ASSAY_ID ASSAY PROJECT PLATE WELL WELL_TYPE RAW_VALUE_A BSUB_VALUE_A Z_SCORE_A RAW_VALUE_B BSUB_VALUE_B Z_SCORE_B COMPOSITE_Z REPRODUCIBILITY CHEMBANK_ID VIRTUAL_ID SMILES 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A01 compound treatment 225360.0 28400.0 1.93 218600.0 22100.0 1.64 2.5292 0.9967 3186889 PK04_093001 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A02 compound treatment 231680.0 34700.0 2.36 226000.0 29500.0 2.19 3.2233 0.9993 3067555 PK04_093002 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A03 compound treatment 197360.0 357.0 0.02 185320.0 -11200.0 -0.83 -0.5721 -0.6862 3186890 PK04_093003 CN(C)C(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A04 compound treatment 222480.0 25500.0 1.74 229160.0 32600.0 2.43 2.9461 0.9865 3186891 PK04_093004 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A05 compound treatment 242120.0 45100.0 3.08 242080.0 45600.0 3.39 4.5729 0.9988 3067558 PK04_093005 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A06 compound treatment 241160.0 44200.0 3.01 239040.0 42500.0 3.16 4.3666 0.9997 3186892 PK04_093006 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A07 compound treatment 264040.0 67000.0 4.57 258720.0 62200.0 4.63 6.5053 1.0 3067559 PK04_093007 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A08 compound treatment 203920.0 6920.0 0.47 207360.0 10800.0 0.81 0.9041 0.9673 3186893 PK04_093008 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A09 compound treatment 181800.0 -15200.0 -1.04 183200.0 -13300.0 -0.99 -1.4338 -0.9997 3186894 PK04_093009 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A10 compound treatment 227040.0 30000.0 2.05 236120.0 39600.0 2.95 3.5323 0.9842 3067560 PK04_093010 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A11 compound treatment 186560.0 -10400.0 -0.71 192520.0 -4000.0 -0.3 -0.7138 -0.925 3186895 PK04_093011 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A12 compound treatment 228080.0 31100.0 2.12 233120.0 36600.0 2.72 3.4245 0.9923 3186896 PK04_093012 NC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A13 mock treatment 181880.0 -15100.0 -1.03 182640.0 -13900.0 -1.03 -1.4594 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A14 mock treatment 184440.0 -12600.0 -0.86 183360.0 -13200.0 -0.98 -1.2981 -0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A15 compound treatment 257840.0 60800.0 4.15 257680.0 61200.0 4.55 6.1517 0.9989 3067562 PK04_093013 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A16 compound treatment 205680.0 8680.0 0.59 214520.0 18000.0 1.34 1.3658 0.9325 3186897 PK04_093014 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A17 compound treatment 188800.0 -8200.0 -0.56 191440.0 -5080.0 -0.38 -0.6626 -0.9818 3067564 PK04_093015 NC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A18 compound treatment 223160.0 26200.0 1.78 237440.0 40900.0 3.05 3.4147 0.9675 3186898 PK04_093016 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A19 compound treatment 229600.0 32600.0 2.22 228480.0 32000.0 2.38 3.2536 0.9994 3186899 PK04_093017 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A20 compound treatment 215440.0 18400.0 1.26 213480.0 17000.0 1.26 1.7815 1.0 3067604 PK04_093018 COCCCNC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A21 compound treatment 229760.0 32800.0 2.23 217480.0 21000.0 1.56 2.6824 0.9846 3186900 PK04_093019 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A22 compound treatment 222720.0 25700.0 1.75 214560.0 18000.0 1.34 2.1893 0.9913 3067607 PK04_093020 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A23 compound treatment 196920.0 -83.1 -0.01 191400.0 -5120.0 -0.38 -0.2733 -0.7175 3186901 PK04_093021 NC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 A24 compound treatment 220880.0 23900.0 1.63 210840.0 14300.0 1.07 1.9049 0.9789 3186902 PK04_093022 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B01 compound treatment 205440.0 8440.0 0.58 210880.0 14400.0 1.07 1.1626 0.9577 3067612 PK04_093023 COC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B02 compound treatment 244680.0 47700.0 3.25 232200.0 35700.0 2.66 4.1763 0.995 3186903 PK04_093024 NC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B03 compound treatment 276200.0 79200.0 5.4 273280.0 76800.0 5.71 7.8578 0.9996 3067614 PK04_093025 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B04 compound treatment 190040.0 -6960.0 -0.47 193320.0 -3200.0 -0.24 -0.5039 -0.949 3186904 PK04_093026 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B05 compound treatment 274080.0 77100.0 5.25 266200.0 69700.0 5.19 7.383 1.0 3186905 PK04_093027 COC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B06 compound treatment 185720.0 -11300.0 -0.77 190080.0 -6440.0 -0.48 -0.8827 -0.974 3068180 PK04_093028 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B07 compound treatment 220840.0 23800.0 1.63 218040.0 21500.0 1.6 2.2819 1.0 3186906 PK04_093029 COC(=O)[C@H]1N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B08 compound treatment 240520.0 43500.0 2.97 235400.0 38900.0 2.89 4.1442 0.9999 3186992 PK04_093030 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B09 compound treatment 265200.0 68200.0 4.65 258880.0 62400.0 4.64 6.5697 1.0 3068181 PK04_093031 COC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B10 compound treatment 247960.0 51000.0 3.47 245160.0 48600.0 3.62 5.0165 0.9998 3186993 PK04_093032 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B11 compound treatment 264920.0 67900.0 4.63 246480.0 50000.0 3.72 5.9036 0.9941 3068182 PK04_093033 COC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B12 compound treatment 242440.0 45400.0 3.1 234800.0 38300.0 2.85 4.2052 0.9991 3186994 PK04_093034 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B13 mock treatment 191240.0 -5760.0 -0.39 188360.0 -8160.0 -0.61 -0.7071 -0.9778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B14 mock treatment 183800.0 -13200.0 -0.9 177280.0 -19200.0 -1.43 -1.6489 -0.975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B15 compound treatment 187760.0 -9240.0 -0.63 192160.0 -4360.0 -0.32 -0.6749 -0.9523 3068183 PK04_093035 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B16 compound treatment 188360.0 -8640.0 -0.59 190440.0 -6080.0 -0.45 -0.7365 -0.9915 3186995 PK04_093036 NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B17 compound treatment 225680.0 28700.0 1.96 218320.0 21800.0 1.62 2.5299 0.9957 3186996 PK04_093037 COC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B18 compound treatment 209080.0 12100.0 0.82 214080.0 17600.0 1.31 1.5065 0.9752 3068184 PK04_093038 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B19 compound treatment 278240.0 81200.0 5.54 276480.0 80000.0 5.95 8.1246 0.9994 3186997 PK04_093039 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B20 compound treatment 244880.0 47900.0 3.26 235120.0 38600.0 2.87 4.3397 0.998 3186998 PK04_093040 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B21 compound treatment 252800.0 55800.0 3.8 250360.0 53800.0 4.01 5.5235 0.9997 3068185 PK04_093041 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B22 compound treatment 196160.0 -843.0 -0.06 190480.0 -6040.0 -0.45 -0.3584 -0.7911 3186999 PK04_093042 CN(C)C(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B23 compound treatment 187960.0 -9040.0 -0.62 181560.0 -15000.0 -1.11 -1.2231 -0.9612 3068186 PK04_093043 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 B24 compound treatment 211880.0 14900.0 1.01 225560.0 29000.0 2.16 2.2457 0.9405 3187000 PK04_093044 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C01 compound treatment 250160.0 53200.0 3.62 241880.0 45400.0 3.38 4.95 0.9994 3187001 PK04_093045 CN(C)C(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C02 compound treatment 220320.0 23300.0 1.59 227760.0 31200.0 2.33 2.7683 0.9828 3068187 PK04_093046 CN(C)C(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C03 compound treatment 217000.0 20000.0 1.36 224880.0 28400.0 2.11 2.4567 0.9776 3187002 PK04_093047 COCCCNC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C04 compound treatment 211360.0 14400.0 0.98 209720.0 13200.0 0.98 1.387 1.0 3068188 PK04_093048 NC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C05 compound treatment 233080.0 36100.0 2.46 248440.0 51900.0 3.86 4.4718 0.9762 3187003 PK04_093049 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C06 compound treatment 235480.0 38500.0 2.62 234320.0 37800.0 2.81 3.8444 0.9994 3187004 PK04_093050 CN(C)C(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C07 compound treatment 198080.0 1080.0 0.07 210920.0 14400.0 1.07 0.8099 0.7538 3068189 PK04_093051 NC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C08 compound treatment 194600.0 -2400.0 -0.16 193720.0 -2800.0 -0.21 -0.263 -0.993 3187005 PK04_093052 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C09 compound treatment 191080.0 -5920.0 -0.4 195280.0 -1240.0 -0.09 -0.3506 -0.8466 3187006 PK04_093053 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C10 compound treatment 237840.0 40800.0 2.78 232320.0 35800.0 2.66 3.8529 0.9998 3068190 PK04_093054 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C11 mock treatment 188680.0 -8320.0 -0.57 191720.0 -4800.0 -0.36 -0.6537 -0.9751 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C12 mock treatment 201200.0 4200.0 0.29 192080.0 -4440.0 -0.33 -0.0312 -0.0714 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C13 compound treatment 222480.0 25500.0 1.74 219080.0 22600.0 1.68 2.4156 0.9999 3187007 PK04_093055 COC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C14 compound treatment 190200.0 -6800.0 -0.46 193080.0 -3440.0 -0.26 -0.5088 -0.9607 3068191 PK04_093056 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C15 mock treatment 188720.0 -8280.0 -0.56 182680.0 -13800.0 -1.03 -1.1275 -0.96 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C16 mock treatment 188680.0 -8320.0 -0.57 185240.0 -11300.0 -0.84 -0.9947 -0.9818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C17 compound treatment 224640.0 27600.0 1.88 219480.0 23000.0 1.71 2.5408 0.9988 3187008 PK04_093057 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C18 compound treatment 222160.0 25200.0 1.72 224080.0 27600.0 2.05 2.6634 0.996 3068193 PK04_093058 COCCCNC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C19 compound treatment 231480.0 34500.0 2.35 222080.0 25600.0 1.9 3.0074 0.9945 3187009 PK04_093059 COC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C20 compound treatment 209800.0 12800.0 0.87 208160.0 11600.0 0.87 1.2297 1.0 3187010 PK04_093060 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C21 compound treatment 241120.0 44100.0 3.01 251440.0 54900.0 4.09 5.0173 0.9886 3068197 PK04_093061 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C22 compound treatment 187560.0 -9440.0 -0.64 186040.0 -10500.0 -0.78 -1.0066 -0.9955 3187011 PK04_093062 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C23 compound treatment 189240.0 -7760.0 -0.53 180720.0 -15800.0 -1.18 -1.2056 -0.935 3068199 PK04_093063 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 C24 compound treatment 211000.0 14000.0 0.95 207480.0 11000.0 0.82 1.2517 0.997 3187012 PK04_093064 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D01 compound treatment 194440.0 -2560.0 -0.17 199160.0 2640.0 0.2 0.0155 0.0591 3187091 PK04_093065 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D02 compound treatment 195520.0 -1480.0 -0.1 190440.0 -6080.0 -0.45 -0.3913 -0.8443 3068202 PK04_093066 CN(C)C(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D03 compound treatment 197720.0 717.0 0.05 202480.0 5960.0 0.44 0.3484 0.7803 3187092 PK04_093067 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D04 compound treatment 220040.0 23000.0 1.57 216920.0 20400.0 1.52 2.1843 0.9999 3187093 PK04_093068 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D05 compound treatment 274480.0 77500.0 5.28 261280.0 64800.0 4.82 7.1434 0.999 3068220 PK04_093069 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D06 compound treatment 232040.0 35000.0 2.39 223800.0 27300.0 2.03 3.1249 0.9967 3187094 PK04_093070 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D07 compound treatment 195800.0 -1200.0 -0.08 194480.0 -2040.0 -0.15 -0.1652 -0.9584 3068223 PK04_093071 COC(=O)[C@H]1COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D08 compound treatment 252160.0 55200.0 3.76 243000.0 46500.0 3.46 5.1053 0.9991 3187095 PK04_093072 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D09 compound treatment 247160.0 50200.0 3.42 239800.0 43300.0 3.22 4.6959 0.9996 3068225 PK04_093073 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D10 compound treatment 195800.0 -1200.0 -0.08 197280.0 763.0 0.06 -0.0178 -0.1788 3187096 PK04_093074 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D11 mock treatment 184840.0 -12200.0 -0.83 188240.0 -8280.0 -0.62 -1.022 -0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D12 mock treatment 189840.0 -7160.0 -0.49 187200.0 -9320.0 -0.69 -0.8356 -0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D13 compound treatment 257640.0 60600.0 4.13 250440.0 53900.0 4.01 5.7611 0.9999 3187097 PK04_093075 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D14 compound treatment 221080.0 24100.0 1.64 218720.0 22200.0 1.65 2.3292 1.0 3068228 PK04_093076 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D15 mock treatment 185920.0 -11100.0 -0.76 191760.0 -4760.0 -0.35 -0.7846 -0.9403 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D16 mock treatment 186920.0 -10100.0 -0.69 188440.0 -8080.0 -0.6 -0.9112 -0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D17 compound treatment 202040.0 5040.0 0.34 200280.0 3760.0 0.28 0.4409 0.9949 3187098 PK04_093077 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D18 compound treatment 214160.0 17200.0 1.17 218720.0 22200.0 1.65 1.9956 0.9857 3187099 PK04_093078 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D19 compound treatment 228920.0 31900.0 2.18 228880.0 32400.0 2.41 3.2419 0.9987 3068229 PK04_093079 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D20 compound treatment 198800.0 1800.0 0.12 207160.0 10600.0 0.79 0.6467 0.8069 3187100 PK04_093080 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D21 compound treatment 238360.0 41400.0 2.82 242600.0 46100.0 3.43 4.419 0.9953 3068232 PK04_093081 COC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D22 compound treatment 186560.0 -10400.0 -0.71 181040.0 -15500.0 -1.15 -1.318 -0.9733 3187101 PK04_093082 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D23 compound treatment 236840.0 39800.0 2.72 218960.0 22400.0 1.67 3.1016 0.9727 3187102 PK04_093083 COC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 D24 compound treatment 179200.0 -17800.0 -1.21 181320.0 -15200.0 -1.13 -1.658 -0.9994 3068234 PK04_093084 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E01 mock treatment 188080.0 -8920.0 -0.61 185480.0 -11000.0 -0.82 -1.011 -0.9891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E02 mock treatment 191000.0 -6000.0 -0.41 190040.0 -6480.0 -0.48 -0.6303 -0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E03 compound treatment 206200.0 9200.0 0.63 213600.0 17100.0 1.27 1.3424 0.9469 3187103 PK04_093085 COC(=O)[C@H]1N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E04 compound treatment 216720.0 19700.0 1.34 219920.0 23400.0 1.74 2.1822 0.9918 3187104 PK04_093086 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E05 compound treatment 207480.0 10500.0 0.71 207600.0 11100.0 0.82 1.0884 0.9974 3068237 PK04_093087 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E06 compound treatment 202800.0 5800.0 0.4 199920.0 3400.0 0.25 0.4586 0.9769 3187105 PK04_093088 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E07 compound treatment 238080.0 41100.0 2.8 234600.0 38100.0 2.83 3.9845 1.0 3068240 PK04_093089 COC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E08 compound treatment 229960.0 33000.0 2.25 223480.0 27000.0 2.01 3.0078 0.9984 3187106 PK04_093090 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E09 mock treatment 189280.0 -7720.0 -0.53 196040.0 -477.0 -0.04 -0.3974 -0.7531 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E10 mock treatment 193640.0 -3360.0 -0.23 192480.0 -4040.0 -0.3 -0.3746 -0.9911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E11 compound treatment 196360.0 -643.0 -0.04 208320.0 11800.0 0.88 0.5902 0.671 3068242 PK04_093091 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E12 compound treatment 270040.0 73000.0 4.98 264560.0 68000.0 5.06 7.1019 1.0 3187107 PK04_093092 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E13 compound treatment 239440.0 42400.0 2.89 229000.0 32500.0 2.42 3.7553 0.996 3068264 PK04_093093 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E14 compound treatment 233160.0 36200.0 2.47 224840.0 28300.0 2.11 3.2336 0.997 3187108 PK04_093094 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E15 compound treatment 234720.0 37700.0 2.57 222200.0 25700.0 1.91 3.1699 0.9893 3187109 PK04_093095 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E16 compound treatment 235520.0 38500.0 2.63 246920.0 50400.0 3.75 4.5094 0.9848 3068267 PK04_093096 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E17 mock treatment 190840.0 -6160.0 -0.42 192600.0 -3920.0 -0.29 -0.5033 -0.984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E18 mock treatment 192600.0 -4400.0 -0.3 197040.0 523.0 0.04 -0.1847 -0.6103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E19 compound treatment 195240.0 -1760.0 -0.12 194400.0 -2120.0 -0.16 -0.1964 -0.9911 3187110 PK04_093097 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E20 compound treatment 201680.0 4680.0 0.32 203040.0 6520.0 0.49 0.5688 0.9792 3187111 PK04_093098 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E21 compound treatment 242960.0 46000.0 3.13 250440.0 53900.0 4.01 5.0534 0.9925 3068269 PK04_093099 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E22 compound treatment 235920.0 38900.0 2.65 234040.0 37500.0 2.79 3.8509 0.9997 3187184 PK04_093100 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E23 compound treatment 208120.0 11100.0 0.76 206360.0 9840.0 0.73 1.0539 0.9999 3068272 PK04_093101 COC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 E24 compound treatment 204480.0 7480.0 0.51 192160.0 -4360.0 -0.32 0.1312 0.2171 3187185 PK04_093102 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F01 mock treatment 190480.0 -6520.0 -0.44 195640.0 -877.0 -0.07 -0.3606 -0.8023 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F02 mock treatment 187320.0 -9680.0 -0.66 195880.0 -637.0 -0.05 -0.5003 -0.7559 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F03 compound treatment 258400.0 61400.0 4.19 251680.0 55200.0 4.11 5.863 1.0 3068274 PK04_093103 COC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F04 compound treatment 223280.0 26300.0 1.79 218680.0 22200.0 1.65 2.4332 0.9992 3187186 PK04_093104 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F05 compound treatment 239320.0 42300.0 2.89 228080.0 31600.0 2.35 3.7011 0.9948 3068276 PK04_093105 COC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F06 compound treatment 272880.0 75900.0 5.17 263200.0 66700.0 4.96 7.1673 0.9998 3187187 PK04_093106 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F07 compound treatment 228480.0 31500.0 2.15 225200.0 28700.0 2.13 3.027 1.0 3187188 PK04_093107 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F08 compound treatment 212640.0 15600.0 1.07 225120.0 28600.0 2.13 2.2591 0.9489 3068278 PK04_093108 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F09 mock treatment 194120.0 -2880.0 -0.2 194200.0 -2320.0 -0.17 -0.2609 -0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F10 mock treatment 195160.0 -1840.0 -0.13 198720.0 2200.0 0.16 0.0271 0.1311 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F11 compound treatment 239600.0 42600.0 2.9 226680.0 30200.0 2.24 3.6409 0.9919 3187189 PK04_093109 COC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F12 compound treatment 205800.0 8800.0 0.6 203600.0 7080.0 0.53 0.7969 0.9979 3068280 PK04_093110 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F13 compound treatment 244680.0 47700.0 3.25 240840.0 44300.0 3.3 4.631 1.0 3187190 PK04_093111 COC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F14 compound treatment 261120.0 64100.0 4.37 252880.0 56400.0 4.19 6.0572 0.9998 3187191 PK04_093112 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F15 compound treatment 235720.0 38700.0 2.64 241880.0 45400.0 3.38 4.2538 0.9926 3068282 PK04_093113 COC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F16 compound treatment 215200.0 18200.0 1.24 220800.0 24300.0 1.81 2.1552 0.9831 3187192 PK04_093114 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F17 mock treatment 189040.0 -7960.0 -0.54 191800.0 -4720.0 -0.35 -0.6321 -0.9777 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F18 mock treatment 192520.0 -4480.0 -0.31 190000.0 -6520.0 -0.49 -0.5591 -0.9752 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F19 compound treatment 296760.0 99800.0 6.8 285880.0 89400.0 6.65 9.5121 0.9999 3187193 PK04_093115 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F20 compound treatment 192600.0 -4400.0 -0.3 194520.0 -2000.0 -0.15 -0.3174 -0.9474 3068312 PK04_093116 NC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F21 compound treatment 247600.0 50600.0 3.45 234240.0 37700.0 2.81 4.4245 0.9948 3068314 PK04_093117 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F22 compound treatment 205040.0 8040.0 0.55 202400.0 5880.0 0.44 0.6971 0.9938 3187194 PK04_093118 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F23 compound treatment 220880.0 23900.0 1.63 247280.0 50800.0 3.78 3.8226 0.9292 3187195 PK04_093119 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 F24 compound treatment 184560.0 -12400.0 -0.85 184560.0 -12000.0 -0.89 -1.2291 -0.9997 3068317 PK04_093120 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G01 compound treatment 229560.0 32600.0 2.22 221200.0 24700.0 1.84 2.8685 0.9956 3187196 PK04_093121 COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G02 compound treatment 205360.0 8360.0 0.57 201640.0 5120.0 0.38 0.6725 0.9809 3068319 PK04_093122 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G03 mock treatment 198360.0 1360.0 0.09 202200.0 5680.0 0.42 0.3645 0.8419 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G04 mock treatment 205280.0 8280.0 0.56 199840.0 3320.0 0.25 0.5739 0.9315 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G05 compound treatment 233360.0 36400.0 2.48 236520.0 40000.0 2.98 3.858 0.9959 3187197 PK04_093123 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G06 compound treatment 215120.0 18100.0 1.24 220040.0 23500.0 1.75 2.1114 0.9854 3187198 PK04_093124 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G07 compound treatment 217160.0 20200.0 1.37 221800.0 25300.0 1.88 2.3023 0.9881 3068323 PK04_093125 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G08 compound treatment 227920.0 30900.0 2.11 229520.0 33000.0 2.46 3.2273 0.9971 3187199 PK04_093126 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G09 compound treatment 232240.0 35200.0 2.4 238040.0 41500.0 3.09 3.884 0.9922 3068325 PK04_093127 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G10 compound treatment 240320.0 43300.0 2.95 232000.0 35500.0 2.64 3.9556 0.9984 3187200 PK04_093128 COCCCNC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G11 compound treatment 239200.0 42200.0 2.88 233120.0 36600.0 2.72 3.9606 0.9996 3187201 PK04_093129 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G12 compound treatment 270320.0 73300.0 5.0 223800.0 27300.0 2.03 4.9703 0.9212 3068327 PK04_093130 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G13 compound treatment 232560.0 35600.0 2.42 224320.0 27800.0 2.07 3.1774 0.9969 3187202 PK04_093131 COC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G14 compound treatment 207200.0 10200.0 0.7 203160.0 6640.0 0.49 0.8412 0.9861 3187203 PK04_093132 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G15 compound treatment 199520.0 2520.0 0.17 201320.0 4800.0 0.36 0.3741 0.9435 3068330 PK04_093133 COC(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G16 compound treatment 234360.0 37400.0 2.55 239840.0 43300.0 3.22 4.0809 0.9932 3068332 PK04_093134 NC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G17 compound treatment 236480.0 39500.0 2.69 240280.0 43800.0 3.26 4.2063 0.9955 3187278 PK04_093135 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G18 compound treatment 193640.0 -3360.0 -0.23 202240.0 5720.0 0.43 0.1391 0.2875 3187279 PK04_093136 COCCCNC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G19 mock treatment 196480.0 -523.0 -0.04 200280.0 3760.0 0.28 0.1728 0.6121 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G20 mock treatment 197680.0 677.0 0.05 200440.0 3920.0 0.29 0.2391 0.8088 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G21 compound treatment 195280.0 -1720.0 -0.12 194760.0 -1760.0 -0.13 -0.1755 -0.9986 3187280 PK04_093137 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G22 compound treatment 205840.0 8840.0 0.6 214960.0 18400.0 1.37 1.3966 0.9317 3068361 PK04_093138 COCCCNC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G23 compound treatment 210120.0 13100.0 0.89 215640.0 19100.0 1.42 1.6388 0.9749 3187281 PK04_093139 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 G24 compound treatment 214560.0 17600.0 1.2 217200.0 20700.0 1.54 1.9349 0.9923 3187282 PK04_093140 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H01 compound treatment 314840.0 118000.0 8.03 303040.0 107000.0 7.93 11.2868 1.0 3068365 PK04_093141 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H02 compound treatment 254400.0 57400.0 3.91 251280.0 54800.0 4.08 5.6491 0.9998 3187283 PK04_093142 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H03 mock treatment 203800.0 6800.0 0.46 198840.0 2320.0 0.17 0.4499 0.9097 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H04 mock treatment 200400.0 3400.0 0.23 201080.0 4560.0 0.34 0.4039 0.9826 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H05 compound treatment 302480.0 105000.0 7.19 282960.0 86400.0 6.43 9.6342 0.9985 3068368 PK04_093143 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H06 compound treatment 205680.0 8680.0 0.59 203880.0 7360.0 0.55 0.8058 0.9993 3187284 PK04_093144 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H07 compound treatment 258720.0 61700.0 4.21 261080.0 64600.0 4.81 6.3731 0.9978 3187285 PK04_093145 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(CC=C)C1=O)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H08 compound treatment 219000.0 22000.0 1.5 206200.0 9680.0 0.72 1.57 0.9436 3068370 PK04_093146 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H09 compound treatment 271240.0 74200.0 5.06 256960.0 60400.0 4.5 6.7598 0.9983 3187286 PK04_093147 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H10 compound treatment 239760.0 42800.0 2.92 236560.0 40000.0 2.98 4.1686 0.9999 3187287 PK04_093148 CN(C)C(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H11 compound treatment 285400.0 88400.0 6.03 271520.0 75000.0 5.58 8.2087 0.9993 3068373 PK04_093149 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H12 compound treatment 203840.0 6840.0 0.47 204760.0 8240.0 0.61 0.7634 0.9908 3187288 PK04_093150 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H13 compound treatment 252920.0 55900.0 3.81 248920.0 52400.0 3.9 5.4535 0.9999 3187289 PK04_093151 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3N(CC=C)C1=O)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H14 compound treatment 251400.0 54400.0 3.71 237880.0 41400.0 3.08 4.7992 0.9957 3068375 PK04_093152 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H15 compound treatment 202280.0 5280.0 0.36 224040.0 27500.0 2.05 1.7029 0.8188 3187290 PK04_093153 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H16 compound treatment 244240.0 47200.0 3.22 247160.0 50600.0 3.77 4.9424 0.9969 3187291 PK04_093154 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H17 compound treatment 281120.0 84100.0 5.73 269360.0 72800.0 5.42 7.8887 0.9996 3068378 PK04_093155 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H18 compound treatment 194640.0 -2360.0 -0.16 200200.0 3680.0 0.27 0.0799 0.2513 3187292 PK04_093156 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H19 mock treatment 198240.0 1240.0 0.08 194840.0 -1680.0 -0.12 -0.0286 -0.19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H20 mock treatment 198440.0 1440.0 0.1 205320.0 8800.0 0.66 0.5326 0.8039 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H21 compound treatment 296720.0 99700.0 6.8 274200.0 77700.0 5.78 8.8955 0.9968 3187293 PK04_093157 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H22 compound treatment 216800.0 19800.0 1.35 230000.0 33500.0 2.49 2.7165 0.9585 3068380 PK04_093158 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H23 compound treatment 226400.0 29400.0 2.0 248080.0 51600.0 3.84 4.1308 0.9541 3068402 PK04_093159 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 H24 compound treatment 191920.0 -5080.0 -0.35 188840.0 -7680.0 -0.57 -0.6491 -0.9713 3187294 PK04_093160 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I01 compound treatment 248640.0 51600.0 3.52 251840.0 55300.0 4.12 5.4009 0.997 3068406 PK04_093161 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I02 compound treatment 238800.0 41800.0 2.85 244160.0 47600.0 3.55 4.5223 0.9941 3187295 PK04_093162 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I03 compound treatment 212120.0 15100.0 1.03 214520.0 18000.0 1.34 1.6762 0.9916 3068409 PK04_093163 COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I04 compound treatment 204400.0 7400.0 0.5 200480.0 3960.0 0.29 0.5652 0.9674 3187296 PK04_093164 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I05 mock treatment 212360.0 15400.0 1.05 211600.0 15100.0 1.12 1.5341 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I06 mock treatment 215520.0 18500.0 1.26 203480.0 6960.0 0.52 1.2591 0.9227 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I07 compound treatment 214480.0 17500.0 1.19 217800.0 21300.0 1.58 1.9626 0.9901 3187297 PK04_093165 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I08 compound treatment 216560.0 19600.0 1.33 212280.0 15800.0 1.17 1.7724 0.998 3068413 PK04_093166 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I09 compound treatment 275000.0 78000.0 5.32 287600.0 91100.0 6.78 8.5536 0.9928 3187298 PK04_093167 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I10 compound treatment 231520.0 34500.0 2.35 237520.0 41000.0 3.05 3.8219 0.9918 3187366 PK04_093168 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I11 compound treatment 252720.0 55700.0 3.8 262280.0 65800.0 4.89 6.147 0.9921 3068416 PK04_093169 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I12 compound treatment 270760.0 73800.0 5.03 270960.0 74400.0 5.54 7.4735 0.9988 3187367 PK04_093170 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I13 compound treatment 204600.0 7600.0 0.52 203480.0 6960.0 0.52 0.7327 1.0 3068419 PK04_093171 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I14 compound treatment 230000.0 33000.0 2.25 239520.0 43000.0 3.2 3.8539 0.9851 3187368 PK04_093172 CN(C)C(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I15 compound treatment 210040.0 13000.0 0.89 209160.0 12600.0 0.94 1.2939 0.9996 3068421 PK04_093173 COC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I16 compound treatment 207080.0 10100.0 0.69 211520.0 15000.0 1.12 1.2754 0.9728 3187369 PK04_093174 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I17 compound treatment 197200.0 197.0 0.01 198120.0 1600.0 0.12 0.0939 0.7817 3068423 PK04_093175 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I18 compound treatment 199600.0 2600.0 0.18 196880.0 363.0 0.03 0.1443 0.8057 3187370 PK04_093176 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I19 compound treatment 180440.0 -16600.0 -1.13 169880.0 -26600.0 -1.98 -2.2003 -0.9644 3187371 PK04_093177 COC(=O)[C@H]1N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I20 compound treatment 217400.0 20400.0 1.39 240880.0 44400.0 3.3 3.318 0.9261 3068425 PK04_093178 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I21 mock treatment 195440.0 -1560.0 -0.11 197400.0 883.0 0.07 -0.0289 -0.2306 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I22 mock treatment 191520.0 -5480.0 -0.37 196400.0 -117.0 -0.01 -0.2705 -0.7234 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I23 compound treatment 218800.0 21800.0 1.49 217600.0 21100.0 1.57 2.1603 0.9996 3187372 PK04_093179 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 I24 compound treatment 180560.0 -16400.0 -1.12 183000.0 -13500.0 -1.01 -1.5041 -0.9985 3068456 PK04_093180 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J01 compound treatment 271160.0 74200.0 5.06 256200.0 59700.0 4.44 6.716 0.9979 3187373 PK04_093181 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3N(CC=C)C1=O)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J02 compound treatment 257360.0 60400.0 4.11 253160.0 56600.0 4.22 5.8907 0.9999 3187374 PK04_093182 CN(C)C(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J03 compound treatment 232960.0 36000.0 2.45 218680.0 22200.0 1.65 2.8998 0.9814 3068460 PK04_093183 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J04 compound treatment 202120.0 5120.0 0.35 201800.0 5280.0 0.39 0.5247 0.9982 3187375 PK04_093184 COCCCNC(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J05 mock treatment 209600.0 12600.0 0.86 204560.0 8040.0 0.6 1.0306 0.9844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J06 mock treatment 210920.0 13900.0 0.95 201120.0 4600.0 0.34 0.9132 0.9052 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J07 compound treatment 322760.0 126000.0 8.57 302800.0 106000.0 7.91 11.656 0.9992 3187376 PK04_093185 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J08 compound treatment 266120.0 69100.0 4.71 252280.0 55800.0 4.15 6.2667 0.998 3068463 PK04_093186 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J09 compound treatment 254560.0 57600.0 3.92 241120.0 44600.0 3.32 5.1221 0.9965 3187377 PK04_093187 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J10 compound treatment 205880.0 8880.0 0.61 204040.0 7520.0 0.56 0.8239 0.9992 3068465 PK04_093188 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J11 compound treatment 275280.0 78300.0 5.34 273760.0 77200.0 5.75 7.8387 0.9993 3187378 PK04_093189 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(Cc5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J12 compound treatment 209840.0 12800.0 0.88 209160.0 12600.0 0.94 1.2842 0.9993 3068467 PK04_093190 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J13 compound treatment 231680.0 34700.0 2.36 262520.0 66000.0 4.91 5.1453 0.9438 3187379 PK04_093191 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(Cc5ccccc5)C3=O)[C@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J14 compound treatment 253760.0 56800.0 3.87 250680.0 54200.0 4.03 5.5866 0.9998 3187380 PK04_093192 COCCCNC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J15 compound treatment 273240.0 76200.0 5.2 257160.0 60600.0 4.51 6.8668 0.9975 3068470 PK04_093193 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J16 compound treatment 218480.0 21500.0 1.46 207200.0 10700.0 0.8 1.5976 0.9588 3187381 PK04_093194 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J17 compound treatment 264960.0 68000.0 4.63 257120.0 60600.0 4.51 6.4655 0.9999 3187382 PK04_093195 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J18 compound treatment 228520.0 31500.0 2.15 225800.0 29300.0 2.18 3.0605 1.0 3068473 PK04_093196 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J19 compound treatment 267040.0 70000.0 4.77 255200.0 58700.0 4.37 6.4647 0.999 3187383 PK04_093197 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J20 compound treatment 203160.0 6160.0 0.42 193880.0 -2640.0 -0.2 0.158 0.3411 3068475 PK04_093198 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J21 mock treatment 193560.0 -3440.0 -0.23 195840.0 -677.0 -0.05 -0.2016 -0.8397 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J22 mock treatment 193280.0 -3720.0 -0.25 188720.0 -7800.0 -0.58 -0.5898 -0.9312 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J23 compound treatment 267280.0 70300.0 4.79 247800.0 51300.0 3.82 6.0868 0.9937 3187384 PK04_093199 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 J24 compound treatment 257720.0 60700.0 4.14 246080.0 49600.0 3.69 5.5355 0.9983 3068477 PK04_093200 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K01 compound treatment 215400.0 18400.0 1.25 212600.0 16100.0 1.2 1.7333 0.9997 3187385 PK04_093201 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K02 compound treatment 264000.0 67000.0 4.57 264600.0 68100.0 5.07 6.8129 0.9987 3187386 PK04_093202 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K03 compound treatment 238320.0 41300.0 2.82 229440.0 32900.0 2.45 3.7245 0.9976 3187447 PK04_093203 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K04 compound treatment 287680.0 90700.0 6.18 301560.0 105000.0 7.82 9.8996 0.9932 3068500 PK04_093204 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K05 compound treatment 296720.0 99700.0 6.8 283120.0 86600.0 6.45 9.3649 0.9996 3187448 PK04_093205 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K06 compound treatment 233960.0 37000.0 2.52 230560.0 34000.0 2.53 3.5732 1.0 3187449 PK04_093206 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K07 mock treatment 209120.0 12100.0 0.83 209920.0 13400.0 1.0 1.2895 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K08 mock treatment 204760.0 7760.0 0.53 202880.0 6360.0 0.47 0.7088 0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K09 compound treatment 250600.0 53600.0 3.65 249680.0 53200.0 3.96 5.3817 0.9992 3068503 PK04_093207 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K10 compound treatment 245240.0 48200.0 3.29 232640.0 36100.0 2.69 4.2265 0.995 3187450 PK04_093208 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K11 compound treatment 293800.0 96800.0 6.6 287480.0 91000.0 6.77 9.4536 0.9999 3068506 PK04_093209 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K12 compound treatment 245160.0 48200.0 3.28 225120.0 28600.0 2.13 3.8269 0.978 3187451 PK04_093210 CN(C)C(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K13 compound treatment 218840.0 21800.0 1.49 233080.0 36600.0 2.72 2.977 0.9597 3187452 PK04_093211 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K14 compound treatment 265880.0 68900.0 4.7 254880.0 58400.0 4.34 6.392 0.9992 3068509 PK04_093212 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K15 mock treatment 199400.0 2400.0 0.16 200120.0 3600.0 0.27 0.3052 0.9718 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K16 mock treatment 198600.0 1600.0 0.11 197440.0 923.0 0.07 0.1256 0.9754 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K17 compound treatment 210760.0 13800.0 0.94 209280.0 12800.0 0.95 1.3349 1.0 3187453 PK04_093213 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K18 compound treatment 202720.0 5720.0 0.39 209280.0 12800.0 0.95 0.9473 0.9226 3187454 PK04_093214 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K19 compound treatment 236080.0 39100.0 2.66 232800.0 36300.0 2.7 3.7933 1.0 3068511 PK04_093215 COC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K20 compound treatment 221240.0 24200.0 1.65 220000.0 23500.0 1.75 2.4043 0.9996 3187455 PK04_093216 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K21 compound treatment 204920.0 7920.0 0.54 200120.0 3600.0 0.27 0.5713 0.9479 3068513 PK04_093217 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K22 compound treatment 202520.0 5520.0 0.38 209960.0 13400.0 1.0 0.9734 0.9107 3187456 PK04_093218 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K23 mock treatment 189280.0 -7720.0 -0.53 183360.0 -13200.0 -0.98 -1.0647 -0.9577 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 K24 mock treatment 185080.0 -11900.0 -0.81 178160.0 -18400.0 -1.37 -1.5409 -0.9692 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L01 compound treatment 311480.0 114000.0 7.8 281320.0 84800.0 6.31 9.9817 0.9945 3187457 PK04_093219 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L02 compound treatment 248960.0 52000.0 3.54 253240.0 56700.0 4.22 5.49 0.9962 3068516 PK04_093220 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L03 compound treatment 323200.0 126000.0 8.6 318720.0 122000.0 9.1 12.515 0.9996 3187458 PK04_093221 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L04 compound treatment 275360.0 78400.0 5.34 267480.0 71000.0 5.28 7.5121 1.0 3187459 PK04_093222 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L05 compound treatment 300560.0 104000.0 7.06 282840.0 86300.0 6.42 9.5353 0.9989 3068518 PK04_093223 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L06 compound treatment 262280.0 65300.0 4.45 253320.0 56800.0 4.23 6.1363 0.9997 3187460 PK04_093224 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L07 mock treatment 200600.0 3600.0 0.25 210360.0 13800.0 1.03 0.9019 0.8516 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L08 mock treatment 205040.0 8040.0 0.55 205440.0 8920.0 0.66 0.857 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L09 compound treatment 251200.0 54200.0 3.69 249160.0 52600.0 3.92 5.3832 0.9996 3068520 PK04_093225 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(CC=C)C1=O)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L10 compound treatment 204200.0 7200.0 0.49 209760.0 13200.0 0.99 1.0439 0.9481 3187461 PK04_093226 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L11 compound treatment 280360.0 83400.0 5.68 271920.0 75400.0 5.61 7.9868 1.0 3187462 PK04_093227 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4N(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L12 compound treatment 231560.0 34600.0 2.36 218560.0 22000.0 1.64 2.826 0.9844 3187463 PK04_093228 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L13 compound treatment 272160.0 75200.0 5.12 265960.0 69400.0 5.17 7.2778 1.0 3068543 PK04_093229 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(Cc5ccccc5)C3=O)[C@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L14 compound treatment 282400.0 85400.0 5.82 264320.0 67800.0 5.05 7.6852 0.9975 3187464 PK04_093230 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L15 mock treatment 203960.0 6960.0 0.47 201040.0 4520.0 0.34 0.5734 0.9859 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L16 mock treatment 197680.0 677.0 0.05 198160.0 1640.0 0.12 0.1191 0.9112 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L17 compound treatment 232600.0 35600.0 2.43 222480.0 26000.0 1.93 3.0824 0.9936 3068545 PK04_093231 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L18 compound treatment 230240.0 33200.0 2.27 239000.0 42500.0 3.16 3.8381 0.9867 3187465 PK04_093232 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L19 compound treatment 260440.0 63400.0 4.32 252560.0 56000.0 4.17 6.0076 0.9998 3187466 PK04_093233 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L20 compound treatment 205800.0 8800.0 0.6 203440.0 6920.0 0.52 0.7884 0.9971 3068547 PK04_093234 NC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L21 compound treatment 224720.0 27700.0 1.89 264880.0 68400.0 5.09 4.934 0.9091 3187467 PK04_093235 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L22 compound treatment 204680.0 7680.0 0.52 217000.0 20500.0 1.52 1.4481 0.8984 3068549 PK04_093236 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L23 mock treatment 186480.0 -10500.0 -0.72 186360.0 -10200.0 -0.76 -1.0418 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 L24 mock treatment 183000.0 -14000.0 -0.95 179960.0 -16600.0 -1.23 -1.5464 -0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M01 compound treatment 246440.0 49400.0 3.37 234360.0 37800.0 2.82 4.3749 0.996 3187528 PK04_093237 COC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M02 compound treatment 271680.0 74700.0 5.09 272040.0 75500.0 5.62 7.5747 0.9988 3187529 PK04_093238 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M03 compound treatment 209080.0 12100.0 0.82 207960.0 11400.0 0.85 1.1844 0.9999 3068551 PK04_093239 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M04 compound treatment 241680.0 44700.0 3.05 252040.0 55500.0 4.13 5.0759 0.9887 3187530 PK04_093240 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M05 compound treatment 212080.0 15100.0 1.03 215640.0 19100.0 1.42 1.7332 0.9872 3068553 PK04_093241 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M06 compound treatment 215320.0 18300.0 1.25 224760.0 28200.0 2.1 2.3694 0.9691 3187531 PK04_093242 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M07 compound treatment 283040.0 86000.0 5.87 285960.0 89400.0 6.66 8.8549 0.998 3187532 PK04_093243 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M08 compound treatment 270640.0 73600.0 5.02 265360.0 68800.0 5.12 7.173 0.9999 3068555 PK04_093244 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M09 mock treatment 208560.0 11600.0 0.79 210040.0 13500.0 1.01 1.2688 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M10 mock treatment 211000.0 14000.0 0.95 207920.0 11400.0 0.85 1.2749 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M11 compound treatment 216760.0 19800.0 1.35 221480.0 25000.0 1.86 2.2662 0.9875 3187533 PK04_093245 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M12 compound treatment 247960.0 51000.0 3.47 247160.0 50600.0 3.77 5.1218 0.9992 3187534 PK04_093246 COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M13 mock treatment 212640.0 15600.0 1.07 204000.0 7480.0 0.56 1.1476 0.9542 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M14 mock treatment 212040.0 15000.0 1.03 211280.0 14800.0 1.1 1.5019 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M15 compound treatment 240200.0 43200.0 2.95 238480.0 42000.0 3.12 4.2909 0.9996 3068558 PK04_093247 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M16 compound treatment 202960.0 5960.0 0.41 206680.0 10200.0 0.76 0.822 0.9575 3187535 PK04_093248 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M17 compound treatment 212520.0 15500.0 1.06 214800.0 18300.0 1.36 1.7102 0.9923 3068560 PK04_093249 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M18 compound treatment 240360.0 43400.0 2.96 257160.0 60600.0 4.51 5.2817 0.9789 3187536 PK04_093250 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M19 compound treatment 226040.0 29000.0 1.98 228840.0 32300.0 2.41 3.1009 0.9953 3187537 PK04_093251 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M20 compound treatment 203720.0 6720.0 0.46 202640.0 6120.0 0.46 0.6461 1.0 3068562 PK04_093252 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)N3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M21 compound treatment 201720.0 4720.0 0.32 207880.0 11400.0 0.85 0.8254 0.9123 3068586 PK04_093253 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M22 compound treatment 216280.0 19300.0 1.31 227600.0 31100.0 2.31 2.5651 0.9641 3187538 PK04_093254 NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M23 compound treatment 230080.0 33100.0 2.26 217000.0 20500.0 1.52 2.6726 0.9818 3068589 PK04_093255 COC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 M24 compound treatment 275280.0 78300.0 5.34 269600.0 73100.0 5.44 7.6198 1.0 3187539 PK04_093256 NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N01 compound treatment 333480.0 136000.0 9.3 324880.0 128000.0 9.55 13.3348 0.9999 3187540 PK04_093257 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3N(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N02 compound treatment 253120.0 56100.0 3.83 255360.0 58800.0 4.38 5.8021 0.9977 3187541 PK04_093258 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N03 compound treatment 302320.0 105000.0 7.18 291440.0 94900.0 7.06 10.0727 1.0 3068594 PK04_093259 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(CC=C)C3=O)[C@@H](O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N04 compound treatment 211920.0 14900.0 1.02 213480.0 17000.0 1.26 1.6118 0.9942 3187542 PK04_093260 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N05 compound treatment 253600.0 56600.0 3.86 251840.0 55300.0 4.12 5.64 0.9995 3068597 PK04_093261 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N06 compound treatment 234840.0 37800.0 2.58 236840.0 40300.0 3.0 3.9462 0.9972 3187543 PK04_093262 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N07 compound treatment 277800.0 80800.0 5.51 276080.0 79600.0 5.92 8.0823 0.9993 3187544 PK04_093263 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(CC=C)C3=O)[C@H](O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N08 compound treatment 263600.0 66600.0 4.54 259040.0 62500.0 4.65 6.501 0.9999 3068600 PK04_093264 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N09 mock treatment 212200.0 15200.0 1.04 209800.0 13300.0 0.99 1.4317 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N10 mock treatment 207920.0 10900.0 0.74 211040.0 14500.0 1.08 1.2906 0.9834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N11 compound treatment 274920.0 77900.0 5.31 272240.0 75700.0 5.64 7.7414 0.9996 3187545 PK04_093265 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N12 compound treatment 249320.0 52300.0 3.57 240040.0 43500.0 3.24 4.8126 0.9988 3187546 PK04_093266 COCCCNC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N13 mock treatment 214840.0 17800.0 1.22 211520.0 15000.0 1.12 1.6495 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N14 mock treatment 207000.0 10000.0 0.68 204160.0 7640.0 0.57 0.8842 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N15 compound treatment 313480.0 116000.0 7.94 303480.0 107000.0 7.96 11.2444 1.0 3068603 PK04_093267 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3N(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N16 compound treatment 216720.0 19700.0 1.34 218840.0 22300.0 1.66 2.1253 0.9945 3187547 PK04_093268 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N17 compound treatment 294880.0 97900.0 6.67 286600.0 90100.0 6.7 9.4594 1.0 3068605 PK04_093269 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N18 compound treatment 260080.0 63100.0 4.3 252640.0 56100.0 4.18 5.9945 0.9999 3187548 PK04_093270 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N19 compound treatment 239720.0 42700.0 2.91 240000.0 43500.0 3.24 4.3477 0.9986 3068607 PK04_093271 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N20 compound treatment 228120.0 31100.0 2.12 237680.0 41200.0 3.06 3.6664 0.9839 3186297 PK04_093272 NC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N21 compound treatment 293440.0 96400.0 6.57 286160.0 89600.0 6.67 9.3668 1.0 3186298 PK04_093273 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(CC=C)C3=O)[C@@H](O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N22 compound treatment 197520.0 517.0 0.04 194080.0 -2440.0 -0.18 -0.1033 -0.5593 3068610 PK04_093274 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N23 compound treatment 266600.0 69600.0 4.74 242120.0 45600.0 3.39 5.7551 0.9865 3068635 PK04_093275 CC(=O)N1Cc2ccccc2C[C@]3(N=C(O[C@@H]3c4ccccc4)c5ccc(OCCCO)cc5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 N24 compound treatment 232920.0 35900.0 2.45 225520.0 29000.0 2.16 3.2579 0.998 3186299 PK04_093276 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O01 compound treatment 236200.0 39200.0 2.67 234760.0 38200.0 2.85 3.9023 0.9995 3068638 PK04_093277 COC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O02 compound treatment 223040.0 26000.0 1.78 233080.0 36600.0 2.72 3.1794 0.9786 3186300 PK04_093278 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O03 compound treatment 241400.0 44400.0 3.03 251920.0 55400.0 4.12 5.056 0.9884 3068640 PK04_093279 COC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O04 compound treatment 225520.0 28500.0 1.94 234440.0 37900.0 2.82 3.3706 0.9834 3186301 PK04_093280 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O05 compound treatment 217040.0 20000.0 1.37 211800.0 15300.0 1.14 1.7703 0.9959 3068642 PK04_093281 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O06 compound treatment 206440.0 9440.0 0.64 206120.0 9600.0 0.71 0.9603 0.9986 3186302 PK04_093282 COCCCNC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O07 compound treatment 203640.0 6640.0 0.45 213840.0 17300.0 1.29 1.2316 0.9014 3186303 PK04_093283 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O08 compound treatment 261520.0 64500.0 4.4 253480.0 57000.0 4.24 6.1081 0.9998 3068645 PK04_093284 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O09 compound treatment 249640.0 52600.0 3.59 243640.0 47100.0 3.51 5.0175 0.9999 3186304 PK04_093285 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O10 compound treatment 250680.0 53700.0 3.66 236840.0 40300.0 3.0 4.7098 0.9952 3186305 PK04_093286 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O11 mock treatment 198120.0 1120.0 0.08 201240.0 4720.0 0.35 0.3024 0.8408 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O12 mock treatment 201520.0 4520.0 0.31 197360.0 843.0 0.06 0.2621 0.8341 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O13 compound treatment 243800.0 46800.0 3.19 245560.0 49000.0 3.65 4.837 0.9977 3068648 PK04_093287 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O14 compound treatment 203040.0 6040.0 0.41 207320.0 10800.0 0.8 0.8596 0.9516 3186306 PK04_093288 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O15 compound treatment 222600.0 25600.0 1.75 243840.0 47300.0 3.52 3.7245 0.9475 3068650 PK04_093289 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O16 compound treatment 228960.0 32000.0 2.18 248560.0 52000.0 3.87 4.2795 0.963 3186307 PK04_093290 CN(C)C(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O17 compound treatment 278000.0 81000.0 5.52 270880.0 74400.0 5.53 7.8183 1.0 3186308 PK04_093291 COC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O18 compound treatment 236680.0 39700.0 2.71 227000.0 30500.0 2.27 3.517 0.9962 3068652 PK04_093292 COCCCNC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O19 compound treatment 236560.0 39600.0 2.7 242360.0 45800.0 3.41 4.3196 0.9932 3186309 PK04_093293 COC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O20 compound treatment 261840.0 64800.0 4.42 265760.0 69200.0 5.15 6.7698 0.9971 3068654 PK04_093294 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O21 compound treatment 250280.0 53300.0 3.63 242200.0 45700.0 3.4 4.9726 0.9995 3186310 PK04_093295 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O22 compound treatment 196120.0 -883.0 -0.06 194000.0 -2520.0 -0.19 -0.175 -0.8896 3186311 PK04_093296 NC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O23 compound treatment 211280.0 14300.0 0.97 218800.0 22300.0 1.66 1.861 0.9677 3068656 PK04_093297 COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 O24 compound treatment 253880.0 56900.0 3.88 215600.0 19100.0 1.42 3.7462 0.9072 3186312 PK04_093298 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P01 compound treatment 278640.0 81600.0 5.57 269240.0 72700.0 5.41 7.7628 0.9999 3186313 PK04_093299 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P02 compound treatment 274640.0 77600.0 5.29 269240.0 72700.0 5.41 7.57 0.9999 3186314 PK04_093300 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P03 compound treatment 263200.0 66200.0 4.51 259280.0 62800.0 4.67 6.4943 0.9999 3067960 PK04_093301 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P04 compound treatment 280480.0 83500.0 5.69 276680.0 80200.0 5.97 8.2431 0.9997 3186315 PK04_093302 CN(C)C(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P05 compound treatment 274400.0 77400.0 5.28 268800.0 72300.0 5.38 7.5353 1.0 3186316 PK04_093303 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P06 compound treatment 245360.0 48400.0 3.3 241640.0 45100.0 3.36 4.7059 1.0 3067963 PK04_093304 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P07 compound treatment 215920.0 18900.0 1.29 217760.0 21200.0 1.58 2.0299 0.9949 3186317 PK04_093305 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P08 compound treatment 217400.0 20400.0 1.39 212880.0 16400.0 1.22 1.8445 0.9978 3186362 PK04_093306 COCCCNC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P09 compound treatment 330960.0 134000.0 9.13 316200.0 120000.0 8.91 12.7565 0.9999 3067965 PK04_093307 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P10 compound treatment 194040.0 -2960.0 -0.2 198200.0 1680.0 0.13 -0.0543 -0.2283 3186363 PK04_093308 COCCCNC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P11 mock treatment 189680.0 -7320.0 -0.5 197520.0 1000.0 0.07 -0.3002 -0.5948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P12 mock treatment 198560.0 1560.0 0.11 197120.0 603.0 0.04 0.1068 0.9267 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P13 compound treatment 298320.0 101000.0 6.91 285760.0 89200.0 6.64 9.581 0.9998 3186364 PK04_093309 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P14 compound treatment 203400.0 6400.0 0.44 209440.0 12900.0 0.96 0.9885 0.936 3067968 PK04_093310 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P15 compound treatment 272920.0 75900.0 5.18 280480.0 84000.0 6.25 8.0786 0.9956 3186365 PK04_093311 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5N(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P16 compound treatment 206000.0 9000.0 0.61 213440.0 16900.0 1.26 1.3244 0.9453 3186366 PK04_093312 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P17 compound treatment 287920.0 90900.0 6.2 283160.0 86600.0 6.45 8.9428 0.9998 3067970 PK04_093313 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(CC=C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P18 compound treatment 206200.0 9200.0 0.63 198040.0 1520.0 0.11 0.5235 0.8216 3186367 PK04_093314 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P19 compound treatment 270760.0 73800.0 5.03 263440.0 66900.0 4.98 7.0777 1.0 3067972 PK04_093315 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(CC=C)C3=O)[C@H](O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P20 compound treatment 225200.0 28200.0 1.92 225400.0 28900.0 2.15 2.8794 0.9984 3186368 PK04_093316 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P21 compound treatment 254440.0 57400.0 3.92 249320.0 52800.0 3.93 5.5478 1.0 3067974 PK04_093317 CC(=O)N1Cc2ccccc2C[C@@]3(N=C(O[C@H]3c4ccccc4)c5ccc(OCCCO)cc5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P22 compound treatment 184280.0 -12700.0 -0.87 187160.0 -9360.0 -0.7 -1.1058 -0.9941 3186369 PK04_093318 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P23 compound treatment 211400.0 14400.0 0.98 210240.0 13700.0 1.02 1.4163 0.9998 3067976 PK04_093319 CC(=O)N1Cc2ccccc2C[C@@]3(COC(=N3)c4ccc(OCCCO)cc4)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2093 P24 compound treatment 228120.0 31100.0 2.12 231960.0 35400.0 2.64 3.3654 0.9942 3186370 PK04_093320 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A01 compound treatment 197560.0 2480.0 0.17 188000.0 -6380.0 -0.47 -0.2162 -0.4292 3186371 PK04_094001 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A02 compound treatment 233920.0 38800.0 2.65 228840.0 34500.0 2.56 3.6859 0.9999 3067979 PK04_094002 COCCCNC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A03 compound treatment 181480.0 -13600.0 -0.93 227280.0 32900.0 2.45 1.0758 0.4108 3068002 PK04_094003 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A04 compound treatment 245720.0 50600.0 3.45 230760.0 36400.0 2.71 4.3559 0.9928 3186372 PK04_094004 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A05 compound treatment 193800.0 -1280.0 -0.09 196000.0 1620.0 0.12 0.0235 0.1578 3068007 PK04_094005 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A06 compound treatment 203040.0 7960.0 0.54 196560.0 2180.0 0.16 0.4985 0.8803 3186373 PK04_094006 CN(C)C(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A07 compound treatment 204160.0 9080.0 0.62 201760.0 7380.0 0.55 0.8261 0.9982 3186374 PK04_094007 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A08 compound treatment 252240.0 57200.0 3.9 253440.0 59100.0 4.4 5.8638 0.9982 3068010 PK04_094008 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A09 compound treatment 182160.0 -12900.0 -0.88 180960.0 -13400.0 -1.0 -1.3291 -0.9981 3186375 PK04_094009 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A10 compound treatment 227480.0 32400.0 2.21 220920.0 26500.0 1.98 2.9587 0.9985 3068013 PK04_094010 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A11 compound treatment 246680.0 51600.0 3.52 241760.0 47400.0 3.53 4.981 1.0 3186376 PK04_094011 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A12 compound treatment 236840.0 41800.0 2.85 234240.0 39900.0 2.97 4.1109 0.9998 3186377 PK04_094012 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A13 mock treatment 182840.0 -12200.0 -0.83 181720.0 -12700.0 -0.94 -1.2564 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A14 mock treatment 178960.0 -16100.0 -1.1 179800.0 -14600.0 -1.08 -1.5444 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A15 compound treatment 208680.0 13600.0 0.93 204080.0 9700.0 0.72 1.1661 0.9924 3068016 PK04_094013 CN(C)C(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A16 compound treatment 220240.0 25200.0 1.72 216320.0 21900.0 1.63 2.3676 0.9997 3186378 PK04_094014 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A17 compound treatment 214560.0 19500.0 1.33 199800.0 5420.0 0.4 1.2243 0.8822 3068018 PK04_094015 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A18 compound treatment 198480.0 3400.0 0.23 193840.0 -537.0 -0.04 0.1355 0.5766 3186379 PK04_094016 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A19 compound treatment 202160.0 7080.0 0.48 199040.0 4660.0 0.35 0.5865 0.9869 3186380 PK04_094017 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A20 compound treatment 227560.0 32500.0 2.21 241080.0 46700.0 3.48 4.0235 0.9763 3068020 PK04_094018 NC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A21 compound treatment 187520.0 -7560.0 -0.52 182520.0 -11900.0 -0.88 -0.9886 -0.9673 3186381 PK04_094019 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A22 compound treatment 177600.0 -17500.0 -1.19 178960.0 -15400.0 -1.15 -1.6542 -0.9998 3186437 PK04_094020 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A23 compound treatment 193040.0 -2040.0 -0.14 207080.0 12700.0 0.95 0.57 0.5965 3068021 PK04_094021 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 A24 compound treatment 174440.0 -20600.0 -1.41 194720.0 343.0 0.03 -0.9771 -0.6942 3186438 PK04_094022 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B01 compound treatment 171880.0 -23200.0 -1.58 169640.0 -24700.0 -1.84 -2.4205 -0.9971 3186439 PK04_094023 CCCN1C(=O)[C@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B02 compound treatment 204880.0 9800.0 0.67 202320.0 7940.0 0.59 0.8903 0.9981 3089331 PK04_094024 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B03 compound treatment 255240.0 60200.0 4.1 246880.0 52500.0 3.91 5.6632 0.9997 3068022 PK04_094025 CCCN1C(=O)[C@]2(Cc3ccccc13)N=C(O[C@@H]2c4ccccc4)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B04 compound treatment 233880.0 38800.0 2.65 223680.0 29300.0 2.18 3.4125 0.9954 3089332 PK04_094026 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B05 compound treatment 262600.0 67500.0 4.6 247280.0 52900.0 3.94 6.039 0.997 3186440 PK04_094027 CCCN1C(=O)[C@@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B06 compound treatment 222760.0 27700.0 1.89 220280.0 25900.0 1.93 2.6974 0.9999 3000708 PK04_094028 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B07 compound treatment 244920.0 49800.0 3.4 235400.0 41000.0 3.05 4.5615 0.9986 3068023 PK04_094029 CN1C(=O)[C@]2(Cc3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B08 compound treatment 201400.0 6320.0 0.43 208200.0 13800.0 1.03 1.032 0.9253 3089333 PK04_094030 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B09 compound treatment 243800.0 48700.0 3.32 236920.0 42500.0 3.17 4.5875 0.9997 3186441 PK04_094031 CN1C(=O)[C@@]2(CC=C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B10 compound treatment 219600.0 24500.0 1.67 222360.0 28000.0 2.08 2.6546 0.9941 3089654 PK04_094032 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B11 compound treatment 282160.0 87100.0 5.94 265680.0 71300.0 5.31 7.9503 0.9984 3186442 PK04_094033 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B12 compound treatment 199400.0 4320.0 0.29 211240.0 16900.0 1.26 1.0955 0.8499 3089334 PK04_094034 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B13 mock treatment 181720.0 -13400.0 -0.91 180760.0 -13600.0 -1.01 -1.3609 -0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B14 mock treatment 178080.0 -17000.0 -1.16 186040.0 -8340.0 -0.62 -1.2585 -0.9571 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B15 compound treatment 258160.0 63100.0 4.3 242120.0 47700.0 3.55 5.5534 0.9955 3068024 PK04_094035 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B16 compound treatment 217840.0 22800.0 1.55 212600.0 18200.0 1.36 2.0561 0.9978 3000709 PK04_094036 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B17 compound treatment 248360.0 53300.0 3.63 240120.0 45700.0 3.4 4.9757 0.9995 3186443 PK04_094037 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B18 compound treatment 271560.0 76500.0 5.21 277120.0 82700.0 6.16 8.0414 0.9966 3089363 PK04_094038 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4)[C@H]1OC(=O)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B19 compound treatment 266680.0 71600.0 4.88 251960.0 57600.0 4.29 6.482 0.9979 3068025 PK04_094039 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B20 compound treatment 231280.0 36200.0 2.47 236600.0 42200.0 3.14 3.9671 0.9928 3089652 PK04_094040 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4)[C@H]1OC(=O)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B21 compound treatment 232880.0 37800.0 2.58 222040.0 27700.0 2.06 3.2779 0.9938 3186444 PK04_094041 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B22 compound treatment 190960.0 -4120.0 -0.28 188240.0 -6140.0 -0.46 -0.5218 -0.9728 3089653 PK04_094042 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4)[C@H]1OC(=O)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B23 compound treatment 228840.0 33800.0 2.3 230040.0 35700.0 2.65 3.5042 0.9975 3186445 PK04_094043 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 B24 compound treatment 267600.0 72500.0 4.94 263080.0 68700.0 5.11 7.1116 0.9999 3089657 PK04_094044 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C01 compound treatment 229080.0 34000.0 2.32 182040.0 -12300.0 -0.92 0.9896 0.397 3068026 PK04_094045 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C02 compound treatment 251040.0 56000.0 3.81 237320.0 42900.0 3.2 4.9576 0.9961 3068051 PK04_094046 CN(C)C(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C03 compound treatment 194040.0 -1040.0 -0.07 201080.0 6700.0 0.5 0.3025 0.6002 3068052 PK04_094047 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C04 compound treatment 190400.0 -4680.0 -0.32 186520.0 -7860.0 -0.58 -0.6393 -0.9595 3068053 PK04_094048 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)N3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C05 compound treatment 228080.0 33000.0 2.25 213240.0 18900.0 1.4 2.5834 0.9742 3068054 PK04_094049 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C06 compound treatment 231880.0 36800.0 2.51 222200.0 27800.0 2.07 3.2382 0.9955 3186446 PK04_094050 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C07 compound treatment 193880.0 -1200.0 -0.08 197680.0 3300.0 0.25 0.1158 0.4468 3068055 PK04_094051 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C08 compound treatment 192640.0 -2440.0 -0.17 193480.0 -897.0 -0.07 -0.165 -0.9194 3186447 PK04_094052 COCCCNC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C09 compound treatment 234720.0 39600.0 2.7 221960.0 27600.0 2.05 3.3624 0.9908 3068056 PK04_094053 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C10 compound treatment 229120.0 34000.0 2.32 223640.0 29300.0 2.18 3.1809 0.9995 3186448 PK04_094054 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C11 mock treatment 189080.0 -6000.0 -0.41 190240.0 -4140.0 -0.31 -0.5071 -0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C12 mock treatment 191040.0 -4040.0 -0.28 187440.0 -6940.0 -0.52 -0.56 -0.9568 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C13 compound treatment 194160.0 -924.0 -0.06 191040.0 -3340.0 -0.25 -0.2201 -0.8592 3186449 PK04_094055 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C14 compound treatment 210840.0 15800.0 1.07 205080.0 10700.0 0.8 1.3229 0.9892 3068057 PK04_094056 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C15 mock treatment 188440.0 -6640.0 -0.45 187080.0 -7300.0 -0.54 -0.7043 -0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C16 mock treatment 190360.0 -4720.0 -0.32 186800.0 -7580.0 -0.56 -0.6265 -0.9647 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C17 compound treatment 188200.0 -6880.0 -0.47 187680.0 -6700.0 -0.5 -0.6843 -0.9995 3186450 PK04_094057 NC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C18 compound treatment 226520.0 31400.0 2.14 217320.0 22900.0 1.71 2.7229 0.9937 3186451 PK04_094058 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C19 compound treatment 191320.0 -3760.0 -0.26 188520.0 -5860.0 -0.44 -0.4897 -0.9681 3068058 PK04_094059 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C20 compound treatment 220360.0 25300.0 1.72 215680.0 21300.0 1.59 2.3397 0.9991 3186452 PK04_094060 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C21 compound treatment 226240.0 31200.0 2.12 217440.0 23100.0 1.72 2.7158 0.9944 3068059 PK04_094061 NC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C22 compound treatment 224120.0 29000.0 1.98 219280.0 24900.0 1.85 2.7104 0.9995 3186453 PK04_094062 NC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C23 compound treatment 177000.0 -18100.0 -1.23 175640.0 -18700.0 -1.39 -1.8579 -0.9981 3186454 PK04_094063 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 C24 compound treatment 174560.0 -20500.0 -1.4 173520.0 -20900.0 -1.55 -2.0871 -0.9987 3068060 PK04_094064 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D01 compound treatment 237520.0 42400.0 2.89 225640.0 31300.0 2.33 3.6911 0.9942 3186455 PK04_094065 CN1C(=O)[C@@]2(CCC(=O)OC(C)(C)C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D02 compound treatment 325840.0 131000.0 8.91 317480.0 123000.0 9.16 12.7822 0.9999 3000713 PK04_094066 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D03 compound treatment 250520.0 55400.0 3.78 234480.0 40100.0 2.98 4.783 0.9932 3186456 PK04_094067 CCCN1C(=O)[C@@]2(CCC(=O)OC(C)(C)C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D04 compound treatment 327320.0 132000.0 9.02 335400.0 141000.0 10.5 13.7966 0.9971 3089658 PK04_094068 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D05 compound treatment 268800.0 73700.0 5.03 255080.0 60700.0 4.52 6.7484 0.9986 3068061 PK04_094069 CCCN1C(=O)[C@@]2(Cc3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D06 compound treatment 359200.0 164000.0 11.19 343280.0 149000.0 11.08 15.7482 1.0 3089659 PK04_094070 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D07 compound treatment 224760.0 29700.0 2.02 221040.0 26700.0 1.98 2.8339 1.0 3186457 PK04_094071 CCCN1C(=O)[C@]2(CCC(=O)OC(C)(C)C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D08 compound treatment 337560.0 142000.0 9.71 325680.0 131000.0 9.77 13.7787 1.0 3089664 PK04_094072 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D09 compound treatment 227520.0 32400.0 2.21 222960.0 28600.0 2.13 3.068 0.9998 3068062 PK04_094073 CCCN1C(=O)[C@@]2(CC=C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D10 compound treatment 289880.0 94800.0 6.46 286520.0 92100.0 6.86 9.4193 0.9996 3000714 PK04_094074 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D11 mock treatment 187200.0 -7880.0 -0.54 186960.0 -7420.0 -0.55 -0.7704 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D12 mock treatment 192280.0 -2800.0 -0.19 184640.0 -9740.0 -0.72 -0.6476 -0.8641 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D13 compound treatment 243920.0 48800.0 3.33 236600.0 42200.0 3.14 4.5764 0.9996 3186504 PK04_094075 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D14 compound treatment 317000.0 122000.0 8.31 330240.0 136000.0 10.11 13.0276 0.9953 3089660 PK04_094076 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D15 mock treatment 193160.0 -1920.0 -0.13 190240.0 -4140.0 -0.31 -0.3105 -0.9277 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D16 mock treatment 189400.0 -5680.0 -0.39 189440.0 -4940.0 -0.37 -0.5338 -0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D17 compound treatment 253800.0 58700.0 4.0 249920.0 55500.0 4.13 5.7537 0.9999 3186505 PK04_094077 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(Cc5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D18 compound treatment 371160.0 176000.0 12.0 371600.0 177000.0 13.19 17.8152 0.9989 3000715 PK04_094078 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@H]1OC(=O)Nc6ccc7OCOc7c6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D19 compound treatment 249120.0 54000.0 3.68 246680.0 52300.0 3.89 5.3576 0.9996 3068063 PK04_094079 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D20 compound treatment 310640.0 116000.0 7.88 309480.0 115000.0 8.57 11.6284 0.9991 3089662 PK04_094080 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@H]1OC(=O)Nc6ccc7OCOc7c6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D21 compound treatment 264040.0 69000.0 4.7 259640.0 65300.0 4.86 6.7589 0.9999 3186506 PK04_094081 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4N(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D22 compound treatment 266080.0 71000.0 4.84 263840.0 69500.0 5.17 7.0783 0.9995 3000716 PK04_094082 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@H]1OC(=O)Nc6ccc7OCOc7c6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D23 compound treatment 245320.0 50200.0 3.42 259840.0 65500.0 4.87 5.867 0.9851 3068064 PK04_094083 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3N(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 D24 compound treatment 190880.0 -4200.0 -0.29 195560.0 1180.0 0.09 -0.1404 -0.4682 3000811 PK04_094084 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E01 mock treatment 192680.0 -2400.0 -0.16 186360.0 -8020.0 -0.6 -0.5378 -0.8691 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E02 mock treatment 185760.0 -9320.0 -0.64 191520.0 -2860.0 -0.21 -0.5998 -0.8949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E03 compound treatment 219120.0 24000.0 1.64 213480.0 19100.0 1.42 2.1641 0.9975 3186507 PK04_094085 CN(C)C(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E04 compound treatment 239400.0 44300.0 3.02 227760.0 33400.0 2.48 3.8933 0.9953 3186508 PK04_094086 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E05 compound treatment 198680.0 3600.0 0.25 199160.0 4780.0 0.36 0.4251 0.9834 3068065 PK04_094087 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E06 compound treatment 261320.0 66200.0 4.52 257880.0 63500.0 4.73 6.5352 0.9997 3186509 PK04_094088 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E07 compound treatment 200000.0 4920.0 0.34 200000.0 5620.0 0.42 0.5329 0.9939 3068066 PK04_094089 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E08 compound treatment 215800.0 20700.0 1.41 213120.0 18700.0 1.39 1.9851 1.0 3186510 PK04_094090 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E09 mock treatment 194440.0 -644.0 -0.04 198200.0 3820.0 0.28 0.1702 0.5911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E10 mock treatment 197040.0 1960.0 0.13 196760.0 2380.0 0.18 0.2197 0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E11 compound treatment 243320.0 48200.0 3.29 235800.0 41400.0 3.08 4.5054 0.9995 3186511 PK04_094091 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E12 compound treatment 199800.0 4720.0 0.32 196120.0 1740.0 0.13 0.3191 0.9203 3068067 PK04_094092 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E13 compound treatment 218480.0 23400.0 1.6 211200.0 16800.0 1.25 2.0133 0.9928 3186512 PK04_094093 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E14 compound treatment 244280.0 49200.0 3.35 231440.0 37100.0 2.76 4.3222 0.9953 3068068 PK04_094094 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E15 compound treatment 200400.0 5320.0 0.36 206520.0 12100.0 0.9 0.8954 0.9195 3186513 PK04_094095 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E16 compound treatment 221560.0 26500.0 1.81 219440.0 25100.0 1.87 2.5954 0.9999 3068069 PK04_094096 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E17 mock treatment 196880.0 1800.0 0.12 199120.0 4740.0 0.35 0.3362 0.8998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E18 mock treatment 192160.0 -2920.0 -0.2 202000.0 7620.0 0.57 0.2602 0.4327 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E19 compound treatment 199120.0 4040.0 0.28 195040.0 663.0 0.05 0.2295 0.8208 3186514 PK04_094097 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E20 compound treatment 221640.0 26600.0 1.81 216840.0 22500.0 1.67 2.4624 0.9992 3186515 PK04_094098 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E21 compound treatment 270720.0 75600.0 5.16 267720.0 73300.0 5.46 7.5062 0.9996 3068070 PK04_094099 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E22 compound treatment 259440.0 64400.0 4.39 248800.0 54400.0 4.05 5.9667 0.9992 3186516 PK04_094100 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E23 compound treatment 188520.0 -6560.0 -0.45 191880.0 -2500.0 -0.19 -0.4478 -0.9242 3068071 PK04_094101 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 E24 compound treatment 226480.0 31400.0 2.14 219640.0 25300.0 1.88 2.8431 0.9979 3186517 PK04_094102 COCCCNC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F01 mock treatment 183160.0 -11900.0 -0.81 182200.0 -12200.0 -0.91 -1.2157 -0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F02 mock treatment 190560.0 -4520.0 -0.31 188120.0 -6260.0 -0.47 -0.5474 -0.98 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F03 compound treatment 246000.0 50900.0 3.47 242840.0 48500.0 3.61 5.0051 0.9998 3068072 PK04_094103 CN1C(=O)[C@]2(CCC(=O)OC(C)(C)C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F04 compound treatment 286520.0 91400.0 6.23 278480.0 84100.0 6.26 8.8341 1.0 3000813 PK04_094104 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]2OC(=O)Nc5ccccc5c6ccccc6)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F05 compound treatment 236360.0 41300.0 2.81 231040.0 36700.0 2.73 3.9194 0.9999 3186518 PK04_094105 CN1C(=O)[C@]2(CC=C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F06 compound treatment 246480.0 51400.0 3.5 246520.0 52100.0 3.88 5.2219 0.9987 3000814 PK04_094106 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F07 compound treatment 255640.0 60600.0 4.13 255880.0 61500.0 4.58 6.1561 0.9987 3186519 PK04_094107 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(C(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F08 compound treatment 319680.0 125000.0 8.49 329320.0 135000.0 10.04 13.1083 0.9965 3089667 PK04_094108 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F09 mock treatment 195440.0 356.0 0.02 198600.0 4220.0 0.31 0.2394 0.7595 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F10 mock treatment 195480.0 396.0 0.03 195360.0 983.0 0.07 0.0708 0.9082 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F11 compound treatment 245760.0 50700.0 3.45 247560.0 53200.0 3.96 5.2419 0.9977 3068073 PK04_094109 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(C(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F12 compound treatment 224440.0 29400.0 2.0 226480.0 32100.0 2.39 3.1047 0.9961 3089654 PK04_094110 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F13 compound treatment 276040.0 81000.0 5.52 267280.0 72900.0 5.43 7.7395 1.0 3186520 PK04_094111 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(C(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F14 compound treatment 273680.0 78600.0 5.36 266520.0 72100.0 5.37 7.5857 1.0 3089708 PK04_094112 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F15 compound treatment 281680.0 86600.0 5.9 265920.0 71500.0 5.32 7.9398 0.9987 3186521 PK04_094113 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(C(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F16 compound treatment 217720.0 22600.0 1.54 208560.0 14200.0 1.06 1.8377 0.9828 3000817 PK04_094114 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F17 mock treatment 194200.0 -884.0 -0.06 197240.0 2860.0 0.21 0.1081 0.488 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F18 mock treatment 196160.0 1080.0 0.07 198880.0 4500.0 0.34 0.2889 0.842 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F19 compound treatment 254240.0 59200.0 4.03 242680.0 48300.0 3.6 5.3939 0.9984 3068074 PK04_094115 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F20 compound treatment 340600.0 146000.0 9.92 348560.0 154000.0 11.48 15.1294 0.9974 3089709 PK04_094116 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F21 compound treatment 232320.0 37200.0 2.54 232800.0 38400.0 2.86 3.8172 0.9982 3186522 PK04_094117 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F22 compound treatment 231800.0 36700.0 2.5 235560.0 41200.0 3.07 3.9374 0.9949 3000821 PK04_094118 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F23 compound treatment 253560.0 58500.0 3.99 256640.0 62300.0 4.63 6.0958 0.9972 3186523 PK04_094119 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 F24 compound treatment 180520.0 -14600.0 -0.99 207040.0 12700.0 0.94 -0.0357 -0.026 3089711 PK04_094120 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G01 compound treatment 227520.0 32400.0 2.21 225080.0 30700.0 2.29 3.1795 0.9999 3068075 PK04_094121 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G02 compound treatment 191920.0 -3160.0 -0.22 192400.0 -1980.0 -0.15 -0.2566 -0.9826 3186524 PK04_094122 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G03 mock treatment 196320.0 1240.0 0.08 195440.0 1060.0 0.08 0.1155 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G04 mock treatment 204320.0 9240.0 0.63 203680.0 9300.0 0.69 0.9349 0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G05 compound treatment 225760.0 30700.0 2.09 227160.0 32800.0 2.44 3.2042 0.9971 3186575 PK04_094123 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G06 compound treatment 219560.0 24500.0 1.67 221760.0 27400.0 2.04 2.6211 0.9951 3186576 PK04_094124 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G07 compound treatment 201000.0 5920.0 0.4 211160.0 16800.0 1.25 1.1685 0.8902 3068110 PK04_094125 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G08 compound treatment 215560.0 20500.0 1.4 215120.0 20700.0 1.54 2.0788 0.9987 3186577 PK04_094126 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G09 compound treatment 223840.0 28800.0 1.96 222440.0 28100.0 2.09 2.8632 0.9995 3068111 PK04_094127 COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G10 compound treatment 199480.0 4400.0 0.3 207760.0 13400.0 1.0 0.9163 0.8809 3186578 PK04_094128 CN(C)C(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G11 compound treatment 213920.0 18800.0 1.28 212320.0 17900.0 1.34 1.8524 0.9998 3186579 PK04_094129 COCCCNC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G12 compound treatment 210640.0 15600.0 1.06 208120.0 13700.0 1.02 1.4732 0.9998 3068112 PK04_094130 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G13 compound treatment 203880.0 8800.0 0.6 205000.0 10600.0 0.79 0.9831 0.9907 3186580 PK04_094131 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G14 compound treatment 270640.0 75600.0 5.15 253960.0 59600.0 4.43 6.7782 0.9972 3186581 PK04_094132 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G15 compound treatment 223360.0 28300.0 1.93 221560.0 27200.0 2.02 2.7937 0.9997 3068113 PK04_094133 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G16 compound treatment 232840.0 37800.0 2.57 221760.0 27400.0 2.04 3.2613 0.9933 3186582 PK04_094134 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G17 compound treatment 199880.0 4800.0 0.33 197120.0 2740.0 0.2 0.3756 0.9743 3186583 PK04_094135 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G18 compound treatment 266960.0 71900.0 4.9 259400.0 65000.0 4.84 6.8871 1.0 3068114 PK04_094136 NC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G19 mock treatment 200640.0 5560.0 0.38 199080.0 4700.0 0.35 0.5154 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G20 mock treatment 197360.0 2280.0 0.16 201920.0 7540.0 0.56 0.5067 0.8699 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G21 compound treatment 202520.0 7440.0 0.51 204880.0 10500.0 0.78 0.9112 0.978 3186584 PK04_094137 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G22 compound treatment 199880.0 4800.0 0.33 206400.0 12000.0 0.89 0.864 0.9068 3068115 PK04_094138 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G23 compound treatment 217000.0 21900.0 1.49 216280.0 21900.0 1.63 2.2093 0.9991 3186585 PK04_094139 CN(C)C(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 G24 compound treatment 186280.0 -8800.0 -0.6 183320.0 -11100.0 -0.82 -1.0063 -0.988 3186586 PK04_094140 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H01 compound treatment 263240.0 68200.0 4.65 246160.0 51800.0 3.85 6.0109 0.9957 3068116 PK04_094141 CCCN1C(=O)[C@]2(Cc3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H02 compound treatment 223520.0 28400.0 1.94 217080.0 22700.0 1.69 2.5657 0.9977 3000914 PK04_094142 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H03 mock treatment 197240.0 2160.0 0.15 194200.0 -177.0 -0.01 0.0946 0.6412 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H04 mock treatment 196440.0 1360.0 0.09 193560.0 -817.0 -0.06 0.0224 0.2023 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H05 compound treatment 235240.0 40200.0 2.74 232080.0 37700.0 2.81 3.9201 0.9999 3068117 PK04_094143 CCCN1C(=O)[C@]2(CC=C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H06 compound treatment 244880.0 49800.0 3.39 232040.0 37700.0 2.8 4.3827 0.9955 3089723 PK04_094144 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H07 compound treatment 265240.0 70200.0 4.78 251080.0 56700.0 4.22 6.3663 0.9981 3186589 PK04_094145 CN1C(=O)[C@@]2(Cc3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H08 compound treatment 224240.0 29200.0 1.99 218960.0 24600.0 1.83 2.6993 0.9991 3089724 PK04_094146 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H09 compound treatment 251120.0 56000.0 3.82 248680.0 54300.0 4.04 5.5593 0.9996 3186590 PK04_094147 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(C(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H10 compound treatment 239720.0 44600.0 3.04 230600.0 36200.0 2.7 4.0582 0.9982 3000917 PK04_094148 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H11 compound treatment 242120.0 47000.0 3.21 244640.0 50300.0 3.74 4.9128 0.9971 3068119 PK04_094149 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(C(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H12 compound treatment 245480.0 50400.0 3.44 245640.0 51300.0 3.82 5.1274 0.9986 3089768 PK04_094150 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H13 compound treatment 270280.0 75200.0 5.13 269240.0 74900.0 5.57 7.565 0.9991 3186593 PK04_094151 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(C(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H14 compound treatment 206240.0 11200.0 0.76 198160.0 3780.0 0.28 0.7369 0.9086 3089763 PK04_094152 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H15 compound treatment 257680.0 62600.0 4.27 244600.0 50200.0 3.74 5.6608 0.9978 3186594 PK04_094153 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H16 compound treatment 220520.0 25400.0 1.73 225320.0 30900.0 2.3 2.8547 0.9902 3089764 PK04_094154 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H17 compound treatment 292320.0 97200.0 6.63 266840.0 72500.0 5.39 8.5012 0.9948 3068121 PK04_094155 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(C(=O)c5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H18 compound treatment 257360.0 62300.0 4.25 265760.0 71400.0 5.31 6.759 0.9938 3000919 PK04_094156 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4)[C@@H]1OC(=O)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H19 mock treatment 195560.0 476.0 0.03 194120.0 -257.0 -0.02 0.0094 0.2505 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H20 mock treatment 195360.0 276.0 0.02 192920.0 -1460.0 -0.11 -0.0634 -0.5757 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H21 compound treatment 267840.0 72800.0 4.96 261400.0 67000.0 4.99 7.0347 1.0 3068122 PK04_094157 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3N(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H22 compound treatment 202080.0 7000.0 0.48 216480.0 22100.0 1.65 1.5005 0.876 3089766 PK04_094158 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4)[C@@H]1OC(=O)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H23 compound treatment 207840.0 12800.0 0.87 228880.0 34500.0 2.57 2.4308 0.8966 3068123 PK04_094159 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 H24 compound treatment 228480.0 33400.0 2.28 280200.0 85800.0 6.39 6.1267 0.9035 3089769 PK04_094160 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I01 compound treatment 208200.0 13100.0 0.89 200400.0 6020.0 0.45 0.9493 0.949 3186651 PK04_094161 COCCCNC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I02 compound treatment 197040.0 1960.0 0.13 191880.0 -2500.0 -0.19 -0.0371 -0.1622 3068124 PK04_094162 COCCCNC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I03 compound treatment 268960.0 73900.0 5.04 262320.0 67900.0 5.06 7.1371 1.0 3186652 PK04_094163 NC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I04 compound treatment 228880.0 33800.0 2.3 227360.0 33000.0 2.45 3.3651 0.9995 3068125 PK04_094164 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I05 mock treatment 200120.0 5040.0 0.34 202440.0 8060.0 0.6 0.6671 0.9649 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I06 mock treatment 200640.0 5560.0 0.38 201760.0 7380.0 0.55 0.6564 0.9835 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I07 compound treatment 226200.0 31100.0 2.12 230240.0 35900.0 2.67 3.3875 0.9935 3186653 PK04_094165 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I08 compound treatment 198520.0 3440.0 0.23 200240.0 5860.0 0.44 0.4742 0.9575 3068126 PK04_094166 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I09 compound treatment 203160.0 8080.0 0.55 200200.0 5820.0 0.43 0.6958 0.993 3186654 PK04_094167 COCCCNC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I10 compound treatment 200440.0 5360.0 0.37 201040.0 6660.0 0.5 0.6089 0.9887 3068572 PK04_094168 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I11 compound treatment 247440.0 52400.0 3.57 249520.0 55100.0 4.1 5.4261 0.9976 3186655 PK04_094169 COCCCNC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I12 compound treatment 268040.0 73000.0 4.97 270920.0 76500.0 5.7 7.5454 0.9977 3186656 PK04_094170 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I13 compound treatment 235680.0 40600.0 2.77 227400.0 33000.0 2.46 3.695 0.9982 3068573 PK04_094171 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I14 compound treatment 225120.0 30000.0 2.05 213480.0 19100.0 1.42 2.4534 0.9841 3186657 PK04_094172 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I15 compound treatment 244120.0 49000.0 3.34 238200.0 43800.0 3.26 4.6703 0.9999 3068574 PK04_094173 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I16 compound treatment 258160.0 63100.0 4.3 244240.0 49900.0 3.71 5.665 0.9973 3186658 PK04_094174 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I17 compound treatment 267680.0 72600.0 4.95 249880.0 55500.0 4.13 6.4207 0.996 3186659 PK04_094175 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I18 compound treatment 265440.0 70400.0 4.8 256240.0 61900.0 4.6 6.6475 0.9998 3068575 PK04_094176 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I19 compound treatment 195400.0 316.0 0.02 200120.0 5740.0 0.43 0.3175 0.7418 3186660 PK04_094177 CN(C)C(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I20 compound treatment 234320.0 39200.0 2.68 253440.0 59100.0 4.4 4.9999 0.9716 3068577 PK04_094178 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I21 mock treatment 195120.0 36.3 0.0 196080.0 1700.0 0.13 0.0914 0.7208 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I22 mock treatment 189400.0 -5680.0 -0.39 186400.0 -7980.0 -0.59 -0.6938 -0.9786 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I23 compound treatment 191360.0 -3720.0 -0.25 192600.0 -1780.0 -0.13 -0.273 -0.9538 3186661 PK04_094179 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 I24 compound treatment 187360.0 -7720.0 -0.53 195080.0 703.0 0.05 -0.3353 -0.6337 3186662 PK04_094180 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J01 compound treatment 261680.0 66600.0 4.54 252040.0 57700.0 4.29 6.2452 0.9996 3068611 PK04_094181 CN1C(=O)[C@@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J02 compound treatment 328000.0 133000.0 9.06 317320.0 123000.0 9.15 12.8779 1.0 3089770 PK04_094182 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J03 compound treatment 267680.0 72600.0 4.95 259440.0 65100.0 4.84 6.9239 0.9999 3068612 PK04_094183 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J04 compound treatment 340920.0 146000.0 9.94 333880.0 140000.0 10.38 14.3723 0.9998 3001007 PK04_094184 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J05 mock treatment 198120.0 3040.0 0.21 200640.0 6260.0 0.47 0.476 0.9332 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J06 mock treatment 197120.0 2040.0 0.14 198320.0 3940.0 0.29 0.3057 0.9416 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J07 compound treatment 265760.0 70700.0 4.82 265440.0 71100.0 5.29 7.1471 0.9989 3186665 PK04_094185 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J08 compound treatment 296680.0 102000.0 6.93 284520.0 90100.0 6.71 9.6418 0.9999 3089771 PK04_094186 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J09 compound treatment 263680.0 68600.0 4.68 264480.0 70100.0 5.22 6.9963 0.9985 3186666 PK04_094187 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(C(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J10 compound treatment 289520.0 94400.0 6.44 293800.0 99400.0 7.4 9.785 0.9976 3089776 PK04_094188 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J11 compound treatment 215280.0 20200.0 1.38 210120.0 15700.0 1.17 1.8022 0.9968 3068615 PK04_094189 CCCN1C(=O)[C@]2(COC(=N2)c3ccc(OCCCO)cc3)Cc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J12 compound treatment 348080.0 153000.0 10.43 352880.0 159000.0 11.8 15.7174 0.9981 3001011 PK04_094190 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J13 compound treatment 260080.0 65000.0 4.43 249520.0 55100.0 4.1 6.0354 0.9993 3068616 PK04_094191 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J14 compound treatment 342160.0 147000.0 10.03 326920.0 133000.0 9.86 14.0658 1.0 3089772 PK04_094192 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J15 compound treatment 274000.0 78900.0 5.38 274000.0 79600.0 5.93 7.9948 0.9988 3068617 PK04_094193 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(C(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J16 compound treatment 353480.0 158000.0 10.8 338600.0 144000.0 10.73 15.2262 1.0 3089773 PK04_094194 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@@H]1OC(=O)Nc6ccc7OCOc7c6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J17 compound treatment 291240.0 96200.0 6.56 286880.0 92500.0 6.88 9.5038 0.9997 3186732 PK04_094195 CN1C(=O)[C@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J18 compound treatment 309880.0 115000.0 7.83 305480.0 111000.0 8.27 11.3812 0.9996 3089774 PK04_094196 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@@H]1OC(=O)Nc6ccc7OCOc7c6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J19 compound treatment 257480.0 62400.0 4.25 250800.0 56400.0 4.2 5.9774 1.0 3186733 PK04_094197 CCCN1C(=O)[C@@]2(Cc3ccccc13)N=C(O[C@H]2c4ccccc4)c5ccc(OCCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J20 compound treatment 238960.0 43900.0 2.99 252880.0 58500.0 4.35 5.1941 0.9832 3089775 PK04_094198 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@@H]1OC(=O)Nc6ccc7OCOc7c6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J21 mock treatment 194480.0 -604.0 -0.04 191960.0 -2420.0 -0.18 -0.1563 -0.847 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J22 mock treatment 187960.0 -7120.0 -0.49 187080.0 -7300.0 -0.54 -0.7274 -0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J23 compound treatment 215240.0 20200.0 1.37 219480.0 25100.0 1.87 2.2928 0.9886 3068619 PK04_094199 COC(=O)C1ON(C(=N1)c2ccc(OCCCO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 J24 compound treatment 222240.0 27200.0 1.85 227280.0 32900.0 2.45 3.0408 0.9905 3089828 PK04_094200 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K01 compound treatment 236000.0 40900.0 2.79 235360.0 41000.0 3.05 4.1294 0.999 3068620 PK04_094201 COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K02 compound treatment 240480.0 45400.0 3.09 238800.0 44400.0 3.31 4.5264 0.9995 3186736 PK04_094202 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K03 compound treatment 239920.0 44800.0 3.06 230640.0 36300.0 2.7 4.0699 0.9981 3186737 PK04_094203 CN(C)C(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K04 compound treatment 207840.0 12800.0 0.87 202880.0 8500.0 0.63 1.0625 0.9878 3068660 PK04_094204 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K05 compound treatment 245280.0 50200.0 3.42 252800.0 58400.0 4.35 5.4946 0.993 3186738 PK04_094205 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K06 compound treatment 210560.0 15500.0 1.06 207880.0 13500.0 1.0 1.4567 0.9997 3068661 PK04_094206 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K07 mock treatment 208040.0 13000.0 0.88 205440.0 11100.0 0.82 1.2068 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K08 mock treatment 202920.0 7840.0 0.53 200440.0 6060.0 0.45 0.6969 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K09 compound treatment 238480.0 43400.0 2.96 241960.0 47600.0 3.54 4.5963 0.996 3186739 PK04_094207 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K10 compound treatment 208280.0 13200.0 0.9 211760.0 17400.0 1.29 1.551 0.9842 3186740 PK04_094208 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K11 compound treatment 251000.0 55900.0 3.81 245560.0 51200.0 3.81 5.3893 1.0 3068664 PK04_094209 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K12 compound treatment 221000.0 25900.0 1.77 215920.0 21500.0 1.6 2.3831 0.9988 3186741 PK04_094210 COCCCNC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K13 compound treatment 248200.0 53100.0 3.62 248560.0 54200.0 4.03 5.4122 0.9986 3068666 PK04_094211 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K14 compound treatment 234200.0 39100.0 2.67 233080.0 38700.0 2.88 3.9226 0.9993 3186742 PK04_094212 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K15 mock treatment 202760.0 7680.0 0.52 207040.0 12700.0 0.94 1.0365 0.9615 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K16 mock treatment 204200.0 9120.0 0.62 199600.0 5220.0 0.39 0.7144 0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K17 compound treatment 230760.0 35700.0 2.43 226400.0 32000.0 2.38 3.4052 0.9999 3186743 PK04_094213 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K18 compound treatment 229840.0 34800.0 2.37 241440.0 47100.0 3.5 4.1524 0.9819 3068667 PK04_094214 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K19 compound treatment 228080.0 33000.0 2.25 222160.0 27800.0 2.07 3.0529 0.9991 3186744 PK04_094215 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K20 compound treatment 213240.0 18200.0 1.24 216800.0 22400.0 1.67 2.0554 0.9892 3186745 PK04_094216 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K21 compound treatment 206560.0 11500.0 0.78 206280.0 11900.0 0.89 1.1797 0.9981 3068668 PK04_094217 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K22 compound treatment 191280.0 -3800.0 -0.26 198920.0 4540.0 0.34 0.0557 0.1308 3186746 PK04_094218 CN(C)C(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K23 mock treatment 191480.0 -3600.0 -0.25 184040.0 -10300.0 -0.77 -0.7177 -0.8887 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 K24 mock treatment 181640.0 -13400.0 -0.92 182000.0 -12400.0 -0.92 -1.2995 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L01 compound treatment 194520.0 -564.0 -0.04 191240.0 -3140.0 -0.23 -0.1923 -0.8126 3068669 PK04_094219 CCOC(=O)N1C(N=C(N1C(=O)OCC)c2ccc(OCCCO)cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L02 compound treatment 261800.0 66700.0 4.55 257560.0 63200.0 4.7 6.5415 0.9999 3001020 PK04_094220 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]2OC(=O)Nc5ccccc5c6ccccc6)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L03 compound treatment 226120.0 31000.0 2.12 226880.0 32500.0 2.42 3.2068 0.9978 3068670 PK04_094221 COCCCNC(=O)C1ON(C(=N1)c2ccc(OCCCO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L04 compound treatment 259720.0 64600.0 4.41 269000.0 74600.0 5.55 7.0433 0.9934 3089829 PK04_094222 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L05 compound treatment 232360.0 37300.0 2.54 238840.0 44500.0 3.31 4.137 0.9915 3186813 PK04_094223 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L06 compound treatment 268320.0 73200.0 4.99 262600.0 68200.0 5.08 7.121 1.0 3001022 PK04_094224 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L07 mock treatment 196760.0 1680.0 0.11 197400.0 3020.0 0.23 0.2399 0.9507 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L08 mock treatment 203000.0 7920.0 0.54 200360.0 5980.0 0.45 0.6965 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L09 compound treatment 216000.0 20900.0 1.43 211400.0 17000.0 1.27 1.9042 0.9983 3067926 PK04_094225 COC(=O)[C@]1(CO)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L10 compound treatment 273440.0 78400.0 5.34 270640.0 76300.0 5.68 7.791 0.9995 3089768 PK04_094226 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L11 compound treatment 210720.0 15600.0 1.07 209920.0 15500.0 1.16 1.5718 0.9992 3186815 PK04_094227 COC(=O)[C@]1(CO)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L12 compound treatment 267560.0 72500.0 4.94 266280.0 71900.0 5.35 7.2781 0.9992 3089830 PK04_094228 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L13 compound treatment 236000.0 40900.0 2.79 227080.0 32700.0 2.43 3.6936 0.9977 3067927 PK04_094229 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L14 compound treatment 275240.0 80200.0 5.46 277920.0 83500.0 6.22 8.2609 0.9979 3089831 PK04_094230 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L15 mock treatment 203600.0 8520.0 0.58 198480.0 4100.0 0.31 0.6265 0.955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L16 mock treatment 199160.0 4080.0 0.28 198880.0 4500.0 0.34 0.4335 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L17 compound treatment 215000.0 19900.0 1.36 219720.0 25300.0 1.89 2.2939 0.987 3067928 PK04_094231 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L18 compound treatment 225080.0 30000.0 2.05 248960.0 54600.0 4.06 4.3187 0.9495 3001180 PK04_094232 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@@H]1OC(=O)Nc6ccccc6c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L19 compound treatment 224720.0 29600.0 2.02 224440.0 30100.0 2.24 3.0109 0.9987 3067929 PK04_094233 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L20 compound treatment 236360.0 41300.0 2.81 242760.0 48400.0 3.6 4.5362 0.9926 3001092 PK04_094234 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@@H]1OC(=O)Nc6ccccc6c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L21 compound treatment 210200.0 15100.0 1.03 217280.0 22900.0 1.7 1.9341 0.971 3067930 PK04_094235 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L22 compound treatment 214040.0 19000.0 1.29 215520.0 21100.0 1.57 2.0266 0.9952 3001093 PK04_094236 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@@H]1OC(=O)Nc6ccccc6c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L23 mock treatment 184760.0 -10300.0 -0.7 189400.0 -4980.0 -0.37 -0.7596 -0.9551 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 L24 mock treatment 176720.0 -18400.0 -1.25 177680.0 -16700.0 -1.24 -1.764 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M01 compound treatment 212560.0 17500.0 1.19 211600.0 17200.0 1.28 1.7489 0.9993 3067931 PK04_094237 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M02 compound treatment 227680.0 32600.0 2.22 215240.0 20900.0 1.55 2.6694 0.9846 3186821 PK04_094238 COCCCNC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M03 compound treatment 226440.0 31400.0 2.14 223200.0 28800.0 2.15 3.0285 1.0 3067933 PK04_094239 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M04 compound treatment 202920.0 7840.0 0.53 199280.0 4900.0 0.36 0.6358 0.9827 3186822 PK04_094240 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M05 compound treatment 205200.0 10100.0 0.69 200520.0 6140.0 0.46 0.811 0.9801 3067934 PK04_094241 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M06 compound treatment 239440.0 44400.0 3.02 234840.0 40500.0 3.01 4.2678 1.0 3186823 PK04_094242 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M07 compound treatment 257360.0 62300.0 4.25 249600.0 55200.0 4.11 5.9085 0.9999 3186824 PK04_094243 CN(C)C(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M08 compound treatment 248360.0 53300.0 3.63 238720.0 44300.0 3.3 4.902 0.9989 3186825 PK04_094244 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M09 mock treatment 209360.0 14300.0 0.97 208120.0 13700.0 1.02 1.4115 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M10 mock treatment 207400.0 12300.0 0.84 203880.0 9500.0 0.71 1.0939 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M11 compound treatment 212480.0 17400.0 1.19 211840.0 17500.0 1.3 1.7577 0.999 3067981 PK04_094245 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M12 compound treatment 205720.0 10600.0 0.73 205320.0 10900.0 0.81 1.0887 0.9983 3186826 PK04_094246 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M13 mock treatment 203560.0 8480.0 0.58 200960.0 6580.0 0.49 0.7551 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M14 mock treatment 207520.0 12400.0 0.85 200200.0 5820.0 0.43 0.906 0.9515 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M15 compound treatment 235640.0 40600.0 2.76 231640.0 37300.0 2.77 3.9162 1.0 3067982 PK04_094247 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M16 compound treatment 258000.0 62900.0 4.29 249640.0 55300.0 4.11 5.9415 0.9998 3186827 PK04_094248 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M17 compound treatment 216120.0 21000.0 1.43 215520.0 21100.0 1.57 2.1268 0.9989 3067983 PK04_094249 CN(C)C(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M18 compound treatment 256760.0 61700.0 4.2 254280.0 59900.0 4.46 6.1259 0.9996 3186828 PK04_094250 NC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M19 compound treatment 220240.0 25200.0 1.72 222960.0 28600.0 2.13 2.717 0.9943 3186829 PK04_094251 CN(C)C(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M20 compound treatment 256360.0 61300.0 4.18 240040.0 45700.0 3.4 5.3572 0.9948 3067984 PK04_094252 NC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M21 compound treatment 240640.0 45600.0 3.11 225800.0 31400.0 2.34 3.8499 0.9902 3186907 PK04_094253 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M22 compound treatment 228600.0 33500.0 2.29 240120.0 45700.0 3.4 4.0231 0.9812 3067985 PK04_094254 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M23 compound treatment 238160.0 43100.0 2.94 218040.0 23700.0 1.76 3.322 0.9701 3186908 PK04_094255 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 M24 compound treatment 256920.0 61800.0 4.22 256360.0 62000.0 4.61 6.2431 0.999 3186909 PK04_094256 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N01 compound treatment 219720.0 24600.0 1.68 212920.0 18500.0 1.38 2.1636 0.9952 3067986 PK04_094257 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N02 compound treatment 229080.0 34000.0 2.32 220600.0 26200.0 1.95 3.019 0.9963 3186910 PK04_094258 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N03 compound treatment 241320.0 46200.0 3.15 234520.0 40100.0 2.99 4.3416 0.9996 3067987 PK04_094259 CN(C)C(=O)C1ON(C(=N1)c2ccc(OCCCO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N04 compound treatment 212760.0 17700.0 1.21 212880.0 18500.0 1.38 1.8259 0.9978 3186911 PK04_094260 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N05 compound treatment 203080.0 8000.0 0.55 193320.0 -1060.0 -0.08 0.3299 0.5989 3414052 PK04_094261 COC(=O)[C@@H]1N=C(O[C@@H]1C)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N06 compound treatment 203680.0 8600.0 0.59 201680.0 7300.0 0.54 0.7988 0.9993 3186912 PK04_094262 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N07 compound treatment 207760.0 12700.0 0.86 204800.0 10400.0 0.78 1.1596 0.9985 3186913 PK04_094263 OCC(NS(=O)(=O)c1ccc(Br)cc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N08 compound treatment 291200.0 96100.0 6.55 278920.0 84500.0 6.29 9.0829 0.9998 1952953 PK04_094264 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N09 mock treatment 203960.0 8880.0 0.61 204160.0 9780.0 0.73 0.9428 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N10 mock treatment 208080.0 13000.0 0.89 207320.0 12900.0 0.96 1.3077 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N11 compound treatment 206280.0 11200.0 0.76 203880.0 9500.0 0.71 1.0399 0.9993 3068027 PK04_094265 CC(=O)OC[C@H](C=C)N(C(=O)OC(C)(C)C)S(=O)(=O)c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N12 compound treatment 251280.0 56200.0 3.83 245440.0 51100.0 3.8 5.3965 1.0 3186914 PK04_094266 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N13 mock treatment 202400.0 7320.0 0.5 196160.0 1780.0 0.13 0.4465 0.8651 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N14 mock treatment 205080.0 10000.0 0.68 199320.0 4940.0 0.37 0.742 0.9581 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N15 compound treatment 199440.0 4360.0 0.3 200080.0 5700.0 0.42 0.5102 0.9847 3068028 PK04_094267 CC(=O)OC[C@@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N16 compound treatment 282960.0 87900.0 5.99 292720.0 98300.0 7.32 9.4119 0.9951 3186915 PK04_094268 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N17 compound treatment 202000.0 6920.0 0.47 201400.0 7020.0 0.52 0.703 0.9987 3068029 PK04_094269 CC(=O)OC[C@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N18 compound treatment 279720.0 84600.0 5.77 269840.0 75500.0 5.62 8.0516 0.9999 1952947 PK04_094270 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@@H]4OC(=O)[C@@H](Cc5ccccc5)C/C=C/C[C@H](Cc6ccccc6)C(=O)O[C@@H]14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N19 compound treatment 206680.0 11600.0 0.79 200760.0 6380.0 0.48 0.895 0.9703 3068030 PK04_094271 OC[C@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N20 compound treatment 208800.0 13700.0 0.94 198160.0 3780.0 0.28 0.8603 0.8809 3186916 PK04_094272 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Br)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N21 compound treatment 195880.0 796.0 0.05 191280.0 -3100.0 -0.23 -0.1246 -0.5262 3068031 PK04_094273 CC(=O)OC[C@@H](C=C)N(C(=O)OC(C)(C)C)S(=O)(=O)c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N22 compound treatment 224160.0 29100.0 1.98 221280.0 26900.0 2.0 2.8176 1.0 1952944 PK04_094274 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(C#N)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N23 compound treatment 194640.0 -444.0 -0.03 192720.0 -1660.0 -0.12 -0.1086 -0.8552 3186917 PK04_094275 CC(=O)OC[C@H](C=C)N(Cc1ccc(cc1)[N+](=O)[O-])S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 N24 compound treatment 186320.0 -8760.0 -0.6 185520.0 -8860.0 -0.66 -0.8886 -0.9988 3413982 PK04_094276 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O01 compound treatment 252360.0 57300.0 3.9 234000.0 39600.0 2.95 4.8465 0.9904 3068032 PK04_094277 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O02 compound treatment 231560.0 36500.0 2.49 227000.0 32600.0 2.43 3.4753 0.9999 3186919 PK04_094278 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O03 compound treatment 191720.0 -3360.0 -0.23 186640.0 -7740.0 -0.58 -0.5693 -0.9186 3068033 PK04_094279 NC(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O04 compound treatment 196760.0 1680.0 0.11 192680.0 -1700.0 -0.13 -0.0085 -0.0499 3186920 PK04_094280 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O05 compound treatment 211320.0 16200.0 1.11 205080.0 10700.0 0.8 1.346 0.987 3068035 PK04_094281 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O06 compound treatment 208520.0 13400.0 0.92 205240.0 10900.0 0.81 1.2194 0.9981 3186921 PK04_094282 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O07 compound treatment 243560.0 48500.0 3.3 236760.0 42400.0 3.15 4.5675 0.9997 3186922 PK04_094283 CN(C)C(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O08 compound treatment 203720.0 8640.0 0.59 205280.0 10900.0 0.81 0.9901 0.9876 3068037 PK04_094284 CN(C)C(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O09 compound treatment 235000.0 39900.0 2.72 230280.0 35900.0 2.67 3.8138 1.0 3186923 PK04_094285 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O10 compound treatment 242520.0 47400.0 3.23 240680.0 46300.0 3.45 4.7237 0.9995 3068038 PK04_094286 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O11 mock treatment 199160.0 4080.0 0.28 196040.0 1660.0 0.12 0.284 0.9336 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O12 mock treatment 195560.0 476.0 0.03 195720.0 1340.0 0.1 0.0936 0.891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O13 compound treatment 208040.0 13000.0 0.88 200640.0 6260.0 0.47 0.9542 0.9554 3186924 PK04_094287 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O14 compound treatment 242520.0 47400.0 3.23 230720.0 36300.0 2.7 4.1995 0.9961 3186925 PK04_094288 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O15 compound treatment 223120.0 28000.0 1.91 218800.0 24400.0 1.82 2.6369 0.9997 3187013 PK04_094289 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O16 compound treatment 233160.0 38100.0 2.6 229360.0 35000.0 2.6 3.6767 1.0 3068077 PK04_094290 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O17 compound treatment 220520.0 25400.0 1.73 207680.0 13300.0 0.99 1.9264 0.9647 3187014 PK04_094291 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O18 compound treatment 257120.0 62000.0 4.23 243720.0 49300.0 3.67 5.5875 0.9975 3187015 PK04_094292 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O19 compound treatment 209160.0 14100.0 0.96 202880.0 8500.0 0.63 1.1261 0.9796 3068081 PK04_094293 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O20 compound treatment 226080.0 31000.0 2.11 222720.0 28300.0 2.11 2.9859 1.0 3187016 PK04_094294 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O21 compound treatment 204560.0 9480.0 0.65 204040.0 9660.0 0.72 0.9654 0.9986 3187017 PK04_094295 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O22 compound treatment 233120.0 38000.0 2.59 228080.0 33700.0 2.51 3.6074 0.9999 3068083 PK04_094296 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O23 compound treatment 221760.0 26700.0 1.82 219120.0 24700.0 1.84 2.5882 1.0 3187018 PK04_094297 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 O24 compound treatment 215640.0 20600.0 1.4 214520.0 20100.0 1.5 2.0511 0.9994 3068084 PK04_094298 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P01 compound treatment 214440.0 19400.0 1.32 204680.0 10300.0 0.77 1.4754 0.9666 3187019 PK04_094299 CC(=O)OC[C@H](C=C)N(Cc1ccccc1[N+](=O)[O-])S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P02 compound treatment 206040.0 11000.0 0.75 206080.0 11700.0 0.87 1.1441 0.9971 3413984 PK04_094300 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P03 compound treatment 197400.0 2320.0 0.16 192800.0 -1580.0 -0.12 0.0287 0.1457 3068086 PK04_094301 COc1ccc(CN([C@H](CO)C=C)S(=O)(=O)c2ccc(Br)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P04 compound treatment 197520.0 2440.0 0.17 193520.0 -857.0 -0.06 0.0724 0.4067 3413986 PK04_094302 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P05 compound treatment 206600.0 11500.0 0.79 202280.0 7900.0 0.59 0.9711 0.9899 3068087 PK04_094303 COc1cc(CN([C@@H](COC(=O)C)C=C)S(=O)(=O)c2ccc(Br)cc2)ccc1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P06 compound treatment 231560.0 36500.0 2.49 234080.0 39700.0 2.95 3.8479 0.9963 1952975 PK04_094304 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P07 compound treatment 197800.0 2720.0 0.19 195720.0 1340.0 0.1 0.2016 0.9581 3068088 PK04_094305 OCCCNS(=O)(=O)c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P08 compound treatment 271240.0 76200.0 5.19 267960.0 73600.0 5.48 7.5439 0.9996 3413993 PK04_094306 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P09 compound treatment 199960.0 4880.0 0.33 195880.0 1500.0 0.11 0.3142 0.8957 3068089 PK04_094307 CC[Si](CC)(CC)OC[C@@H](C=C)N(Cc1ccc(OC(=O)C)c(OC)c1)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P10 compound treatment 286800.0 91700.0 6.25 287480.0 93100.0 6.93 9.3213 0.9987 1952969 PK04_094308 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@@H]4OC(=O)[C@H](Cc5ccccc5)C/C=C/C[C@@H](Cc6ccccc6)C(=O)O[C@@H]14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P11 mock treatment 191680.0 -3400.0 -0.23 190920.0 -3460.0 -0.26 -0.346 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P12 mock treatment 193840.0 -1240.0 -0.08 191440.0 -2940.0 -0.22 -0.2145 -0.915 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P13 compound treatment 197680.0 2600.0 0.18 192200.0 -2180.0 -0.16 0.0106 0.0442 3068090 PK04_094309 COc1cc(CO)ccc1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P14 compound treatment 205880.0 10800.0 0.74 201560.0 7180.0 0.53 0.8985 0.9877 3068091 PK04_094310 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P15 compound treatment 260640.0 65600.0 4.47 252040.0 57700.0 4.29 6.195 0.9998 3187025 PK04_094311 COc1ccc(CN(C2=CC[C@@]3(C(=O)N)C(=O)C(=C(Cl)C(=O)[C@]3(C2)C#N)Cl)S(=O)(=O)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P16 compound treatment 202680.0 7600.0 0.52 203800.0 9420.0 0.7 0.8621 0.9889 3187026 PK04_094312 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P17 compound treatment 194160.0 -924.0 -0.06 190200.0 -4180.0 -0.31 -0.2644 -0.8334 3068092 PK04_094313 CC(C)(C)OC(=O)N1[C@H](COC1(C)C)C=C(Br)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P18 compound treatment 200640.0 5560.0 0.38 195640.0 1260.0 0.09 0.3343 0.8566 3187027 PK04_094314 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P19 compound treatment 188760.0 -6320.0 -0.43 187240.0 -7140.0 -0.53 -0.6805 -0.9946 1003211 PK04_094315 CNS(=O)(=O)c1ccc(C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P20 compound treatment 214520.0 19400.0 1.33 213120.0 18700.0 1.39 1.9234 0.9997 3187028 PK04_094316 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P21 compound treatment 188800.0 -6280.0 -0.43 181640.0 -12700.0 -0.95 -0.9732 -0.9356 3068127 PK04_094317 COc1cc(COC(=O)C)ccc1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P22 compound treatment 250680.0 55600.0 3.79 251520.0 57100.0 4.25 5.6875 0.9984 3187029 PK04_094318 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P23 compound treatment 179560.0 -15500.0 -1.06 181560.0 -12800.0 -0.95 -1.4229 -0.9987 3068129 PK04_094319 OC[C@@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2094 P24 compound treatment 179160.0 -15900.0 -1.09 180040.0 -14300.0 -1.07 -1.5222 -1.0 3413981 PK04_094320 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A01 compound treatment 174040.0 -18700.0 -1.28 177920.0 -12300.0 -0.92 -1.5528 -0.9869 3067957 PK04_095001 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NC4CC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A02 compound treatment 189840.0 -2940.0 -0.2 185760.0 -4500.0 -0.34 -0.3785 -0.9696 3187176 PK04_095002 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2OC)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A03 compound treatment 208840.0 16100.0 1.1 174560.0 -15700.0 -1.17 -0.052 -0.0324 3067577 PK04_095003 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCc6ccccc6)c7ccc(cc7)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A04 compound treatment 201720.0 8940.0 0.61 193800.0 3540.0 0.26 0.6174 0.9295 3187436 PK04_095004 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A05 compound treatment 226080.0 33300.0 2.27 209640.0 19400.0 1.44 2.6253 0.976 3186425 PK04_095005 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc6I)c7ccc(cc7)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A06 compound treatment 184480.0 -8300.0 -0.57 186800.0 -3460.0 -0.26 -0.5821 -0.9367 3187069 PK04_095006 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A07 compound treatment 188720.0 -4060.0 -0.28 182160.0 -8100.0 -0.6 -0.6219 -0.9375 3187427 PK04_095007 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A08 compound treatment 226920.0 34100.0 2.33 224320.0 34100.0 2.53 3.4384 0.9991 3187515 PK04_095008 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc6)c7ccc(cc7)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A09 compound treatment 180800.0 -12000.0 -0.82 179120.0 -11100.0 -0.83 -1.1637 -1.0 3187425 PK04_095009 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A10 compound treatment 185800.0 -6980.0 -0.48 179440.0 -10800.0 -0.81 -0.9058 -0.9684 3068592 PK04_095010 CCCNC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A11 compound treatment 177360.0 -15400.0 -1.05 211200.0 20900.0 1.56 0.3587 0.1909 3187517 PK04_095011 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A12 compound treatment 192760.0 -15.6 0.0 196560.0 6300.0 0.47 0.3307 0.7055 3187344 PK04_095012 COCCCNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A13 mock treatment 179240.0 -13500.0 -0.92 175560.0 -14700.0 -1.09 -1.4263 -0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A14 mock treatment 178360.0 -14400.0 -0.98 179000.0 -11300.0 -0.84 -1.2877 -0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A15 compound treatment 174880.0 -17900.0 -1.22 189600.0 -663.0 -0.05 -0.8976 -0.7351 3186552 PK04_095013 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A16 compound treatment 177400.0 -15400.0 -1.05 173800.0 -16500.0 -1.23 -1.6076 -0.997 3187439 PK04_095014 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A17 compound treatment 174720.0 -18100.0 -1.23 186160.0 -4100.0 -0.31 -1.0863 -0.8565 3187073 PK04_095015 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5cc(cc(c5)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A18 compound treatment 184560.0 -8220.0 -0.56 181480.0 -8780.0 -0.65 -0.8583 -0.997 3187272 PK04_095016 COCCCNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A19 compound treatment 180720.0 -12100.0 -0.82 176680.0 -13600.0 -1.01 -1.296 -0.9947 3187508 PK04_095017 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NC3CC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A20 compound treatment 175160.0 -17600.0 -1.2 199520.0 9260.0 0.69 -0.362 -0.2615 3186432 PK04_095018 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(Cc5ccccc5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A21 compound treatment 211600.0 18800.0 1.28 192160.0 1900.0 0.14 1.0074 0.7802 3068646 PK04_095019 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A22 compound treatment 176560.0 -16200.0 -1.11 173480.0 -16800.0 -1.25 -1.665 -0.9981 3068651 PK04_095020 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A23 compound treatment 182480.0 -10300.0 -0.7 166760.0 -23500.0 -1.75 -1.7332 -0.9196 3187585 PK04_095021 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 A24 compound treatment 181720.0 -11100.0 -0.75 175480.0 -14800.0 -1.1 -1.3109 -0.983 3187430 PK04_095022 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B01 compound treatment 209320.0 16500.0 1.13 218320.0 28100.0 2.09 2.2742 0.9582 3187519 PK04_095023 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)O)c4ccc(cc4)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B02 compound treatment 181160.0 -11600.0 -0.79 177720.0 -12500.0 -0.93 -1.2201 -0.9967 3186885 PK04_095024 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B03 compound treatment 184480.0 -8300.0 -0.57 184840.0 -5420.0 -0.4 -0.6853 -0.9863 3187435 PK04_095025 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B04 compound treatment 205400.0 12600.0 0.86 207880.0 17600.0 1.31 1.5358 0.9792 3186491 PK04_095026 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B05 compound treatment 181680.0 -11100.0 -0.76 182040.0 -8220.0 -0.61 -0.9676 -0.9945 3068539 PK04_095027 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4cc(F)cc(c4)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B06 compound treatment 217320.0 24500.0 1.67 211160.0 20900.0 1.56 2.283 0.9993 3186559 PK04_095028 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B07 compound treatment 218320.0 25500.0 1.74 220520.0 30300.0 2.25 2.8238 0.9919 3068561 PK04_095029 CCCNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B08 compound treatment 189120.0 -3660.0 -0.25 189840.0 -423.0 -0.03 -0.1985 -0.7901 3068322 PK04_095030 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B09 compound treatment 174440.0 -18300.0 -1.25 176520.0 -13700.0 -1.02 -1.6072 -0.995 3187432 PK04_095031 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B10 compound treatment 197760.0 4980.0 0.34 205000.0 14700.0 1.1 1.0159 0.8847 3068145 PK04_095032 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCC(F)(F)F)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B11 compound treatment 179640.0 -13100.0 -0.9 178840.0 -11400.0 -0.85 -1.2344 -0.9997 3187265 PK04_095033 CC(C)N1[C@H]([C@H](C(=O)NCCCN(C)C)c2ccccc2C1=O)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B12 compound treatment 189400.0 -3380.0 -0.23 180520.0 -9740.0 -0.73 -0.6755 -0.8879 3186629 PK04_095034 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B13 mock treatment 178280.0 -14500.0 -0.99 180920.0 -9340.0 -0.7 -1.1905 -0.9852 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B14 mock treatment 179200.0 -13600.0 -0.93 178400.0 -11900.0 -0.88 -1.2788 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B15 compound treatment 197680.0 4900.0 0.33 194080.0 3820.0 0.28 0.4373 0.9967 3187269 PK04_095035 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C3CCCCC3)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B16 compound treatment 187760.0 -5020.0 -0.34 189280.0 -983.0 -0.07 -0.2935 -0.8393 3186887 PK04_095036 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B17 compound treatment 189480.0 -3300.0 -0.22 184920.0 -5340.0 -0.4 -0.44 -0.9635 3068417 PK04_095037 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B18 compound treatment 180680.0 -12100.0 -0.82 179240.0 -11000.0 -0.82 -1.1632 -1.0 3067610 PK04_095038 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(C7CC7)c2c1)c8ccc(cc8)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B19 compound treatment 196320.0 3540.0 0.24 187480.0 -2780.0 -0.21 0.0244 0.0768 3068639 PK04_095039 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3cc(F)cc(c3)C(F)(F)F)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B20 compound treatment 184440.0 -8340.0 -0.57 183000.0 -7260.0 -0.54 -0.7841 -0.9997 3068006 PK04_095040 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B21 compound treatment 181960.0 -10800.0 -0.74 171600.0 -18700.0 -1.39 -1.5036 -0.9561 3068601 PK04_095041 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NCc4ccccc4)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B22 compound treatment 177560.0 -15200.0 -1.04 172160.0 -18100.0 -1.35 -1.6862 -0.9917 3068203 PK04_095042 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5Cl)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B23 compound treatment 171200.0 -21600.0 -1.47 168360.0 -21900.0 -1.63 -2.1928 -0.9987 3187355 PK04_095043 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NCC(F)(F)F)c4ccccc4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 B24 compound treatment 173760.0 -19000.0 -1.3 169200.0 -21100.0 -1.57 -2.0252 -0.9955 3068156 PK04_095044 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C01 compound treatment 186080.0 -6700.0 -0.46 181200.0 -9060.0 -0.67 -0.7997 -0.9819 3187590 PK04_095045 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C02 compound treatment 185760.0 -7020.0 -0.48 179000.0 -11300.0 -0.84 -0.9309 -0.9646 3187180 PK04_095046 CC(C)NC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C03 compound treatment 196400.0 3620.0 0.25 191960.0 1700.0 0.13 0.2641 0.9515 3186493 PK04_095047 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C04 compound treatment 164000.0 -28800.0 -1.96 160000.0 -30300.0 -2.25 -2.9799 -0.9976 3186427 PK04_095048 CN(C)CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C05 compound treatment 209880.0 17100.0 1.17 200760.0 10500.0 0.78 1.377 0.981 3187172 PK04_095049 COc1ccccc1CN2[C@H]([C@H](C(=O)NCCN3CCOCC3)c4ccccc4C2=O)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C06 compound treatment 191200.0 -1580.0 -0.11 191320.0 1060.0 0.08 -0.0203 -0.1525 3187080 PK04_095050 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C07 compound treatment 181960.0 -10800.0 -0.74 184000.0 -6260.0 -0.47 -0.851 -0.9755 3186988 PK04_095051 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C08 compound treatment 199000.0 6220.0 0.42 186000.0 -4260.0 -0.32 0.0757 0.143 3068011 PK04_095052 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C09 compound treatment 184680.0 -8100.0 -0.55 179200.0 -11100.0 -0.82 -0.9725 -0.9811 3068498 PK04_095053 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C10 compound treatment 163080.0 -29700.0 -2.02 158720.0 -31500.0 -2.35 -3.0916 -0.9973 3186550 PK04_095054 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C11 mock treatment 184960.0 -7820.0 -0.53 178760.0 -11500.0 -0.86 -0.9821 -0.974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C12 mock treatment 184000.0 -8780.0 -0.6 179840.0 -10400.0 -0.78 -0.9716 -0.9918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C13 compound treatment 186920.0 -5860.0 -0.4 184920.0 -5340.0 -0.4 -0.5635 -1.0 3187361 PK04_095055 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C14 compound treatment 185760.0 -7020.0 -0.48 180000.0 -10300.0 -0.76 -0.8783 -0.9746 3068504 PK04_095056 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccc(OC(F)(F)F)cc3)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C15 mock treatment 187440.0 -5340.0 -0.36 181640.0 -8620.0 -0.64 -0.711 -0.9638 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C16 mock treatment 184040.0 -8740.0 -0.6 178160.0 -12100.0 -0.9 -1.0581 -0.9798 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C17 compound treatment 185600.0 -7180.0 -0.49 183400.0 -6860.0 -0.51 -0.7071 -0.9998 3067969 PK04_095057 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCCCN(C)C)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C18 compound treatment 212480.0 19700.0 1.34 209080.0 18800.0 1.4 1.9402 0.9998 3187359 PK04_095058 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3ccc(OC(F)(F)F)cc3)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C19 compound treatment 175600.0 -17200.0 -1.17 178960.0 -11300.0 -0.84 -1.4228 -0.9868 3187087 PK04_095059 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C20 compound treatment 183840.0 -8940.0 -0.61 183160.0 -7100.0 -0.53 -0.8046 -0.9975 3187443 PK04_095060 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C21 compound treatment 201840.0 9060.0 0.62 196960.0 6700.0 0.5 0.7895 0.9943 3067571 PK04_095061 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C22 compound treatment 180400.0 -12400.0 -0.84 177080.0 -13200.0 -0.98 -1.2904 -0.9972 3187181 PK04_095062 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NCC(F)(F)F)c3ccccc3C2=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C23 compound treatment 176880.0 -15900.0 -1.08 173720.0 -16500.0 -1.23 -1.6369 -0.998 3187509 PK04_095063 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C(C)C)[C@@H]2c3ccc(CO)cc3)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 C24 compound treatment 188320.0 -4460.0 -0.3 182600.0 -7660.0 -0.57 -0.6181 -0.9565 3068474 PK04_095064 CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D01 compound treatment 230360.0 37600.0 2.56 213400.0 23100.0 1.72 3.0296 0.9813 3068587 PK04_095065 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(CC3(CC4CC5CC(C4)C3)C5)C(=O)c6ccccc26)c7ccc(CO)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D02 compound treatment 180400.0 -12400.0 -0.84 180000.0 -10300.0 -0.76 -1.1367 -0.9988 3068318 PK04_095066 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D03 compound treatment 183320.0 -9460.0 -0.64 184320.0 -5940.0 -0.44 -0.7686 -0.9831 3187363 PK04_095067 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D04 compound treatment 192840.0 64.4 0.0 184400.0 -5860.0 -0.44 -0.3054 -0.7 3186486 PK04_095068 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(CCN7CCOCC7)c2c1)c8ccc(cc8)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D05 compound treatment 190000.0 -2780.0 -0.19 192320.0 2060.0 0.15 -0.0255 -0.1049 3187179 PK04_095069 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C(=O)c3ccccc23)c4ccc(C)cn4)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D06 compound treatment 247640.0 54900.0 3.74 228840.0 38600.0 2.87 4.6752 0.9915 3187522 PK04_095070 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D07 compound treatment 188680.0 -4100.0 -0.28 182320.0 -7940.0 -0.59 -0.6154 -0.9414 3068515 PK04_095071 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NC3CC3)c4ccccc4C2=O)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D08 compound treatment 192200.0 -576.0 -0.04 185680.0 -4580.0 -0.34 -0.2689 -0.7833 3186872 PK04_095072 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D09 compound treatment 180440.0 -12300.0 -0.84 168640.0 -21600.0 -1.61 -1.7326 -0.9542 3068609 PK04_095073 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D10 compound treatment 187840.0 -4940.0 -0.34 180400.0 -9860.0 -0.73 -0.757 -0.9374 3186795 PK04_095074 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D11 mock treatment 183440.0 -9340.0 -0.64 180640.0 -9620.0 -0.72 -0.9565 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D12 mock treatment 189400.0 -3380.0 -0.23 185280.0 -4980.0 -0.37 -0.425 -0.9737 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D13 compound treatment 184880.0 -7900.0 -0.54 189320.0 -943.0 -0.07 -0.4302 -0.7926 3067964 PK04_095075 CCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D14 compound treatment 187240.0 -5540.0 -0.38 187120.0 -3140.0 -0.23 -0.4322 -0.9735 3068230 PK04_095076 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D15 mock treatment 183600.0 -9180.0 -0.63 181440.0 -8820.0 -0.66 -0.9067 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D16 mock treatment 189960.0 -2820.0 -0.19 181920.0 -8340.0 -0.62 -0.5748 -0.8844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D17 compound treatment 179040.0 -13700.0 -0.94 179160.0 -11100.0 -0.83 -1.2465 -0.9981 3068595 PK04_095077 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCc3ccccc3)c4ccccc4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D18 compound treatment 195240.0 2460.0 0.17 198240.0 7980.0 0.59 0.5386 0.8729 3186982 PK04_095078 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D19 compound treatment 183800.0 -8980.0 -0.61 190520.0 258.0 0.02 -0.4191 -0.6846 3187440 PK04_095079 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D20 compound treatment 185360.0 -7420.0 -0.51 182240.0 -8020.0 -0.6 -0.7797 -0.9966 3068415 PK04_095080 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D21 compound treatment 187760.0 -5020.0 -0.34 177360.0 -12900.0 -0.96 -0.9208 -0.9033 3068596 PK04_095081 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCC(F)(F)F)c3ccccc3C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D22 compound treatment 183840.0 -8940.0 -0.61 184240.0 -6020.0 -0.45 -0.7477 -0.9886 3186713 PK04_095082 CC(C)CNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D23 compound treatment 176640.0 -16100.0 -1.1 174600.0 -15700.0 -1.17 -1.6022 -0.9996 3187357 PK04_095083 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 D24 compound treatment 169920.0 -22900.0 -1.56 172360.0 -17900.0 -1.33 -2.044 -0.997 3068270 PK04_095084 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCCN6CCOCC6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E01 mock treatment 187280.0 -5500.0 -0.37 182440.0 -7820.0 -0.58 -0.6766 -0.9773 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E02 mock treatment 181720.0 -11100.0 -0.75 188080.0 -2180.0 -0.16 -0.6478 -0.8402 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E03 compound treatment 188680.0 -4100.0 -0.28 186720.0 -3540.0 -0.26 -0.3839 -0.9996 3068636 PK04_095085 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E04 compound treatment 195800.0 3020.0 0.21 192080.0 1820.0 0.14 0.2415 0.9791 3186556 PK04_095086 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E05 compound treatment 244080.0 51300.0 3.5 224880.0 34600.0 2.58 4.2951 0.9887 3187587 PK04_095087 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E06 compound treatment 229960.0 37200.0 2.54 212840.0 22600.0 1.68 2.9808 0.9801 3186428 PK04_095088 COCCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E07 compound treatment 216760.0 24000.0 1.64 207360.0 17100.0 1.27 2.056 0.9923 3187266 PK04_095089 CCCNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E08 compound treatment 189600.0 -3180.0 -0.22 190960.0 698.0 0.05 -0.1164 -0.5227 3187351 PK04_095090 CC(C)CNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E09 mock treatment 190600.0 -2180.0 -0.15 188840.0 -1420.0 -0.11 -0.1797 -0.9863 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E10 mock treatment 187320.0 -5460.0 -0.37 186040.0 -4220.0 -0.31 -0.4852 -0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E11 compound treatment 194880.0 2100.0 0.14 190400.0 138.0 0.01 0.1087 0.7556 3068004 PK04_095091 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E12 compound treatment 222680.0 29900.0 2.04 207240.0 17000.0 1.26 2.3351 0.9735 3186500 PK04_095092 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E13 compound treatment 199760.0 6980.0 0.48 191840.0 1580.0 0.12 0.4197 0.8558 3187346 PK04_095093 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCCN3CCOCC3)c4ccccc4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E14 compound treatment 201760.0 8980.0 0.61 199520.0 9260.0 0.69 0.9203 0.9983 3187262 PK04_095094 CC(C)N1[C@H]([C@H](C(=O)NCCN2CCOCC2)c3ccccc3C1=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E15 compound treatment 278520.0 85700.0 5.85 255760.0 65500.0 4.87 7.5806 0.9959 3067574 PK04_095095 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NC6CC6)c7ccc(cc7)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E16 compound treatment 194520.0 1740.0 0.12 191120.0 858.0 0.06 0.1292 0.9574 3187350 PK04_095096 COCCCNC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E17 mock treatment 193440.0 664.0 0.05 192520.0 2260.0 0.17 0.1508 0.8668 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E18 mock treatment 192600.0 -176.0 -0.01 190120.0 -143.0 -0.01 -0.016 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E19 compound treatment 206880.0 14100.0 0.96 203760.0 13500.0 1.0 1.3903 0.9998 3068657 PK04_095097 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E20 compound treatment 206960.0 14200.0 0.97 212400.0 22100.0 1.65 1.8489 0.9678 3068140 PK04_095098 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E21 compound treatment 206360.0 13600.0 0.93 196320.0 6060.0 0.45 0.9737 0.9453 3186562 PK04_095099 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E22 compound treatment 192520.0 -256.0 -0.02 185600.0 -4660.0 -0.35 -0.2577 -0.7417 3187591 PK04_095100 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E23 compound treatment 190720.0 -2060.0 -0.14 186040.0 -4220.0 -0.31 -0.3213 -0.9338 3187263 PK04_095101 CC(C)N1[C@H]([C@H](C(=O)NCc2ccccc2)c3ccccc3C1=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 E24 compound treatment 186840.0 -5940.0 -0.4 182200.0 -8060.0 -0.6 -0.7105 -0.9816 3068517 PK04_095102 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NCc3ccccc3)c4ccccc4C2=O)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F01 mock treatment 182720.0 -10100.0 -0.69 180760.0 -9500.0 -0.71 -0.9849 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F02 mock treatment 187640.0 -5140.0 -0.35 187160.0 -3100.0 -0.23 -0.4109 -0.9796 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F03 compound treatment 203720.0 10900.0 0.75 197720.0 7460.0 0.56 0.9201 0.9894 3187079 PK04_095103 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F04 compound treatment 190760.0 -2020.0 -0.14 174080.0 -16200.0 -1.2 -0.9488 -0.7827 3068331 PK04_095104 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F05 compound treatment 225400.0 32600.0 2.22 210040.0 19800.0 1.47 2.6136 0.9799 3068563 PK04_095105 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2CC5(CC6CC7CC(C6)C5)C7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F06 compound treatment 199640.0 6860.0 0.47 198680.0 8420.0 0.63 0.7739 0.9897 3186879 PK04_095106 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NCCN6CCOCC6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F07 compound treatment 211000.0 18200.0 1.24 202720.0 12500.0 0.93 1.5342 0.9896 3187523 PK04_095107 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F08 compound treatment 204640.0 11900.0 0.81 197320.0 7060.0 0.53 0.9434 0.9781 3186563 PK04_095108 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F09 mock treatment 198240.0 5460.0 0.37 189480.0 -783.0 -0.06 0.2222 0.5894 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F10 mock treatment 189960.0 -2820.0 -0.19 191280.0 1020.0 0.08 -0.0822 -0.3983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F11 compound treatment 201480.0 8700.0 0.59 207880.0 17600.0 1.31 1.3468 0.9358 3187257 PK04_095109 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2C5Cc6ccccc6C5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F12 compound treatment 199880.0 7100.0 0.48 189680.0 -583.0 -0.04 0.3118 0.6413 3068241 PK04_095110 CCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F13 compound treatment 194680.0 1900.0 0.13 194160.0 3900.0 0.29 0.2969 0.9343 3068554 PK04_095111 COCCCNC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F14 compound treatment 197560.0 4780.0 0.33 196280.0 6020.0 0.45 0.5473 0.9879 3068362 PK04_095112 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C(C)C)[C@@H]2c3ccc(CO)cc3)Sc4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F15 compound treatment 244520.0 51700.0 3.53 233960.0 43700.0 3.25 4.7942 0.9992 3186423 PK04_095113 CC(C)CNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F16 compound treatment 212440.0 19700.0 1.34 225520.0 35300.0 2.62 2.8035 0.9514 3068012 PK04_095114 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)O)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F17 mock treatment 196480.0 3700.0 0.25 188160.0 -2100.0 -0.16 0.0679 0.2286 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F18 mock treatment 192840.0 64.4 0.0 189960.0 -303.0 -0.02 -0.0128 -0.5587 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F19 compound treatment 240800.0 48000.0 3.27 228680.0 38400.0 2.86 4.337 0.9977 3067568 PK04_095115 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F20 compound treatment 197680.0 4900.0 0.33 189040.0 -1220.0 -0.09 0.1721 0.4966 3068266 PK04_095116 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F21 compound treatment 223040.0 30300.0 2.06 211000.0 20700.0 1.54 2.5504 0.9898 3186419 PK04_095117 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCc4ccccc4)c5ccc(cc5)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F22 compound treatment 187840.0 -4940.0 -0.34 184320.0 -5940.0 -0.44 -0.5507 -0.9909 3187524 PK04_095118 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F23 compound treatment 187120.0 -5660.0 -0.39 182680.0 -7580.0 -0.56 -0.6717 -0.9828 3068017 PK04_095119 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)O)c4ccccc4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 F24 compound treatment 176360.0 -16400.0 -1.12 179640.0 -10600.0 -0.79 -1.3504 -0.9855 3186554 PK04_095120 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G01 compound treatment 245720.0 52900.0 3.61 228760.0 38500.0 2.87 4.5784 0.9935 3186418 PK04_095121 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCCN4CCOCC4)c5ccc(cc5)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G02 compound treatment 196600.0 3820.0 0.26 195920.0 5660.0 0.42 0.4821 0.9734 3067966 PK04_095122 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCCN3CCOCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G03 mock treatment 193120.0 344.0 0.02 191000.0 738.0 0.05 0.0554 0.9282 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G04 mock treatment 198520.0 5740.0 0.39 193600.0 3340.0 0.25 0.4526 0.9759 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G05 compound treatment 215240.0 22500.0 1.53 208080.0 17800.0 1.33 2.0207 0.9974 3068153 PK04_095123 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G06 compound treatment 198920.0 6140.0 0.42 191520.0 1260.0 0.09 0.3624 0.8443 3187356 PK04_095124 COCCCNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G07 compound treatment 214720.0 21900.0 1.5 211400.0 21100.0 1.57 2.1703 0.9997 3187173 PK04_095125 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3OC)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G08 compound treatment 202000.0 9220.0 0.63 192280.0 2020.0 0.15 0.5509 0.852 3068514 PK04_095126 CCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G09 compound treatment 218760.0 26000.0 1.77 220560.0 30300.0 2.25 2.8472 0.9929 3187442 PK04_095127 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G10 compound treatment 207280.0 14500.0 0.99 210960.0 20700.0 1.54 1.7885 0.977 3068420 PK04_095128 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G11 compound treatment 203880.0 11100.0 0.76 192560.0 2300.0 0.17 0.6562 0.8455 3187434 PK04_095129 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G12 compound treatment 220080.0 27300.0 1.86 205640.0 15400.0 1.14 2.1256 0.9727 3186416 PK04_095130 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G13 compound treatment 198680.0 5900.0 0.4 202800.0 12500.0 0.93 0.9445 0.9294 3068507 PK04_095131 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G14 compound treatment 209920.0 17100.0 1.17 206840.0 16600.0 1.23 1.6989 0.9996 3187162 PK04_095132 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5cc(F)cc(c5)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G15 compound treatment 196640.0 3860.0 0.26 193920.0 3660.0 0.27 0.3788 0.9999 3068602 PK04_095133 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G16 compound treatment 193240.0 464.0 0.03 194640.0 4380.0 0.33 0.2528 0.7722 3187426 PK04_095134 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G17 compound treatment 211360.0 18600.0 1.27 210480.0 20200.0 1.5 1.9599 0.9963 3067567 PK04_095135 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G18 compound treatment 211200.0 18400.0 1.26 204880.0 14600.0 1.09 1.6575 0.9974 3187525 PK04_095136 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G19 mock treatment 199920.0 7140.0 0.49 195320.0 5060.0 0.38 0.6106 0.9919 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G20 mock treatment 195360.0 2580.0 0.18 190520.0 258.0 0.02 0.1381 0.7794 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G21 compound treatment 194000.0 1220.0 0.08 193120.0 2860.0 0.21 0.2094 0.9166 3187167 PK04_095137 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccc(OC(F)(F)F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G22 compound treatment 200240.0 7460.0 0.51 200760.0 10500.0 0.78 0.9123 0.9784 3187174 PK04_095138 COc1ccccc1CN2[C@H]([C@H](C(=O)NC(C)C)c3ccccc3C2=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G23 compound treatment 196520.0 3740.0 0.26 195800.0 5540.0 0.41 0.4719 0.9735 3068478 PK04_095139 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 G24 compound treatment 193640.0 864.0 0.06 185080.0 -5180.0 -0.39 -0.2311 -0.5922 3068471 PK04_095140 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccccc5Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H01 compound treatment 200520.0 7740.0 0.53 190880.0 618.0 0.05 0.4058 0.7658 3068149 PK04_095141 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H02 compound treatment 238800.0 46000.0 3.14 228280.0 38000.0 2.83 4.2195 0.9987 3068236 PK04_095142 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H03 mock treatment 190400.0 -2380.0 -0.16 189320.0 -943.0 -0.07 -0.1641 -0.9299 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H04 mock treatment 202320.0 9540.0 0.65 191640.0 1380.0 0.1 0.5326 0.8085 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H05 compound treatment 208440.0 15700.0 1.07 205120.0 14900.0 1.11 1.5371 0.9998 3187083 PK04_095143 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H06 compound treatment 211240.0 18500.0 1.26 202840.0 12600.0 0.94 1.5521 0.9894 3068265 PK04_095144 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H07 compound treatment 209480.0 16700.0 1.14 204360.0 14100.0 1.05 1.5472 0.9992 3068458 PK04_095145 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H08 compound treatment 201520.0 8740.0 0.6 191840.0 1580.0 0.12 0.5046 0.8304 3068401 PK04_095146 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H09 compound treatment 202640.0 9860.0 0.67 199000.0 8740.0 0.65 0.9354 0.9999 3187071 PK04_095147 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H10 compound treatment 225040.0 32300.0 2.2 223920.0 33700.0 2.51 3.3267 0.9979 3068139 PK04_095148 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H11 compound treatment 196360.0 3580.0 0.24 196000.0 5740.0 0.43 0.4747 0.9649 3187589 PK04_095149 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H12 compound treatment 198800.0 6020.0 0.41 197080.0 6820.0 0.51 0.6492 0.9945 3186627 PK04_095150 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4OC)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H13 compound treatment 207280.0 14500.0 0.99 206240.0 16000.0 1.19 1.5401 0.9958 3187261 PK04_095151 CC(C)N1[C@H]([C@H](C(=O)NC2CC2)c3ccccc3C1=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H14 compound treatment 193480.0 704.0 0.05 194600.0 4340.0 0.32 0.2622 0.8035 3186980 PK04_095152 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H15 compound treatment 209160.0 16400.0 1.12 200680.0 10400.0 0.78 1.3381 0.9841 3187166 PK04_095153 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccc(OC(F)(F)F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H16 compound treatment 200800.0 8020.0 0.55 192720.0 2460.0 0.18 0.5162 0.8948 3186978 PK04_095154 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H17 compound treatment 194120.0 1340.0 0.09 191400.0 1140.0 0.08 0.1247 0.9992 3187349 PK04_095155 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCCCN(C)C)c3ccccc3C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H18 compound treatment 203000.0 10200.0 0.7 214880.0 24600.0 1.83 1.7885 0.9123 3068412 PK04_095156 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H19 mock treatment 194480.0 1700.0 0.12 194640.0 4380.0 0.33 0.3125 0.9036 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H20 mock treatment 192240.0 -536.0 -0.04 191360.0 1100.0 0.08 0.0319 0.3569 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H21 compound treatment 191600.0 -1180.0 -0.08 194880.0 4620.0 0.34 0.1863 0.528 3187512 PK04_095157 COCCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H22 compound treatment 188680.0 -4100.0 -0.28 186920.0 -3340.0 -0.25 -0.3734 -0.9983 3186806 PK04_095158 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H23 compound treatment 186200.0 -6580.0 -0.45 186480.0 -3780.0 -0.28 -0.5161 -0.9749 3068599 PK04_095159 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NC4CC4)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 H24 compound treatment 184760.0 -8020.0 -0.55 189000.0 -1260.0 -0.09 -0.4529 -0.8167 3187586 PK04_095160 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I01 compound treatment 201160.0 8380.0 0.57 196920.0 6660.0 0.5 0.7546 0.9975 3187165 PK04_095161 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccc(OC(F)(F)F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I02 compound treatment 208880.0 16100.0 1.1 200120.0 9860.0 0.73 1.2951 0.9808 3068418 PK04_095162 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I03 compound treatment 205520.0 12700.0 0.87 201480.0 11200.0 0.83 1.2047 0.9998 3187178 PK04_095163 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NCCN3CCOCC3)c4ccccc4C2=O)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I04 compound treatment 201720.0 8940.0 0.61 202960.0 12700.0 0.95 1.0994 0.9775 3068019 PK04_095164 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I05 mock treatment 200480.0 7700.0 0.53 198240.0 7980.0 0.59 0.7913 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I06 mock treatment 196120.0 3340.0 0.23 195760.0 5500.0 0.41 0.4505 0.9619 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I07 compound treatment 225160.0 32400.0 2.21 223120.0 32900.0 2.45 3.2904 0.9987 3068542 PK04_095165 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C3Cc4ccccc4C3)C(=O)c5ccccc25)c6ccc(CO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I08 compound treatment 200040.0 7260.0 0.5 198480.0 8220.0 0.61 0.7827 0.9945 3187345 PK04_095166 CC(C)CNC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I09 compound treatment 262920.0 70100.0 4.78 258560.0 68300.0 5.08 6.9759 0.9995 3067971 PK04_095167 CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I10 compound treatment 197800.0 5020.0 0.34 199440.0 9180.0 0.68 0.7252 0.9491 3068641 PK04_095168 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I11 compound treatment 192360.0 -416.0 -0.03 189120.0 -1140.0 -0.09 -0.0802 -0.8944 3187358 PK04_095169 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I12 compound treatment 200960.0 8180.0 0.56 195680.0 5420.0 0.4 0.6797 0.9873 3068653 PK04_095170 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I13 compound treatment 207600.0 14800.0 1.01 199240.0 8980.0 0.67 1.1871 0.9798 3067962 PK04_095171 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I14 compound treatment 208360.0 15600.0 1.06 208560.0 18300.0 1.36 1.7143 0.9925 3068606 PK04_095172 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I15 compound treatment 212960.0 20200.0 1.38 210600.0 20300.0 1.51 2.0434 0.9989 3068476 PK04_095173 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5cc(F)cc(c5)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I16 compound treatment 241040.0 48300.0 3.29 222080.0 31800.0 2.37 4.0012 0.987 3186417 PK04_095174 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NC4CC4)c5ccc(cc5)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I17 compound treatment 215920.0 23100.0 1.58 208800.0 18500.0 1.38 2.0913 0.9978 3187268 PK04_095175 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2C5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I18 compound treatment 197040.0 4260.0 0.29 201760.0 11500.0 0.86 0.8107 0.897 3187264 PK04_095176 CC(C)N1[C@H]([C@H](C(=O)NCC(F)(F)F)c2ccccc2C1=O)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I19 compound treatment 211840.0 19100.0 1.3 201880.0 11600.0 0.86 1.5305 0.9804 3186499 PK04_095177 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3OC)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I20 compound treatment 182200.0 -10600.0 -0.72 179840.0 -10400.0 -0.78 -1.0583 -0.9993 3068422 PK04_095178 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I21 mock treatment 192560.0 -216.0 -0.01 189960.0 -303.0 -0.02 -0.0263 -0.9787 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I22 mock treatment 188720.0 -4060.0 -0.28 185560.0 -4700.0 -0.35 -0.443 -0.9932 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I23 compound treatment 195720.0 2940.0 0.2 187480.0 -2780.0 -0.21 -0.0045 -0.0156 3068550 PK04_095179 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C(C)C)C(=O)c3ccccc23)c4ccc(CO)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 I24 compound treatment 188440.0 -4340.0 -0.3 175360.0 -14900.0 -1.11 -0.9933 -0.8653 3187258 PK04_095180 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2C4Cc5ccccc5C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J01 compound treatment 215080.0 22300.0 1.52 208720.0 18500.0 1.37 2.0466 0.9987 3187273 PK04_095181 CC(C)CNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J02 compound treatment 194560.0 1780.0 0.12 194400.0 4140.0 0.31 0.3038 0.9175 3186630 PK04_095182 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J03 compound treatment 194080.0 1300.0 0.09 198960.0 8700.0 0.65 0.5206 0.7968 3187353 PK04_095183 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(C(=O)c3ccccc32)c4ccc(C)cn4)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J04 compound treatment 203320.0 10500.0 0.72 203920.0 13700.0 1.02 1.2271 0.9856 3187588 PK04_095184 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)O)c3ccccc3C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J05 mock treatment 201400.0 8620.0 0.59 198160.0 7900.0 0.59 0.8314 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J06 mock treatment 207560.0 14800.0 1.01 202320.0 12100.0 0.9 1.3473 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J07 compound treatment 236720.0 43900.0 3.0 224640.0 34400.0 2.56 3.9277 0.9969 3186420 PK04_095185 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c4ccc(cc4)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J08 compound treatment 208040.0 15300.0 1.04 201800.0 11500.0 0.86 1.3431 0.9954 3186722 PK04_095186 COCCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J09 compound treatment 254200.0 61400.0 4.19 243720.0 53500.0 3.98 5.7745 0.9997 3186426 PK04_095187 CC(C)NC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J10 compound treatment 200320.0 7540.0 0.51 198440.0 8180.0 0.61 0.7941 0.9965 3186639 PK04_095188 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J11 compound treatment 209440.0 16700.0 1.14 209200.0 18900.0 1.41 1.8 0.9943 3187270 PK04_095189 CC(C)NC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J12 compound treatment 220480.0 27700.0 1.89 212920.0 22700.0 1.69 2.528 0.9984 3067980 PK04_095190 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J13 compound treatment 203480.0 10700.0 0.73 188320.0 -1940.0 -0.14 0.4138 0.5562 3186421 PK04_095191 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J14 compound treatment 229560.0 36800.0 2.51 222160.0 31900.0 2.37 3.452 0.9996 3068150 PK04_095192 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J15 compound treatment 199080.0 6300.0 0.43 194520.0 4260.0 0.32 0.528 0.9888 3068598 PK04_095193 CCCNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J16 compound treatment 201880.0 9100.0 0.62 197360.0 7100.0 0.53 0.8124 0.9968 3068324 PK04_095194 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J17 compound treatment 210240.0 17500.0 1.19 211440.0 21200.0 1.58 1.9565 0.9904 3067973 PK04_095195 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCCN6CCOCC6)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J18 compound treatment 210440.0 17700.0 1.2 207480.0 17200.0 1.28 1.7577 0.9995 3068414 PK04_095196 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J19 compound treatment 204880.0 12100.0 0.83 206920.0 16700.0 1.24 1.4602 0.9804 3187085 PK04_095197 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J20 compound treatment 195600.0 2820.0 0.19 193840.0 3580.0 0.27 0.3244 0.9873 3186884 PK04_095198 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J21 mock treatment 187920.0 -4860.0 -0.33 184200.0 -6060.0 -0.45 -0.5531 -0.9884 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J22 mock treatment 184400.0 -8380.0 -0.57 183960.0 -6300.0 -0.47 -0.7355 -0.9952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J23 compound treatment 186240.0 -6540.0 -0.45 181360.0 -8900.0 -0.66 -0.7836 -0.9814 3187082 PK04_095199 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 J24 compound treatment 183400.0 -9380.0 -0.64 180360.0 -9900.0 -0.74 -0.9731 -0.9975 3068227 PK04_095200 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K01 compound treatment 242720.0 49900.0 3.41 242840.0 52600.0 3.91 5.1748 0.9976 3187514 PK04_095201 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NC6CC6)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K02 compound treatment 203800.0 11000.0 0.75 196520.0 6260.0 0.47 0.8608 0.9735 3187168 PK04_095202 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccc(OC(F)(F)F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K03 compound treatment 245960.0 53200.0 3.63 254760.0 64500.0 4.8 5.9583 0.9904 3068143 PK04_095203 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NC5CC5)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K04 compound treatment 184400.0 -8380.0 -0.57 179040.0 -11200.0 -0.84 -0.9944 -0.9828 3187275 PK04_095204 CN(C)CCCNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K05 compound treatment 277240.0 84500.0 5.76 271440.0 81200.0 6.04 8.3441 0.9997 3187271 PK04_095205 CN(C)CCCNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K06 compound treatment 224880.0 32100.0 2.19 223480.0 33200.0 2.47 3.2959 0.9982 3186561 PK04_095206 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K07 mock treatment 205680.0 12900.0 0.88 198400.0 8140.0 0.61 1.0504 0.9834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K08 mock treatment 194280.0 1500.0 0.1 188280.0 -1980.0 -0.15 -0.0318 -0.177 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K09 compound treatment 201000.0 8220.0 0.56 195040.0 4780.0 0.36 0.6479 0.9758 3068519 PK04_095207 CN(C)CCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K10 compound treatment 209120.0 16300.0 1.11 203840.0 13600.0 1.01 1.5025 0.9988 3068466 PK04_095208 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccccc4C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K11 compound treatment 224240.0 31500.0 2.15 224840.0 34600.0 2.57 3.3366 0.9959 3068556 PK04_095209 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2C5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K12 compound treatment 259320.0 66500.0 4.54 274240.0 84000.0 6.25 7.6275 0.9876 3067978 PK04_095210 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)O)c6ccc(cc6)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K13 compound treatment 207160.0 14400.0 0.98 203200.0 12900.0 0.96 1.3743 1.0 3068499 PK04_095211 COCCCNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K14 compound treatment 261880.0 69100.0 4.71 251560.0 61300.0 4.56 6.5574 0.9999 3068588 PK04_095212 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2CC5(CC6CC7CC(C6)C5)C7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K15 mock treatment 202920.0 10100.0 0.69 199200.0 8940.0 0.67 0.9594 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K16 mock treatment 193200.0 424.0 0.03 200320.0 10100.0 0.75 0.5498 0.7339 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K17 compound treatment 211240.0 18500.0 1.26 209480.0 19200.0 1.43 1.9015 0.998 3068009 PK04_095213 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K18 compound treatment 186480.0 -6300.0 -0.43 184360.0 -5900.0 -0.44 -0.6141 -0.9999 3186498 PK04_095214 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCCCN(C)C)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K19 compound treatment 202000.0 9220.0 0.63 197120.0 6860.0 0.51 0.8056 0.9946 3068472 PK04_095215 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K20 compound treatment 196600.0 3820.0 0.26 188800.0 -1460.0 -0.11 0.1074 0.3801 3187259 PK04_095216 COCCCNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K21 compound treatment 199120.0 6340.0 0.43 193920.0 3660.0 0.27 0.4983 0.9751 3187078 PK04_095217 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccccc5C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K22 compound treatment 204520.0 11700.0 0.8 210040.0 19800.0 1.47 1.607 0.959 3068508 PK04_095218 COc1ccccc1CN2[C@H]([C@H](C(=O)NC3CC3)c4ccccc4C2=O)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K23 mock treatment 184640.0 -8140.0 -0.55 182480.0 -7780.0 -0.58 -0.8018 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 K24 mock treatment 181360.0 -11400.0 -0.78 179600.0 -10700.0 -0.79 -1.1115 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L01 compound treatment 165720.0 -27100.0 -1.84 165120.0 -25100.0 -1.87 -2.6275 -1.0 3187175 PK04_095219 COc1ccccc1CN2[C@H]([C@H](C(=O)NCCCN(C)C)c3ccccc3C2=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L02 compound treatment 206080.0 13300.0 0.91 202880.0 12600.0 0.94 1.3054 0.9998 3186714 PK04_095220 CC(C)NC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L03 compound treatment 200000.0 7220.0 0.49 196720.0 6460.0 0.48 0.6881 0.9999 3067967 PK04_095221 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCc3ccccc3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L04 compound treatment 208480.0 15700.0 1.07 196920.0 6660.0 0.5 1.1075 0.9387 3186429 PK04_095222 CC(C)CN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L05 compound treatment 212680.0 19900.0 1.36 215400.0 25100.0 1.87 2.2825 0.9876 3068540 PK04_095223 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2C5Cc6ccccc6C5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L06 compound treatment 210640.0 17900.0 1.22 206760.0 16500.0 1.23 1.7294 1.0 3186551 PK04_095224 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L07 mock treatment 197640.0 4860.0 0.33 200040.0 9780.0 0.73 0.7491 0.9367 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L08 mock treatment 195600.0 2820.0 0.19 193520.0 3260.0 0.24 0.3076 0.9935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L09 compound treatment 182200.0 -10600.0 -0.72 176600.0 -13700.0 -1.02 -1.2289 -0.9858 3187518 PK04_095225 CN(C)CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L10 compound treatment 214520.0 21700.0 1.48 210920.0 20700.0 1.54 2.1354 0.9998 3068144 PK04_095226 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCc5ccccc5)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L11 compound treatment 201320.0 8540.0 0.58 201400.0 11100.0 0.83 0.9981 0.9851 3187076 PK04_095227 COCCCNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L12 compound treatment 201520.0 8740.0 0.6 197800.0 7540.0 0.56 0.8182 0.9995 3068313 PK04_095228 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L13 compound treatment 199320.0 6540.0 0.45 196760.0 6500.0 0.48 0.6574 0.9992 3187347 PK04_095229 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(C(C)C)C(=O)c3ccccc32)c4ccc(CO)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L14 compound treatment 201560.0 8780.0 0.6 197200.0 6940.0 0.52 0.7886 0.9973 3068194 PK04_095230 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CC(C)C)C4=O)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L15 mock treatment 199680.0 6900.0 0.47 198480.0 8220.0 0.61 0.7653 0.9916 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L16 mock treatment 196400.0 3620.0 0.25 195200.0 4940.0 0.37 0.4346 0.9814 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L17 compound treatment 210480.0 17700.0 1.21 199280.0 9020.0 0.67 1.3281 0.9616 3068510 PK04_095231 COc1ccccc1CN2[C@H]([C@H](C(=O)NCc3ccccc3)c4ccccc4C2=O)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L18 compound treatment 200240.0 7460.0 0.51 202240.0 12000.0 0.89 0.9902 0.9647 3068263 PK04_095232 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C(C)C)[C@@H]2c3ccc(CO)cc3I)Sc4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L19 compound treatment 200800.0 8020.0 0.55 197000.0 6740.0 0.5 0.7414 0.9991 3067958 PK04_095233 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCCN4CCOCC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L20 compound treatment 189440.0 -3340.0 -0.23 189960.0 -303.0 -0.02 -0.1767 -0.7733 3068403 PK04_095234 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L21 compound treatment 216200.0 23400.0 1.6 200760.0 10500.0 0.78 1.6817 0.9459 3187163 PK04_095235 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3cc(F)cc(c3)C(F)(F)F)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L22 compound treatment 191480.0 -1300.0 -0.09 187680.0 -2580.0 -0.19 -0.1984 -0.9378 3186433 PK04_095236 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(CC(F)(F)F)c2c1)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L23 mock treatment 181840.0 -10900.0 -0.75 176880.0 -13400.0 -1.0 -1.2315 -0.9898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 L24 mock treatment 177920.0 -14900.0 -1.01 176200.0 -14100.0 -1.05 -1.4562 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M01 compound treatment 195480.0 2700.0 0.18 190800.0 538.0 0.04 0.1587 0.841 3187444 PK04_095237 CC(C)CNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M02 compound treatment 202480.0 9700.0 0.66 203560.0 13300.0 0.99 1.1676 0.9808 3068593 PK04_095238 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NC3CC3)c4ccccc4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M03 compound treatment 213160.0 20400.0 1.39 210800.0 20500.0 1.53 2.0635 0.9989 3187441 PK04_095239 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M04 compound treatment 194760.0 1980.0 0.14 197880.0 7620.0 0.57 0.4966 0.8519 3068649 PK04_095240 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M05 compound treatment 184120.0 -8660.0 -0.59 177440.0 -12800.0 -0.95 -1.0921 -0.9733 3068152 PK04_095241 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M06 compound treatment 209400.0 16600.0 1.13 202280.0 12000.0 0.89 1.4339 0.9931 3068655 PK04_095242 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M07 compound treatment 212720.0 19900.0 1.36 208440.0 18200.0 1.35 1.9181 1.0 3068005 PK04_095243 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M08 compound treatment 218520.0 25700.0 1.76 215520.0 25300.0 1.88 2.5703 0.9994 3187084 PK04_095244 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccccc5Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M09 mock treatment 208480.0 15700.0 1.07 202880.0 12600.0 0.94 1.4211 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M10 mock treatment 205600.0 12800.0 0.87 205200.0 14900.0 1.11 1.4044 0.9929 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M11 compound treatment 263160.0 70400.0 4.8 249880.0 59600.0 4.44 6.5306 0.9992 3186422 PK04_095245 CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M12 compound treatment 202960.0 10200.0 0.69 194680.0 4420.0 0.33 0.7235 0.9417 3068142 PK04_095246 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M13 mock treatment 195720.0 2940.0 0.2 206360.0 16100.0 1.2 0.9891 0.8142 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M14 mock treatment 203240.0 10500.0 0.71 200680.0 10400.0 0.78 1.0527 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M15 compound treatment 216080.0 23300.0 1.59 214840.0 24600.0 1.83 2.4169 0.9975 3068557 PK04_095247 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2C5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M16 compound treatment 225800.0 33000.0 2.25 218200.0 27900.0 2.08 3.0623 0.9992 3187170 PK04_095248 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2OC)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M17 compound treatment 220560.0 27800.0 1.89 213440.0 23200.0 1.73 2.5592 0.9989 3187431 PK04_095249 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M18 compound treatment 218960.0 26200.0 1.79 212000.0 21700.0 1.62 2.4063 0.9988 3187074 PK04_095250 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5cc(cc(c5)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M19 compound treatment 204160.0 11400.0 0.78 200720.0 10500.0 0.78 1.0992 1.0 3068552 PK04_095251 CC(C)NC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M20 compound treatment 245560.0 52800.0 3.6 240560.0 50300.0 3.74 5.1917 0.9998 3068014 PK04_095252 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)O)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M21 compound treatment 203720.0 10900.0 0.75 201080.0 10800.0 0.81 1.0969 0.9993 3187086 PK04_095253 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M22 compound treatment 206480.0 13700.0 0.93 198960.0 8700.0 0.65 1.1184 0.9839 3187428 PK04_095254 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M23 compound treatment 183840.0 -8940.0 -0.61 184680.0 -5580.0 -0.42 -0.7246 -0.9826 3187081 PK04_095255 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 M24 compound treatment 214440.0 21700.0 1.48 210720.0 20500.0 1.52 2.121 0.9999 3068003 PK04_095256 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N01 compound treatment 218040.0 25300.0 1.72 205280.0 15000.0 1.12 2.0083 0.9781 3187360 PK04_095257 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N02 compound treatment 198200.0 5420.0 0.37 193880.0 3620.0 0.27 0.4519 0.9878 3068231 PK04_095258 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N03 compound treatment 210920.0 18100.0 1.24 209960.0 19700.0 1.47 1.9113 0.9964 3068544 PK04_095259 CC(C)NC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N04 compound treatment 284640.0 91900.0 6.26 285640.0 95400.0 7.1 9.4481 0.9981 3187527 PK04_095260 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)O)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N05 compound treatment 207760.0 15000.0 1.02 203760.0 13500.0 1.0 1.4327 1.0 3187260 PK04_095261 CCCNC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N06 compound treatment 204480.0 11700.0 0.8 212880.0 22600.0 1.68 1.7546 0.9418 3186724 PK04_095262 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N07 compound treatment 212720.0 19900.0 1.36 210240.0 20000.0 1.49 2.0129 0.999 3068501 PK04_095263 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N08 compound treatment 216800.0 24000.0 1.64 218560.0 28300.0 2.11 2.6474 0.9923 3186871 PK04_095264 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N09 mock treatment 209800.0 17000.0 1.16 203160.0 12900.0 0.96 1.4995 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N10 mock treatment 210800.0 18000.0 1.23 206560.0 16300.0 1.21 1.7266 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N11 compound treatment 212200.0 19400.0 1.32 208680.0 18400.0 1.37 1.9057 0.9999 3187070 PK04_095265 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N12 compound treatment 217440.0 24700.0 1.68 206040.0 15800.0 1.17 2.0194 0.9846 3186804 PK04_095266 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N13 mock treatment 199880.0 7100.0 0.48 198080.0 7820.0 0.58 0.7539 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N14 mock treatment 203280.0 10500.0 0.72 202040.0 11800.0 0.88 1.1262 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N15 compound treatment 233800.0 41000.0 2.8 222600.0 32300.0 2.41 3.6796 0.9972 3186424 PK04_095267 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCCN6CCOCC6)c7ccc(cc7)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N16 compound treatment 200080.0 7300.0 0.5 201720.0 11500.0 0.85 0.9551 0.9672 3068226 PK04_095268 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N17 compound treatment 236440.0 43700.0 2.98 230000.0 39700.0 2.96 4.1963 1.0 3068455 PK04_095269 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N18 compound treatment 209800.0 17000.0 1.16 203600.0 13300.0 0.99 1.5226 0.997 3068137 PK04_095270 CN(C)CCCN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N19 compound treatment 191640.0 -1140.0 -0.08 183320.0 -6940.0 -0.52 -0.4201 -0.8041 3068647 PK04_095271 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N20 compound treatment 208560.0 15800.0 1.08 212960.0 22700.0 1.69 1.9555 0.9763 3186492 PK04_095272 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N21 compound treatment 199240.0 6460.0 0.44 198760.0 8500.0 0.63 0.7588 0.9844 3067959 PK04_095273 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N22 compound treatment 193280.0 504.0 0.03 191840.0 1580.0 0.12 0.1073 0.8773 3187526 PK04_095274 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)O)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N23 compound treatment 204640.0 11900.0 0.81 196560.0 6300.0 0.47 0.9034 0.9663 3068468 PK04_095275 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 N24 compound treatment 183480.0 -9300.0 -0.63 180080.0 -10200.0 -0.76 -0.984 -0.996 3068222 PK04_095276 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O01 compound treatment 227760.0 35000.0 2.39 222000.0 31700.0 2.36 3.3568 1.0 3068590 PK04_095277 CC(C)NC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O02 compound treatment 216480.0 23700.0 1.62 199400.0 9140.0 0.68 1.6236 0.926 3067977 PK04_095278 COCCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O03 compound treatment 204400.0 11600.0 0.79 192560.0 2300.0 0.17 0.6813 0.8403 3068512 PK04_095279 COc1ccccc1CN2[C@H]([C@H](C(=O)NCC(F)(F)F)c3ccccc3C2=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O04 compound treatment 248960.0 56200.0 3.83 224880.0 34600.0 2.58 4.5304 0.9814 3068637 PK04_095280 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O05 compound treatment 221240.0 28500.0 1.94 218960.0 28700.0 2.14 2.8825 0.9989 3068459 PK04_095281 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4cc(cc(c4)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O06 compound treatment 215240.0 22500.0 1.53 212040.0 21800.0 1.62 2.2291 0.9996 3187520 PK04_095282 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O07 compound treatment 216640.0 23900.0 1.63 215160.0 24900.0 1.85 2.4608 0.9979 3186989 PK04_095283 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O08 compound treatment 204360.0 11600.0 0.79 195480.0 5220.0 0.39 0.833 0.9466 3187364 PK04_095284 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O09 compound treatment 210920.0 18100.0 1.24 203480.0 13200.0 0.98 1.5703 0.9936 3068604 PK04_095285 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O10 compound treatment 190440.0 -2340.0 -0.16 191400.0 1140.0 0.08 -0.0527 -0.2924 3187362 PK04_095286 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O11 mock treatment 196040.0 3260.0 0.22 193080.0 2820.0 0.21 0.3056 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O12 mock treatment 193640.0 864.0 0.06 192320.0 2060.0 0.15 0.15 0.9139 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O13 compound treatment 208000.0 15200.0 1.04 216760.0 26500.0 1.97 2.1284 0.9551 3068644 PK04_095287 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O14 compound treatment 209160.0 16400.0 1.12 206320.0 16100.0 1.2 1.6349 0.9994 3068464 PK04_095288 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccccc5C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O15 compound treatment 248080.0 55300.0 3.77 247680.0 57400.0 4.27 5.6879 0.9981 3187516 PK04_095289 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCc6ccccc6)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O16 compound treatment 208400.0 15600.0 1.07 194120.0 3860.0 0.29 0.9562 0.8668 3187164 PK04_095290 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5cc(F)cc(c5)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O17 compound treatment 201160.0 8380.0 0.57 196880.0 6620.0 0.49 0.7525 0.9972 3187177 PK04_095291 CC(C)CNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O18 compound treatment 185080.0 -7700.0 -0.52 181360.0 -8900.0 -0.66 -0.8395 -0.9933 3068546 PK04_095292 CN(C)CCCNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O19 compound treatment 208560.0 15800.0 1.08 200240.0 9980.0 0.74 1.286 0.9836 3187256 PK04_095293 CC(C)CNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O20 compound treatment 197040.0 4260.0 0.29 194120.0 3860.0 0.29 0.4086 1.0 3187088 PK04_095294 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O21 compound treatment 192880.0 104.0 0.01 193720.0 3460.0 0.26 0.187 0.7264 3186494 PK04_095295 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCC(C)C)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O22 compound treatment 186200.0 -6580.0 -0.45 180320.0 -9940.0 -0.74 -0.8403 -0.9712 3187161 PK04_095296 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O23 compound treatment 187320.0 -5460.0 -0.37 185720.0 -4540.0 -0.34 -0.5021 -0.9989 3187267 PK04_095297 CC(C)CNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 O24 compound treatment 183960.0 -8820.0 -0.6 183400.0 -6860.0 -0.51 -0.7861 -0.9967 3068502 PK04_095298 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P01 compound treatment 204200.0 11400.0 0.78 199760.0 9500.0 0.71 1.0506 0.9988 3068591 PK04_095299 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2CC4(CC5CC6CC(C5)C4)C6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P02 compound treatment 216760.0 24000.0 1.64 218360.0 28100.0 2.09 2.635 0.9926 3187521 PK04_095300 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P03 compound treatment 221600.0 28800.0 1.97 210760.0 20500.0 1.53 2.4683 0.9922 3186990 PK04_095301 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P04 compound treatment 201720.0 8940.0 0.61 201360.0 11100.0 0.83 1.0152 0.9889 3186985 PK04_095302 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P05 compound treatment 237320.0 44500.0 3.04 226520.0 36300.0 2.7 4.0556 0.9983 3067579 PK04_095303 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c6ccc(cc6)[N+](=O)[O-])c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P06 compound treatment 202160.0 9380.0 0.64 202400.0 12100.0 0.9 1.0912 0.9857 3186975 PK04_095304 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P07 compound treatment 208840.0 16100.0 1.1 212400.0 22100.0 1.65 1.9395 0.9803 3068548 PK04_095305 CC(C)CNC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P08 compound treatment 211760.0 19000.0 1.29 199480.0 9220.0 0.69 1.4003 0.9559 3067563 PK04_095306 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(CCN5CCOCC5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P09 compound treatment 208400.0 15600.0 1.07 195960.0 5700.0 0.42 1.0531 0.9185 3067961 PK04_095307 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCc4ccccc4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P10 compound treatment 214040.0 21300.0 1.45 216040.0 25800.0 1.92 2.3817 0.9905 3068015 PK04_095308 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P11 mock treatment 191400.0 -1380.0 -0.09 192240.0 1980.0 0.15 0.0378 0.2163 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P12 mock treatment 200320.0 7540.0 0.51 193640.0 3380.0 0.25 0.5415 0.9458 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P13 compound treatment 198720.0 5940.0 0.41 190520.0 258.0 0.02 0.3001 0.7397 3187510 PK04_095309 CC(C)NC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P14 compound treatment 231880.0 39100.0 2.67 231520.0 41300.0 3.07 4.0564 0.9975 3186495 PK04_095310 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCCN5CCOCC5)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P15 compound treatment 200240.0 7460.0 0.51 193760.0 3500.0 0.26 0.5439 0.9515 3187437 PK04_095311 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P16 compound treatment 198320.0 5540.0 0.38 185800.0 -4460.0 -0.33 0.0324 0.0645 3186625 PK04_095312 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(C(C)C)C4=O)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P17 compound treatment 211240.0 18500.0 1.26 207520.0 17300.0 1.28 1.7984 0.9999 3068541 PK04_095313 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2C5Cc6ccccc6C5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P18 compound treatment 193280.0 504.0 0.03 188480.0 -1780.0 -0.13 -0.0695 -0.5071 3186878 PK04_095314 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NC6CC6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P19 compound treatment 209400.0 16600.0 1.13 200400.0 10100.0 0.75 1.3349 0.9804 3187513 PK04_095315 CC(C)CNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P20 compound treatment 194360.0 1580.0 0.11 185920.0 -4340.0 -0.32 -0.1522 -0.4465 3068271 PK04_095316 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCc6ccccc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P21 compound treatment 197680.0 4900.0 0.33 189800.0 -463.0 -0.03 0.2121 0.631 3068008 PK04_095317 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P22 compound treatment 181880.0 -10900.0 -0.74 175680.0 -14600.0 -1.09 -1.2927 -0.9829 3068262 PK04_095318 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P23 compound treatment 190160.0 -2620.0 -0.18 186560.0 -3700.0 -0.28 -0.3209 -0.9778 3068469 PK04_095319 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccccc5Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2095 P24 compound treatment 174440.0 -18300.0 -1.25 175040.0 -15200.0 -1.13 -1.6851 -0.9988 3186794 PK04_095320 CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A01 compound treatment 184640.0 -10200.0 -0.69 207440.0 14700.0 1.09 0.2844 0.2195 3186490 PK04_096001 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A02 compound treatment 190120.0 -4680.0 -0.32 182520.0 -10200.0 -0.76 -0.7629 -0.9257 3186641 PK04_096002 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A03 compound treatment 186280.0 -8520.0 -0.58 184560.0 -8170.0 -0.61 -0.8406 -0.9997 3068261 PK04_096003 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NC4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A04 compound treatment 182480.0 -12300.0 -0.84 179680.0 -13100.0 -0.97 -1.2807 -0.9974 3186971 PK04_096004 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A05 compound treatment 183240.0 -11600.0 -0.79 181360.0 -11400.0 -0.85 -1.1556 -0.9994 3186883 PK04_096005 COCCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A06 compound treatment 181360.0 -13400.0 -0.92 178880.0 -13900.0 -1.03 -1.3768 -0.9983 3068309 PK04_096006 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A07 compound treatment 185440.0 -9360.0 -0.64 185320.0 -7410.0 -0.55 -0.8411 -0.9974 3186716 PK04_096007 COCCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A08 compound treatment 235760.0 41000.0 2.79 220960.0 28200.0 2.1 3.4604 0.9902 3068367 PK04_096008 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)Sc6ccc(C)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A09 compound treatment 182520.0 -12300.0 -0.84 173000.0 -19700.0 -1.47 -1.6303 -0.9645 3068224 PK04_096009 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A10 compound treatment 185800.0 -9000.0 -0.61 178600.0 -14100.0 -1.05 -1.1774 -0.9671 3186633 PK04_096010 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5C(F)(F)F)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A11 compound treatment 184440.0 -10400.0 -0.71 181000.0 -11700.0 -0.87 -1.1167 -0.9945 3186986 PK04_096011 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A12 compound treatment 193040.0 -1760.0 -0.12 191320.0 -1410.0 -0.1 -0.159 -0.9978 3186640 PK04_096012 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A13 mock treatment 184840.0 -9960.0 -0.68 178000.0 -14700.0 -1.1 -1.2553 -0.9735 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A14 mock treatment 179560.0 -15200.0 -1.04 179000.0 -13700.0 -1.02 -1.4572 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A15 compound treatment 183400.0 -11400.0 -0.78 179400.0 -13300.0 -0.99 -1.251 -0.9927 3186881 PK04_096013 CC(C)NC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A16 compound treatment 192320.0 -2480.0 -0.17 186360.0 -6370.0 -0.47 -0.4547 -0.9035 3186790 PK04_096014 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A17 compound treatment 180960.0 -13800.0 -0.94 178160.0 -14600.0 -1.08 -1.4339 -0.9976 3186485 PK04_096015 CC(C)CN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A18 compound treatment 186880.0 -7920.0 -0.54 179640.0 -13100.0 -0.97 -1.0706 -0.9612 3186802 PK04_096016 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A19 compound treatment 181880.0 -12900.0 -0.88 179960.0 -12800.0 -0.95 -1.2948 -0.9993 3068405 PK04_096017 CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A20 compound treatment 189200.0 -5600.0 -0.38 183960.0 -8770.0 -0.65 -0.7315 -0.9673 3068141 PK04_096018 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A21 compound treatment 184880.0 -9920.0 -0.68 183360.0 -9370.0 -0.7 -0.9713 -0.9999 3186624 PK04_096019 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5OC)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A22 compound treatment 184400.0 -10400.0 -0.71 178920.0 -13800.0 -1.03 -1.2281 -0.9836 3068200 PK04_096020 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CCCN(C)C)C4=O)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A23 compound treatment 177960.0 -16800.0 -1.15 173600.0 -19100.0 -1.42 -1.8185 -0.9943 3068358 PK04_096021 CC(C)CNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 A24 compound treatment 173440.0 -21400.0 -1.46 172960.0 -19800.0 -1.47 -2.0701 -1.0 3068371 PK04_096022 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B01 compound treatment 178680.0 -16100.0 -1.1 178400.0 -14300.0 -1.07 -1.5312 -0.9999 3187511 PK04_096023 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCC(F)(F)F)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B02 compound treatment 195160.0 361.0 0.02 192160.0 -570.0 -0.04 -0.0126 -0.2565 3187030 PK04_096024 OCCCc1cc[n+](Cc2cccc(OC(F)(F)F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B03 compound treatment 186640.0 -8160.0 -0.56 183160.0 -9570.0 -0.71 -0.897 -0.9925 3187169 PK04_096025 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B04 compound treatment 223920.0 29100.0 1.99 214080.0 21400.0 1.59 2.5275 0.9939 3068853 PK04_096026 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B05 compound treatment 228720.0 33900.0 2.31 226720.0 34000.0 2.53 3.4241 0.999 3068457 PK04_096027 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5cc(cc(c5)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B06 compound treatment 240560.0 45800.0 3.12 234160.0 41400.0 3.08 4.3864 1.0 3068854 PK04_096028 C[n+]1ccc2ccc(O)cc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B07 compound treatment 182720.0 -12100.0 -0.82 178600.0 -14100.0 -1.05 -1.3259 -0.9927 3187352 PK04_096029 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NCCN4CCOCC4)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B08 compound treatment 224000.0 29200.0 1.99 221480.0 28800.0 2.14 2.9208 0.9994 3187112 PK04_096030 COc1cc2CC[N+](=Cc2cc1O)Cc3cc4OCOc4cc3Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B09 compound treatment 209200.0 14400.0 0.98 177920.0 -14800.0 -1.1 -0.0852 -0.0577 3068505 PK04_096031 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B10 compound treatment 187800.0 -7000.0 -0.48 189680.0 -3050.0 -0.23 -0.4979 -0.9423 3068855 PK04_096032 C[n+]1ccc(CCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B11 compound treatment 203760.0 8960.0 0.61 201600.0 8870.0 0.66 0.8988 0.9993 3068374 PK04_096033 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B12 compound treatment 245720.0 50900.0 3.47 242480.0 49800.0 3.7 5.0731 0.9995 3187113 PK04_096034 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(C=C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B13 mock treatment 184720.0 -10100.0 -0.69 180360.0 -12400.0 -0.92 -1.1369 -0.9896 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B14 mock treatment 176600.0 -18200.0 -1.24 175960.0 -16800.0 -1.25 -1.7599 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B15 compound treatment 182760.0 -12000.0 -0.82 173840.0 -18900.0 -1.41 -1.5745 -0.9672 3187255 PK04_096035 COCCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B16 compound treatment 228600.0 33800.0 2.3 229640.0 36900.0 2.75 3.572 0.9962 3068856 PK04_096036 Oc1ccc2cc[n+](Cc3sc4ccccc4c3Cl)cc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B17 compound treatment 183280.0 -11500.0 -0.79 181600.0 -11100.0 -0.83 -1.141 -0.9996 3068608 PK04_096037 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B18 compound treatment 222520.0 27700.0 1.89 219840.0 27100.0 2.02 2.7631 0.9995 3187114 PK04_096038 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(C5CC5)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B19 compound treatment 195000.0 201.0 0.01 193560.0 830.0 0.06 0.0534 0.8436 3187171 PK04_096039 COc1ccccc1CN2[C@H]([C@H](C(=O)NCC(C)C)c3ccccc3C2=O)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B20 compound treatment 220800.0 26000.0 1.77 217920.0 25200.0 1.87 2.5792 0.9996 3068857 PK04_096040 OCCCc1cc[n+](Cc2ccc(o2)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B21 compound treatment 185640.0 -9160.0 -0.62 177800.0 -14900.0 -1.11 -1.2273 -0.9628 3068424 PK04_096041 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B22 compound treatment 208080.0 13300.0 0.91 214840.0 22100.0 1.65 1.8039 0.9604 3187115 PK04_096042 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B23 compound treatment 182280.0 -12500.0 -0.85 179960.0 -12800.0 -0.95 -1.2756 -0.9986 3187072 PK04_096043 CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 B24 compound treatment 201600.0 6800.0 0.46 206560.0 13800.0 1.03 1.0557 0.9351 3187116 PK04_096044 COC(=O)C1=CN(C)C(C=C(C=C1C(=O)OC)c2ccc(CO)cc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C01 compound treatment 184440.0 -10400.0 -0.71 178080.0 -14700.0 -1.09 -1.2704 -0.9779 3068218 PK04_096045 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C02 compound treatment 195200.0 401.0 0.03 186160.0 -6570.0 -0.49 -0.3264 -0.6665 3186566 PK04_096046 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C03 compound treatment 209880.0 15100.0 1.03 206120.0 13400.0 1.0 1.4317 0.9999 3186549 PK04_096047 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C04 compound treatment 189480.0 -5320.0 -0.36 188320.0 -4410.0 -0.33 -0.4885 -0.9988 3186726 PK04_096048 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C05 compound treatment 192960.0 -1840.0 -0.13 186320.0 -6410.0 -0.48 -0.426 -0.8636 3186792 PK04_096049 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C06 compound treatment 187760.0 -7040.0 -0.48 188400.0 -4330.0 -0.32 -0.5672 -0.9812 3186987 PK04_096050 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C07 compound treatment 194760.0 -38.8 0.0 192000.0 -730.0 -0.05 -0.0403 -0.7406 3068275 PK04_096051 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C08 compound treatment 220000.0 25200.0 1.72 214200.0 21500.0 1.6 2.3448 0.9993 3186560 PK04_096052 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C09 compound treatment 243520.0 48700.0 3.32 209080.0 16400.0 1.22 3.2092 0.9072 3068147 PK04_096053 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C10 compound treatment 182320.0 -12500.0 -0.85 185320.0 -7410.0 -0.55 -0.9916 -0.978 3186976 PK04_096054 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C11 mock treatment 200880.0 6080.0 0.41 196000.0 3270.0 0.24 0.4653 0.9678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C12 mock treatment 186680.0 -8120.0 -0.55 189080.0 -3650.0 -0.27 -0.5835 -0.9463 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C13 compound treatment 191440.0 -3360.0 -0.23 200360.0 7630.0 0.57 0.2396 0.3914 3186974 PK04_096055 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C14 compound treatment 180360.0 -14400.0 -0.98 186520.0 -6210.0 -0.46 -1.0229 -0.9406 3186876 PK04_096056 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C15 mock treatment 189960.0 -4840.0 -0.33 185520.0 -7210.0 -0.54 -0.6127 -0.9727 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C16 mock treatment 184880.0 -9920.0 -0.68 182000.0 -10700.0 -0.8 -1.0429 -0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C17 compound treatment 195160.0 361.0 0.02 202640.0 9910.0 0.74 0.539 0.7303 3186553 PK04_096057 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C18 compound treatment 186160.0 -8640.0 -0.59 190600.0 -2130.0 -0.16 -0.5286 -0.8666 3186634 PK04_096058 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C19 compound treatment 188200.0 -6600.0 -0.45 185560.0 -7170.0 -0.53 -0.6955 -0.9964 3186638 PK04_096059 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C20 compound treatment 189560.0 -5240.0 -0.36 184280.0 -8450.0 -0.63 -0.6973 -0.9641 3068219 PK04_096060 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C21 compound treatment 202880.0 8080.0 0.55 210600.0 17900.0 1.33 1.33 0.9239 3068151 PK04_096061 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C22 compound treatment 178120.0 -16700.0 -1.14 180480.0 -12300.0 -0.91 -1.4487 -0.994 3068158 PK04_096062 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C23 compound treatment 178640.0 -16200.0 -1.1 173040.0 -19700.0 -1.47 -1.8152 -0.9901 3186800 PK04_096063 COCCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 C24 compound treatment 172440.0 -22400.0 -1.52 168600.0 -24100.0 -1.8 -2.3478 -0.9967 3068376 PK04_096064 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D01 compound treatment 193640.0 -1160.0 -0.08 188040.0 -4690.0 -0.35 -0.3027 -0.8457 3068407 PK04_096065 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D02 compound treatment 179960.0 -14800.0 -1.01 182680.0 -10100.0 -0.75 -1.2443 -0.989 3187117 PK04_096066 CN1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5ccc(CN6CCCC6)cc5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D03 compound treatment 259640.0 64800.0 4.42 252680.0 60000.0 4.46 6.2809 1.0 3187274 PK04_096067 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2CC5(CC6CC7CC(C6)C5)C7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D04 compound treatment 230200.0 35400.0 2.41 224240.0 31500.0 2.35 3.3649 0.9999 3068858 PK04_096068 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(C=C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D05 compound treatment 207360.0 12600.0 0.86 192960.0 230.0 0.02 0.6177 0.7211 3187075 PK04_096069 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D06 compound treatment 215920.0 21100.0 1.44 205480.0 12800.0 0.95 1.6892 0.9795 3187118 PK04_096070 OCCCC1=CC(N(Cc2cc3OCOc3cc2Br)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C1)c6ccc(CN7CCCC7)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D07 compound treatment 194480.0 -319.0 -0.02 184840.0 -7890.0 -0.59 -0.4306 -0.7328 3068634 PK04_096071 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D08 compound treatment 214520.0 19700.0 1.34 214240.0 21500.0 1.6 2.0828 0.9962 3068859 PK04_096072 OCc1ccc(cc1)c2cc[n+](Cc3ccc(o3)[N+](=O)[O-])cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D09 compound treatment 261360.0 66600.0 4.54 239800.0 47100.0 3.5 5.686 0.9918 3067975 PK04_096073 CC(C)NC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D10 compound treatment 260000.0 65200.0 4.45 246240.0 53500.0 3.98 5.9594 0.9985 3068860 PK04_096074 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D11 mock treatment 185200.0 -9600.0 -0.65 184800.0 -7930.0 -0.59 -0.8801 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D12 mock treatment 189000.0 -5800.0 -0.4 187440.0 -5290.0 -0.39 -0.5579 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D13 compound treatment 206760.0 12000.0 0.82 202160.0 9430.0 0.7 1.0729 0.9972 3187429 PK04_096075 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D14 compound treatment 187560.0 -7240.0 -0.49 182440.0 -10300.0 -0.77 -0.8905 -0.9774 3187119 PK04_096076 CN1C(=O)C2C(C3C(C4CC4)N(Cc5cccc(OC(F)(F)F)c5)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D15 mock treatment 183200.0 -11600.0 -0.79 186120.0 -6610.0 -0.49 -0.907 -0.9739 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D16 mock treatment 187960.0 -6840.0 -0.47 182840.0 -9890.0 -0.74 -0.8502 -0.9757 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D17 compound treatment 189480.0 -5320.0 -0.36 191320.0 -1410.0 -0.1 -0.3306 -0.8758 3187348 PK04_096077 CC(C)NC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D18 compound treatment 254400.0 59600.0 4.06 252360.0 59600.0 4.44 6.0115 0.999 3068861 PK04_096078 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C4CC4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D19 compound treatment 186440.0 -8360.0 -0.57 188960.0 -3770.0 -0.28 -0.6014 -0.9467 3187354 PK04_096079 CC(C)NC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D20 compound treatment 205680.0 10900.0 0.74 207440.0 14700.0 1.09 1.2987 0.982 3187120 PK04_096080 OCc1ccc(cc1)c2cc[n+](Cc3sc4ccccc4c3Cl)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D21 compound treatment 188720.0 -6080.0 -0.41 186600.0 -6130.0 -0.46 -0.6157 -0.9988 3187433 PK04_096081 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D22 compound treatment 255480.0 60700.0 4.14 251400.0 58700.0 4.37 6.013 0.9996 3068862 PK04_096082 COc1cc2CCN(C)C(C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D23 compound treatment 201680.0 6880.0 0.47 200880.0 8150.0 0.61 0.7606 0.9919 3068462 PK04_096083 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccccc5C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 D24 compound treatment 171520.0 -23300.0 -1.59 174160.0 -18600.0 -1.38 -2.0995 -0.9976 3187121 PK04_096084 COC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(C=C1C(=O)OC)c4ccc(CO)cc4)C5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E01 mock treatment 189240.0 -5560.0 -0.38 185600.0 -7130.0 -0.53 -0.6432 -0.9864 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E02 mock treatment 189760.0 -5040.0 -0.34 182800.0 -9930.0 -0.74 -0.7655 -0.9393 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E03 compound treatment 236760.0 42000.0 2.86 219040.0 26300.0 1.96 3.4075 0.9829 3186708 PK04_096085 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E04 compound treatment 240440.0 45600.0 3.11 234680.0 42000.0 3.12 4.408 1.0 3186710 PK04_096086 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E05 compound treatment 214720.0 19900.0 1.36 200840.0 8110.0 0.6 1.3872 0.9333 3186888 PK04_096087 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E06 compound treatment 201120.0 6320.0 0.43 200640.0 7910.0 0.59 0.721 0.9882 3186565 PK04_096088 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E07 compound treatment 206760.0 12000.0 0.82 198960.0 6230.0 0.46 0.9045 0.9642 3186983 PK04_096089 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E08 compound treatment 208480.0 13700.0 0.93 205200.0 12500.0 0.93 1.3158 1.0 3067581 PK04_096090 CCCN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E09 mock treatment 199040.0 4240.0 0.29 195520.0 2790.0 0.21 0.3513 0.9868 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E10 mock treatment 193280.0 -1520.0 -0.1 197640.0 4910.0 0.37 0.1852 0.4876 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E11 compound treatment 199600.0 4800.0 0.33 194720.0 1990.0 0.15 0.3362 0.9357 3186717 PK04_096091 CC(C)CNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E12 compound treatment 205960.0 11200.0 0.76 205000.0 12300.0 0.91 1.1838 0.9959 3068221 PK04_096092 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E13 compound treatment 210440.0 15600.0 1.07 192600.0 -130.0 -0.01 0.7472 0.7007 3068273 PK04_096093 CN(C)CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E14 compound treatment 211160.0 16400.0 1.12 207280.0 14600.0 1.08 1.5545 0.9999 3068377 PK04_096094 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E15 compound treatment 203840.0 9040.0 0.62 199640.0 6910.0 0.51 0.7995 0.9959 3068408 PK04_096095 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E16 compound treatment 203720.0 8920.0 0.61 202640.0 9910.0 0.74 0.9516 0.9954 3186635 PK04_096096 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E17 mock treatment 191840.0 -2960.0 -0.2 197440.0 4710.0 0.35 0.1052 0.2602 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E18 mock treatment 195840.0 1040.0 0.07 198480.0 5750.0 0.43 0.3528 0.8133 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E19 compound treatment 190160.0 -4640.0 -0.32 197680.0 4950.0 0.37 0.0369 0.076 3186791 PK04_096097 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E20 compound treatment 199080.0 4280.0 0.29 197240.0 4510.0 0.34 0.4437 0.9976 3068233 PK04_096098 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E21 compound treatment 203280.0 8480.0 0.58 198480.0 5750.0 0.43 0.7115 0.989 3186719 PK04_096099 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)Sc6ccc(C)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E22 compound treatment 192480.0 -2320.0 -0.16 195720.0 2990.0 0.22 0.0456 0.167 3186789 PK04_096100 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E23 compound treatment 195480.0 681.0 0.05 188440.0 -4290.0 -0.32 -0.1929 -0.598 3186803 PK04_096101 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 E24 compound treatment 175560.0 -19200.0 -1.31 176400.0 -16300.0 -1.22 -1.7869 -0.9993 3186711 PK04_096102 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F01 mock treatment 183240.0 -11600.0 -0.79 182280.0 -10500.0 -0.78 -1.1072 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F02 mock treatment 189520.0 -5280.0 -0.36 185600.0 -7130.0 -0.53 -0.6297 -0.9821 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F03 compound treatment 218000.0 23200.0 1.58 211960.0 19200.0 1.43 2.1305 0.9988 3068521 PK04_096103 CCCNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F04 compound treatment 237360.0 42600.0 2.9 237560.0 44800.0 3.34 4.4111 0.9976 3187122 PK04_096104 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F05 compound treatment 220920.0 26100.0 1.78 211600.0 18900.0 1.4 2.2523 0.9931 3068461 PK04_096105 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F06 compound treatment 236200.0 41400.0 2.82 227800.0 35100.0 2.61 3.8415 0.9992 3068863 PK04_096106 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(c5ccc(CN6CCCC6)cc5)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F07 compound treatment 202880.0 8080.0 0.55 196120.0 3390.0 0.25 0.568 0.9373 3187077 PK04_096107 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F08 compound treatment 202360.0 7560.0 0.52 197120.0 4390.0 0.33 0.5956 0.9758 3187123 PK04_096108 CN/1C(C=C(CCCO)C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F09 mock treatment 195240.0 441.0 0.03 188880.0 -3850.0 -0.29 -0.1813 -0.6294 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F10 mock treatment 192040.0 -2760.0 -0.19 198520.0 5790.0 0.43 0.1717 0.3652 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F11 compound treatment 188200.0 -6600.0 -0.45 194880.0 2150.0 0.16 -0.205 -0.4293 3187438 PK04_096109 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F12 compound treatment 241880.0 47100.0 3.21 245360.0 52600.0 3.92 5.0395 0.9951 3187124 PK04_096110 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(C=C1C(=O)OC)c3ccc(CO)cc3)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F13 compound treatment 218600.0 23800.0 1.62 205160.0 12400.0 0.93 1.8016 0.9645 3068559 PK04_096111 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2C4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F14 compound treatment 223280.0 28500.0 1.94 222600.0 29900.0 2.22 2.945 0.9977 3068864 PK04_096112 COC(=O)C1=CN(C)C(C=C(CCCO)C=C1C(=O)OC)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F15 compound treatment 222680.0 27900.0 1.9 215320.0 22600.0 1.68 2.533 0.9981 3186801 PK04_096113 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F16 compound treatment 240120.0 45300.0 3.09 220640.0 27900.0 2.08 3.6537 0.9813 3187125 PK04_096114 COC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(CCCO)C=C1C(=O)OC)C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F17 mock treatment 195280.0 481.0 0.03 191360.0 -1370.0 -0.1 -0.0489 -0.4565 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F18 mock treatment 190240.0 -4560.0 -0.31 194760.0 2030.0 0.15 -0.1129 -0.3268 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F19 compound treatment 201760.0 6960.0 0.47 200000.0 7270.0 0.54 0.7182 0.9979 3186718 PK04_096115 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NC6CC6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F20 compound treatment 277080.0 82300.0 5.61 272400.0 79700.0 5.93 8.1595 0.9996 3068865 PK04_096116 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F21 compound treatment 216600.0 21800.0 1.49 217760.0 25000.0 1.86 2.3683 0.9937 3067569 PK04_096117 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F22 compound treatment 263120.0 68300.0 4.66 258880.0 66200.0 4.92 6.775 0.9996 3187126 PK04_096118 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C=C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F23 compound treatment 184560.0 -10200.0 -0.7 183800.0 -8930.0 -0.66 -0.9636 -0.9997 3068643 PK04_096119 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 F24 compound treatment 210560.0 15800.0 1.07 216240.0 23500.0 1.75 1.9971 0.9726 3187127 PK04_096120 CN/1C(C=C(C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CO)cc4)c5cccs5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G01 compound treatment 197320.0 2520.0 0.17 191720.0 -1010.0 -0.08 0.0684 0.3645 3186434 PK04_096121 CN(C)CCCN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G02 compound treatment 200040.0 5240.0 0.36 197760.0 5030.0 0.37 0.5174 0.9997 3067602 PK04_096122 CC(C)N1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G03 mock treatment 190080.0 -4720.0 -0.32 194480.0 1750.0 0.13 -0.1354 -0.3901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G04 mock treatment 201760.0 6960.0 0.47 191600.0 -1130.0 -0.08 0.2761 0.5729 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G05 compound treatment 257640.0 62800.0 4.28 241880.0 49200.0 3.66 5.6161 0.9969 3068238 PK04_096123 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G06 compound treatment 213880.0 19100.0 1.3 207160.0 14400.0 1.07 1.6793 0.9955 3068315 PK04_096124 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G07 compound treatment 208040.0 13200.0 0.9 197480.0 4750.0 0.35 0.8883 0.9163 3186805 PK04_096125 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G08 compound treatment 222920.0 28100.0 1.92 224800.0 32100.0 2.39 3.0435 0.9941 3186712 PK04_096126 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G09 compound treatment 197480.0 2680.0 0.18 200680.0 7950.0 0.59 0.5476 0.8843 3068360 PK04_096127 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G10 compound treatment 208920.0 14100.0 0.96 206280.0 13600.0 1.01 1.3939 0.9997 3186431 PK04_096128 COc1ccc(CCN2C(=O)[C@]3(CC(=O)N([C@@H]3c4ccc(CO)cc24)C5CCCCC5)c6ccc(cc6)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G11 compound treatment 245800.0 51000.0 3.48 231240.0 38500.0 2.87 4.4854 0.9954 3186642 PK04_096129 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G12 compound treatment 221640.0 26800.0 1.83 206400.0 13700.0 1.02 2.0134 0.9616 3068326 PK04_096130 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G13 compound treatment 215600.0 20800.0 1.42 208080.0 15400.0 1.14 1.8106 0.9943 3186484 PK04_096131 CCCN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G14 compound treatment 221440.0 26600.0 1.82 224680.0 32000.0 2.38 2.9658 0.9912 3068146 PK04_096132 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G15 compound treatment 203360.0 8560.0 0.58 200960.0 8230.0 0.61 0.8459 0.9997 3068195 PK04_096133 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(C6CC6)C4=O)c7ccccc7C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G16 compound treatment 208120.0 13300.0 0.91 211120.0 18400.0 1.37 1.61 0.9802 3068279 PK04_096134 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G17 compound treatment 210080.0 15300.0 1.04 203000.0 10300.0 0.76 1.2772 0.9884 3068328 PK04_096135 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G18 compound treatment 202160.0 7360.0 0.5 196680.0 3950.0 0.29 0.5628 0.9675 3068311 PK04_096136 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G19 mock treatment 200840.0 6040.0 0.41 198320.0 5590.0 0.42 0.5854 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G20 mock treatment 200800.0 6000.0 0.41 194200.0 1470.0 0.11 0.3667 0.8658 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G21 compound treatment 201000.0 6200.0 0.42 198320.0 5590.0 0.42 0.5931 1.0 3068284 PK04_096137 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G22 compound treatment 202920.0 8120.0 0.55 209400.0 16700.0 1.24 1.2688 0.9339 3186501 PK04_096138 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G23 compound treatment 206400.0 11600.0 0.79 200240.0 7510.0 0.56 0.9545 0.9856 3186555 PK04_096139 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 G24 compound treatment 189760.0 -5040.0 -0.34 192360.0 -370.0 -0.03 -0.2624 -0.7613 3186877 PK04_096140 CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H01 compound treatment 197880.0 3080.0 0.21 190240.0 -2490.0 -0.19 0.0175 0.0625 3186629 PK04_096141 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H02 compound treatment 217680.0 22900.0 1.56 210480.0 17800.0 1.32 2.0372 0.9966 3068866 PK04_096142 OCc1ccc(cc1)c2cc[n+](Cc3cc4OCOc4cc3Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H03 mock treatment 198000.0 3200.0 0.22 193800.0 1070.0 0.08 0.2106 0.9066 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H04 mock treatment 193200.0 -1600.0 -0.11 194960.0 2230.0 0.17 0.0403 0.2029 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H05 compound treatment 202520.0 7720.0 0.53 196400.0 3670.0 0.27 0.5654 0.9533 3186432 PK04_096143 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(Cc5ccccc5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H06 compound treatment 225960.0 31200.0 2.12 216080.0 23400.0 1.74 2.7311 0.995 3068867 PK04_096144 OCc1ccc(cc1)c2cc[n+](Cc3cccc(OC(F)(F)F)c3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H07 compound treatment 244800.0 50000.0 3.41 235760.0 43000.0 3.2 4.675 0.9995 3187128 PK04_096145 CC(C)CN1C(=O)[C@]2(CC(=O)N(CC3C4CC5CC(C4)CC3C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H08 compound treatment 232520.0 37700.0 2.57 233600.0 40900.0 3.04 3.9694 0.9965 3068868 PK04_096146 COc1cc2CC[N+](=Cc2cc1O)Cc3sc4ccccc4c3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H09 compound treatment 251000.0 56200.0 3.83 232760.0 40000.0 2.98 4.8161 0.9923 3186637 PK04_096147 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H10 compound treatment 241400.0 46600.0 3.18 234400.0 41700.0 3.1 4.4396 0.9999 3187129 PK04_096148 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(C4CC4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H11 compound treatment 206200.0 11400.0 0.78 205320.0 12600.0 0.94 1.2122 0.9957 3187130 PK04_096149 CC1(C)OB(OC1(C)C)/C=C\CC(OC(=O)c2ccncc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H12 compound treatment 229560.0 34800.0 2.37 213720.0 21000.0 1.56 2.7804 0.9795 3187131 PK04_096150 C[n+]1ccc(cc1)c2ccc(CO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H13 compound treatment 221360.0 26600.0 1.81 217440.0 24700.0 1.84 2.5809 1.0 3068898 PK04_096151 COC(=O)c1ccc(OC)c(/C=C\CC(OC(=O)C)c2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H14 compound treatment 298800.0 104000.0 7.09 281880.0 89200.0 6.64 9.7055 0.9995 3187132 PK04_096152 CN1C(=O)C2C(C3C(N(Cc4cc5OCOc5cc4Br)C2C=C3CCCO)c6cccs6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H15 compound treatment 209160.0 14400.0 0.98 207000.0 14300.0 1.06 1.4433 0.9992 3187133 PK04_096153 COC(=O)c1ccc(OC)c(/C=C\CC(CCc2ccccc2)OC(=O)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H16 compound treatment 283160.0 88400.0 6.02 275160.0 82400.0 6.14 8.5979 1.0 3187134 PK04_096154 OCc1ccc(cc1)C2=CC(N(Cc3cccc(OC(F)(F)F)c3)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C2)c6cccs6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H17 compound treatment 251000.0 56200.0 3.83 230640.0 37900.0 2.82 4.7045 0.9887 3068899 PK04_096155 COC(=O)c1ccc(OC)c(/C=C\CC(CCc2ccccc2)OC(=O)c3ccncc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H18 compound treatment 274920.0 80100.0 5.46 255320.0 62600.0 4.66 7.1565 0.9969 3068900 PK04_096156 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(C5CC5)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H19 mock treatment 200000.0 5200.0 0.35 195080.0 2350.0 0.17 0.3744 0.947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H20 mock treatment 190720.0 -4080.0 -0.28 196080.0 3350.0 0.25 -0.0203 -0.0544 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H21 compound treatment 246120.0 51300.0 3.5 226800.0 34100.0 2.54 4.2671 0.9875 3187204 PK04_096157 CC(C)(C)OC(=O)COc1cccc(c1)C(=O)CCN2CCOCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H22 compound treatment 213400.0 18600.0 1.27 217920.0 25200.0 1.87 2.2224 0.9819 3187205 PK04_096158 OCCCc1cc[n+](Cc2cc3OCOc3cc2Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H23 compound treatment 193760.0 -1040.0 -0.07 190400.0 -2330.0 -0.17 -0.1727 -0.922 3068901 PK04_096159 COc1ccc(/C=C/C(=O)c2cccc(OCC(=O)OC(C)(C)C)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 H24 compound treatment 226880.0 32100.0 2.19 224600.0 31900.0 2.37 3.2238 0.9992 3187206 PK04_096160 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I01 compound treatment 193640.0 -1160.0 -0.08 187280.0 -5450.0 -0.41 -0.3427 -0.8292 3186796 PK04_096161 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I02 compound treatment 200080.0 5280.0 0.36 195640.0 2910.0 0.22 0.4077 0.9704 3186628 PK04_096162 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I03 compound treatment 202960.0 8160.0 0.56 191280.0 -1450.0 -0.11 0.3171 0.5595 3186882 PK04_096163 CN(C)CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I04 compound treatment 204640.0 9840.0 0.67 203840.0 11100.0 0.83 1.0591 0.9946 3186797 PK04_096164 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I05 mock treatment 212680.0 17900.0 1.22 206240.0 13500.0 1.01 1.573 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I06 mock treatment 198400.0 3600.0 0.25 199360.0 6630.0 0.49 0.5225 0.9481 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I07 compound treatment 210080.0 15300.0 1.04 208360.0 15600.0 1.16 1.5593 0.9985 3186430 PK04_096165 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(C5CC5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I08 compound treatment 226960.0 32200.0 2.19 220960.0 28200.0 2.1 3.0361 0.9998 3186557 PK04_096166 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I09 compound treatment 235680.0 40900.0 2.79 226760.0 34000.0 2.53 3.7617 0.9989 3186558 PK04_096167 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I10 compound treatment 217080.0 22300.0 1.52 211640.0 18900.0 1.41 2.0693 0.9993 3068320 PK04_096168 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I11 compound treatment 208400.0 13600.0 0.93 204920.0 12200.0 0.91 1.2972 0.9999 3068364 PK04_096169 COCCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I12 compound treatment 244800.0 50000.0 3.41 239720.0 47000.0 3.5 4.8835 0.9999 3186489 PK04_096170 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I13 compound treatment 229120.0 34300.0 2.34 214200.0 21500.0 1.6 2.7845 0.9827 3186807 PK04_096171 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I14 compound treatment 203720.0 8920.0 0.61 200480.0 7750.0 0.58 0.8379 0.9996 3068281 PK04_096172 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I15 compound treatment 205920.0 11100.0 0.76 203600.0 10900.0 0.81 1.1082 0.9995 3186567 PK04_096173 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I16 compound treatment 198120.0 3320.0 0.23 197080.0 4350.0 0.32 0.389 0.9847 3068410 PK04_096174 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I17 compound treatment 202880.0 8080.0 0.55 197440.0 4710.0 0.35 0.6375 0.9762 3186973 PK04_096175 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I18 compound treatment 234920.0 40100.0 2.74 233080.0 40400.0 3.0 4.0577 0.9989 3068148 PK04_096176 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I19 compound treatment 218240.0 23400.0 1.6 206480.0 13800.0 1.02 1.8537 0.9768 3068239 PK04_096177 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I20 compound treatment 219480.0 24700.0 1.68 209320.0 16600.0 1.23 2.0629 0.9884 3068268 PK04_096178 CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I21 mock treatment 198720.0 3920.0 0.27 194400.0 1670.0 0.12 0.2769 0.9393 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I22 mock treatment 194320.0 -479.0 -0.03 189000.0 -3730.0 -0.28 -0.2194 -0.7848 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I23 compound treatment 188880.0 -5920.0 -0.4 186600.0 -6130.0 -0.46 -0.6079 -0.9981 3186564 PK04_096179 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 I24 compound treatment 187960.0 -6840.0 -0.47 184040.0 -8690.0 -0.65 -0.787 -0.9871 3068366 PK04_096180 CC(C)CNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J01 compound treatment 200960.0 6160.0 0.42 200600.0 7870.0 0.59 0.7112 0.9867 1230870 PK04_096181 Oc1cccc(c1)C(=O)CCN2CCOCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J02 compound treatment 216480.0 21700.0 1.48 210520.0 17800.0 1.32 1.9815 0.9985 3187207 PK04_096182 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OC)C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J03 compound treatment 241080.0 46300.0 3.16 230040.0 37300.0 2.78 4.1947 0.998 3068902 PK04_096183 COc1ccc(CC[C@H](O)c2cccc(OCC(=O)OC(C)(C)C)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J04 compound treatment 237800.0 43000.0 2.93 234200.0 41500.0 3.09 4.2555 0.9997 3187208 PK04_096184 CN1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5cccs5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J05 mock treatment 195560.0 761.0 0.05 199560.0 6830.0 0.51 0.3961 0.7753 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J06 mock treatment 198240.0 3440.0 0.23 202040.0 9310.0 0.69 0.6559 0.8965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J07 compound treatment 231800.0 37000.0 2.52 224680.0 32000.0 2.38 3.4652 0.9996 3187209 PK04_096185 CCCN1C(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@H](N2C1=O)c5cccc(O)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J08 compound treatment 296440.0 102000.0 6.93 286640.0 93900.0 6.99 9.8422 1.0 3068903 PK04_096186 OCc1ccc(cc1)C2=CC(C3CC3)N(Cc4cc5OCOc5cc4Br)/C(=N\P(=O)(Oc6ccccc6)Oc7ccccc7)/C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J09 compound treatment 204600.0 9800.0 0.67 201160.0 8430.0 0.63 0.9162 0.9995 1032549 PK04_096187 CCOC(=O)C1CCCCN1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J10 compound treatment 244200.0 49400.0 3.37 240600.0 47900.0 3.56 4.9008 0.9996 3187210 PK04_096188 COc1cc2CCN(C)C(C=C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J11 compound treatment 201200.0 6400.0 0.44 199800.0 7070.0 0.53 0.6807 0.9957 3187211 PK04_096189 CCOC(=O)[C@@H]1CCCCN1C(=O)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J12 compound treatment 263280.0 68500.0 4.67 258160.0 65400.0 4.87 6.7448 0.9998 3187212 PK04_096190 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(c4ccc(CN5CCCC5)cc4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J13 compound treatment 204480.0 9680.0 0.66 201480.0 8750.0 0.65 0.9272 1.0 3068904 PK04_096191 [O-][N+](=O)c1cc(Br)ccc1C(=O)NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J14 compound treatment 262920.0 68100.0 4.64 248480.0 55800.0 4.15 6.218 0.9984 3068905 PK04_096192 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(C=C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J15 compound treatment 211640.0 16800.0 1.15 205680.0 13000.0 0.96 1.4934 0.9962 3187213 PK04_096193 CC(=O)Nc1cc(Br)ccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J16 compound treatment 262080.0 67300.0 4.59 247600.0 54900.0 4.08 6.1312 0.9983 3187214 PK04_096194 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(c5cccs5)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J17 compound treatment 205320.0 10500.0 0.72 201040.0 8310.0 0.62 0.9445 0.9973 3068906 PK04_096195 CC(=O)Nc1cc(Br)ccc1C(=O)NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J18 compound treatment 270320.0 75500.0 5.15 259880.0 67200.0 5.0 7.1747 0.9999 3187215 PK04_096196 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(c5cccs5)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J19 compound treatment 194840.0 41.3 0.0 193360.0 630.0 0.05 0.0351 0.7482 3068907 PK04_096197 Brc1ccc2c(=O)oc(nc2c1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J20 compound treatment 221920.0 27100.0 1.85 223560.0 30800.0 2.29 2.93 0.9943 3187216 PK04_096198 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(c4ccc(CN5CCCC5)cc4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J21 mock treatment 189680.0 -5120.0 -0.35 190440.0 -2290.0 -0.17 -0.3673 -0.9457 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J22 mock treatment 188640.0 -6160.0 -0.42 188040.0 -4690.0 -0.35 -0.5437 -0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J23 compound treatment 188240.0 -6560.0 -0.45 188640.0 -4090.0 -0.3 -0.5314 -0.9824 3068908 PK04_096199 Nc1cc(Br)ccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 J24 compound treatment 260880.0 66100.0 4.51 264240.0 71500.0 5.32 6.9491 0.9966 3068910 PK04_096200 Oc1ccc2cc[n+](Cc3ccc(o3)[N+](=O)[O-])cc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K01 compound treatment 196200.0 1400.0 0.1 193160.0 430.0 0.03 0.0902 0.8951 3068198 PK04_096201 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(Cc6ccccc6)C4=O)c7ccccc7C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K02 compound treatment 234120.0 39300.0 2.68 229960.0 37200.0 2.77 3.8549 0.9999 3186870 PK04_096202 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K03 compound treatment 224000.0 29200.0 1.99 220280.0 27600.0 2.05 2.8576 0.9999 3068155 PK04_096203 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K04 compound treatment 196800.0 2000.0 0.14 192400.0 -330.0 -0.02 0.0791 0.5706 3186875 PK04_096204 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCC(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K05 compound treatment 210360.0 15600.0 1.06 201880.0 9150.0 0.68 1.2317 0.977 3068359 PK04_096205 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NC4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K06 compound treatment 209240.0 14400.0 0.98 210880.0 18200.0 1.35 1.6514 0.9879 3186626 PK04_096206 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CC(F)(F)F)C4=O)c6ccccc6C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K07 mock treatment 203720.0 8920.0 0.61 201880.0 9150.0 0.68 0.9116 0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K08 mock treatment 200520.0 5720.0 0.39 197080.0 4350.0 0.32 0.5047 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K09 compound treatment 265080.0 70300.0 4.79 255920.0 63200.0 4.7 6.7137 1.0 3186869 PK04_096207 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K10 compound treatment 213480.0 18700.0 1.27 205240.0 12500.0 0.93 1.559 0.9881 3068235 PK04_096208 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K11 compound treatment 209760.0 15000.0 1.02 202000.0 9270.0 0.69 1.2091 0.9819 3186487 PK04_096209 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(Cc7ccccc7)c2c1)c8ccc(cc8)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K12 compound treatment 215520.0 20700.0 1.41 213440.0 20700.0 1.54 2.0889 0.9991 3068411 PK04_096210 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K13 compound treatment 222280.0 27500.0 1.87 216960.0 24200.0 1.8 2.6 0.9998 3068329 PK04_096211 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K14 compound treatment 211640.0 16800.0 1.15 207560.0 14800.0 1.1 1.5924 0.9998 3067608 PK04_096212 COCCCN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K15 mock treatment 201080.0 6280.0 0.43 198960.0 6230.0 0.46 0.6307 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K16 mock treatment 203040.0 8240.0 0.56 195760.0 3030.0 0.23 0.5568 0.9196 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K17 compound treatment 219480.0 24700.0 1.68 211240.0 18500.0 1.38 2.164 0.9951 3186979 PK04_096213 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K18 compound treatment 204680.0 9880.0 0.67 207840.0 15100.0 1.12 1.2716 0.97 3186636 PK04_096214 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K19 compound treatment 203240.0 8440.0 0.58 202520.0 9790.0 0.73 0.9222 0.9932 3186793 PK04_096215 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K20 compound treatment 199840.0 5040.0 0.34 200160.0 7430.0 0.55 0.6341 0.9738 3186637 PK04_096216 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K21 compound treatment 214280.0 19500.0 1.33 208560.0 15800.0 1.18 1.7723 0.9982 3067613 PK04_096217 COc1ccc(CCN2C(=O)[C@]3(CC(=O)N(CC4(CC5CC6CC(C5)C4)C6)[C@@H]3c7ccc(CO)cc27)c8ccc(cc8)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K22 compound treatment 195880.0 1080.0 0.07 196640.0 3910.0 0.29 0.2579 0.8591 3186873 PK04_096218 CCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K23 mock treatment 189840.0 -4960.0 -0.34 185840.0 -6890.0 -0.51 -0.6017 -0.9796 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 K24 mock treatment 186560.0 -8240.0 -0.56 180640.0 -12100.0 -0.9 -1.0334 -0.9743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L01 compound treatment 200880.0 6080.0 0.41 194240.0 1510.0 0.11 0.3726 0.8675 3068940 PK04_096219 Cc1nc2cc(Br)ccc2c(=O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L02 compound treatment 238800.0 44000.0 3.0 236640.0 43900.0 3.27 4.4321 0.9991 3187217 PK04_096220 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(c5ccc(CN6CCCC6)cc5)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L03 compound treatment 202000.0 7200.0 0.49 192280.0 -450.0 -0.03 0.3235 0.6573 3068941 PK04_096221 CC(C)c1nc2cc(Br)ccc2c(=O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L04 compound treatment 228520.0 33700.0 2.3 228000.0 35300.0 2.63 3.4818 0.9978 3068942 PK04_096222 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L05 compound treatment 202760.0 7960.0 0.54 198720.0 5990.0 0.45 0.699 0.9952 3187218 PK04_096223 Cc1nc2cc(Br)ccc2c(=O)n1Cc3cccc(O)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L06 compound treatment 255280.0 60500.0 4.12 241560.0 48800.0 3.63 5.4855 0.998 3068943 PK04_096224 COc1cc2CCN(C)C(c3cccs3)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L07 mock treatment 196640.0 1840.0 0.13 193040.0 310.0 0.02 0.1051 0.8233 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L08 mock treatment 201880.0 7080.0 0.48 196400.0 3670.0 0.27 0.5345 0.9636 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L09 compound treatment 265800.0 71000.0 4.84 261960.0 69200.0 5.15 7.0663 0.9995 3187219 PK04_096225 Oc1cccc(CNC(=O)c2ccc(Br)cc2NC(=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L10 compound treatment 307040.0 112000.0 7.65 293160.0 100000.0 7.47 10.6964 0.9999 3187220 PK04_096226 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(C=C1C(=O)OC)c4ccc(CO)cc4)C5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L11 compound treatment 207600.0 12800.0 0.87 207160.0 14400.0 1.07 1.3765 0.9947 3068944 PK04_096227 Oc1cccc(Cn2c(nc3cc(Br)ccc3c2=O)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L12 compound treatment 237280.0 42500.0 2.9 230040.0 37300.0 2.78 4.0115 0.9998 3187221 PK04_096228 CN1C(=O)C2C(C3C(N(Cc4cc5OCOc5cc4Br)C2C=C3CCCO)c6ccc(CN7CCCC7)cc6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L13 compound treatment 209520.0 14700.0 1.0 203160.0 10400.0 0.78 1.2586 0.9919 1980253 PK04_096229 Cc1c(NC(=O)/C(=C/C=C/c2ccccc2)/C#N)c(=O)n(c3ccccc3)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L14 compound treatment 258520.0 63700.0 4.34 256280.0 63600.0 4.73 6.4164 0.9991 3068945 PK04_096230 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OC)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L15 mock treatment 197880.0 3080.0 0.21 196200.0 3470.0 0.26 0.3312 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L16 mock treatment 198560.0 3760.0 0.26 196880.0 4150.0 0.31 0.3997 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L17 compound treatment 224000.0 29200.0 1.99 212200.0 19500.0 1.45 2.4324 0.9878 3187222 PK04_096231 Cc1c(NC(=O)/C(=C/C=C/c2ccccc2[N+](=O)[O-])/C#N)c(=O)n(c3ccccc3)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L18 compound treatment 263920.0 69100.0 4.71 264000.0 71300.0 5.3 7.083 0.9983 3187223 PK04_096232 OCCCC1=CC(N(Cc2cc3OCOc3cc2Br)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C1)c6cccs6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L19 compound treatment 208640.0 13800.0 0.94 201760.0 9030.0 0.67 1.1425 0.9862 3068946 PK04_096233 Cc1c(NC(=O)/C(=C/C=C/c2ccc(cc2)[N+](=O)[O-])/C#N)c(=O)n(c3ccccc3)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L20 compound treatment 226520.0 31700.0 2.16 224040.0 31300.0 2.33 3.177 0.9993 3187224 PK04_096234 OCCCC1=CC(N(Cc2cccc(OC(F)(F)F)c2)/C(=N\P(=O)(Oc3ccccc3)Oc4ccccc4)/C1)c5cccs5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L21 compound treatment 195800.0 1000.0 0.07 192800.0 70.0 0.01 0.052 0.7589 3068947 PK04_096235 CN(C)c1ccc(/C=C/C=C(\C#N)/C(=O)Nc2c(C)n(C)n(c3ccccc3)c2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L22 compound treatment 223000.0 28200.0 1.92 218360.0 25600.0 1.91 2.7084 1.0 3187225 PK04_096236 COc1cc2CCN(C)C(C3CC3)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L23 mock treatment 183520.0 -11300.0 -0.77 182360.0 -10400.0 -0.77 -1.0895 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 L24 mock treatment 181960.0 -12800.0 -0.88 176000.0 -16700.0 -1.25 -1.4994 -0.9851 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M01 compound treatment 198720.0 3920.0 0.27 200960.0 8230.0 0.61 0.6222 0.9309 3186502 PK04_096237 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M02 compound treatment 245920.0 51100.0 3.49 243120.0 50400.0 3.75 5.1164 0.9993 3186497 PK04_096238 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NC(C)C)c5ccccc5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M03 compound treatment 199160.0 4360.0 0.3 198280.0 5550.0 0.41 0.5023 0.987 3068404 PK04_096239 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M04 compound treatment 256200.0 61400.0 4.19 240400.0 47700.0 3.55 5.4688 0.9966 3186643 PK04_096240 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M05 compound treatment 217280.0 22500.0 1.53 206960.0 14200.0 1.06 1.8327 0.9837 3186723 PK04_096241 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M06 compound treatment 228720.0 33900.0 2.31 232760.0 40000.0 2.98 3.742 0.9922 3186868 PK04_096242 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M07 compound treatment 210000.0 15200.0 1.04 213800.0 21100.0 1.57 1.8417 0.9798 3186798 PK04_096243 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M08 compound treatment 205160.0 10400.0 0.71 200520.0 7790.0 0.58 0.9095 0.9952 3186799 PK04_096244 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M09 mock treatment 202920.0 8120.0 0.55 208040.0 15300.0 1.14 1.1972 0.945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M10 mock treatment 200160.0 5360.0 0.37 202160.0 9430.0 0.7 0.7547 0.9538 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M11 compound treatment 246040.0 51200.0 3.49 238560.0 45800.0 3.41 4.8822 0.9999 3186496 PK04_096245 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4OC)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M12 compound treatment 204120.0 9320.0 0.64 201920.0 9190.0 0.68 0.933 0.9993 3068379 PK04_096246 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M13 mock treatment 209520.0 14700.0 1.0 206120.0 13400.0 1.0 1.4144 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M14 mock treatment 205160.0 10400.0 0.71 200160.0 7430.0 0.55 0.8905 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M15 compound treatment 209520.0 14700.0 1.0 204920.0 12200.0 0.91 1.3512 0.9987 3186488 PK04_096247 CC(C)N1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M16 compound treatment 220480.0 25700.0 1.75 214880.0 22200.0 1.65 2.4038 0.9995 3186886 PK04_096248 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M17 compound treatment 209480.0 14700.0 1.0 204560.0 11800.0 0.88 1.3303 0.998 3068154 PK04_096249 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M18 compound treatment 216880.0 22100.0 1.51 207880.0 15200.0 1.13 1.8618 0.9899 3068369 PK04_096250 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M19 compound treatment 207640.0 12800.0 0.88 204840.0 12100.0 0.9 1.2564 0.9999 3186727 PK04_096251 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M20 compound treatment 227560.0 32800.0 2.23 224240.0 31500.0 2.35 3.2377 0.9997 3186984 PK04_096252 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M21 compound treatment 209160.0 14400.0 0.98 202720.0 9990.0 0.74 1.2181 0.9908 3068372 PK04_096253 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M22 compound treatment 201560.0 6760.0 0.46 189360.0 -3370.0 -0.25 0.1486 0.2832 3186721 PK04_096254 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M23 compound treatment 207480.0 12700.0 0.86 187600.0 -5130.0 -0.38 0.3414 0.3612 3068316 PK04_096255 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 M24 compound treatment 198880.0 4080.0 0.28 189520.0 -3210.0 -0.24 0.0278 0.0758 3068283 PK04_096256 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N01 compound treatment 192840.0 -1960.0 -0.13 190960.0 -1770.0 -0.13 -0.1876 -1.0 1694663 PK04_096257 Cc1c(NC(=O)CC#N)c(=O)n(c2ccccc2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N02 compound treatment 222120.0 27300.0 1.86 205160.0 12400.0 0.93 1.9713 0.9478 3187226 PK04_096258 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C)C=C(CCCO)C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N03 compound treatment 213160.0 18400.0 1.25 203760.0 11000.0 0.82 1.4656 0.9791 3068949 PK04_096259 Cc1ccccc1/C=C/C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N04 compound treatment 212560.0 17800.0 1.21 215960.0 23200.0 1.73 2.0788 0.9848 3187227 PK04_096260 COC(=O)C1=CN(C)C(C=C(CCCO)C=C1C(=O)OC)c2ccc(CN3CCCC3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N05 compound treatment 219520.0 24700.0 1.69 213720.0 21000.0 1.56 2.2964 0.9993 3068950 PK04_096261 CCOc1ccc(cc1)N2C(SCC2=O)c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N06 compound treatment 252240.0 57400.0 3.92 238760.0 46000.0 3.43 5.1916 0.9978 3187228 PK04_096262 Oc1ccc2cc[n+](Cc3cccc(OC(F)(F)F)c3)cc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N07 compound treatment 206200.0 11400.0 0.78 203440.0 10700.0 0.8 1.1133 0.9999 3068951 PK04_096263 [O-][N+](=O)c1cccc(c1)C2SCC(=O)N2c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N08 compound treatment 226720.0 31900.0 2.18 219840.0 27100.0 2.02 2.9656 0.9993 3187299 PK04_096264 CN1C(=O)C2C(C3C(N(C)C2C=C3CCCO)c4cccs4)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N09 mock treatment 202560.0 7760.0 0.53 202480.0 9750.0 0.73 0.8873 0.988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N10 mock treatment 201840.0 7040.0 0.48 201960.0 9230.0 0.69 0.8252 0.9846 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N11 compound treatment 215560.0 20800.0 1.42 210000.0 17300.0 1.29 1.9097 0.9988 3068985 PK04_096265 Cc1cc(C)cc(c1)N2C(SCC2=O)c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N12 compound treatment 238000.0 43200.0 2.95 231920.0 39200.0 2.92 4.1451 1.0 3187300 PK04_096266 COc1cc2CCN(C)C(c3ccc(CN4CCCC4)cc3)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N13 mock treatment 204560.0 9760.0 0.67 200320.0 7590.0 0.56 0.87 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N14 mock treatment 206800.0 12000.0 0.82 200600.0 7870.0 0.59 0.9927 0.9866 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N15 compound treatment 205160.0 10400.0 0.71 201200.0 8470.0 0.63 0.9453 0.9984 3068986 PK04_096267 COc1ccc(/C=C/C=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N16 compound treatment 251600.0 56800.0 3.87 235000.0 42300.0 3.15 4.9629 0.9947 3187301 PK04_096268 OCCCC1=CC(C2CC2)N(Cc3sc4ccccc4c3Cl)/C(=N\P(=O)(Oc5ccccc5)Oc6ccccc6)/C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N17 compound treatment 211560.0 16800.0 1.14 203280.0 10600.0 0.79 1.3633 0.9832 3068987 PK04_096269 Cc1cccc(/C=C/C=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N18 compound treatment 217160.0 22400.0 1.52 206000.0 13300.0 0.99 1.7764 0.9779 3068988 PK04_096270 OCCCc1cc[n+](Cc2sc3ccccc3c2Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N19 compound treatment 204960.0 10200.0 0.69 201320.0 8590.0 0.64 0.9419 0.9992 3068989 PK04_096271 Cc1ccc(/C=C/C=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N20 compound treatment 297880.0 103000.0 7.03 288120.0 95400.0 7.1 9.9895 1.0 3187302 PK04_096272 CN1C(=O)C2C(C3C(C4CC4)N(Cc5sc6ccccc6c5Cl)C2C=C3c7ccc(CO)cc7)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N21 compound treatment 200080.0 5280.0 0.36 197080.0 4350.0 0.32 0.4835 0.9986 3068990 PK04_096273 COc1cccc(/C=C/C=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N22 compound treatment 231480.0 36700.0 2.5 223720.0 31000.0 2.31 3.3993 0.9992 3068991 PK04_096274 Oc1ccc2cc[n+](Cc3cc4OCOc4cc3Br)cc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N23 compound treatment 190000.0 -4800.0 -0.33 186680.0 -6050.0 -0.45 -0.5497 -0.9877 3187303 PK04_096275 Clc1ccccc1/C=C/C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 N24 compound treatment 207880.0 13100.0 0.89 203360.0 10600.0 0.79 1.1901 0.9982 3187304 PK04_096276 CN/1C(C=C(C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CO)cc4)C5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O01 compound treatment 196240.0 1440.0 0.1 192760.0 30.0 0.0 0.0711 0.723 3186631 PK04_096277 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O02 compound treatment 205600.0 10800.0 0.74 196880.0 4150.0 0.31 0.7391 0.9256 3067615 PK04_096278 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(CC(F)(F)F)c2c1)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O03 compound treatment 192960.0 -1840.0 -0.13 187640.0 -5090.0 -0.38 -0.3565 -0.8934 3186715 PK04_096279 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O04 compound treatment 205520.0 10700.0 0.73 196520.0 3790.0 0.28 0.7163 0.9143 3068363 PK04_096280 CC(C)NC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O05 compound treatment 206720.0 11900.0 0.81 195320.0 2590.0 0.19 0.711 0.8512 3068310 PK04_096281 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O06 compound treatment 206400.0 11600.0 0.79 204440.0 11700.0 0.87 1.1755 0.9988 3068196 PK04_096282 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CCN6CCOCC6)C4=O)c7ccccc7C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O07 compound treatment 216680.0 21900.0 1.49 205160.0 12400.0 0.93 1.709 0.9736 3068277 PK04_096283 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O08 compound treatment 204760.0 9960.0 0.68 199280.0 6550.0 0.49 0.8249 0.9868 3186720 PK04_096284 CC(C)NC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O09 compound treatment 198640.0 3840.0 0.26 196760.0 4030.0 0.3 0.3973 0.9977 3186632 PK04_096285 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O10 compound treatment 207680.0 12900.0 0.88 201600.0 8870.0 0.66 1.0878 0.9901 3068157 PK04_096286 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(C5CCCCC5)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O11 mock treatment 203320.0 8520.0 0.58 196400.0 3670.0 0.27 0.6039 0.9408 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O12 mock treatment 203200.0 8400.0 0.57 195520.0 2790.0 0.21 0.5518 0.9058 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O13 compound treatment 197800.0 3000.0 0.2 200880.0 8150.0 0.61 0.5736 0.896 3186874 PK04_096287 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O14 compound treatment 216120.0 21300.0 1.45 201560.0 8830.0 0.66 1.4926 0.9356 3068138 PK04_096288 COCCCN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O15 compound treatment 202440.0 7640.0 0.52 193760.0 1030.0 0.08 0.4226 0.8025 3186972 PK04_096289 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O16 compound treatment 201640.0 6840.0 0.47 194160.0 1430.0 0.11 0.4051 0.8467 3186981 PK04_096290 COCCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O17 compound treatment 265800.0 71000.0 4.84 247360.0 54600.0 4.07 6.2979 0.9962 3186709 PK04_096291 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O18 compound treatment 196520.0 1720.0 0.12 198520.0 5790.0 0.43 0.3877 0.8681 3186725 PK04_096292 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O19 compound treatment 200560.0 5760.0 0.39 207520.0 14800.0 1.1 1.0561 0.9036 3068321 PK04_096293 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O20 compound treatment 198160.0 3360.0 0.23 193520.0 790.0 0.06 0.2036 0.8607 3068192 PK04_096294 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O21 compound treatment 195800.0 1000.0 0.07 197080.0 4350.0 0.32 0.2772 0.8378 3068201 PK04_096295 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O22 compound treatment 190680.0 -4120.0 -0.28 183880.0 -8850.0 -0.66 -0.6643 -0.9278 3068381 PK04_096296 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O23 compound treatment 204800.0 10000.0 0.68 198840.0 6110.0 0.45 0.8037 0.9806 3186880 PK04_096297 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NCc6ccccc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 O24 compound treatment 180080.0 -14700.0 -1.0 179680.0 -13100.0 -0.97 -1.3964 -0.9999 3186977 PK04_096298 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P01 compound treatment 200640.0 5840.0 0.4 194720.0 1990.0 0.15 0.3863 0.9092 3068992 PK04_096299 Cc1c(NC(=O)/C(=C/c2cccc(c2)[N+](=O)[O-])/C#N)c(=O)n(c3ccccc3)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P02 compound treatment 197440.0 2640.0 0.18 194040.0 1310.0 0.1 0.1963 0.9585 3187305 PK04_096300 COC(=O)C1=CN(C)C(C=C(CCCO)C=C1C(=O)OC)C2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P03 compound treatment 203360.0 8560.0 0.58 196680.0 3950.0 0.29 0.6206 0.9496 3187306 PK04_096301 COc1cccc(/C=C(\C#N)/C(=O)Nc2c(C)n(C)n(c3ccccc3)c2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P04 compound treatment 238880.0 44100.0 3.01 229200.0 36500.0 2.71 4.0444 0.9987 3068993 PK04_096302 COc1cc2CC[N+](=Cc2cc1O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P05 compound treatment 203040.0 8240.0 0.56 195240.0 2510.0 0.19 0.5294 0.8941 3068994 PK04_096303 Cc1c(NC(=O)/C(=C/c2ccccc2Cl)/C#N)c(=O)n(c3ccccc3)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P06 compound treatment 252000.0 57200.0 3.9 241520.0 48800.0 3.63 5.3253 0.9994 3187307 PK04_096304 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(c4cccs4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P07 compound treatment 207880.0 13100.0 0.89 199360.0 6630.0 0.49 0.9795 0.961 3187308 PK04_096305 Cc1c(NC(=O)/C(=C/c2ccc(Cl)cc2)/C#N)c(=O)n(c3ccccc3)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P08 compound treatment 201880.0 7080.0 0.48 192400.0 -330.0 -0.02 0.324 0.6703 3068995 PK04_096306 CN1C(=O)C2C(C3C(C4CC4)N(C)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P09 compound treatment 221000.0 26200.0 1.79 202280.0 9550.0 0.71 1.7657 0.9184 1972122 PK04_096307 Cc1cc(C)cc(c1)N2C(c3cccc(c3)[N+](=O)[O-])S(=O)(=O)CC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P10 compound treatment 206040.0 11200.0 0.77 200720.0 7990.0 0.59 0.9624 0.9921 3187309 PK04_096308 CN/1C(C=C(CCCO)C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P11 mock treatment 198720.0 3920.0 0.27 193520.0 790.0 0.06 0.2306 0.8425 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P12 mock treatment 193480.0 -1320.0 -0.09 192800.0 70.0 0.01 -0.0599 -0.665 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P13 compound treatment 192640.0 -2160.0 -0.15 195680.0 2950.0 0.22 0.0512 0.1936 3068996 PK04_096309 Clc1ccc(/C=C/C=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P14 compound treatment 234960.0 40200.0 2.74 227960.0 35200.0 2.62 3.7902 0.9998 3187310 PK04_096310 COc1cc2CC[N+](=Cc2cc1O)Cc3cccc(OC(F)(F)F)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P15 compound treatment 215800.0 21000.0 1.43 206600.0 13900.0 1.03 1.7424 0.9871 3068997 PK04_096311 O=C/C=C/c1ccc2OCOc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P16 compound treatment 206800.0 12000.0 0.82 205320.0 12600.0 0.94 1.2411 0.9977 3187311 PK04_096312 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OC)c3ccc(CN4CCCC4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P17 compound treatment 205520.0 10700.0 0.73 198280.0 5550.0 0.41 0.8089 0.9635 3068998 PK04_096313 O=C/C=C/c1ccc(cc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P18 compound treatment 271840.0 77000.0 5.25 280840.0 88100.0 6.56 8.3511 0.9939 3187312 PK04_096314 CN1C(=O)C2C(C3C(C4CC4)N(Cc5cc6OCOc6cc5Br)C2C=C3c7ccc(CO)cc7)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P19 compound treatment 200760.0 5960.0 0.41 194120.0 1390.0 0.1 0.3605 0.8597 3187313 PK04_096315 O=C/C=C/c1ccc(\C=C\c2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P20 compound treatment 244160.0 49400.0 3.37 249040.0 56300.0 4.19 5.3431 0.9941 3187314 PK04_096316 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(c4cccs4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P21 compound treatment 195840.0 1040.0 0.07 203160.0 10400.0 0.78 0.5991 0.7686 3069028 PK04_096317 [O-][N+](=O)c1cccc(c1)C2N(C(=O)CS2(=O)=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P22 compound treatment 236280.0 41500.0 2.83 224800.0 32100.0 2.39 3.6875 0.9964 3187315 PK04_096318 COC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(CCCO)C=C1C(=O)OC)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P23 compound treatment 190400.0 -4400.0 -0.3 192400.0 -330.0 -0.02 -0.2294 -0.7625 3069029 PK04_096319 CCOc1ccc(cc1)N2C(c3cccc(c3)[N+](=O)[O-])S(=O)(=O)/C(=C\C=C\c4ccccc4OC)/C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2096 P24 compound treatment 189840.0 -4960.0 -0.34 189080.0 -3650.0 -0.27 -0.4311 -0.9941 3187316 PK04_096320 COC(=O)C1=CN(C)C(C=C(C=C1C(=O)OC)c2ccc(CO)cc2)C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A01 compound treatment 271160.0 76000.0 5.18 223800.0 34800.0 2.59 5.4914 0.9485 2141518 PK04_097001 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A02 compound treatment 266760.0 71600.0 4.88 249240.0 60200.0 4.48 6.6181 0.9991 2141905 PK04_097002 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A03 compound treatment 395200.0 200000.0 13.64 405440.0 216000.0 16.11 21.0305 0.9966 2141091 PK04_097003 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A04 compound treatment 263240.0 68000.0 4.64 295880.0 107000.0 7.95 8.903 0.9671 2141692 PK04_097004 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A05 compound treatment 245360.0 50200.0 3.42 274360.0 85300.0 6.35 6.9085 0.9579 2141533 PK04_097005 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A06 compound treatment 263440.0 68200.0 4.65 270400.0 81400.0 6.06 7.5717 0.9915 2141714 PK04_097006 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A07 compound treatment 251880.0 56700.0 3.86 269280.0 80200.0 5.97 6.9555 0.9778 2141463 PK04_097007 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A08 compound treatment 247960.0 52800.0 3.6 231480.0 42400.0 3.16 4.7772 0.9979 2141076 PK04_097008 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A09 compound treatment 296280.0 101000.0 6.89 290120.0 101000.0 7.52 10.1927 0.999 2141109 PK04_097009 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A10 compound treatment 274880.0 79700.0 5.43 264600.0 75600.0 5.62 7.818 0.9999 2141546 PK04_097010 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A11 compound treatment 236600.0 41400.0 2.82 228040.0 39000.0 2.9 4.0485 0.9999 2141079 PK04_097011 OC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A12 compound treatment 408040.0 213000.0 14.51 373960.0 185000.0 13.76 19.9928 0.9996 2141141 PK04_097012 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A13 mock treatment 174040.0 -21200.0 -1.44 180280.0 -8760.0 -0.65 -1.4809 -0.9357 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A14 mock treatment 175240.0 -20000.0 -1.36 177360.0 -11700.0 -0.87 -1.5768 -0.9766 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A15 compound treatment 210760.0 15600.0 1.06 253920.0 64900.0 4.83 4.1648 0.8424 2141882 PK04_097013 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A16 compound treatment 206160.0 11000.0 0.75 201960.0 12900.0 0.96 1.2085 0.9923 2141936 PK04_097014 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A17 compound treatment 244640.0 49400.0 3.37 230520.0 41500.0 3.09 4.5666 0.999 2141372 PK04_097015 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A18 compound treatment 236200.0 41000.0 2.8 231960.0 42900.0 3.19 4.2355 0.9978 2141092 PK04_097016 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A19 compound treatment 277240.0 82000.0 5.59 256760.0 67700.0 5.04 7.5191 0.9986 2141344 PK04_097017 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A20 compound treatment 327560.0 132000.0 9.02 322720.0 134000.0 9.95 13.4163 0.9988 2141115 PK04_097018 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A21 compound treatment 232880.0 37700.0 2.57 212720.0 23700.0 1.76 3.0629 0.9831 2141570 PK04_097019 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A22 compound treatment 290720.0 95500.0 6.51 272320.0 83300.0 6.2 8.9879 0.9997 2141549 PK04_097020 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A23 compound treatment 229800.0 34600.0 2.36 223520.0 34500.0 2.57 3.4828 0.9991 2141876 PK04_097021 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 A24 compound treatment 234240.0 39000.0 2.66 236160.0 47100.0 3.51 4.362 0.9908 2141753 PK04_097022 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B01 compound treatment 227880.0 32700.0 2.23 235280.0 46200.0 3.44 4.0091 0.9779 2141940 PK04_097023 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccccc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B02 compound treatment 278760.0 83600.0 5.7 266280.0 77200.0 5.75 8.0934 1.0 2142685 PK04_097024 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B03 compound treatment 271280.0 76100.0 5.19 259520.0 70500.0 5.25 7.3771 1.0 2141335 PK04_097025 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B04 compound treatment 280520.0 85300.0 5.82 253200.0 64200.0 4.77 7.4899 0.9952 2143933 PK04_097026 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B05 compound treatment 227800.0 32600.0 2.22 216480.0 27400.0 2.04 3.0159 0.9991 2141445 PK04_097027 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B06 compound treatment 237760.0 42600.0 2.9 254720.0 65700.0 4.89 5.5085 0.969 2144925 PK04_097028 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B07 compound treatment 248280.0 53100.0 3.62 255400.0 66400.0 4.94 6.0514 0.9883 2141881 PK04_097029 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccccc3OCCO)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B08 compound treatment 210880.0 15700.0 1.07 224720.0 35700.0 2.66 2.6338 0.9201 2144289 PK04_097030 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B09 compound treatment 255040.0 59800.0 4.08 280760.0 91700.0 6.83 7.712 0.9697 2141150 PK04_097031 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B10 compound treatment 229000.0 33800.0 2.3 250160.0 61100.0 4.55 4.8462 0.9504 2144633 PK04_097032 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B11 compound treatment 287320.0 92100.0 6.28 300880.0 112000.0 8.32 10.327 0.9904 2141161 PK04_097033 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B12 compound treatment 219240.0 24000.0 1.64 233680.0 44600.0 3.32 3.5084 0.947 2144765 PK04_097034 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B13 mock treatment 181040.0 -14200.0 -0.96 174120.0 -14900.0 -1.11 -1.4677 -0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B14 mock treatment 176040.0 -19200.0 -1.31 173520.0 -15500.0 -1.16 -1.7403 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B15 compound treatment 237720.0 42500.0 2.9 235040.0 46000.0 3.42 4.4709 0.9966 2141135 PK04_097035 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B16 compound treatment 221360.0 26200.0 1.78 201040.0 12000.0 0.89 1.8928 0.9488 2144753 PK04_097036 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B17 compound treatment 270280.0 75100.0 5.12 270320.0 81300.0 6.05 7.8972 0.9966 2141225 PK04_097037 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B18 compound treatment 288600.0 93400.0 6.37 266600.0 77600.0 5.77 8.5846 0.9988 2144045 PK04_097038 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B19 compound treatment 277040.0 81800.0 5.58 251880.0 62800.0 4.68 7.2527 0.9961 2141420 PK04_097039 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B20 compound treatment 239880.0 44700.0 3.05 219640.0 30600.0 2.28 3.7645 0.9897 2144377 PK04_097040 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B21 compound treatment 274120.0 78900.0 5.38 223720.0 34700.0 2.58 5.6299 0.9434 2141808 PK04_097041 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B22 compound treatment 253960.0 58800.0 4.01 250240.0 61200.0 4.55 6.0537 0.998 2143265 PK04_097042 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B23 compound treatment 211360.0 16200.0 1.1 231320.0 42300.0 3.15 3.0043 0.9011 2141931 PK04_097043 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 B24 compound treatment 207040.0 11800.0 0.81 215040.0 26000.0 1.93 1.9393 0.9249 2142705 PK04_097044 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C01 compound treatment 259440.0 64200.0 4.38 263320.0 74300.0 5.53 7.0063 0.9934 2141223 PK04_097045 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C02 compound treatment 180160.0 -15000.0 -1.02 268040.0 79000.0 5.88 3.4327 0.5752 2141108 PK04_097046 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C03 compound treatment 292480.0 97300.0 6.63 230240.0 41200.0 3.07 6.8581 0.9386 2141329 PK04_097047 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C04 compound treatment 261760.0 66600.0 4.54 262320.0 73300.0 5.45 7.0655 0.9958 2141703 PK04_097048 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C05 compound treatment 277480.0 82300.0 5.61 273640.0 84600.0 6.3 8.4191 0.9983 2065845 PK04_097049 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C06 compound treatment 235200.0 40000.0 2.73 224560.0 35500.0 2.64 3.7978 0.9999 2141782 PK04_097050 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C07 compound treatment 302400.0 107000.0 7.31 311760.0 123000.0 9.13 11.6266 0.9939 2141574 PK04_097051 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C08 compound treatment 285800.0 90600.0 6.18 272000.0 83000.0 6.17 8.7338 1.0 2141856 PK04_097052 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C09 compound treatment 290120.0 94900.0 6.47 285840.0 96800.0 7.2 9.6705 0.9986 2141751 PK04_097053 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C10 compound treatment 202720.0 7530.0 0.51 208040.0 19000.0 1.41 1.3626 0.9059 2141441 PK04_097054 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C11 mock treatment 184000.0 -11200.0 -0.76 182640.0 -6400.0 -0.48 -0.8766 -0.9743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C12 mock treatment 184240.0 -11000.0 -0.75 183360.0 -5680.0 -0.42 -0.8271 -0.9638 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C13 compound treatment 215440.0 20200.0 1.38 232200.0 43200.0 3.21 3.2473 0.9288 2141937 PK04_097055 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C14 compound treatment 287960.0 92800.0 6.32 299360.0 110000.0 8.21 10.2779 0.9917 2141727 PK04_097056 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C15 mock treatment 190840.0 -4350.0 -0.3 188200.0 -843.0 -0.06 -0.2542 -0.8381 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C16 mock treatment 183840.0 -11400.0 -0.77 179840.0 -9200.0 -0.68 -1.0317 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C17 compound treatment 217520.0 22300.0 1.52 227400.0 38400.0 2.85 3.095 0.9566 2141078 PK04_097057 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C18 compound treatment 220960.0 25800.0 1.76 207280.0 18200.0 1.36 2.2019 0.9919 2141467 PK04_097058 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C19 compound treatment 261960.0 66800.0 4.55 277560.0 88500.0 6.59 7.8772 0.9837 2141339 PK04_097059 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C20 compound treatment 254560.0 59400.0 4.05 268360.0 79300.0 5.9 7.0362 0.983 2141364 PK04_097060 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C21 compound treatment 255160.0 60000.0 4.09 257920.0 68900.0 5.13 6.5157 0.9937 2141370 PK04_097061 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C22 compound treatment 273720.0 78500.0 5.35 255000.0 66000.0 4.91 7.2568 0.9991 2141489 PK04_097062 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C23 compound treatment 177840.0 -17400.0 -1.18 168080.0 -21000.0 -1.56 -1.9398 -0.9907 2141706 PK04_097063 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 C24 compound treatment 257040.0 61800.0 4.22 232320.0 43300.0 3.22 5.2591 0.9912 2141172 PK04_097064 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D01 compound treatment 206640.0 11400.0 0.78 199040.0 10000.0 0.74 1.0779 0.9997 2141788 PK04_097065 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D02 compound treatment 211680.0 16500.0 1.12 221480.0 32400.0 2.41 2.5019 0.9395 2143973 PK04_097066 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D03 compound treatment 277200.0 82000.0 5.59 265640.0 76600.0 5.7 7.9845 1.0 2141854 PK04_097067 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D04 compound treatment 315280.0 120000.0 8.19 274000.0 85000.0 6.32 10.2603 0.9918 2141969 PK04_097068 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D05 compound treatment 271160.0 76000.0 5.18 249960.0 60900.0 4.53 6.8682 0.9978 2141087 PK04_097069 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D06 compound treatment 298200.0 103000.0 7.02 261960.0 72900.0 5.43 8.8032 0.9919 2144657 PK04_097070 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D07 compound treatment 268920.0 73700.0 5.03 257360.0 68300.0 5.08 7.1496 1.0 2141768 PK04_097071 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D08 compound treatment 268400.0 73200.0 4.99 266200.0 77200.0 5.74 7.5898 0.9976 2144733 PK04_097072 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D09 compound treatment 343000.0 148000.0 10.08 304440.0 115000.0 8.59 13.1986 0.9968 2141552 PK04_097073 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D10 compound treatment 271000.0 75800.0 5.17 264040.0 75000.0 5.58 7.6014 0.9993 2143885 PK04_097074 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D11 mock treatment 179960.0 -15200.0 -1.04 181440.0 -7600.0 -0.57 -1.1345 -0.9592 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D12 mock treatment 190120.0 -5070.0 -0.35 178840.0 -10200.0 -0.76 -0.7815 -0.9366 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D13 compound treatment 274480.0 79300.0 5.41 242440.0 53400.0 3.97 6.6324 0.9886 2141513 PK04_097075 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D14 compound treatment 271720.0 76500.0 5.22 261560.0 72500.0 5.4 7.5056 0.9999 2144449 PK04_097076 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D15 mock treatment 186360.0 -8830.0 -0.6 186440.0 -2600.0 -0.19 -0.5628 -0.8897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D16 mock treatment 185520.0 -9670.0 -0.66 179400.0 -9640.0 -0.72 -0.9738 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D17 compound treatment 231160.0 36000.0 2.45 235600.0 46600.0 3.47 4.1841 0.9857 2141816 PK04_097077 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D18 compound treatment 270600.0 75400.0 5.14 263360.0 74300.0 5.53 7.5464 0.9993 2142085 PK04_097078 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D19 compound treatment 255840.0 60600.0 4.13 251280.0 62200.0 4.63 6.1991 0.9984 2141432 PK04_097079 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D20 compound treatment 259600.0 64400.0 4.39 243280.0 54200.0 4.04 5.9593 0.9991 2144825 PK04_097080 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D21 compound treatment 419000.0 224000.0 15.26 406560.0 218000.0 16.19 22.2368 0.9996 2141123 PK04_097081 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D22 compound treatment 227040.0 31800.0 2.17 239720.0 50700.0 3.77 4.2023 0.9656 2144893 PK04_097082 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D23 compound treatment 238160.0 43000.0 2.93 225160.0 36100.0 2.69 3.9721 0.9991 2141421 PK04_097083 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 D24 compound treatment 175800.0 -19400.0 -1.32 205160.0 16100.0 1.2 -0.0867 -0.0486 2143085 PK04_097084 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E01 mock treatment 187400.0 -7790.0 -0.53 186280.0 -2760.0 -0.21 -0.5211 -0.9147 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E02 mock treatment 185640.0 -9550.0 -0.65 178320.0 -10700.0 -0.8 -1.0249 -0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E03 compound treatment 290840.0 95600.0 6.52 279040.0 90000.0 6.7 9.3473 0.9999 2141878 PK04_097085 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E04 compound treatment 314480.0 119000.0 8.13 268280.0 79200.0 5.9 9.9207 0.9875 2141520 PK04_097086 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E05 compound treatment 286800.0 91600.0 6.25 258960.0 69900.0 5.2 8.0958 0.9959 2141359 PK04_097087 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E06 compound treatment 321960.0 127000.0 8.64 300960.0 112000.0 8.33 12.0012 0.9998 2141507 PK04_097088 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E07 compound treatment 297960.0 103000.0 7.01 274240.0 85200.0 6.34 9.4379 0.9988 2141863 PK04_097089 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccccc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E08 compound treatment 288360.0 93200.0 6.35 290240.0 101000.0 7.53 9.8172 0.9964 2141163 PK04_097090 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E09 mock treatment 197320.0 2130.0 0.15 188560.0 -483.0 -0.04 0.0771 0.5161 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E10 mock treatment 191400.0 -3790.0 -0.26 192960.0 3920.0 0.29 0.0233 0.0597 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E11 compound treatment 246080.0 50900.0 3.47 228440.0 39400.0 2.93 4.5265 0.9965 2141456 PK04_097091 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E12 compound treatment 296280.0 101000.0 6.89 287600.0 98600.0 7.34 10.0601 0.9995 2141683 PK04_097092 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E13 compound treatment 285560.0 90400.0 6.16 267920.0 78900.0 5.87 8.5075 0.9997 2141357 PK04_097093 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E14 compound treatment 273400.0 78200.0 5.33 248560.0 59500.0 4.43 6.9025 0.9958 2141366 PK04_097094 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E15 compound treatment 331160.0 136000.0 9.27 277040.0 88000.0 6.55 11.1858 0.9855 2141575 PK04_097095 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E16 compound treatment 293440.0 98200.0 6.7 276680.0 87600.0 6.52 9.3484 0.9999 2141485 PK04_097096 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E17 mock treatment 195840.0 647.0 0.04 190600.0 1560.0 0.12 0.1131 0.9124 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E18 mock treatment 193680.0 -1510.0 -0.1 186040.0 -3000.0 -0.22 -0.231 -0.9383 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E19 compound treatment 268600.0 73400.0 5.0 256280.0 67200.0 5.0 7.0773 1.0 2141377 PK04_097097 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E20 compound treatment 265720.0 70500.0 4.81 236640.0 47600.0 3.54 5.9049 0.9887 2141326 PK04_097098 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E21 compound treatment 296000.0 101000.0 6.87 287760.0 98700.0 7.35 10.055 0.9994 2141702 PK04_097099 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E22 compound treatment 256520.0 61300.0 4.18 241760.0 52700.0 3.92 5.7308 0.9995 2141417 PK04_097100 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E23 compound treatment 189800.0 -5390.0 -0.37 249560.0 60500.0 4.5 2.9249 0.6472 2141167 PK04_097101 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 E24 compound treatment 471400.0 276000.0 18.83 428720.0 240000.0 17.84 25.9291 0.9996 2141113 PK04_097102 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F01 mock treatment 186080.0 -9110.0 -0.62 176680.0 -12400.0 -0.92 -1.09 -0.9817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F02 mock treatment 190960.0 -4230.0 -0.29 181000.0 -8040.0 -0.6 -0.6274 -0.944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F03 compound treatment 328720.0 134000.0 9.1 317360.0 128000.0 9.55 13.1901 0.9997 2141216 PK04_097103 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F04 compound treatment 276040.0 80800.0 5.51 260440.0 71400.0 5.31 7.6549 0.9998 2142933 PK04_097104 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F05 compound treatment 270280.0 75100.0 5.12 259000.0 70000.0 5.21 7.3015 1.0 2141355 PK04_097105 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F06 compound treatment 305080.0 110000.0 7.49 277840.0 88800.0 6.61 9.9706 0.998 2142833 PK04_097106 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F07 compound treatment 255120.0 59900.0 4.09 228720.0 39700.0 2.95 4.9771 0.9873 2141414 PK04_097107 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F08 compound treatment 278720.0 83500.0 5.69 255760.0 66700.0 4.97 7.5378 0.9977 2144249 PK04_097108 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F09 mock treatment 196440.0 1250.0 0.09 187840.0 -1200.0 -0.09 -0.0032 -0.026 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F10 mock treatment 202040.0 6850.0 0.47 193200.0 4160.0 0.31 0.5488 0.98 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F11 compound treatment 312120.0 117000.0 7.97 296880.0 108000.0 8.03 11.3121 1.0 2141568 PK04_097109 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F12 compound treatment 318240.0 123000.0 8.39 295600.0 107000.0 7.93 11.5397 0.9996 2142765 PK04_097110 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F13 compound treatment 278600.0 83400.0 5.69 271480.0 82400.0 6.14 8.3594 0.9993 2141348 PK04_097111 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F14 compound treatment 330600.0 135000.0 9.23 313120.0 124000.0 9.23 13.0576 1.0 2142645 PK04_097112 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F15 compound treatment 322440.0 127000.0 8.68 301760.0 113000.0 8.39 12.0664 0.9999 2141505 PK04_097113 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F16 compound treatment 244280.0 49100.0 3.35 230320.0 41300.0 3.07 4.5387 0.9991 2142977 PK04_097114 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F17 mock treatment 192480.0 -2710.0 -0.18 186080.0 -2960.0 -0.22 -0.2867 -0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F18 mock treatment 195720.0 527.0 0.04 186880.0 -2160.0 -0.16 -0.0884 -0.5361 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F19 compound treatment 342240.0 147000.0 10.03 308880.0 120000.0 8.92 13.3956 0.9983 2141200 PK04_097115 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F20 compound treatment 302800.0 108000.0 7.34 283360.0 94300.0 7.02 10.1512 0.9998 2142045 PK04_097116 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F21 compound treatment 235760.0 40600.0 2.77 231920.0 42900.0 3.19 4.2122 0.9975 2141938 PK04_097117 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F22 compound treatment 250320.0 55100.0 3.76 228120.0 39100.0 2.91 4.7141 0.992 2144373 PK04_097118 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F23 compound treatment 241840.0 46600.0 3.18 228360.0 39300.0 2.93 4.3179 0.9991 2141419 PK04_097119 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 F24 compound treatment 244480.0 49300.0 3.36 251200.0 62200.0 4.63 5.6472 0.9877 2142769 PK04_097120 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G01 compound treatment 307920.0 113000.0 7.69 311640.0 123000.0 9.12 11.8864 0.9964 2141178 PK04_097121 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G02 compound treatment 296440.0 101000.0 6.9 286760.0 97700.0 7.27 10.0236 0.9997 2141487 PK04_097122 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G03 mock treatment 194040.0 -1150.0 -0.08 187440.0 -1600.0 -0.12 -0.14 -0.9795 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G04 mock treatment 199720.0 4530.0 0.31 190640.0 1600.0 0.12 0.3023 0.914 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G05 compound treatment 321560.0 126000.0 8.62 294000.0 105000.0 7.81 11.6156 0.9988 2141519 PK04_097123 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G06 compound treatment 281640.0 86400.0 5.89 270280.0 81200.0 6.05 8.4428 0.9999 2141537 PK04_097124 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G07 compound treatment 279480.0 84300.0 5.75 267880.0 78800.0 5.87 8.2123 0.9999 2141722 PK04_097125 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G08 compound treatment 347920.0 153000.0 10.41 320480.0 131000.0 9.78 14.2799 0.9995 2141577 PK04_097126 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G09 compound treatment 255440.0 60200.0 4.11 232160.0 43100.0 3.21 5.1735 0.9925 2141458 PK04_097127 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G10 compound treatment 288280.0 93100.0 6.35 272600.0 83600.0 6.22 8.885 0.9999 2141190 PK04_097128 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G11 compound treatment 285240.0 90000.0 6.14 267600.0 78600.0 5.85 8.4753 0.9997 2141333 PK04_097129 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G12 compound treatment 355280.0 160000.0 10.91 326000.0 137000.0 10.19 14.9253 0.9994 2141508 PK04_097130 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G13 compound treatment 264240.0 69000.0 4.71 245360.0 56300.0 4.19 6.2925 0.9983 2141118 PK04_097131 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G14 compound treatment 285240.0 90000.0 6.14 281160.0 92100.0 6.86 9.1889 0.9985 2141927 PK04_097132 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G15 compound treatment 267280.0 72100.0 4.91 257400.0 68400.0 5.09 7.0727 0.9999 2141159 PK04_097133 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G16 compound treatment 295760.0 101000.0 6.86 287480.0 98400.0 7.33 10.0287 0.9995 2141713 PK04_097134 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G17 compound treatment 254240.0 59000.0 4.03 235240.0 46200.0 3.44 5.2778 0.9969 2141795 PK04_097135 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G18 compound treatment 258600.0 63400.0 4.32 271560.0 82500.0 6.14 7.3994 0.9852 2141553 PK04_097136 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G19 mock treatment 199080.0 3890.0 0.27 191680.0 2640.0 0.2 0.3261 0.9891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G20 mock treatment 196880.0 1690.0 0.12 190200.0 1160.0 0.09 0.1422 0.9898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G21 compound treatment 227520.0 32300.0 2.2 235920.0 46900.0 3.49 4.0254 0.9755 2141819 PK04_097137 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G22 compound treatment 268480.0 73300.0 5.0 282200.0 93200.0 6.93 8.4357 0.9871 2141516 PK04_097138 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G23 compound treatment 299920.0 105000.0 7.14 289600.0 101000.0 7.48 10.3408 0.9997 2141691 PK04_097139 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 G24 compound treatment 250080.0 54900.0 3.74 269680.0 80600.0 6.0 6.8897 0.9741 2141155 PK04_097140 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H01 compound treatment 273440.0 78200.0 5.33 268280.0 79200.0 5.9 7.9422 0.9987 2141157 PK04_097141 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H02 compound treatment 242640.0 47400.0 3.23 234680.0 45600.0 3.4 4.6891 0.9997 2143037 PK04_097142 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H03 mock treatment 198480.0 3290.0 0.22 187040.0 -2000.0 -0.15 0.053 0.197 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H04 mock treatment 201800.0 6610.0 0.45 187360.0 -1680.0 -0.13 0.2299 0.4918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H05 compound treatment 311520.0 116000.0 7.93 294840.0 106000.0 7.87 11.1758 1.0 2141926 PK04_097143 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H06 compound treatment 286960.0 91800.0 6.26 281640.0 92600.0 6.89 9.2971 0.9988 2143177 PK04_097144 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H07 compound treatment 337680.0 142000.0 9.71 300960.0 112000.0 8.33 12.759 0.9971 2141694 PK04_097145 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H08 compound treatment 304480.0 109000.0 7.45 285080.0 96000.0 7.15 10.3227 0.9998 2143025 PK04_097146 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H09 compound treatment 343800.0 149000.0 10.13 321800.0 133000.0 9.88 14.1508 0.9999 2141749 PK04_097147 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H10 compound treatment 281200.0 86000.0 5.86 268960.0 79900.0 5.95 8.3521 1.0 2143077 PK04_097148 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H11 compound treatment 480440.0 285000.0 19.45 437480.0 248000.0 18.49 26.826 0.9997 2141097 PK04_097149 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H12 compound treatment 271520.0 76300.0 5.2 264240.0 75200.0 5.6 7.637 0.9993 2142913 PK04_097150 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H13 compound treatment 336840.0 142000.0 9.66 321000.0 132000.0 9.82 13.7732 1.0 2141401 PK04_097151 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H14 compound treatment 275520.0 80300.0 5.48 261480.0 72400.0 5.39 7.6846 1.0 2143093 PK04_097152 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H15 compound treatment 264800.0 69600.0 4.75 246920.0 57900.0 4.31 6.4016 0.9988 2141777 PK04_097153 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H16 compound treatment 271480.0 76300.0 5.2 266960.0 77900.0 5.8 7.7783 0.9985 2143865 PK04_097154 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H17 compound treatment 294240.0 99000.0 6.75 268480.0 79400.0 5.91 8.9555 0.9978 2141142 PK04_097155 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H18 compound treatment 324160.0 129000.0 8.79 299320.0 110000.0 8.21 12.0209 0.9994 2143925 PK04_097156 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H19 mock treatment 193400.0 -1790.0 -0.12 187120.0 -1920.0 -0.14 -0.1877 -0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H20 mock treatment 194440.0 -753.0 -0.05 194800.0 5760.0 0.43 0.2667 0.618 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H21 compound treatment 313600.0 118000.0 8.07 291800.0 103000.0 7.65 11.1161 0.9996 2141168 PK04_097157 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H22 compound treatment 220880.0 25700.0 1.75 220640.0 31600.0 2.35 2.9012 0.9895 2143057 PK04_097158 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H23 compound treatment 224640.0 29400.0 2.01 222120.0 33100.0 2.46 3.1603 0.9949 2141804 PK04_097159 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 H24 compound treatment 233040.0 37800.0 2.58 223720.0 34700.0 2.58 3.6495 1.0 2142649 PK04_097160 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I01 compound treatment 247520.0 52300.0 3.57 238280.0 49200.0 3.66 5.1138 0.9999 2141890 PK04_097161 O[C@@H](CNC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I02 compound treatment 232680.0 37500.0 2.56 224360.0 35300.0 2.63 3.6658 0.9999 2141465 PK04_097162 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I03 compound treatment 300400.0 105000.0 7.17 274960.0 85900.0 6.39 9.5935 0.9984 2141772 PK04_097163 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I04 compound treatment 340240.0 145000.0 9.89 308440.0 119000.0 8.89 13.2761 0.9986 2141343 PK04_097164 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I05 mock treatment 201240.0 6050.0 0.41 196920.0 7880.0 0.59 0.706 0.9852 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I06 mock treatment 200120.0 4930.0 0.34 192480.0 3440.0 0.26 0.4184 0.991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I07 compound treatment 264960.0 69800.0 4.76 258000.0 69000.0 5.13 6.9924 0.9993 2141794 PK04_097165 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I08 compound treatment 301640.0 106000.0 7.26 288080.0 99000.0 7.37 10.3437 1.0 2141922 PK04_097166 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I09 compound treatment 349680.0 154000.0 10.53 336240.0 147000.0 10.96 15.1942 0.9998 2141780 PK04_097167 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I10 compound treatment 255960.0 60800.0 4.14 242880.0 53800.0 4.01 5.7628 0.9999 2141799 PK04_097168 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I11 compound treatment 307520.0 112000.0 7.66 281040.0 92000.0 6.85 10.2567 0.9984 2141177 PK04_097169 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I12 compound treatment 333600.0 138000.0 9.44 316120.0 127000.0 9.46 13.3601 1.0 2141747 PK04_097170 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I13 compound treatment 272760.0 77600.0 5.29 269240.0 80200.0 5.97 7.9599 0.9982 2141423 PK04_097171 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I14 compound treatment 274440.0 79200.0 5.4 264280.0 75200.0 5.6 7.7799 0.9998 2141775 PK04_097172 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I15 compound treatment 312480.0 117000.0 8.0 298400.0 109000.0 8.14 11.4094 1.0 2141538 PK04_097173 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I16 compound treatment 476200.0 281000.0 19.16 433160.0 244000.0 18.17 26.3942 0.9996 2065871 PK04_097174 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I17 compound treatment 282240.0 87000.0 5.93 278200.0 89200.0 6.64 8.8885 0.9984 2141729 PK04_097175 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I18 compound treatment 230160.0 35000.0 2.38 232480.0 43400.0 3.23 3.9717 0.9888 2141892 PK04_097176 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I19 compound treatment 237440.0 42200.0 2.88 225000.0 36000.0 2.68 3.929 0.9993 2141687 PK04_097177 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I20 compound treatment 288560.0 93400.0 6.37 267040.0 78000.0 5.81 8.6059 0.9989 2141680 PK04_097178 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I21 mock treatment 197480.0 2290.0 0.16 184600.0 -4440.0 -0.33 -0.1236 -0.338 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I22 mock treatment 191000.0 -4190.0 -0.29 178920.0 -10100.0 -0.75 -0.7349 -0.912 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I23 compound treatment 302160.0 107000.0 7.29 270040.0 81000.0 6.03 9.4194 0.9955 2141841 PK04_097179 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 I24 compound treatment 220720.0 25500.0 1.74 250240.0 61200.0 4.55 4.4513 0.9129 2141766 PK04_097180 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J01 compound treatment 275840.0 80600.0 5.5 274840.0 85800.0 6.39 8.4031 0.9972 2141705 PK04_097181 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J02 compound treatment 304560.0 109000.0 7.46 284640.0 95600.0 7.11 10.3034 0.9997 2143397 PK04_097182 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J03 compound treatment 291360.0 96200.0 6.56 261760.0 72700.0 5.41 8.463 0.9955 2141179 PK04_097183 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J04 compound treatment 249360.0 54200.0 3.69 238360.0 49300.0 3.67 5.2067 1.0 2144337 PK04_097184 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J05 mock treatment 195960.0 767.0 0.05 192000.0 2960.0 0.22 0.1926 0.8514 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J06 mock treatment 201400.0 6210.0 0.42 198480.0 9440.0 0.7 0.7959 0.9706 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J07 compound treatment 269880.0 74700.0 5.09 269800.0 80800.0 6.01 7.8506 0.9966 2141805 PK04_097185 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J08 compound treatment 293520.0 98300.0 6.7 287600.0 98600.0 7.34 9.927 0.999 2143365 PK04_097186 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J09 compound treatment 328520.0 133000.0 9.09 314040.0 125000.0 9.3 13.0058 0.9999 2141901 PK04_097187 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J10 compound treatment 279800.0 84600.0 5.77 269360.0 80300.0 5.98 8.3057 0.9998 2144881 PK04_097188 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J11 compound treatment 353520.0 158000.0 10.79 307680.0 119000.0 8.83 13.8763 0.995 2141717 PK04_097189 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J12 compound treatment 322720.0 128000.0 8.69 300320.0 111000.0 8.28 12.0041 0.9997 2143405 PK04_097190 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J13 compound treatment 313760.0 119000.0 8.08 301920.0 113000.0 8.4 11.6564 0.9998 2141188 PK04_097191 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J14 compound treatment 301280.0 106000.0 7.23 280120.0 91100.0 6.78 9.9074 0.9995 2142929 PK04_097192 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J15 compound treatment 353440.0 158000.0 10.79 328200.0 139000.0 10.36 14.9523 0.9998 2141365 PK04_097193 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J16 compound treatment 370160.0 175000.0 11.93 332920.0 144000.0 10.71 16.0068 0.9985 2144325 PK04_097194 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J17 compound treatment 356720.0 162000.0 11.01 342560.0 154000.0 11.43 15.8662 0.9998 2141221 PK04_097195 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J18 compound treatment 279840.0 84600.0 5.77 264480.0 75400.0 5.61 8.0508 0.9999 2143377 PK04_097196 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J19 compound treatment 242040.0 46800.0 3.19 238640.0 49600.0 3.69 4.8686 0.9974 2141815 PK04_097197 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J20 compound treatment 266400.0 71200.0 4.85 237920.0 48900.0 3.64 6.005 0.9899 2142585 PK04_097198 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J21 mock treatment 190440.0 -4750.0 -0.32 185800.0 -3240.0 -0.24 -0.3998 -0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J22 mock treatment 186920.0 -8270.0 -0.56 188560.0 -483.0 -0.04 -0.4243 -0.7507 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J23 compound treatment 287960.0 92800.0 6.32 268000.0 79000.0 5.88 8.6275 0.9993 2141186 PK04_097199 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 J24 compound treatment 206360.0 11200.0 0.76 240360.0 51300.0 3.82 3.239 0.8317 2144237 PK04_097200 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K01 compound treatment 327320.0 132000.0 9.01 315400.0 126000.0 9.4 13.0195 0.9998 2141164 PK04_097201 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K02 compound treatment 438800.0 244000.0 16.61 421920.0 233000.0 17.33 23.9997 0.9998 2141443 PK04_097202 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K03 compound treatment 325160.0 130000.0 8.86 303880.0 115000.0 8.55 12.3091 0.9998 2141548 PK04_097203 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K04 compound treatment 300160.0 105000.0 7.16 295520.0 106000.0 7.92 10.6639 0.9987 2141351 PK04_097204 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K05 compound treatment 285680.0 90500.0 6.17 269520.0 80500.0 5.99 8.5975 0.9999 2141786 PK04_097205 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K06 compound treatment 312320.0 117000.0 7.99 297760.0 109000.0 8.09 11.368 1.0 2141746 PK04_097206 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K07 mock treatment 211360.0 16200.0 1.1 206400.0 17400.0 1.29 1.6928 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K08 mock treatment 215400.0 20200.0 1.38 208680.0 19600.0 1.46 2.0076 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K09 compound treatment 298920.0 104000.0 7.07 281120.0 92100.0 6.85 9.8463 0.9999 2141350 PK04_097207 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K10 compound treatment 302920.0 108000.0 7.34 305200.0 116000.0 8.65 11.3064 0.9967 2141331 PK04_097208 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K11 compound treatment 268920.0 73700.0 5.03 259120.0 70100.0 5.22 7.2422 0.9998 2141806 PK04_097209 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K12 compound treatment 281200.0 86000.0 5.86 269640.0 80600.0 6.0 8.3879 0.9999 2141720 PK04_097210 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K13 compound treatment 341000.0 146000.0 9.94 318480.0 129000.0 9.63 13.8411 0.9999 2141904 PK04_097211 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K14 compound treatment 387720.0 193000.0 13.13 367880.0 179000.0 13.31 18.6932 1.0 2141222 PK04_097212 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K15 mock treatment 211760.0 16600.0 1.13 210440.0 21400.0 1.59 1.9247 0.9858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K16 mock treatment 199480.0 4290.0 0.29 194680.0 5640.0 0.42 0.5033 0.9844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K17 compound treatment 267600.0 72400.0 4.94 272720.0 83700.0 6.23 7.8943 0.9934 2141773 PK04_097213 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K18 compound treatment 271120.0 75900.0 5.18 238920.0 49900.0 3.71 6.2852 0.9867 2141524 PK04_097214 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K19 compound treatment 300560.0 105000.0 7.18 275000.0 86000.0 6.4 9.6033 0.9983 2141218 PK04_097215 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K20 compound treatment 240560.0 45400.0 3.09 229280.0 40200.0 2.99 4.3046 0.9999 2141861 PK04_097216 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K21 compound treatment 220480.0 25300.0 1.72 211760.0 22700.0 1.69 2.4146 1.0 2141117 PK04_097217 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K22 compound treatment 256320.0 61100.0 4.17 236280.0 47200.0 3.52 5.4328 0.9964 2141354 PK04_097218 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K23 mock treatment 194320.0 -873.0 -0.06 183760.0 -5280.0 -0.39 -0.3201 -0.805 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 K24 mock treatment 181440.0 -13800.0 -0.94 182800.0 -6240.0 -0.46 -0.9916 -0.9476 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L01 compound treatment 364560.0 169000.0 11.55 325440.0 136000.0 10.15 15.3432 0.9979 2141684 PK04_097219 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L02 compound treatment 355560.0 160000.0 10.93 351960.0 163000.0 12.13 16.305 0.9987 2143489 PK04_097220 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L03 compound treatment 333200.0 138000.0 9.41 318800.0 130000.0 9.66 13.4819 0.9999 2141375 PK04_097221 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccccc3OCCO)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L04 compound treatment 314960.0 120000.0 8.17 293640.0 105000.0 7.78 11.2785 0.9997 2143313 PK04_097222 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L05 compound treatment 310080.0 115000.0 7.83 288800.0 99800.0 7.42 10.7885 0.9996 2141889 PK04_097223 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L06 compound treatment 272560.0 77400.0 5.27 274120.0 85100.0 6.33 8.2071 0.9959 2144793 PK04_097224 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L07 mock treatment 216040.0 20800.0 1.42 215160.0 26100.0 1.94 2.3795 0.9882 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L08 mock treatment 203720.0 8530.0 0.58 199160.0 10100.0 0.75 0.9435 0.9918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L09 compound treatment 297360.0 102000.0 6.97 286360.0 97300.0 7.24 10.0469 0.9998 2141438 PK04_097225 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L10 compound treatment 259560.0 64400.0 4.39 253840.0 64800.0 4.82 6.5131 0.9989 2142993 PK04_097226 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L11 compound treatment 319800.0 125000.0 8.5 299800.0 111000.0 8.24 11.836 0.9999 2141185 PK04_097227 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L12 compound treatment 312400.0 117000.0 7.99 288520.0 99500.0 7.4 10.8856 0.9993 2144653 PK04_097228 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L13 compound treatment 261080.0 65900.0 4.49 246240.0 57200.0 4.26 6.1864 0.9996 2141893 PK04_097229 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L14 compound treatment 321640.0 126000.0 8.62 309440.0 120000.0 8.96 12.432 0.9998 2143417 PK04_097230 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L15 mock treatment 243720.0 48500.0 3.31 234440.0 45400.0 3.38 4.7285 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L16 mock treatment 197680.0 2490.0 0.17 191800.0 2760.0 0.21 0.265 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L17 compound treatment 314360.0 119000.0 8.12 290920.0 102000.0 7.58 11.1064 0.9994 2141152 PK04_097231 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L18 compound treatment 282400.0 87200.0 5.95 283480.0 94400.0 7.03 9.1741 0.9965 2143325 PK04_097232 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L19 compound treatment 273560.0 78400.0 5.34 266080.0 77000.0 5.73 7.8322 0.9994 2141709 PK04_097233 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L20 compound treatment 264720.0 69500.0 4.74 244880.0 55800.0 4.16 6.2903 0.9978 2142773 PK04_097234 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L21 compound treatment 286560.0 91400.0 6.23 285760.0 96700.0 7.2 9.4946 0.9974 2141174 PK04_097235 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L22 compound treatment 217440.0 22200.0 1.52 205040.0 16000.0 1.19 1.9144 0.9928 2142985 PK04_097236 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L23 mock treatment 187560.0 -7630.0 -0.52 177240.0 -11800.0 -0.88 -0.9892 -0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 L24 mock treatment 177000.0 -18200.0 -1.24 175800.0 -13200.0 -0.99 -1.574 -0.9935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M01 compound treatment 303560.0 108000.0 7.39 290040.0 101000.0 7.52 10.5394 1.0 2141838 PK04_097237 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M02 compound treatment 329400.0 134000.0 9.15 297280.0 108000.0 8.06 12.1662 0.998 2141189 PK04_097238 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M03 compound treatment 309480.0 114000.0 7.79 289240.0 100000.0 7.46 10.7827 0.9998 2141724 PK04_097239 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M04 compound treatment 326560.0 131000.0 8.96 319640.0 131000.0 9.72 13.206 0.9992 2141153 PK04_097240 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M05 compound treatment 225720.0 30500.0 2.08 219640.0 30600.0 2.28 3.0819 0.999 2141436 PK04_097241 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M06 compound treatment 280120.0 84900.0 5.79 275480.0 86400.0 6.43 8.6432 0.9986 2141769 PK04_097242 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M07 compound treatment 264960.0 69800.0 4.76 266680.0 77600.0 5.78 7.4492 0.9953 2141771 PK04_097243 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M08 compound treatment 298360.0 103000.0 7.03 297400.0 108000.0 8.06 10.6761 0.9977 2141480 PK04_097244 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M09 mock treatment 217760.0 22600.0 1.54 209600.0 20600.0 1.53 2.1698 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M10 mock treatment 209720.0 14500.0 0.99 207480.0 18400.0 1.37 1.6706 0.9872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M11 compound treatment 338440.0 143000.0 9.77 319760.0 131000.0 9.73 13.785 1.0 2141571 PK04_097245 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M12 compound treatment 308320.0 113000.0 7.71 292960.0 104000.0 7.73 10.9226 1.0 2141879 PK04_097246 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M13 mock treatment 214880.0 19700.0 1.34 205880.0 16800.0 1.25 1.8352 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M14 mock treatment 207280.0 12100.0 0.82 199840.0 10800.0 0.8 1.1509 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M15 compound treatment 282040.0 86800.0 5.92 271640.0 82600.0 6.15 8.5336 0.9998 2141832 PK04_097247 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M16 compound treatment 277520.0 82300.0 5.61 272520.0 83500.0 6.21 8.362 0.9987 2141542 PK04_097248 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M17 compound treatment 313120.0 118000.0 8.04 287760.0 98700.0 7.35 10.8803 0.999 2141399 PK04_097249 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M18 compound treatment 284680.0 89500.0 6.1 277480.0 88400.0 6.58 8.9682 0.9993 2141903 PK04_097250 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M19 compound treatment 320160.0 125000.0 8.52 305520.0 116000.0 8.67 12.1544 1.0 2141716 PK04_097251 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M20 compound treatment 267160.0 72000.0 4.91 276800.0 87800.0 6.53 8.0878 0.9901 2141203 PK04_097252 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M21 compound treatment 344760.0 150000.0 10.2 325840.0 137000.0 10.18 14.4097 1.0 2141110 PK04_097253 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M22 compound treatment 277240.0 82000.0 5.59 280560.0 91500.0 6.81 8.7717 0.9952 2141731 PK04_097254 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M23 compound treatment 422360.0 227000.0 15.49 395880.0 207000.0 15.39 21.8367 1.0 2141095 PK04_097255 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 M24 compound treatment 239200.0 44000.0 3.0 233920.0 44900.0 3.34 4.4833 0.9986 2141894 PK04_097256 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N01 compound treatment 307880.0 113000.0 7.68 302400.0 113000.0 8.44 11.3982 0.9989 2141340 PK04_097257 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N02 compound treatment 329160.0 134000.0 9.13 298760.0 110000.0 8.17 12.2325 0.9984 2142089 PK04_097258 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N03 compound treatment 328040.0 133000.0 9.06 310360.0 121000.0 9.03 12.789 1.0 2141511 PK04_097259 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N04 compound treatment 251960.0 56800.0 3.87 254440.0 65400.0 4.87 6.1783 0.9936 2144305 PK04_097260 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N05 compound treatment 317000.0 122000.0 8.3 273560.0 84500.0 6.29 10.32 0.9906 2141839 PK04_097261 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N06 compound treatment 293400.0 98200.0 6.7 269520.0 80500.0 5.99 8.9697 0.9985 2142057 PK04_097262 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N07 compound treatment 405800.0 211000.0 14.36 377920.0 189000.0 14.06 20.0932 0.9999 2141431 PK04_097263 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N08 compound treatment 281200.0 86000.0 5.86 262080.0 73000.0 5.44 7.99 0.9993 2144369 PK04_097264 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N09 mock treatment 204840.0 9650.0 0.66 197320.0 8280.0 0.62 0.9007 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N10 mock treatment 208280.0 13100.0 0.89 197320.0 8280.0 0.62 1.0665 0.9836 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N11 compound treatment 311600.0 116000.0 7.94 302480.0 113000.0 8.44 11.5817 0.9995 2141527 PK04_097265 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N12 compound treatment 314360.0 119000.0 8.12 285760.0 96700.0 7.2 10.8348 0.9982 2144009 PK04_097266 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N13 mock treatment 201080.0 5890.0 0.4 200080.0 11000.0 0.82 0.8646 0.9457 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N14 mock treatment 198640.0 3450.0 0.24 193960.0 4920.0 0.37 0.4249 0.9771 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N15 compound treatment 323880.0 129000.0 8.77 313280.0 124000.0 9.25 12.7421 0.9997 2141907 PK04_097267 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccccc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N16 compound treatment 302240.0 107000.0 7.3 274480.0 85400.0 6.36 9.6569 0.9976 2143157 PK04_097268 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N17 compound treatment 324640.0 129000.0 8.83 293480.0 104000.0 7.77 11.7367 0.998 2141544 PK04_097269 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N18 compound treatment 262760.0 67600.0 4.61 251760.0 62700.0 4.67 6.5579 1.0 2144297 PK04_097270 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N19 compound treatment 291480.0 96300.0 6.56 274600.0 85600.0 6.37 9.1445 0.9999 2141483 PK04_097271 O[C@@H](CNC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N20 compound treatment 264640.0 69400.0 4.73 269120.0 80100.0 5.96 7.5622 0.9935 2142217 PK04_097272 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N21 compound treatment 230240.0 35000.0 2.39 225680.0 36600.0 2.73 3.6177 0.9978 2141887 PK04_097273 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N22 compound treatment 235000.0 39800.0 2.71 218640.0 29600.0 2.2 3.4766 0.9946 2143065 PK04_097274 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N23 compound treatment 247480.0 52300.0 3.56 232960.0 43900.0 3.27 4.8319 0.9991 2141817 PK04_097275 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 N24 compound treatment 221160.0 26000.0 1.77 208720.0 19700.0 1.46 2.2874 0.9956 2144333 PK04_097276 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O01 compound treatment 291480.0 96300.0 6.56 276680.0 87600.0 6.52 9.254 1.0 2141166 PK04_097277 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O02 compound treatment 304120.0 109000.0 7.43 273400.0 84400.0 6.28 9.6907 0.9965 2141900 PK04_097278 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O03 compound treatment 276480.0 81300.0 5.54 261600.0 72600.0 5.4 7.7372 0.9999 2141790 PK04_097279 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O04 compound treatment 294560.0 99400.0 6.77 277400.0 88400.0 6.58 9.4403 0.9999 2141883 PK04_097280 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O05 compound treatment 303400.0 108000.0 7.38 286360.0 97300.0 7.24 10.338 1.0 2141427 PK04_097281 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O06 compound treatment 260720.0 65500.0 4.47 251600.0 62600.0 4.66 6.4512 0.9998 2141093 PK04_097282 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O07 compound treatment 299000.0 104000.0 7.08 283680.0 94600.0 7.04 9.9849 1.0 2141812 PK04_097283 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O08 compound treatment 249640.0 54400.0 3.71 234400.0 45400.0 3.38 5.0118 0.9989 2141430 PK04_097284 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O09 compound treatment 253960.0 58800.0 4.01 248120.0 59100.0 4.4 5.9421 0.9989 2141454 PK04_097285 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O10 compound treatment 306280.0 111000.0 7.57 275920.0 86900.0 6.47 9.9274 0.9969 2141529 PK04_097286 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O11 mock treatment 200600.0 5410.0 0.37 192040.0 3000.0 0.22 0.4184 0.971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O12 mock treatment 194200.0 -993.0 -0.07 193640.0 4600.0 0.34 0.194 0.5564 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O13 compound treatment 269520.0 74300.0 5.07 256560.0 67500.0 5.03 7.1364 1.0 2141368 PK04_097287 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O14 compound treatment 276680.0 81500.0 5.56 255800.0 66800.0 4.97 7.4416 0.9984 2141362 PK04_097288 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O15 compound treatment 282200.0 87000.0 5.93 267680.0 78600.0 5.85 8.3329 1.0 2141460 PK04_097289 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O16 compound treatment 290040.0 94800.0 6.47 282560.0 93500.0 6.96 9.494 0.9993 2141860 PK04_097290 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O17 compound treatment 316680.0 121000.0 8.28 305000.0 116000.0 8.63 11.9592 0.9998 2141175 PK04_097291 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O18 compound treatment 321920.0 127000.0 8.64 295920.0 107000.0 7.95 11.734 0.9991 2141486 PK04_097292 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O19 compound treatment 310840.0 116000.0 7.88 337680.0 149000.0 11.06 13.3976 0.9862 2141156 PK04_097293 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O20 compound treatment 264640.0 69400.0 4.73 238440.0 49400.0 3.68 5.9476 0.9922 2141685 PK04_097294 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O21 compound treatment 280560.0 85400.0 5.82 289120.0 100000.0 7.45 9.3822 0.9926 2141094 PK04_097295 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O22 compound treatment 252720.0 57500.0 3.92 253840.0 64800.0 4.82 6.1834 0.9947 2141379 PK04_097296 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O23 compound treatment 323680.0 128000.0 8.76 289240.0 100000.0 7.46 11.4673 0.9968 2141397 PK04_097297 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccccc3OCCO)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 O24 compound treatment 275600.0 80400.0 5.48 293440.0 104000.0 7.77 9.3705 0.9854 2065842 PK04_097298 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P01 compound treatment 291280.0 96100.0 6.55 263640.0 74600.0 5.55 8.5581 0.9966 2141898 PK04_097299 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P02 compound treatment 274520.0 79300.0 5.41 246560.0 57500.0 4.28 6.8512 0.9933 2143305 PK04_097300 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P03 compound treatment 316560.0 121000.0 8.27 295040.0 106000.0 7.89 11.4293 0.9997 2141555 PK04_097301 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P04 compound treatment 253080.0 57900.0 3.95 250040.0 61000.0 4.54 6.0008 0.9976 2144945 PK04_097302 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P05 compound treatment 315200.0 120000.0 8.18 302000.0 113000.0 8.41 11.73 0.9999 2141923 PK04_097303 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P06 compound treatment 299520.0 104000.0 7.11 271160.0 82100.0 6.11 9.351 0.9971 2144433 PK04_097304 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P07 compound treatment 327320.0 132000.0 9.01 311240.0 122000.0 9.09 12.8006 1.0 2141482 PK04_097305 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P08 compound treatment 306440.0 111000.0 7.58 267000.0 78000.0 5.8 9.4657 0.9913 2143929 PK04_097306 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P09 compound treatment 308800.0 114000.0 7.75 301320.0 112000.0 8.36 11.3857 0.9993 2141698 PK04_097307 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P10 compound treatment 279120.0 83900.0 5.72 261800.0 72800.0 5.42 7.875 0.9996 2142653 PK04_097308 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P11 mock treatment 198240.0 3050.0 0.21 189880.0 837.0 0.06 0.1909 0.8804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P12 mock treatment 197240.0 2050.0 0.14 190360.0 1320.0 0.1 0.168 0.985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P13 compound treatment 288040.0 92800.0 6.33 263400.0 74400.0 5.53 8.3892 0.9978 2141449 PK04_097309 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P14 compound treatment 243600.0 48400.0 3.3 211080.0 22000.0 1.64 3.4934 0.9479 2144933 PK04_097310 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P15 compound treatment 297880.0 103000.0 7.0 278920.0 89900.0 6.69 9.6804 0.9997 2141416 PK04_097311 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P16 compound treatment 299560.0 104000.0 7.12 264360.0 75300.0 5.61 8.9951 0.993 2144445 PK04_097312 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P17 compound treatment 238760.0 43600.0 2.97 235920.0 46900.0 3.49 4.5673 0.9968 2141453 PK04_097313 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P18 compound treatment 271760.0 76600.0 5.22 253960.0 64900.0 4.83 7.1076 0.9993 2142745 PK04_097314 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P19 compound treatment 294160.0 99000.0 6.75 273160.0 84100.0 6.26 9.1979 0.9993 2141541 PK04_097315 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P20 compound treatment 283040.0 87800.0 5.99 267400.0 78400.0 5.83 8.3587 0.9999 2142193 PK04_097316 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P21 compound treatment 330320.0 135000.0 9.21 318080.0 129000.0 9.6 13.3052 0.9998 2141134 PK04_097317 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P22 compound treatment 241880.0 46700.0 3.18 239600.0 50600.0 3.76 4.9114 0.9965 2142729 PK04_097318 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P23 compound treatment 330600.0 135000.0 9.23 301000.0 112000.0 8.33 12.4198 0.9987 2141121 PK04_097319 OC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2097 P24 compound treatment 229920.0 34700.0 2.37 225080.0 36000.0 2.68 3.5707 0.9981 2144273 PK04_097320 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A01 compound treatment 274560.0 81100.0 5.53 278200.0 86000.0 6.4 8.4395 0.9973 2141696 PK04_098001 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A02 compound treatment 234160.0 40700.0 2.78 235040.0 42900.0 3.19 4.2205 0.9976 2144133 PK04_098002 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A03 compound treatment 247760.0 54300.0 3.7 246040.0 53900.0 4.01 5.455 0.9992 2141089 PK04_098003 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A04 compound treatment 236360.0 42900.0 2.93 224640.0 32500.0 2.42 3.7792 0.9955 2142093 PK04_098004 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A05 compound treatment 289800.0 96400.0 6.57 281280.0 89100.0 6.63 9.3363 1.0 2141744 PK04_098005 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A06 compound treatment 259360.0 65900.0 4.5 260240.0 68100.0 5.07 6.7616 0.9982 2143237 PK04_098006 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A07 compound treatment 265040.0 71600.0 4.88 281320.0 89200.0 6.64 8.1448 0.9886 2141337 PK04_098007 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A08 compound treatment 259320.0 65900.0 4.49 173840.0 -18300.0 -1.36 2.2126 0.4712 2144129 PK04_098008 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A09 compound treatment 175600.0 -17800.0 -1.21 176280.0 -15900.0 -1.18 -1.695 -0.9999 2141791 PK04_098009 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A10 compound treatment 247600.0 54200.0 3.69 246680.0 54500.0 4.06 5.481 0.9989 2144193 PK04_098010 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A11 compound treatment 431480.0 238000.0 16.23 418240.0 226000.0 16.83 23.3744 0.9998 2141133 PK04_098011 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A12 compound treatment 254840.0 61400.0 4.19 236480.0 44300.0 3.3 5.2932 0.993 2143993 PK04_098012 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A13 mock treatment 177160.0 -16300.0 -1.11 177560.0 -14600.0 -1.09 -1.5524 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A14 mock treatment 183520.0 -9900.0 -0.67 183280.0 -8890.0 -0.66 -0.9448 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A15 compound treatment 294000.0 101000.0 6.86 291480.0 99300.0 7.39 10.0756 0.9993 2141695 PK04_098013 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A16 compound treatment 247920.0 54500.0 3.72 236800.0 44600.0 3.32 4.9765 0.9984 2144913 PK04_098014 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A17 compound treatment 173560.0 -19900.0 -1.35 170400.0 -21800.0 -1.62 -2.1028 -0.996 2141801 PK04_098015 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A18 compound treatment 268640.0 75200.0 5.13 252920.0 60800.0 4.52 6.8237 0.998 2142117 PK04_098016 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A19 compound treatment 278600.0 85200.0 5.81 267680.0 75500.0 5.62 8.0807 0.9999 2141835 PK04_098017 O[C@@H](CNC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A20 compound treatment 176960.0 -16500.0 -1.12 172680.0 -19500.0 -1.45 -1.8189 -0.992 2144205 PK04_098018 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A21 compound treatment 269720.0 76300.0 5.2 232160.0 40000.0 2.98 5.7832 0.9649 2141920 PK04_098019 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A22 compound treatment 225120.0 31700.0 2.16 219520.0 27400.0 2.04 2.9679 0.9996 2141945 PK04_098020 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A23 compound treatment 402320.0 209000.0 14.24 402760.0 211000.0 15.67 21.154 0.9989 2141111 PK04_098021 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 A24 compound treatment 219360.0 25900.0 1.77 216160.0 24000.0 1.79 2.5134 1.0 2143385 PK04_098022 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B01 compound treatment 284680.0 91300.0 6.22 240440.0 48300.0 3.59 6.9402 0.9659 2142845 PK04_098023 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B02 compound treatment 239520.0 46100.0 3.14 224640.0 32500.0 2.42 3.9316 0.9916 2143009 PK04_098024 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B03 compound treatment 233360.0 39900.0 2.72 228240.0 36100.0 2.68 3.8241 1.0 2144209 PK04_098025 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B04 compound treatment 259200.0 65800.0 4.48 238760.0 46600.0 3.47 5.6234 0.9919 2142037 PK04_098026 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B05 compound treatment 226960.0 33500.0 2.29 227360.0 35200.0 2.62 3.4692 0.9977 2144313 PK04_098027 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B06 compound treatment 266000.0 72600.0 4.95 284920.0 92800.0 6.9 8.3805 0.9867 2143245 PK04_098028 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B07 compound treatment 231680.0 38300.0 2.61 219720.0 27600.0 2.05 3.2947 0.9929 2144661 PK04_098029 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B08 compound treatment 283720.0 90300.0 6.16 282720.0 90600.0 6.74 9.119 0.999 2143409 PK04_098030 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B09 compound treatment 235280.0 41900.0 2.85 229480.0 37300.0 2.78 3.9819 0.9999 2144745 PK04_098031 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B10 compound treatment 227480.0 34100.0 2.32 220480.0 28300.0 2.11 3.1322 0.9988 2143049 PK04_098032 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B11 compound treatment 239960.0 46500.0 3.17 253840.0 61700.0 4.59 5.4895 0.9837 2143257 PK04_098033 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B12 compound treatment 272360.0 78900.0 5.38 272520.0 80400.0 5.98 8.0346 0.9986 2141502 PK04_098034 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B13 mock treatment 178160.0 -15300.0 -1.04 176480.0 -15700.0 -1.17 -1.561 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B14 mock treatment 178120.0 -15300.0 -1.04 176920.0 -15200.0 -1.13 -1.5398 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B15 compound treatment 247600.0 54200.0 3.69 241080.0 48900.0 3.64 5.1863 1.0 2142113 PK04_098035 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B16 compound treatment 239640.0 46200.0 3.15 241400.0 49200.0 3.66 4.8194 0.9972 2141859 PK04_098036 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B17 compound treatment 217320.0 23900.0 1.63 211880.0 19700.0 1.47 2.1898 0.9986 2144033 PK04_098037 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B18 compound treatment 259320.0 65900.0 4.49 268280.0 76100.0 5.66 7.1828 0.9934 2141540 PK04_098038 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B19 compound treatment 258040.0 64600.0 4.41 237880.0 45700.0 3.4 5.5212 0.9918 2144437 PK04_098039 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B20 compound treatment 236720.0 43300.0 2.95 239720.0 47600.0 3.54 4.5902 0.9959 2144725 PK04_098040 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B21 compound treatment 209640.0 16200.0 1.11 196920.0 4750.0 0.35 1.0323 0.889 2143413 PK04_098041 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B22 compound treatment 231000.0 37600.0 2.56 218920.0 26800.0 1.99 3.2198 0.9922 2141509 PK04_098042 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B23 compound treatment 266040.0 72600.0 4.95 264600.0 72400.0 5.39 7.3131 0.9991 2142009 PK04_098043 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 B24 compound treatment 271840.0 78400.0 5.35 249320.0 57200.0 4.25 6.7885 0.9936 2141342 PK04_098044 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C01 compound treatment 234200.0 40800.0 2.78 254680.0 62500.0 4.65 5.256 0.9697 2141145 PK04_098045 OC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C02 compound treatment 175800.0 -17600.0 -1.2 180360.0 -11800.0 -0.88 -1.4706 -0.9882 2143097 PK04_098046 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C03 compound treatment 277800.0 84400.0 5.75 276360.0 84200.0 6.27 8.4989 0.9991 2141834 PK04_098047 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C04 compound treatment 265080.0 71700.0 4.89 248840.0 56700.0 4.22 6.4374 0.9973 2142605 PK04_098048 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C05 compound treatment 334320.0 141000.0 9.61 313280.0 121000.0 9.01 13.1667 0.9995 2141398 PK04_098049 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C06 compound treatment 253920.0 60500.0 4.12 235280.0 43100.0 3.21 5.1857 0.9923 2143013 PK04_098050 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C07 compound treatment 206560.0 13100.0 0.9 220200.0 28000.0 2.09 2.109 0.9287 2141793 PK04_098051 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C08 compound treatment 275720.0 82300.0 5.61 285920.0 93800.0 6.98 8.9017 0.9942 2143277 PK04_098052 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C09 compound treatment 271680.0 78300.0 5.34 260480.0 68300.0 5.08 7.3681 0.9997 2141681 PK04_098053 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C10 compound treatment 286360.0 92900.0 6.34 281120.0 89000.0 6.62 9.1621 0.9998 2144125 PK04_098054 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C11 mock treatment 183480.0 -9940.0 -0.68 190520.0 -1650.0 -0.12 -0.5657 -0.8216 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C12 mock treatment 185680.0 -7740.0 -0.53 189520.0 -2650.0 -0.2 -0.5122 -0.9097 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C13 compound treatment 186320.0 -7100.0 -0.48 179120.0 -13000.0 -0.97 -1.0287 -0.9483 2141376 PK04_098055 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C14 compound treatment 207280.0 13900.0 0.95 231360.0 39200.0 2.92 2.731 0.8906 2143897 PK04_098056 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C15 mock treatment 183280.0 -10100.0 -0.69 181440.0 -10700.0 -0.8 -1.0532 -0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C16 mock treatment 188640.0 -4780.0 -0.33 185680.0 -6490.0 -0.48 -0.5716 -0.9817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C17 compound treatment 244880.0 51500.0 3.51 237120.0 45000.0 3.35 4.8468 0.9997 2141461 PK04_098057 O[C@@H](CNC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C18 compound treatment 244600.0 51200.0 3.49 217360.0 25200.0 1.88 3.7933 0.9576 2143145 PK04_098058 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C19 compound treatment 290880.0 97500.0 6.64 298320.0 106000.0 7.9 10.2852 0.9963 2141551 PK04_098059 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C20 compound treatment 221800.0 28400.0 1.93 209280.0 17100.0 1.27 2.269 0.9794 2144941 PK04_098060 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C21 compound treatment 262360.0 68900.0 4.7 249960.0 57800.0 4.3 6.3652 0.999 2141535 PK04_098061 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C22 compound treatment 241920.0 48500.0 3.31 233560.0 41400.0 3.08 4.5167 0.9994 2142185 PK04_098062 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C23 compound treatment 171360.0 -22100.0 -1.5 170600.0 -21600.0 -1.61 -2.1983 -0.9995 2141425 PK04_098063 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 C24 compound treatment 242560.0 49100.0 3.35 237560.0 45400.0 3.38 4.7581 1.0 2144353 PK04_098064 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D01 compound treatment 264120.0 70700.0 4.82 259840.0 67700.0 5.04 6.97 0.9998 2143317 PK04_098065 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D02 compound treatment 279600.0 86200.0 5.88 264160.0 72000.0 5.36 7.9436 0.9989 2144805 PK04_098066 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D03 compound treatment 219800.0 26400.0 1.8 213680.0 21500.0 1.6 2.4041 0.9983 2142937 PK04_098067 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D04 compound treatment 270480.0 77100.0 5.25 259480.0 67300.0 5.01 7.2577 0.9997 2141997 PK04_098068 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D05 compound treatment 217320.0 23900.0 1.63 218840.0 26700.0 1.99 2.5561 0.9952 2144781 PK04_098069 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D06 compound treatment 244560.0 51100.0 3.49 227960.0 35800.0 2.66 4.3493 0.9912 2144025 PK04_098070 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D07 compound treatment 258960.0 65500.0 4.47 233960.0 41800.0 3.11 5.3592 0.9843 2144817 PK04_098071 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D08 compound treatment 253760.0 60300.0 4.11 244680.0 52500.0 3.91 5.6727 0.9997 2144197 PK04_098072 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D09 compound treatment 256800.0 63400.0 4.32 237560.0 45400.0 3.38 5.4446 0.9926 2144761 PK04_098073 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D10 compound treatment 275520.0 82100.0 5.6 263400.0 71200.0 5.3 7.7069 0.9996 2142125 PK04_098074 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D11 mock treatment 189200.0 -4220.0 -0.29 183800.0 -8370.0 -0.62 -0.6436 -0.9384 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D12 mock treatment 183200.0 -10200.0 -0.7 183880.0 -8290.0 -0.62 -0.9286 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D13 compound treatment 246120.0 52700.0 3.59 229800.0 37600.0 2.8 4.5213 0.9924 2143225 PK04_098075 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D14 compound treatment 248400.0 55000.0 3.75 230000.0 37800.0 2.82 4.6418 0.9901 2144233 PK04_098076 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D15 mock treatment 185000.0 -8420.0 -0.57 183120.0 -9050.0 -0.67 -0.8818 -0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D16 mock treatment 183720.0 -9700.0 -0.66 181440.0 -10700.0 -0.8 -1.032 -0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D17 compound treatment 195520.0 2100.0 0.14 206400.0 14200.0 1.06 0.8505 0.7955 2143045 PK04_098077 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D18 compound treatment 271680.0 78300.0 5.34 243200.0 51000.0 3.8 6.4587 0.9861 2142013 PK04_098078 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D19 compound treatment 217520.0 24100.0 1.64 226560.0 34400.0 2.56 2.972 0.977 2142213 PK04_098079 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D20 compound treatment 223320.0 29900.0 2.04 212440.0 20300.0 1.51 2.5085 0.989 2141447 PK04_098080 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D21 compound treatment 246920.0 53500.0 3.65 236880.0 44700.0 3.33 4.9325 0.999 2143393 PK04_098081 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D22 compound treatment 247920.0 54500.0 3.72 259640.0 67500.0 5.02 6.1785 0.989 2065844 PK04_098082 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D23 compound treatment 220800.0 27400.0 1.87 220520.0 28400.0 2.11 2.8123 0.9981 2144185 PK04_098083 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 D24 compound treatment 207600.0 14200.0 0.97 224640.0 32500.0 2.42 2.3928 0.9192 2141197 PK04_098084 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E01 mock treatment 186760.0 -6660.0 -0.45 182640.0 -9530.0 -0.71 -0.8223 -0.9768 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E02 mock treatment 180000.0 -13400.0 -0.91 185160.0 -7010.0 -0.52 -1.0155 -0.9645 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E03 compound treatment 273680.0 80300.0 5.47 258440.0 66300.0 4.93 7.3572 0.9987 2141526 PK04_098085 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E04 compound treatment 294440.0 101000.0 6.89 281360.0 89200.0 6.64 9.5642 0.9998 2142637 PK04_098086 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E05 compound treatment 266080.0 72700.0 4.95 281120.0 89000.0 6.62 8.1844 0.9898 2141181 PK04_098087 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E06 compound treatment 260920.0 67500.0 4.6 264840.0 72700.0 5.41 7.0789 0.9968 2142777 PK04_098088 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E07 compound treatment 229280.0 35900.0 2.44 226080.0 33900.0 2.52 3.5137 0.9999 2141090 PK04_098089 OC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E08 compound treatment 294720.0 101000.0 6.91 299120.0 107000.0 7.96 10.5124 0.9975 2144801 PK04_098090 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E09 mock treatment 199120.0 5700.0 0.39 192200.0 34.9 0.0 0.2767 0.7118 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E10 mock treatment 199320.0 5900.0 0.4 201960.0 9790.0 0.73 0.8 0.9608 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E11 compound treatment 267880.0 74500.0 5.08 247160.0 55000.0 4.09 6.4839 0.9943 2141328 PK04_098091 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E12 compound treatment 282600.0 89200.0 6.08 279720.0 87600.0 6.52 8.9071 0.9994 2144117 PK04_098092 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E13 compound treatment 320640.0 127000.0 8.67 329600.0 137000.0 10.23 13.366 0.9966 2141750 PK04_098093 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E14 compound treatment 284840.0 91400.0 6.23 284960.0 92800.0 6.91 9.2909 0.9987 2142133 PK04_098094 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E15 compound treatment 265040.0 71600.0 4.88 275200.0 83000.0 6.18 7.8227 0.9932 2141837 PK04_098095 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E16 compound treatment 230200.0 36800.0 2.51 255720.0 63600.0 4.73 5.1179 0.9559 2143333 PK04_098096 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E17 mock treatment 189760.0 -3660.0 -0.25 198840.0 6670.0 0.5 0.1749 0.3147 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E18 mock treatment 194720.0 1300.0 0.09 195840.0 3670.0 0.27 0.2562 0.8908 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E19 compound treatment 297880.0 104000.0 7.12 289640.0 97500.0 7.25 10.1658 1.0 2141392 PK04_098097 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E20 compound treatment 254040.0 60600.0 4.13 245480.0 53300.0 3.97 5.7283 0.9998 2144457 PK04_098098 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E21 compound treatment 322240.0 129000.0 8.78 327160.0 135000.0 10.05 13.3148 0.9978 2141783 PK04_098099 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E22 compound treatment 269560.0 76100.0 5.19 262120.0 70000.0 5.21 7.3522 1.0 2142073 PK04_098100 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E23 compound treatment 248680.0 55300.0 3.77 228840.0 36700.0 2.73 4.5942 0.9875 2141929 PK04_098101 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccccc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 E24 compound treatment 215240.0 21800.0 1.49 257320.0 65200.0 4.85 4.481 0.8834 2141993 PK04_098102 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F01 mock treatment 186880.0 -6540.0 -0.45 181840.0 -10300.0 -0.77 -0.8586 -0.9664 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F02 mock treatment 187080.0 -6340.0 -0.43 187280.0 -4890.0 -0.36 -0.5626 -0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F03 compound treatment 241720.0 48300.0 3.29 226800.0 34600.0 2.58 4.1513 0.9927 2142917 PK04_098103 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F04 compound treatment 268920.0 75500.0 5.15 242600.0 50400.0 3.75 6.2941 0.988 2142953 PK04_098104 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F05 compound treatment 242680.0 49300.0 3.36 235480.0 43300.0 3.22 4.6544 0.9998 2144897 PK04_098105 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F06 compound treatment 230080.0 36700.0 2.5 228640.0 36500.0 2.71 3.687 0.9991 2144329 PK04_098106 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F07 compound treatment 251280.0 57900.0 3.94 246880.0 54700.0 4.07 5.6689 0.9999 2144721 PK04_098107 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F08 compound treatment 258640.0 65200.0 4.45 250440.0 58300.0 4.34 6.2111 0.9999 2143969 PK04_098108 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F09 mock treatment 190760.0 -2660.0 -0.18 193840.0 1670.0 0.12 -0.04 -0.1818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F10 mock treatment 189880.0 -3540.0 -0.24 192680.0 515.0 0.04 -0.1435 -0.5874 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F11 compound treatment 239680.0 46300.0 3.15 227360.0 35200.0 2.62 4.0824 0.9957 2141973 PK04_098109 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F12 compound treatment 294600.0 101000.0 6.9 231520.0 39400.0 2.93 6.949 0.9272 2141515 PK04_098110 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F13 compound treatment 261960.0 68500.0 4.67 261800.0 69600.0 5.18 6.969 0.9987 2144053 PK04_098111 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F14 compound treatment 298240.0 105000.0 7.15 300120.0 108000.0 8.03 10.7347 0.9983 2143249 PK04_098112 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F15 compound treatment 268840.0 75400.0 5.14 253760.0 61600.0 4.58 6.8776 0.9984 2144873 PK04_098113 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F16 compound treatment 271760.0 78300.0 5.34 270240.0 78100.0 5.81 7.8856 0.9991 2141199 PK04_098114 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F17 mock treatment 195280.0 1860.0 0.13 192640.0 475.0 0.04 0.1148 0.8709 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F18 mock treatment 194960.0 1540.0 0.11 199920.0 7750.0 0.58 0.4825 0.8224 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F19 compound treatment 252240.0 58800.0 4.01 246000.0 53800.0 4.01 5.6689 1.0 2142825 PK04_098115 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F20 compound treatment 247200.0 53800.0 3.67 238840.0 46700.0 3.47 5.0491 0.9996 2144217 PK04_098116 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F21 compound treatment 245040.0 51600.0 3.52 228400.0 36200.0 2.7 4.3956 0.9914 2144057 PK04_098117 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F22 compound treatment 259560.0 66100.0 4.51 257920.0 65800.0 4.89 6.6491 0.9992 2141689 PK04_098118 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F23 compound treatment 274680.0 81300.0 5.54 277520.0 85400.0 6.35 8.4095 0.9977 2144037 PK04_098119 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 F24 compound treatment 208440.0 15000.0 1.02 202760.0 10600.0 0.79 1.2818 0.9917 2141464 PK04_098120 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G01 compound treatment 340800.0 147000.0 10.05 339240.0 147000.0 10.95 14.8453 0.9991 2141573 PK04_098121 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G02 compound treatment 249440.0 56000.0 3.82 246120.0 54000.0 4.02 5.5402 0.9997 2144113 PK04_098122 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G03 mock treatment 193880.0 462.0 0.03 198720.0 6550.0 0.49 0.3672 0.7512 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G04 mock treatment 192440.0 -978.0 -0.07 195800.0 3630.0 0.27 0.1441 0.5173 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G05 compound treatment 276320.0 82900.0 5.65 251440.0 59300.0 4.41 7.1161 0.9925 2141531 PK04_098123 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G06 compound treatment 258240.0 64800.0 4.42 264400.0 72200.0 5.38 6.9265 0.9953 2143985 PK04_098124 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G07 compound treatment 461600.0 268000.0 18.28 439440.0 247000.0 18.4 25.9421 1.0 2065843 PK04_098125 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G08 compound treatment 267160.0 73700.0 5.03 259800.0 67600.0 5.03 7.1144 1.0 2144713 PK04_098126 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G09 compound treatment 284400.0 91000.0 6.2 286000.0 93800.0 6.98 9.3244 0.9983 2141779 PK04_098127 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G10 compound treatment 291520.0 98100.0 6.69 277880.0 85700.0 6.38 9.2403 0.9997 2142633 PK04_098128 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G11 compound treatment 277560.0 84100.0 5.74 262840.0 70700.0 5.26 7.7758 0.9991 2141711 PK04_098129 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G12 compound treatment 285200.0 91800.0 6.26 213800.0 21600.0 1.61 5.5632 0.861 2142689 PK04_098130 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G13 compound treatment 263160.0 69700.0 4.75 259600.0 67400.0 5.02 6.9111 0.9996 2141802 PK04_098131 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G14 compound treatment 242000.0 48600.0 3.31 253480.0 61300.0 4.56 5.5689 0.9876 2142905 PK04_098132 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G15 compound treatment 239160.0 45700.0 3.12 249680.0 57500.0 4.28 5.232 0.9879 2141192 PK04_098133 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G16 compound treatment 358320.0 165000.0 11.24 324200.0 132000.0 9.83 14.8983 0.9978 2142129 PK04_098134 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G17 compound treatment 302480.0 109000.0 7.44 321400.0 129000.0 9.62 12.059 0.9919 2141728 PK04_098135 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G18 compound treatment 290120.0 96700.0 6.59 298160.0 106000.0 7.89 10.2401 0.996 2144641 PK04_098136 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G19 mock treatment 195840.0 2420.0 0.17 200040.0 7870.0 0.59 0.5312 0.8724 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G20 mock treatment 193200.0 -218.0 -0.01 189160.0 -3010.0 -0.22 -0.1687 -0.7525 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G21 compound treatment 218600.0 25200.0 1.72 291320.0 99200.0 7.38 6.4323 0.8489 2141885 PK04_098137 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccccc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G22 compound treatment 215440.0 22000.0 1.5 251600.0 59400.0 4.42 4.1896 0.8969 2144357 PK04_098138 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G23 compound treatment 288440.0 95000.0 6.48 300360.0 108000.0 8.05 10.2749 0.9942 2141361 PK04_098139 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 G24 compound treatment 233640.0 40200.0 2.74 233400.0 41200.0 3.07 4.1091 0.9984 2142625 PK04_098140 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H01 compound treatment 247440.0 54000.0 3.68 247240.0 55100.0 4.1 5.5028 0.9986 2142737 PK04_098141 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H02 compound treatment 241840.0 48400.0 3.3 237800.0 45600.0 3.4 4.736 0.9999 2144017 PK04_098142 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H03 mock treatment 192600.0 -818.0 -0.06 188920.0 -3250.0 -0.24 -0.2102 -0.8481 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H04 mock treatment 195840.0 2420.0 0.17 190680.0 -1490.0 -0.11 0.0386 0.1943 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H05 compound treatment 259240.0 65800.0 4.49 301840.0 110000.0 8.16 8.9451 0.9603 2143493 PK04_098143 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H06 compound treatment 284120.0 90700.0 6.18 276000.0 83800.0 6.24 8.7846 1.0 2141857 PK04_098144 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H07 compound treatment 303320.0 110000.0 7.49 317080.0 125000.0 9.3 11.8722 0.9943 2143497 PK04_098145 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H08 compound treatment 292040.0 98600.0 6.72 279320.0 87200.0 6.49 9.3412 0.9998 2141183 PK04_098146 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H09 compound treatment 332640.0 139000.0 9.49 279760.0 87600.0 6.52 11.3216 0.9832 2143289 PK04_098147 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H10 compound treatment 298040.0 105000.0 7.13 264720.0 72600.0 5.4 8.862 0.9906 2142033 PK04_098148 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H11 compound treatment 263640.0 70200.0 4.79 248120.0 56000.0 4.16 6.3301 0.9976 2143345 PK04_098149 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H12 compound treatment 325520.0 132000.0 9.01 289920.0 97800.0 7.28 11.513 0.9944 2141965 PK04_098150 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H13 compound treatment 278360.0 84900.0 5.79 264360.0 72200.0 5.37 7.8944 0.9993 2142053 PK04_098151 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H14 compound treatment 293920.0 101000.0 6.85 277240.0 85100.0 6.33 9.3223 0.9992 2143285 PK04_098152 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H15 compound treatment 258200.0 64800.0 4.42 240440.0 48300.0 3.59 5.6636 0.9948 2143953 PK04_098153 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H16 compound treatment 279320.0 85900.0 5.86 280360.0 88200.0 6.56 8.7827 0.9984 2142849 PK04_098154 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H17 compound treatment 345560.0 152000.0 10.37 330160.0 138000.0 10.27 14.5969 1.0 2142197 PK04_098155 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H18 compound treatment 275920.0 82500.0 5.62 268560.0 76400.0 5.69 7.9978 1.0 2141678 PK04_098156 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H19 mock treatment 193880.0 462.0 0.03 195920.0 3750.0 0.28 0.2199 0.7818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H20 mock treatment 193800.0 382.0 0.03 192080.0 -85.1 -0.01 0.0139 0.52 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H21 compound treatment 269200.0 75800.0 5.17 260960.0 68800.0 5.12 7.2738 1.0 2142657 PK04_098157 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H22 compound treatment 288640.0 95200.0 6.49 274480.0 82300.0 6.13 8.9225 0.9996 2141194 PK04_098158 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H23 compound treatment 240640.0 47200.0 3.22 246840.0 54700.0 4.07 5.1539 0.9933 2142665 PK04_098159 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 H24 compound treatment 193040.0 -378.0 -0.03 203840.0 11700.0 0.87 0.5962 0.6858 2141813 PK04_098160 O[C@@H](CNC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I01 compound treatment 309720.0 116000.0 7.93 298840.0 107000.0 7.94 11.2208 1.0 2141395 PK04_098161 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I02 compound treatment 257800.0 64400.0 4.39 275080.0 82900.0 6.17 7.4674 0.9861 2144813 PK04_098162 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I03 compound treatment 417800.0 224000.0 15.3 391760.0 200000.0 14.86 21.3213 0.9999 2141107 PK04_098163 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I04 compound treatment 260040.0 66600.0 4.54 266760.0 74600.0 5.55 7.1375 0.995 2142597 PK04_098164 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I05 mock treatment 194920.0 1500.0 0.1 198320.0 6150.0 0.46 0.3963 0.8443 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I06 mock treatment 199600.0 6180.0 0.42 201960.0 9790.0 0.73 0.8135 0.9661 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I07 compound treatment 258840.0 65400.0 4.46 256600.0 64400.0 4.8 6.5449 0.9993 2141144 PK04_098165 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I08 compound treatment 267320.0 73900.0 5.04 259000.0 66800.0 4.97 7.0801 1.0 2142693 PK04_098166 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I09 compound treatment 274480.0 81100.0 5.53 269960.0 77800.0 5.79 8.002 0.9997 2141896 PK04_098167 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccccc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I10 compound treatment 292280.0 98900.0 6.74 270920.0 78800.0 5.86 8.9107 0.9976 2141957 PK04_098168 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I11 compound treatment 293960.0 101000.0 6.85 286480.0 94300.0 7.02 9.8105 0.9999 2141394 PK04_098169 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I12 compound treatment 335080.0 142000.0 9.66 319040.0 127000.0 9.44 13.5064 0.9999 2142049 PK04_098170 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I13 compound treatment 309800.0 116000.0 7.93 295400.0 103000.0 7.68 11.0436 0.9999 2141346 PK04_098171 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I14 compound treatment 304240.0 111000.0 7.56 287520.0 95400.0 7.1 10.3609 0.9995 2143477 PK04_098172 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I15 compound treatment 305480.0 112000.0 7.64 296480.0 104000.0 7.76 10.8922 1.0 2141373 PK04_098173 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I16 compound treatment 291080.0 97700.0 6.66 278360.0 86200.0 6.42 9.2444 0.9998 2144645 PK04_098174 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I17 compound treatment 250200.0 56800.0 3.87 245720.0 53600.0 3.99 5.5558 0.9999 2141116 PK04_098175 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I18 compound treatment 270400.0 77000.0 5.25 272520.0 80400.0 5.98 7.9401 0.9979 2142097 PK04_098176 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I19 compound treatment 214880.0 21500.0 1.46 218240.0 26100.0 1.94 2.4069 0.9903 2141442 PK04_098177 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I20 compound treatment 308280.0 115000.0 7.83 301240.0 109000.0 8.12 11.2777 0.9998 2142005 PK04_098178 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I21 mock treatment 193680.0 262.0 0.02 194640.0 2470.0 0.18 0.1429 0.772 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I22 mock treatment 188760.0 -4660.0 -0.32 188520.0 -3650.0 -0.27 -0.4164 -0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I23 compound treatment 395880.0 202000.0 13.8 422360.0 230000.0 17.13 21.875 0.9943 2141137 PK04_098179 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 I24 compound treatment 178320.0 -15100.0 -1.03 179920.0 -12200.0 -0.91 -1.3723 -0.9982 2144905 PK04_098180 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J01 compound treatment 239800.0 46400.0 3.16 240560.0 48400.0 3.6 4.7829 0.9979 2142853 PK04_098181 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J02 compound treatment 253120.0 59700.0 4.07 256120.0 64000.0 4.76 6.2439 0.997 2141434 PK04_098182 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J03 compound treatment 240720.0 47300.0 3.22 237400.0 45200.0 3.37 4.661 0.9998 2142925 PK04_098183 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J04 compound treatment 230720.0 37300.0 2.54 226240.0 34100.0 2.54 3.5915 1.0 2141810 PK04_098184 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J05 mock treatment 198200.0 4780.0 0.33 197840.0 5670.0 0.42 0.5292 0.9918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J06 mock treatment 196800.0 3380.0 0.23 199320.0 7150.0 0.53 0.5396 0.9298 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J07 compound treatment 264840.0 71400.0 4.87 241160.0 49000.0 3.65 6.0216 0.9898 2143253 PK04_098185 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J08 compound treatment 313520.0 120000.0 8.19 303400.0 111000.0 8.28 11.644 1.0 2141219 PK04_098186 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J09 compound treatment 273480.0 80100.0 5.46 253400.0 61200.0 4.56 7.0823 0.996 2142945 PK04_098187 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J10 compound treatment 243440.0 50000.0 3.41 235120.0 43000.0 3.2 4.6721 0.9995 2141450 PK04_098188 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J11 compound treatment 213360.0 19900.0 1.36 210000.0 17800.0 1.33 1.9 0.9999 2144285 PK04_098189 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J12 compound treatment 403640.0 210000.0 14.33 446600.0 254000.0 18.94 23.5248 0.9906 2141139 PK04_098190 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J13 compound treatment 302040.0 109000.0 7.41 298240.0 106000.0 7.89 10.819 0.9995 2143473 PK04_098191 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J14 compound treatment 263120.0 69700.0 4.75 251520.0 59400.0 4.42 6.4839 0.9993 2144013 PK04_098192 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J15 compound treatment 303560.0 110000.0 7.51 279240.0 87100.0 6.48 9.8923 0.9973 2142837 PK04_098193 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J16 compound treatment 285080.0 91700.0 6.25 255960.0 63800.0 4.75 7.7763 0.9908 2141784 PK04_098194 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J17 compound treatment 277120.0 83700.0 5.71 267720.0 75600.0 5.62 8.0114 1.0 2144425 PK04_098195 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J18 compound treatment 312560.0 119000.0 8.12 289440.0 97300.0 7.24 10.863 0.9984 2141332 PK04_098196 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J19 compound treatment 270040.0 76600.0 5.22 270800.0 78600.0 5.85 7.8322 0.9984 2143957 PK04_098197 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J20 compound treatment 283640.0 90200.0 6.15 273400.0 81200.0 6.05 8.6247 1.0 2141933 PK04_098198 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J21 mock treatment 188320.0 -5100.0 -0.35 187880.0 -4290.0 -0.32 -0.4713 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J22 mock treatment 182000.0 -11400.0 -0.78 184320.0 -7850.0 -0.58 -0.9633 -0.99 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J23 compound treatment 259400.0 66000.0 4.5 252880.0 60700.0 4.52 6.3762 1.0 2144049 PK04_098199 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 J24 compound treatment 234600.0 41200.0 2.81 224760.0 32600.0 2.43 3.7007 0.9974 2141196 PK04_098200 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K01 compound treatment 327120.0 134000.0 9.12 313360.0 121000.0 9.02 12.8238 1.0 2141522 PK04_098201 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K02 compound treatment 268600.0 75200.0 5.13 257920.0 65800.0 4.89 7.0849 0.9997 2142617 PK04_098202 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K03 compound treatment 236320.0 42900.0 2.92 230520.0 38400.0 2.85 4.0868 0.9999 2141439 PK04_098203 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K04 compound treatment 320040.0 127000.0 8.63 291920.0 99800.0 7.42 11.3541 0.9972 2143329 PK04_098204 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K05 compound treatment 313560.0 120000.0 8.19 304360.0 112000.0 8.35 11.6964 1.0 2141725 PK04_098205 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K06 compound treatment 322680.0 129000.0 8.81 323480.0 131000.0 9.77 13.1423 0.9987 2142973 PK04_098206 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K07 mock treatment 204000.0 10600.0 0.72 195280.0 3110.0 0.23 0.6741 0.8895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K08 mock treatment 202520.0 9100.0 0.62 199920.0 7750.0 0.58 0.8469 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K09 compound treatment 421000.0 228000.0 15.52 402960.0 211000.0 15.69 22.065 1.0 2141136 PK04_098207 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K10 compound treatment 284200.0 90800.0 6.19 276120.0 84000.0 6.25 8.7948 1.0 2143005 PK04_098208 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K11 compound treatment 306320.0 113000.0 7.7 296000.0 104000.0 7.73 10.9074 1.0 2141925 PK04_098209 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K12 compound treatment 268040.0 74600.0 5.09 271000.0 78800.0 5.87 7.7463 0.9975 2144741 PK04_098210 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K13 compound treatment 391480.0 198000.0 13.5 371000.0 179000.0 13.31 18.9599 1.0 2141147 PK04_098211 OC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K14 compound treatment 332120.0 139000.0 9.46 320320.0 128000.0 9.54 13.4311 1.0 2143465 PK04_098212 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K15 mock treatment 209240.0 15800.0 1.08 206960.0 14800.0 1.1 1.5414 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K16 mock treatment 206960.0 13500.0 0.92 197200.0 5030.0 0.37 0.9178 0.9211 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K17 compound treatment 330480.0 137000.0 9.34 316560.0 124000.0 9.26 13.1542 1.0 2141530 PK04_098213 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K18 compound treatment 256240.0 62800.0 4.28 286160.0 94000.0 7.0 7.9753 0.9723 2143169 PK04_098214 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K19 compound treatment 276880.0 83500.0 5.69 269840.0 77700.0 5.78 8.1114 1.0 2141707 PK04_098215 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K20 compound treatment 211640.0 18200.0 1.24 208760.0 16600.0 1.24 1.7518 1.0 2143073 PK04_098216 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K21 compound treatment 194360.0 942.0 0.06 190640.0 -1530.0 -0.11 -0.0349 -0.2673 2141428 PK04_098217 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K22 compound treatment 266320.0 72900.0 4.97 266040.0 73900.0 5.5 7.4024 0.9987 2142725 PK04_098218 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K23 mock treatment 183520.0 -9900.0 -0.67 183240.0 -8930.0 -0.66 -0.9469 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 K24 mock treatment 182040.0 -11400.0 -0.78 180600.0 -11600.0 -0.86 -1.1572 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L01 compound treatment 260240.0 66800.0 4.56 252280.0 60100.0 4.47 6.3851 1.0 2143889 PK04_098219 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L02 compound treatment 297800.0 104000.0 7.12 273640.0 81500.0 6.06 9.3199 0.9968 2141700 PK04_098220 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L03 compound treatment 254880.0 61500.0 4.19 226920.0 34800.0 2.59 4.792 0.9731 2142733 PK04_098221 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L04 compound treatment 261680.0 68300.0 4.65 279560.0 87400.0 6.5 7.8902 0.9865 2141934 PK04_098222 O[C@@H](CNC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L05 compound treatment 277560.0 84100.0 5.74 263520.0 71400.0 5.31 7.8116 0.9993 2143873 PK04_098223 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L06 compound treatment 271680.0 78300.0 5.34 255400.0 63200.0 4.71 7.1008 0.998 2141797 PK04_098224 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L07 mock treatment 192360.0 -1060.0 -0.07 193800.0 1630.0 0.12 0.035 0.2476 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L08 mock treatment 196320.0 2900.0 0.2 194760.0 2590.0 0.19 0.2765 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L09 compound treatment 260920.0 67500.0 4.6 243840.0 51700.0 3.85 5.9737 0.996 2142957 PK04_098225 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L10 compound treatment 216240.0 22800.0 1.56 212200.0 20000.0 1.49 2.1546 0.9998 3413983 PK04_098226 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L11 compound treatment 266760.0 73300.0 5.0 258960.0 66800.0 4.97 7.051 1.0 2142717 PK04_098227 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L12 compound treatment 210960.0 17500.0 1.2 214520.0 22400.0 1.66 2.0222 0.9869 3413985 PK04_098228 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L13 compound treatment 285760.0 92300.0 6.3 276320.0 84200.0 6.26 8.8805 1.0 2143357 PK04_098229 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L14 compound treatment 225800.0 32400.0 2.21 231280.0 39100.0 2.91 3.6196 0.9907 3413987 PK04_098230 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L15 mock treatment 199160.0 5740.0 0.39 196800.0 4630.0 0.34 0.5207 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L16 mock treatment 200280.0 6860.0 0.47 196080.0 3910.0 0.29 0.5368 0.974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L17 compound treatment 228400.0 35000.0 2.38 217520.0 25400.0 1.89 3.0208 0.9933 2143089 PK04_098231 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L18 compound treatment 222800.0 29400.0 2.0 219600.0 27400.0 2.04 2.8603 1.0 3413990 PK04_098232 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L19 compound treatment 254680.0 61300.0 4.18 253080.0 60900.0 4.53 6.1591 0.9992 2144137 PK04_098233 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L20 compound treatment 226680.0 33300.0 2.27 226560.0 34400.0 2.56 3.4136 0.9982 3413992 PK04_098234 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L21 compound treatment 279400.0 86000.0 5.86 277200.0 85000.0 6.33 8.6202 0.9993 2143369 PK04_098235 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L22 compound treatment 233880.0 40500.0 2.76 226960.0 34800.0 2.59 3.7818 0.9995 3413998 PK04_098236 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@@H]4OC(=O)[C@H](Cc5cccc(Br)c5)C/C=C/C[C@@H](Cc6cccc(Br)c6)C(=O)O[C@@H]14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L23 mock treatment 200160.0 6740.0 0.46 194600.0 2430.0 0.18 0.4532 0.9172 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 L24 mock treatment 214840.0 21400.0 1.46 243360.0 51200.0 3.81 3.727 0.9133 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M01 compound treatment 254240.0 60800.0 4.15 249280.0 57100.0 4.25 5.938 0.9999 2141977 PK04_098237 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M02 compound treatment 242520.0 49100.0 3.35 256560.0 64400.0 4.79 5.7561 0.9846 2144277 PK04_098238 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M03 compound treatment 289480.0 96100.0 6.55 274560.0 82400.0 6.13 8.9672 0.9995 2143353 PK04_098239 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M04 compound treatment 293000.0 99600.0 6.79 265600.0 73400.0 5.47 8.6654 0.9942 2142753 PK04_098240 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9(O)CCCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M05 compound treatment 278760.0 85300.0 5.82 275000.0 82800.0 6.17 8.4736 0.9996 2142713 PK04_098241 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M06 compound treatment 275640.0 82200.0 5.61 263960.0 71800.0 5.34 7.7422 0.9997 2143893 PK04_098242 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M07 compound treatment 210480.0 17100.0 1.16 206400.0 14200.0 1.06 1.5717 0.9989 2143173 PK04_098243 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M08 compound treatment 286400.0 93000.0 6.34 302960.0 111000.0 8.25 10.3134 0.9916 2143913 PK04_098244 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M09 mock treatment 203320.0 9900.0 0.68 198240.0 6070.0 0.45 0.7971 0.981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M10 mock treatment 203560.0 10100.0 0.69 203560.0 11400.0 0.85 1.0886 0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M11 compound treatment 293520.0 100000.0 6.82 290000.0 97800.0 7.28 9.9746 0.9995 2143965 PK04_098245 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M12 compound treatment 287760.0 94300.0 6.43 266640.0 74500.0 5.54 8.4675 0.9973 2144453 PK04_098246 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M13 mock treatment 206480.0 13100.0 0.89 204720.0 12600.0 0.93 1.2904 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M14 mock treatment 203720.0 10300.0 0.7 199320.0 7150.0 0.53 0.8732 0.9907 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M15 compound treatment 277040.0 83600.0 5.7 263280.0 71100.0 5.29 7.7739 0.9993 2142065 PK04_098247 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M16 compound treatment 300880.0 107000.0 7.33 259640.0 67500.0 5.02 8.7316 0.983 2143293 PK04_098248 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M17 compound treatment 275000.0 81600.0 5.56 270040.0 77900.0 5.8 8.0313 0.9998 2142857 PK04_098249 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M18 compound treatment 288840.0 95400.0 6.51 259960.0 67800.0 5.05 8.168 0.9921 2142613 PK04_098250 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M19 compound treatment 245600.0 52200.0 3.56 251920.0 59800.0 4.45 5.6604 0.9939 2142697 PK04_098251 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M20 compound treatment 249680.0 56300.0 3.84 248600.0 56400.0 4.2 5.6823 0.999 2144821 PK04_098252 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M21 compound treatment 199080.0 5660.0 0.39 190160.0 -2010.0 -0.15 0.1674 0.4046 2142965 PK04_098253 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M22 compound treatment 234400.0 41000.0 2.79 236400.0 44200.0 3.29 4.3037 0.9967 2144777 PK04_098254 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M23 compound treatment 210360.0 16900.0 1.16 215440.0 23300.0 1.73 2.0416 0.9806 2141143 PK04_098255 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 M24 compound treatment 316240.0 123000.0 8.37 299920.0 108000.0 8.02 11.5919 0.9998 2144937 PK04_098256 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N01 compound treatment 249520.0 56100.0 3.82 230480.0 38300.0 2.85 4.721 0.9895 2144901 PK04_098257 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N02 compound treatment 217320.0 23900.0 1.63 211960.0 19800.0 1.47 2.194 0.9987 3413999 PK04_098258 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Br)cc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N03 compound treatment 283240.0 89800.0 6.12 263120.0 71000.0 5.28 8.0644 0.9973 2143297 PK04_098259 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N04 compound treatment 233000.0 39600.0 2.7 225440.0 33300.0 2.48 3.6594 0.9991 3414005 PK04_098260 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(C#N)cc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N05 compound treatment 302680.0 109000.0 7.45 255000.0 62800.0 4.68 8.5742 0.9748 2142017 PK04_098261 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N06 compound treatment 210840.0 17400.0 1.19 212760.0 20600.0 1.53 1.9237 0.9921 3188747 PK04_098262 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)CCc3ccccc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N07 compound treatment 257520.0 64100.0 4.37 246400.0 54200.0 4.04 5.9445 0.9992 2143017 PK04_098263 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N08 compound treatment 228800.0 35400.0 2.41 214680.0 22500.0 1.68 2.8906 0.9842 3188748 PK04_098264 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)c3ccc(Br)cc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N09 mock treatment 198600.0 5180.0 0.35 195880.0 3710.0 0.28 0.4453 0.9926 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N10 mock treatment 200960.0 7540.0 0.51 203320.0 11200.0 0.83 0.9506 0.9735 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N11 compound treatment 237760.0 44300.0 3.02 233480.0 41300.0 3.07 4.312 1.0 2144265 PK04_098265 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N12 compound treatment 230480.0 37100.0 2.53 225080.0 32900.0 2.45 3.5189 0.9999 3069249 PK04_098266 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)c3c(OC)cccc3OC)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N13 mock treatment 200360.0 6940.0 0.47 197200.0 5030.0 0.37 0.5996 0.9933 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N14 mock treatment 197720.0 4300.0 0.29 195880.0 3710.0 0.28 0.4029 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N15 compound treatment 284160.0 90700.0 6.19 261360.0 69200.0 5.15 8.0161 0.9958 2143165 PK04_098267 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N16 compound treatment 229240.0 35800.0 2.44 219640.0 27500.0 2.04 3.1729 0.9961 3188751 PK04_098268 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccccc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N17 compound treatment 255880.0 62500.0 4.26 240320.0 48200.0 3.58 5.5455 0.9963 2144365 PK04_098269 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N18 compound treatment 191880.0 -1540.0 -0.1 195600.0 3430.0 0.26 0.1066 0.3859 3188752 PK04_098270 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3cccc(F)c3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N19 compound treatment 249520.0 56100.0 3.82 239040.0 46900.0 3.49 5.1715 0.9989 2142105 PK04_098271 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N20 compound treatment 246240.0 52800.0 3.6 234120.0 42000.0 3.12 4.7544 0.9975 3068687 PK04_098272 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccc(OC)cc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N21 compound treatment 248920.0 55500.0 3.78 249480.0 57300.0 4.27 5.692 0.9982 2144245 PK04_098273 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N22 compound treatment 231640.0 38200.0 2.61 220520.0 28400.0 2.11 3.3349 0.9945 3068689 PK04_098274 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N23 compound treatment 236720.0 43300.0 2.95 222880.0 30700.0 2.29 3.704 0.992 2143153 PK04_098275 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 N24 compound treatment 184440.0 -8980.0 -0.61 182000.0 -10200.0 -0.76 -0.9678 -0.9945 3188876 PK04_098276 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccc(Br)cc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O01 compound treatment 252760.0 59300.0 4.05 239280.0 47100.0 3.51 5.3403 0.9975 2143373 PK04_098277 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O02 compound treatment 299640.0 106000.0 7.24 298040.0 106000.0 7.88 10.6927 0.9991 2142209 PK04_098278 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O03 compound treatment 186920.0 -6500.0 -0.44 185240.0 -6930.0 -0.52 -0.6777 -0.9972 2144345 PK04_098279 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O04 compound treatment 274760.0 81300.0 5.55 257960.0 65800.0 4.9 7.384 0.9981 2142673 PK04_098280 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O05 compound treatment 264880.0 71500.0 4.87 249880.0 57700.0 4.3 6.4825 0.998 2143977 PK04_098281 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O06 compound treatment 275760.0 82300.0 5.61 274000.0 81800.0 6.09 8.2764 0.9992 2142077 PK04_098282 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O07 compound treatment 292640.0 99200.0 6.76 300720.0 109000.0 8.08 10.4963 0.9961 2141985 PK04_098283 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O08 compound treatment 323240.0 130000.0 8.85 300000.0 108000.0 8.03 11.9336 0.9988 2143485 PK04_098284 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O09 compound treatment 271200.0 77800.0 5.3 260040.0 67900.0 5.05 7.3218 0.9997 2144665 PK04_098285 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O10 compound treatment 311360.0 118000.0 8.04 295640.0 103000.0 7.7 11.1314 0.9998 2143273 PK04_098286 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O11 mock treatment 195120.0 1700.0 0.12 191440.0 -725.0 -0.05 0.0439 0.3429 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O12 mock treatment 210720.0 17300.0 1.18 199680.0 7510.0 0.56 1.2296 0.9419 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O13 compound treatment 231440.0 38000.0 2.59 231480.0 39300.0 2.93 3.902 0.9982 2144773 PK04_098287 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O14 compound treatment 267840.0 74400.0 5.07 253720.0 61600.0 4.58 6.8273 0.9987 2143945 PK04_098288 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O15 compound treatment 245080.0 51700.0 3.52 242720.0 50600.0 3.76 5.1511 0.9995 2144317 PK04_098289 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O16 compound treatment 253800.0 60400.0 4.12 260840.0 68700.0 5.11 6.5251 0.9942 2143905 PK04_098290 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O17 compound treatment 299400.0 106000.0 7.23 284400.0 92200.0 6.86 9.9633 0.9997 2143917 PK04_098291 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O18 compound treatment 196120.0 2700.0 0.18 192440.0 275.0 0.02 0.1447 0.7808 2144253 PK04_098292 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O19 compound treatment 268440.0 75000.0 5.11 257720.0 65600.0 4.88 7.0667 0.9997 2144105 PK04_098293 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8=CCCCC8)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O20 compound treatment 253760.0 60300.0 4.11 245920.0 53800.0 4.0 5.738 0.9999 2144293 PK04_098294 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O21 compound treatment 254880.0 61500.0 4.19 243680.0 51500.0 3.83 5.6741 0.999 2142997 PK04_098295 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O22 compound treatment 244640.0 51200.0 3.49 222000.0 29800.0 2.22 4.0395 0.9761 2144737 PK04_098296 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O23 compound treatment 186320.0 -7100.0 -0.48 186200.0 -5970.0 -0.44 -0.6561 -0.9991 2141452 PK04_098297 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 O24 compound treatment 494360.0 301000.0 20.52 480000.0 288000.0 21.42 29.656 0.9998 2142677 PK04_098298 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCCO)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P01 compound treatment 256120.0 62700.0 4.27 252840.0 60700.0 4.52 6.2159 0.9996 2144005 PK04_098299 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P02 compound treatment 203960.0 10500.0 0.72 203760.0 11600.0 0.86 1.1184 0.9959 3068772 PK04_098300 CCOC(=O)[C@H]1C/C=C/C[C@H](C(=O)OCC)C(=O)O[C@H]2[C@H](OC(=O)Nc3ccc(C#N)cc3)[C@@H](CO)O[C@H](OC)[C@@H]2OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P03 compound treatment 232880.0 39500.0 2.69 224280.0 32100.0 2.39 3.5925 0.9983 2142593 PK04_098301 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P04 compound treatment 205160.0 11700.0 0.8 198520.0 6350.0 0.47 0.9005 0.9685 3000699 PK04_098302 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P05 compound treatment 275920.0 82500.0 5.62 247960.0 55800.0 4.15 6.9136 0.9889 2144921 PK04_098303 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P06 compound treatment 213960.0 20500.0 1.4 210840.0 18700.0 1.39 1.9731 1.0 3000700 PK04_098304 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P07 compound treatment 261760.0 68300.0 4.66 240560.0 48400.0 3.6 5.8416 0.9919 2143937 PK04_098305 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P08 compound treatment 167960.0 -25500.0 -1.74 166200.0 -26000.0 -1.93 -2.5938 -0.9986 3000701 PK04_098306 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P09 compound treatment 243080.0 49700.0 3.39 247040.0 54900.0 4.08 5.2821 0.9957 2144785 PK04_098307 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P10 compound treatment 190600.0 -2820.0 -0.19 190560.0 -1610.0 -0.12 -0.2203 -0.9739 3089322 PK04_098308 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P11 mock treatment 191720.0 -1700.0 -0.12 189160.0 -3010.0 -0.22 -0.24 -0.953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P12 mock treatment 187640.0 -5780.0 -0.39 186160.0 -6010.0 -0.45 -0.5946 -0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P13 compound treatment 237760.0 44300.0 3.02 228920.0 36800.0 2.74 4.072 0.9988 2144213 PK04_098309 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P14 compound treatment 233640.0 40200.0 2.74 241320.0 49200.0 3.66 4.5259 0.9899 3089323 PK04_098310 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P15 compound treatment 245720.0 52300.0 3.57 248160.0 56000.0 4.17 5.4683 0.997 2144225 PK04_098311 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P16 compound treatment 211000.0 17600.0 1.2 220680.0 28500.0 2.12 2.3483 0.9634 3000703 PK04_098312 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P17 compound treatment 276640.0 83200.0 5.67 264360.0 72200.0 5.37 7.8114 0.9996 2141953 PK04_098313 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P18 compound treatment 296960.0 104000.0 7.06 283960.0 91800.0 6.83 9.8225 0.9999 3000704 PK04_098314 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)c4cc5ccccc5[nH]4)[C@H]1OC(=O)c6cc7ccccc7[nH]6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P19 compound treatment 220600.0 27200.0 1.85 217080.0 24900.0 1.85 2.6216 1.0 2143337 PK04_098315 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P20 compound treatment 219440.0 26000.0 1.77 214080.0 21900.0 1.63 2.4078 0.9991 3089326 PK04_098316 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Br)cc2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P21 compound treatment 383120.0 190000.0 12.93 376320.0 184000.0 13.71 18.8369 0.9996 2143233 PK04_098317 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P22 compound treatment 210760.0 17300.0 1.18 206600.0 14400.0 1.07 1.5957 0.9989 3089328 PK04_098318 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(C#N)cc2)[C@H](OC(=O)c3cc4ccccc4[nH]3)[C@H]1OC(=O)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P23 compound treatment 229560.0 36100.0 2.46 222640.0 30500.0 2.27 3.3462 0.9991 2142969 PK04_098319 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2098 P24 compound treatment 196800.0 3380.0 0.23 191000.0 -1170.0 -0.09 0.1017 0.4129 3189006 PK04_098320 CC(C)[Si](OCCCNS(=O)(=O)c1ccc(Br)cc1)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A01 mock treatment 175360.0 -5530.0 -0.38 172480.0 -9240.0 -0.69 -0.7529 -0.9599 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A02 mock treatment 172320.0 -8570.0 -0.58 171040.0 -10700.0 -0.79 -0.9752 -0.9885 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A03 compound treatment 168280.0 -12600.0 -0.86 175960.0 -5760.0 -0.43 -0.911 -0.9484 3076292 SMP2_000001 C[C@H](CCCC(C)(C)O)C1CCC2C3CC=C4CC(O)CCC4(C)C3CCC12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A04 compound treatment 176440.0 -4450.0 -0.3 174440.0 -7280.0 -0.54 -0.5976 -0.9624 170 SMP2_000002 CCCCCCCC[C@@H](O)/C=C/C=C/C=C\[C@@H](O)CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A05 compound treatment 174640.0 -6250.0 -0.43 171280.0 -10400.0 -0.78 -0.8507 -0.96 3076293 SMP2_000003 CN(C)CC/C=C/1\c2ccccc2CC(O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A06 compound treatment 203320.0 22400.0 1.53 196680.0 15000.0 1.11 1.8686 0.9878 2153 SMP2_000004 C[C@@H]1[C@@H](OC(=O)/C=C/C=C/c2ccccc2)[C@@]3(OC4(O[C@@H]3[C@@H]5[C@@H]6O[C@]6(CO)[C@@H](O)[C@@]7(O)[C@@H](C=C(C)C7=O)[C@@]15O4)c8ccccc8)C(=C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A07 compound treatment 172080.0 -8810.0 -0.6 173920.0 -7800.0 -0.58 -0.8352 -0.9999 3471112 SMP2_000005 CCOC(=O)CCC(=O)OC1C(CC(C)OC1OC2C(C)C(OC3CC(C)(OC)C(O)C(C)O3)C(C)C(=O)OC(CC)C(C)(O)C(O)C(C)C(=O)C(C)CC2(C)O)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A08 compound treatment 178960.0 -1930.0 -0.13 177320.0 -4400.0 -0.33 -0.3246 -0.9196 2199 SMP2_000006 CC(C(C)c1ccc(O)cn1)C(N)C(=O)NC([C@H]2O[C@H]([C@@H](O)[C@H]2O)N3C=CC(=O)CC3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A09 compound treatment 175600.0 -5290.0 -0.36 172720.0 -9000.0 -0.67 -0.7287 -0.9578 698 SMP2_000007 NC[C@H]1O[C@H](O[C@@H]2[C@@H](N)C[C@@H](N)[C@H](O[C@H]3O[C@H](CO)[C@@H](O)[C@H](N)[C@H]3O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A10 compound treatment 190560.0 9670.0 0.66 188280.0 6560.0 0.49 0.8114 0.9891 3199281 SMP2_000008 CC(=C[C@@H](O)C1=C[C@@H](O)[C@@H]2O[C@@H]2C1=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A11 compound treatment 176240.0 -4650.0 -0.32 180560.0 -1160.0 -0.09 -0.2852 -0.8682 1001979 SMP2_000009 NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A12 compound treatment 176080.0 -4810.0 -0.33 173120.0 -8600.0 -0.64 -0.6845 -0.9517 3199282 SMP2_000010 C[C@@H]1[C@@H](OC(=O)C)[C@]2(OC(=O)C)[C@H]([C@@H]3C=C(CO)C[C@]4(O)[C@@H](C=C(C)C4=O)[C@]13O)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A13 compound treatment 172960.0 -7930.0 -0.54 176640.0 -5080.0 -0.38 -0.6496 -0.9847 1497 SMP2_000011 NC[C@H]1O[C@H](O[C@@H]2[C@@H](N)C[C@@H](N)[C@H](O)C2O[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)[C@H](N)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A14 compound treatment 173600.0 -7290.0 -0.5 179080.0 -2640.0 -0.2 -0.4904 -0.9176 1000212 SMP2_000012 C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@@H]3[C@@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A15 compound treatment 210320.0 29400.0 2.01 211960.0 30200.0 2.25 3.0102 0.9984 3199283 SMP2_000013 COC1/C=C\OC2(C)Oc3c(C2=O)c4c(O)cc(NC(=O)\C(=C/C=C\C(C)C(O)C(C)C(O)C(C)C(OC(=O)C)C1C)\C)c(O)c4c(O)c3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A16 compound treatment 232240.0 51400.0 3.5 244120.0 62400.0 4.64 5.7595 0.9903 2267 SMP2_000014 CO[C@H]1[C@H](O)C(O)[C@@H](OC1CO)n2c3c(Cl)cccc3c4c5C(=O)NC(=O)c5c6c7cccc(Cl)c7[nH]c6c24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A17 compound treatment 178920.0 -1970.0 -0.13 174520.0 -7200.0 -0.54 -0.4739 -0.8577 706 SMP2_000015 Nc1ccc(cc1)S(=O)(=O)Nc2cnc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A18 compound treatment 183480.0 2590.0 0.18 177760.0 -3960.0 -0.29 -0.0835 -0.243 1098997 SMP2_000016 CCC1(O)C(=O)OCc2c1cc3-c4nc5ccccc5cc4Cn3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A19 compound treatment 236080.0 55200.0 3.76 237040.0 55300.0 4.12 5.572 0.999 1001956 SMP2_000017 CC(C)C1N(C)c2cccc3[nH]cc(CC(CO)NC1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A20 compound treatment 177360.0 -3530.0 -0.24 179720.0 -2000.0 -0.15 -0.2754 -0.9734 1912779 SMP2_000018 CC(NC(=O)c1ccccc1/N=C/c2c(O)ccc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A21 compound treatment 173880.0 -7010.0 -0.48 176560.0 -5160.0 -0.38 -0.6095 -0.9941 230 SMP2_000019 CCCCCC(=O)/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C\C=C/CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A22 compound treatment 170280.0 -10600.0 -0.72 171440.0 -10300.0 -0.77 -1.0525 -0.9996 464 SMP2_000020 CN(Cc1cnc2nc(N)nc(N)c2n1)c3ccc(cc3)C(=O)N[C@@H](CCC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A23 compound treatment 239920.0 59000.0 4.02 235400.0 53700.0 4.0 5.6708 1.0 548 SMP2_000021 N[C@H]1C[C@H]([C@H](O)[C@@H]1O)n2cc(I)c3c(N)ncnc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 A24 compound treatment 195040.0 14200.0 0.96 197280.0 15600.0 1.16 1.501 0.9959 3199284 SMP2_000022 C/C(=C/CNc1ncnc2[nH]cnc12)/CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B01 mock treatment 168120.0 -12800.0 -0.87 164800.0 -16900.0 -1.26 -1.5061 -0.9837 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B02 mock treatment 168280.0 -12600.0 -0.86 169920.0 -11800.0 -0.88 -1.2289 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B03 compound treatment 172280.0 -8610.0 -0.59 169120.0 -12600.0 -0.94 -1.0782 -0.9745 1001866 SMP2_000023 NC(CCCNC(=N)N)C(=O)CC(Cc1ccccc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B04 compound treatment 176960.0 -3930.0 -0.27 173160.0 -8560.0 -0.64 -0.6399 -0.9259 3076299 SMP2_000024 C[C@@H]1CCOC(=O)/C=C\C=C/C(=O)O[C@@H]2C[C@@H]3OC4C=C(C)CCC4(COC(=O)[C@H]1O)[C@]2(C)[C@@]53CO5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B05 compound treatment 169720.0 -11200.0 -0.76 172280.0 -9440.0 -0.7 -1.0353 -0.9992 3199377 SMP2_000025 CO[C@@H]1C[C@H](C)O[C@@H](CC[C@H](C)[C@H](O)[C@H](C)[C@H]2OC(=O)/C(=C/C[C@H](O)C[C@H]3O[C@@H](CC=C3)C[C@H](OC)[C@@H](C)[C@@H](O)C[C@@H](O)[C@H](C)[C@H](OC(=O)/C(=C/C[C@H](O)C[C@H]4O[C@@H](CC=C4)C[C@H](OC)[C@@H](C)[C@@H](O)C[C@@H](O)[C@@H]2C)/C)[C@@H](C)[C@@H](O)[C@@H](C)CC[C@@H]5C[C@@H](C[C@H](C)O5)OC)/C)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B06 compound treatment 173080.0 -7810.0 -0.53 171160.0 -10600.0 -0.79 -0.9322 -0.982 3076300 SMP2_000026 CC1(C)C(O)C2(C)CCC1C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B07 compound treatment 171560.0 -9330.0 -0.64 173640.0 -8080.0 -0.6 -0.875 -0.9996 3199378 SMP2_000027 CC(CO)C1CC(O)C2(C)OC3CC4OC5CC6(C)OC7CCC8OC9CC%10(C)OC%11C(CC%10OC9CC(C)C8OC7CC6OC5(C)CC=CC4OC3CC2O1)OC(=O)C=C%11C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B08 compound treatment 176600.0 -4290.0 -0.29 173240.0 -8480.0 -0.63 -0.6531 -0.9388 3076301 SMP2_000028 Cn1cc(C[C@@H](N)C(=O)O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B09 compound treatment 229040.0 48200.0 3.28 215040.0 33300.0 2.48 4.0748 0.9904 28 SMP2_000029 CNc1ccc2oc(C[C@@H]3OC4(CC[C@@H]3C)O[C@H](C(C)C(=O)c5ccc[nH]5)[C@H](C)C[C@H]4C)nc2c1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B10 compound treatment 141600.0 -39300.0 -2.68 137600.0 -44100.0 -3.28 -4.216 -0.9949 3199379 SMP2_000030 CC(C)CC(CO)NC(=O)C(CCC(=O)N)NC(=O)C(C)(C)NC(=O)C(CC(C)C)NC(=O)C(CCC(=O)N)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)C(CCC(=O)N)NC(=O)C(C)(C)NC(=O)C(CC(C)C)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)C(C)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B11 compound treatment 172200.0 -8690.0 -0.59 175320.0 -6400.0 -0.48 -0.7557 -0.9942 2006 SMP2_000031 O[C@H]1C2OC2[C@H](O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B12 compound treatment 254960.0 74100.0 5.05 247920.0 66200.0 4.93 7.0548 0.9999 3076303 SMP2_000032 CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B13 compound treatment 478400.0 298000.0 20.28 485280.0 304000.0 22.59 30.3182 0.9986 3076304 SMP2_000033 CCN(CC)CCNC(=O)c1c(C)[nH]c(/C=C/2\C(=O)Nc3ccc(Cl)cc23)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B14 compound treatment 170000.0 -10900.0 -0.74 171480.0 -10200.0 -0.76 -1.0639 -0.9999 1000114 SMP2_000034 CCN(CC)CCCC(C)Nc1ccnc2cc(Cl)ccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B15 compound treatment 176000.0 -4890.0 -0.33 175840.0 -5880.0 -0.44 -0.5452 -0.9909 277 SMP2_000035 OC[C@H]1O[C@H]([C@H](O)[C@H]1O)n2cnc3cc(Cl)c(Cl)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B16 compound treatment 177640.0 -3250.0 -0.22 175200.0 -6520.0 -0.49 -0.4998 -0.9368 3076306 SMP2_000036 CC(=O)c1ccc(cc1O)N2CCOCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B17 compound treatment 209160.0 28300.0 1.93 205120.0 23400.0 1.74 2.5943 0.9987 2095622 SMP2_000037 CC(=CCC/C(=C/CC/C(=C/Cc1c(O)c2ccccc2oc1=O)/C)/C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B18 compound treatment 172280.0 -8610.0 -0.59 170800.0 -10900.0 -0.81 -0.9898 -0.9872 1670 SMP2_000038 Nc1nc2n(COC(CO)CO)cnc2c(=O)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B19 compound treatment 186800.0 5910.0 0.4 179480.0 -2240.0 -0.17 0.167 0.3829 2090 SMP2_000039 CCOC(=O)C(C#N)C1C(=C(N)Oc2ccc(Br)cc12)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B20 compound treatment 187600.0 6710.0 0.46 187480.0 5760.0 0.43 0.6266 0.9995 1096696 SMP2_000040 Oc1ccc(cc1CC=C)c2cc(CC=C)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B21 compound treatment 291280.0 110000.0 7.53 332160.0 150000.0 11.2 13.239 0.9813 3199380 SMP2_000041 NC1=NC(=O)/C(=C\2/CCNC(=O)c3[nH]c(Br)cc23)/N1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B22 compound treatment 169120.0 -11800.0 -0.8 167240.0 -14500.0 -1.08 -1.3295 -0.9894 2137 SMP2_000042 Oc1cc(O)c2c(=O)cc(oc2c1)c3ccc(O)c(O)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B23 compound treatment 166920.0 -14000.0 -0.95 167560.0 -14200.0 -1.05 -1.4187 -0.9987 3104545 SMP2_000043 CC1CC(C)/C=C(/C)\CC(C)C(=O)NC(C)C(=O)N(C)C(Cc2c(Br)[nH]c3ccccc23)C(=O)NC(CC(=O)O1)c4ccc(O)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 B24 compound treatment 144320.0 -36600.0 -2.49 142000.0 -39700.0 -2.96 -3.8533 -0.9964 907437 SMP2_000044 CCCCCCCCCCCCC(=O)N1CCCCC1CNC(=O)[C@@H](N)CCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C01 mock treatment 173280.0 -7610.0 -0.52 175360.0 -6360.0 -0.47 -0.7016 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C02 mock treatment 174160.0 -6730.0 -0.46 178360.0 -3360.0 -0.25 -0.5013 -0.9593 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C03 compound treatment 231400.0 50500.0 3.44 232480.0 50800.0 3.78 5.1064 0.9989 907417 SMP2_000045 COc1cc2[C@H]3CC[C@]4(C)[C@@H](O)CC[C@H]4[C@@H]3CCc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C04 compound treatment 181280.0 392.0 0.03 174840.0 -6880.0 -0.51 -0.3433 -0.6693 180 SMP2_000046 CCCCC/C=C\C/C=C\C=C\C=C\[C@@H](SCC(N)C(=O)NCC(=O)O)[C@@H](O)CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C05 compound treatment 173640.0 -7250.0 -0.49 179760.0 -1960.0 -0.15 -0.4527 -0.8784 3199382 SMP2_000047 C[C@@H]1CCC2[C@H](C[C@]3(C)C(=CCC4[C@]5(C)C[C@@H](O)[C@H](O)[C@@](C)(CO)C5CC[C@]43C)C2[C@H]1C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C06 compound treatment 229560.0 48700.0 3.32 230000.0 48300.0 3.59 4.8872 0.9992 3104900 SMP2_000048 C/C(=C\CCC1C=CC(OC1O)C2=CC(=O)OC2O)/CCC3=C(C)CCCC3(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C07 compound treatment 231600.0 50700.0 3.46 223520.0 41800.0 3.11 4.6445 0.9986 907313 SMP2_000049 Oc1c(I)cc2c(Oc3c(I)c(O)c(I)cc3C42OC(=O)c5ccccc54)c1I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C08 compound treatment 185160.0 4270.0 0.29 180200.0 -1520.0 -0.11 0.1259 0.4028 3076308 SMP2_000050 CCCCCCCCCCCCCCCCCCCCCCCC(=O)N[C@@H](CO)[C@H](O)CCCCCCCCCCCCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C09 compound treatment 185600.0 4710.0 0.32 182160.0 439.0 0.03 0.2502 0.775 1002910 SMP2_000051 OC(C(O)C(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C10 compound treatment 178720.0 -2170.0 -0.15 179800.0 -1920.0 -0.14 -0.2056 -0.9999 453 SMP2_000052 COc1cccc(c1N)c2cc(=O)c3ccccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C11 compound treatment 178480.0 -2410.0 -0.16 181640.0 -81.2 -0.01 -0.1204 -0.7326 3199383 SMP2_000053 C[C@@H]1C[C@H]2[C@@H](CC[C@@H]3C[C@@H](O)CC[C@@]32C)[C@]45O[C@@H]5C[C@@H](C14)c6ccc(=O)oc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C12 compound treatment 179880.0 -1010.0 -0.07 181880.0 159.0 0.01 -0.0403 -0.5771 3199384 SMP2_000054 CC[C@H]1OC(=O)C[C@@H](O)C[C@@H](OC[C@]2(C)OC(C)[C@@H](O[C@@]3(C)C[C@@](C)(O)[C@@H](O)C(C)O3)[C@H](C2O)N(C)C)[C@@H](CC=O)C[C@@H](C)C(=O)/C=C\C(=C/C1CO[C@@H]4OC(C)[C@@H](O)[C@H](OC)C4OC)\C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C13 compound treatment 184680.0 3790.0 0.26 183840.0 2120.0 0.16 0.2943 0.9719 3076309 SMP2_000055 C[C@]12CC[C@H](C3CCC(C)(C)OC3)[C@@]2(C)[C@H](O)C[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5[C@@H](O)C[C@]41C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C14 compound treatment 173240.0 -7650.0 -0.52 180280.0 -1440.0 -0.11 -0.4446 -0.8351 222 SMP2_000056 CCCCC[C@H](O)/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C15 compound treatment 203200.0 22300.0 1.52 213040.0 31300.0 2.33 2.7238 0.9786 3076310 SMP2_000057 CC1(C)CC[C@H](F)[C@@]2(CO[C@@]3(O)[C@H](O)[C@H]12)[C@@H]4CC[C@@H]5[C@@H](O)[C@@]43C(=O)C5=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C16 compound treatment 214160.0 33300.0 2.27 215520.0 33800.0 2.52 3.3827 0.9987 3199385 SMP2_000058 OC[C@@H]1C[C@H](N[C@@H]2C=C(CO)[C@@H](O)[C@H](O)[C@H]2O)C(O)C(O)[C@@H]1O[C@@H]3OC(CO)[C@@H](O)[C@H](O)[C@@H]3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C17 compound treatment 198240.0 17400.0 1.18 195200.0 13500.0 1.0 1.5458 0.9966 1448 SMP2_000059 OC(=O)c1cc(N=Nc2ccc(cc2)S(=O)(=O)Nc3ccccn3)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C18 compound treatment 186920.0 6030.0 0.41 181240.0 -481.0 -0.04 0.2654 0.6431 31 SMP2_000060 CCCCCCCCCCCCCCC[C@H](O)[C@@H](N)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C19 compound treatment 178480.0 -2410.0 -0.16 175000.0 -6720.0 -0.5 -0.4698 -0.8924 95 SMP2_000061 CCCCCC(O)/C=C/C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C20 compound treatment 227400.0 46500.0 3.17 227000.0 45300.0 3.37 4.6252 0.9995 2065223 SMP2_000062 CN(C)c1ccc(cc1)C(O)(c2ccccc2)c3ccc(cc3)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C21 compound treatment 177280.0 -3610.0 -0.25 187520.0 5800.0 0.43 0.1312 0.2641 3199386 SMP2_000063 CO[C@H]1C[C@H](C)CC2=C(NCC=C)C(=O)C=C(NC(=O)/C(=C\C=C/[C@H](O)[C@@H](OC(=O)N)/C(=C\[C@H](C)[C@H]1O)/C)/C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C22 compound treatment 180800.0 -88.5 -0.01 179000.0 -2720.0 -0.2 -0.1475 -0.7278 2041 SMP2_000064 OC(=O)CNC(=O)C(CS)Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C23 compound treatment 170480.0 -10400.0 -0.71 165920.0 -15800.0 -1.18 -1.3334 -0.9707 3076311 SMP2_000065 COc1cc2ccnc3cc[nH]c(c1OC)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 C24 compound treatment 169800.0 -11100.0 -0.76 170520.0 -11200.0 -0.83 -1.1241 -0.9988 907566 SMP2_000066 C/C(=C\CNc1ncnc2n(cnc12)C3OC(CO)[C@@H](O)[C@H]3O)/CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D01 mock treatment 170520.0 -10400.0 -0.71 171040.0 -10700.0 -0.79 -1.062 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D02 mock treatment 175560.0 -5330.0 -0.36 173040.0 -8680.0 -0.65 -0.7138 -0.9629 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D03 compound treatment 172800.0 -8090.0 -0.55 177000.0 -4720.0 -0.35 -0.6384 -0.9763 3199387 SMP2_000067 CCC1/C=C(/C)\CC(C)CC(OC)C2OC(O)(C(C)CC2OC)C(=O)C(=O)N3CCCCC3C(=O)OC(C(C)C(O)CC1=O)/C(=C/C4CCC(O)C(C4)OC)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D04 compound treatment 180360.0 -528.0 -0.04 180560.0 -1160.0 -0.09 -0.0866 -0.9248 907555 SMP2_000068 CC1=C[C@H]2O[C@@H]3C[C@@H](O)C(C)(C43CO4)[C@@]2(CO)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D05 compound treatment 183600.0 2710.0 0.18 187400.0 5680.0 0.42 0.4296 0.9312 1962 SMP2_000069 CN(CC[C@H](N)CC(=O)N[C@H]1C=C[C@H](O[C@@H]1C(=O)O)n2ccc(N)nc2=O)C(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D06 compound treatment 183280.0 2390.0 0.16 187200.0 5480.0 0.41 0.4036 0.9191 852250 SMP2_000070 C1CCC(NC1)c2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D07 compound treatment 213640.0 32800.0 2.23 221080.0 39400.0 2.93 3.6503 0.991 3076314 SMP2_000071 O[C@@H]1C=CC(Br)[C@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D08 compound treatment 187840.0 6950.0 0.47 190440.0 8720.0 0.65 0.794 0.9881 3076315 SMP2_000072 OC[C@H]1O[C@H](C[C@@H]1O)n2cc(I)c(O)nc2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D09 compound treatment 198960.0 18100.0 1.23 199600.0 17900.0 1.33 1.8121 0.9993 3199389 SMP2_000073 CCCCCCCc1c(C)c(O)cc2c3ccccc3[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D10 compound treatment 188360.0 7470.0 0.51 186960.0 5240.0 0.39 0.6359 0.9913 3199390 SMP2_000074 COc1ccc(cc1)C(O)(C2CC2)c3cncnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D11 compound treatment 218040.0 37200.0 2.53 221440.0 39700.0 2.96 3.8813 0.997 832324 SMP2_000075 COc1cc(OC)c2c(=O)c(C)c(CC[C@@H](C)[C@@H](C)[C@@H](C)[C@@H](C)/C=C/C=C/C(=C/C)/C)oc2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D12 compound treatment 254280.0 73400.0 5.0 249680.0 68000.0 5.06 7.1146 1.0 2085117 SMP2_000076 COc1ccc(OC)c2c(=S)c3ccccc3[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D13 compound treatment 185920.0 5030.0 0.34 181840.0 119.0 0.01 0.2488 0.7251 251 SMP2_000077 Nc1ncnc2n(cnc12)C3(CO)OC(=C)C(O)C3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D14 compound treatment 199800.0 18900.0 1.29 202760.0 21000.0 1.57 2.0189 0.9953 2007 SMP2_000078 CO[C@@H]1[C@@H](OC(=O)c2ccc(C)[nH]2)[C@@H](O)[C@H](CC1(C)C)Oc3ccc4CC(NC(=O)c5[nH]cc(CC(=O)Nc6cc7ccc(O[C@@H]8OC(C)(C)[C@H](OC)[C@@H](OC(=O)c9ccc(C)[nH]9)[C@H]8O)c(C)c7oc6=O)c5C)C(=O)Oc4c3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D15 compound treatment 178000.0 -2890.0 -0.2 177720.0 -4000.0 -0.3 -0.3498 -0.9798 751 SMP2_000079 COc1cc(NS(=O)(=O)c2ccc(N)cc2)nc(OC)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D16 compound treatment 232560.0 51700.0 3.52 232000.0 50300.0 3.74 5.1371 0.9995 3076316 SMP2_000080 Oc1cc(ccc1C(=O)c2ccccc2)N3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D17 compound treatment 175280.0 -5610.0 -0.38 171480.0 -10200.0 -0.76 -0.8093 -0.9491 3076317 SMP2_000081 CO[C@@H]1C[C@@H](CC[C@H]1O)/C=C(\C)/[C@H]2OC(=O)[C@@H]3CCCCN3C(=O)C(=O)[C@]4(O)O[C@H](C[C@H](C[C@@H](C)C\C(=C/[C@@H](CC=C)C(=O)C[C@H](O)[C@H]2C)\C)OC)[C@H](C[C@H]4C)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D18 compound treatment 182480.0 1590.0 0.11 181880.0 159.0 0.01 0.0851 0.7795 1392 SMP2_000082 CNC(C)[C@@H]1CC[C@@H](N)[C@@H](O[C@@H]2[C@@H](N)C[C@@H](N)[C@H](O[C@@H]3OC[C@](C)(O)[C@H](NC)[C@H]3O)[C@H]2O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D19 compound treatment 193880.0 13000.0 0.89 200400.0 18700.0 1.39 1.6093 0.9763 610 SMP2_000083 O=S(=O)(N1CCCNCC1)c2cccc3cnccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D20 compound treatment 211440.0 30600.0 2.08 210640.0 28900.0 2.15 2.9948 0.9999 3076318 SMP2_000084 Oc1nccc2c(cccc12)S(=O)(=O)N3CCCNCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D21 compound treatment 209120.0 28200.0 1.92 156560.0 -25200.0 -1.87 0.0368 0.0137 616 SMP2_000085 COc1cc(O)c2c(=O)c(OC)c3CC(C)C(C(=O)C)c4c(OC)c(=O)c5c(O)cc(OC)c6c1c2c3c4c56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D22 compound treatment 194240.0 13400.0 0.91 199720.0 18000.0 1.34 1.5909 0.9823 1096695 SMP2_000086 Oc1ccc(CC=C)cc1c2cc(CC=C)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D23 compound treatment 173080.0 -7810.0 -0.53 170280.0 -11400.0 -0.85 -0.9786 -0.9744 3176136 SMP2_000087 C[C@@H]1C2NCC(C)C[C@H]2O[C@@]31CCC4C5CC=C6CC(O)CCC6(C)C5C(=O)C4=C3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 D24 compound treatment 214920.0 34000.0 2.32 202600.0 20900.0 1.55 2.7394 0.981 3076319 SMP2_000088 Nc1nc(OCC2CCCCC2)c3[nH]cnc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E01 mock treatment 181640.0 752.0 0.05 180800.0 -921.0 -0.07 -0.0123 -0.1431 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E02 mock treatment 178640.0 -2250.0 -0.15 186120.0 4400.0 0.33 0.1231 0.3405 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E03 compound treatment 189760.0 8870.0 0.6 192400.0 10700.0 0.79 0.9897 0.9909 445 SMP2_000089 NC(=O)c1cccc(N)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E04 compound treatment 335120.0 154000.0 10.52 317800.0 136000.0 10.13 14.5968 0.9998 1057045 SMP2_000090 COC(=O)c1ccc(O)c2nc3c(C=O)c(O)cc(O)c3nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E05 compound treatment 538400.0 358000.0 24.37 528080.0 346000.0 25.78 35.4631 0.9996 1949 SMP2_000091 NOC(=O)C1=CC(=C(c2ccc(O)c(c2)C(=O)ON)c3ccc(O)c(c3)C(=O)ON)C=CC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E06 compound treatment 233800.0 52900.0 3.61 240840.0 59100.0 4.4 5.6621 0.9951 2180 SMP2_000092 COc1ccc(CNc2nc(NCc3ccc(OC)cc3)c4ncn(C(C)C)c4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E07 compound treatment 397240.0 216000.0 14.75 454120.0 272000.0 20.27 24.7657 0.9878 1020463 SMP2_000093 Oc1cc2ccc(=O)oc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E08 compound treatment 193280.0 12400.0 0.84 188320.0 6600.0 0.49 0.9447 0.9667 3076699 SMP2_000094 CN1CCC[C@H]1CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E09 compound treatment 215280.0 34400.0 2.34 209400.0 27700.0 2.06 3.1146 0.9979 1694 SMP2_000095 Oc1ccc(cc1)c2sc3cc(O)ccc3c2C(=O)c4ccc(OCCN5CCCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E10 compound treatment 195360.0 14500.0 0.99 203360.0 21600.0 1.61 1.8364 0.9723 2345 SMP2_000096 Nc1ncnc2n(ccc12)[C@@H]3O[C@H](CO)[C@H](O)[C@H]3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E11 compound treatment 194280.0 13400.0 0.91 185920.0 4200.0 0.31 0.8666 0.898 3199487 SMP2_000097 C[C@@H]1CC[C@@]2(C[C@H](C)C3C(=CCC4[C@@]3(C)C[C@@H](O)C5[C@](C)(CO)[C@@H](O)[C@H](O)C[C@]45C)C2[C@H]1C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E12 compound treatment 198920.0 18000.0 1.23 191880.0 10200.0 0.76 1.4039 0.9727 2240 SMP2_000098 CC(C)C[C@H](NP(=O)(O)OC1OC(C)C(O)C(O)C1O)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E13 compound treatment 197120.0 16200.0 1.11 194200.0 12500.0 0.93 1.4392 0.9962 1000145 SMP2_000099 NC[C@@H]1O[C@H](O[C@H]2[C@@H](O)[C@@H](O[C@@H]3[C@@H](O)[C@H](N)C[C@H](N)[C@H]3OC4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4N)O[C@@H]2CO)[C@H](N)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E14 compound treatment 213000.0 32100.0 2.19 210680.0 29000.0 2.16 3.0721 1.0 267 SMP2_000100 CCCCC[C@H](O)/C=C/[C@@H]1[C@@H](C/C=C\CCCC(=O)O)C=CC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E15 compound treatment 259280.0 78400.0 5.34 262840.0 81100.0 6.04 8.0482 0.9982 1114632 SMP2_000101 CC1OC(OCC2OC(Oc3c(oc4cc(O)cc(O)c4c3=O)c5ccc(O)c(O)c5)C(O)C(O)C2O)C(O)C(O)C1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E16 compound treatment 189640.0 8750.0 0.6 199280.0 17600.0 1.31 1.346 0.9369 1000121 SMP2_000102 C/C(=C\CO)/C=C/C=C(\C)/C=C/C1=C(C)CCCC1(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E17 compound treatment 205080.0 24200.0 1.65 208200.0 26500.0 1.97 2.5598 0.9961 1599897 SMP2_000103 O=c1n2CCc3c([nH]c4ccccc34)-c2nc5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E18 compound treatment 183040.0 2150.0 0.15 189440.0 7720.0 0.57 0.5099 0.8601 2354 SMP2_000104 COc1ccc2C3C4[C@H](CC(C)(C)OO[C@H](C=C(C)C)N4c2c1)N5C(=O)[C@@H]6CCCN6C(=O)[C@]5(O)[C@H]3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E19 compound treatment 185640.0 4750.0 0.32 185000.0 3280.0 0.24 0.4016 0.9902 1001870 SMP2_000105 C/C(=C/C(=O)O)/C=C/[C@@]1(O)C(=CC(=O)CC1(C)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E20 compound treatment 218160.0 37300.0 2.54 214200.0 32500.0 2.42 3.5061 0.9997 296 SMP2_000106 Nc1ncnc2N(=CNc21)C3CCCO3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E21 compound treatment 471240.0 290000.0 19.8 475920.0 294000.0 21.9 29.4804 0.9987 600 SMP2_000107 COC(=O)/C=C/c1cc(O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E22 compound treatment 293280.0 112000.0 7.66 263040.0 81300.0 6.05 9.6978 0.9932 2327 SMP2_000108 CCC(C)C1NC2C=Cc3c(cc(nc3C2O)C(=O)OC(C)C(NCC(=O)c4csc(n4)C(NC(=O)c5csc(n5)/C(=C\C)/NC(=O)C(NC(=O)c6csc(n6)C7(CCC(=NC7)c8nc(cs8)C(=O)NC(=C)C(=O)NC(=C)C(=O)N)NC(=C)C(C)NC(=O)C(=C)NCC(C)NC1=O)C(C)O)C(C)(O)C(C)O)c9nccs9)C(C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E23 compound treatment 141520.0 -39400.0 -2.68 146480.0 -35200.0 -2.62 -3.7526 -0.9999 3076759 SMP2_000109 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](COP(=O)(O)OCC[N+](C)(C)C)NC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 E24 compound treatment 194160.0 13300.0 0.9 192160.0 10400.0 0.78 1.1892 0.9971 3199491 SMP2_000110 C/C=C/C1OC2=C(C(=O)C[C@H](C)O2)C(=O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F01 mock treatment 177240.0 -3650.0 -0.25 177200.0 -4520.0 -0.34 -0.4138 -0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F02 mock treatment 176800.0 -4090.0 -0.28 180880.0 -841.0 -0.06 -0.2414 -0.8449 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F03 compound treatment 182160.0 1270.0 0.09 190920.0 9200.0 0.68 0.5454 0.7903 907179 SMP2_000111 C/C(=C\C=C\C=C(/C)\C=C\C=C(/C)\C=C\C1=C(C)C(=O)C(O)CC1(C)C)/C=C/C=C(\C)/C=C/C2=C(C)C(=O)C(O)CC2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F04 compound treatment 523080.0 342000.0 23.33 533480.0 352000.0 26.18 35.0088 0.9983 3076760 SMP2_000112 COc1cc(O)c2c3oc4cc(O)c(O)cc4c3c(=O)oc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F05 compound treatment 192000.0 11100.0 0.76 196000.0 14300.0 1.06 1.2871 0.9862 328 SMP2_000113 C/C=C(/C)\C=C\1/CN=C2N(CCC2(O)C1=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F06 compound treatment 192280.0 11400.0 0.78 192400.0 10700.0 0.79 1.1112 0.9999 3076761 SMP2_000114 CNCC/C=C/1\c2ccccc2CC(O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F07 compound treatment 193600.0 12700.0 0.87 193640.0 11900.0 0.89 1.2401 0.9999 3199493 SMP2_000115 CCC/C=C/C=C/C(=O)O[C@H]1\C(=C\C(=O)OC)\C[C@H]2C[C@@H](OC(=O)C[C@H](O)C[C@H]3C[C@H](OC(=O)C)C(C)(C)[C@](O)(C[C@@H]4C/C(=C/C(=O)OC)/C[C@@H](O4)/C=C\C(C)(C)[C@]1(O)O2)O3)[C@@H](C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F08 compound treatment 203440.0 22600.0 1.54 197200.0 15500.0 1.15 1.9018 0.9899 1046629 SMP2_000116 Nc1cc2c3ccccc3ccc2c4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F09 compound treatment 190200.0 9310.0 0.63 187920.0 6200.0 0.46 0.7751 0.9877 1037664 SMP2_000117 CSCS(=O)CC(CO)NC(=O)C=Cc1c(C)nc(O)nc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F10 compound treatment 192040.0 11200.0 0.76 194240.0 12500.0 0.93 1.1964 0.9949 1943 SMP2_000118 CN[C@H]1[C@@H](O)[C@H]2O[C@H](O[C@@H]3[C@@H](N)C[C@@H](N)[C@H](O)[C@H]3O)[C@H](N)C[C@@H]2O[C@@H]1O[C@@]4(C)O[C@H](CO)[C@@H](N)[C@H](O)[C@H]4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F11 compound treatment 190320.0 9430.0 0.64 190440.0 8720.0 0.65 0.9135 1.0 3199494 SMP2_000119 CC[C@@H]1C[C@@]1(NC(=O)C2=C[C@H](CC)C[C@H]3[C@@H]2CCC3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F12 compound treatment 402240.0 221000.0 15.09 397520.0 216000.0 16.06 22.028 0.9995 1320 SMP2_000120 C[C@]1(CC[C@]2(C)CC[C@]3(C)C4=CC=C5C=C(O)C(=O)C=C5[C@]4(C)CC[C@@]3(C)[C@@H]2C1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F13 compound treatment 217720.0 36800.0 2.51 212680.0 31000.0 2.3 3.4049 0.9991 745 SMP2_000121 CC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F14 compound treatment 265880.0 85000.0 5.79 274880.0 93200.0 6.93 9.0 0.996 2008 SMP2_000122 CC1=C(SCCO)C(=O)c2ccccc2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F15 compound treatment 188440.0 7550.0 0.51 190400.0 8680.0 0.65 0.8208 0.9937 3199495 SMP2_000123 CCCCCCCCCCCCCC[C@@H](O)[C@@H](O)[C@@H](N)COP(=O)(O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F16 compound treatment 192360.0 11500.0 0.78 187600.0 5880.0 0.44 0.8624 0.9623 3076763 SMP2_000124 Oc1ccc2c(Oc3cc(O)ccc3C42OC(=O)c5ccc(Nc6nc(Cl)nc(Cl)n6)cc54)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F17 compound treatment 190600.0 9710.0 0.66 193160.0 11400.0 0.85 1.0702 0.9923 1433 SMP2_000125 CS(=O)(=O)c1ccc(cc1)[C@@H](O)[C@@H](CO)NC(=O)C(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F18 compound treatment 184360.0 3470.0 0.24 186640.0 4920.0 0.37 0.4262 0.9777 1100216 SMP2_000126 CC(=CCCC(C)(OC1OC(COC2OC(CO)C(O)C2O)C(O)C(O)C1O)C3CCC4(C)C3C(O)CC5C6(C)CCC(OC7OC(CO)C(O)C(O)C7OC8OC(CO)C(O)C(O)C8O)C(C)(C)C6CCC54C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F19 compound treatment 184520.0 3630.0 0.25 191080.0 9360.0 0.7 0.6676 0.9031 3000453 SMP2_000127 C[C@@H]1CC2OC(=O)C(=C)C2[C@H](O)[C@@]3(C)[C@H]1C=CC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F20 compound treatment 230720.0 49800.0 3.4 228720.0 47000.0 3.5 4.8757 0.9999 3060680 SMP2_000128 Oc1ccccc1N2CC=C(NC2=O)c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F21 compound treatment 187840.0 6950.0 0.47 191720.0 10000.0 0.74 0.8613 0.9763 1907753 SMP2_000129 CC[C@@H]1[C@H](C)C[C@@H]2[C@H]3C[C@H]4CCC(=O)C5=C(O)[C@H](CCCNC(=O)/C=C\C[C@@H]4[C@H]3C=C[C@@H]12)NC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F22 compound treatment 279200.0 98300.0 6.7 267800.0 86100.0 6.41 9.2696 0.9997 1001972 SMP2_000130 CCCC[C@@H](C)/C=C(\C)/C=C(\C)/C(=O)NC1=C[C@@](O)(\C=C\C=C\C=C\C(=O)NC2=C(O)CCC2=O)[C@@H]3O[C@@H]3C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F23 compound treatment 177000.0 -3890.0 -0.27 174600.0 -7120.0 -0.53 -0.5622 -0.9487 3076765 SMP2_000131 CO[C@H]1[C@@H](CC(=O)O[C@H](C)C/C=C\C=C/[C@H](O)[C@H](C)C[C@H](CC=O)[C@@H]1O[C@@H]2O[C@H](C)[C@@H](O[C@H]3C[C@@](C)(O)[C@@H](OC(=O)CC(C)C)[C@H](C)O3)[C@@H]([C@H]2O)N(C)C)OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 F24 compound treatment 179040.0 -1850.0 -0.13 183200.0 1480.0 0.11 -0.0113 -0.0675 288 SMP2_000132 C[C@@H]1Cc2c(Cl)cc(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)c(O)c2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G01 mock treatment 184120.0 3230.0 0.22 189280.0 7560.0 0.56 0.5536 0.9163 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G02 mock treatment 186480.0 5590.0 0.38 189440.0 7720.0 0.57 0.6758 0.9802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G03 compound treatment 193520.0 12600.0 0.86 194880.0 13200.0 0.98 1.3015 0.9979 2407 SMP2_000133 CN1C(=C(O)c2ccccc2S1(=O)=O)C(=O)Nc3ncc(C)s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G04 compound treatment 251640.0 70800.0 4.82 243560.0 61800.0 4.6 6.6653 0.9997 907364 SMP2_000134 CCC(C(=O)NC/C=C\C=C(\C)/C(OC)C(C)C1OC(\C=C/C=C\C=C(\C)/C(=O)c2c(O)cc[nH]c2=O)C(O)C1O)C3(O)OC(\C=C/C=C\C)C(C)(C)C(O)C3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G05 compound treatment 265920.0 85000.0 5.8 268920.0 87200.0 6.49 8.6883 0.9984 1978 SMP2_000135 OC(=O)/C=C/c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G06 compound treatment 195160.0 14300.0 0.97 194120.0 12400.0 0.92 1.3405 0.9996 3076766 SMP2_000136 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CO)[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G07 compound treatment 194240.0 13400.0 0.91 191920.0 10200.0 0.76 1.1804 0.9959 1117 SMP2_000137 Nc1nc(=O)c2nc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)O)C(=O)O)cnc2[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G08 compound treatment 192640.0 11800.0 0.8 191200.0 9480.0 0.71 1.0654 0.998 313 SMP2_000138 CCCCCCCCCCCCCCC[C@@H](O)[C@H](CO)NC(=O)CCCCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G09 compound treatment 191800.0 10900.0 0.74 193040.0 11300.0 0.84 1.1217 0.9981 3076819 SMP2_000139 COCC(=O)c1ncn-2c1[C@@H]3CCNC3C(=O)c4cc(OC)ccc42 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G10 compound treatment 210280.0 29400.0 2.0 216840.0 35100.0 2.61 3.2651 0.9914 3199591 SMP2_000140 CCCCCCCCCC(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H]3C=C(C)C(=O)[C@]3(O)CC(=C[C@H]2[C@@H]4C(C)(C)[C@@]41OC(=O)CCCCCCCCC)COC(=O)Cc5ccc(O)c(OC)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G11 compound treatment 200200.0 19300.0 1.32 198440.0 16700.0 1.24 1.8108 0.9996 939 SMP2_000141 Cc1cccc(Nc2ccccc2C(=O)O)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G12 compound treatment 219480.0 38600.0 2.63 213440.0 31700.0 2.36 3.5297 0.9985 3076821 SMP2_000142 CCCCCCCCCCCCCC[C@@H](O)[C@@H](O)[C@@H](N)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G13 compound treatment 192040.0 11200.0 0.76 191400.0 9680.0 0.72 1.047 0.9996 1012954 SMP2_000143 OC(Cc1ccncc1)C(Cl)(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G14 compound treatment 209000.0 28100.0 1.92 216760.0 35000.0 2.61 3.1992 0.9885 4637 SMP2_000144 C[C@@H]1C[C@]2(OC(=O)C)[C@H]([C@@H]3C=C(CO)C[C@@]4(O)[C@@H](C=C(C)C4=O)[C@@]13O)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G15 compound treatment 195600.0 14700.0 1.0 195600.0 13900.0 1.03 1.4396 0.9999 942 SMP2_000145 OC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G16 compound treatment 195760.0 14900.0 1.01 187120.0 5400.0 0.4 1.0011 0.9179 3199592 SMP2_000146 CCCC[C@]1(CC[C@]2(CC[C@H](C)[C@@H](C/C=C(\C)/C=C/[C@H](O)[C@@H](C)/C=C/C(=O)O)O2)O[C@H]1\C=C\C(=C\C(=O)O)\C)OC(=O)CCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G17 compound treatment 233040.0 52200.0 3.56 206200.0 24500.0 1.82 3.8024 0.9518 1011013 SMP2_000147 Nc1ccc2nc3ccc(N)cc3[s+]c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G18 compound treatment 223200.0 42300.0 2.88 219320.0 37600.0 2.8 4.0185 0.9999 3076824 SMP2_000148 NC(=O)OCC1N=C(N)N2CCC(O)(O)C32NC(=NC13)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G19 compound treatment 274240.0 93400.0 6.36 280120.0 98400.0 7.32 9.6788 0.9976 3199593 SMP2_000149 COc1cc(ccc1O)[C@H]2Oc3cc(ccc3O[C@H]2CO)[C@H]4Oc5cc(O)cc(O)c5C(=O)[C@@H]4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G20 compound treatment 190080.0 9190.0 0.63 191960.0 10200.0 0.76 0.982 0.9953 3185114 SMP2_000150 CC[C@]1(C=CCN2CC[C@]3([C@H]4N(C)c5cc(OC)ccc53)[C@@H]21)[C@@H](OC(=O)C)[C@]4(O)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G21 compound treatment 188800.0 7910.0 0.54 183400.0 1680.0 0.12 0.4698 0.8484 3199594 SMP2_000151 C[C@@H]1[C@@H](O)[C@]2(O)[C@H]([C@@H]3C=C(CO)C[C@@]4(O)[C@@H](C=C(C)C4=O)[C@@]13O)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G22 compound treatment 183240.0 2350.0 0.16 188800.0 7080.0 0.53 0.4859 0.8823 3076825 SMP2_000152 NC(=O)C1CCCN1C(=O)C(Cc2c[nH]cn2)NC(=O)C3CCC(=O)N3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G23 compound treatment 223880.0 43000.0 2.93 229200.0 47500.0 3.53 4.5713 0.9957 1095351 SMP2_000153 COC1=C(Br)C(O)C(O)(CC#N)C=C1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 G24 compound treatment 238760.0 57900.0 3.95 234560.0 52800.0 3.93 5.5707 1.0 3 SMP2_000154 Oc1ccc(/C=C(\C#N)/C(=O)NCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H01 mock treatment 182240.0 1350.0 0.09 182080.0 359.0 0.03 0.084 0.876 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H02 mock treatment 182320.0 1430.0 0.1 184400.0 2680.0 0.2 0.21 0.946 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H03 compound treatment 186760.0 5870.0 0.4 183200.0 1480.0 0.11 0.3609 0.8693 3199595 SMP2_000155 CCC(C)C(NC(=O)C1CC(=O)NCC(=O)NC(Cc2ccccc2)C(=O)NC(C(C)CC)C(=O)NCC(=O)NC(Cc3c[nH]c4ccccc34)C(=O)NCC(=O)NC(CC(=O)N)C(=O)N1)C(=O)NC(Cc5ccccc5)C(=O)NCC(=O)NC(Cc6c[nH]cn6)C(=O)NC(Cc7ccc(O)cc7)C(=O)NC(CO)C(=O)NCC(=O)NC(CC(=O)O)C(=O)NC(Cc8ccccc8)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H04 compound treatment 189240.0 8350.0 0.57 187920.0 6200.0 0.46 0.7288 0.9946 1303231 SMP2_000156 CN(C)CC(O)Cn1c2ccc(Br)cc2c3cc(Br)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H05 compound treatment 198280.0 17400.0 1.19 191840.0 10100.0 0.75 1.3709 0.976 3076826 SMP2_000157 Nc1ccccc1NC(=O)CCCCCCC(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H06 compound treatment 190080.0 9190.0 0.63 193280.0 11600.0 0.86 1.0514 0.9879 3076827 SMP2_000158 OC[C@H]1CC2CCN1CC2C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H07 compound treatment 271360.0 90500.0 6.17 255880.0 74200.0 5.52 8.2643 0.9985 3199596 SMP2_000159 OC(=O)c1cc(/C=C/c2ccc(/C=C/c3ccc(O)c(c3)C(=O)O)c(Br)c2)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H08 compound treatment 204880.0 24000.0 1.64 206480.0 24800.0 1.84 2.4596 0.9982 1088673 SMP2_000160 CC(C)C1NC(=O)C(NC(=O)c2cc(N)c(C)c3oc4c(C)c(=O)c(N)c(C(=O)NC5C(C)OC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C6CCCN6C(=O)C(NC5=O)C(C)C)c4nc23)C(C)OC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C7CCCN7C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H09 compound treatment 198520.0 17600.0 1.2 187920.0 6200.0 0.46 1.1762 0.9135 3069011 SMP2_000161 NCCC(=O)NCCc1c[nH]cn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H10 compound treatment 197440.0 16600.0 1.13 200400.0 18700.0 1.39 1.7809 0.9946 1025 SMP2_000162 CC(C)CC(=O)OC1C(O[C@@H]2C[C@H]([C@H]3CC[C@]4(C[C@@H]5CC[C@H]4[C@]3(C)C2)[C@@H](O)C5=C)C(=O)O)OC(CO)C(OS(=O)(=O)O)C1OS(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H11 compound treatment 236960.0 56100.0 3.82 244560.0 62800.0 4.68 6.0102 0.995 1018447 SMP2_000163 Oc1ccc2c(c1)oc3c2c(=O)oc4cc(O)ccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H12 compound treatment 206520.0 25600.0 1.75 204800.0 23100.0 1.72 2.4502 1.0 1000068 SMP2_000164 CC1=C(N2[C@H](SC1)C(NC(=O)C(N)c3ccccc3)C2=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H13 compound treatment 191560.0 10700.0 0.73 181440.0 -281.0 -0.02 0.4997 0.6865 526 SMP2_000165 C[C@@H](O)[C@@H]1O[C@H]1/C=C/[C@@H]2O[C@H]2[C@H](O)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H14 compound treatment 204680.0 23800.0 1.62 196080.0 14400.0 1.07 1.9026 0.9795 460 SMP2_000166 CCC1NC(=O)C([C@H](O)[C@H](C)C/C=C/C)N(C)C(=O)C(C(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)C(C)NC(=O)C(CC(C)C)N(C)C(=O)C(NC(=O)C(CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H15 compound treatment 194160.0 13300.0 0.9 197240.0 15500.0 1.16 1.4565 0.9927 907301 SMP2_000167 CCC(C)C(O)C(C)C(=O)C(C)/C=C(\C)/CC(C)C1OC(=O)C1CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H16 compound treatment 190360.0 9470.0 0.65 189880.0 8160.0 0.61 0.886 0.9995 3076266 SMP2_000168 CO[C@@H]1[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H17 compound treatment 197240.0 16400.0 1.11 195000.0 13300.0 0.99 1.4871 0.9982 1001938 SMP2_000169 COC[C@H]1CC[C@H]2[C@@H](C)[C@@H](O)[C@H](OC3OC(COC(C)(C)C=C)[C@H](O)C(OC(=O)C)[C@@H]3O)C4=C(CC(O)[C@]4(C)C=C12)C(C)COC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H18 compound treatment 425440.0 245000.0 16.67 421000.0 239000.0 17.81 24.3821 0.9995 829 SMP2_000170 CC(C)c1c(O)c(O)c(C=O)c2c(O)c(c(C)cc12)c3c(C)cc4c(C(C)C)c(O)c(O)c(C=O)c4c3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H19 compound treatment 194160.0 13300.0 0.9 193840.0 12100.0 0.9 1.2776 1.0 2334 SMP2_000171 C/C(=C\1/C(=O)NC(Cc2ccccc2)C1=O)/Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H20 compound treatment 196440.0 15600.0 1.06 194800.0 13100.0 0.97 1.438 0.9991 2109 SMP2_000172 OCc1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H21 compound treatment 186120.0 5230.0 0.36 180560.0 -1160.0 -0.09 0.1911 0.5207 2106 SMP2_000173 COC1=CC(=O)C(=C(C[C@]2(C)[C@@H](C)CC[C@@]3(C)[C@H]2CCCC3=C)C1=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H22 compound treatment 219440.0 38600.0 2.63 216800.0 35100.0 2.61 3.7046 1.0 1260 SMP2_000174 N[C@@H](Cc1ccc(cc1)N(CCCl)CCCl)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H23 compound treatment 212280.0 31400.0 2.14 205640.0 23900.0 1.78 2.7721 0.9958 3076270 SMP2_000175 C[C@]12C=Cc3occc3C2CC[C@]4(C[C@H]5CCC41)C[C@]5(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 H24 compound treatment 183960.0 3070.0 0.21 186080.0 4360.0 0.32 0.3775 0.9776 3199601 SMP2_000176 CCC(C)C1NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(N)CSSCC(NC(=O)C(CC(=O)N)NC(=O)C(CCC(=O)N)NC1=O)C(=O)N3CCCC3C(=O)NC(CC(C)C)C(=O)NCC(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I01 mock treatment 185800.0 4910.0 0.33 186120.0 4400.0 0.33 0.4683 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I02 mock treatment 185480.0 4590.0 0.31 184160.0 2440.0 0.18 0.3497 0.9664 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I03 compound treatment 191120.0 10200.0 0.7 198040.0 16300.0 1.21 1.3521 0.9653 3076271 SMP2_000177 OC(=O)/C=C/c1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I04 compound treatment 247120.0 66200.0 4.52 246280.0 64600.0 4.8 6.5905 0.9995 3199602 SMP2_000178 C/C(=C\CCC1=CC(=O)OC1O)/CC/C=C(\C)/CCC2=C(C)CCCC2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I05 compound treatment 194040.0 13200.0 0.9 192920.0 11200.0 0.83 1.2234 0.9993 1135 SMP2_000179 OCCNCCNc1ccc(NCCNCCO)c2C(=O)c3c(O)ccc(O)c3C(=O)c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I06 compound treatment 207640.0 26800.0 1.82 202200.0 20500.0 1.52 2.3674 0.996 252 SMP2_000180 CCCCCCOC(=O)[C@]1(O)C[C@H]2O[C@@]1(C)n3c4ccccc4c5c6CNC(=O)c6c7c8ccccc8n2c7c35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I07 compound treatment 200560.0 19700.0 1.34 205840.0 24100.0 1.8 2.2176 0.9897 3076272 SMP2_000181 COC(=O)C1=CO[C@@H](O[C@@H]2OC(CO)[C@H](O)[C@@H](O)[C@H]2O)[C@H]3[C@@H]1CC=C3CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I08 compound treatment 192960.0 12100.0 0.82 195440.0 13700.0 1.02 1.3039 0.9943 3199603 SMP2_000182 CCCCCCCCCCCCCCC[C@@H](O)[C@H](CO)NC(=O)CCCCCCCCCCCCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I09 compound treatment 220720.0 39800.0 2.72 221000.0 39300.0 2.92 3.9874 0.9993 2129 SMP2_000183 OCC(O)C1OC(=O)C(=C1O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I10 compound treatment 222560.0 41700.0 2.84 218560.0 36800.0 2.74 3.9477 0.9998 3199692 SMP2_000184 CCCCCCCCC(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H]3C=C(C)C(=O)[C@]3(O)CC(=C[C@H]2[C@@H]4C(C)(C)[C@@]41OC(=O)CCCCCCCC)COC(=O)Cc5ccc(O)c(OC)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I11 compound treatment 226840.0 46000.0 3.13 215480.0 33800.0 2.51 3.9919 0.994 1865 SMP2_000185 Clc1cccc(Nc2nnc(c3ccccc3)c4ccccc24)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I12 mock treatment 200200.0 19300.0 1.32 192360.0 10600.0 0.79 1.4909 0.9704 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I13 compound treatment 196200.0 15300.0 1.04 195920.0 14200.0 1.06 1.4854 1.0 3472730 SMP2_000186 CC12CCC3C(CC=C4CC(O)CCC34C)C2CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I14 compound treatment 203040.0 22200.0 1.51 202080.0 20400.0 1.52 2.1393 1.0 3076274 SMP2_000187 Oc1ccc(cc1)C2COc3cc(O)ccc3C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I15 compound treatment 230480.0 49600.0 3.38 242360.0 60600.0 4.51 5.582 0.9899 2288 SMP2_000188 CC(=CCC(O)C1=CC(=O)c2c(O)ccc(O)c2C1=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I16 compound treatment 189160.0 8270.0 0.56 193840.0 12100.0 0.9 1.0365 0.9744 3199693 SMP2_000189 COC(C(C)C1CC(O)C2(C)OC2/C=C\C(C)C3CC(CC(=O)O3)CC4OC4C(=O)O1)C(=CC=CC(=Cc5coc(C)n5)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I17 compound treatment 191120.0 10200.0 0.7 191440.0 9720.0 0.72 1.0047 0.9998 1025605 SMP2_000190 OCCN(CCO)CCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I18 compound treatment 213960.0 33100.0 2.25 219280.0 37600.0 2.8 3.571 0.9943 3060146 SMP2_000191 Oc1ccc(cc1)c2nc(c([nH]2)c3ccc(F)cc3)c4ccncc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I19 compound treatment 211440.0 30600.0 2.08 206080.0 24400.0 1.81 2.7548 0.9976 1874 SMP2_000192 Oc1cccc2c(O)nccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I20 compound treatment 197880.0 17000.0 1.16 198920.0 17200.0 1.28 1.7243 0.9988 1080610 SMP2_000193 COc1ccc(O)c2c(=O)c3c(OC)cc4OC5OC=CC5c4c3oc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I21 compound treatment 191000.0 10100.0 0.69 186320.0 4600.0 0.34 0.7295 0.9478 2290 SMP2_000194 C[C@]1(CC(N)CCC(N)C(=O)O)O[C@](C)([C@@H](O)[C@H]1O)n2cnc3c(N)ncnc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I22 compound treatment 214520.0 33600.0 2.29 217200.0 35500.0 2.64 3.4885 0.9975 3076167 SMP2_000195 CC(C)C1OC(=O)C2=CCCN2C(=O)c3coc(CC(=O)C[C@H](O)/C=C(/C)\C=C/CNC(=O)\C=C/C1C)n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I23 compound treatment 249960.0 69100.0 4.71 239920.0 58200.0 4.33 6.3927 0.9991 1077786 SMP2_000196 CC(C)CC1N2C(=O)C(NC(=O)C3CN(C)C4Cc5c[nH]c6cccc(C4=C3)c56)(OC2(O)C7CCCN7C1=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 I24 compound treatment 261840.0 81000.0 5.52 264080.0 82400.0 6.13 8.2369 0.9986 325 SMP2_000197 N/C(=C(/C#N)\C(=C(/N)\Sc1ccccc1N)\C#N)/Sc2ccccc2N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J01 mock treatment 179840.0 -1050.0 -0.07 181960.0 239.0 0.02 -0.038 -0.5156 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J02 mock treatment 182120.0 1230.0 0.08 185040.0 3320.0 0.25 0.234 0.8971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J03 compound treatment 187800.0 6910.0 0.47 184640.0 2920.0 0.22 0.4868 0.9382 3076170 SMP2_000198 OC[C@@H]1[C@@H](O)[C@H](O)[C@H]2[C@@H](O)CCN12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J04 compound treatment 204080.0 23200.0 1.58 195480.0 13800.0 1.02 1.8421 0.9779 677 SMP2_000199 C[C@@H](N)[C@H]1CC[C@@H](CC1)C(=O)Nc2ccncc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J05 compound treatment 188440.0 7550.0 0.51 192080.0 10400.0 0.77 0.9092 0.9807 2060246 SMP2_000200 C[C@@]1(CO)[C@H](O)CC[C@@]2(C)[C@H](C/C=C/3\[C@H](O)COC3=O)C(=C)CCC12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J06 compound treatment 207120.0 26200.0 1.79 200960.0 19200.0 1.43 2.2771 0.9939 414 SMP2_000201 CC1CNCCN1S(=O)(=O)c2cccc3cnccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J07 compound treatment 200160.0 19300.0 1.31 192720.0 11000.0 0.82 1.5079 0.9741 1972 SMP2_000202 COC(=O)/C(=C\Nc1ccc(Oc2ccccc2OC(C)C)nc1)/NC(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J08 compound treatment 221120.0 40200.0 2.74 214320.0 32600.0 2.43 3.6551 0.9981 3189311 SMP2_000203 CC(=O)OCC1=C(N2[C@H](SC1)[C@H](N)C2=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J09 compound treatment 367680.0 187000.0 12.73 362440.0 181000.0 13.45 18.5157 0.9996 2109607 SMP2_000204 CC(C)c1cc2CC[C@H]3C(C)(C)CCC[C@]3(C(=O)O)c2c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J10 compound treatment 203920.0 23000.0 1.57 206520.0 24800.0 1.85 2.4154 0.9968 1960 SMP2_000205 CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J11 compound treatment 196120.0 15200.0 1.04 195440.0 13700.0 1.02 1.4563 1.0 3199694 SMP2_000206 CC1[C@H]2NC[C@@H](C)C[C@H]2O[C@@]31CC[C@H]4[C@@H]5CC=C6C[C@@H](O)CC[C@]6(C)[C@H]5CC4=C3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J12 compound treatment 173720.0 -7170.0 -0.49 179720.0 -2000.0 -0.15 -0.4509 -0.8825 874122 SMP2_000207 COc1c(O)c2c(=O)cc3OCOc4cc(O)c5c(=O)c(OC)c(CC(C)O)c6c(c1CC(C)O)c2c3c4c56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J13 compound treatment 222360.0 41500.0 2.83 223560.0 41800.0 3.11 4.2012 0.9988 1301 SMP2_000208 OCCN(CCO)c1nc(N2CCCCC2)c3nc(nc(N4CCCCC4)c3n1)N(CCO)CCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J14 compound treatment 193680.0 12800.0 0.87 195560.0 13800.0 1.03 1.345 0.9966 1001900 SMP2_000209 Nc1ccn(C2OC(CO)C(O)C2O)c(=O)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J15 compound treatment 207400.0 26500.0 1.81 211360.0 29600.0 2.21 2.8379 0.9951 2056 SMP2_000210 CC(C)CC(NC(=O)NC(C1CCNC(=N1)N)C(=O)NC(CCC(=O)N)C(=O)NC(C)C=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J16 compound treatment 196160.0 15300.0 1.04 195960.0 14200.0 1.06 1.4856 1.0 599 SMP2_000211 Cc1cc(O)c2C(=O)c3c(O)cc(O)cc3C(=O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J17 compound treatment 202880.0 22000.0 1.5 196880.0 15200.0 1.13 1.8579 0.9902 162 SMP2_000212 CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(C)C)CC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J18 compound treatment 195240.0 14400.0 0.98 197200.0 15500.0 1.15 1.5065 0.9967 3076285 SMP2_000213 CN1C(=O)/C(=C/2\Nc3ccccc3\C2=N\O)/c4ccc(Br)cc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J19 compound treatment 191320.0 10400.0 0.71 190200.0 8480.0 0.63 0.9491 0.9982 3199695 SMP2_000214 CC1O[C@@H](O[C@H]2C[C@@H](C=O)C3C(CCC4C3CC[C@]5(C)[C@H](CC[C@]45O)c6ccc(=O)oc6)[C@H]2O)[C@H](O)[C@@H](O)[C@H]1O[C@@H]7OC(CO)[C@@H](O)[C@@H](O)[C@H]7O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J20 compound treatment 185520.0 4630.0 0.32 183600.0 1880.0 0.14 0.3222 0.9329 3076287 SMP2_000215 COc1cc(O)c(CC=C(C)C)c2OC(CC(=O)c12)c3ccc(O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J21 compound treatment 184000.0 3110.0 0.21 177880.0 -3840.0 -0.29 -0.0522 -0.1465 2411 SMP2_000216 NCC1O[C@@H](O[C@@H]2[C@H](N)C[C@@H](N)C(O[C@H]3OC(CO)[C@@H](O)[C@@H](N)[C@H]3O)C2O)[C@H](N)C[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J22 compound treatment 180360.0 -528.0 -0.04 181480.0 -241.0 -0.02 -0.0382 -0.9482 3199697 SMP2_000217 CCC(=O)O[C@H]1C(C)O[C@](C)(C[C@]1(C)O)O[C@@H]2C(C)O[C@@H](CO[C@@H]3[C@@H](C)[C@@H](CC(=O)O[C@H](C)C/C=C\C=C/[C@H](O)[C@H](C)C[C@@H]3CC(=O)C)OC(=O)CC)[C@H](O)[C@@H]2N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J23 compound treatment 284400.0 104000.0 7.06 273040.0 91300.0 6.8 9.796 0.9998 3076290 SMP2_000218 C[C@@H]1[C@H](O)[C@@H](C)[C@H]2O[C@@H]1CC[C@H](C)/C=C(/C)\C[C@@H](C)C[C@H](C)[C@]3(O)OC4=C(C)C(=O)C(=C2C4=C3)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 J24 compound treatment 175360.0 -5530.0 -0.38 177920.0 -3800.0 -0.28 -0.4666 -0.99 3199698 SMP2_000219 CC(NC(=O)C(NC(=O)c1nc(nc(N)c1C)C(CC(=O)N)NCC(N)C(=O)N)C(OC2OC(CO)C(O)C(O)C2(C)OC3OC(CO)C(O)C(O)(C3O)C(=O)N)c4cnc[nH]4)C(O)C(C)C(=O)NC(C(=O)C)C(=O)NCCC5=NC(CS5)c6nc(cs6)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K01 mock treatment 181440.0 552.0 0.04 184040.0 2320.0 0.17 0.1486 0.8414 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K02 mock treatment 185600.0 4710.0 0.32 186320.0 4600.0 0.34 0.4692 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K03 compound treatment 180320.0 -568.0 -0.04 185400.0 3680.0 0.27 0.1662 0.601 3076443 SMP2_000220 CC(C)CCC[C@@H](C)C1CCC2C3C(O)C=C4CC(O)CCC4(C)C3CCC12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K04 compound treatment 159880.0 -21000.0 -1.43 158040.0 -23700.0 -1.76 -2.2591 -0.9947 25 SMP2_000221 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@@H](N)COP(=O)(O)OCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K05 compound treatment 197800.0 16900.0 1.15 203240.0 21500.0 1.6 1.9478 0.987 3076448 SMP2_000222 CCC1=CC2C[C@@H]3c4[nH]c5ccccc5c4CCN(C2)[C@@]31C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K06 compound treatment 203640.0 22800.0 1.55 208560.0 26800.0 2.0 2.5093 0.9922 309 SMP2_000223 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CO)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K07 compound treatment 267280.0 86400.0 5.89 270240.0 88500.0 6.59 8.8233 0.9984 1000097 SMP2_000224 Cc1c(C)c2OC(C)(COc3ccc(CC4SC(=O)NC4=O)cc3)CCc2c(C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K08 compound treatment 269720.0 88800.0 6.06 262040.0 80300.0 5.98 8.5094 1.0 2113458 SMP2_000225 CCC(=O)NCCc1c2scnc2c3nccc4c5ccccc5[nH]c1c43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K09 compound treatment 356320.0 175000.0 11.96 353360.0 172000.0 12.77 17.4902 0.9995 3076491 SMP2_000226 CCCCCCCCCCCCCCCC(=O)OCC(O)[C@H]1OC(=O)C(=C1O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K10 compound treatment 201880.0 21000.0 1.43 199280.0 17600.0 1.31 1.936 0.999 3184 SMP2_000227 CCCCC[C@H](O)/C=C/[C@H]1[C@H](O)C[C@@H]2O/C(=C\CCCC(=O)O)/C[C@H]12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K11 compound treatment 197520.0 16600.0 1.13 201000.0 19300.0 1.43 1.8164 0.9932 1313 SMP2_000228 Oc1ccc(Cl)cc1C(=O)Nc2ccc(cc2Cl)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K12 compound treatment 232240.0 51400.0 3.5 229760.0 48000.0 3.58 5.0037 0.9999 3199699 SMP2_000229 CC(C)Nc1cccnc1N2CCN(CC2)C(=O)c3cc4cc(O)ccc4[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K13 compound treatment 202240.0 21400.0 1.46 198520.0 16800.0 1.25 1.9134 0.9971 2709 SMP2_000230 Cc1ncc(CO)c(CO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K14 compound treatment 217320.0 36400.0 2.48 219040.0 37300.0 2.78 3.7203 0.9984 3076498 SMP2_000231 CC1CC2OC2/C=C\C=C/C(=O)Cc3c(Cl)c(O)cc(O)c3C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K15 compound treatment 199440.0 18600.0 1.26 200960.0 19200.0 1.43 1.9068 0.9981 3076544 SMP2_000232 CCN(CC)CCCC(C)Nc1nc(C)cc(Nc2ccc3nc(C)cc(N)c3c2)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K16 compound treatment 235560.0 54700.0 3.73 235440.0 53700.0 4.0 5.4627 0.9994 633 SMP2_000233 OC(=O)c1cc(ccc1O)N(Cc2ccccc2O)Cc3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K17 compound treatment 176440.0 -4450.0 -0.3 175000.0 -6720.0 -0.5 -0.5682 -0.9712 3199700 SMP2_000234 CC1OC2OC3[C@@H](O)[C@@H](O)CO[C@H]3OC(=O)[C@@]45CCC(C)(C)C[C@H]5C6=CC[C@@H]7[C@@]8(C)C[C@H](O)[C@H](O[C@@H]9OC(CO)[C@@H](O)[C@H](O)C9O[C@@H]%10OC[C@@H](OC(=O)C[C@](C)(O)CC(=O)O[C@@H]1C(O[C@@H]%11OC[C@@H](O)[C@H](O)C%11O)[C@@H]2O)C(O)C%10O)[C@@](C)(CO)[C@@H]8CC[C@@]7(C)[C@]6(C)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K18 compound treatment 207160.0 26300.0 1.79 198640.0 16900.0 1.26 2.1569 0.9851 3076548 SMP2_000235 NC1N=CC(=N1)[C@H]2[C@H](CNC(=O)c3cc(Br)c[nH]3)[C@@H](CNC(=O)c4cc(Br)c[nH]4)[C@@H]2C5=NC(N)N=C5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K19 compound treatment 187120.0 6230.0 0.42 188320.0 6600.0 0.49 0.6477 0.9974 3076550 SMP2_000236 CCCCC[C@H](O)[C@H](SCC(N)C(=O)O)/C=C/C=C/C=C\C/C=C\CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K20 compound treatment 219600.0 38700.0 2.64 216080.0 34400.0 2.56 3.6744 0.9999 3199701 SMP2_000237 CO[C@@H]1C[C@H](C)O[C@@H](CC[C@H](C)[C@H](O)[C@H](C)[C@H]2OC(=O)/C=C\C(=C/C[C@@H](O)C[C@@H]3CCC[C@@H](C[C@H](OC)[C@@H](C)[C@@H](O)C[C@@H](O)[C@H](C)[C@H](OC(=O)/C=C\C(=C/C[C@@H](O)C[C@@H]4CCC[C@@H](CC(OC)[C@@H](C)[C@@H](O)C[C@@H](O)[C@@H]2C)O4)\C)[C@@H](C)[C@@H](O)[C@@H](C)CC[C@H]5C[C@@H](C[C@H](C)O5)OC)O3)\C)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K21 compound treatment 187080.0 6190.0 0.42 181560.0 -161.0 -0.01 0.29 0.6867 3076553 SMP2_000238 CC(C)CCC[C@@H](C)[C@H]1C[C@H](O)C2=C3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K22 compound treatment 233800.0 52900.0 3.61 233960.0 52200.0 3.89 5.3 0.9993 2329 SMP2_000239 C[C@@H]1C[C@@]2(OC3(Cc4ccccc4)O[C@@H]2[C@@H]5C=C(COC(=O)Cc6ccc(O)cc6)C[C@@]7(O)[C@@H](C=C(C)C7=O)[C@@]15O3)C(=C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K23 compound treatment 402760.0 222000.0 15.13 409600.0 228000.0 16.96 22.6888 0.9984 1000035 SMP2_000240 O=C1c2ccccc2-c3n[nH]c4cccc1c34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 K24 compound treatment 181160.0 272.0 0.02 179600.0 -2120.0 -0.16 -0.0985 -0.62 1100080 SMP2_000241 OCC1OC(C(O)C1O)n2cccnc2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L01 mock treatment 180800.0 -88.5 -0.01 181520.0 -201.0 -0.01 -0.0149 -0.9201 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L02 mock treatment 184480.0 3590.0 0.24 181360.0 -361.0 -0.03 0.1541 0.6257 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L03 compound treatment 230200.0 49300.0 3.36 222440.0 40700.0 3.03 4.5202 0.9987 155 SMP2_000242 CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC[C@@H](NC[C@@H](N)CS)C(C)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L04 compound treatment 222160.0 41300.0 2.81 220360.0 38600.0 2.88 4.0231 0.9999 410 SMP2_000243 CC(=N)NCc1cccc(CN)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L05 compound treatment 195200.0 14300.0 0.98 195200.0 13500.0 1.0 1.3993 0.9999 1000029 SMP2_000244 CSCCC(NC(=O)C(CC(C)C)NC(=O)C(Cc1c[nH]cn1)NC(=O)CNC(=O)C(NC(=O)C(C)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(CCC(=O)N)NC(=O)C(CC(=O)N)NC(=O)CNC(=O)C(CC(C)C)NC(=O)C(CCCNC(=N)N)NC(=O)C(CCC(=O)N)NC(=O)C4CCC(=O)N4)C(C)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L06 compound treatment 191720.0 10800.0 0.74 187080.0 5360.0 0.4 0.8042 0.9582 3199703 SMP2_000245 CCC1OC2(C[C@@H]3CC(C/C=C(/C)\C(O[C@@H]4C[C@@H](C)C(O[C@H]5C[C@H](OC)C(O)[C@H](C)O5)[C@H](C4)OC)C(C)\C=C/C=C\6/COC7C6[C@@H](C=C(C)[C@H]7O)C(=O)O3)O2)C=CC1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L07 compound treatment 196840.0 16000.0 1.09 197160.0 15400.0 1.15 1.5815 0.9996 3076615 SMP2_000246 COC1/C=C\C=C(\C)/Cc2cc(OC)c(Cl)c(c2)N(C)C(=O)CC(OC(=O)C(C)C)C3(C)OC3C(C)C4CC1(O)NC(=O)O4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L08 compound treatment 253280.0 72400.0 4.94 248200.0 66500.0 4.95 6.9885 1.0 3199793 SMP2_000247 CCN1C[C@]2(COC)CCC(OC)[C@]3(C4C[C@@]5(O)[C@H](OC(=O)c6ccc(OC)cc6)C4[C@](C[C@H]5OC)(OC(=O)C)[C@H]7[C@H](OC)C32)[C@@H]71 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L09 compound treatment 355440.0 175000.0 11.9 345280.0 164000.0 12.17 17.0226 0.9999 1983 SMP2_000248 CC(C)c1cc2C3CC4C(C)(C)CCCC4(C(=O)O3)c2c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L10 compound treatment 202040.0 21200.0 1.44 198360.0 16600.0 1.24 1.8953 0.9971 3199794 SMP2_000249 C[C@@H]1C[C@H]2[C@@H](CC[C@@H]3C[C@@H](O)CC[C@@]32C)[C@]45O[C@@H]5[C@H](OC(=O)C)[C@@H](C14)c6ccc(=O)oc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L11 compound treatment 196040.0 15200.0 1.03 198680.0 17000.0 1.26 1.6229 0.9951 3199795 SMP2_000250 CC1C2C(Cc3ccccc3)NC(=O)C24C(/C=C\CC(C)CC(C)(O)/C=C\C4O)C(O)C1=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L12 compound treatment 196120.0 15200.0 1.04 196120.0 14400.0 1.07 1.4921 0.9999 964 SMP2_000251 CN(C)N=Nc1[nH]cnc1C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L13 compound treatment 167480.0 -13400.0 -0.91 167160.0 -14600.0 -1.08 -1.4127 -0.9964 3076672 SMP2_000252 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@@H](N)CO[C@@H]1O[C@H](CO)[C@@H](O[C@@H]2O[C@H](CO)[C@H](O)C(O)C2O)C(O)C1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L14 compound treatment 198040.0 17200.0 1.17 195760.0 14000.0 1.04 1.5657 0.9984 1001931 SMP2_000253 C[C@@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CC[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L15 compound treatment 232720.0 51800.0 3.53 227840.0 46100.0 3.43 4.9258 0.9999 831956 SMP2_000254 COc1c(O)ccc2c1cc([N+](=O)[O-])c3c(cc4OCOc4c23)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L16 compound treatment 191360.0 10500.0 0.71 193480.0 11800.0 0.88 1.1237 0.9949 604 SMP2_000255 Oc1c(Br)cc(/C=C\2/C3C=C(I)C=CC3NC2=O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L17 compound treatment 198240.0 17400.0 1.18 202040.0 20300.0 1.51 1.9058 0.9926 3199797 SMP2_000256 C[C@@]1([C@H]2[C@H](C(=O)O)[C@]3(CC4CC[C@H]3[C@@]52CC[C@@H]1O)CC4=C)C(=O)O5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L18 compound treatment 368560.0 188000.0 12.79 361480.0 180000.0 13.38 18.5076 0.9998 604 SMP2_000257 Oc1c(Br)cc(/C=C\2/C3C=C(I)C=CC3NC2=O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L19 compound treatment 191760.0 10900.0 0.74 185640.0 3920.0 0.29 0.7303 0.9169 97 SMP2_000258 CCCCC/C=C\C[C@@H]1O[C@H]1\C=C\C(O)C/C=C\CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L20 compound treatment 186920.0 6030.0 0.41 192120.0 10400.0 0.77 0.838 0.9562 3199798 SMP2_000259 CC1CC(OC2C(O)C(O)C(O)C(O)C2O)C(N)CC1NC(=N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L21 compound treatment 240000.0 59100.0 4.03 239840.0 58100.0 4.33 5.9083 0.9994 2108 SMP2_000260 COc1cc2C/C(=C\c3cc(C)c(O)c(C)c3)/C(=O)c2c(N)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L22 compound treatment 181920.0 1030.0 0.07 185800.0 4080.0 0.3 0.2644 0.8484 440 SMP2_000261 COC(=O)Nc1nc2cc(ccc2[nH]1)C(=O)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L23 compound treatment 187720.0 6830.0 0.47 186240.0 4520.0 0.34 0.5671 0.9872 1201 SMP2_000262 COc1cc(Cc2cnc(N)nc2N)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 L24 compound treatment 355760.0 175000.0 11.92 352840.0 171000.0 12.74 17.4359 0.9995 648 SMP2_000263 Oc1cc(O)cc(/C=C/c2ccc(O)c(O)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M01 mock treatment 181200.0 312.0 0.02 190760.0 9040.0 0.67 0.4907 0.7291 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M02 mock treatment 189960.0 9070.0 0.62 191680.0 9960.0 0.74 0.9614 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M03 compound treatment 222760.0 41900.0 2.85 223960.0 42200.0 3.14 4.2415 0.9988 549 SMP2_000264 Nc1ncnc2nc(cc(c3cccc(Br)c3)c12)c4ccc(nc4)N5CCOCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M04 compound treatment 228200.0 47300.0 3.23 225680.0 44000.0 3.27 4.5943 1.0 1092656 SMP2_000265 CC1OC(CC(=O)O)CC2=C1C(=O)c3c(O)cccc3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M05 compound treatment 225840.0 45000.0 3.06 230200.0 48500.0 3.61 4.7184 0.9967 1000067 SMP2_000266 NC(C(=O)NC1[C@H]2SCC(=C(N2C1=O)C(=O)O)Cl)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M06 compound treatment 234320.0 53400.0 3.64 233000.0 51300.0 3.82 5.2745 0.9997 535 SMP2_000267 ONC(=O)CCCN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M07 compound treatment 246520.0 65600.0 4.47 239800.0 58100.0 4.32 6.2205 0.9999 3177114 SMP2_000268 CN(C)c1cc2c(Nc3ccc4n(Cc5ccccc5)ncc4c3)ncnc2cn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M08 compound treatment 220200.0 39300.0 2.68 215000.0 33300.0 2.48 3.6465 0.9992 241 SMP2_000269 CC[C@@H](C)[C@@H](CO[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCS(=O)(=O)C)C(=O)OC(C)C)NCC(N)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M09 compound treatment 204000.0 23100.0 1.58 199280.0 17600.0 1.31 2.0382 0.9957 3076808 SMP2_000270 CC1(C)[C@H]2C[C@@H]1C(=C)[C@H](O)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M10 compound treatment 227760.0 46900.0 3.2 225640.0 43900.0 3.27 4.5709 0.9999 220 SMP2_000271 CCCCC[C@H](O)/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M11 compound treatment 541080.0 360000.0 24.56 530600.0 349000.0 25.97 35.7249 0.9996 1579 SMP2_000272 CC(Cc1ccc(O)c(O)c1)C(C)Cc2ccc(O)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M12 compound treatment 205920.0 25000.0 1.71 202360.0 20600.0 1.54 2.2929 0.9986 284 SMP2_000273 OC(=O)c1cc(ccc1O)N(Cc2ccccc2O)Cc3cc(O)ccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M13 compound treatment 202040.0 21200.0 1.44 196680.0 15000.0 1.11 1.8069 0.9918 3076815 SMP2_000274 CC(O)CCCCn1c(=O)n(C)c2ncn(C)c2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M14 compound treatment 484120.0 303000.0 20.67 485680.0 304000.0 22.62 30.615 0.999 1102317 SMP2_000275 COc1ccc(cc1)C23Oc4cc(OC)cc(OC)c4C3(O)C(O)C(C2c5ccccc5)C(=O)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M15 compound treatment 203680.0 22800.0 1.55 201000.0 19300.0 1.43 2.1133 0.9992 1907751 SMP2_000276 CN/C(=N\c1ccc(cc1)C2=NNC(=O)CC2C)/NC#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M16 compound treatment 196720.0 15800.0 1.08 200280.0 18600.0 1.38 1.7399 0.9926 536 SMP2_000277 ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M17 compound treatment 243360.0 62500.0 4.26 236680.0 55000.0 4.09 5.904 0.9998 3076873 SMP2_000278 COc1cc(O)c(CC=C(C)C)c(O)c1C(=O)/C=C/c2ccc(O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M18 compound treatment 219120.0 38200.0 2.61 216760.0 35000.0 2.61 3.6871 1.0 536 SMP2_000279 ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M19 compound treatment 194240.0 13400.0 0.91 192880.0 11200.0 0.83 1.2309 0.999 3199800 SMP2_000280 CC(C)CCC[C@@H](C)[C@H]1CC(=O)[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M20 compound treatment 189320.0 8430.0 0.57 189360.0 7640.0 0.57 0.8085 1.0 3199801 SMP2_000281 CO[C@@H]([C@H](O)CC(=O)[C@@H](C)[C@@H](O)CC[C@@H](C)C1O[C@]2(CC[C@@H](C)C(CC[C@H](C)C(=O)C)O2)CC[C@@H]1C)[C@H](OC(=O)C[C@@H](O)C3=C(C)C(=O)OC3=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M21 compound treatment 185080.0 4190.0 0.29 190720.0 9000.0 0.67 0.6757 0.9279 257 SMP2_000282 CCCCC[C@H](O)/C=C/[C@H]1[C@H](O)C[C@H](O)[C@@H]1CC(=O)CCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M22 compound treatment 197480.0 16600.0 1.13 198560.0 16800.0 1.25 1.686 0.9987 3076883 SMP2_000283 CCC(C)C1NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(N)CSSCC(NC(=O)C(CC(=O)N)NC(=O)C(CCC(=O)N)NC1=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M23 compound treatment 184720.0 3830.0 0.26 185520.0 3800.0 0.28 0.3846 0.9992 2059 SMP2_000284 CC(C)CC(N)C(O)C(=O)NC(C(C)C)C(=O)NC(C(C)C)C(=O)NC(CC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 M24 compound treatment 233600.0 52700.0 3.59 236640.0 54900.0 4.09 5.4314 0.9979 2350 SMP2_000285 Cc1c(C)c2OC(C)(CN3CCN(CC3)c4cc(nc(n4)N5CCCC5)N6CCCC6)CCc2c(C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N01 mock treatment 184880.0 3990.0 0.27 185680.0 3960.0 0.29 0.4008 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N02 mock treatment 185480.0 4590.0 0.31 181640.0 -81.2 -0.01 0.2171 0.6933 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N03 compound treatment 197960.0 17100.0 1.16 187000.0 5280.0 0.39 1.1008 0.8961 3076955 SMP2_000286 CC(C)(C)[C@]1(O)C[C@@H]2OC(=O)CC23C(=O)O[C@@H]4OC(=O)[C@H](O)C413 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N04 compound treatment 258160.0 77300.0 5.27 261080.0 79400.0 5.91 7.9016 0.9984 907302 SMP2_000287 CN1CC[C@]2(C)C1N(C)c3ccc(O)cc32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N05 compound treatment 203280.0 22400.0 1.53 200480.0 18800.0 1.4 2.0667 0.999 3199802 SMP2_000288 CSC(=S)NCc1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N06 compound treatment 190720.0 9830.0 0.67 200720.0 19000.0 1.41 1.4738 0.9418 398 SMP2_000289 OC[C@H]1NC[C@@H](O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N07 compound treatment 199960.0 19100.0 1.3 198520.0 16800.0 1.25 1.8035 0.9998 1975 SMP2_000290 C[C@@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@@H](O)CC[C@@]43C)[C@@]2(O)CC[C@@H]1c5ccc(=O)oc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N08 compound treatment 253760.0 72900.0 4.97 250960.0 69200.0 5.15 7.1569 0.9998 1026746 SMP2_000291 OCc1cc(O)c2C(=O)c3c(O)cccc3C(=O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N09 compound treatment 272040.0 91200.0 6.21 273440.0 91700.0 6.83 9.2212 0.9989 810 SMP2_000292 CCCCC[C@@H]1[C@@H](OC(=O)CC(C)C)[C@H](C)OC(=O)[C@@H](NC(=O)c2cccc(NC=O)c2O)[C@@H](C)OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N10 compound treatment 193600.0 12700.0 0.87 198800.0 17100.0 1.27 1.5116 0.9826 3176068 SMP2_000293 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CO)NC(=O)CCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N11 compound treatment 303520.0 123000.0 8.36 304320.0 123000.0 9.12 12.364 0.999 2018 SMP2_000294 NC1=NC(=O)/C(=C/2\CCNC(=O)c3[nH]ccc23)/N1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N12 compound treatment 208320.0 27400.0 1.87 202360.0 20600.0 1.54 2.4086 0.9952 1090 SMP2_000295 CCC[C@@H]1C[C@H](N(C)C1)C(=O)NC(C(C)Cl)C2O[C@H](SC)[C@H](O)[C@@H](O)[C@H]2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N13 compound treatment 202640.0 21800.0 1.48 193960.0 12200.0 0.91 1.6927 0.9726 3199804 SMP2_000296 CC(C)CC(NC(=O)C(Cc1ccc(OP(O)(O)O)cc1)NC(=O)C2CCCN2C(=O)C)C(=O)NC(CCCCN)C(=O)NC(C(C)O)C(=O)NC(CCCCN)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N14 compound treatment 184640.0 3750.0 0.26 189080.0 7360.0 0.55 0.5681 0.9399 1000674 SMP2_000297 COc1cccc2C(=O)c3c(O)c4CC(O)(CC(OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N15 compound treatment 292440.0 112000.0 7.61 294080.0 112000.0 8.36 11.2909 0.9989 1084811 SMP2_000298 Cc1c2[nH]c3ccc(O)cc3c2c(C)c4cnccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N16 compound treatment 262000.0 81100.0 5.53 258960.0 77200.0 5.75 7.9752 0.9998 3077040 SMP2_000299 CC(C)[C@H]1CN2CCC[C@H]2[C@@]3(O)O[C@](CC(=O)[C@H]4CN(C)[C@@H]5Cc6c[nH]c7cccc(C5=C4)c67)(C(C)C)C(=O)N13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N17 compound treatment 196640.0 15800.0 1.07 190880.0 9160.0 0.68 1.2414 0.9759 1108916 SMP2_000300 NCCCCC(NC(=O)C(Cc1c[nH]cn1)NC(=O)CN)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N18 compound treatment 410840.0 230000.0 15.68 394720.0 213000.0 15.85 22.2952 1.0 3177114 SMP2_000301 CN(C)c1cc2c(Nc3ccc4n(Cc5ccccc5)ncc4c3)ncnc2cn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N19 compound treatment 194240.0 13400.0 0.91 190920.0 9200.0 0.68 1.1278 0.9901 3076041 SMP2_000302 COc1cc(/C=C/c2cccc[n+]2C)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N20 compound treatment 190880.0 9990.0 0.68 192640.0 10900.0 0.81 1.0563 0.9962 1734 SMP2_000303 Nc1nnc(c(N)n1)c2cccc(Cl)c2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N21 compound treatment 205360.0 24500.0 1.67 204240.0 22500.0 1.68 2.3648 1.0 3076048 SMP2_000304 OC[C@H]1O[C@@H](Oc2c[nH]c3ccccc23)[C@H](O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N22 compound treatment 195520.0 14600.0 1.0 192960.0 11200.0 0.84 1.2968 0.9962 1000089 SMP2_000305 COC1C(C)OC(OC2CC(C)(O)C(C(=O)OC)c3cc4C(=O)c5c6OC7OC(C)(C(O)C(C7O)N(C)C)c6cc(O)c5C(=O)c4c(O)c23)C(OC)C1(C)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N23 compound treatment 266840.0 86000.0 5.86 267960.0 86200.0 6.42 8.6821 0.999 628 SMP2_000306 Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc34)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 N24 compound treatment 179440.0 -1450.0 -0.1 178760.0 -2960.0 -0.22 -0.2257 -0.9344 1273 SMP2_000307 C[C@@]12CC(=O)C3C(CCC4=CC(=O)C=C[C@]34C)C2CC[C@]1(O)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O01 mock treatment 184160.0 3270.0 0.22 185000.0 3280.0 0.24 0.3303 0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O02 mock treatment 184000.0 3110.0 0.21 185920.0 4200.0 0.31 0.371 0.9822 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O03 compound treatment 188360.0 7470.0 0.51 186040.0 4320.0 0.32 0.5875 0.9754 1059696 SMP2_000308 CC1CCC2(C)CCC3(C)C(=CCC4C5(C)CCC(O)C(C)(C)C5CCC43C)C2C1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O04 compound treatment 186000.0 5110.0 0.35 192640.0 10900.0 0.81 0.821 0.9286 988 SMP2_000309 COc1ccc2[nH]cc(CCNC(=O)C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O05 compound treatment 201560.0 20700.0 1.41 192000.0 10300.0 0.77 1.5375 0.9588 413 SMP2_000310 CCCCCC[C@@H]([C@@H](C)O)n1cnc2c(N)ncnc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O06 compound treatment 208480.0 27600.0 1.88 207000.0 25300.0 1.88 2.6605 1.0 3199805 SMP2_000311 NC(=O)OC[C@H]1[C@@H]2NC(=N)N[C@]23N(CCC3(O)O)C(=N)N1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O07 compound treatment 205880.0 25000.0 1.7 202560.0 20800.0 1.55 2.3015 0.9989 2081802 SMP2_000312 CC[C@@]1(O)C(=O)OCc2c1cc3-c4nc5ccc(O)c(CN(C)C)c5cc4Cn3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O08 compound treatment 190400.0 9510.0 0.65 191200.0 9480.0 0.71 0.9574 0.9991 1080649 SMP2_000313 CC1(CC2(O)OC3O1)C4(CC2C34COC(=O)c5ccccc5)OC6OC(CO)C(O)C(O)C6O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O09 compound treatment 184560.0 3670.0 0.25 188680.0 6960.0 0.52 0.5432 0.9443 3076119 SMP2_000314 CNc1ccc2ccccc2c1N=Nc3ccc(N=Nc4ccccc4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O10 compound treatment 187960.0 7070.0 0.48 191040.0 9320.0 0.69 0.8313 0.9842 1072985 SMP2_000315 CC1C(O)C2(O)C(C3C=C(CO)CC4(O)C(C=C(C)C4=O)C13O)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O11 compound treatment 198120.0 17200.0 1.17 199720.0 18000.0 1.34 1.7779 0.9979 3076122 SMP2_000316 CC(=C[C@H](C=C)C(C)(C)O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O12 compound treatment 195360.0 14500.0 0.99 202120.0 20400.0 1.52 1.7712 0.9782 3001166 SMP2_000317 C[C@H]/1CC[C@@H]2C[C@H](C[C@@](O)(O2)[C@@H]3CSC(=O)N3)OC(=O)\C=C(\C)/CC/C=C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O13 compound treatment 233360.0 52500.0 3.58 225680.0 44000.0 3.27 4.843 0.999 189 SMP2_000318 CCCCCC(O)c1cccc(OCc2ccc3ccccc3n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O14 compound treatment 196160.0 15300.0 1.04 197160.0 15400.0 1.15 1.5487 0.9988 3199895 SMP2_000319 CSCCC(NC(=O)C(CC(C)C)NC(=O)CNC(=O)C(Cc1ccc(O)cc1)NC(=O)C(Cc2ccccc2)NC(=O)C(CCCNC(=N)N)NC(=O)C(CCC(=O)O)NC(=O)C3CCCN3C(=O)C(CC(=O)N)NC(=O)C4CCCN4C(=O)C(N)CCCCN)C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O15 compound treatment 181720.0 832.0 0.06 183320.0 1600.0 0.12 0.1242 0.9425 2305 SMP2_000320 COC1=C(N)C(=O)c2nc(ccc2C1=O)c3nc(C(=O)O)c(C)c(c3N)c4ccc(OC)c(OC)c4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O16 compound treatment 192000.0 11100.0 0.76 195360.0 13600.0 1.02 1.2534 0.9896 3076126 SMP2_000321 Nc1ncnc2n([C@@H]3OC4COP(O)(S)O[C@@H]4C3O)c(nc12)N5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O17 compound treatment 217120.0 36200.0 2.47 216600.0 34900.0 2.6 3.5823 0.9997 2080871 SMP2_000322 CC1=C(O)C(=O)[C@@H]2O[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O18 compound treatment 231720.0 50800.0 3.47 231120.0 49400.0 3.68 5.0503 0.9996 3076175 SMP2_000323 COc1cc(ccc1O)[C@H]2Oc3cc(ccc3O[C@@H]2CO)[C@H]4Oc5cc(O)cc(O)c5C(=O)[C@@H]4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O19 compound treatment 193480.0 12600.0 0.86 190760.0 9040.0 0.67 1.0827 0.9927 3199896 SMP2_000324 CC(C)CCC[C@@H](C)[C@H]1CC(=O)C2=C3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O20 compound treatment 219680.0 38800.0 2.64 219280.0 37600.0 2.8 3.8467 0.9996 3076177 SMP2_000325 COc1cc(ccc1O)c2cc(=O)c3c(O)cc(OC4OC(CO)C(O)C(O)C4OS(=O)(=O)O)cc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O21 compound treatment 226680.0 45800.0 3.12 222600.0 40900.0 3.04 4.3589 0.9999 2119025 SMP2_000326 Nc1nc(S)c2nc[nH]c2n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O22 compound treatment 213000.0 32100.0 2.19 216200.0 34500.0 2.57 3.3626 0.9969 2081802 SMP2_000327 CC[C@@]1(O)C(=O)OCc2c1cc3-c4nc5ccc(O)c(CN(C)C)c5cc4Cn3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O23 compound treatment 157880.0 -23000.0 -1.57 159160.0 -22600.0 -1.68 -2.2965 -0.9994 316 SMP2_000328 CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 O24 compound treatment 182920.0 2030.0 0.14 184880.0 3160.0 0.24 0.2642 0.9682 1004963 SMP2_000329 CC1CCC2(CCC3(C)C(=CCC4C5(C)CCC(O)C(C)(C)C5CCC43C)C2C1C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P01 mock treatment 183040.0 2150.0 0.15 184600.0 2880.0 0.21 0.2552 0.9829 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P02 mock treatment 183760.0 2870.0 0.2 182400.0 679.0 0.05 0.1742 0.8614 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P03 compound treatment 224520.0 43600.0 2.97 223200.0 41500.0 3.09 4.2863 0.9998 3199897 SMP2_000330 CS[C@]12CC3=CC=CC(O)[C@H]3N2C(=O)[C@@](CO)(SC)N(C)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P04 compound treatment 186560.0 5670.0 0.39 187880.0 6160.0 0.46 0.5975 0.9964 2060488 SMP2_000331 CC(=CCC[C@@](C)(O)C=C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P05 compound treatment 184480.0 3590.0 0.24 185160.0 3440.0 0.26 0.3541 0.9998 1968 SMP2_000332 C[C@@H]1CC2OC3CC4OC(=O)C=C(C)C4O[C@@]3(C)CC2OC5CC[C@@]6(C)O[C@@]7(C)CC8OC9CC%10O[C@@]%11(C)[C@@H](O)C[C@@H](CC(=C)C=O)OC%11CC%10OC9C=CC[C@]8(C)OC7CC6OC15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P06 compound treatment 187400.0 6510.0 0.44 187840.0 6120.0 0.46 0.6359 0.9999 1000053 SMP2_000333 OC[C@H]1NC[C@H](O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P07 compound treatment 194760.0 13900.0 0.95 196400.0 14700.0 1.09 1.4412 0.9974 1977 SMP2_000334 CC12CCc3occc3[C@H]2CCC4(CC5CC[C@H]41)C[C@]5(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P08 compound treatment 184840.0 3950.0 0.27 186240.0 4520.0 0.34 0.4283 0.994 1693 SMP2_000335 NCCCNCCSP(=O)(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P09 compound treatment 188680.0 7790.0 0.53 192040.0 10300.0 0.77 0.9187 0.9838 3199899 SMP2_000336 CC[C@@H]1[C@H](O)[C@@H](C)C/C(=C\C=C/C(=C(\OC(=O)\C(=C/C(=C\[C@H](C)C1O)/C)\OC)/[C@@H](C)[C@@H](O)[C@H](C)[C@@]2(O)C[C@@H](OC3CC(O)C(OC(=O)N)C(C)O3)[C@H](C)[C@H](O2)/C=C/C)/OC)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P10 compound treatment 222960.0 42100.0 2.87 221160.0 39400.0 2.94 4.1038 0.9999 446 SMP2_000337 COc1cc(CNC(=O)CCCC/C=C/C(C)C)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P11 compound treatment 312600.0 132000.0 8.98 315400.0 134000.0 9.95 13.3848 0.9987 360 SMP2_000338 Oc1ccc(cc1)c2cc(=O)c3c(O)cc(O)cc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P12 compound treatment 196680.0 15800.0 1.08 196600.0 14900.0 1.11 1.5443 0.9999 3068886 SMP2_000339 CC(C)/N=c/1\cc2n(c3ccc(Cl)cc3)c4ccccc4nc2cc1Nc5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P13 compound treatment 200640.0 19800.0 1.35 191800.0 10100.0 0.75 1.4826 0.9618 1817 SMP2_000340 CC(=O)O[C@@]12CO[C@H]2C[C@@H](O)[C@@]3(C)[C@H]1[C@H](OC(=O)c4ccccc4)[C@@]5(O)C[C@H](OC(=O)[C@@H](O)[C@H](NC(=O)OC(C)(C)C)c6ccccc6)C(=C([C@H](O)C3=O)C5(C)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P14 compound treatment 192440.0 11600.0 0.79 192800.0 11100.0 0.82 1.1399 0.9997 3076236 SMP2_000341 COc1ccc(C=Cc2cc(O)cc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P15 compound treatment 188560.0 7670.0 0.52 191320.0 9600.0 0.71 0.875 0.9882 832320 SMP2_000342 CC[C@H](C)[C@H](NC(=O)[C@H]([C@@H](C)CC)N(C)C(=O)C)C(=O)N[C@@H](C(=O)C)C(=O)N[C@@H](CC(C)C)[C@@]1(O)O[C@H](C)[C@H](N[C@@]1(C)CO)C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P16 compound treatment 188160.0 7270.0 0.5 185520.0 3800.0 0.28 0.5505 0.9645 2069 SMP2_000343 CC12CCC3C(CCC4=C(O)C(=O)CCC34C)C2CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P17 compound treatment 186520.0 5630.0 0.38 188560.0 6840.0 0.51 0.6314 0.9903 3199902 SMP2_000344 CCC(C)C(NC(=O)C(Cc1ccc(O)cc1)NC(=O)C(CCCNC(=N)N)NC(=O)C(CCCNC(=N)N)NC(=O)C2CCCN2C(=O)C(C)NC(=O)C(N)CO)C(=O)N3CCCC3C(=O)NC(CC(C)C)C(=O)NC(Cc4ccccc4)C(=O)NCC(=O)NC(Cc5ccccc5)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P18 compound treatment 187040.0 6150.0 0.42 188560.0 6840.0 0.51 0.6565 0.9954 2100 SMP2_000345 COC(=O)CC(O)(CCCC(C)(C)O)C(=O)O[C@H]1[C@H]2c3cc4OCOc4cc3CCN5CCC[C@]25C=C1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P19 compound treatment 334560.0 154000.0 10.48 330880.0 149000.0 11.1 15.2581 0.9996 613 SMP2_000346 Oc1cc(/C=C/c2ccc(O)c(O)c2)oc(=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P20 compound treatment 188640.0 7750.0 0.53 185600.0 3880.0 0.29 0.5778 0.9595 3076242 SMP2_000347 CC1(C)O[C@H]2CC(=O)OC[C@]23[C@H]4CC[C@@](C)([C@@H](OC5OC(CO)C(O)C(O)C5O)c6ccoc6)[C@@]7(O[C@@H]7C(=O)O)[C@]4(C)C(=O)C[C@]13C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P21 compound treatment 182160.0 1270.0 0.09 182960.0 1240.0 0.09 0.1265 0.9995 3199903 SMP2_000348 C/C=C(/C)\C(=O)O[C@H]1C(=C[C@]2([C@H](C)C[C@H]3[C@@H](C3(C)C)[C@]4(C)C=C(CO)[C@@H](O)[C@@]12O)C4=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P22 compound treatment 207640.0 26800.0 1.82 209800.0 28100.0 2.09 2.7674 0.9977 1048361 SMP2_000349 c1ccc2c(c1)[nH]c3cnccc32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P23 compound treatment 175520.0 -5370.0 -0.37 177640.0 -4080.0 -0.3 -0.4736 -0.9957 832145 SMP2_000350 OC[C@@H]1[C@@H](O)[C@H](O)[C@H](O)[C@H]2NC(=O)C(=O)N21 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2099 P24 compound treatment 296480.0 116000.0 7.88 285680.0 104000.0 7.74 11.0436 1.0 2260 SMP2_000351 Cc1cc(O)c2c(=O)c3c(O)cc(O)c4c5c(O)cc(O)c6c(=O)c7c(O)cc(CO)c8c1c2c(c34)c(c65)c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A01 compound treatment 222840.0 33200.0 2.26 205320.0 16800.0 1.25 2.4827 0.961 3052787 PK04_100001 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A02 compound treatment 206600.0 16900.0 1.15 196960.0 8440.0 0.63 1.2599 0.9592 3052649 PK04_100002 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A03 compound treatment 208200.0 18500.0 1.26 200840.0 12300.0 0.92 1.5412 0.9877 3176622 PK04_100003 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A04 compound treatment 217000.0 27300.0 1.86 199440.0 10900.0 0.81 1.8917 0.9309 3175961 PK04_100004 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A05 compound treatment 191840.0 2160.0 0.15 185760.0 -2760.0 -0.21 -0.0411 -0.1627 3176556 PK04_100005 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A06 compound treatment 206280.0 16600.0 1.13 200320.0 11800.0 0.88 1.4213 0.9921 3176630 PK04_100006 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A07 compound treatment 217360.0 27700.0 1.89 214440.0 25900.0 1.93 2.6985 0.9999 3175901 PK04_100007 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A08 compound treatment 203640.0 14000.0 0.95 192920.0 4400.0 0.33 0.9046 0.8987 3176729 PK04_100008 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A09 compound treatment 246960.0 57300.0 3.91 286040.0 97500.0 7.26 7.8936 0.9577 3052580 PK04_100009 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A10 compound treatment 219560.0 29900.0 2.04 210840.0 22300.0 1.66 2.6151 0.9949 3176731 PK04_100010 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A11 compound treatment 263480.0 73800.0 5.03 220480.0 32000.0 2.38 5.2398 0.9415 3176633 PK04_100011 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A12 compound treatment 265280.0 75600.0 5.15 243880.0 55400.0 4.12 6.558 0.9938 3176445 PK04_100012 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A13 mock treatment 180080.0 -9600.0 -0.65 172920.0 -15600.0 -1.16 -1.2838 -0.9632 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A14 mock treatment 176920.0 -12800.0 -0.87 175000.0 -13500.0 -1.01 -1.3267 -0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A15 compound treatment 287400.0 97700.0 6.66 227800.0 39300.0 2.92 6.7781 0.9316 3175963 PK04_100013 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A16 compound treatment 279280.0 89600.0 6.11 244160.0 55600.0 4.14 7.2477 0.9821 3052785 PK04_100014 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A17 compound treatment 189360.0 -320.0 -0.02 185000.0 -3520.0 -0.26 -0.2007 -0.7633 3052837 PK04_100015 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A18 compound treatment 214320.0 24600.0 1.68 210400.0 21900.0 1.63 2.3393 0.9999 3176262 PK04_100016 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A19 compound treatment 193320.0 3640.0 0.25 186120.0 -2400.0 -0.18 0.0492 0.1608 3176686 PK04_100017 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A20 compound treatment 198360.0 8680.0 0.59 189760.0 1240.0 0.09 0.4837 0.8076 3176371 PK04_100018 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A21 compound treatment 200400.0 10700.0 0.73 192520.0 4000.0 0.3 0.7273 0.9216 3052829 PK04_100019 OC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A22 compound treatment 185360.0 -4320.0 -0.29 168360.0 -20200.0 -1.5 -1.2692 -0.8301 3052833 PK04_100020 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A23 compound treatment 185040.0 -4640.0 -0.32 167720.0 -20800.0 -1.55 -1.3183 -0.8344 3052878 PK04_100021 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 A24 compound treatment 192360.0 2680.0 0.18 185880.0 -2640.0 -0.2 -0.0097 -0.0363 3052694 PK04_100022 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B01 compound treatment 191240.0 1560.0 0.11 189200.0 680.0 0.05 0.111 0.9423 3052928 PK04_100023 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B02 compound treatment 305880.0 116000.0 7.92 285680.0 97200.0 7.23 10.7151 0.999 3052800 PK04_100024 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B03 compound treatment 189200.0 -480.0 -0.03 191440.0 2920.0 0.22 0.1305 0.5939 3052842 PK04_100025 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B04 compound treatment 179760.0 -9920.0 -0.68 177240.0 -11300.0 -0.84 -1.0719 -0.9943 3176782 PK04_100026 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B05 compound treatment 191440.0 1760.0 0.12 186920.0 -1600.0 -0.12 6.0E-4 0.0038 3175971 PK04_100027 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B06 compound treatment 277120.0 87400.0 5.96 256920.0 68400.0 5.09 7.8151 0.9969 3176561 PK04_100028 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B07 compound treatment 207160.0 17500.0 1.19 203120.0 14600.0 1.09 1.611 0.9989 3176369 PK04_100029 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B08 compound treatment 216920.0 27200.0 1.86 211280.0 22800.0 1.69 2.511 0.9989 3176441 PK04_100030 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B09 compound treatment 275840.0 86200.0 5.87 272440.0 83900.0 6.25 8.5702 0.9995 3052641 PK04_100031 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B10 compound treatment 211640.0 22000.0 1.5 199360.0 10800.0 0.81 1.6291 0.9579 3176555 PK04_100032 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B11 compound treatment 269440.0 79800.0 5.44 277760.0 89200.0 6.64 8.5416 0.9951 3176554 PK04_100033 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B12 compound treatment 213720.0 24000.0 1.64 217640.0 29100.0 2.17 2.6914 0.9905 3052747 PK04_100034 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B13 mock treatment 175640.0 -14000.0 -0.96 172000.0 -16500.0 -1.23 -1.5463 -0.9923 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B14 mock treatment 174680.0 -15000.0 -1.02 169320.0 -19200.0 -1.43 -1.7336 -0.9865 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B15 compound treatment 177880.0 -11800.0 -0.8 168760.0 -19800.0 -1.47 -1.6088 -0.9597 3052707 PK04_100035 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B16 compound treatment 279800.0 90100.0 6.14 260120.0 71600.0 5.33 8.1127 0.9975 3176447 PK04_100036 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B17 compound treatment 191040.0 1360.0 0.09 187720.0 -800.0 -0.06 0.0235 0.2129 3176194 PK04_100037 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B18 compound treatment 238600.0 48900.0 3.34 231960.0 43400.0 3.23 4.6445 0.9999 3176504 PK04_100038 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B19 compound treatment 185240.0 -4440.0 -0.3 183640.0 -4880.0 -0.36 -0.4709 -0.9959 3176439 PK04_100039 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B20 compound treatment 212720.0 23000.0 1.57 212320.0 23800.0 1.77 2.3633 0.9982 3176678 PK04_100040 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B21 compound treatment 185080.0 -4600.0 -0.31 177880.0 -10600.0 -0.79 -0.7817 -0.9178 3176260 PK04_100041 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B22 compound treatment 199600.0 9920.0 0.68 190360.0 1840.0 0.14 0.5751 0.8334 3176621 PK04_100042 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B23 compound treatment 185480.0 -4200.0 -0.29 183720.0 -4800.0 -0.36 -0.4551 -0.994 3176370 PK04_100043 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 B24 compound treatment 258280.0 68600.0 4.68 255680.0 67200.0 5.0 6.8416 0.9994 3176636 PK04_100044 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C01 compound treatment 212120.0 22400.0 1.53 201560.0 13000.0 0.97 1.7681 0.9759 3052532 PK04_100045 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C02 compound treatment 219640.0 30000.0 2.04 207440.0 18900.0 1.41 2.44 0.9835 3052638 PK04_100046 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C03 compound treatment 213280.0 23600.0 1.61 207400.0 18900.0 1.41 2.1313 0.9977 3052540 PK04_100047 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C04 compound treatment 220560.0 30900.0 2.11 205240.0 16700.0 1.24 2.3686 0.9685 3052751 PK04_100048 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C05 compound treatment 206240.0 16600.0 1.13 197080.0 8560.0 0.64 1.2488 0.9633 3052702 PK04_100049 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C06 compound treatment 223760.0 34100.0 2.32 214440.0 25900.0 1.93 3.0071 0.9957 3176680 PK04_100050 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C07 compound treatment 214880.0 25200.0 1.72 204480.0 16000.0 1.19 2.0548 0.9838 3052743 PK04_100051 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C08 compound treatment 222560.0 32900.0 2.24 214160.0 25600.0 1.91 2.9345 0.9968 3176043 PK04_100052 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C09 compound treatment 292600.0 103000.0 7.02 290720.0 102000.0 7.61 10.3402 0.9992 3052925 PK04_100053 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C10 compound treatment 213000.0 23300.0 1.59 209600.0 21100.0 1.57 2.2336 1.0 3176324 PK04_100054 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C11 mock treatment 182640.0 -7040.0 -0.48 176920.0 -11600.0 -0.86 -0.9499 -0.9616 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C12 mock treatment 177920.0 -11800.0 -0.8 182080.0 -6440.0 -0.48 -0.9059 -0.9698 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C13 compound treatment 254840.0 65200.0 4.44 281040.0 92500.0 6.89 8.0104 0.9775 3176376 PK04_100055 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C14 compound treatment 212120.0 22400.0 1.53 207200.0 18700.0 1.39 2.0649 0.9989 3176324 PK04_100056 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C15 mock treatment 177480.0 -12200.0 -0.83 182520.0 -6000.0 -0.45 -0.9039 -0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C16 mock treatment 188720.0 -960.0 -0.07 175120.0 -13400.0 -1.0 -0.7515 -0.7519 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C17 compound treatment 208280.0 18600.0 1.27 199000.0 10500.0 0.78 1.4482 0.9728 3052884 PK04_100057 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C18 compound treatment 274160.0 84500.0 5.76 268760.0 80200.0 5.97 8.2955 0.9998 3176562 PK04_100058 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C19 compound treatment 196680.0 7000.0 0.48 189160.0 640.0 0.05 0.3711 0.7738 3176124 PK04_100059 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C20 compound treatment 213720.0 24000.0 1.64 198480.0 9960.0 0.74 1.6831 0.9357 3052784 PK04_100060 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C21 compound treatment 200320.0 10600.0 0.73 196880.0 8360.0 0.62 0.9529 0.9971 3052792 PK04_100061 OC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C22 compound treatment 194600.0 4920.0 0.34 189640.0 1120.0 0.08 0.2961 0.8568 3052749 PK04_100062 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C23 compound treatment 170760.0 -18900.0 -1.29 171440.0 -17100.0 -1.27 -1.811 -1.0 3176204 PK04_100063 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 C24 compound treatment 256360.0 66700.0 4.55 229560.0 41000.0 3.05 5.3744 0.9813 3176041 PK04_100064 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D01 compound treatment 194600.0 4920.0 0.34 193560.0 5040.0 0.38 0.5024 0.9984 3052926 PK04_100065 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D02 compound treatment 263240.0 73600.0 5.02 259880.0 71400.0 5.31 7.3017 0.9996 3176201 PK04_100066 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D03 compound treatment 210520.0 20800.0 1.42 210760.0 22200.0 1.66 2.1751 0.9971 3052885 PK04_100067 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D04 compound treatment 176480.0 -13200.0 -0.9 183480.0 -5040.0 -0.38 -0.9016 -0.9247 3176377 PK04_100068 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D05 compound treatment 310840.0 121000.0 8.26 306720.0 118000.0 8.8 12.0615 0.9995 3052790 PK04_100069 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D06 compound treatment 231440.0 41800.0 2.85 224160.0 35600.0 2.65 3.8888 0.9994 3052881 PK04_100070 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D07 compound treatment 252640.0 63000.0 4.29 228440.0 39900.0 2.97 5.1361 0.9839 3052536 PK04_100071 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D08 compound treatment 219360.0 29700.0 2.02 223360.0 34800.0 2.59 3.2644 0.9925 3052923 PK04_100072 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D09 compound treatment 200520.0 10800.0 0.74 196920.0 8400.0 0.63 0.9647 0.9965 3052690 PK04_100073 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D10 compound treatment 217720.0 28000.0 1.91 214840.0 26300.0 1.96 2.7369 0.9999 3052841 PK04_100074 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D11 mock treatment 172640.0 -17000.0 -1.16 177640.0 -10900.0 -0.81 -1.3941 -0.9844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D12 mock treatment 187640.0 -2040.0 -0.14 175160.0 -13400.0 -0.99 -0.8015 -0.7982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D13 compound treatment 233000.0 43300.0 2.95 216320.0 27800.0 2.07 3.5514 0.9848 3176624 PK04_100075 NCCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D14 compound treatment 183680.0 -6000.0 -0.41 184280.0 -4240.0 -0.32 -0.5124 -0.9918 3176375 PK04_100076 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D15 mock treatment 180560.0 -9120.0 -0.62 176720.0 -11800.0 -0.88 -1.0607 -0.9857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D16 mock treatment 179120.0 -10600.0 -0.72 178120.0 -10400.0 -0.77 -1.0564 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D17 compound treatment 207240.0 17600.0 1.2 204320.0 15800.0 1.18 1.6781 1.0 3176503 PK04_100077 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D18 compound treatment 244880.0 55200.0 3.76 246800.0 58300.0 4.34 5.7282 0.9975 3052543 PK04_100078 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D19 compound treatment 211720.0 22000.0 1.5 212800.0 24300.0 1.81 2.3403 0.9958 3052538 PK04_100079 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D20 compound treatment 214000.0 24300.0 1.66 205400.0 16900.0 1.26 2.0608 0.9906 3052705 PK04_100080 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D21 compound treatment 189760.0 80.0 0.01 186080.0 -2440.0 -0.18 -0.1246 -0.6856 3052691 PK04_100081 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D22 compound treatment 204920.0 15200.0 1.04 192040.0 3520.0 0.26 0.9199 0.8585 3052534 PK04_100082 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D23 compound treatment 280200.0 90500.0 6.17 274920.0 86400.0 6.43 8.9109 0.9998 3176202 PK04_100083 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 D24 compound treatment 218800.0 29100.0 1.99 212000.0 23500.0 1.75 2.6395 0.998 3176197 PK04_100084 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E01 mock treatment 182240.0 -7440.0 -0.51 184400.0 -4120.0 -0.31 -0.5755 -0.9709 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E02 mock treatment 187920.0 -1760.0 -0.12 191040.0 2520.0 0.19 0.0478 0.2146 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E03 compound treatment 225680.0 36000.0 2.45 214160.0 25600.0 1.91 3.0849 0.9923 3176672 PK04_100085 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E04 compound treatment 231840.0 42200.0 2.87 220520.0 32000.0 2.38 3.7166 0.9956 3052883 PK04_100086 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E05 compound treatment 238840.0 49200.0 3.35 230120.0 41600.0 3.1 4.5592 0.9992 3176126 PK04_100087 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E06 compound treatment 231640.0 42000.0 2.86 223200.0 34700.0 2.58 3.848 0.9987 3052533 PK04_100088 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E07 compound treatment 245000.0 55300.0 3.77 213800.0 25300.0 1.88 3.9973 0.9484 3175839 PK04_100089 NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E08 compound treatment 209040.0 19400.0 1.32 206320.0 17800.0 1.32 1.8701 1.0 3052695 PK04_100090 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E09 mock treatment 185760.0 -3920.0 -0.27 192920.0 4400.0 0.33 0.0426 0.1007 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E10 mock treatment 187480.0 -2200.0 -0.15 185520.0 -3000.0 -0.22 -0.2639 -0.9813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E11 compound treatment 186800.0 -2880.0 -0.2 184400.0 -4120.0 -0.31 -0.3557 -0.9768 3176568 PK04_100091 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E12 compound treatment 218920.0 29200.0 1.99 210160.0 21600.0 1.61 2.5485 0.9944 3176044 PK04_100092 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E13 compound treatment 276600.0 86900.0 5.93 293640.0 105000.0 7.82 9.7225 0.9906 3052753 PK04_100093 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E14 compound treatment 214440.0 24800.0 1.69 217040.0 28500.0 2.12 2.6946 0.9936 3175962 PK04_100094 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E15 compound treatment 224000.0 34300.0 2.34 224320.0 35800.0 2.66 3.5386 0.9979 3176325 PK04_100095 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E16 compound treatment 283640.0 94000.0 6.41 271360.0 82800.0 6.17 8.8893 0.9998 3052542 PK04_100096 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E17 mock treatment 185040.0 -4640.0 -0.32 185360.0 -3160.0 -0.24 -0.39 -0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E18 mock treatment 181000.0 -8680.0 -0.59 184160.0 -4360.0 -0.32 -0.6479 -0.96 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E19 compound treatment 183280.0 -6400.0 -0.44 183200.0 -5320.0 -0.4 -0.5885 -0.9988 3052746 PK04_100097 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E20 compound treatment 211120.0 21400.0 1.46 202000.0 13500.0 1.0 1.743 0.9831 3176676 PK04_100098 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E21 compound treatment 212280.0 22600.0 1.54 214640.0 26100.0 1.94 2.4641 0.9934 3052756 PK04_100099 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E22 compound treatment 214280.0 24600.0 1.68 209920.0 21400.0 1.59 2.3122 0.9997 3176560 PK04_100100 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E23 compound treatment 197320.0 7640.0 0.52 197320.0 8800.0 0.65 0.8314 0.9936 3052487 PK04_100101 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 E24 compound treatment 180160.0 -9520.0 -0.65 258320.0 69800.0 5.19 3.2145 0.614 3176563 PK04_100102 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F01 mock treatment 184880.0 -4800.0 -0.33 179280.0 -9240.0 -0.69 -0.7177 -0.9423 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F02 mock treatment 187480.0 -2200.0 -0.15 189480.0 960.0 0.07 -0.0555 -0.3343 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F03 compound treatment 281200.0 91500.0 6.24 273240.0 84700.0 6.31 8.8707 1.0 3176684 PK04_100103 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F04 compound treatment 288240.0 98600.0 6.72 265840.0 77300.0 5.75 8.8206 0.997 3176121 PK04_100104 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F05 compound treatment 226120.0 36400.0 2.48 223800.0 35300.0 2.63 3.6134 0.9996 3176435 PK04_100105 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F06 compound treatment 238280.0 48600.0 3.31 244640.0 56100.0 4.18 5.2964 0.9934 3176627 PK04_100106 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F07 compound treatment 208680.0 19000.0 1.3 222280.0 33800.0 2.51 2.6927 0.9525 3176774 PK04_100107 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F08 compound treatment 231920.0 42200.0 2.88 231960.0 43400.0 3.23 4.3225 0.9983 3174822 PK04_100108 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F09 mock treatment 192640.0 2960.0 0.2 193200.0 4680.0 0.35 0.389 0.9663 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F10 mock treatment 190920.0 1240.0 0.08 188160.0 -360.0 -0.03 0.0408 0.4604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F11 compound treatment 213840.0 24200.0 1.65 211480.0 23000.0 1.71 2.373 0.9998 3176192 PK04_100109 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F12 compound treatment 223160.0 33500.0 2.28 218360.0 29800.0 2.22 3.1844 0.9999 3052594 PK04_100110 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F13 compound treatment 229680.0 40000.0 2.73 229240.0 40700.0 3.03 4.0713 0.9986 3052748 PK04_100111 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F14 compound treatment 296880.0 107000.0 7.31 303120.0 115000.0 8.53 11.1991 0.997 3176567 PK04_100112 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F15 compound treatment 242680.0 53000.0 3.61 239560.0 51000.0 3.8 5.2412 0.9997 3052759 PK04_100113 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F16 compound treatment 195320.0 5640.0 0.38 195800.0 7280.0 0.54 0.655 0.9859 3176780 PK04_100114 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F17 mock treatment 185720.0 -3960.0 -0.27 188800.0 280.0 0.02 -0.1762 -0.6506 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F18 mock treatment 186200.0 -3480.0 -0.24 187760.0 -760.0 -0.06 -0.2078 -0.8518 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F19 compound treatment 223040.0 33400.0 2.27 219640.0 31100.0 2.32 3.246 1.0 3176625 PK04_100115 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F20 compound treatment 228240.0 38600.0 2.63 229600.0 41100.0 3.06 4.0209 0.9972 3052750 PK04_100116 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F21 compound treatment 218280.0 28600.0 1.95 214640.0 26100.0 1.94 2.7534 1.0 3052889 PK04_100117 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F22 compound treatment 221640.0 32000.0 2.18 217800.0 29300.0 2.18 3.0817 1.0 3052696 PK04_100118 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F23 compound treatment 191760.0 2080.0 0.14 201080.0 12600.0 0.93 0.7613 0.8052 3176674 PK04_100119 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 F24 compound treatment 208880.0 19200.0 1.31 203520.0 15000.0 1.12 1.715 0.9969 3176436 PK04_100120 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G01 compound treatment 221960.0 32300.0 2.2 219680.0 31200.0 2.32 3.196 0.9997 3052845 PK04_100121 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G02 compound treatment 235640.0 46000.0 3.13 240720.0 52200.0 3.89 4.9628 0.9943 3052835 PK04_100122 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G03 mock treatment 193120.0 3440.0 0.23 190880.0 2360.0 0.18 0.29 0.9899 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G04 mock treatment 196000.0 6320.0 0.43 192760.0 4240.0 0.32 0.5278 0.9883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G05 compound treatment 244600.0 54900.0 3.74 232400.0 43900.0 3.27 4.9569 0.9977 3176502 PK04_100123 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G06 compound treatment 244160.0 54500.0 3.71 240040.0 51500.0 3.83 5.3378 0.9999 3176265 PK04_100124 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G07 compound treatment 207560.0 17900.0 1.22 202000.0 13500.0 1.0 1.5714 0.9953 3052742 PK04_100125 NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G08 compound treatment 231480.0 41800.0 2.85 224120.0 35600.0 2.65 3.8887 0.9993 3052639 PK04_100126 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G09 compound treatment 247960.0 58300.0 3.97 260440.0 71900.0 5.35 6.5946 0.9892 3176200 PK04_100127 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G10 compound treatment 235120.0 45400.0 3.1 232240.0 43700.0 3.25 4.4915 0.9997 3052650 PK04_100128 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G11 compound treatment 282440.0 92800.0 6.32 293320.0 105000.0 7.8 9.9872 0.9946 3176683 PK04_100129 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G12 compound treatment 230120.0 40400.0 2.76 218440.0 29900.0 2.23 3.5242 0.9944 3176631 PK04_100130 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G13 compound treatment 280840.0 91200.0 6.22 285920.0 97400.0 7.25 9.5206 0.9971 3176045 PK04_100131 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G14 compound treatment 250720.0 61000.0 4.16 255960.0 67400.0 5.02 6.4919 0.9957 3176196 PK04_100132 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G15 compound treatment 193960.0 4280.0 0.29 198960.0 10400.0 0.78 0.7558 0.9106 3176446 PK04_100133 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G16 compound treatment 270640.0 81000.0 5.52 262600.0 74100.0 5.51 7.8016 1.0 3052834 PK04_100134 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G17 compound treatment 217520.0 27800.0 1.9 221800.0 33300.0 2.48 3.0936 0.9914 3052640 PK04_100135 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G18 compound treatment 233040.0 43400.0 2.96 234720.0 46200.0 3.44 4.5217 0.9972 3176727 PK04_100136 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G19 mock treatment 194240.0 4560.0 0.31 195680.0 7160.0 0.53 0.5966 0.9671 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G20 mock treatment 193880.0 4200.0 0.29 185880.0 -2640.0 -0.2 0.0635 0.183 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G21 compound treatment 195160.0 5480.0 0.37 197280.0 8760.0 0.65 0.7252 0.9651 3176272 PK04_100137 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G22 compound treatment 204960.0 15300.0 1.04 202480.0 14000.0 1.04 1.4713 1.0 3176261 PK04_100138 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G23 compound treatment 218880.0 29200.0 1.99 211840.0 23300.0 1.74 2.635 0.9977 3176513 PK04_100139 OC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 G24 compound treatment 204920.0 15200.0 1.04 200400.0 11900.0 0.88 1.3599 0.9968 3052924 PK04_100140 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H01 compound treatment 197960.0 8280.0 0.56 192600.0 4080.0 0.3 0.6139 0.9577 3176557 PK04_100141 NCCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H02 compound treatment 301000.0 111000.0 7.59 304640.0 116000.0 8.64 11.4777 0.9979 3052875 PK04_100142 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H03 mock treatment 195800.0 6120.0 0.42 188520.0 0.0 0.0 0.295 0.7071 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H04 mock treatment 191480.0 1800.0 0.12 191840.0 3320.0 0.25 0.2615 0.9478 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H05 compound treatment 267200.0 77500.0 5.29 288320.0 99800.0 7.43 8.9894 0.9861 3052652 PK04_100143 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H06 compound treatment 268760.0 79100.0 5.39 282640.0 94100.0 7.01 8.7656 0.9916 3052786 PK04_100144 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H07 compound treatment 207720.0 18000.0 1.23 201280.0 12800.0 0.95 1.5412 0.9918 3176328 PK04_100145 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H08 compound treatment 234640.0 45000.0 3.07 230600.0 42100.0 3.13 4.382 0.9999 3176321 PK04_100146 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H09 compound treatment 233080.0 43400.0 2.96 225280.0 36800.0 2.74 4.0268 0.9992 3176735 PK04_100147 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H10 compound treatment 236840.0 47200.0 3.22 237520.0 49000.0 3.65 4.8523 0.998 3175969 PK04_100148 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H11 compound treatment 226560.0 36900.0 2.51 219680.0 31200.0 2.32 3.4178 0.9992 3176193 PK04_100149 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H12 compound treatment 220400.0 30700.0 2.09 219880.0 31400.0 2.33 3.1314 0.9985 3176050 PK04_100150 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H13 compound treatment 317120.0 127000.0 8.69 315240.0 127000.0 9.43 12.8127 0.9992 3176569 PK04_100151 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H14 compound treatment 297840.0 108000.0 7.37 317640.0 129000.0 9.61 12.0095 0.9914 3052874 PK04_100152 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H15 compound treatment 234400.0 44700.0 3.05 238120.0 49600.0 3.69 4.7662 0.9955 3052832 PK04_100153 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H16 compound treatment 286840.0 97200.0 6.62 307520.0 119000.0 8.86 10.9466 0.9898 3176267 PK04_100154 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H17 compound treatment 194520.0 4840.0 0.33 192160.0 3640.0 0.27 0.4249 0.9952 3176378 PK04_100155 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H18 compound treatment 213160.0 23500.0 1.6 214760.0 26200.0 1.95 2.5129 0.9951 3176322 PK04_100156 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H19 mock treatment 189960.0 280.0 0.02 194520.0 6000.0 0.45 0.3293 0.7367 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H20 mock treatment 191640.0 1960.0 0.13 187920.0 -600.0 -0.04 0.0629 0.4465 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H21 compound treatment 299720.0 110000.0 7.5 297240.0 109000.0 8.09 11.0265 0.9993 3052801 PK04_100157 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H22 compound treatment 209040.0 19400.0 1.32 203080.0 14600.0 1.08 1.6996 0.9952 3176726 PK04_100158 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H23 compound treatment 228600.0 38900.0 2.65 223440.0 34900.0 2.6 3.714 0.9999 3176558 PK04_100159 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 H24 compound treatment 188440.0 -1240.0 -0.08 186720.0 -1800.0 -0.13 -0.1545 -0.9754 3052704 PK04_100160 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I01 compound treatment 210680.0 21000.0 1.43 211400.0 22900.0 1.7 2.2165 0.9963 3052648 PK04_100161 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I02 compound treatment 231400.0 41700.0 2.84 218120.0 29600.0 2.2 3.569 0.992 3176506 PK04_100162 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I03 compound treatment 241880.0 52200.0 3.56 236640.0 48100.0 3.58 5.0489 1.0 3176274 PK04_100163 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I04 compound treatment 240840.0 51200.0 3.49 228520.0 40000.0 2.98 4.5714 0.9969 3176679 PK04_100164 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I05 mock treatment 197480.0 7800.0 0.53 193280.0 4760.0 0.35 0.6265 0.9805 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I06 mock treatment 200440.0 10800.0 0.73 200040.0 11500.0 0.86 1.125 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I07 compound treatment 273840.0 84200.0 5.74 291800.0 103000.0 7.69 9.4926 0.9896 3052930 PK04_100165 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I08 compound treatment 243040.0 53400.0 3.64 239960.0 51400.0 3.83 5.2796 0.9997 3176444 PK04_100166 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I09 compound treatment 303640.0 114000.0 7.77 298120.0 110000.0 8.16 11.2618 0.9997 3052697 PK04_100167 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I10 compound treatment 223040.0 33400.0 2.27 218560.0 30000.0 2.24 3.1892 1.0 3176731 PK04_100168 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I11 compound treatment 274440.0 84800.0 5.78 301400.0 113000.0 8.4 10.0268 0.9833 3052535 PK04_100169 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I12 compound treatment 228080.0 38400.0 2.62 222760.0 34200.0 2.55 3.6532 0.9999 3176198 PK04_100170 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I13 compound treatment 313840.0 124000.0 8.46 318680.0 130000.0 9.69 12.8356 0.9977 3176119 PK04_100171 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I14 compound treatment 234840.0 45200.0 3.08 230800.0 42300.0 3.15 4.4022 0.9999 3176442 PK04_100172 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I15 compound treatment 287120.0 97400.0 6.64 306680.0 118000.0 8.79 10.9159 0.9904 3176566 PK04_100173 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I16 compound treatment 235240.0 45600.0 3.11 230960.0 42400.0 3.16 4.4299 1.0 3052844 PK04_100174 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I17 compound treatment 226880.0 37200.0 2.54 226160.0 37600.0 2.8 3.7743 0.9988 3176781 PK04_100175 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I18 compound treatment 236480.0 46800.0 3.19 231120.0 42600.0 3.17 4.4981 1.0 3052891 PK04_100176 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I19 compound treatment 210960.0 21300.0 1.45 206400.0 17900.0 1.33 1.9669 0.9991 3052840 PK04_100177 OC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I20 compound treatment 207040.0 17400.0 1.18 205840.0 17300.0 1.29 1.7484 0.9991 3174821 PK04_100178 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I21 mock treatment 189920.0 240.0 0.02 188960.0 440.0 0.03 0.0347 0.9486 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I22 mock treatment 184760.0 -4920.0 -0.34 183200.0 -5320.0 -0.4 -0.5172 -0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I23 compound treatment 223080.0 33400.0 2.28 219080.0 30600.0 2.27 3.2185 1.0 3176670 PK04_100179 OC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 I24 compound treatment 203880.0 14200.0 0.97 200160.0 11600.0 0.87 1.2971 0.9985 3176728 PK04_100180 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J01 compound treatment 207840.0 18200.0 1.24 206000.0 17500.0 1.3 1.7954 0.9997 3176783 PK04_100181 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J02 compound treatment 292080.0 102000.0 6.98 300920.0 112000.0 8.37 10.8519 0.996 3176448 PK04_100182 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J03 compound treatment 265840.0 76200.0 5.19 278720.0 90200.0 6.71 8.4186 0.9919 3176047 PK04_100183 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J04 compound treatment 302200.0 113000.0 7.67 267680.0 79200.0 5.89 9.5904 0.9915 3176269 PK04_100184 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J05 mock treatment 200240.0 10600.0 0.72 198120.0 9600.0 0.71 1.0143 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J06 mock treatment 201880.0 12200.0 0.83 200400.0 11900.0 0.88 1.2134 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J07 compound treatment 275720.0 86000.0 5.87 318600.0 130000.0 9.68 10.9937 0.9712 3176635 PK04_100185 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J08 compound treatment 268440.0 78800.0 5.37 270560.0 82000.0 6.11 8.1145 0.9979 3176114 PK04_100186 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J09 compound treatment 282360.0 92700.0 6.32 273840.0 85300.0 6.35 8.9581 1.0 3175966 PK04_100187 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J10 compound treatment 220040.0 30400.0 2.07 227880.0 39400.0 2.93 3.535 0.9855 3052757 PK04_100188 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J11 compound treatment 256160.0 66500.0 4.53 250600.0 62100.0 4.62 6.472 1.0 3174819 PK04_100189 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J12 compound treatment 213760.0 24100.0 1.64 214280.0 25800.0 1.92 2.5165 0.997 3176738 PK04_100190 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J13 compound treatment 212320.0 22600.0 1.54 207680.0 19200.0 1.43 2.0998 0.9992 3176380 PK04_100191 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J14 compound treatment 296160.0 106000.0 7.26 297440.0 109000.0 8.11 10.8654 0.9985 3176199 PK04_100192 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J15 compound treatment 236560.0 46900.0 3.2 239920.0 51400.0 3.83 4.9651 0.996 3176623 PK04_100193 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J16 compound treatment 282400.0 92700.0 6.32 304360.0 116000.0 8.62 10.5663 0.9884 3176632 PK04_100194 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J17 compound treatment 249480.0 59800.0 4.08 251080.0 62600.0 4.66 6.1753 0.9978 3052795 PK04_100195 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J18 compound treatment 231920.0 42200.0 2.88 241400.0 52900.0 3.94 4.8193 0.9882 3052636 PK04_100196 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J19 compound treatment 246200.0 56500.0 3.85 282320.0 93800.0 6.98 7.6612 0.9608 3052591 PK04_100197 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J20 compound treatment 226400.0 36700.0 2.5 225920.0 37400.0 2.78 3.7385 0.9986 3176629 PK04_100198 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J21 mock treatment 184720.0 -4960.0 -0.34 185080.0 -3440.0 -0.26 -0.4202 -0.9906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J22 mock treatment 180000.0 -9680.0 -0.66 183640.0 -4880.0 -0.36 -0.7235 -0.9604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J23 compound treatment 213680.0 24000.0 1.64 212640.0 24100.0 1.8 2.4264 0.9989 3176776 PK04_100199 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 J24 compound treatment 214560.0 24900.0 1.7 219480.0 31000.0 2.3 2.8288 0.9886 3052544 PK04_100200 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K01 compound treatment 205560.0 15900.0 1.08 208400.0 19900.0 1.48 1.8118 0.9882 3176739 PK04_100201 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K02 compound treatment 232080.0 42400.0 2.89 233880.0 45400.0 3.38 4.4312 0.997 3176042 PK04_100202 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K03 compound treatment 235040.0 45400.0 3.09 227040.0 38500.0 2.87 4.214 0.9993 3052528 PK04_100203 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K04 compound treatment 239680.0 50000.0 3.41 235480.0 47000.0 3.5 4.8818 0.9999 3176564 PK04_100204 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K05 compound treatment 261440.0 71800.0 4.89 248200.0 59700.0 4.44 6.6003 0.9988 3176329 PK04_100205 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K06 compound treatment 244480.0 54800.0 3.74 243000.0 54500.0 4.05 5.509 0.9992 3052588 PK04_100206 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K07 mock treatment 199600.0 9920.0 0.68 195800.0 7280.0 0.54 0.8614 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K08 mock treatment 198080.0 8400.0 0.57 195360.0 6840.0 0.51 0.7649 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K09 compound treatment 209160.0 19500.0 1.33 211400.0 22900.0 1.7 2.1432 0.9924 3176733 PK04_100207 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K10 compound treatment 222360.0 32700.0 2.23 219360.0 30800.0 2.3 3.1985 0.9999 3052589 PK04_100208 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K11 compound treatment 309680.0 120000.0 8.18 322720.0 134000.0 9.99 12.8476 0.9951 3052651 PK04_100209 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K12 compound treatment 230560.0 40900.0 2.79 236360.0 47800.0 3.56 4.4885 0.9927 3176507 PK04_100210 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K13 compound treatment 311320.0 122000.0 8.29 319680.0 131000.0 9.76 12.7667 0.9967 3052706 PK04_100211 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K14 compound treatment 234560.0 44900.0 3.06 234400.0 45900.0 3.41 4.5782 0.9985 3175959 PK04_100212 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K15 mock treatment 196400.0 6720.0 0.46 193400.0 4880.0 0.36 0.5808 0.9934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K16 mock treatment 193760.0 4080.0 0.28 194160.0 5640.0 0.42 0.4935 0.98 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K17 compound treatment 248960.0 59300.0 4.04 248880.0 60400.0 4.49 6.0344 0.9986 3174817 PK04_100213 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K18 compound treatment 210400.0 20700.0 1.41 208760.0 20200.0 1.51 2.0641 0.9995 3176725 PK04_100214 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K19 compound treatment 221720.0 32000.0 2.18 212520.0 24000.0 1.79 2.8077 0.995 3052537 PK04_100215 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K20 compound treatment 207160.0 17500.0 1.19 197360.0 8840.0 0.66 1.3079 0.9608 3052596 PK04_100216 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K21 compound treatment 218880.0 29200.0 1.99 211440.0 22900.0 1.71 2.6139 0.997 3176049 PK04_100217 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K22 compound treatment 225440.0 35800.0 2.44 222440.0 33900.0 2.52 3.5091 0.9998 3052637 PK04_100218 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K23 mock treatment 181120.0 -8560.0 -0.58 179000.0 -9520.0 -0.71 -0.9137 -0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 K24 mock treatment 169880.0 -19800.0 -1.35 174600.0 -13900.0 -1.04 -1.6871 -0.9915 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L01 compound treatment 195640.0 5960.0 0.41 201080.0 12600.0 0.93 0.9483 0.9304 3052595 PK04_100219 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L02 compound treatment 309240.0 120000.0 8.15 314440.0 126000.0 9.37 12.3907 0.9976 3176046 PK04_100220 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L03 compound treatment 200480.0 10800.0 0.74 206040.0 17500.0 1.3 1.4427 0.9634 3052585 PK04_100221 NCCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L04 compound treatment 229480.0 39800.0 2.71 228320.0 39800.0 2.96 4.0133 0.999 3176734 PK04_100222 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L05 compound treatment 230040.0 40400.0 2.75 233160.0 44600.0 3.32 4.295 0.9956 3176688 PK04_100223 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L06 compound treatment 238520.0 48800.0 3.33 240160.0 51600.0 3.84 5.0722 0.9974 3176372 PK04_100224 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L07 mock treatment 199760.0 10100.0 0.69 199840.0 11300.0 0.84 1.0817 0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L08 mock treatment 199000.0 9320.0 0.64 202800.0 14300.0 1.06 1.2008 0.9698 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L09 compound treatment 259520.0 69800.0 4.76 254160.0 65600.0 4.89 6.8214 0.9999 3176559 PK04_100225 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L10 compound treatment 239600.0 49900.0 3.4 234520.0 46000.0 3.42 4.8274 1.0 3052527 PK04_100226 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L11 compound treatment 219560.0 29900.0 2.04 216080.0 27600.0 2.05 2.8909 1.0 3176432 PK04_100227 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L12 compound treatment 216760.0 27100.0 1.85 211200.0 22700.0 1.69 2.4991 0.999 3176326 PK04_100228 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L13 compound treatment 214360.0 24700.0 1.68 209960.0 21400.0 1.6 2.3181 0.9996 3176737 PK04_100229 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L14 compound treatment 273920.0 84200.0 5.74 280120.0 91600.0 6.82 8.8818 0.9964 3175964 PK04_100230 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L15 mock treatment 194920.0 5240.0 0.36 193040.0 4520.0 0.34 0.4905 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L16 mock treatment 194560.0 4880.0 0.33 192800.0 4280.0 0.32 0.4605 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L17 compound treatment 207640.0 18000.0 1.22 208120.0 19600.0 1.46 1.8973 0.9962 3176787 PK04_100231 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L18 compound treatment 210640.0 21000.0 1.43 216200.0 27700.0 2.06 2.4672 0.984 3175960 PK04_100232 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L19 compound treatment 206520.0 16800.0 1.15 216080.0 27600.0 2.05 2.2622 0.9624 3176273 PK04_100233 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L20 compound treatment 213320.0 23600.0 1.61 207960.0 19400.0 1.45 2.1627 0.9986 3052882 PK04_100234 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L21 compound treatment 203280.0 13600.0 0.93 201160.0 12600.0 0.94 1.3208 1.0 3176053 PK04_100235 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L22 compound treatment 205840.0 16200.0 1.1 207320.0 18800.0 1.4 1.7684 0.993 3052696 PK04_100236 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L23 mock treatment 180360.0 -9320.0 -0.64 178360.0 -10200.0 -0.76 -0.984 -0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 L24 mock treatment 173880.0 -15800.0 -1.08 176080.0 -12400.0 -0.93 -1.4164 -0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M01 compound treatment 217840.0 28200.0 1.92 210720.0 22200.0 1.65 2.5259 0.9972 3176052 PK04_100237 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M02 compound treatment 219560.0 29900.0 2.04 213480.0 25000.0 1.86 2.7541 0.9989 3176323 PK04_100238 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M03 compound treatment 214440.0 24800.0 1.69 216840.0 28300.0 2.11 2.6841 0.9939 3176206 PK04_100239 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M04 compound treatment 214840.0 25200.0 1.72 213360.0 24800.0 1.85 2.5202 0.9993 3052883 PK04_100240 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M05 compound treatment 228280.0 38600.0 2.63 226200.0 37700.0 2.8 3.8439 0.9995 3052744 PK04_100241 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M06 compound treatment 253680.0 64000.0 4.36 248120.0 59600.0 4.44 6.2219 1.0 3176505 PK04_100242 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M07 compound treatment 236920.0 47200.0 3.22 245560.0 57000.0 4.25 5.2792 0.9907 3176434 PK04_100243 NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M08 compound treatment 229840.0 40200.0 2.74 224360.0 35800.0 2.67 3.8222 0.9999 3176729 PK04_100244 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M09 mock treatment 199880.0 10200.0 0.7 197640.0 9120.0 0.68 0.9717 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M10 mock treatment 198760.0 9080.0 0.62 199520.0 11000.0 0.82 1.0166 0.9905 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M11 compound treatment 202560.0 12900.0 0.88 195280.0 6760.0 0.5 0.9767 0.9651 3052590 PK04_100245 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M12 compound treatment 223880.0 34200.0 2.33 227600.0 39100.0 2.91 3.7054 0.994 3176565 PK04_100246 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M13 mock treatment 195600.0 5920.0 0.4 195800.0 7280.0 0.54 0.6685 0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M14 mock treatment 205800.0 16100.0 1.1 202760.0 14200.0 1.06 1.5265 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M15 compound treatment 206880.0 17200.0 1.17 218920.0 30400.0 2.26 2.4291 0.9532 3176508 PK04_100247 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M16 compound treatment 287840.0 98200.0 6.69 274600.0 86100.0 6.41 9.2623 0.9998 3052587 PK04_100248 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M17 compound treatment 208080.0 18400.0 1.25 207640.0 19100.0 1.42 1.8933 0.998 3052643 PK04_100249 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M18 compound treatment 222480.0 32800.0 2.24 215600.0 27100.0 2.02 3.0064 0.9987 3176777 PK04_100250 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M19 compound treatment 211600.0 21900.0 1.49 207560.0 19000.0 1.42 2.0588 0.9996 3052583 PK04_100251 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M20 compound treatment 226080.0 36400.0 2.48 214920.0 26400.0 1.96 3.1442 0.9933 3052586 PK04_100252 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M21 compound treatment 211360.0 21700.0 1.48 209360.0 20800.0 1.55 2.1419 0.9997 3052593 PK04_100253 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M22 compound treatment 218360.0 28700.0 1.96 218200.0 29700.0 2.21 2.9446 0.9981 3176374 PK04_100254 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M23 compound treatment 206760.0 17100.0 1.16 209960.0 21400.0 1.6 1.9517 0.988 3052699 PK04_100255 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 M24 compound treatment 212960.0 23300.0 1.59 233440.0 44900.0 3.34 3.4863 0.942 3176628 PK04_100256 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N01 compound treatment 247080.0 57400.0 3.91 241200.0 52700.0 3.92 5.5396 1.0 3052530 PK04_100257 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N02 compound treatment 301880.0 112000.0 7.65 303440.0 115000.0 8.55 11.457 0.9984 3176510 PK04_100258 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N03 compound treatment 217760.0 28100.0 1.91 213520.0 25000.0 1.86 2.6694 0.9999 3052646 PK04_100259 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N04 compound treatment 277360.0 87700.0 5.98 276400.0 87900.0 6.54 8.8518 0.999 3176040 PK04_100260 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N05 compound treatment 321400.0 132000.0 8.98 320560.0 132000.0 9.83 13.299 0.999 3052838 PK04_100261 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N06 compound treatment 239720.0 50000.0 3.41 239560.0 51000.0 3.8 5.0985 0.9986 3176263 PK04_100262 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N07 compound treatment 296840.0 107000.0 7.31 313360.0 125000.0 9.29 11.7361 0.9929 3176511 PK04_100263 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N08 compound treatment 230400.0 40700.0 2.78 227080.0 38600.0 2.87 3.9924 0.9999 3052644 PK04_100264 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N09 mock treatment 200080.0 10400.0 0.71 195640.0 7120.0 0.53 0.8761 0.9897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N10 mock treatment 199600.0 9920.0 0.68 204320.0 15800.0 1.18 1.3097 0.9655 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N11 compound treatment 221840.0 32200.0 2.19 215240.0 26700.0 1.99 2.9566 0.9988 3052880 PK04_100265 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N12 compound treatment 249600.0 59900.0 4.09 243160.0 54600.0 4.07 5.7642 1.0 3176732 PK04_100266 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N13 mock treatment 202200.0 12500.0 0.85 198800.0 10300.0 0.77 1.1446 0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N14 mock treatment 201920.0 12200.0 0.83 199320.0 10800.0 0.8 1.1584 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N15 compound treatment 217160.0 27500.0 1.87 213120.0 24600.0 1.83 2.6194 0.9999 3052703 PK04_100267 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N16 compound treatment 267400.0 77700.0 5.3 271120.0 82600.0 6.15 8.0938 0.9973 3176120 PK04_100268 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N17 compound treatment 209880.0 20200.0 1.38 212640.0 24100.0 1.8 2.2432 0.9914 3052843 PK04_100269 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N18 compound treatment 244560.0 54900.0 3.74 238680.0 50200.0 3.73 5.2855 1.0 3176116 PK04_100270 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N19 compound treatment 208640.0 19000.0 1.29 210480.0 22000.0 1.63 2.0697 0.9933 3176319 PK04_100271 NCCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N20 compound treatment 263320.0 73600.0 5.02 259880.0 71400.0 5.31 7.3056 0.9996 3052797 PK04_100272 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N21 compound treatment 279720.0 90000.0 6.14 299480.0 111000.0 8.26 10.1803 0.9893 3052581 PK04_100273 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N22 compound treatment 206440.0 16800.0 1.14 204840.0 16300.0 1.21 1.6669 0.9995 3176118 PK04_100274 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N23 compound treatment 196600.0 6920.0 0.47 196040.0 7520.0 0.56 0.7294 0.9964 3176207 PK04_100275 NCCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 N24 compound treatment 202560.0 12900.0 0.88 207000.0 18500.0 1.38 1.5935 0.9765 3176266 PK04_100276 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O01 compound treatment 221920.0 32200.0 2.2 220600.0 32100.0 2.39 3.2425 0.9991 3176687 PK04_100277 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O02 compound treatment 214120.0 24400.0 1.67 211200.0 22700.0 1.69 2.3718 1.0 3176323 PK04_100278 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O03 compound treatment 227000.0 37300.0 2.54 222960.0 34400.0 2.56 3.6116 1.0 3176438 PK04_100279 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O04 compound treatment 244040.0 54400.0 3.71 234080.0 45600.0 3.39 5.0183 0.999 3176117 PK04_100280 C[N+](C)(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O05 compound treatment 233800.0 44100.0 3.01 226400.0 37900.0 2.82 4.1205 0.9995 3176384 PK04_100281 NCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O06 compound treatment 217560.0 27900.0 1.9 219040.0 30500.0 2.27 2.9502 0.9961 3052695 PK04_100282 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O07 compound treatment 277480.0 87800.0 5.99 308000.0 119000.0 8.89 10.5207 0.9814 3052929 PK04_100283 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O08 compound treatment 233680.0 44000.0 3.0 228200.0 39700.0 2.95 4.2094 1.0 3052798 PK04_100284 C[N+](C)(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O09 compound treatment 262400.0 72700.0 4.96 268920.0 80400.0 5.98 7.737 0.9956 3176509 PK04_100285 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O10 compound treatment 217480.0 27800.0 1.9 212520.0 24000.0 1.79 2.6033 0.9996 3176681 PK04_100286 C[N+](C)(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O11 mock treatment 195400.0 5720.0 0.39 197080.0 8560.0 0.64 0.7262 0.9723 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O12 mock treatment 194440.0 4760.0 0.32 192120.0 3600.0 0.27 0.4189 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O13 compound treatment 256480.0 66800.0 4.55 256360.0 67800.0 5.05 6.7906 0.9987 3176682 PK04_100287 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O14 compound treatment 223960.0 34300.0 2.34 233120.0 44600.0 3.32 3.9998 0.9853 3176320 PK04_100288 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O15 compound treatment 261280.0 71600.0 4.88 280240.0 91700.0 6.83 8.2787 0.9865 3176268 PK04_100289 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O16 compound treatment 227720.0 38000.0 2.59 220960.0 32400.0 2.41 3.5411 0.9994 3176373 PK04_100290 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O17 compound treatment 214280.0 24600.0 1.68 210640.0 22100.0 1.65 2.3501 1.0 3052700 PK04_100291 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O18 compound treatment 209440.0 19800.0 1.35 212360.0 23800.0 1.77 2.2072 0.9908 3176275 PK04_100292 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O19 compound treatment 222680.0 33000.0 2.25 228160.0 39600.0 2.95 3.677 0.991 3052887 PK04_100293 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O20 compound treatment 224960.0 35300.0 2.41 214240.0 25700.0 1.91 3.0544 0.9936 3176039 PK04_100294 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O21 compound treatment 212440.0 22800.0 1.55 211920.0 23400.0 1.74 2.3287 0.9983 3176637 PK04_100295 OC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O22 compound treatment 226160.0 36500.0 2.49 218040.0 29500.0 2.2 3.3122 0.9981 3176115 PK04_100296 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O23 compound treatment 246480.0 56800.0 3.87 237120.0 48600.0 3.62 5.2959 0.9994 3052755 PK04_100297 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 O24 compound treatment 204920.0 15200.0 1.04 209800.0 21300.0 1.58 1.8546 0.9791 3176443 PK04_100298 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P01 compound treatment 198520.0 8840.0 0.6 192120.0 3600.0 0.27 0.6156 0.9334 3052698 PK04_100299 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P02 compound treatment 283920.0 94200.0 6.42 288040.0 99500.0 7.41 9.7807 0.9975 3176634 PK04_100300 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccc(I)cc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P03 compound treatment 210560.0 20900.0 1.42 206480.0 18000.0 1.34 1.9518 0.9995 3174820 PK04_100301 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P04 compound treatment 242520.0 52800.0 3.6 245480.0 57000.0 4.24 5.545 0.9967 3052597 PK04_100302 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P05 compound treatment 308800.0 119000.0 8.12 282560.0 94000.0 7.0 10.6917 0.9973 3176270 PK04_100303 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P06 compound treatment 224000.0 34300.0 2.34 223440.0 34900.0 2.6 3.4923 0.9986 3176677 PK04_100304 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)NCCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P07 compound treatment 218520.0 28800.0 1.97 201240.0 12700.0 0.95 2.0598 0.9439 3176122 PK04_100305 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@@H]6N7[C@H]([C@H](C(=O)OCC=C)[C@@]68C(=O)Nc9ccccc98)C(=O)O[C@H]([C@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P08 compound treatment 218360.0 28700.0 1.96 219320.0 30800.0 2.29 3.0036 0.9969 3052701 PK04_100306 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P09 compound treatment 215480.0 25800.0 1.76 225400.0 36900.0 2.74 3.1847 0.9769 3175972 PK04_100307 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P10 compound treatment 206000.0 16300.0 1.11 207840.0 19300.0 1.44 1.8035 0.992 3052830 PK04_100308 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P11 mock treatment 195080.0 5400.0 0.37 196120.0 7600.0 0.57 0.6603 0.9784 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P12 mock treatment 192560.0 2880.0 0.2 186600.0 -1920.0 -0.14 0.0378 0.1556 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P13 compound treatment 210600.0 20900.0 1.43 203200.0 14700.0 1.09 1.7811 0.9913 3052541 PK04_100309 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P14 compound treatment 286440.0 96800.0 6.6 306760.0 118000.0 8.8 10.8873 0.9899 3052545 PK04_100310 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P15 compound treatment 209800.0 20100.0 1.37 209000.0 20500.0 1.52 2.0478 0.9986 3176381 PK04_100311 CN(C)CCCCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P16 compound treatment 299320.0 110000.0 7.47 277960.0 89400.0 6.66 9.9926 0.9983 3052789 PK04_100312 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P17 compound treatment 207840.0 18200.0 1.24 211680.0 23200.0 1.72 2.0943 0.9868 3052890 PK04_100313 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P18 compound treatment 229200.0 39500.0 2.69 236000.0 47500.0 3.53 4.404 0.991 3176779 PK04_100314 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P19 compound treatment 273800.0 84100.0 5.74 282160.0 93600.0 6.97 8.9833 0.9953 3052876 PK04_100315 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P20 compound treatment 214400.0 24700.0 1.69 212120.0 23600.0 1.76 2.4337 0.9998 3176264 PK04_100316 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)NCCCCCNC(=O)CS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P21 compound treatment 195680.0 6000.0 0.41 195200.0 6680.0 0.5 0.6408 0.9953 3052692 PK04_100317 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P22 compound treatment 195280.0 5600.0 0.38 201120.0 12600.0 0.94 0.9331 0.9215 3176051 PK04_100318 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P23 compound treatment 261200.0 71500.0 4.88 256920.0 68400.0 5.09 7.0476 0.9998 3052754 PK04_100319 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@@H]5N6[C@H]([C@H](C(=O)OCC=C)[C@@]57C(=O)Nc8ccccc87)C(=O)O[C@H]([C@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2100 P24 compound treatment 195360.0 5680.0 0.39 201440.0 12900.0 0.96 0.9538 0.9201 3176127 PK04_100320 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A01 compound treatment 202480.0 16000.0 1.09 197600.0 16800.0 1.25 1.6538 0.9977 3189007 PK04_101001 CC(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A02 compound treatment 199520.0 13000.0 0.89 199880.0 19100.0 1.42 1.6311 0.9745 3069619 PK04_101002 OCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A03 compound treatment 179720.0 -6780.0 -0.46 170280.0 -10500.0 -0.78 -0.8813 -0.9681 3189008 PK04_101003 CCCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A04 compound treatment 205880.0 19400.0 1.32 192040.0 11200.0 0.84 1.5251 0.9755 3189009 PK04_101004 CC(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A05 compound treatment 212200.0 25700.0 1.75 202080.0 21300.0 1.58 2.3581 0.9987 3069620 PK04_101005 OCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A06 compound treatment 189960.0 3460.0 0.24 185200.0 4380.0 0.33 0.3976 0.9874 3189010 PK04_101006 CCCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A07 compound treatment 195760.0 9260.0 0.63 192800.0 12000.0 0.89 1.0772 0.9857 3189011 PK04_101007 OCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCOC(=O)[C@@H]6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A08 compound treatment 193160.0 6660.0 0.45 191840.0 11000.0 0.82 0.9013 0.9612 3069621 PK04_101008 OCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A09 compound treatment 198280.0 11800.0 0.8 192840.0 12000.0 0.89 1.2008 0.9986 3189120 PK04_101009 CCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A10 compound treatment 188200.0 1700.0 0.12 183960.0 3140.0 0.23 0.2475 0.9479 3069622 PK04_101010 CCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A11 compound treatment 193320.0 6820.0 0.47 191080.0 10300.0 0.76 0.869 0.9717 3189121 PK04_101011 CC(C)(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A12 compound treatment 196320.0 9820.0 0.67 194080.0 13300.0 0.99 1.1715 0.9822 3069678 PK04_101012 CC(C)(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A13 mock treatment 176040.0 -10500.0 -0.71 164440.0 -16400.0 -1.22 -1.366 -0.9674 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A14 mock treatment 177520.0 -8980.0 -0.61 170200.0 -10600.0 -0.79 -0.9915 -0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A15 compound treatment 179320.0 -7180.0 -0.49 183680.0 2860.0 0.21 -0.1953 -0.366 3189122 PK04_101013 OCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A16 compound treatment 179000.0 -7500.0 -0.51 172880.0 -7940.0 -0.59 -0.7791 -0.9974 3069679 PK04_101014 OCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A17 compound treatment 182920.0 -3580.0 -0.24 177160.0 -3660.0 -0.27 -0.3649 -0.9985 3189123 PK04_101015 OCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A18 compound treatment 194440.0 7940.0 0.54 189840.0 9020.0 0.67 0.8578 0.9943 3189124 PK04_101016 OCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A19 compound treatment 201320.0 14800.0 1.01 193520.0 12700.0 0.95 1.3831 0.9994 3069680 PK04_101017 OCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A20 compound treatment 189920.0 3420.0 0.23 180880.0 62.0 0.0 0.1683 0.7209 3189125 PK04_101018 OCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A21 compound treatment 210240.0 23700.0 1.62 183880.0 3060.0 0.23 1.3058 0.7988 3069681 PK04_101019 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C(=O)N(CCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A22 compound treatment 191600.0 5100.0 0.35 184320.0 3500.0 0.26 0.4304 0.9899 3189126 PK04_101020 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCCOC(=O)C5[C@H]4C(=O)N(CCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A23 compound treatment 193160.0 6660.0 0.45 184280.0 3460.0 0.26 0.5035 0.9639 3189127 PK04_101021 OCCCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 A24 compound treatment 189680.0 3180.0 0.22 185920.0 5100.0 0.38 0.422 0.9648 3069682 PK04_101022 OCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B01 compound treatment 191800.0 5300.0 0.36 183000.0 2180.0 0.16 0.3705 0.9347 3189128 PK04_101023 CCCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B02 compound treatment 114160.0 -72300.0 -4.93 118560.0 -62300.0 -4.63 -6.7637 -0.9995 3189129 PK04_101024 CCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4c(Cl)cccc4CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B03 compound treatment 196720.0 10200.0 0.7 196160.0 15300.0 1.14 1.3003 0.972 3069683 PK04_101025 OCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B04 compound treatment 177480.0 -9020.0 -0.61 173960.0 -6860.0 -0.51 -0.7956 -0.9957 3189130 PK04_101026 CC(C)(C)N(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4c(Cl)cccc4CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B05 compound treatment 202800.0 16300.0 1.11 199560.0 18700.0 1.39 1.7723 0.9937 3069684 PK04_101027 CCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B06 compound treatment 185080.0 -1420.0 -0.1 179840.0 -978.0 -0.07 -0.1197 -0.9903 3189131 PK04_101028 COc1ccc(cc1)N(CC=C)C(=O)C2N(C(=O)C3C(C4OC23C=C4)C(=O)O)c5c(Cl)cccc5CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B07 compound treatment 206160.0 19700.0 1.34 199240.0 18400.0 1.37 1.9175 0.9999 3189132 PK04_101029 CC(C)(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B08 compound treatment 178120.0 -8380.0 -0.57 177000.0 -3820.0 -0.28 -0.6047 -0.9481 3069685 PK04_101030 OCc1cccc(Cl)c1N2C(C(=O)N(CC=C)Cc3ccccc3)C4(OC5C=C4)C(C5C(=O)O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B09 compound treatment 188320.0 1820.0 0.12 192840.0 12000.0 0.89 0.7206 0.7977 3189133 PK04_101031 OCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B10 compound treatment 177600.0 -8900.0 -0.61 172840.0 -7980.0 -0.59 -0.8487 -0.9999 3189129 PK04_101032 CCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4c(Cl)cccc4CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B11 compound treatment 202000.0 15500.0 1.06 191720.0 10900.0 0.81 1.3212 0.9915 3189134 PK04_101033 OCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B12 compound treatment 185160.0 -1340.0 -0.09 180240.0 -578.0 -0.04 -0.0948 -0.9414 3069686 PK04_101034 CCCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4c(Cl)cccc4CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B13 mock treatment 173600.0 -12900.0 -0.88 167480.0 -13300.0 -0.99 -1.3236 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B14 mock treatment 172720.0 -13800.0 -0.94 165040.0 -15800.0 -1.17 -1.4945 -0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B15 compound treatment 194880.0 8380.0 0.57 191240.0 10400.0 0.78 0.9527 0.9887 3189135 PK04_101035 C[C@]12C3[C@H](OC24C=CCN(C(=O)[C@H]4N(CCO)C1=O)c5ccc(Cl)cc5)/C=C\CCCOC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B16 compound treatment 174240.0 -12300.0 -0.84 167040.0 -13800.0 -1.03 -1.3159 -0.9948 3069686 PK04_101036 CCCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4c(Cl)cccc4CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B17 compound treatment 206880.0 20400.0 1.39 201640.0 20800.0 1.55 2.0785 0.9985 3189136 PK04_101037 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C(=O)N(CCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B18 compound treatment 179080.0 -7420.0 -0.51 174320.0 -6500.0 -0.48 -0.6995 -0.9998 3069687 PK04_101038 COc1ccc(cc1)N(CC=C)C(=O)C2N(C(=O)C3C(C4OC23C=C4)C(=O)O)c5ccc(CCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B19 compound treatment 192040.0 5540.0 0.38 184200.0 3380.0 0.25 0.4453 0.9805 3189137 PK04_101039 CC1CC/C=C\[C@H]2OC34C=CCN(Cc5ccccc5)C(=O)[C@H]4N(CCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B20 compound treatment 174440.0 -12100.0 -0.82 171600.0 -9220.0 -0.69 -1.0663 -0.996 3069688 PK04_101040 OCCc1ccc(cc1)N2C(C(=O)N(CC=C)Cc3ccccc3)C4(OC5C=C4)C(C5C(=O)O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B21 compound treatment 196720.0 10200.0 0.7 185680.0 4860.0 0.36 0.7488 0.9534 3189138 PK04_101041 CC(C)N1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B22 compound treatment 104400.0 -82100.0 -5.6 117160.0 -63700.0 -4.74 -7.3079 -0.9966 3189139 PK04_101042 CCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4ccc(CCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B23 compound treatment 185040.0 -1460.0 -0.1 177840.0 -2980.0 -0.22 -0.2269 -0.9344 3069689 PK04_101043 CCCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 B24 compound treatment 116480.0 -70000.0 -4.77 123480.0 -57300.0 -4.27 -6.3929 -0.9984 3189140 PK04_101044 CC(C)(C)N(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4ccc(CCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C01 compound treatment 192600.0 6100.0 0.42 188240.0 7420.0 0.55 0.6849 0.9903 3189247 PK04_101045 CC(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C02 compound treatment 189400.0 2900.0 0.2 197280.0 16500.0 1.23 1.0064 0.8109 3069724 PK04_101046 CC(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C03 compound treatment 204360.0 17900.0 1.22 194280.0 13500.0 1.0 1.5697 0.9953 3189248 PK04_101047 CCCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C04 compound treatment 198600.0 12100.0 0.83 185680.0 4860.0 0.36 0.8394 0.9316 3189249 PK04_101048 OCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C05 compound treatment 201480.0 15000.0 1.02 192840.0 12000.0 0.89 1.355 0.9978 3069725 PK04_101049 OCCCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCOC(=O)[C@@H]6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C06 compound treatment 201080.0 14600.0 0.99 193720.0 12900.0 0.96 1.3821 0.9998 3189250 PK04_101050 CCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C07 compound treatment 200080.0 13600.0 0.93 194720.0 13900.0 1.03 1.3865 0.9985 3069726 PK04_101051 CCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C08 compound treatment 196280.0 9780.0 0.67 195560.0 14700.0 1.1 1.2475 0.9715 3189251 PK04_101052 CC(C)(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C09 compound treatment 199560.0 13100.0 0.89 191760.0 10900.0 0.81 1.2056 0.999 3189252 PK04_101053 CC(C)(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C10 compound treatment 194560.0 8060.0 0.55 192560.0 11700.0 0.87 1.0067 0.975 3069727 PK04_101054 OCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C11 mock treatment 171960.0 -14500.0 -0.99 171680.0 -9140.0 -0.68 -1.1817 -0.9831 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C12 mock treatment 176840.0 -9660.0 -0.66 177440.0 -3380.0 -0.25 -0.6433 -0.9128 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C13 compound treatment 197440.0 10900.0 0.75 194920.0 14100.0 1.05 1.2697 0.986 3189253 PK04_101055 OCCCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C14 compound treatment 192320.0 5820.0 0.4 193080.0 12300.0 0.91 0.9261 0.9305 3069728 PK04_101056 OCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C15 mock treatment 177480.0 -9020.0 -0.61 174760.0 -6060.0 -0.45 -0.7535 -0.9884 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C16 mock treatment 176360.0 -10100.0 -0.69 169440.0 -11400.0 -0.85 -1.0874 -0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C17 compound treatment 198800.0 12300.0 0.84 188920.0 8100.0 0.6 1.0195 0.9869 3189254 PK04_101057 OCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C18 compound treatment 197160.0 10700.0 0.73 190240.0 9420.0 0.7 1.01 0.9998 3189255 PK04_101058 OCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C19 compound treatment 194840.0 8340.0 0.57 190640.0 9820.0 0.73 0.9192 0.9923 3069729 PK04_101059 OCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C20 compound treatment 207160.0 20700.0 1.41 198320.0 17500.0 1.3 1.9173 0.9992 3189256 PK04_101060 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCCOC(=O)C5[C@H]4C(=O)N(CCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C21 compound treatment 212680.0 26200.0 1.79 203480.0 22700.0 1.69 2.4549 0.9996 3189257 PK04_101061 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C(=O)N(CCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C22 compound treatment 195440.0 8940.0 0.61 195280.0 14500.0 1.08 1.1923 0.9638 3069730 PK04_101062 CC(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C23 compound treatment 169400.0 -17100.0 -1.17 166600.0 -14200.0 -1.06 -1.5724 -0.9988 3189258 PK04_101063 CC(C)C(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 C24 compound treatment 196160.0 9660.0 0.66 192920.0 12100.0 0.9 1.1028 0.9882 3069731 PK04_101064 CC(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D01 compound treatment 202520.0 16000.0 1.09 199360.0 18500.0 1.38 1.7483 0.9933 3189259 PK04_101065 CC1CC/C=C\[C@H]2OC34C=CCN(Cn5nnc6ccccc56)C(=O)[C@H]4N(CCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D02 compound treatment 110360.0 -76100.0 -5.19 122760.0 -58100.0 -4.32 -6.7259 -0.9958 3069687 PK04_101066 COc1ccc(cc1)N(CC=C)C(=O)C2N(C(=O)C3C(C4OC23C=C4)C(=O)O)c5ccc(CCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D03 compound treatment 202840.0 16300.0 1.11 191600.0 10800.0 0.8 1.3553 0.987 3189260 PK04_101067 CCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D04 compound treatment 109960.0 -76500.0 -5.22 106600.0 -74200.0 -5.52 -7.5956 -0.9996 3069688 PK04_101068 OCCc1ccc(cc1)N2C(C(=O)N(CC=C)Cc3ccccc3)C4(OC5C=C4)C(C5C(=O)O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D05 compound treatment 203560.0 17100.0 1.16 183680.0 2860.0 0.21 0.9732 0.8229 3069732 PK04_101069 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCO)C(=O)[C@@H]3C2C(=O)O1)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D06 compound treatment 184720.0 -1780.0 -0.12 176640.0 -4180.0 -0.31 -0.3055 -0.9155 3189139 PK04_101070 CCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4ccc(CCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D07 compound treatment 197480.0 11000.0 0.75 192440.0 11600.0 0.86 1.1412 0.9974 3189261 PK04_101071 CC1CC/C=C\[C@H]2OC34C=CCN(CCN5CCOCC5)C(=O)[C@H]4N(CCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D08 compound treatment 182880.0 -3620.0 -0.25 175280.0 -5540.0 -0.41 -0.4658 -0.9698 3069733 PK04_101072 CCCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4ccc(CCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D09 compound treatment 199760.0 13300.0 0.9 197240.0 16400.0 1.22 1.5037 0.989 3189262 PK04_101073 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCO)C(=O)[C@@H]3C2C(=O)O1)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D10 compound treatment 185880.0 -616.0 -0.04 183560.0 2740.0 0.2 0.1146 0.5501 3069733 PK04_101074 CCCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4ccc(CCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D11 mock treatment 177360.0 -9140.0 -0.62 168240.0 -12600.0 -0.94 -1.1024 -0.9804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D12 mock treatment 176360.0 -10100.0 -0.69 169240.0 -11600.0 -0.86 -1.098 -0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D13 compound treatment 204320.0 17800.0 1.22 191120.0 10300.0 0.77 1.4014 0.9753 3189263 PK04_101075 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCO)C(=O)[C@]3(C)C2C(=O)O1)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D14 compound treatment 182240.0 -4260.0 -0.29 174080.0 -6740.0 -0.5 -0.5598 -0.9662 3069734 PK04_101076 CC(C)(C)N(CC=C)C(=O)C1N(CCOCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D15 mock treatment 175560.0 -10900.0 -0.75 175280.0 -5540.0 -0.41 -0.8187 -0.9609 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D16 mock treatment 176840.0 -9660.0 -0.66 171720.0 -9100.0 -0.68 -0.9443 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D17 compound treatment 205560.0 19100.0 1.3 200560.0 19700.0 1.47 1.958 0.9981 3189264 PK04_101077 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C(=O)N(CCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D18 compound treatment 171680.0 -14800.0 -1.01 171120.0 -9700.0 -0.72 -1.2246 -0.9864 3069734 PK04_101078 CC(C)(C)N(CC=C)C(=O)C1N(CCOCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D19 compound treatment 203880.0 17400.0 1.19 195400.0 14600.0 1.09 1.6055 0.999 3069735 PK04_101079 CC1CC/C=C\[C@H]2OC34C=CCN(Cc5ccccc5)C(=O)[C@H]4N(CCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D20 compound treatment 184800.0 -1700.0 -0.12 174920.0 -5900.0 -0.44 -0.3922 -0.8639 3189265 PK04_101080 COc1ccc(cc1)N(CC=C)C(=O)C2N(CCOCCO)C(=O)C3C(C4OC23C=C4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D21 compound treatment 196360.0 9860.0 0.67 188600.0 7780.0 0.58 0.8851 0.9972 3189266 PK04_101081 CC(C)N1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D22 compound treatment 101840.0 -84700.0 -5.77 100560.0 -80300.0 -5.97 -8.3049 -0.9999 3189265 PK04_101082 COc1ccc(cc1)N(CC=C)C(=O)C2N(CCOCCO)C(=O)C3C(C4OC23C=C4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D23 compound treatment 198480.0 12000.0 0.82 187960.0 7140.0 0.53 0.9536 0.9783 3069736 PK04_101083 CCCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 D24 compound treatment 144720.0 -41800.0 -2.85 148440.0 -32400.0 -2.41 -3.7179 -0.9965 3189267 PK04_101084 OCCOCCN1C(C(=O)N(CC=C)Cc2ccccc2)C3(OC4C=C3)C(C4C(=O)O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E01 mock treatment 182040.0 -4460.0 -0.3 181760.0 942.0 0.07 -0.1652 -0.53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E02 mock treatment 179040.0 -7460.0 -0.51 179320.0 -1500.0 -0.11 -0.4383 -0.8422 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E03 compound treatment 208880.0 22400.0 1.53 207960.0 27100.0 2.02 2.5075 0.9904 3189373 PK04_101085 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E04 compound treatment 216960.0 30500.0 2.08 211680.0 30900.0 2.3 3.0928 0.9987 3189374 PK04_101086 CCCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E05 compound treatment 223320.0 36800.0 2.51 209240.0 28400.0 2.12 3.271 0.9964 3069761 PK04_101087 CCCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(C(CO)C(C)C)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E06 compound treatment 209440.0 22900.0 1.56 203280.0 22500.0 1.67 2.2882 0.9994 3189375 PK04_101088 CC(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E07 compound treatment 219920.0 33400.0 2.28 201280.0 20500.0 1.52 2.6882 0.9808 3189376 PK04_101089 CC(C)C(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCOC(=O)[C@@H]6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E08 compound treatment 217160.0 30700.0 2.09 209080.0 28300.0 2.1 2.9656 1.0 3069762 PK04_101090 CCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E09 mock treatment 191800.0 5300.0 0.36 181040.0 222.0 0.02 0.2674 0.7386 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E10 mock treatment 186600.0 104.0 0.01 184880.0 4060.0 0.3 0.2188 0.7235 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E11 compound treatment 215240.0 28700.0 1.96 206560.0 25700.0 1.92 2.7404 0.9999 3189377 PK04_101091 CCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(C(CO)C(C)C)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E12 compound treatment 221480.0 35000.0 2.39 209840.0 29000.0 2.16 3.2139 0.9988 3069763 PK04_101092 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E13 compound treatment 219040.0 32500.0 2.22 206120.0 25300.0 1.88 2.9005 0.9967 3189378 PK04_101093 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E14 compound treatment 213480.0 27000.0 1.84 205600.0 24800.0 1.84 2.6051 1.0 3189379 PK04_101094 CC(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E15 compound treatment 220360.0 33900.0 2.31 211040.0 30200.0 2.25 3.223 0.9999 3069764 PK04_101095 CC(C)C(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E16 compound treatment 219720.0 33200.0 2.27 216720.0 35900.0 2.67 3.4911 0.9966 3189380 PK04_101096 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E17 mock treatment 184560.0 -1940.0 -0.13 177360.0 -3460.0 -0.26 -0.2753 -0.9519 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E18 mock treatment 182440.0 -4060.0 -0.28 182440.0 1620.0 0.12 -0.1102 -0.3651 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E19 compound treatment 203240.0 16700.0 1.14 190680.0 9860.0 0.73 1.3262 0.9772 3069765 PK04_101097 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E20 compound treatment 219280.0 32800.0 2.24 202160.0 21300.0 1.59 2.7036 0.986 3189381 PK04_101098 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E21 compound treatment 209000.0 22500.0 1.53 198400.0 17600.0 1.31 2.0102 0.9969 3189382 PK04_101099 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E22 compound treatment 204920.0 18400.0 1.26 202680.0 21900.0 1.63 2.0387 0.9918 3069730 PK04_101100 CC(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E23 compound treatment 202080.0 15600.0 1.06 196040.0 15200.0 1.13 1.5524 0.9995 3069766 PK04_101101 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C(=O)N(C(CO)C(C)C)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 E24 compound treatment 196680.0 10200.0 0.69 169720.0 -11100.0 -0.83 -0.0931 -0.0863 3069731 PK04_101102 CC(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F01 mock treatment 177680.0 -8820.0 -0.6 174600.0 -6220.0 -0.46 -0.7522 -0.9917 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F02 mock treatment 101000.0 -85500.0 -5.83 111080.0 -69700.0 -5.19 -7.7918 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F03 compound treatment 218880.0 32400.0 2.21 206080.0 25300.0 1.88 2.8907 0.9968 3189383 PK04_101103 CC1CC/C=C\[C@H]2OC34C=CCN(Cn5nnc6ccccc56)C(=O)[C@H]4N(CCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F04 compound treatment 193840.0 7340.0 0.5 186360.0 5540.0 0.41 0.6457 0.9954 3189267 PK04_101104 OCCOCCN1C(C(=O)N(CC=C)Cc2ccccc2)C3(OC4C=C3)C(C4C(=O)O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F05 compound treatment 219680.0 33200.0 2.26 204840.0 24000.0 1.79 2.864 0.9932 3189384 PK04_101105 CCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F06 compound treatment 190720.0 4220.0 0.29 179080.0 -1740.0 -0.13 0.1122 0.3553 3069767 PK04_101106 CCCCN(CC=C)C(=O)C1N(CCOCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F07 compound treatment 216080.0 29600.0 2.02 201880.0 21100.0 1.57 2.5346 0.9922 3189385 PK04_101107 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCO)C(=O)[C@@H]3C2C(=O)O1)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F08 compound treatment 193080.0 6580.0 0.45 183760.0 2940.0 0.22 0.4722 0.9455 3069767 PK04_101108 CCCCN(CC=C)C(=O)C1N(CCOCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F09 mock treatment 190560.0 4060.0 0.28 185240.0 4420.0 0.33 0.4286 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F10 mock treatment 185960.0 -536.0 -0.04 185360.0 4540.0 0.34 0.2132 0.627 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F11 compound treatment 219200.0 32700.0 2.23 205960.0 25100.0 1.87 2.8998 0.9962 3069768 PK04_101109 CC1CC/C=C\[C@H]2OC34C=CCN(CCN5CCOCC5)C(=O)[C@H]4N(CCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F12 compound treatment 194760.0 8260.0 0.56 184080.0 3260.0 0.24 0.5701 0.9292 3189386 PK04_101110 CCCCCN(CC=C)C(=O)C1N(CCOCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F13 compound treatment 219800.0 33300.0 2.27 207560.0 26700.0 1.99 3.0129 0.9978 3189387 PK04_101111 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCO)C(=O)[C@@H]3C2C(=O)O1)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F14 compound treatment 194640.0 8140.0 0.56 190480.0 9660.0 0.72 0.9011 0.9918 3189386 PK04_101112 CCCCCN(CC=C)C(=O)C1N(CCOCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F15 compound treatment 212200.0 25700.0 1.75 206240.0 25400.0 1.89 2.5771 0.9993 3069769 PK04_101113 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCO)C(=O)[C@]3(C)C2C(=O)O1)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F16 compound treatment 194000.0 7500.0 0.51 179840.0 -978.0 -0.07 0.3103 0.6005 3189388 PK04_101114 CC(C)(C)N(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F17 mock treatment 184640.0 -1860.0 -0.13 181040.0 222.0 0.02 -0.0778 -0.6096 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F18 mock treatment 181800.0 -4700.0 -0.32 171480.0 -9340.0 -0.69 -0.7178 -0.9381 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F19 compound treatment 215480.0 29000.0 1.98 209680.0 28900.0 2.15 2.9162 0.9991 3189389 PK04_101115 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C(=O)N(CCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F20 compound treatment 95960.0 -90500.0 -6.17 98400.0 -82400.0 -6.13 -8.7021 -1.0 3189388 PK04_101116 CC(C)(C)N(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F21 compound treatment 204520.0 18000.0 1.23 192320.0 11500.0 0.86 1.4742 0.9844 3069770 PK04_101117 OCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F22 compound treatment 99360.0 -87100.0 -5.94 94040.0 -86800.0 -6.46 -8.7676 -0.9991 3189390 PK04_101118 COc1ccc(cc1)N(CC=C)C(=O)C2N(C(=O)C3C(C4OC23C=C4)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F23 compound treatment 206520.0 20000.0 1.37 191080.0 10300.0 0.76 1.5054 0.9623 3189391 PK04_101119 CC(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 F24 compound treatment 118840.0 -67700.0 -4.61 103480.0 -77300.0 -5.76 -7.3317 -0.994 3189390 PK04_101120 COc1ccc(cc1)N(CC=C)C(=O)C2N(C(=O)C3C(C4OC23C=C4)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G01 compound treatment 203120.0 16600.0 1.13 193920.0 13100.0 0.98 1.4909 0.9972 3189392 PK04_101121 CC(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G02 compound treatment 211560.0 25100.0 1.71 207320.0 26500.0 1.97 2.603 0.9974 3189374 PK04_101122 CCCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G03 mock treatment 195840.0 9340.0 0.64 185240.0 4420.0 0.33 0.6832 0.9528 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G04 mock treatment 200480.0 14000.0 0.95 185200.0 4380.0 0.33 0.9048 0.8979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G05 compound treatment 222920.0 36400.0 2.48 207360.0 26500.0 1.98 3.1528 0.9936 3069794 PK04_101123 CC(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G06 compound treatment 222840.0 36300.0 2.48 213280.0 32500.0 2.42 3.4605 0.9999 3189375 PK04_101124 CC(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G07 compound treatment 222760.0 36300.0 2.47 208560.0 27700.0 2.06 3.2082 0.996 3189393 PK04_101125 CCCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G08 compound treatment 222720.0 36200.0 2.47 210000.0 29200.0 2.17 3.2821 0.9979 3069762 PK04_101126 CCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G09 compound treatment 211400.0 24900.0 1.7 199720.0 18900.0 1.41 2.1954 0.9956 3069795 PK04_101127 CC(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCOC(=O)[C@@H]6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G10 compound treatment 228800.0 42300.0 2.88 216760.0 35900.0 2.68 3.931 0.9993 3069763 PK04_101128 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G11 compound treatment 227240.0 40700.0 2.78 214480.0 33700.0 2.51 3.7358 0.9987 3189504 PK04_101129 CCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G12 compound treatment 218720.0 32200.0 2.2 216160.0 35300.0 2.63 3.4134 0.996 3189379 PK04_101130 CC(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G13 compound treatment 209800.0 23300.0 1.59 207480.0 26700.0 1.98 2.5266 0.9939 3069796 PK04_101131 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G14 compound treatment 225720.0 39200.0 2.67 211400.0 30600.0 2.28 3.5004 0.9968 3189380 PK04_101132 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G15 compound treatment 221480.0 35000.0 2.39 203440.0 22600.0 1.68 2.8771 0.9855 3189505 PK04_101133 CC(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G16 compound treatment 228800.0 42300.0 2.88 212680.0 31900.0 2.37 3.7162 0.9953 3189381 PK04_101134 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G17 compound treatment 209600.0 23100.0 1.58 205080.0 24300.0 1.81 2.3907 0.9977 3189506 PK04_101135 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G18 compound treatment 230480.0 44000.0 3.0 223120.0 42300.0 3.15 4.3467 0.9997 3069797 PK04_101136 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCCOC(=O)C5[C@H]4C(=O)N(C(C)CO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G19 mock treatment 188000.0 1500.0 0.1 184240.0 3420.0 0.25 0.2526 0.92 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G20 mock treatment 186520.0 24.0 0.0 178200.0 -2620.0 -0.19 -0.1366 -0.7011 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G21 compound treatment 203200.0 16700.0 1.14 185840.0 5020.0 0.37 1.0696 0.8924 3189507 PK04_101137 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G22 compound treatment 209280.0 22800.0 1.55 203200.0 22400.0 1.67 2.2763 0.9994 3189508 PK04_101138 CC(C)C(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G23 compound treatment 211400.0 24900.0 1.7 200480.0 19700.0 1.46 2.2353 0.9973 3069798 PK04_101139 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C(=O)N(C(C)CO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 G24 compound treatment 197720.0 11200.0 0.77 188920.0 8100.0 0.6 0.9675 0.993 3189509 PK04_101140 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H01 compound treatment 209720.0 23200.0 1.58 199640.0 18800.0 1.4 2.1102 0.9981 3069799 PK04_101141 CCCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H02 compound treatment 142200.0 -44300.0 -3.02 146480.0 -34300.0 -2.56 -3.9426 -0.9966 3189510 PK04_101142 CC(C)(CO)N1C(C(=O)N(CC=C)Cc2ccccc2)C3(OC4C=C3)C(C4C(=O)O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H03 mock treatment 185480.0 -1020.0 -0.07 181480.0 662.0 0.05 -0.0141 -0.1663 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H04 mock treatment 121440.0 -65100.0 -4.44 127600.0 -53200.0 -3.96 -5.937 -0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H05 compound treatment 217000.0 30500.0 2.08 213400.0 32600.0 2.42 3.1853 0.9971 3189511 PK04_101143 OCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H06 compound treatment 194600.0 8100.0 0.55 190680.0 9860.0 0.73 0.9097 0.9902 3069800 PK04_101144 CCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H07 compound treatment 218280.0 31800.0 2.17 218480.0 37700.0 2.8 3.5143 0.9919 3189512 PK04_101145 CCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H08 compound treatment 194480.0 7980.0 0.54 188280.0 7460.0 0.56 0.7776 0.9999 3069800 PK04_101146 CCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H09 compound treatment 213440.0 26900.0 1.84 205960.0 25100.0 1.87 2.6221 1.0 3189513 PK04_101147 CC(C)(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H10 compound treatment 197720.0 11200.0 0.77 190720.0 9900.0 0.74 1.0622 0.9998 3189510 PK04_101148 CC(C)(CO)N1C(C(=O)N(CC=C)Cc2ccccc2)C3(OC4C=C3)C(C4C(=O)O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H11 compound treatment 220440.0 33900.0 2.31 214320.0 33500.0 2.49 3.3995 0.9993 3069801 PK04_101149 OCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H12 compound treatment 197320.0 10800.0 0.74 188440.0 7620.0 0.57 0.9229 0.9916 3189514 PK04_101150 CCCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H13 compound treatment 219120.0 32600.0 2.22 210480.0 29700.0 2.21 3.1338 1.0 3189515 PK04_101151 OCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H14 compound treatment 195680.0 9180.0 0.63 188760.0 7940.0 0.59 0.8607 0.9996 3189514 PK04_101152 CCCCCN(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)C(C)(C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H15 compound treatment 216960.0 30500.0 2.08 208840.0 28000.0 2.09 2.9434 1.0 3069802 PK04_101153 C[C@]12C3[C@H](OC24C=CCN(C(=O)[C@H]4N(CCCO)C1=O)c5ccc(Cl)cc5)/C=C\CCCOC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H16 compound treatment 192200.0 5700.0 0.39 190800.0 9980.0 0.74 0.8003 0.9544 3189516 PK04_101154 CC(C)(C)N(CC=C)C(=O)C1N(CCCCCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H17 compound treatment 233560.0 47100.0 3.21 223440.0 42600.0 3.17 4.512 1.0 3189517 PK04_101155 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C(=O)N(CCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H18 compound treatment 148400.0 -38100.0 -2.6 148880.0 -31900.0 -2.38 -3.5174 -0.999 3189516 PK04_101156 CC(C)(C)N(CC=C)C(=O)C1N(CCCCCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H19 mock treatment 186600.0 104.0 0.01 186200.0 5380.0 0.4 0.2883 0.7195 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H20 mock treatment 176720.0 -9780.0 -0.67 167560.0 -13300.0 -0.99 -1.169 -0.9817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H21 compound treatment 212720.0 26200.0 1.79 205480.0 24700.0 1.84 2.5621 0.9999 3069803 PK04_101157 OCCCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H22 compound treatment 79800.0 -107000.0 -7.27 81920.0 -98900.0 -7.36 -10.3484 -1.0 3189518 PK04_101158 COc1ccc(cc1)N(CC=C)C(=O)C2N(CCCCCCO)C(=O)C3C(C4OC23C=C4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H23 compound treatment 198920.0 12400.0 0.85 197960.0 17100.0 1.28 1.5011 0.9802 3069804 PK04_101159 CC(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 H24 compound treatment 94480.0 -92000.0 -6.27 95880.0 -84900.0 -6.32 -8.906 -1.0 3189518 PK04_101160 COc1ccc(cc1)N(CC=C)C(=O)C2N(CCCCCCO)C(=O)C3C(C4OC23C=C4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I01 compound treatment 216760.0 30300.0 2.06 209120.0 28300.0 2.11 2.9484 0.9999 3189519 PK04_101161 OCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I02 compound treatment 214640.0 28100.0 1.92 203680.0 22900.0 1.7 2.56 0.9982 3189520 PK04_101162 CCCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(C(CO)C(C)C)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I03 compound treatment 225960.0 39500.0 2.69 215440.0 34600.0 2.58 3.7246 0.9998 3069839 PK04_101163 CC(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I04 compound treatment 219080.0 32600.0 2.22 212480.0 31700.0 2.36 3.2371 0.9996 3189521 PK04_101164 CC(C)C(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I05 mock treatment 194680.0 8180.0 0.56 189360.0 8540.0 0.64 0.8441 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I06 mock treatment 197160.0 10700.0 0.73 189320.0 8500.0 0.63 0.9615 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I07 compound treatment 226840.0 40300.0 2.75 226000.0 45200.0 3.36 4.3227 0.995 3069840 PK04_101165 CCCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I08 compound treatment 224320.0 37800.0 2.58 215000.0 34200.0 2.54 3.6224 1.0 3189522 PK04_101166 CCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(C(CO)C(C)C)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I09 compound treatment 232840.0 46300.0 3.16 220720.0 39900.0 2.97 4.3341 0.9995 3189523 PK04_101167 OCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCOC(=O)[C@@H]6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I10 compound treatment 222560.0 36100.0 2.46 212080.0 31300.0 2.33 3.3838 0.9996 3069841 PK04_101168 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I11 compound treatment 226440.0 39900.0 2.72 216840.0 36000.0 2.68 3.8214 1.0 3189524 PK04_101169 CCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I12 compound treatment 225360.0 38900.0 2.65 220320.0 39500.0 2.94 3.9525 0.9987 3189640 PK04_101170 CC(C)C(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I13 compound treatment 234000.0 47500.0 3.24 217920.0 37100.0 2.76 4.2427 0.9969 3069842 PK04_101171 CC(C)(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I14 compound treatment 215360.0 28900.0 1.97 214240.0 33400.0 2.49 3.1504 0.9933 3189641 PK04_101172 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I15 compound treatment 227360.0 40900.0 2.79 218480.0 37700.0 2.8 3.9521 1.0 3069843 PK04_101173 OCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I16 compound treatment 219920.0 33400.0 2.28 211960.0 31100.0 2.32 3.2502 1.0 3189642 PK04_101174 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@@]3(C)C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I17 compound treatment 234800.0 48300.0 3.29 218120.0 37300.0 2.78 4.2918 0.9964 3069844 PK04_101175 OCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I18 compound treatment 227080.0 40600.0 2.77 210400.0 29600.0 2.2 3.5133 0.9936 3189643 PK04_101176 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C(=O)N(C(CO)C(C)C)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I19 compound treatment 212880.0 26400.0 1.8 202600.0 21800.0 1.62 2.4183 0.9987 3069845 PK04_101177 OCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I20 compound treatment 209120.0 22600.0 1.54 203240.0 22400.0 1.67 2.2707 0.9992 3189644 PK04_101178 CC(C)C(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I21 mock treatment 189600.0 3100.0 0.21 180080.0 -738.0 -0.05 0.1108 0.5068 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I22 mock treatment 182040.0 -4460.0 -0.3 174520.0 -6300.0 -0.47 -0.5463 -0.978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I23 compound treatment 221320.0 34800.0 2.37 213880.0 33100.0 2.46 3.4188 0.9998 3189645 PK04_101179 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C(=O)N(CCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 I24 compound treatment 188880.0 2380.0 0.16 191920.0 11100.0 0.83 0.6992 0.8303 3069846 PK04_101180 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C1=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J01 compound treatment 209120.0 22600.0 1.54 201280.0 20500.0 1.52 2.1675 1.0 3189646 PK04_101181 CCCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J02 compound treatment 110160.0 -76300.0 -5.2 110160.0 -70700.0 -5.26 -7.3986 -1.0 3189647 PK04_101182 OCCCCCCN1C(C(=O)N(CC=C)Cc2ccccc2)C3(OC4C=C3)C(C4C(=O)O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J03 compound treatment 220200.0 33700.0 2.3 207800.0 27000.0 2.01 3.0448 0.9977 3069847 PK04_101183 OCCCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J04 compound treatment 193560.0 7060.0 0.48 185280.0 4460.0 0.33 0.5754 0.9835 3189647 PK04_101184 OCCCCCCN1C(C(=O)N(CC=C)Cc2ccccc2)C3(OC4C=C3)C(C4C(=O)O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J05 mock treatment 194000.0 7500.0 0.51 181920.0 1100.0 0.08 0.4198 0.8101 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J06 mock treatment 191440.0 4940.0 0.34 180920.0 102.0 0.01 0.2437 0.7228 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J07 compound treatment 219280.0 32800.0 2.24 214200.0 33400.0 2.48 3.3373 0.9986 3189648 PK04_101185 CCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J08 compound treatment 195720.0 9220.0 0.63 190920.0 10100.0 0.75 0.9763 0.9961 3189649 PK04_101186 CCCCN(CC=C)C(=O)C1N(CCCCCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J09 compound treatment 223840.0 37300.0 2.55 219560.0 38700.0 2.88 3.8392 0.9981 3069848 PK04_101187 CC(C)(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J10 compound treatment 196640.0 10100.0 0.69 196240.0 15400.0 1.15 1.3007 0.9706 3189649 PK04_101188 CCCCN(CC=C)C(=O)C1N(CCCCCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J11 compound treatment 221520.0 35000.0 2.39 212480.0 31700.0 2.36 3.3547 1.0 3189650 PK04_101189 OCCCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J12 compound treatment 196040.0 9540.0 0.65 184760.0 3940.0 0.29 0.6676 0.9353 3189651 PK04_101190 CCCCCN(CC=C)C(=O)C1N(CCCCCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J13 compound treatment 222120.0 35600.0 2.43 209440.0 28600.0 2.13 3.2237 0.9979 3069849 PK04_101191 OCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J14 compound treatment 197680.0 11200.0 0.76 191840.0 11000.0 0.82 1.1192 0.9993 3189651 PK04_101192 CCCCCN(CC=C)C(=O)C1N(CCCCCCO)C(=O)C2C(C3OC12C=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J15 compound treatment 215520.0 29000.0 1.98 207480.0 26700.0 1.98 2.8024 1.0 3189652 PK04_101193 C[C@]12C3[C@H](OC24C=CCN(C(=O)[C@H]4N(CCCCCO)C1=O)c5ccc(Cl)cc5)/C=C\CCCOC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J16 compound treatment 199280.0 12800.0 0.87 191000.0 10200.0 0.76 1.1522 0.9976 3069850 PK04_101194 CC(C)(C)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1c(Cl)cccc1CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J17 compound treatment 217840.0 31300.0 2.14 212360.0 31500.0 2.35 3.171 0.9989 3189653 PK04_101195 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C(=O)N(CCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J18 compound treatment 102120.0 -84400.0 -5.75 112120.0 -68700.0 -5.11 -7.683 -0.9983 3069850 PK04_101196 CC(C)(C)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1c(Cl)cccc1CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J19 compound treatment 208480.0 22000.0 1.5 197760.0 16900.0 1.26 1.9514 0.9963 3189654 PK04_101197 CC1CC/C=C\[C@H]2OC34C=CCN(Cc5ccccc5)C(=O)[C@H]4N(CCCCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J20 compound treatment 89800.0 -96700.0 -6.59 93120.0 -87700.0 -6.53 -9.2769 -1.0 3069851 PK04_101198 COc1ccc(cc1)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c2c(Cl)cccc2CO)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J21 mock treatment 183840.0 -2660.0 -0.18 174840.0 -5980.0 -0.44 -0.4427 -0.9215 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J22 mock treatment 75080.0 -111000.0 -7.6 77800.0 -103000.0 -7.67 -10.7928 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J23 compound treatment 201640.0 15100.0 1.03 190880.0 10100.0 0.75 1.2596 0.9876 3189655 PK04_101199 CC(C)N1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 J24 compound treatment 93440.0 -93100.0 -6.34 90800.0 -90000.0 -6.7 -9.2235 -0.9996 3069851 PK04_101200 COc1ccc(cc1)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c2c(Cl)cccc2CO)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K01 compound treatment 214880.0 28400.0 1.94 206320.0 25500.0 1.9 2.7105 1.0 3189656 PK04_101201 OCCCCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K02 compound treatment 207200.0 20700.0 1.41 206360.0 25500.0 1.9 2.3423 0.9893 3189657 PK04_101202 CCCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(C(CO)C(C)C)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K03 compound treatment 223760.0 37300.0 2.54 206800.0 26000.0 1.93 3.1638 0.9909 3069890 PK04_101203 CC(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K04 compound treatment 226440.0 39900.0 2.72 215080.0 34300.0 2.55 3.7288 0.9995 3189658 PK04_101204 CC(C)C(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCC(C)OC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K05 compound treatment 219560.0 33100.0 2.25 208960.0 28100.0 2.09 3.075 0.9993 3069891 PK04_101205 CCCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K06 compound treatment 216560.0 30100.0 2.05 207320.0 26500.0 1.97 2.8441 0.9998 3189659 PK04_101206 CCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(C(CO)C(C)C)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K07 mock treatment 196760.0 10300.0 0.7 186240.0 5420.0 0.4 0.7802 0.9658 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K08 mock treatment 191320.0 4820.0 0.33 187040.0 6220.0 0.46 0.56 0.9859 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K09 compound treatment 228920.0 42400.0 2.89 222280.0 41500.0 3.09 4.2272 0.9995 3187684 PK04_101207 OCCCCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCOC(=O)[C@@H]6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K10 compound treatment 217320.0 30800.0 2.1 218320.0 37500.0 2.79 3.4596 0.9902 3069892 PK04_101208 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K11 compound treatment 217000.0 30500.0 2.08 215040.0 34200.0 2.55 3.2716 0.9949 3187685 PK04_101209 CCCCN1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K12 compound treatment 222680.0 36200.0 2.47 218160.0 37300.0 2.78 3.7096 0.9982 3187686 PK04_101210 CC(C)C(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K13 compound treatment 221720.0 35200.0 2.4 213960.0 33100.0 2.47 3.4423 0.9999 3069893 PK04_101211 CC(C)(C)N1CC=CC23O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K14 compound treatment 217480.0 31000.0 2.11 210680.0 29900.0 2.22 3.0653 0.9997 3187687 PK04_101212 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K15 mock treatment 199280.0 12800.0 0.87 191640.0 10800.0 0.81 1.1858 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K16 mock treatment 200920.0 14400.0 0.98 183520.0 2700.0 0.2 0.8376 0.8344 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K17 compound treatment 225640.0 39100.0 2.67 220000.0 39200.0 2.92 3.9491 0.999 3069894 PK04_101213 OCCCCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K18 compound treatment 205520.0 19000.0 1.3 201280.0 20500.0 1.52 1.994 0.9968 3187688 PK04_101214 CC(C)C(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@@]3(C)C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K19 compound treatment 210720.0 24200.0 1.65 202120.0 21300.0 1.59 2.2889 0.9998 3069895 PK04_101215 OCCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K20 compound treatment 210880.0 24400.0 1.66 199920.0 19100.0 1.42 2.1808 0.997 3187689 PK04_101216 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C(=O)N(C(CO)C(C)C)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K21 compound treatment 198320.0 11800.0 0.81 201920.0 21100.0 1.57 1.6806 0.952 3187690 PK04_101217 OCCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCOC(=O)[C@@H]4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K22 compound treatment 211840.0 25300.0 1.73 195640.0 14800.0 1.1 2.0018 0.9765 3069896 PK04_101218 CC(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K23 mock treatment 182120.0 -4380.0 -0.3 175280.0 -5540.0 -0.41 -0.5024 -0.9874 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 K24 mock treatment 179520.0 -6980.0 -0.48 166680.0 -14100.0 -1.05 -1.0804 -0.9356 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L01 compound treatment 211040.0 24500.0 1.67 204080.0 23300.0 1.73 2.4075 0.9999 3187691 PK04_101219 CCCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L02 compound treatment 181800.0 -4700.0 -0.32 176440.0 -4380.0 -0.33 -0.4568 -1.0 3187692 PK04_101220 OCc1cccc(Cl)c1N(C(C(=O)N(CC=C)Cc2ccccc2)c3cccs3)C(=O)/C=C\C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L03 compound treatment 214680.0 28200.0 1.92 208640.0 27800.0 2.07 2.8229 0.9993 3069897 PK04_101221 CC1CC/C=C\[C@H]2OC34C=CCN(Cn5nnc6ccccc56)C(=O)[C@H]4N(CCCCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L04 compound treatment 190120.0 3620.0 0.25 189200.0 8380.0 0.62 0.6158 0.9178 3187693 PK04_101222 CCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1c(Cl)cccc1CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L05 compound treatment 213080.0 26600.0 1.81 211320.0 30500.0 2.27 2.8868 0.9938 3187694 PK04_101223 CCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L06 compound treatment 190160.0 3660.0 0.25 184560.0 3740.0 0.28 0.3736 0.9985 3187693 PK04_101224 CCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1c(Cl)cccc1CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L07 mock treatment 190400.0 3900.0 0.27 184800.0 3980.0 0.3 0.3978 0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L08 mock treatment 189200.0 2700.0 0.18 189520.0 8700.0 0.65 0.5883 0.8737 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L09 compound treatment 219400.0 32900.0 2.24 216160.0 35300.0 2.63 3.4462 0.9969 3069898 PK04_101225 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCCCO)C(=O)[C@@H]3C2C(=O)O1)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L10 compound treatment 194400.0 7900.0 0.54 190400.0 9580.0 0.71 0.8853 0.9904 3187692 PK04_101226 OCc1cccc(Cl)c1N(C(C(=O)N(CC=C)Cc2ccccc2)c3cccs3)C(=O)/C=C\C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L11 compound treatment 219480.0 33000.0 2.25 221480.0 40700.0 3.03 3.7301 0.9893 3187695 PK04_101227 CC1CC/C=C\[C@H]2OC34C=CCN(CCN5CCOCC5)C(=O)[C@H]4N(CCCCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L12 compound treatment 196440.0 9940.0 0.68 189800.0 8980.0 0.67 0.9521 1.0 3187696 PK04_101228 CCCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1c(Cl)cccc1CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L13 compound treatment 216080.0 29600.0 2.02 207280.0 26500.0 1.97 2.8188 0.9999 3069899 PK04_101229 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCCCO)C(=O)[C@@H]3C2C(=O)O1)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L14 compound treatment 194640.0 8140.0 0.56 191000.0 10200.0 0.76 0.9285 0.9883 3187696 PK04_101230 CCCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1c(Cl)cccc1CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L15 mock treatment 195040.0 8540.0 0.58 185840.0 5020.0 0.37 0.6762 0.977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L16 mock treatment 175320.0 -11200.0 -0.76 172080.0 -8740.0 -0.65 -0.9986 -0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L17 compound treatment 206840.0 20300.0 1.39 202960.0 22100.0 1.65 2.146 0.9963 3187697 PK04_101231 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCCCO)C(=O)[C@]3(C)C2C(=O)O1)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L18 compound treatment 101080.0 -85400.0 -5.82 102200.0 -78600.0 -5.85 -8.2553 -1.0 3187698 PK04_101232 CC(C)(C)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1ccc(CCO)cc1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L19 compound treatment 218160.0 31700.0 2.16 205200.0 24400.0 1.81 2.8096 0.9963 3069900 PK04_101233 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C(=O)N(CCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L20 compound treatment 77280.0 -109000.0 -7.45 75680.0 -105000.0 -7.83 -10.7983 -0.9997 3187698 PK04_101234 CC(C)(C)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1ccc(CCO)cc1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L21 compound treatment 208480.0 22000.0 1.5 201240.0 20400.0 1.52 2.1346 1.0 3187699 PK04_101235 CC1CC/C=C\[C@H]2OC34C=CCN(Cc5ccccc5)C(=O)[C@H]4N(CCCCCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L22 compound treatment 82040.0 -104000.0 -7.12 83760.0 -97100.0 -7.22 -10.1436 -1.0 3187700 PK04_101236 COc1ccc(cc1)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c2ccc(CCO)cc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L23 mock treatment 176960.0 -9540.0 -0.65 171600.0 -9220.0 -0.69 -0.9448 -0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 L24 mock treatment 89040.0 -97500.0 -6.64 91600.0 -89200.0 -6.64 -9.3935 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M01 compound treatment 224200.0 37700.0 2.57 211640.0 30800.0 2.29 3.4397 0.9984 3187701 PK04_101237 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCOC(=O)[C@@H]5[C@H]4C(=O)N(CCCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M02 compound treatment 229480.0 43000.0 2.93 227840.0 47000.0 3.5 4.5469 0.9961 3069926 PK04_101238 CC(C)N1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M03 compound treatment 217520.0 31000.0 2.12 217760.0 36900.0 2.75 3.4398 0.9916 3187702 PK04_101239 OCCCCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M04 compound treatment 222280.0 35800.0 2.44 214560.0 33700.0 2.51 3.5009 0.9999 3069927 PK04_101240 CCCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M05 compound treatment 225840.0 39300.0 2.68 211760.0 30900.0 2.3 3.5251 0.9971 3187703 PK04_101241 CC(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M06 compound treatment 226120.0 39600.0 2.7 218880.0 38100.0 2.83 3.9133 0.9997 3187824 PK04_101242 CC(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCC(C)OC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M07 compound treatment 222080.0 35600.0 2.43 213480.0 32700.0 2.43 3.4344 1.0 3069928 PK04_101243 CCCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M08 compound treatment 229480.0 43000.0 2.93 226080.0 45300.0 3.37 4.4542 0.9976 3187825 PK04_101244 CCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M09 mock treatment 200640.0 14100.0 0.96 191880.0 11100.0 0.82 1.264 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M10 mock treatment 195360.0 8860.0 0.6 192040.0 11200.0 0.84 1.0179 0.9874 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M11 compound treatment 221040.0 34500.0 2.36 225720.0 44900.0 3.34 4.0284 0.9853 3187826 PK04_101245 OCCCCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M12 compound treatment 231800.0 45300.0 3.09 222800.0 42000.0 3.12 4.3934 1.0 3069929 PK04_101246 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M13 mock treatment 204280.0 17800.0 1.21 194160.0 13300.0 0.99 1.5595 0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M14 mock treatment 192600.0 6100.0 0.42 189320.0 8500.0 0.63 0.7417 0.9793 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M15 compound treatment 223280.0 36800.0 2.51 215440.0 34600.0 2.58 3.5954 0.9999 3187827 PK04_101247 CCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M16 compound treatment 226440.0 39900.0 2.72 220480.0 39700.0 2.95 4.013 0.9992 3187828 PK04_101248 CC(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M17 compound treatment 215880.0 29400.0 2.0 205720.0 24900.0 1.85 2.7271 0.9992 3069930 PK04_101249 CC(C)(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M18 compound treatment 234240.0 47700.0 3.26 213400.0 32600.0 2.42 4.0164 0.9895 3187829 PK04_101250 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M19 compound treatment 216960.0 30500.0 2.08 214480.0 33700.0 2.51 3.2402 0.9957 3069931 PK04_101251 OCCCCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M20 compound treatment 208840.0 22300.0 1.52 205520.0 24700.0 1.84 2.3772 0.9956 3187830 PK04_101252 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@@]3(C)C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M21 compound treatment 208600.0 22100.0 1.51 204280.0 23500.0 1.75 2.3003 0.9973 3187831 PK04_101253 OCCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M22 compound treatment 213760.0 27300.0 1.86 213160.0 32300.0 2.41 3.0164 0.9918 3069932 PK04_101254 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C(=O)N(C(C)CO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M23 compound treatment 206280.0 19800.0 1.35 202040.0 21200.0 1.58 2.0706 0.9969 3187832 PK04_101255 OCCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 M24 compound treatment 199200.0 12700.0 0.87 193920.0 13100.0 0.98 1.302 0.9983 3187833 PK04_101256 CC(CO)N1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N01 compound treatment 218280.0 31800.0 2.17 216120.0 35300.0 2.63 3.3901 0.9954 3069933 PK04_101257 CC(C)N1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N02 compound treatment 168640.0 -17900.0 -1.22 167640.0 -13200.0 -0.98 -1.5543 -0.9943 3187700 PK04_101258 COc1ccc(cc1)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c2ccc(CCO)cc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N03 compound treatment 212720.0 26200.0 1.79 216840.0 36000.0 2.68 3.16 0.9806 3187834 PK04_101259 CCCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N04 compound treatment 196520.0 10000.0 0.68 184880.0 4060.0 0.3 0.697 0.9327 3069934 PK04_101260 OCCc1ccc(cc1)N(C(C(=O)N(CC=C)Cc2ccccc2)c3cccs3)C(=O)/C=C\C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N05 compound treatment 216520.0 30000.0 2.05 221080.0 40300.0 3.0 3.5663 0.9827 3187835 PK04_101261 CC1CC/C=C\[C@H]2OC34C=CCN(Cn5nnc6ccccc56)C(=O)[C@H]4N(CCCCCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N06 compound treatment 195280.0 8780.0 0.6 192280.0 11500.0 0.85 1.0267 0.985 3069934 PK04_101262 OCCc1ccc(cc1)N(C(C(=O)N(CC=C)Cc2ccccc2)c3cccs3)C(=O)/C=C\C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N07 compound treatment 222760.0 36300.0 2.47 222400.0 41600.0 3.09 3.9366 0.9938 3187836 PK04_101263 CCCCN1CC=CC23O[C@@H]4/C=C\CCC(C)OC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N08 compound treatment 198000.0 11500.0 0.78 198320.0 17500.0 1.3 1.4757 0.9705 3069935 PK04_101264 CCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1ccc(CCO)cc1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N09 mock treatment 195520.0 9020.0 0.62 191880.0 11100.0 0.82 1.0172 0.9897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N10 mock treatment 194400.0 7900.0 0.54 186640.0 5820.0 0.43 0.6874 0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N11 compound treatment 217720.0 31200.0 2.13 222640.0 41800.0 3.11 3.7063 0.9828 3187837 PK04_101265 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCCCCO)C(=O)[C@@H]3C2C(=O)O1)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N12 compound treatment 209640.0 23100.0 1.58 200960.0 20100.0 1.5 2.1758 0.9997 3069935 PK04_101266 CCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1ccc(CCO)cc1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N13 mock treatment 197560.0 11100.0 0.75 191120.0 10300.0 0.77 1.0755 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N14 mock treatment 195200.0 8700.0 0.59 187200.0 6380.0 0.47 0.7555 0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N15 compound treatment 219080.0 32600.0 2.22 206960.0 26100.0 1.95 2.9466 0.9978 3069936 PK04_101267 CC1CC/C=C\[C@H]2OC34C=CCN(CCN5CCOCC5)C(=O)[C@H]4N(CCCCCCO)C(=O)[C@@H]3C2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N16 compound treatment 197520.0 11000.0 0.75 187120.0 6300.0 0.47 0.8631 0.9742 3187838 PK04_101268 CCCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1ccc(CCO)cc1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N17 compound treatment 218680.0 32200.0 2.19 213360.0 32500.0 2.42 3.2641 0.9988 3187839 PK04_101269 CC1CC/C=C\[C@H]2OC34C=CCN(C(=O)[C@H]4N(CCCCCCO)C(=O)[C@]3(C)C2C(=O)O1)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N18 compound treatment 199840.0 13300.0 0.91 188560.0 7740.0 0.58 1.0507 0.9757 3187838 PK04_101270 CCCCCN(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)c1ccc(CCO)cc1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N19 compound treatment 222040.0 35500.0 2.42 217400.0 36600.0 2.72 3.6387 0.9983 3187840 PK04_101271 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCC(C)OC(=O)C5[C@H]4C(=O)N(CCCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N20 compound treatment 170720.0 -15800.0 -1.08 167760.0 -13100.0 -0.97 -1.4477 -0.9987 3187841 PK04_101272 CC(C)(C)N(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N21 compound treatment 207360.0 20900.0 1.42 195480.0 14700.0 1.09 1.7774 0.9914 3069973 PK04_101273 OCCCCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N22 compound treatment 104160.0 -82300.0 -5.61 105520.0 -75300.0 -5.6 -7.932 -1.0 3187841 PK04_101274 CC(C)(C)N(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N23 compound treatment 194560.0 8060.0 0.55 194640.0 13800.0 1.03 1.1162 0.9569 3187842 PK04_101275 CC(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 N24 compound treatment 98400.0 -88100.0 -6.01 108360.0 -72500.0 -5.39 -8.0603 -0.9986 3187843 PK04_101276 COc1ccc(cc1)N(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O01 compound treatment 223000.0 36500.0 2.49 216760.0 35900.0 2.68 3.6513 0.9993 3069974 PK04_101277 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCCOC(=O)C5[C@H]4C(=O)N(CCCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O02 compound treatment 213080.0 26600.0 1.81 209560.0 28700.0 2.14 2.7942 0.9966 3187957 PK04_101278 CC(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O03 compound treatment 213440.0 26900.0 1.84 206320.0 25500.0 1.9 2.641 0.9999 3187958 PK04_101279 OCCCCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O04 compound treatment 218720.0 32200.0 2.2 213000.0 32200.0 2.4 3.2471 0.9991 3069975 PK04_101280 CCCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O05 compound treatment 214120.0 27600.0 1.88 214200.0 33400.0 2.48 3.0885 0.9907 3187959 PK04_101281 CC(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O06 compound treatment 210000.0 23500.0 1.6 205200.0 24400.0 1.81 2.4163 0.9981 3187960 PK04_101282 CC(CO)N1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O07 compound treatment 211760.0 25300.0 1.72 203000.0 22200.0 1.65 2.3853 0.9998 3069976 PK04_101283 CCCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O08 compound treatment 222240.0 35700.0 2.44 204080.0 23300.0 1.73 2.9474 0.986 3187961 PK04_101284 CCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(C(C)CO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O09 compound treatment 215920.0 29400.0 2.01 208520.0 27700.0 2.06 2.8764 0.9999 3069977 PK04_101285 OCCCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6C=CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O10 compound treatment 218200.0 31700.0 2.16 214680.0 33900.0 2.52 3.3105 0.9971 3187962 PK04_101286 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O11 mock treatment 186800.0 304.0 0.02 195080.0 14300.0 1.06 0.7652 0.7208 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O12 mock treatment 192920.0 6420.0 0.44 190280.0 9460.0 0.7 0.8077 0.9739 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O13 compound treatment 220360.0 33900.0 2.31 202400.0 21600.0 1.61 2.7683 0.9843 3187963 PK04_101287 CCCCN1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O14 compound treatment 217160.0 30700.0 2.09 208280.0 27500.0 2.04 2.9235 0.9999 3069978 PK04_101288 CC(CO)N1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O15 compound treatment 210360.0 23900.0 1.63 206880.0 26100.0 1.94 2.522 0.9962 3187964 PK04_101289 CC(C)(C)N1CC=CC23O[C@@H]4C=CCCOC(=O)C4[C@H]3C(=O)N(CCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O16 compound treatment 207240.0 20700.0 1.41 200440.0 19600.0 1.46 2.0327 0.9999 3187965 PK04_101290 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O17 compound treatment 219280.0 32800.0 2.24 211000.0 30200.0 2.25 3.1689 1.0 3069979 PK04_101291 OCCCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5C=CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O18 compound treatment 205880.0 19400.0 1.32 195600.0 14800.0 1.1 1.7124 0.9958 3187966 PK04_101292 CC(CO)N1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@@]3(C)C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O19 compound treatment 205560.0 19100.0 1.3 199800.0 19000.0 1.41 1.918 0.9991 3187967 PK04_101293 OCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O20 compound treatment 215280.0 28800.0 1.96 208080.0 27300.0 2.03 2.8224 0.9999 3069980 PK04_101294 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C(=O)N(C(C)CO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O21 compound treatment 206960.0 20500.0 1.4 202800.0 22000.0 1.64 2.1434 0.9969 3187968 PK04_101295 OCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4C=CCCOC(=O)C4[C@H]3C1=O)c5ccc(Cl)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O22 compound treatment 197080.0 10600.0 0.72 194240.0 13400.0 1.0 1.2166 0.9873 3069981 PK04_101296 OCCN1[C@@H]2C(=O)N(Cc3ccccc3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O23 compound treatment 200120.0 13600.0 0.93 205120.0 24300.0 1.81 1.9358 0.952 3187969 PK04_101297 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5C=CCCOC(=O)C5[C@H]4C(=O)N(CCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 O24 compound treatment 203000.0 16500.0 1.13 191000.0 10200.0 0.76 1.3315 0.9815 3187970 PK04_101298 CC(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P01 compound treatment 208080.0 21600.0 1.47 203000.0 22200.0 1.65 2.2079 0.9984 3069982 PK04_101299 CCCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P02 compound treatment 189520.0 3020.0 0.21 182240.0 1420.0 0.11 0.2206 0.952 3187843 PK04_101300 COc1ccc(cc1)N(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P03 compound treatment 207320.0 20800.0 1.42 207360.0 26500.0 1.98 2.4007 0.9869 3187971 PK04_101301 OCCCCCCN1[C@@H]2C(=O)N(Cn3nnc4ccccc34)CC=CC52O[C@@H]6/C=C\CCCOC(=O)C6[C@H]5C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P04 compound treatment 187560.0 1060.0 0.07 189480.0 8660.0 0.64 0.5072 0.7817 3069983 PK04_101302 OCCOCCN(C(C(=O)N(CC=C)Cc1ccccc1)c2cccs2)C(=O)/C=C\C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P05 compound treatment 203880.0 17400.0 1.19 197840.0 17000.0 1.27 1.7339 0.9994 3187972 PK04_101303 CCCCN1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P06 compound treatment 191160.0 4660.0 0.32 184960.0 4140.0 0.31 0.4428 0.9999 3187973 PK04_101304 OCCOCCc1ccc(cc1)N(C(C(=O)N(CC=C)Cc2ccccc2)c3cccs3)C(=O)/C=C\C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P07 compound treatment 207720.0 21200.0 1.45 197680.0 16900.0 1.25 1.9106 0.9975 3069985 PK04_101305 CC(C)(C)N1CC=CC23O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C(=O)N(CCCCCCO)[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P08 compound treatment 194280.0 7780.0 0.53 183600.0 2780.0 0.21 0.5217 0.9158 3187974 PK04_101306 CCCCN(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P09 compound treatment 210480.0 24000.0 1.64 213480.0 32700.0 2.43 2.8752 0.9814 3187975 PK04_101307 OCCCCCCN1[C@@H]2C(=O)N(CCN3CCOCC3)CC=CC42O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P10 compound treatment 186400.0 -96.0 -0.01 185920.0 5100.0 0.38 0.2639 0.6948 3187974 PK04_101308 CCCCN(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P11 mock treatment 183960.0 -2540.0 -0.17 188080.0 7260.0 0.54 0.2599 0.458 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P12 mock treatment 185520.0 -976.0 -0.07 188600.0 7780.0 0.58 0.3625 0.6218 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P13 compound treatment 203840.0 17300.0 1.18 205680.0 24900.0 1.85 2.1446 0.9766 3069986 PK04_101309 OCCCCCCN1[C@@H]2C(=O)N(CC=CC32O[C@@H]4/C=C\CCCOC(=O)C4[C@H]3C1=O)c5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P14 compound treatment 190280.0 3780.0 0.26 190520.0 9700.0 0.72 0.693 0.9038 3069301 PK04_101310 CCCCCN(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P15 compound treatment 200520.0 14000.0 0.96 197640.0 16800.0 1.25 1.5614 0.9911 3187976 PK04_101311 C[C@]12C3[C@H](OC24C=CCN(C(=O)[C@H]4N(CCCCCCO)C1=O)c5ccc(Cl)cc5)/C=C\CCCOC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P16 compound treatment 189800.0 3300.0 0.23 186920.0 6100.0 0.45 0.4804 0.9477 3069301 PK04_101312 CCCCCN(CC=C)C(=O)C(N(CCOCCO)C(=O)/C=C\C(=O)O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P17 compound treatment 208320.0 21800.0 1.49 203480.0 22700.0 1.69 2.2447 0.998 3187977 PK04_101313 CCN(CC)c1ccc(cc1)N2CC=CC34O[C@@H]5/C=C\CCCOC(=O)C5[C@H]4C(=O)N(CCCCCCO)[C@@H]3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P18 compound treatment 185920.0 -576.0 -0.04 183440.0 2620.0 0.2 0.1102 0.5537 3069302 PK04_101314 CC(C)(C)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)C(C)(C)CO)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P19 compound treatment 189080.0 2580.0 0.18 181840.0 1020.0 0.08 0.1784 0.9295 3189130 PK04_101315 CC(C)(C)N(CC=C)C(=O)C1N(C(=O)C2C(C3OC12C=C3)C(=O)O)c4c(Cl)cccc4CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P20 compound treatment 154000.0 -32500.0 -2.22 156160.0 -24700.0 -1.84 -2.8643 -0.9956 3069302 PK04_101316 CC(C)(C)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)C(C)(C)CO)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P21 compound treatment 176920.0 -9580.0 -0.65 178600.0 -2220.0 -0.17 -0.5784 -0.8589 3189131 PK04_101317 COc1ccc(cc1)N(CC=C)C(=O)C2N(C(=O)C3C(C4OC23C=C4)C(=O)O)c5c(Cl)cccc5CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P22 compound treatment 97120.0 -89400.0 -6.09 102800.0 -78000.0 -5.81 -8.4146 -0.9997 3069303 PK04_101318 COc1ccc(cc1)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)C(C)(C)CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P23 compound treatment 178760.0 -7740.0 -0.53 179280.0 -1540.0 -0.11 -0.4539 -0.841 3069685 PK04_101319 OCc1cccc(Cl)c1N2C(C(=O)N(CC=C)Cc3ccccc3)C4(OC5C=C4)C(C5C(=O)O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2101 P24 compound treatment 160960.0 -25500.0 -1.74 168080.0 -12700.0 -0.95 -1.9014 -0.9592 3069303 PK04_101320 COc1ccc(cc1)N(CC=C)C(=O)C(N(C(=O)/C=C\C(=O)O)C(C)(C)CO)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A01 compound treatment 213560.0 32500.0 2.21 212720.0 32400.0 2.41 3.2676 0.9991 3188092 PK04_102001 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A02 compound treatment 246160.0 65100.0 4.44 249440.0 69100.0 5.14 6.7717 0.9973 3188093 PK04_102002 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6CCCCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A03 compound treatment 256680.0 75600.0 5.15 252040.0 71700.0 5.33 7.4157 0.9999 3069304 PK04_102003 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccccc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A04 compound treatment 240040.0 58900.0 4.02 230240.0 49900.0 3.71 5.4662 0.9992 3188094 PK04_102004 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5ccc(cc5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A05 compound treatment 174360.0 -6740.0 -0.46 172120.0 -8250.0 -0.61 -0.7588 -0.9898 3069305 PK04_102005 COc1ccc(cc1)[Si](C)(C)[C@H](CC(=O)N2CCC[C@H]2CO)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A06 compound treatment 226520.0 45400.0 3.1 225440.0 45100.0 3.35 4.5618 0.9992 3188095 PK04_102006 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CCn5cc(nn5)[C@H](O)c6ccccc6)[C@H]([C@@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A07 compound treatment 239200.0 58100.0 3.96 241320.0 61000.0 4.54 6.0088 0.9977 3069306 PK04_102007 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(c5ccccc53)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A08 compound treatment 258760.0 77700.0 5.29 252640.0 72300.0 5.38 7.5475 1.0 3188096 PK04_102008 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(NC(=O)C)cc4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A09 compound treatment 224040.0 42900.0 2.93 225800.0 45400.0 3.38 4.4612 0.9974 3188097 PK04_102009 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(C)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A10 compound treatment 243840.0 62700.0 4.28 241400.0 61000.0 4.54 6.2367 0.9995 3069307 PK04_102010 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6CCOC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A11 compound treatment 207680.0 26600.0 1.81 210440.0 30100.0 2.24 2.8642 0.9945 3188098 PK04_102011 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(c6ccccc63)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A12 compound treatment 224880.0 43800.0 2.98 225000.0 44600.0 3.32 4.4596 0.9986 3069308 PK04_102012 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N(C=O)c5ccccc5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A13 mock treatment 167120.0 -14000.0 -0.95 170000.0 -10400.0 -0.77 -1.2194 -0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A14 mock treatment 169200.0 -11900.0 -0.81 167840.0 -12500.0 -0.93 -1.2328 -0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A15 compound treatment 204360.0 23300.0 1.59 214440.0 34100.0 2.54 2.9146 0.9744 3188099 PK04_102013 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(c4ccccc43)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A16 compound treatment 236840.0 55700.0 3.8 233640.0 53300.0 3.97 5.4909 0.9998 3188100 PK04_102014 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A17 compound treatment 254960.0 73900.0 5.04 239800.0 59400.0 4.42 6.6886 0.9979 3069309 PK04_102015 COc1ccc(cc1)C(=O)Nc2ccc3N(Cc4ccccc4)C(=O)[C@]5(O[C@H](CCO)[C@H]([C@@H]5C)[Si](C)(C)c6ccc(OC)cc6)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A18 compound treatment 245880.0 64800.0 4.42 244200.0 63800.0 4.75 6.4824 0.9993 3188101 PK04_102016 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(NC(=O)[C@H](C)O)cc4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A19 compound treatment 216000.0 34900.0 2.38 213840.0 33500.0 2.49 3.4442 0.9997 3069310 PK04_102017 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5C(=O)COc6ccccc56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A20 compound treatment 252200.0 71100.0 4.85 252440.0 72100.0 5.36 7.2208 0.9987 3188102 PK04_102018 COc1ccc(cc1)C(=O)Nc2ccc3N(Cc4ccccc4)C(=O)[C@@]5(O[C@@H](CCO)[C@@H]([C@H]5C)[Si](C)(C)c6ccc(OC)cc6)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A21 compound treatment 196920.0 15800.0 1.08 187760.0 7390.0 0.55 1.1518 0.9512 3188103 PK04_102019 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6ccc(cc6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A22 compound treatment 254760.0 73700.0 5.02 245680.0 65300.0 4.86 6.9884 0.9999 3069311 PK04_102020 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(NC(=O)[C@H](C)O)cc4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A23 compound treatment 238400.0 57300.0 3.91 216080.0 35700.0 2.66 4.6419 0.9824 3188104 PK04_102021 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccc(cc63)N7CCOC7=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 A24 compound treatment 231120.0 50000.0 3.41 229800.0 49400.0 3.68 5.013 0.9993 3188105 PK04_102022 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccc(cc63)N7CCOC7=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B01 compound treatment 261480.0 80400.0 5.48 253960.0 73600.0 5.48 7.7481 1.0 3069350 PK04_102023 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5CCC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B02 compound treatment 259280.0 78200.0 5.33 257440.0 77100.0 5.74 7.8252 0.9993 3188106 PK04_102024 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B03 compound treatment 223600.0 42500.0 2.9 235560.0 55200.0 4.11 4.9536 0.9854 3069351 PK04_102025 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6CCCCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B04 compound treatment 243880.0 62800.0 4.28 221560.0 41200.0 3.07 5.1945 0.9866 3188107 PK04_102026 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CC(=O)N5Cc6ccccc6C[C@H]5CO)[C@H]([C@@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B05 compound treatment 225280.0 44200.0 3.01 217960.0 37600.0 2.8 4.1084 0.9993 3188221 PK04_102027 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B06 compound treatment 231000.0 49900.0 3.4 230480.0 50100.0 3.73 5.043 0.9989 3069352 PK04_102028 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(I)c5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B07 compound treatment 208960.0 27900.0 1.9 211680.0 31300.0 2.33 2.9911 0.9948 3188222 PK04_102029 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CC(=O)N(CCO)Cc5ccccc5)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B08 compound treatment 224480.0 43400.0 2.96 215160.0 34800.0 2.59 3.9225 0.9978 3069353 PK04_102030 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(I)cc5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B09 compound treatment 204480.0 23400.0 1.59 199960.0 19600.0 1.46 2.1583 0.999 3188223 PK04_102031 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B10 compound treatment 230440.0 49300.0 3.36 228720.0 48400.0 3.6 4.9234 0.9994 3188224 PK04_102032 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B11 compound treatment 208040.0 26900.0 1.84 565400.0 385000.0 28.66 21.5623 0.7509 3069354 PK04_102033 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B12 compound treatment 256760.0 75700.0 5.16 253680.0 73300.0 5.46 7.5058 0.9996 3188225 PK04_102034 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7CCCCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B13 mock treatment 163440.0 -17700.0 -1.2 169800.0 -10600.0 -0.79 -1.4074 -0.9787 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B14 mock treatment 167440.0 -13700.0 -0.93 163240.0 -17100.0 -1.27 -1.5598 -0.9881 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B15 compound treatment 200760.0 19700.0 1.34 190960.0 10600.0 0.79 1.5054 0.968 3188226 PK04_102035 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B16 compound treatment 251120.0 70000.0 4.77 235880.0 55500.0 4.13 6.2972 0.9974 3069355 PK04_102036 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(I)c5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B17 compound treatment 222400.0 41300.0 2.82 214600.0 34200.0 2.55 3.7927 0.9988 3188227 PK04_102037 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CC(=O)N5Cc6ccccc6C[C@H]5CO)[C@H]([C@@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B18 compound treatment 238000.0 56900.0 3.88 231360.0 51000.0 3.8 5.4268 0.9999 3069356 PK04_102038 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(I)c5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B19 compound treatment 246240.0 65100.0 4.44 238960.0 58600.0 4.36 6.224 1.0 3188228 PK04_102039 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B20 compound treatment 249960.0 68900.0 4.69 245840.0 65500.0 4.87 6.7654 0.9998 3188229 PK04_102040 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B21 compound treatment 207920.0 26800.0 1.83 206360.0 26000.0 1.93 2.661 0.9996 3069357 PK04_102041 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(C)c6c3cc(C)cc6Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B22 compound treatment 253120.0 72000.0 4.91 247560.0 67200.0 5.0 7.0083 1.0 3188230 PK04_102042 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(I)c6)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B23 compound treatment 234560.0 53500.0 3.64 230800.0 50400.0 3.75 5.2315 0.9999 3069358 PK04_102043 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7C(=O)COc8ccccc78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 B24 compound treatment 227240.0 46100.0 3.15 211320.0 31000.0 2.3 3.8534 0.9883 3188231 PK04_102044 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(I)cc5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C01 compound treatment 187360.0 6260.0 0.43 182280.0 1910.0 0.14 0.4026 0.8946 3188232 PK04_102045 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(c5ccccc53)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C02 compound treatment 166920.0 -14200.0 -0.97 208600.0 28200.0 2.1 0.8023 0.3469 3069359 PK04_102046 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6C(=O)COc7ccccc67 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C03 compound treatment 212760.0 31700.0 2.16 216640.0 36300.0 2.7 3.4353 0.9939 3188233 PK04_102047 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(c6ccccc63)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C04 compound treatment 219600.0 38500.0 2.62 216360.0 36000.0 2.68 3.7504 0.9999 3188234 PK04_102048 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6ccc(cc6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C05 compound treatment 228480.0 47400.0 3.23 218520.0 38200.0 2.84 4.2921 0.9979 3069360 PK04_102049 COc1ccc(cc1)[Si](C)(C)[C@H](CCn2cc(nn2)[C@H](O)c3ccccc3)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C06 compound treatment 249280.0 68200.0 4.65 252120.0 71800.0 5.34 7.0631 0.9976 3188235 PK04_102050 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CCO)[C@H]([C@@H]4C)[Si](C)(C)c5ccc(OC)cc5)c6ccccc36)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C07 compound treatment 210400.0 29300.0 2.0 216200.0 35800.0 2.67 3.2984 0.9899 3069393 PK04_102051 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C08 compound treatment 223120.0 42000.0 2.86 204360.0 24000.0 1.79 3.2885 0.9741 3188236 PK04_102052 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6C(=O)c7ccccc7Oc8ccccc68 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C09 compound treatment 231280.0 50200.0 3.42 229400.0 49000.0 3.65 4.9997 0.9995 3069394 PK04_102053 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(C)c4c3cc(C)cc4Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C10 compound treatment 205120.0 24000.0 1.64 215640.0 35300.0 2.63 3.0144 0.9742 3188352 PK04_102054 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5C(=O)COc6ccccc56)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C11 mock treatment 169800.0 -11300.0 -0.77 179560.0 -806.0 -0.06 -0.5871 -0.7599 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C12 mock treatment 176240.0 -4860.0 -0.33 177040.0 -3330.0 -0.25 -0.4093 -0.9897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C13 compound treatment 223680.0 42600.0 2.9 228640.0 48300.0 3.59 4.5933 0.9944 3188353 PK04_102055 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(C)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C14 compound treatment 226760.0 45700.0 3.11 215120.0 34800.0 2.59 4.0303 0.9958 3069395 PK04_102056 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5C(=O)c6ccccc6Oc7ccccc57 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C15 mock treatment 176480.0 -4620.0 -0.31 169560.0 -10800.0 -0.8 -0.7914 -0.9162 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C16 mock treatment 174960.0 -6140.0 -0.42 175840.0 -4530.0 -0.34 -0.5341 -0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C17 compound treatment 211880.0 30800.0 2.1 202440.0 22100.0 1.64 2.6456 0.9927 3188354 PK04_102057 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N5C(=O)c6cccc7cccc5c67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C18 compound treatment 211960.0 30900.0 2.1 216480.0 36100.0 2.69 3.3884 0.9927 3069396 PK04_102058 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(NC(=O)[C@H](C)O)cc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C19 compound treatment 221000.0 39900.0 2.72 209880.0 29500.0 2.2 3.4768 0.9944 3188355 PK04_102059 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5C(=O)COc6ccccc56)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C20 compound treatment 224400.0 43300.0 2.95 207680.0 27300.0 2.03 3.5249 0.9834 3188356 PK04_102060 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N5C(=O)c6ccccc6Oc7ccccc57)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C21 compound treatment 257360.0 76300.0 5.2 253880.0 73500.0 5.47 7.5453 0.9997 3069397 PK04_102061 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C22 compound treatment 209040.0 27900.0 1.9 204920.0 24600.0 1.83 2.6392 0.9998 3188357 PK04_102062 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6C(=O)COc7ccccc67 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C23 compound treatment 166560.0 -14500.0 -0.99 164560.0 -15800.0 -1.18 -1.5327 -0.9964 3188358 PK04_102063 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N5C(=O)c6cccc7cccc5c67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 C24 compound treatment 239920.0 58800.0 4.01 231480.0 51100.0 3.8 5.5257 0.9997 3069398 PK04_102064 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5ccc(cc5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D01 compound treatment 200800.0 19700.0 1.34 201560.0 21200.0 1.58 2.0651 0.9968 3188359 PK04_102065 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D02 compound treatment 258360.0 77300.0 5.27 242920.0 62600.0 4.66 7.0167 0.9981 3069399 PK04_102066 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(I)cc6)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D03 compound treatment 226800.0 45700.0 3.12 226720.0 46400.0 3.45 4.6427 0.9987 3188360 PK04_102067 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(cc6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D04 compound treatment 255400.0 74300.0 5.07 234160.0 53800.0 4.0 6.413 0.9932 3188361 PK04_102068 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D05 compound treatment 228240.0 47100.0 3.21 217240.0 36900.0 2.74 4.2132 0.9969 3069400 PK04_102069 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D06 compound treatment 238400.0 57300.0 3.91 253880.0 73500.0 5.47 6.6313 0.9864 3188362 PK04_102070 C[C@H](C=C)[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D07 compound treatment 221040.0 39900.0 2.72 218720.0 38400.0 2.85 3.944 0.9997 3188363 PK04_102071 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6ccc(cc6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D08 compound treatment 196520.0 15400.0 1.05 192360.0 12000.0 0.89 1.3746 0.9967 3069401 PK04_102072 CO[C@H](C=C)[C@H](O)c1ccc(OC)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D09 compound treatment 222600.0 41500.0 2.83 223720.0 43400.0 3.23 4.2823 0.9979 3188364 PK04_102073 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D10 compound treatment 231560.0 50500.0 3.44 230960.0 50600.0 3.77 5.0953 0.999 3069402 PK04_102074 CO[C@H](C=C)[C@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D11 mock treatment 172080.0 -9020.0 -0.61 174320.0 -6050.0 -0.45 -0.753 -0.9882 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D12 mock treatment 173240.0 -7860.0 -0.54 170480.0 -9890.0 -0.74 -0.8991 -0.9879 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D13 compound treatment 209600.0 28500.0 1.94 204080.0 23700.0 1.76 2.622 0.9988 3069403 PK04_102075 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6CCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D14 compound treatment 348040.0 167000.0 11.38 324520.0 144000.0 10.73 15.6344 0.9996 3188365 PK04_102076 CSc1ccc(NC(=O)O[C@@H]([C@@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D15 mock treatment 172120.0 -8980.0 -0.61 175880.0 -4490.0 -0.33 -0.669 -0.9594 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D16 mock treatment 168400.0 -12700.0 -0.87 172760.0 -7610.0 -0.57 -1.0125 -0.9788 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D17 compound treatment 236000.0 54900.0 3.74 244200.0 63800.0 4.75 6.0061 0.993 3188366 PK04_102077 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D18 compound treatment 180280.0 -819.0 -0.06 177120.0 -3250.0 -0.24 -0.2103 -0.8481 3069404 PK04_102078 C[C@@H](C=C)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D19 compound treatment 238760.0 57700.0 3.93 234080.0 53700.0 4.0 5.6066 1.0 3188367 PK04_102079 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CC(=O)N5CCC[C@H]5CO)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D20 compound treatment 348080.0 167000.0 11.38 332280.0 152000.0 11.31 16.0448 1.0 3069405 PK04_102080 COc1ccc(NC(=O)O[C@H]([C@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D21 compound treatment 250040.0 68900.0 4.7 241960.0 61600.0 4.58 6.5651 0.9999 3188368 PK04_102081 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(cc6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D22 compound treatment 202680.0 21600.0 1.47 202560.0 22200.0 1.65 2.2084 0.9983 3069440 PK04_102082 COc1ccc(NC(=O)O[C@@H]([C@@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D23 compound treatment 240640.0 59500.0 4.06 240360.0 60000.0 4.47 6.0277 0.9989 3188485 PK04_102083 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 D24 compound treatment 177280.0 -3820.0 -0.26 193880.0 13500.0 1.01 0.5271 0.5073 3069441 PK04_102084 O[C@H](CC=C)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E01 mock treatment 175760.0 -5340.0 -0.36 173960.0 -6410.0 -0.48 -0.5945 -0.9911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E02 mock treatment 173880.0 -7220.0 -0.49 172000.0 -8370.0 -0.62 -0.7883 -0.9932 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E03 compound treatment 225160.0 44100.0 3.0 217600.0 37200.0 2.77 4.0836 0.9992 3069442 PK04_102085 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(c6ccccc63)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E04 compound treatment 257280.0 76200.0 5.19 253240.0 72900.0 5.42 7.5078 0.9998 3188486 PK04_102086 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5CCCCC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E05 compound treatment 272280.0 91200.0 6.22 269720.0 89400.0 6.65 9.0982 0.9994 3188487 PK04_102087 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(c6ccccc63)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E06 compound treatment 280960.0 99900.0 6.81 265600.0 85200.0 6.34 9.2998 0.9994 3069443 PK04_102088 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@@]4(O[C@@H](CCn5cc(nn5)[C@H](O)c6ccccc6)[C@@H]([C@H]4C)[Si](C)(C)c7ccc(OC)cc7)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E07 compound treatment 250040.0 68900.0 4.7 248160.0 67800.0 5.05 6.8914 0.9994 3188488 PK04_102089 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(c5ccccc53)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E08 compound treatment 241520.0 60400.0 4.12 236520.0 56200.0 4.18 5.8681 1.0 3188489 PK04_102090 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CCn5cc(CCO)nn5)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E09 mock treatment 184000.0 2900.0 0.2 177960.0 -2410.0 -0.18 0.0132 0.0496 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E10 mock treatment 183160.0 2060.0 0.14 184880.0 4510.0 0.34 0.3369 0.9252 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E11 compound treatment 233280.0 52200.0 3.56 228320.0 48000.0 3.57 5.0393 1.0 3069444 PK04_102091 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E12 compound treatment 249560.0 68500.0 4.67 232840.0 52500.0 3.91 6.062 0.9961 3188490 PK04_102092 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N(C=O)c5ccccc5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E13 compound treatment 239080.0 58000.0 3.95 234200.0 53800.0 4.01 5.6283 1.0 3069445 PK04_102093 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(C)c5c3cc(C)cc5Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E14 compound treatment 255120.0 74000.0 5.05 254400.0 74000.0 5.51 7.4647 0.999 3188491 PK04_102094 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N(C=O)c5ccccc5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E15 compound treatment 254040.0 72900.0 4.97 253360.0 73000.0 5.43 7.3579 0.999 3188492 PK04_102095 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(C)c6c3cc(C)cc6Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E16 compound treatment 210520.0 29400.0 2.01 211360.0 31000.0 2.31 3.0495 0.9976 3069446 PK04_102096 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6cccc(c6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E17 mock treatment 190640.0 9540.0 0.65 178480.0 -1890.0 -0.14 0.3607 0.542 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E18 mock treatment 183400.0 2300.0 0.16 178040.0 -2330.0 -0.17 -0.0115 -0.0492 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E19 compound treatment 269680.0 88600.0 6.04 258280.0 77900.0 5.8 8.3708 0.9998 3188493 PK04_102097 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCCCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E20 compound treatment 228720.0 47600.0 3.25 217480.0 37100.0 2.76 4.249 0.9968 3188494 PK04_102098 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6ccc(cc6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E21 compound treatment 285520.0 104000.0 7.12 281200.0 101000.0 7.5 10.3406 0.9997 3069448 PK04_102099 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCOC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E22 compound treatment 247280.0 66200.0 4.51 245120.0 64800.0 4.82 6.5983 0.9995 3188495 PK04_102100 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5CCOC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E23 compound treatment 271000.0 89900.0 6.13 263120.0 82800.0 6.16 8.6891 1.0 3069450 PK04_102101 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCOC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 E24 compound treatment 239240.0 58100.0 3.96 241360.0 61000.0 4.54 6.0129 0.9977 3188496 PK04_102102 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@]4(O[C@H](CCn5cc(CCO)nn5)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F01 mock treatment 172080.0 -9020.0 -0.61 167680.0 -12700.0 -0.94 -1.1024 -0.9784 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F02 mock treatment 175160.0 -5940.0 -0.4 177600.0 -2770.0 -0.21 -0.4319 -0.9508 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F03 compound treatment 252480.0 71400.0 4.87 240720.0 60400.0 4.49 6.6175 0.9992 3188497 PK04_102103 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccc(cc63)N7CCC7=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F04 compound treatment 306320.0 125000.0 8.54 306960.0 127000.0 9.42 12.6991 0.9988 3069264 PK04_102104 C[C@H](C=C)[C@@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F05 compound treatment 266120.0 85000.0 5.8 251600.0 71200.0 5.3 7.8476 0.999 3069265 PK04_102105 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F06 compound treatment 382560.0 201000.0 13.73 369360.0 189000.0 14.07 19.6584 0.9999 3188498 PK04_102106 CSc1ccc(NC(=O)O[C@H]([C@@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F07 compound treatment 268440.0 87300.0 5.95 263480.0 83100.0 6.19 8.5847 0.9998 3188499 PK04_102107 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F08 compound treatment 218600.0 37500.0 2.56 210000.0 29600.0 2.21 3.3674 0.9973 3069441 PK04_102108 O[C@H](CC=C)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F09 mock treatment 182360.0 1260.0 0.09 179640.0 -726.0 -0.05 0.0226 0.2223 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F10 mock treatment 178400.0 -2700.0 -0.18 178560.0 -1810.0 -0.13 -0.2252 -0.9881 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F11 compound treatment 240440.0 59300.0 4.05 225280.0 44900.0 3.34 5.2245 0.9955 3188500 PK04_102109 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F12 compound treatment 181880.0 781.0 0.05 184920.0 4550.0 0.34 0.2773 0.8083 3069270 PK04_102110 CO[C@@H](C=C)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F13 compound treatment 242800.0 61700.0 4.21 236560.0 56200.0 4.18 5.9319 1.0 3188501 PK04_102111 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(C)c5c3cc(C)cc5Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F14 compound treatment 218080.0 37000.0 2.52 220160.0 39800.0 2.96 3.8771 0.9968 3188502 PK04_102112 CSc1ccc(NC(=O)O[C@H]([C@@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F15 compound treatment 265360.0 84300.0 5.74 246560.0 66200.0 4.93 7.5457 0.9971 3188623 PK04_102113 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F16 compound treatment 241280.0 60200.0 4.1 236280.0 55900.0 4.16 5.8439 1.0 3069312 PK04_102114 CO[C@H](C=C)[C@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F17 mock treatment 183240.0 2140.0 0.15 175880.0 -4490.0 -0.33 -0.1329 -0.3646 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F18 mock treatment 183360.0 2260.0 0.15 182040.0 1670.0 0.12 0.1971 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F19 compound treatment 247000.0 65900.0 4.49 237360.0 57000.0 4.24 6.1764 0.9996 3188624 PK04_102115 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F20 compound treatment 200080.0 19000.0 1.29 194920.0 14600.0 1.08 1.681 0.9961 3069314 PK04_102116 CO[C@H](C=C)[C@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F21 compound treatment 249400.0 68300.0 4.66 247880.0 67500.0 5.02 6.8458 0.9993 3069316 PK04_102117 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccc(cc63)N7CCC7=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F22 compound treatment 346720.0 166000.0 11.29 333000.0 153000.0 11.36 16.0171 1.0 3188625 PK04_102118 O[C@@H](CC=C)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F23 compound treatment 240640.0 59500.0 4.06 243040.0 62700.0 4.66 6.1688 0.9976 3188626 PK04_102119 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 F24 compound treatment 192840.0 11700.0 0.8 198840.0 18500.0 1.37 1.5383 0.9669 3069318 PK04_102120 CO[C@@H](C=C)[C@@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G01 compound treatment 232080.0 51000.0 3.48 218240.0 37900.0 2.82 4.4509 0.9946 3069320 PK04_102121 COc1ccc(cc1)[Si](C)(C)[C@H](CCn2cc(CCO)nn2)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G02 compound treatment 218320.0 37200.0 2.54 217520.0 37200.0 2.77 3.7497 0.9991 3188627 PK04_102122 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6CCOC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G03 mock treatment 183880.0 2780.0 0.19 178160.0 -2210.0 -0.16 0.018 0.0716 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G04 mock treatment 191600.0 10500.0 0.72 183120.0 2750.0 0.2 0.6512 0.8744 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G05 compound treatment 244680.0 63600.0 4.33 244600.0 64200.0 4.78 6.4456 0.9988 3069321 PK04_102123 COc1ccc(cc1)[Si](C)(C)[C@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G06 compound treatment 254640.0 73500.0 5.01 248240.0 67900.0 5.05 7.1173 1.0 3188628 PK04_102124 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G07 compound treatment 241800.0 60700.0 4.14 239320.0 59000.0 4.39 6.0289 0.9996 3069362 PK04_102125 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(C)c4ccccc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G08 compound treatment 283760.0 103000.0 7.0 267320.0 87000.0 6.47 9.5253 0.9992 3188629 PK04_102126 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6CCOC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G09 compound treatment 230600.0 49500.0 3.37 224640.0 44300.0 3.3 4.7164 0.9999 3188630 PK04_102127 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(I)cc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G10 compound treatment 252400.0 71300.0 4.86 246000.0 65600.0 4.88 6.8915 1.0 3188631 PK04_102128 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@@]4(O[C@@H](CCn5cc(nn5)[C@H](O)c6ccccc6)[C@@H]([C@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G11 compound treatment 226880.0 45800.0 3.12 231400.0 51000.0 3.8 4.8928 0.9952 3069365 PK04_102129 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(C)c4c3cc(C)cc4Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G12 compound treatment 228440.0 47300.0 3.23 212280.0 31900.0 2.38 3.9618 0.9886 3188632 PK04_102130 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6cccc(c6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G13 compound treatment 258400.0 77300.0 5.27 251120.0 70800.0 5.27 7.4502 1.0 3069368 PK04_102131 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccccc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G14 compound treatment 269320.0 88200.0 6.01 261320.0 81000.0 6.03 8.5134 1.0 3069370 PK04_102132 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(NC(=O)C)c4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G15 compound treatment 238720.0 57600.0 3.93 231240.0 50900.0 3.79 5.4552 0.9998 3188633 PK04_102133 COc1ccc(cc1)[Si](C)(C)[C@@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G16 compound treatment 241600.0 60500.0 4.12 235360.0 55000.0 4.09 5.8109 1.0 3188634 PK04_102134 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N5C(=O)COc6ccccc56)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G17 compound treatment 266480.0 85400.0 5.82 263360.0 83000.0 6.18 8.4839 0.9996 3188635 PK04_102135 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(NC(=O)[C@H](C)O)c4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G18 compound treatment 221280.0 40200.0 2.74 219960.0 39600.0 2.95 4.0208 0.9993 3069408 PK04_102136 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6CCOC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G19 mock treatment 185000.0 3900.0 0.27 183760.0 3390.0 0.25 0.3667 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G20 mock treatment 182400.0 1300.0 0.09 187240.0 6870.0 0.51 0.4245 0.8175 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G21 compound treatment 236080.0 55000.0 3.75 242400.0 62000.0 4.62 5.9153 0.9947 3188636 PK04_102137 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N(C=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G22 compound treatment 268360.0 87300.0 5.95 244680.0 64300.0 4.79 7.5914 0.9942 3188637 PK04_102138 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G23 compound treatment 238160.0 57100.0 3.89 233280.0 52900.0 3.94 5.5356 1.0 3069412 PK04_102139 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@@]4(O[C@@H](CCn5cc(CCO)nn5)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 G24 compound treatment 239080.0 58000.0 3.95 239160.0 58800.0 4.38 5.8894 0.9987 3188638 PK04_102140 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCCCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H01 compound treatment 225360.0 44300.0 3.02 224320.0 44000.0 3.27 4.4469 0.9992 3188639 PK04_102141 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@@]4(O[C@@H](CC(=O)N(CCO)Cc5ccccc5)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H02 compound treatment 219440.0 38300.0 2.61 223000.0 42600.0 3.17 4.0921 0.9954 3069414 PK04_102142 CSc1ccc(NC(=O)O[C@H]([C@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H03 mock treatment 182080.0 981.0 0.07 179000.0 -1370.0 -0.1 -0.0246 -0.2021 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H04 mock treatment 184520.0 3420.0 0.23 179640.0 -726.0 -0.05 0.1267 0.5292 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H05 compound treatment 249800.0 68700.0 4.68 253120.0 72800.0 5.41 7.1408 0.9974 3188755 PK04_102143 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@@]4(O[C@@H](CC(=O)N5Cc6ccccc6C[C@H]5CO)[C@@H]([C@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H06 compound treatment 257480.0 76400.0 5.21 251640.0 71300.0 5.3 7.4332 1.0 3188362 PK04_102144 C[C@H](C=C)[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H07 compound treatment 276000.0 94900.0 6.47 268560.0 88200.0 6.56 9.2165 1.0 3188756 PK04_102145 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7CCCCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H08 compound treatment 265440.0 84300.0 5.75 264800.0 84400.0 6.28 8.5095 0.999 3069452 PK04_102146 CSc1ccc(NC(=O)O[C@@H](CC=C)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H09 compound treatment 280240.0 99100.0 6.76 266560.0 86200.0 6.42 9.3156 0.9997 3188757 PK04_102147 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(cc6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H10 compound treatment 314280.0 133000.0 9.08 308040.0 128000.0 9.5 13.1396 0.9997 3069454 PK04_102148 COc1ccc(NC(=O)O[C@@H]([C@@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H11 compound treatment 264400.0 83300.0 5.68 268320.0 88000.0 6.55 8.6446 0.9975 3188758 PK04_102149 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H12 compound treatment 240400.0 59300.0 4.04 233600.0 53200.0 3.96 5.6604 0.9999 3069456 PK04_102150 COc1ccc(NC(=O)O[C@H](CC=C)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H13 compound treatment 262760.0 81700.0 5.57 259840.0 79500.0 5.91 8.1193 0.9995 3188759 PK04_102151 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6C(=O)COc7ccccc67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H14 compound treatment 492320.0 311000.0 21.22 488680.0 308000.0 22.95 31.2293 0.9992 3069458 PK04_102152 CSc1ccc(NC(=O)O[C@@H](CC=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H15 compound treatment 220320.0 39200.0 2.67 218640.0 38300.0 2.85 3.9051 0.9995 3188760 PK04_102153 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6CCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H16 compound treatment 228960.0 47900.0 3.26 230080.0 49700.0 3.7 4.9236 0.998 3069460 PK04_102154 COc1ccc(NC(=O)O[C@H](CC=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H17 compound treatment 286040.0 105000.0 7.15 283200.0 103000.0 7.65 10.471 0.9994 3188761 PK04_102155 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6CCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H18 compound treatment 394760.0 214000.0 14.57 384880.0 205000.0 15.22 21.0634 0.9998 3069461 PK04_102156 COc1ccc(NC(=O)O[C@H](CC=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H19 mock treatment 184520.0 3420.0 0.23 186200.0 5830.0 0.43 0.472 0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H20 mock treatment 181200.0 101.0 0.01 182240.0 1870.0 0.14 0.1035 0.7412 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H21 compound treatment 256360.0 75300.0 5.13 248800.0 68400.0 5.09 7.2297 1.0 3188762 PK04_102157 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6CCCCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H22 compound treatment 359080.0 178000.0 12.13 340920.0 161000.0 11.95 17.0298 1.0 3069504 PK04_102158 O[C@H](CC=C)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H23 compound treatment 205200.0 24100.0 1.64 207680.0 27300.0 2.03 2.5993 0.9944 3188763 PK04_102159 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 H24 compound treatment 178360.0 -2740.0 -0.19 183160.0 2790.0 0.21 0.015 0.0537 3069401 PK04_102160 CO[C@H](C=C)[C@H](O)c1ccc(OC)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I01 compound treatment 241240.0 60100.0 4.1 237480.0 57100.0 4.25 5.9051 0.9998 3069507 PK04_102161 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I02 compound treatment 230280.0 49200.0 3.35 220040.0 39700.0 2.95 4.4589 0.998 3188764 PK04_102162 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6C(=O)c7ccccc7Oc8ccccc68 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I03 compound treatment 210560.0 29500.0 2.01 210360.0 30000.0 2.23 2.9988 0.9986 3188765 PK04_102163 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I04 compound treatment 250800.0 69700.0 4.75 253760.0 73400.0 5.46 7.2227 0.9976 3069594 PK04_102164 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(NC(=O)C)c4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I05 mock treatment 183840.0 2740.0 0.19 189920.0 9550.0 0.71 0.6349 0.8636 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I06 mock treatment 184280.0 3180.0 0.22 184000.0 3630.0 0.27 0.3446 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I07 compound treatment 248280.0 67200.0 4.58 247040.0 66700.0 4.96 6.7476 0.9992 3188766 PK04_102165 COc1ccc(cc1)[Si](C)(C)[C@@H](CCn2cc(nn2)[C@H](O)c3ccccc3)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I08 compound treatment 248440.0 67300.0 4.59 233560.0 53200.0 3.96 6.0459 0.9973 3188767 PK04_102166 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6cccc(c6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I09 compound treatment 206640.0 25500.0 1.74 204840.0 24500.0 1.82 2.5193 0.9997 3069598 PK04_102167 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I10 compound treatment 259240.0 78100.0 5.33 247320.0 67000.0 4.98 7.2907 0.9994 3188768 PK04_102168 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@@]4(O[C@@H](CCn5cc(CCO)nn5)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I11 compound treatment 255200.0 74100.0 5.05 239240.0 58900.0 4.38 6.6707 0.9975 3188769 PK04_102169 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(I)cc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I12 compound treatment 289440.0 108000.0 7.39 283280.0 103000.0 7.66 10.6391 0.9998 3069636 PK04_102170 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCOC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I13 compound treatment 250800.0 69700.0 4.75 246720.0 66400.0 4.94 6.8522 0.9998 3188770 PK04_102171 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(c5ccccc53)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I14 compound treatment 251640.0 70500.0 4.81 235720.0 55400.0 4.12 6.3138 0.997 3188771 PK04_102172 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5C(=O)c6ccccc6Oc7ccccc57)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I15 compound treatment 226400.0 45300.0 3.09 226240.0 45900.0 3.41 4.5981 0.9987 3069640 PK04_102173 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I16 compound treatment 292520.0 111000.0 7.6 288640.0 108000.0 8.06 11.0696 0.9996 3188888 PK04_102174 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@]4(O[C@H](CCO)[C@H]([C@@H]4C)[Si](C)(C)c5ccc(OC)cc5)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I17 compound treatment 234480.0 53400.0 3.64 234160.0 53800.0 4.0 5.4045 0.9989 3069645 PK04_102175 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(NC(=O)C)cc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I18 compound treatment 237080.0 56000.0 3.82 227120.0 46800.0 3.48 5.1593 0.9989 3188889 PK04_102176 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccc(cc63)N7C(=O)c8cccc9cccc7c89 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I19 compound treatment 243200.0 62100.0 4.23 214880.0 34500.0 2.57 4.8102 0.9713 3069647 PK04_102177 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5C(=O)c6cccc7cccc5c67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I20 compound treatment 239120.0 58000.0 3.96 229960.0 49600.0 3.69 5.4071 0.9994 3188890 PK04_102178 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(cc4)N5C(=O)c6ccccc6Oc7ccccc57)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I21 mock treatment 181800.0 701.0 0.05 182480.0 2110.0 0.16 0.145 0.8822 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I22 mock treatment 180680.0 -419.0 -0.03 180000.0 -366.0 -0.03 -0.0395 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I23 compound treatment 220560.0 39500.0 2.69 224280.0 43900.0 3.27 4.2134 0.9953 3188891 PK04_102179 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5C(=O)c6cccc7cccc5c67 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 I24 compound treatment 225640.0 44500.0 3.04 224880.0 44500.0 3.31 4.4899 0.9991 3069706 PK04_102180 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N(C=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J01 compound treatment 233400.0 52300.0 3.57 228520.0 48200.0 3.58 5.0556 1.0 3188892 PK04_102181 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J02 compound treatment 234160.0 53100.0 3.62 237960.0 57600.0 4.29 5.589 0.9964 3069707 PK04_102182 CSc1ccc(NC(=O)O[C@@H](CC=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J03 compound treatment 231520.0 50400.0 3.44 230720.0 50400.0 3.75 5.0807 0.9991 3188893 PK04_102183 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6CCCCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J04 compound treatment 225920.0 44800.0 3.06 222520.0 42200.0 3.14 4.3792 0.9999 3069711 PK04_102184 CO[C@H](C=C)[C@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J05 mock treatment 185680.0 4580.0 0.31 185160.0 4790.0 0.36 0.4731 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J06 mock treatment 189720.0 8620.0 0.59 189640.0 9270.0 0.69 0.9037 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J07 compound treatment 237560.0 56500.0 3.85 238640.0 58300.0 4.34 5.7887 0.9982 3188894 PK04_102185 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6cccc(c6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J08 compound treatment 389320.0 208000.0 14.2 374600.0 194000.0 14.46 20.2601 1.0 3069714 PK04_102186 COc1ccc(NC(=O)O[C@@H](CC=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J09 compound treatment 273240.0 92100.0 6.28 263720.0 83400.0 6.2 8.8287 1.0 3188895 PK04_102187 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J10 compound treatment 200840.0 19700.0 1.35 197480.0 17100.0 1.27 1.8524 0.9996 3069716 PK04_102188 CO[C@@H](C=C)[C@@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J11 compound treatment 239880.0 58800.0 4.01 232240.0 51900.0 3.86 5.5637 0.9998 3188896 PK04_102189 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J12 compound treatment 334840.0 154000.0 10.48 326920.0 147000.0 10.91 15.1244 0.9998 3069744 PK04_102190 COc1ccc(NC(=O)O[C@H]([C@@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J13 compound treatment 270080.0 89000.0 6.07 261080.0 80700.0 6.01 8.5374 1.0 3188897 PK04_102191 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J14 compound treatment 190480.0 9380.0 0.64 195840.0 15500.0 1.15 1.2666 0.9615 3069746 PK04_102192 OCCOc1ccc(cc1)[C@@H](O)CC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J15 compound treatment 267680.0 86600.0 5.9 262880.0 82500.0 6.14 8.5165 0.9998 3069749 PK04_102193 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J16 compound treatment 233960.0 52900.0 3.6 230920.0 50600.0 3.76 5.2089 0.9998 3188898 PK04_102194 CO[C@H](C=C)[C@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J17 compound treatment 252200.0 71100.0 4.85 244160.0 63800.0 4.75 6.785 0.9999 3188899 PK04_102195 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CC(=O)N5CCC[C@H]5CO)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J18 compound treatment 357520.0 176000.0 12.03 334360.0 154000.0 11.46 16.6093 0.9997 3069504 PK04_102196 O[C@H](CC=C)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J19 compound treatment 271800.0 90700.0 6.18 246280.0 65900.0 4.91 7.8414 0.9934 3188900 PK04_102197 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(cc6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J20 compound treatment 279760.0 98700.0 6.73 277400.0 97000.0 7.22 9.863 0.9994 3069264 PK04_102198 C[C@H](C=C)[C@@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J21 mock treatment 176920.0 -4180.0 -0.28 175200.0 -5170.0 -0.38 -0.4733 -0.9891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J22 mock treatment 173800.0 -7300.0 -0.5 172280.0 -8090.0 -0.6 -0.7774 -0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J23 compound treatment 241840.0 60700.0 4.14 234400.0 54000.0 4.02 5.7719 0.9999 3069786 PK04_102199 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 J24 compound treatment 236680.0 55600.0 3.79 237960.0 57600.0 4.29 5.7105 0.9981 3188901 PK04_102200 CSc1ccc(NC(=O)O[C@H](CC=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K01 compound treatment 228040.0 46900.0 3.2 216440.0 36100.0 2.68 4.1614 0.9962 3069787 PK04_102201 COc1ccc(cc1)[Si](C)(C)[C@@H](CCn2cc(CCO)nn2)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K02 compound treatment 261920.0 80800.0 5.51 253800.0 73400.0 5.47 7.7609 1.0 3188902 PK04_102202 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(NC(=O)[C@H](C)O)cc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K03 compound treatment 254960.0 73900.0 5.04 237960.0 57600.0 4.29 6.5918 0.9968 3188903 PK04_102203 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(C)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K04 compound treatment 264000.0 82900.0 5.65 244840.0 64500.0 4.8 7.3896 0.9967 3069790 PK04_102204 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N(C=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K05 compound treatment 221560.0 40500.0 2.76 220320.0 40000.0 2.97 4.0532 0.9993 3188904 PK04_102205 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(C)c5c3cc(C)cc5Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K06 compound treatment 275080.0 94000.0 6.41 269560.0 89200.0 6.64 9.2247 0.9998 3189012 PK04_102206 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CCO)[C@H]([C@@H]4C)[Si](C)(C)c5ccc(OC)cc5)c6ccccc36)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K07 mock treatment 190520.0 9420.0 0.64 195360.0 15000.0 1.12 1.2433 0.9656 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K08 mock treatment 183760.0 2660.0 0.18 188080.0 7710.0 0.57 0.5343 0.8873 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K09 compound treatment 237160.0 56100.0 3.82 232800.0 52400.0 3.9 5.4621 0.9999 3069821 PK04_102207 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K10 compound treatment 236520.0 55400.0 3.78 225640.0 45300.0 3.37 5.0544 0.9984 3189013 PK04_102208 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(NC(=O)C)cc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K11 compound treatment 249720.0 68600.0 4.68 243360.0 63000.0 4.69 6.6233 1.0 3069825 PK04_102209 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N4c5c3cc(OC)cc5C(=CC4(C)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K12 compound treatment 283200.0 102000.0 6.96 277880.0 97500.0 7.26 10.0541 0.9998 3189014 PK04_102210 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@@]4(O[C@@H](CCO)[C@@H]([C@H]4C)[Si](C)(C)c5ccc(OC)cc5)c6ccccc36)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K13 compound treatment 213480.0 32400.0 2.21 222320.0 42000.0 3.12 3.769 0.9856 3189015 PK04_102211 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(C)c5c3cc(C)cc5Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K14 compound treatment 286680.0 106000.0 7.2 288160.0 108000.0 8.02 10.7628 0.9985 3069831 PK04_102212 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCOC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K15 mock treatment 191320.0 10200.0 0.7 186800.0 6430.0 0.48 0.8313 0.9832 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K16 mock treatment 189240.0 8140.0 0.56 185840.0 5470.0 0.41 0.6805 0.9884 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K17 compound treatment 239480.0 58400.0 3.98 230360.0 50000.0 3.72 5.4455 0.9994 3189016 PK04_102213 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5C(=O)COc6ccccc56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K18 compound treatment 250920.0 69800.0 4.76 224160.0 43800.0 3.26 5.6707 0.9829 3069867 PK04_102214 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(NC(=O)C)cc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K19 compound treatment 229920.0 48800.0 3.33 233720.0 53400.0 3.97 5.1615 0.9961 3189017 PK04_102215 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K20 compound treatment 243720.0 62600.0 4.27 226520.0 46200.0 3.44 5.4478 0.9942 3069873 PK04_102216 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@@]4(O[C@@H](CCO)[C@@H]([C@H]4C)[Si](C)(C)c5ccc(OC)cc5)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K21 compound treatment 229520.0 48400.0 3.3 225880.0 45500.0 3.39 4.7296 0.9999 3189018 PK04_102217 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5C(=O)c6cccc7cccc5c67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K22 compound treatment 247400.0 66300.0 4.52 215320.0 35000.0 2.6 5.0358 0.9656 3189019 PK04_102218 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CCn5cc(CCO)nn5)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K23 mock treatment 178000.0 -3100.0 -0.21 177800.0 -2570.0 -0.19 -0.2844 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 K24 mock treatment 173840.0 -7260.0 -0.49 172000.0 -8370.0 -0.62 -0.7902 -0.9935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L01 compound treatment 261600.0 80500.0 5.49 248520.0 68200.0 5.07 7.4676 0.9992 3069879 PK04_102219 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L02 compound treatment 173200.0 -7900.0 -0.54 171760.0 -8610.0 -0.64 -0.8337 -0.9963 3189020 PK04_102220 C[C@@H](C=C)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L03 compound treatment 276280.0 95200.0 6.49 253800.0 73400.0 5.47 8.4532 0.9964 3189021 PK04_102221 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(cc6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L04 compound treatment 194320.0 13200.0 0.9 188240.0 7870.0 0.59 1.0518 0.9783 3069907 PK04_102222 C[C@H](C=C)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L05 compound treatment 276920.0 95800.0 6.53 267640.0 87300.0 6.5 9.2124 1.0 3189022 PK04_102223 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6ccc(cc6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L06 compound treatment 257400.0 76300.0 5.2 263280.0 82900.0 6.17 8.0419 0.9964 3069909 PK04_102224 C[C@@H](C=C)[C@@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L07 mock treatment 186800.0 5700.0 0.39 189480.0 9110.0 0.68 0.7545 0.9651 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L08 mock treatment 183120.0 2020.0 0.14 184960.0 4590.0 0.34 0.3392 0.9202 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L09 compound treatment 275640.0 94500.0 6.45 272640.0 92300.0 6.87 9.4138 0.9995 3189023 PK04_102225 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L10 compound treatment 228160.0 47100.0 3.21 233760.0 53400.0 3.97 5.0787 0.9944 3069912 PK04_102226 COc1ccc(NC(=O)O[C@H]([C@@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L11 compound treatment 283520.0 102000.0 6.98 290200.0 110000.0 8.17 10.7179 0.9969 3189024 PK04_102227 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@@]4(O[C@@H](CC(=O)N5CCC[C@H]5CO)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L12 compound treatment 208120.0 27000.0 1.84 208440.0 28100.0 2.09 2.7801 0.998 3069746 PK04_102228 OCCOc1ccc(cc1)[C@@H](O)CC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L13 compound treatment 261320.0 80200.0 5.47 259600.0 79200.0 5.9 8.0372 0.9993 3069917 PK04_102229 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5CCC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L14 compound treatment 223000.0 41900.0 2.86 218280.0 37900.0 2.82 4.0153 1.0 3069920 PK04_102230 O[C@@H](CC=C)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L15 mock treatment 181000.0 -98.8 -0.01 188520.0 8150.0 0.61 0.4244 0.6992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L16 mock treatment 187920.0 6820.0 0.47 183640.0 3270.0 0.24 0.5011 0.9545 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L17 compound treatment 237840.0 56700.0 3.87 207880.0 27500.0 2.05 4.1834 0.9558 3189025 PK04_102231 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L18 compound treatment 191240.0 10100.0 0.69 188680.0 8310.0 0.62 0.9264 0.9985 3069953 PK04_102232 CO[C@H](C=C)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L19 compound treatment 272040.0 90900.0 6.2 264120.0 83800.0 6.23 8.7919 1.0 3189026 PK04_102233 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5ccc(cc5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L20 compound treatment 198080.0 17000.0 1.16 202400.0 22000.0 1.64 1.9782 0.9855 3069956 PK04_102234 CO[C@@H](C=C)[C@@H](O)c1ccc(OC)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L21 compound treatment 285520.0 104000.0 7.12 271360.0 91000.0 6.77 9.8228 0.9997 3189027 PK04_102235 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6CCCCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L22 compound treatment 212520.0 31400.0 2.14 200480.0 20100.0 1.5 2.5733 0.9846 3069961 PK04_102236 CO[C@H](C=C)[C@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L23 mock treatment 173920.0 -7180.0 -0.49 172840.0 -7530.0 -0.56 -0.7422 -0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 L24 mock treatment 169480.0 -11600.0 -0.79 167920.0 -12400.0 -0.93 -1.2151 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M01 compound treatment 240160.0 59100.0 4.03 226480.0 46100.0 3.43 5.2741 0.9968 3069962 PK04_102237 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(c5ccccc53)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M02 compound treatment 253920.0 72800.0 4.96 238800.0 58400.0 4.35 6.5858 0.9978 3188628 PK04_102238 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M03 compound treatment 269400.0 88300.0 6.02 254360.0 74000.0 5.51 8.151 0.999 3189028 PK04_102239 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(C)c6c3cc(C)cc6Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M04 compound treatment 269320.0 88200.0 6.01 255640.0 75300.0 5.6 8.2145 0.9994 3189141 PK04_102240 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5CCCCC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M05 compound treatment 261280.0 80200.0 5.47 259800.0 79400.0 5.91 8.0458 0.9992 3069277 PK04_102241 COc1ccc(cc1)[Si](C)(C)[C@@H](CC(=O)N(CCO)Cc2ccccc2)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M06 compound treatment 268080.0 87000.0 5.93 265920.0 85600.0 6.37 8.6957 0.9994 3189142 PK04_102242 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@@]4(O[C@@H](CCn5cc(CCO)nn5)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M07 compound treatment 293840.0 113000.0 7.69 283040.0 103000.0 7.64 10.8386 1.0 3189143 PK04_102243 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N4c5c3cc(OC)cc5C(=CC4(C)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M08 compound treatment 255160.0 74100.0 5.05 243840.0 63500.0 4.72 6.9109 0.9994 3069284 PK04_102244 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(NC(=O)[C@H](C)O)cc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M09 mock treatment 191800.0 10700.0 0.73 187480.0 7110.0 0.53 0.8903 0.9876 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M10 mock treatment 186080.0 4980.0 0.34 189200.0 8830.0 0.66 0.705 0.9528 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M11 compound treatment 222960.0 41900.0 2.85 219880.0 39500.0 2.94 4.0976 0.9999 3189144 PK04_102245 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M12 compound treatment 257280.0 76200.0 5.19 255400.0 75000.0 5.58 7.6214 0.9993 3189145 PK04_102246 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CCn5cc(nn5)[C@H](O)c6ccccc6)[C@H]([C@@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M13 mock treatment 195160.0 14100.0 0.96 194320.0 14000.0 1.04 1.4122 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M14 mock treatment 191560.0 10500.0 0.71 186520.0 6150.0 0.46 0.8282 0.9771 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M15 compound treatment 258920.0 77800.0 5.31 251200.0 70800.0 5.27 7.4795 1.0 3189146 PK04_102247 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M16 compound treatment 244640.0 63500.0 4.33 242800.0 62400.0 4.65 6.349 0.9994 3189147 PK04_102248 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@@]4(O[C@@H](CCn5cc(nn5)[C@H](O)c6ccccc6)[C@@H]([C@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M17 compound treatment 243760.0 62700.0 4.27 245920.0 65600.0 4.88 6.4707 0.9978 3069327 PK04_102249 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(NC(=O)C)cc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M18 compound treatment 273320.0 92200.0 6.29 272800.0 92400.0 6.88 9.3104 0.999 3189148 PK04_102250 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5CCOC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M19 compound treatment 236480.0 55400.0 3.78 229560.0 49200.0 3.66 5.2588 0.9999 3069330 PK04_102251 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6ccc(cc6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M20 compound treatment 269320.0 88200.0 6.01 264320.0 84000.0 6.25 8.6713 0.9998 3189149 PK04_102252 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCCCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M21 compound treatment 230560.0 49500.0 3.37 228360.0 48000.0 3.57 4.9102 0.9996 3189150 PK04_102253 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4cccc(c4)N5C(=O)c6ccccc6Oc7ccccc57)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M22 compound treatment 236240.0 55100.0 3.76 229400.0 49000.0 3.65 5.2388 0.9999 3189151 PK04_102254 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6cccc(c6)N7CCOC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M23 compound treatment 210520.0 29400.0 2.01 212320.0 32000.0 2.38 3.1 0.9964 3189152 PK04_102255 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 M24 compound treatment 262040.0 80900.0 5.52 265360.0 85000.0 6.33 8.3751 0.9977 3069375 PK04_102256 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@@]4(O[C@@H](CCO)[C@@H]([C@H]4C)[Si](C)(C)c5ccc(OC)cc5)c6ccccc36)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N01 compound treatment 247560.0 66500.0 4.53 227480.0 47100.0 3.51 5.6835 0.992 3189153 PK04_102257 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N02 compound treatment 207280.0 26200.0 1.78 209640.0 29300.0 2.18 2.8028 0.9951 3069379 PK04_102258 CSc1ccc(NC(=O)O[C@@H]([C@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N03 compound treatment 226360.0 45300.0 3.09 231080.0 50700.0 3.77 4.8509 0.995 3189154 PK04_102259 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6ccc(cc6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N04 compound treatment 213840.0 32700.0 2.23 203360.0 23000.0 1.71 2.7885 0.9914 3069716 PK04_102260 CO[C@@H](C=C)[C@@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N05 compound treatment 234000.0 52900.0 3.61 225280.0 44900.0 3.34 4.914 0.9993 3069403 PK04_102261 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6CCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N06 compound treatment 181360.0 261.0 0.02 184360.0 3990.0 0.3 0.2228 0.7481 3069417 PK04_102262 C[C@H](C=C)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N07 compound treatment 251480.0 70400.0 4.8 237360.0 57000.0 4.24 6.3924 0.9981 3189155 PK04_102263 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CC(=O)N(CCO)Cc5ccccc5)[C@H]([C@@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N08 compound treatment 219200.0 38100.0 2.6 215800.0 35400.0 2.64 3.7016 1.0 3069421 PK04_102264 CO[C@@H](C=C)[C@@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N09 mock treatment 190440.0 9340.0 0.64 186200.0 5830.0 0.43 0.7573 0.9826 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N10 mock treatment 188680.0 7580.0 0.52 194280.0 13900.0 1.04 1.0977 0.9485 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N11 compound treatment 270720.0 89600.0 6.11 268440.0 88100.0 6.56 8.9556 0.9994 3189156 PK04_102265 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@@]4(O[C@@H](CC(=O)N5Cc6ccccc6C[C@H]5CO)[C@@H]([C@H]4C)[Si](C)(C)c7ccc(OC)cc7)c8ccccc38)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N12 compound treatment 249600.0 68500.0 4.67 250920.0 70600.0 5.25 7.0154 0.9983 3069424 PK04_102266 CO[C@@H](C=C)[C@@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N13 mock treatment 189520.0 8420.0 0.57 192000.0 11600.0 0.87 1.0182 0.9801 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N14 mock treatment 187400.0 6300.0 0.43 189600.0 9230.0 0.69 0.7897 0.9744 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N15 compound treatment 259640.0 78500.0 5.35 241800.0 61400.0 4.57 7.0195 0.9969 3189268 PK04_102267 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7C(=O)c8cccc9cccc7c89)c%10ccccc%103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N16 compound treatment 189280.0 8180.0 0.56 190800.0 10400.0 0.78 0.9435 0.9868 3069404 PK04_102268 C[C@@H](C=C)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N17 compound treatment 247640.0 66500.0 4.54 253160.0 72800.0 5.42 7.0388 0.9961 3069428 PK04_102269 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N18 compound treatment 211080.0 30000.0 2.04 214960.0 34600.0 2.57 3.2659 0.9935 3189269 PK04_102270 CO[C@@H](C=C)[C@@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N19 compound treatment 247720.0 66600.0 4.54 248560.0 68200.0 5.08 6.8006 0.9985 3070277 PK04_102271 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@@]4(O[C@@H](CC(=O)N5CCC[C@H]5CO)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N20 compound treatment 186000.0 4900.0 0.33 187120.0 6750.0 0.5 0.5917 0.9803 3069270 PK04_102272 CO[C@@H](C=C)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N21 compound treatment 270880.0 89800.0 6.12 271080.0 90700.0 6.75 9.1023 0.9988 3070278 PK04_102273 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N5CCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N22 compound treatment 290480.0 109000.0 7.46 280080.0 99700.0 7.42 10.5208 1.0 3070279 PK04_102274 CSc1ccc(NC(=O)O[C@H](CC=C)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N23 compound treatment 216960.0 35900.0 2.44 212240.0 31900.0 2.37 3.4063 0.9999 3070280 PK04_102275 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6C(=O)COc7ccccc67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 N24 compound treatment 197520.0 16400.0 1.12 196680.0 16300.0 1.21 1.6502 0.9992 3189270 PK04_102276 CO[C@@H](C=C)[C@@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O01 compound treatment 197320.0 16200.0 1.11 190600.0 10200.0 0.76 1.3206 0.9834 3189271 PK04_102277 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(c5ccccc53)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O02 compound treatment 239200.0 58100.0 3.96 231800.0 51400.0 3.83 5.5078 0.9999 3070281 PK04_102278 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N(C=O)c5ccccc5)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O03 compound treatment 208520.0 27400.0 1.87 187600.0 7230.0 0.54 1.7026 0.8752 3189272 PK04_102279 COc1ccc(cc1)[Si](C)(C)[C@@H](CC(=O)N2CCC[C@H]2CO)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O04 compound treatment 275440.0 94300.0 6.43 270520.0 90200.0 6.71 9.2926 0.9998 3189273 PK04_102280 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(NC(=O)[C@H](C)O)c4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O05 compound treatment 254240.0 73100.0 4.99 256880.0 76500.0 5.69 7.5528 0.9978 3070282 PK04_102281 COc1ccc(cc1)[Si](C)(C)[C@H](CC(=O)N(CCO)Cc2ccccc2)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O06 compound treatment 242320.0 61200.0 4.17 223680.0 43300.0 3.22 5.2309 0.9919 3189274 PK04_102282 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5C(=O)c6cccc7cccc5c67 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O07 compound treatment 248960.0 67900.0 4.63 245120.0 64800.0 4.82 6.6793 0.9998 3070283 PK04_102283 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(C)c5c3cc(C)cc5Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O08 compound treatment 238360.0 57300.0 3.9 238840.0 58500.0 4.35 5.8378 0.9985 3189275 PK04_102284 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N(C=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O09 compound treatment 268520.0 87400.0 5.96 265360.0 85000.0 6.33 8.6875 0.9996 3189276 PK04_102285 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(C)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O10 compound treatment 280000.0 98900.0 6.74 272840.0 92500.0 6.88 9.6346 0.9999 3070284 PK04_102286 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O11 mock treatment 185000.0 3900.0 0.27 177200.0 -3170.0 -0.24 0.0214 0.0603 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O12 mock treatment 190080.0 8980.0 0.61 185240.0 4870.0 0.36 0.6895 0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O13 compound treatment 266360.0 85300.0 5.81 254800.0 74400.0 5.54 8.0276 0.9997 3189277 PK04_102287 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(C)c4ccccc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O14 compound treatment 244640.0 63500.0 4.33 231760.0 51400.0 3.83 5.768 0.9981 3189278 PK04_102288 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(NC(=O)[C@H](C)O)cc43 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O15 compound treatment 253000.0 71900.0 4.9 251520.0 71200.0 5.3 7.2109 0.9993 3070285 PK04_102289 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(c4ccccc43)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O16 compound treatment 258880.0 77800.0 5.3 256840.0 76500.0 5.69 7.7743 0.9994 3189279 PK04_102290 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@]4(O[C@H](CCn5cc(nn5)[C@H](O)c6ccccc6)[C@H]([C@@H]4C)[Si](C)(C)c7ccc(OC)cc7)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O17 compound treatment 224760.0 43700.0 2.98 222840.0 42500.0 3.16 4.3401 0.9995 3070286 PK04_102291 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(CC=C)c6ccc(cc63)N7C(=O)c8cccc9cccc7c89 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O18 compound treatment 255680.0 74600.0 5.08 253960.0 73600.0 5.48 7.4685 0.9993 3189280 PK04_102292 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6CCCCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O19 compound treatment 237760.0 56700.0 3.86 242480.0 62100.0 4.62 6.0005 0.996 3189281 PK04_102293 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5cccc(c5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O20 compound treatment 262720.0 81600.0 5.56 261800.0 81400.0 6.06 8.2205 0.9991 3070287 PK04_102294 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccc(cc4)N5CCCCC5=O)c6ccccc63 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O21 compound treatment 218360.0 37300.0 2.54 210680.0 30300.0 2.26 3.3916 0.9982 3189282 PK04_102295 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4cccc(c4)N5C(=O)COc6ccccc56)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O22 compound treatment 220640.0 39500.0 2.7 214800.0 34400.0 2.56 3.7184 0.9997 3070288 PK04_102296 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(CC=C)c4ccc(cc43)N5C(=O)c6ccccc6Oc7ccccc57 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O23 compound treatment 232760.0 51700.0 3.52 227520.0 47200.0 3.51 4.9721 1.0 3189283 PK04_102297 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(CC=C)c5ccc(cc53)N6C(=O)c7cccc8cccc6c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 O24 compound treatment 176400.0 -4700.0 -0.32 233680.0 53300.0 3.97 2.5793 0.6479 3189284 PK04_102298 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCO)C(=O)N(Cc4ccc(NC(=O)C)cc4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P01 compound treatment 266000.0 84900.0 5.79 264040.0 83700.0 6.23 8.4965 0.9993 3070289 PK04_102299 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(CCO)nn4)C(=O)N(Cc5ccc(cc5)N6CCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P02 compound treatment 187800.0 6700.0 0.46 181480.0 1110.0 0.08 0.3817 0.822 3069953 PK04_102300 CO[C@H](C=C)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P03 compound treatment 241120.0 60000.0 4.09 235640.0 55300.0 4.11 5.8025 1.0 3189285 PK04_102301 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4Cc5ccccc5C[C@H]4CO)C(=O)N(Cc6cccc(c6)N7C(=O)COc8ccccc78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P04 compound treatment 277920.0 96800.0 6.6 262200.0 81800.0 6.09 8.9743 0.9992 3070290 PK04_102302 C[C@@H](C=C)[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P05 compound treatment 253960.0 72900.0 4.97 249080.0 68700.0 5.11 7.1288 0.9999 3189394 PK04_102303 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(CCO)nn4)C(=O)N(C)c5c3cc(C)cc5Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P06 compound treatment 184640.0 3540.0 0.24 185080.0 4710.0 0.35 0.4188 0.9834 3069907 PK04_102304 C[C@H](C=C)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P07 compound treatment 233640.0 52500.0 3.58 235320.0 55000.0 4.09 5.425 0.9978 3189395 PK04_102305 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(Cc6cccc(c6)N7CCC7=O)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P08 compound treatment 210800.0 29700.0 2.02 207520.0 27200.0 2.02 2.8609 1.0 3069314 PK04_102306 CO[C@H](C=C)[C@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P09 compound treatment 235520.0 54400.0 3.71 233080.0 52700.0 3.92 5.3978 0.9996 3070291 PK04_102307 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6CCCCC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P10 compound treatment 214200.0 33100.0 2.26 224440.0 44100.0 3.28 3.9153 0.9833 3189396 PK04_102308 CSc1ccc(NC(=O)O[C@@H]([C@@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P11 mock treatment 177560.0 -3540.0 -0.24 177800.0 -2570.0 -0.19 -0.3057 -0.9933 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P12 mock treatment 180240.0 -859.0 -0.06 179280.0 -1090.0 -0.08 -0.0986 -0.9874 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P13 compound treatment 239000.0 57900.0 3.95 224080.0 43700.0 3.25 5.0919 0.9954 3189397 PK04_102309 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N(CCO)Cc4ccccc4)C(=O)N(Cc5cccc(c5)N6C(=O)c7cccc8cccc6c78)c9ccccc93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P14 compound treatment 184280.0 3180.0 0.22 183880.0 3510.0 0.26 0.3383 0.9957 3070292 PK04_102310 OCCOc1ccc(cc1)[C@H](O)CC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P15 compound treatment 228960.0 47900.0 3.26 222960.0 42600.0 3.17 4.5489 0.9999 3070293 PK04_102311 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@@]4(O[C@@H](CC(=O)N(CCO)Cc5ccccc5)[C@@H]([C@H]4C)[Si](C)(C)c6ccc(OC)cc6)c7ccccc37)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P16 compound treatment 177040.0 -4060.0 -0.28 174120.0 -6250.0 -0.46 -0.5244 -0.9693 3070292 PK04_102312 OCCOc1ccc(cc1)[C@H](O)CC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P17 compound treatment 250200.0 69100.0 4.71 238040.0 57700.0 4.29 6.3665 0.9989 3189398 PK04_102313 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5ccc(cc5)N6CCOC6=O)c7ccccc73 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P18 compound treatment 259960.0 78900.0 5.38 258120.0 77800.0 5.79 7.8938 0.9993 3070294 PK04_102314 CO[C@@H](C=C)[C@@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P19 compound treatment 216520.0 35400.0 2.41 227680.0 47300.0 3.52 4.1976 0.9831 3189399 PK04_102315 COc1ccc(cc1)[Si](C)(C)[C@@H]2[C@@H](C)[C@@]3(O[C@H]2CC(=O)N4CCC[C@H]4CO)C(=O)N(Cc5cccc(c5)N6C(=O)COc7ccccc67)c8ccccc83 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P20 compound treatment 247840.0 66700.0 4.55 247880.0 67500.0 5.02 6.7706 0.9988 3070290 PK04_102316 C[C@@H](C=C)[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P21 compound treatment 260960.0 79900.0 5.44 256600.0 76200.0 5.67 7.862 0.9998 3189400 PK04_102317 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccc(cc53)N6CCC6=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P22 compound treatment 194920.0 13800.0 0.94 199280.0 18900.0 1.41 1.6617 0.9809 3070295 PK04_102318 COc1ccc(NC(=O)O[C@@H]([C@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P23 compound treatment 213320.0 32200.0 2.2 211280.0 30900.0 2.3 3.1803 0.9997 3189401 PK04_102319 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCn4cc(nn4)[C@H](O)c5ccccc5)C(=O)N(C)c6c3cc(C)cc6Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2102 P24 compound treatment 200200.0 19100.0 1.3 194240.0 13900.0 1.03 1.651 0.9934 3414053 PK04_102320 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A01 mock treatment 169640.0 -8580.0 -0.58 167840.0 -11500.0 -0.86 -1.0193 -0.9826 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A02 mock treatment 170440.0 -7780.0 -0.53 171080.0 -8270.0 -0.62 -0.8102 -0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A03 mock treatment 169800.0 -8420.0 -0.57 168160.0 -11200.0 -0.83 -0.9947 -0.9834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A04 mock treatment 199440.0 21200.0 1.45 202160.0 22800.0 1.7 2.2235 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A05 mock treatment 172280.0 -5940.0 -0.4 170080.0 -9270.0 -0.69 -0.7741 -0.9676 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A06 mock treatment 193960.0 15700.0 1.07 193760.0 14400.0 1.07 1.5173 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A07 mock treatment 171720.0 -6500.0 -0.44 172040.0 -7310.0 -0.54 -0.6979 -0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A08 mock treatment 167560.0 -10700.0 -0.73 168120.0 -11200.0 -0.84 -1.1048 -0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A09 mock treatment 167240.0 -11000.0 -0.75 167960.0 -11400.0 -0.85 -1.1286 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A10 mock treatment 166240.0 -12000.0 -0.82 167000.0 -12400.0 -0.92 -1.2274 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A11 mock treatment 164600.0 -13600.0 -0.93 172600.0 -6750.0 -0.5 -1.0117 -0.9585 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A12 mock treatment 166160.0 -12100.0 -0.82 172720.0 -6630.0 -0.49 -0.9302 -0.9702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A13 mock treatment 165160.0 -13100.0 -0.89 170680.0 -8670.0 -0.65 -1.0858 -0.9875 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A14 mock treatment 163880.0 -14300.0 -0.98 167160.0 -12200.0 -0.91 -1.3327 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A15 mock treatment 160160.0 -18100.0 -1.23 169480.0 -9870.0 -0.73 -1.39 -0.9696 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A16 mock treatment 164680.0 -13500.0 -0.92 173440.0 -5910.0 -0.44 -0.9637 -0.9426 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A17 mock treatment 163720.0 -14500.0 -0.99 171040.0 -8310.0 -0.62 -1.1362 -0.9746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A18 mock treatment 172520.0 -5700.0 -0.39 166040.0 -13300.0 -0.99 -0.9751 -0.9164 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A19 mock treatment 194880.0 16700.0 1.14 199560.0 20200.0 1.5 1.8669 0.9904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A20 mock treatment 166560.0 -11700.0 -0.79 171760.0 -7590.0 -0.57 -0.9614 -0.986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A21 mock treatment 169360.0 -8860.0 -0.6 170280.0 -9070.0 -0.68 -0.9043 -0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A22 mock treatment 166440.0 -11800.0 -0.8 169760.0 -9590.0 -0.71 -1.0725 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A23 mock treatment 118440.0 -59800.0 -4.08 133800.0 -45600.0 -3.39 -5.279 -0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 A24 mock treatment 163080.0 -15100.0 -1.03 164600.0 -14800.0 -1.1 -1.506 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B01 mock treatment 163880.0 -14300.0 -0.98 158360.0 -21000.0 -1.56 -1.7959 -0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B02 mock treatment 165360.0 -12900.0 -0.88 165080.0 -14300.0 -1.06 -1.3708 -0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B03 compound treatment 176400.0 -1820.0 -0.12 175280.0 -4070.0 -0.3 -0.3018 -0.9219 2277 HSCI1_000001 CCc1nc([nH]c1c2ccncc2)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B04 compound treatment 306560.0 128000.0 8.75 310880.0 132000.0 9.79 13.1093 0.9984 656 HSCI1_000002 Oc1c(Br)cc(/C=C/2\C(=O)Nc3ccc(I)cc23)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B05 compound treatment 171120.0 -7100.0 -0.48 169840.0 -9510.0 -0.71 -0.8427 -0.9828 2114187 HSCI1_000003 CCOC(=O)c1cccc(NC(=O)CBr)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B06 compound treatment 171360.0 -6860.0 -0.47 172440.0 -6910.0 -0.51 -0.6943 -0.9989 1362420 HSCI1_000004 Oc1c(I)cc(Cl)cc1C(=O)Nc2cc(ccc2Cl)S(=O)(=O)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B07 compound treatment 456920.0 279000.0 19.0 451520.0 272000.0 20.26 27.7595 0.9995 3175973 HSCI1_000005 COC(=O)c1cc(NCc2cc(O)ccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B08 compound treatment 164080.0 -14100.0 -0.96 162400.0 -17000.0 -1.26 -1.5736 -0.9912 3175974 HSCI1_000006 CCCCCCCCCCCCCCCCCCOC[C@H](COP(=O)(O)OC1CCC(O)C(O)C1O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B09 compound treatment 258800.0 80600.0 5.49 257960.0 78600.0 5.85 8.0218 0.9995 9 HSCI1_000007 [O-][N+](=O)c1ccc2[nH]c-3c(CC(=O)Nc4ccccc34)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B10 compound treatment 159920.0 -18300.0 -1.25 159040.0 -20300.0 -1.51 -1.951 -0.9954 571 HSCI1_000008 CCCCCCCCCCCCCCCCCCOC[C@H](COC(=O)OC1C(O)C(O)C(O)C(CO)C1O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B11 mock treatment 165960.0 -12300.0 -0.84 166760.0 -12600.0 -0.94 -1.2535 -0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B12 mock treatment 166560.0 -11700.0 -0.79 170240.0 -9110.0 -0.68 -1.0414 -0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B13 mock treatment 163440.0 -14800.0 -1.01 168880.0 -10500.0 -0.78 -1.2634 -0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B14 mock treatment 162120.0 -16100.0 -1.1 166360.0 -13000.0 -0.97 -1.4597 -0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B15 compound treatment 166760.0 -11500.0 -0.78 166640.0 -12700.0 -0.95 -1.2213 -0.9955 3055039 HSCI1_000009 Cn1cnc2nc(NCCO)nc(NCc3ccccc3)c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B16 compound treatment 146920.0 -31300.0 -2.13 147800.0 -31600.0 -2.35 -3.1692 -0.9989 3175975 HSCI1_000010 CCCCCCCCCCCCCCCCCCOC[C@H](COP(=O)(O)OC1C(O)C(O)C(O)CC1OC)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B17 compound treatment 193160.0 14900.0 1.02 196080.0 16700.0 1.25 1.6008 0.995 3055043 HSCI1_000011 CCCCCCCCCCCCCCC[C@@H](O)[C@H](N)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B18 compound treatment 165120.0 -13100.0 -0.89 164960.0 -14400.0 -1.07 -1.3887 -0.9959 2326 HSCI1_000012 CCCCCC(=O)O[C@@H]1[C@@H](OC(=O)/C(=C\C)/C)C(=C2[C@@H]3OC(=O)[C@@](C)(O)[C@@]3(O)[C@H](C[C@](C)(OC(=O)C)[C@@H]12)OC(=O)CCC)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B19 compound treatment 177240.0 -975.0 -0.07 182000.0 2650.0 0.2 0.0923 0.4439 2026 HSCI1_000013 CCCCCCCCCCNc1cc(CO)c2cc[nH]c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B20 compound treatment 171160.0 -7060.0 -0.48 171240.0 -8110.0 -0.6 -0.767 -0.9937 193 HSCI1_000014 COc1cc2CCN(C)[C@H]3Cc4ccc(OC)c(Oc5ccc(C[C@@H]6N(C)CCc7cc(OC)c(Oc(c1OC)c32)cc67)cc5)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B21 compound treatment 171120.0 -7100.0 -0.48 174000.0 -5350.0 -0.4 -0.6237 -0.9953 3055048 HSCI1_000015 Nc1nc(Cl)nc2n(cnc12)C3OC(CO)[C@H](O)[C@H]3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B22 compound treatment 170760.0 -7460.0 -0.51 171480.0 -7870.0 -0.59 -0.7737 -0.9975 3175977 HSCI1_000016 CCCCCCCCCC(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H]3C=C(C)C(=O)[C@@]3(O)CC(=C[C@H]2[C@@H]4C(C)(C)[C@]41OC(=O)CCCCCCCCC)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B23 mock treatment 166560.0 -11700.0 -0.79 166760.0 -12600.0 -0.94 -1.2246 -0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 B24 mock treatment 161040.0 -17200.0 -1.17 168080.0 -11300.0 -0.84 -1.4212 -0.9866 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C01 mock treatment 172440.0 -5780.0 -0.39 163240.0 -16100.0 -1.2 -1.1264 -0.8924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C02 mock treatment 175160.0 -3060.0 -0.21 171280.0 -8070.0 -0.6 -0.5721 -0.8997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C03 compound treatment 179120.0 905.0 0.06 175160.0 -4190.0 -0.31 -0.177 -0.5566 2257 HSCI1_000017 COc1ccc(cc1)C(=O)CBr 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C04 compound treatment 232960.0 54700.0 3.73 235560.0 56200.0 4.18 5.5972 0.9984 561 HSCI1_000018 C[C@@H](NC(=O)/C(=C/c1ccc(O)c(O)c1)/C#N)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C05 compound treatment 180200.0 1980.0 0.14 179800.0 448.0 0.03 0.1192 0.8557 2256 HSCI1_000019 Oc1ccc(cc1)C(=O)CBr 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C06 compound treatment 232720.0 54500.0 3.72 230880.0 51500.0 3.84 5.3394 0.9999 1000099 HSCI1_000020 C[C@H](NC(=O)/C(=C/c1ccc(O)c(O)c1)/C#N)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C07 compound treatment 180920.0 2700.0 0.18 182880.0 3530.0 0.26 0.3161 0.985 2258 HSCI1_000021 OC(=O)COc1ccc(cc1)C(=O)CBr 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C08 compound treatment 158520.0 -19700.0 -1.34 162480.0 -16900.0 -1.26 -1.8374 -0.9994 2227 HSCI1_000022 CCCCCCCCCCCCCCCC(=O)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C09 compound treatment 172120.0 -6100.0 -0.42 175240.0 -4110.0 -0.31 -0.5103 -0.9887 2147 HSCI1_000023 CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCCP(=O)(F)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C10 compound treatment 178480.0 265.0 0.02 183200.0 3850.0 0.29 0.2153 0.7502 617 HSCI1_000024 COc1cc(OC)c(/C=C\2/C(=O)Nc3ccccc23)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C11 mock treatment 171560.0 -6660.0 -0.45 175880.0 -3470.0 -0.26 -0.5036 -0.9644 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C12 mock treatment 166400.0 -11800.0 -0.81 175640.0 -3710.0 -0.28 -0.765 -0.8983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C13 mock treatment 222360.0 44100.0 3.01 223920.0 44600.0 3.32 4.4736 0.9988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C14 mock treatment 169800.0 -8420.0 -0.57 171800.0 -7550.0 -0.56 -0.8031 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C15 mock treatment 172160.0 -6060.0 -0.41 170840.0 -8510.0 -0.63 -0.7399 -0.9785 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C16 mock treatment 169040.0 -9180.0 -0.63 171560.0 -7790.0 -0.58 -0.8524 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C17 compound treatment 182760.0 4540.0 0.31 176960.0 -2390.0 -0.18 0.0932 0.2608 3055108 HSCI1_000025 CSCC1OC([C@@H](O)[C@H]1O)n2ccc3c(N)ncnc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C18 compound treatment 208800.0 30600.0 2.09 219200.0 39800.0 2.97 3.5715 0.9851 3055110 HSCI1_000026 ClCC(=O)c1cc(Br)c(Br)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C19 compound treatment 288040.0 110000.0 7.49 285400.0 106000.0 7.89 10.8755 0.9997 2121 HSCI1_000027 Oc1ccc(cc1)c2oc3cc(O)cc(O)c3c(=O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C20 compound treatment 182120.0 3900.0 0.27 187400.0 8050.0 0.6 0.6118 0.9333 1916983 HSCI1_000028 CC(C)C(N1C(=O)/C(=C/c2ccccc2)/SC1=S)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C21 compound treatment 240640.0 62400.0 4.26 233040.0 53700.0 4.0 5.8349 0.9995 2188 HSCI1_000029 Oc1ccc(O)c2C(=O)C(=C(Cl)C(=O)c12)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C22 compound treatment 310280.0 132000.0 9.0 302560.0 123000.0 9.17 12.8508 1.0 563 HSCI1_000030 Oc1ccc(/C=C(\C#N)/C(=O)NCCCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C23 compound treatment 170080.0 -8140.0 -0.55 178200.0 -1150.0 -0.09 -0.4528 -0.8068 1031143 HSCI1_000031 CS(=O)(=O)SCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 C24 mock treatment 166440.0 -11800.0 -0.8 167240.0 -12100.0 -0.9 -1.2051 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D01 mock treatment 165160.0 -13100.0 -0.89 170880.0 -8470.0 -0.63 -1.0752 -0.9857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D02 mock treatment 163880.0 -14300.0 -0.98 166480.0 -12900.0 -0.96 -1.3685 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D03 compound treatment 187120.0 8900.0 0.61 191440.0 12100.0 0.9 1.0654 0.9817 551 HSCI1_000032 CC(C)(C)c1cc(C=C(C#N)C#N)cc(Br)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D04 compound treatment 169800.0 -8420.0 -0.57 175040.0 -4310.0 -0.32 -0.6326 -0.9623 3479696 HSCI1_000033 OC(=O)C(CCCCNC(=O)CNC(=O)c1cccc(c1)C(=O)NCC(=O)NCCCCC(NC(=O)OCc2ccc(cc2)C(F)(F)F)C(=O)O)NC(=O)OCc3ccc(cc3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D05 compound treatment 209560.0 31300.0 2.14 218280.0 38900.0 2.9 3.5598 0.9888 674 HSCI1_000034 CCOC(=O)c1c(C)[nH]c(/C=C/2\C(=O)Nc3ccccc23)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D06 compound treatment 329680.0 151000.0 10.33 321040.0 142000.0 10.55 14.7586 0.9999 146 HSCI1_000035 CCCCCC#CCC#CCC#CCC#CCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D07 compound treatment 193280.0 15100.0 1.03 196320.0 17000.0 1.26 1.6192 0.9947 3175981 HSCI1_000036 O=c1sn(Cc2ccccc2)c(=S)n1Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D08 compound treatment 217000.0 38800.0 2.64 224080.0 44700.0 3.33 4.2237 0.9935 1000097 HSCI1_000037 Cc1c(C)c2OC(C)(COc3ccc(CC4SC(=O)NC4=O)cc3)CCc2c(C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D09 compound treatment 245760.0 67500.0 4.6 245960.0 66600.0 4.96 6.7616 0.9993 628 HSCI1_000038 Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc34)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D10 compound treatment 182840.0 4620.0 0.32 188440.0 9090.0 0.68 0.7012 0.9396 3175982 HSCI1_000039 COc1ccc(Nc2nccc(NCCO)n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D11 mock treatment 172600.0 -5620.0 -0.38 175680.0 -3670.0 -0.27 -0.464 -0.9864 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D12 mock treatment 169360.0 -8860.0 -0.6 170520.0 -8830.0 -0.66 -0.8917 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D13 mock treatment 176280.0 -1940.0 -0.13 178080.0 -1270.0 -0.09 -0.1602 -0.9868 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D14 mock treatment 171680.0 -6540.0 -0.45 171160.0 -8190.0 -0.61 -0.7462 -0.9881 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D15 mock treatment 166720.0 -11500.0 -0.78 172200.0 -7150.0 -0.53 -0.9306 -0.9822 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D16 mock treatment 165320.0 -12900.0 -0.88 173320.0 -6030.0 -0.45 -0.9391 -0.9513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D17 compound treatment 179280.0 1060.0 0.07 179600.0 248.0 0.02 0.0644 0.8595 584 HSCI1_000040 Nc1cc2ncnc(Nc3cccc(Br)c3)c2cc1N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D18 compound treatment 208880.0 30700.0 2.09 204920.0 25600.0 1.9 2.8239 0.9989 2180 HSCI1_000041 COc1ccc(CNc2nc(NCc3ccc(OC)cc3)c4ncn(C(C)C)c4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D19 compound treatment 188920.0 10700.0 0.73 193160.0 13800.0 1.03 1.2427 0.9859 3055161 HSCI1_000042 COc1cc2ncnc(Nc3ccc(Cl)cc3F)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D20 compound treatment 175720.0 -2500.0 -0.17 174400.0 -4950.0 -0.37 -0.3809 -0.9384 2067 HSCI1_000043 CC(C)C(C(=O)OC(C#N)c1cccc(Oc2ccccc2)c1)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D21 compound treatment 179160.0 945.0 0.06 180480.0 1130.0 0.08 0.1049 0.9914 3055164 HSCI1_000044 N/C(=C(/C#N)\c1ccccc1C(F)(F)F)/Sc2ccc(N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D22 compound treatment 180040.0 1820.0 0.12 179920.0 568.0 0.04 0.1179 0.897 2407 HSCI1_000045 CN1C(=C(O)c2ccccc2S1(=O)=O)C(=O)Nc3ncc(C)s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D23 compound treatment 213160.0 34900.0 2.38 215800.0 36400.0 2.71 3.6028 0.9979 550 HSCI1_000046 COC1=C(Br)[C@H](O)[C@](O)(CC#N)C=C1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 D24 mock treatment 169960.0 -8260.0 -0.56 170000.0 -9350.0 -0.7 -0.8902 -0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E01 mock treatment 176600.0 -1620.0 -0.11 173920.0 -5430.0 -0.4 -0.3638 -0.8681 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E02 mock treatment 175520.0 -2700.0 -0.18 174120.0 -5230.0 -0.39 -0.4053 -0.9412 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E03 mock treatment 178720.0 505.0 0.03 180040.0 688.0 0.05 0.0605 0.9813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E04 mock treatment 185120.0 6900.0 0.47 178200.0 -1150.0 -0.09 0.2722 0.5689 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E05 compound treatment 181880.0 3660.0 0.25 182840.0 3490.0 0.26 0.3602 0.9998 2294 HSCI1_000047 CC(=O)NC(C(=O)O)C(C)(C)SN=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E06 compound treatment 182080.0 3860.0 0.26 186360.0 7010.0 0.52 0.5551 0.95 3175983 HSCI1_000048 CCCCCCCCCCCCCCCCCC(=O)OCC(CO)OC(=O)CCC/C=C/C/C=C/C\C=C\C\C=C\CCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E07 compound treatment 379280.0 201000.0 13.71 390320.0 211000.0 15.7 20.7958 0.9977 640 HSCI1_000049 O=C/1Nc2ccccc2\C1=C\c3ccc[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E08 compound treatment 278000.0 99800.0 6.8 279640.0 100000.0 7.46 10.0884 0.9989 1907779 HSCI1_000050 CC(C)n1cnc2c(NCc3ccccc3)nc(NCCO)nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E09 mock treatment 185720.0 7500.0 0.51 185840.0 6490.0 0.48 0.7032 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E10 mock treatment 179720.0 1500.0 0.1 183680.0 4330.0 0.32 0.3003 0.8883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E11 compound treatment 341960.0 164000.0 11.16 344400.0 165000.0 12.28 16.58 0.9989 627 HSCI1_000051 C=CC(=O)c1ccc2ccccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E12 compound treatment 216840.0 38600.0 2.63 216280.0 36900.0 2.75 3.8055 0.9998 536 HSCI1_000052 ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E13 compound treatment 277360.0 99100.0 6.76 302720.0 123000.0 9.18 11.2722 0.9886 593 HSCI1_000053 Oc1ccc2ccc(=O)oc2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E14 compound treatment 189320.0 11100.0 0.76 194760.0 15400.0 1.15 1.3462 0.9797 3055208 HSCI1_000054 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CO)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E15 mock treatment 178200.0 -15.3 0.0 183440.0 4090.0 0.3 0.2144 0.7047 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E16 mock treatment 181920.0 3700.0 0.25 179680.0 328.0 0.02 0.1959 0.7718 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E17 mock treatment 175600.0 -2620.0 -0.18 182040.0 2690.0 0.2 0.0154 0.0574 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E18 mock treatment 185880.0 7660.0 0.52 182240.0 2890.0 0.21 0.5215 0.9229 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E19 compound treatment 184200.0 5980.0 0.41 185440.0 6090.0 0.45 0.6089 0.9986 1912 HSCI1_000055 [O-][N+](=O)c1cccc2cn[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E20 compound treatment 184840.0 6620.0 0.45 184680.0 5330.0 0.4 0.5998 0.9979 3175984 HSCI1_000056 CCCC(=O)OCSC(=S)OC1CC2CC1C3CCCC23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E21 compound treatment 276000.0 97800.0 6.67 272920.0 93600.0 6.96 9.6383 0.9998 596 HSCI1_000057 CN(C)c1ccc(/C=C\2/C(=O)Nc3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E22 compound treatment 350440.0 172000.0 11.74 337560.0 158000.0 11.77 16.6288 1.0 564 HSCI1_000058 Oc1ccc(/C=C(\C#N)/C(=O)NCCCCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E23 compound treatment 197560.0 19300.0 1.32 197600.0 18200.0 1.36 1.8929 0.9999 2175 HSCI1_000059 CCCCCCCCN1C(=O)C(=C(C)C1(C)O)C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 E24 mock treatment 178440.0 225.0 0.02 171000.0 -8350.0 -0.62 -0.4287 -0.6895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F01 mock treatment 170640.0 -7580.0 -0.52 169400.0 -9950.0 -0.74 -0.889 -0.9845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F02 mock treatment 175160.0 -3060.0 -0.21 175840.0 -3510.0 -0.26 -0.3321 -0.9937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F03 mock treatment 179960.0 1740.0 0.12 177240.0 -2110.0 -0.16 -0.027 -0.1372 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F04 mock treatment 180400.0 2180.0 0.15 185880.0 6530.0 0.49 0.4489 0.8833 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F05 compound treatment 229360.0 51100.0 3.49 229680.0 50300.0 3.75 5.1142 0.9994 2108 HSCI1_000060 COc1cc2C/C(=C\c3cc(C)c(O)c(C)c3)/C(=O)c2c(N)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F06 compound treatment 203560.0 25300.0 1.73 212640.0 33300.0 2.48 2.9737 0.9845 2303 HSCI1_000061 COc1cc2CCN3Cc4c(OC)c(O)ccc4CC3c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F07 compound treatment 206800.0 28600.0 1.95 214160.0 34800.0 2.59 3.2099 0.9902 1967 HSCI1_000062 Brc1cccc(Nc2ncnc3cc4[nH]cnc4cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F08 compound treatment 197160.0 18900.0 1.29 198120.0 18800.0 1.4 1.901 0.9992 1918768 HSCI1_000063 Clc1ccc(C(=O)n2nnc3ccccc23)c(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F09 mock treatment 178800.0 585.0 0.04 181400.0 2050.0 0.15 0.136 0.863 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F10 mock treatment 178400.0 185.0 0.01 183920.0 4570.0 0.34 0.2493 0.7328 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F11 compound treatment 303320.0 125000.0 8.53 307560.0 128000.0 9.54 12.7784 0.9984 583 HSCI1_000064 CC(C)n1cnc2c(NCc3ccccc3)nc(NCCCO)nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F12 compound treatment 186280.0 8060.0 0.55 185720.0 6370.0 0.47 0.7239 0.9973 1085933 HSCI1_000065 COC(=O)c1ccccc1NC(=O)c2ccc(F)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F13 compound treatment 291000.0 113000.0 7.69 294960.0 116000.0 8.6 11.5213 0.9984 675 HSCI1_000066 Brc1ccc2NC(=O)/C(=C\c3cc4CCCCc4[nH]3)/c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F14 compound treatment 198400.0 20200.0 1.38 203840.0 24500.0 1.82 2.2618 0.9904 2144 HSCI1_000067 O=C(Nc1ccccc1)C2C(=O)NC(=S)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F15 mock treatment 180760.0 2540.0 0.17 186920.0 7570.0 0.56 0.521 0.8839 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F16 mock treatment 179520.0 1300.0 0.09 185880.0 6530.0 0.49 0.4064 0.8229 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F17 mock treatment 181640.0 3420.0 0.23 183600.0 4250.0 0.32 0.3887 0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F18 mock treatment 178560.0 345.0 0.02 182000.0 2650.0 0.2 0.156 0.7859 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F19 compound treatment 193200.0 15000.0 1.02 197080.0 17700.0 1.32 1.6554 0.992 643 HSCI1_000068 CNc1cc2ncnc(Nc3cccc(Br)c3)c2cc1N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F20 compound treatment 197560.0 19300.0 1.32 195040.0 15700.0 1.17 1.7582 0.9982 122 HSCI1_000069 C(c1c[nH]c2ccccc12)c3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F21 compound treatment 448720.0 271000.0 18.44 444880.0 266000.0 19.76 27.0147 0.9994 590 HSCI1_000070 CC(C)n1cnc2c(Nc3cccc(Cl)c3)nc(NCCO)nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F22 compound treatment 180240.0 2020.0 0.14 188360.0 9010.0 0.67 0.5717 0.8352 2060831 HSCI1_000071 O=C1CCCC(=O)C1CC2C(=O)CCCC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F23 compound treatment 209080.0 30900.0 2.1 211400.0 32000.0 2.39 3.1745 0.998 3176054 HSCI1_000072 N/C(=C(/C#N)\C(=C(/N)\Sc1ccccc1)\[N+]#[C-])/Sc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 F24 mock treatment 177120.0 -1100.0 -0.07 167760.0 -11600.0 -0.86 -0.6629 -0.7654 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G01 mock treatment 179240.0 1020.0 0.07 178360.0 -992.0 -0.07 -0.0028 -0.0277 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G02 compound treatment 176000.0 -2220.0 -0.15 172240.0 -7110.0 -0.53 -0.4811 -0.874 305 HSCI1_000073 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CO)NC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G03 mock treatment 188760.0 10500.0 0.72 190680.0 11300.0 0.84 1.1045 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G04 mock treatment 232640.0 54400.0 3.71 238400.0 59000.0 4.39 5.7313 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G05 mock treatment 190960.0 12700.0 0.87 185760.0 6410.0 0.48 0.9516 0.9601 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G06 mock treatment 189960.0 11700.0 0.8 189080.0 9730.0 0.72 1.0781 0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G07 compound treatment 222720.0 44500.0 3.03 221560.0 42200.0 3.14 4.3668 0.9998 2073 HSCI1_000074 CC(=CCC/C(=C/CC/C(=C/CSc1nc[nH]n1)/C)/C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G08 compound treatment 302800.0 125000.0 8.49 301240.0 122000.0 9.07 12.4207 0.9995 3176055 HSCI1_000075 CCOc1cc(/C=C(/C#N)\C(=O)N)cc(CSc2ccccc2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G09 compound treatment 191520.0 13300.0 0.91 190440.0 11100.0 0.83 1.2249 0.9989 2335 HSCI1_000076 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G10 compound treatment 192160.0 13900.0 0.95 200040.0 20700.0 1.54 1.761 0.9732 3055275 HSCI1_000077 CC(C)(C)OC(=O)NC(CC(=O)CCl)C(=O)Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G11 compound treatment 258280.0 80100.0 5.46 260560.0 81200.0 6.04 8.1336 0.9987 2134 HSCI1_000078 COc1cc(O)c(cc1/C=C/C(=O)c2ccc(O)cc2)C(C)(C)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G12 compound treatment 248360.0 70100.0 4.78 248800.0 69400.0 5.17 7.0364 0.9992 3055277 HSCI1_000079 COc1cc(cc(CN(C)CCc2ccc(cc2)[N+](=O)[O-])c1O)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G13 compound treatment 186520.0 8300.0 0.57 186040.0 6690.0 0.5 0.7523 0.9979 1002387 HSCI1_000080 Oc1ccc(C=C(C#N)C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G14 compound treatment 181680.0 3460.0 0.24 185920.0 6570.0 0.49 0.5127 0.9443 3176058 HSCI1_000081 C[C@@H]1[C@@H](O)[C@@]2(O)[C@H]([C@@H]3C=C(CO)C[C@@]4(O)[C@@H](C=C(C)C4=O)[C@]13O)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G15 compound treatment 187720.0 9500.0 0.65 185480.0 6130.0 0.46 0.7807 0.9852 672 HSCI1_000082 Oc1ccc(CC(C#N)C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G16 compound treatment 311960.0 134000.0 9.12 308240.0 129000.0 9.59 13.2307 0.9997 3176059 HSCI1_000083 OCc1cc2ncnc(Nc3ccc(O)c(Br)c3)c2cc1CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G17 mock treatment 185640.0 7420.0 0.51 189040.0 9690.0 0.72 0.8678 0.985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G18 mock treatment 179400.0 1180.0 0.08 185720.0 6370.0 0.47 0.3922 0.8158 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G19 mock treatment 182440.0 4220.0 0.29 189960.0 10600.0 0.79 0.7619 0.9066 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G20 mock treatment 181560.0 3340.0 0.23 189920.0 10600.0 0.79 0.7174 0.876 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G21 compound treatment 219400.0 41200.0 2.81 198080.0 18700.0 1.39 2.9711 0.9478 3415700 HSCI1_000084 CCCCCCCC(=O)OCC(CO)OC(=O)CCCCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G22 compound treatment 420120.0 242000.0 16.49 413920.0 235000.0 17.46 24.0066 0.9996 3176060 HSCI1_000085 CCn1cnc2c(Nc3cccc(Cl)c3)nc(N[C@@H]4CCCC[C@@H]4N)nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G23 compound treatment 218120.0 39900.0 2.72 212960.0 33600.0 2.5 3.6924 0.9991 3055326 HSCI1_000086 Cc1ccc(cc1)c2cn3c4CCCCc4sc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 G24 mock treatment 174920.0 -3300.0 -0.22 180240.0 888.0 0.07 -0.1121 -0.4788 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H01 mock treatment 182000.0 3780.0 0.26 176520.0 -2830.0 -0.21 0.0334 0.1003 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H02 compound treatment 189720.0 11500.0 0.78 188120.0 8770.0 0.65 1.0161 0.9958 1886 HSCI1_000087 NCCOB(c1ccccc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H03 mock treatment 186120.0 7900.0 0.54 180400.0 1050.0 0.08 0.4362 0.8011 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H04 mock treatment 190040.0 11800.0 0.81 185160.0 5810.0 0.43 0.8757 0.9573 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H05 mock treatment 190960.0 12700.0 0.87 185200.0 5850.0 0.44 0.9222 0.9489 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H06 mock treatment 189760.0 11500.0 0.79 182200.0 2850.0 0.21 0.7064 0.8667 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H07 compound treatment 204840.0 26600.0 1.82 215760.0 36400.0 2.71 3.1996 0.981 2278 HSCI1_000088 Oc1cc(ccc1NC(=O)Nc2ccccc2Br)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H08 compound treatment 190680.0 12500.0 0.85 197040.0 17700.0 1.32 1.5318 0.9776 1891 HSCI1_000089 Clc1oc(=O)c2ccccc2c1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H09 compound treatment 212440.0 34200.0 2.33 216760.0 37400.0 2.78 3.6186 0.9961 1966 HSCI1_000090 Cn1cnc2cc3c(Nc4cccc(Br)c4)ncnc3cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H10 compound treatment 188760.0 10500.0 0.72 189920.0 10600.0 0.79 1.0645 0.999 3176061 HSCI1_000091 CC1(CCC2(C)O1)C(C2C(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H11 compound treatment 299520.0 121000.0 8.27 303680.0 124000.0 9.25 12.391 0.9984 291 HSCI1_000092 CC[C@H](CO)Nc1nc(NCc2ccccc2)c3ncn(C(C)C)c3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H12 compound treatment 370520.0 192000.0 13.11 367840.0 188000.0 14.03 19.1904 0.9994 3055333 HSCI1_000093 O=C/1Nc2ccccc2\C1=C/c3c[nH]cn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H13 compound treatment 324720.0 147000.0 9.99 325720.0 146000.0 10.89 14.7658 0.9991 3176062 HSCI1_000094 CC[C@@H](CO)Nc1nc(NCc2ccccc2)c3ncn(C(C)C)c3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H14 compound treatment 199520.0 21300.0 1.45 188160.0 8810.0 0.66 1.4906 0.9354 1040138 HSCI1_000095 COc1cc(C=O)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H15 compound treatment 234840.0 56600.0 3.86 233600.0 54200.0 4.04 5.5847 0.9997 3176063 HSCI1_000096 CC(C)n1cnc2c(NCc3ccccc3O)nc(NCCCO)nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H16 compound treatment 184440.0 6220.0 0.42 182520.0 3170.0 0.24 0.4668 0.9615 2109 HSCI1_000097 OCc1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H17 mock treatment 186760.0 8540.0 0.58 183520.0 4170.0 0.31 0.6313 0.9565 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H18 mock treatment 184200.0 5980.0 0.41 182800.0 3450.0 0.26 0.47 0.975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H19 mock treatment 185480.0 7260.0 0.5 188920.0 9570.0 0.71 0.8538 0.9843 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H20 mock treatment 185280.0 7060.0 0.48 186320.0 6970.0 0.52 0.7073 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H21 compound treatment 420360.0 242000.0 16.51 416040.0 237000.0 17.62 24.1297 0.9995 3176064 HSCI1_000098 O/N=C\1/C(=C\2/C(=O)Nc3ccc(cc23)S(=O)(=O)O)/Nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H22 compound treatment 183360.0 5140.0 0.35 183480.0 4130.0 0.31 0.4653 0.9978 2069332 HSCI1_000099 CC(=O)/C(=N/O)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H23 compound treatment 198600.0 20400.0 1.39 196320.0 17000.0 1.26 1.8757 0.9989 642 HSCI1_000100 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 H24 mock treatment 174720.0 -3500.0 -0.24 168160.0 -11200.0 -0.83 -0.7575 -0.8743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I01 mock treatment 179400.0 1180.0 0.08 181600.0 2250.0 0.17 0.1754 0.9442 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I02 compound treatment 185040.0 6820.0 0.47 180000.0 648.0 0.05 0.3631 0.7762 666 HSCI1_000101 CC(C)c1cc(/C=C(\C#N)/C(=O)NCCCc2ccccc2)cc(C(C)C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I03 compound treatment 190840.0 12600.0 0.86 192160.0 12800.0 0.95 1.2827 0.9987 3176066 HSCI1_000102 CCCCC/C=C/C/C=C/C\C=C\C\C=C\CCCC(=O)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I04 compound treatment 450760.0 273000.0 18.58 462800.0 283000.0 21.1 28.0562 0.998 2104844 HSCI1_000103 Oc1ccc(O)c(CNc2ccc(cc2)C(=O)OC3(CC4CC5CC(C4)C3)C5)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I05 mock treatment 220000.0 41800.0 2.85 218240.0 38900.0 2.89 4.061 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I06 mock treatment 215720.0 37500.0 2.56 214280.0 34900.0 2.6 3.6462 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I07 mock treatment 192560.0 14300.0 0.98 192720.0 13400.0 0.99 1.3951 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I08 mock treatment 183240.0 5020.0 0.34 189800.0 10400.0 0.78 0.7921 0.9322 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I09 compound treatment 416920.0 239000.0 16.27 415880.0 237000.0 17.6 23.9555 0.9992 626 HSCI1_000104 CC(C)N(CCC(=O)c1ccc2ccccc2c1)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I10 compound treatment 227280.0 49100.0 3.35 226440.0 47100.0 3.5 4.8435 0.9997 3055340 HSCI1_000105 Cc1ccc(N/N=C/2\C(=O)Nc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I11 compound treatment 188320.0 10100.0 0.69 198480.0 19100.0 1.42 1.4938 0.9445 568 HSCI1_000106 COc1ccc(C=C(C#N)C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I12 compound treatment 227800.0 49600.0 3.38 230840.0 51500.0 3.83 5.1001 0.998 3176067 HSCI1_000107 Ic1cccc(CSc2nnc(o2)c3ccncc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I13 compound treatment 262840.0 84600.0 5.77 266320.0 87000.0 6.47 8.6565 0.9984 558 HSCI1_000108 Oc1ccc(C=C(C#N)C#N)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I14 compound treatment 172520.0 -5700.0 -0.39 175560.0 -3790.0 -0.28 -0.4741 -0.9877 3176068 HSCI1_000109 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CO)NC(=O)CCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I15 compound treatment 200160.0 21900.0 1.5 204840.0 25500.0 1.9 2.3993 0.9931 1975 HSCI1_000110 C[C@@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@@H](O)CC[C@@]43C)[C@@]2(O)CC[C@@H]1c5ccc(=O)oc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I16 compound treatment 160040.0 -18200.0 -1.24 169320.0 -10000.0 -0.75 -1.4042 -0.9706 1001980 HSCI1_000111 CCCCCCCC/C=C/CCCCCCCC(=O)OCC(CO)OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I17 compound treatment 178000.0 -215.0 -0.01 181720.0 2370.0 0.18 0.1142 0.646 130 HSCI1_000112 C/C(=C\C=C\C(=C\C(=O)Nc1ccc(O)cc1)\C)/C=C/C2=C(C)CCCC2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I18 compound treatment 192600.0 14400.0 0.98 194960.0 15600.0 1.16 1.5149 0.9965 1922639 HSCI1_000113 CC(C)C(N1C(=O)/C(=C/c2ccc(Br)cc2)/SC1=S)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I19 mock treatment 182560.0 4340.0 0.3 186800.0 7450.0 0.55 0.6014 0.9569 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I20 mock treatment 183440.0 5220.0 0.36 185600.0 6250.0 0.47 0.5807 0.9913 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I21 mock treatment 188240.0 10000.0 0.68 183320.0 3970.0 0.3 0.6921 0.9296 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I22 mock treatment 179920.0 1700.0 0.12 179000.0 -352.0 -0.03 0.0636 0.5342 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I23 compound treatment 253480.0 75300.0 5.13 248360.0 69000.0 5.14 7.2601 1.0 565 HSCI1_000114 Oc1cc(C=C(C#N)C#N)cc(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 I24 mock treatment 175040.0 -3180.0 -0.22 174640.0 -4710.0 -0.35 -0.4011 -0.9731 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J01 mock treatment 179360.0 1140.0 0.08 171960.0 -7390.0 -0.55 -0.3338 -0.6008 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J02 compound treatment 213600.0 35400.0 2.41 215000.0 35600.0 2.65 3.5819 0.9989 3176070 HSCI1_000115 OC(=O)c1c(Br)c(Br)c(Br)c(Br)c1c2c3ccc(O)cc3oc4cc(=O)ccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J03 compound treatment 186720.0 8500.0 0.58 185080.0 5730.0 0.43 0.7114 0.9886 294 HSCI1_000116 [O-][N+](=O)c1ccc(cc1)c2nc(c([nH]2)c3ccncc3)c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J04 compound treatment 196960.0 18700.0 1.28 195960.0 16600.0 1.24 1.7777 0.9999 3055387 HSCI1_000117 C[C@@]12CCC3C(CCC4=C[C@H](O)CCC34)C2CC[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J05 mock treatment 183520.0 5300.0 0.36 187000.0 7650.0 0.57 0.6582 0.976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J06 mock treatment 187480.0 9260.0 0.63 185360.0 6010.0 0.45 0.7628 0.9857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J07 mock treatment 185800.0 7580.0 0.52 195800.0 16400.0 1.22 1.2313 0.9265 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J08 mock treatment 185520.0 7300.0 0.5 192640.0 13300.0 0.99 1.0515 0.9496 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J09 compound treatment 225680.0 47500.0 3.24 228440.0 49100.0 3.65 4.8716 0.9982 633 HSCI1_000118 OC(=O)c1cc(ccc1O)N(Cc2ccccc2O)Cc3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J10 compound treatment 184120.0 5900.0 0.4 187520.0 8170.0 0.61 0.7145 0.98 2251 HSCI1_000119 O=C(NC1=CC(=O)c2ccccc2C1=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J11 compound treatment 201880.0 23700.0 1.61 209680.0 30300.0 2.26 2.7369 0.9864 645 HSCI1_000120 Brc1cccc(Nc2ncnc3ccc(NC(=O)C=C)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J12 compound treatment 195480.0 17300.0 1.18 198320.0 19000.0 1.41 1.8305 0.9959 3176071 HSCI1_000121 Nc1nc(Cl)nc2n(cnc12)C3C[C@@H](O)C(CO)O3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J13 compound treatment 195960.0 17700.0 1.21 204680.0 25300.0 1.89 2.1884 0.977 646 HSCI1_000122 CCC(=O)Nc1ccc2ncnc(Nc3cccc(Br)c3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J14 compound treatment 270960.0 92700.0 6.32 259600.0 80200.0 5.97 8.6943 0.9996 854065 HSCI1_000123 CCCCCCCCCCCC1=C(O)C(=O)C=C(O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J15 compound treatment 499280.0 321000.0 21.89 503280.0 324000.0 24.11 32.5256 0.9988 670 HSCI1_000124 CN(C)S(=O)(=O)c1ccc2NC(=O)/C(=C\c3cc4CCCCc4[nH]3)/c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J16 compound treatment 204160.0 25900.0 1.77 197880.0 18500.0 1.38 2.2258 0.9924 3176072 HSCI1_000125 CN(C)c1ccc(/C=C/2\C(=O)Nc3ccccc23)c4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J17 compound treatment 197320.0 19100.0 1.3 199440.0 20100.0 1.5 1.9782 0.9976 1996 HSCI1_000126 CC#CC(=O)Nc1ccc2ncnc(Nc3cccc(Br)c3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J18 compound treatment 184800.0 6580.0 0.45 183480.0 4130.0 0.31 0.5347 0.9829 2268 HSCI1_000127 CC(=CC1C(C(=O)OCc2coc(Cc3ccccc3)c2)C1(C)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J19 mock treatment 181760.0 3540.0 0.24 181120.0 1770.0 0.13 0.2639 0.9591 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J20 mock treatment 177720.0 -495.0 -0.03 178840.0 -512.0 -0.04 -0.0508 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J21 mock treatment 180160.0 1940.0 0.13 187280.0 7930.0 0.59 0.511 0.8449 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J22 mock treatment 178880.0 665.0 0.05 178680.0 -672.0 -0.05 -0.0033 -0.0493 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J23 compound treatment 464800.0 287000.0 19.54 458120.0 279000.0 20.75 28.4867 0.9995 654 HSCI1_000128 CC(C)C(CO)Nc1nc(Nc2cccc(Cl)c2)c3ncn(C(C)C)c3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 J24 mock treatment 175000.0 -3220.0 -0.22 173200.0 -6150.0 -0.46 -0.4788 -0.9431 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K01 mock treatment 178520.0 305.0 0.02 178360.0 -992.0 -0.07 -0.0375 -0.4892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K02 compound treatment 219840.0 41600.0 2.84 215240.0 35900.0 2.67 3.8954 0.9995 3055432 HSCI1_000129 CCOC(=O)c1cc(OC)c(OC)cc1NC(=O)c2cc(OC)c(OC)c(OC)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K03 compound treatment 269720.0 91500.0 6.24 271440.0 92100.0 6.85 9.2577 0.9989 570 HSCI1_000130 NC(=O)/C(=C/c1ccc(O)c(O)c1)/C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K04 compound treatment 234200.0 56000.0 3.82 232600.0 53200.0 3.96 5.5012 0.9998 1005921 HSCI1_000131 OCC1OC(Oc2cc(O)c3c(=O)c(coc3c2)c4ccc(O)cc4)C(O)C(O)C1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K05 compound treatment 214440.0 36200.0 2.47 209120.0 29800.0 2.22 3.3129 0.9985 559 HSCI1_000132 OC(=O)/C(=C/c1ccc(O)c(O)c1)/C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K06 compound treatment 353080.0 175000.0 11.92 343880.0 165000.0 12.25 17.0887 0.9999 620 HSCI1_000133 COc1cc(/C=C(\C#N)/C(=O)c2ccc(O)c(O)c2)cc(I)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K07 mock treatment 190680.0 12500.0 0.85 192800.0 13400.0 1.0 1.3086 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K08 mock treatment 189480.0 11300.0 0.77 188880.0 9530.0 0.71 1.0445 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K09 mock treatment 190080.0 11900.0 0.81 184400.0 5050.0 0.38 0.8376 0.9392 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K10 mock treatment 189880.0 11700.0 0.8 186880.0 7530.0 0.56 0.9585 0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K11 compound treatment 191160.0 12900.0 0.88 189520.0 10200.0 0.76 1.1592 0.9971 553 HSCI1_000134 Oc1cc(C=C(C#N)C#N)ccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K12 compound treatment 366480.0 188000.0 12.84 359080.0 180000.0 13.38 18.5346 0.9998 3176129 HSCI1_000135 Oc1cc(/C=C(\C#N)/C(=O)NCCCc2ccccc2)cc(I)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K13 compound treatment 414080.0 236000.0 16.08 405200.0 226000.0 16.81 23.2565 0.9998 1000035 HSCI1_000136 O=C1c2ccccc2-c3n[nH]c4cccc1c34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K14 compound treatment 441520.0 263000.0 17.95 448640.0 269000.0 20.04 26.8655 0.9985 1 HSCI1_000137 Oc1ccc(/C=C(\C#N)/C(=O)NCCCNC(=O)\C(=C\c2ccc(O)c(O)c2)\C#N)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K15 mock treatment 222760.0 44500.0 3.04 215040.0 35700.0 2.66 4.0256 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K16 mock treatment 232800.0 54600.0 3.72 231080.0 51700.0 3.85 5.3538 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K17 compound treatment 259440.0 81200.0 5.54 254000.0 74600.0 5.56 7.8443 1.0 554 HSCI1_000138 Oc1cc(C=C(C#N)C#N)cc([N+](=O)[O-])c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K18 compound treatment 91680.0 -86500.0 -5.9 91600.0 -87800.0 -6.53 -8.7899 -0.9987 3176130 HSCI1_000139 CN(C)c1ccc2c(c3ccccc3C(=O)O)c4ccc(=[N+](C)C)cc4oc2c1.CC(=O)NCCSS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K19 compound treatment 184120.0 5900.0 0.4 180680.0 1330.0 0.1 0.3545 0.8553 555 HSCI1_000140 Cc1cc2ncc(nc2cc1C)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K20 compound treatment 186880.0 8660.0 0.59 180960.0 1610.0 0.12 0.5023 0.8334 2311 HSCI1_000141 COC(=O)c1c(c2cc(OC)c(OC)c(OC)c2)c3ccnc(OCc4ncccn4)c3c(=O)n1Cc5ccnc(C)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K21 mock treatment 207440.0 29200.0 1.99 211240.0 31900.0 2.37 3.0871 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K22 mock treatment 179760.0 1540.0 0.11 182800.0 3450.0 0.26 0.2559 0.9226 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K23 mock treatment 180760.0 2540.0 0.17 179080.0 -272.0 -0.02 0.1084 0.6203 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 K24 mock treatment 170880.0 -7340.0 -0.5 175120.0 -4230.0 -0.31 -0.5764 -0.9752 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L01 mock treatment 178480.0 265.0 0.02 179240.0 -112.0 -0.01 0.0069 0.345 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L02 compound treatment 182120.0 3900.0 0.27 183960.0 4610.0 0.34 0.4307 0.9922 1995 HSCI1_000142 CN(C1CCCCC1)C(=O)CCCOc2ccc3[nH]c(=O)ccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L03 compound treatment 342520.0 164000.0 11.2 345960.0 167000.0 12.4 16.6891 0.9987 3176131 HSCI1_000143 Nc1ncnc2n(cc(I)c12)C3OC(CO)[C@H](O)[C@@H]3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L04 compound treatment 213200.0 35000.0 2.39 209880.0 30500.0 2.27 3.2932 0.9997 3055484 HSCI1_000144 COc1cc(SC)ccc1c2nc3ccncc3[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L05 compound treatment 196040.0 17800.0 1.22 194880.0 15500.0 1.16 1.6765 0.9997 1907775 HSCI1_000145 CS(=O)(=O)c1ccc(cc1)c2nc(c([nH]2)c3ccncc3)c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L06 compound treatment 208760.0 30500.0 2.08 215040.0 35700.0 2.66 3.3507 0.9928 3176132 HSCI1_000146 COc1ccc(cc1)C(=C2C(=O)Nc3ccccc23)c4ccc(OC)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L07 mock treatment 185520.0 7300.0 0.5 187560.0 8210.0 0.61 0.7841 0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L08 mock treatment 183800.0 5580.0 0.38 184640.0 5290.0 0.39 0.5475 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L09 mock treatment 188840.0 10600.0 0.72 183240.0 3890.0 0.29 0.7168 0.919 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L10 mock treatment 184840.0 6620.0 0.45 184040.0 4690.0 0.35 0.5661 0.9919 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L11 compound treatment 430440.0 252000.0 17.2 430960.0 252000.0 18.73 25.4009 0.9991 3055486 HSCI1_000147 O=C1NC(=O)c2c1c3c4ccccc4n5C6CCC(O6)n7c8ccccc8c2c7c53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L12 compound treatment 188040.0 9820.0 0.67 192640.0 13300.0 0.99 1.1729 0.982 3176133 HSCI1_000148 OC(=O)c1ccc(Cl)cc1NC(=O)Nc2cccc(c2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L13 compound treatment 302400.0 124000.0 8.47 309320.0 130000.0 9.67 12.8267 0.9978 3176134 HSCI1_000149 O/N=C\1/C(=C\2/C(=O)Nc3ccc(I)cc23)/Nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L14 compound treatment 200960.0 22700.0 1.55 199760.0 20400.0 1.52 2.1705 0.9999 3055490 HSCI1_000150 COc1cc(ccc1c2nc3ccncc3[nH]2)S(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L15 mock treatment 182520.0 4300.0 0.29 184040.0 4690.0 0.35 0.4542 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L16 mock treatment 189720.0 11500.0 0.78 187400.0 8050.0 0.6 0.9782 0.9911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L17 compound treatment 189560.0 11300.0 0.77 190120.0 10800.0 0.8 1.1136 0.9998 3176135 HSCI1_000151 C[S+](O)c1ccc(CSc2nc(c([nH]2)c3ccc(F)cc3)c4ccncc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L18 compound treatment 254240.0 76000.0 5.18 254480.0 75100.0 5.59 7.6188 0.9993 2109556 HSCI1_000152 Nc1n[nH]c2nc3ccccc3nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L19 compound treatment 182680.0 4460.0 0.3 184600.0 5250.0 0.39 0.4914 0.9924 3176136 HSCI1_000153 C[C@@H]1C2NCC(C)C[C@H]2O[C@@]31CCC4C5CC=C6CC(O)CCC6(C)C5C(=O)C4=C3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L20 compound treatment 187240.0 9020.0 0.62 188400.0 9050.0 0.67 0.9112 0.999 3055494 HSCI1_000154 OB(O)c1ccc(cc1)C(=O)/C=C/c2ccc(I)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L21 mock treatment 185480.0 7260.0 0.5 182560.0 3210.0 0.24 0.519 0.944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L22 mock treatment 184880.0 6660.0 0.45 177760.0 -1590.0 -0.12 0.2375 0.5058 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L23 mock treatment 178080.0 -135.0 -0.01 173640.0 -5710.0 -0.43 -0.3071 -0.7223 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 L24 mock treatment 169920.0 -8300.0 -0.57 171840.0 -7510.0 -0.56 -0.7953 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M01 mock treatment 183160.0 4940.0 0.34 181560.0 2210.0 0.16 0.3546 0.9454 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M02 compound treatment 273520.0 95300.0 6.5 273160.0 93800.0 6.98 9.5314 0.9994 2095175 HSCI1_000155 Oc1ccc(/C=C(\C#N)/C(=O)NC2CCC(CC3CCC(CC3)NC(=O)\C(=C\c4ccc(O)c(O)c4)\C#N)CC2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M03 compound treatment 227120.0 48900.0 3.33 225480.0 46100.0 3.43 4.7852 0.9999 552 HSCI1_000156 NC(=C(C#N)C#N)/C(=C/c1ccc(O)cc1)/C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M04 compound treatment 351920.0 174000.0 11.84 353160.0 174000.0 12.94 17.5211 0.999 613 HSCI1_000157 Oc1cc(/C=C/c2ccc(O)c(O)c2)oc(=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M05 compound treatment 200960.0 22700.0 1.55 204480.0 25100.0 1.87 2.4189 0.9957 657 HSCI1_000158 COc1ccc(/C=C(\C#N)/c2cccnc2)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M06 compound treatment 204920.0 26700.0 1.82 200080.0 20700.0 1.54 2.3782 0.9966 3176139 HSCI1_000159 CCCCCCCCCC(=O)O[C@@H]1[C@@H](C)[C@]2(O)[C@@H]3C=C(C)C(=O)[C@@]3(O)CC(=C[C@H]2[C@@H]4C(C)(C)[C@@]41OC(=O)CCCCCCCCC)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M07 compound treatment 292760.0 115000.0 7.81 286000.0 107000.0 7.94 11.1346 1.0 671 HSCI1_000160 NC(=C(C#N)C#N)/C(=C/c1cc(O)c(O)c(O)c1)/C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M08 compound treatment 213040.0 34800.0 2.37 209680.0 30300.0 2.26 3.2749 0.9997 3176140 HSCI1_000161 Nc1ncnc2n(cnc12)C3OC(CO)[C@H](O)[C@@H]3S 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M09 mock treatment 201920.0 23700.0 1.62 196920.0 17600.0 1.31 2.0673 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M10 mock treatment 191720.0 13500.0 0.92 194640.0 15300.0 1.14 1.4556 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M11 mock treatment 190280.0 12100.0 0.82 200880.0 21500.0 1.6 1.7146 0.952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M12 mock treatment 184160.0 5940.0 0.41 189440.0 10100.0 0.75 0.8175 0.9581 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M13 mock treatment 190240.0 12000.0 0.82 194120.0 14800.0 1.1 1.3569 0.9896 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M14 mock treatment 190000.0 11800.0 0.8 190000.0 10600.0 0.79 1.1285 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M15 compound treatment 250480.0 72300.0 4.93 244680.0 65300.0 4.86 6.9218 1.0 585 HSCI1_000162 Oc1ccc(C(=O)/C=C/c2ccc(O)c(O)c2)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M16 compound treatment 506400.0 328000.0 22.37 506200.0 327000.0 24.33 33.0225 0.9991 2024 HSCI1_000163 CN(N=O)c1cc(O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M17 compound treatment 496320.0 318000.0 21.69 489560.0 310000.0 23.09 31.6608 0.9995 569 HSCI1_000164 COC(=O)c1ccc(NCc2cc(O)ccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M18 compound treatment 326840.0 149000.0 10.13 328760.0 149000.0 11.12 15.028 0.9989 1890 HSCI1_000165 CN(N=O)c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M19 compound treatment 193960.0 15700.0 1.07 198040.0 18700.0 1.39 1.7425 0.9918 1008455 HSCI1_000166 BrCC(=O)c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M20 compound treatment 380360.0 202000.0 13.78 372120.0 193000.0 14.35 19.89 0.9998 3176141 HSCI1_000167 CCN(N=O)c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M21 compound treatment 271880.0 93700.0 6.39 262720.0 83400.0 6.2 8.9029 0.9999 560 HSCI1_000168 Oc1ccc(/C=C(\C#N)/C(=O)Nc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M22 compound treatment 323880.0 146000.0 9.93 302800.0 123000.0 9.19 13.519 0.9992 566 HSCI1_000169 COc1cc(/C=C(\C#N)/C(=O)N)cc(CSc2nc3ccccc3s2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M23 mock treatment 180320.0 2100.0 0.14 183880.0 4530.0 0.34 0.3398 0.9276 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 M24 mock treatment 172480.0 -5740.0 -0.39 173400.0 -5950.0 -0.44 -0.5897 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N01 mock treatment 182000.0 3780.0 0.26 180640.0 1290.0 0.1 0.2502 0.9091 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N02 compound treatment 211800.0 33600.0 2.29 218520.0 39200.0 2.92 3.6804 0.9929 837968 HSCI1_000170 Nc1ncnc2n(cnc12)C3CCCO3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N03 compound treatment 192640.0 14400.0 0.98 190320.0 11000.0 0.82 1.2726 0.9957 3176143 HSCI1_000171 CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)CCC(=O)O)[C@@]3(C)O[C@](C)(CC(=O)[C@@]32O)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N04 compound treatment 350920.0 173000.0 11.77 338880.0 160000.0 11.87 16.7214 1.0 831810 HSCI1_000172 Brc1c(Br)c(Br)c2[nH]nnc2c1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N05 compound treatment 329200.0 151000.0 10.29 312120.0 133000.0 9.88 14.266 0.9998 3054768 HSCI1_000173 C[C@H]1[C@H]2[C@H](Cc3ccccc3)NC(=O)[C@@]42OC(=O)/C=C\[C@H](O)CCC[C@@H](C)C/C=C\[C@H]4C(=O)C1=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N06 compound treatment 271400.0 93200.0 6.35 264280.0 84900.0 6.32 8.9618 1.0 3054769 HSCI1_000174 Cn1sc(=O)n(Cc2ccccc2)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N07 compound treatment 218760.0 40500.0 2.76 214800.0 35400.0 2.64 3.8201 0.9997 621 HSCI1_000175 CS(=O)c1ccc(cc1)c2nc(c([nH]2)c3ccncc3)c4cccc(I)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N08 compound treatment 208800.0 30600.0 2.09 207120.0 27800.0 2.07 2.9358 1.0 3054770 HSCI1_000176 c1ccc(cc1)c2n[nH]c3c2oc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N09 mock treatment 186680.0 8460.0 0.58 191760.0 12400.0 0.92 1.0611 0.9744 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N10 mock treatment 187320.0 9100.0 0.62 188960.0 9610.0 0.72 0.9446 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N11 mock treatment 185240.0 7020.0 0.48 192840.0 13500.0 1.0 1.0485 0.9427 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N12 mock treatment 192080.0 13900.0 0.95 191640.0 12300.0 0.91 1.3151 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N13 mock treatment 183640.0 5420.0 0.37 191120.0 11800.0 0.88 0.8808 0.9265 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N14 mock treatment 183320.0 5100.0 0.35 189880.0 10500.0 0.78 0.8001 0.9333 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N15 compound treatment 187120.0 8900.0 0.61 193320.0 14000.0 1.04 1.1644 0.9672 3176144 HSCI1_000177 CC1C2C(Cc3ccccc3)NC(=O)C42OC(=O)O/C=C\C(C)(O)C(=O)C(C)C/C=C\C4C5OC51C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N16 compound treatment 244360.0 66100.0 4.51 239880.0 60500.0 4.5 6.3742 1.0 1056418 HSCI1_000178 Nc1ncnc2n(cnc12)C3CCC(CO)O3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N17 compound treatment 196440.0 18200.0 1.24 195960.0 16600.0 1.24 1.7526 1.0 2177 HSCI1_000179 CC(C)CC[C@@H](O)[C@](C)(O)C1CC[C@@]2(O)C3=CC(=O)[C@]4(O)C[C@@H](O)[C@@H](O)C[C@]4(C)C3[C@H](O)C[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N18 compound treatment 382360.0 204000.0 13.92 377200.0 198000.0 14.73 20.2538 0.9996 3054771 HSCI1_000180 COc1ccc2NC(=O)/C(=C\c3c[nH]cn3)/c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N19 compound treatment 183440.0 5220.0 0.36 187280.0 7930.0 0.59 0.6691 0.9708 3176146 HSCI1_000181 CCCC(=O)O[C@@H]1[C@@H](C)[C@]2(O)[C@@H]3C=C(C)C(=O)[C@@]3(O)CC(=C[C@H]2[C@@H]4C(C)(C)[C@@]41OC(=O)CCC)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N20 compound treatment 190960.0 12700.0 0.87 185840.0 6490.0 0.48 0.9558 0.9616 2127 HSCI1_000182 CC1(C)CCC2=C(O1)c3ccccc3C(=O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N21 compound treatment 182320.0 4100.0 0.28 182120.0 2770.0 0.21 0.3435 0.9886 3054772 HSCI1_000183 CC(C)(O)/C=C/C(=O)[C@](C)(O)C1[C@H](O)C[C@@]2(C)[C@@H]3CC=C4C(C=C(O)C(=O)C4(C)C)[C@]3(C)C(=O)C[C@@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N22 compound treatment 247720.0 69500.0 4.74 240080.0 60700.0 4.52 6.5467 0.9997 1937872 HSCI1_000184 [O-][N+](=O)c1ccccc1c2ccc(C=C3C(=O)N(C(=S)N(C3=O)c4ccccc4)c5ccccc5)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N23 mock treatment 176480.0 -1740.0 -0.12 175680.0 -3670.0 -0.27 -0.2769 -0.9298 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 N24 mock treatment 171760.0 -6460.0 -0.44 172800.0 -6550.0 -0.49 -0.656 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O01 mock treatment 177720.0 -495.0 -0.03 177120.0 -2230.0 -0.17 -0.1414 -0.8338 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O02 mock treatment 175200.0 -3020.0 -0.21 183080.0 3730.0 0.28 0.0508 0.1472 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O03 compound treatment 203120.0 24900.0 1.7 203160.0 23800.0 1.77 2.4536 0.9998 5 HSCI1_000185 CC(C)(C)c1cc(C=C(C#N)C#N)cc(c1O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O04 compound treatment 201800.0 23600.0 1.61 203120.0 23800.0 1.77 2.3878 0.9989 2090 HSCI1_000186 CCOC(=O)C(C#N)C1C(=C(N)Oc2ccc(Br)cc12)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O05 compound treatment 321720.0 144000.0 9.78 333280.0 154000.0 11.46 15.019 0.9969 2107241 HSCI1_000187 ClC1=C(N2C(=O)CCC2=O)C(=O)c3ccccc3C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O06 compound treatment 204360.0 26100.0 1.78 204480.0 25100.0 1.87 2.5828 0.9997 651 HSCI1_000188 Nc1ncnc2n(ncc12)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O07 compound treatment 406840.0 229000.0 15.59 402200.0 223000.0 16.59 22.7496 0.9995 562 HSCI1_000189 Oc1ccc(/C=C(\C#N)/C(=O)c2ccc(O)c(O)c2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O08 compound treatment 189720.0 11500.0 0.78 192360.0 13000.0 0.97 1.2392 0.9945 3176147 HSCI1_000190 CS/C(=C(\C#N)/C(=C(\N)/SC)/[N+]#[C-])/N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O09 compound treatment 254800.0 76600.0 5.22 251200.0 71800.0 5.35 7.4732 0.9999 3176148 HSCI1_000191 OCc1cc2ncnc(Nc3ccc(O)cc3)c2cc1CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O10 compound treatment 225840.0 47600.0 3.25 223080.0 43700.0 3.25 4.5972 1.0 3054774 HSCI1_000192 Nc1ccc(cc1)c2cc(=O)c3cc(O)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O11 mock treatment 180880.0 2660.0 0.18 188080.0 8730.0 0.65 0.5878 0.8714 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O12 mock treatment 177840.0 -375.0 -0.03 186320.0 6970.0 0.52 0.3486 0.6714 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O13 mock treatment 207440.0 29200.0 1.99 210280.0 30900.0 2.3 3.0365 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O14 mock treatment 187320.0 9100.0 0.62 186240.0 6890.0 0.51 0.8014 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O15 compound treatment 207560.0 29300.0 2.0 205240.0 25900.0 1.93 2.7771 0.9998 3176208 HSCI1_000193 COc1ccc(N=O)c(CCc2cc(OC)ccc2N=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O16 compound treatment 182440.0 4220.0 0.29 189520.0 10200.0 0.76 0.7388 0.9124 3054775 HSCI1_000194 CC(C)(C)OC(=O)NC(CC(=O)O)C(=O)OCCF 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O17 compound treatment 221920.0 43700.0 2.98 221520.0 42200.0 3.14 4.3261 0.9997 1860 HSCI1_000195 CC(C)[C@@H]1N(C)c2cccc3[nH]cc(C[C@@H](CO)NC1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O18 compound treatment 462440.0 284000.0 19.38 465280.0 286000.0 21.28 28.7497 0.9989 634 HSCI1_000196 OC(=O)c1cc(NCc2cc(O)ccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O19 compound treatment 197000.0 18800.0 1.28 195200.0 15800.0 1.18 1.7396 0.9992 589 HSCI1_000197 Nc1cc(Nc2ccc(cc2)S(=O)(=O)N)ncn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O20 compound treatment 258720.0 80500.0 5.49 251840.0 72500.0 5.4 7.6959 1.0 3054776 HSCI1_000198 Oc1ccc2[nH]c(cc2c1)C(=O)c3cc4ccccc4[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O21 compound treatment 388840.0 211000.0 14.36 368000.0 189000.0 14.04 20.082 0.9999 557 HSCI1_000199 Cc1cc2ncc(nc2cc1C)c3ccc(O)c(O)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O22 compound treatment 383560.0 205000.0 14.0 387360.0 208000.0 15.48 20.8463 0.9987 1000586 HSCI1_000200 O/N=C\1/C(=C\2/C(=O)Nc3ccccc23)/Nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O23 mock treatment 171520.0 -6700.0 -0.46 172360.0 -6990.0 -0.52 -0.6908 -0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 O24 mock treatment 166120.0 -12100.0 -0.82 165400.0 -14000.0 -1.04 -1.3174 -0.9935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P01 mock treatment 181280.0 3060.0 0.21 178440.0 -912.0 -0.07 0.0997 0.454 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P02 mock treatment 179040.0 825.0 0.06 178520.0 -832.0 -0.06 -0.004 -0.0483 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P03 mock treatment 181800.0 3580.0 0.24 181320.0 1970.0 0.15 0.2764 0.97 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P04 mock treatment 187240.0 9020.0 0.62 180880.0 1530.0 0.11 0.5155 0.8238 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P05 mock treatment 185280.0 7060.0 0.48 184560.0 5210.0 0.39 0.6147 0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P06 mock treatment 178640.0 425.0 0.03 179960.0 608.0 0.05 0.0525 0.9767 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P07 mock treatment 182680.0 4460.0 0.3 182680.0 3330.0 0.25 0.3904 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P08 mock treatment 184960.0 6740.0 0.46 182000.0 2650.0 0.2 0.4645 0.9285 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P09 mock treatment 181120.0 2900.0 0.2 183520.0 4170.0 0.31 0.3594 0.9765 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P10 mock treatment 179240.0 1020.0 0.07 179400.0 47.9 0.0 0.0519 0.7422 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P11 mock treatment 180040.0 1820.0 0.12 180760.0 1410.0 0.1 0.1621 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P12 mock treatment 174720.0 -3500.0 -0.24 182840.0 3490.0 0.26 0.0151 0.0427 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P13 mock treatment 180000.0 1780.0 0.12 184000.0 4650.0 0.35 0.3306 0.9017 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P14 mock treatment 181720.0 3500.0 0.24 181360.0 2010.0 0.15 0.2746 0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P15 mock treatment 179120.0 905.0 0.06 180880.0 1530.0 0.11 0.124 0.9587 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P16 mock treatment 176800.0 -1420.0 -0.1 180080.0 728.0 0.05 -0.0299 -0.2704 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P17 mock treatment 179640.0 1420.0 0.1 176880.0 -2470.0 -0.18 -0.0614 -0.2952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P18 mock treatment 180360.0 2140.0 0.15 182360.0 3010.0 0.22 0.2617 0.9787 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P19 mock treatment 173360.0 -4860.0 -0.33 179000.0 -352.0 -0.03 -0.2526 -0.7607 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P20 mock treatment 172400.0 -5820.0 -0.4 175760.0 -3590.0 -0.27 -0.4694 -0.9816 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P21 mock treatment 173880.0 -4340.0 -0.3 174120.0 -5230.0 -0.39 -0.4844 -0.9907 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P22 mock treatment 173440.0 -4780.0 -0.33 173400.0 -5950.0 -0.44 -0.5435 -0.9885 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P23 mock treatment 165760.0 -12500.0 -0.85 165680.0 -13700.0 -1.02 -1.32 -0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2104 P24 mock treatment 165040.0 -13200.0 -0.9 166000.0 -13400.0 -0.99 -1.3379 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A01 mock treatment 190240.0 13100.0 0.89 180000.0 4310.0 0.32 0.8587 0.9043 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A02 mock treatment 166240.0 -10900.0 -0.74 165560.0 -10100.0 -0.75 -1.0583 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A03 mock treatment 166480.0 -10600.0 -0.73 167240.0 -8450.0 -0.63 -0.9583 -0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A04 mock treatment 173480.0 -3650.0 -0.25 165440.0 -10300.0 -0.76 -0.7156 -0.8915 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A05 mock treatment 212040.0 34900.0 2.38 206120.0 30400.0 2.26 3.2843 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A06 mock treatment 169320.0 -7810.0 -0.53 164480.0 -11200.0 -0.83 -0.9666 -0.9764 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A07 mock treatment 175360.0 -1770.0 -0.12 178520.0 2830.0 0.21 0.0634 0.2616 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A08 mock treatment 166120.0 -11000.0 -0.75 166040.0 -9650.0 -0.72 -1.0388 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A09 mock treatment 165640.0 -11500.0 -0.78 167160.0 -8530.0 -0.64 -1.003 -0.9946 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A10 mock treatment 166760.0 -10400.0 -0.71 167800.0 -7890.0 -0.59 -0.9153 -0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A11 mock treatment 170880.0 -6250.0 -0.43 167320.0 -8370.0 -0.62 -0.742 -0.9828 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A12 mock treatment 165680.0 -11400.0 -0.78 167480.0 -8210.0 -0.61 -0.9842 -0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A13 mock treatment 169280.0 -7850.0 -0.54 165960.0 -9730.0 -0.72 -0.8907 -0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A14 mock treatment 166240.0 -10900.0 -0.74 168520.0 -7170.0 -0.53 -0.9025 -0.9869 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A15 mock treatment 169440.0 -7690.0 -0.52 167720.0 -7970.0 -0.59 -0.7903 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A16 mock treatment 171200.0 -5930.0 -0.4 168000.0 -7690.0 -0.57 -0.6907 -0.9855 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A17 mock treatment 164360.0 -12800.0 -0.87 167720.0 -7970.0 -0.59 -1.0352 -0.9825 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A18 mock treatment 164880.0 -12200.0 -0.84 163000.0 -12700.0 -0.94 -1.2586 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A19 mock treatment 171160.0 -5970.0 -0.41 170840.0 -4850.0 -0.36 -0.5432 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A20 mock treatment 171520.0 -5610.0 -0.38 166160.0 -9530.0 -0.71 -0.7722 -0.9579 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A21 mock treatment 164920.0 -12200.0 -0.83 167360.0 -8330.0 -0.62 -1.0272 -0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A22 mock treatment 163720.0 -13400.0 -0.91 162240.0 -13500.0 -1.0 -1.3545 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A23 mock treatment 165880.0 -11200.0 -0.77 162640.0 -13100.0 -0.97 -1.2293 -0.9931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 A24 mock treatment 162520.0 -14600.0 -1.0 164240.0 -11500.0 -0.85 -1.3071 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B01 mock treatment 158280.0 -18800.0 -1.29 156720.0 -19000.0 -1.41 -1.9072 -0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B02 mock treatment 165600.0 -11500.0 -0.79 162680.0 -13000.0 -0.97 -1.2407 -0.9946 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B03 compound treatment 209480.0 32400.0 2.21 204760.0 29100.0 2.16 3.0893 1.0 577 HSCI1_000201 CN1C(=O)C(=C(C1=O)c2c[nH]c3ccccc23)c4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B04 compound treatment 216920.0 39800.0 2.71 223120.0 47400.0 3.53 4.4142 0.9915 614 HSCI1_000202 Cc1cc(O)c2c(=O)c3c(O)cc(O)c4c5c(O)cc(O)c6c(=O)c7c(O)cc(C)c8c1c2c(c34)c(c78)c65 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B05 compound treatment 170240.0 -6890.0 -0.47 170360.0 -5330.0 -0.4 -0.6128 -0.9965 907102 HSCI1_000203 NCCCCCCNS(=O)(=O)c1cccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B06 compound treatment 165120.0 -12000.0 -0.82 169520.0 -6170.0 -0.46 -0.9039 -0.9627 1012954 HSCI1_000204 OC(Cc1ccncc1)C(Cl)(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B07 compound treatment 187320.0 10200.0 0.69 183680.0 7990.0 0.59 0.9116 0.997 3176210 HSCI1_000205 CCCC(=O)Oc1ccc2[nH]c(cc2c1)C(=O)c3cc4ccccc4[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B08 compound treatment 176040.0 -1090.0 -0.07 171320.0 -4370.0 -0.33 -0.2827 -0.8467 321 HSCI1_000206 O=c1cc(oc2c(cccc12)c3ccccc3)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B09 compound treatment 186200.0 9070.0 0.62 187280.0 11600.0 0.86 1.047 0.9867 3176211 HSCI1_000207 C[C@@H](O)[C@]1(C)CC[C@@H](O1)[C@]2(C)CC[C@@H](C[C@H](O)[C@H](C)[C@H](O)[C@H](C)/C=C/C[C@@H](C)C[C@@H](C)/C(=C/C(=O)[C@@H](C)C[C@@H](C)C[C@H](C)CCC(=O)O)/O)O2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B10 compound treatment 168200.0 -8930.0 -0.61 165280.0 -10400.0 -0.78 -0.9785 -0.9929 3103895 HSCI1_000208 C[C@@H]1CC2C3CCC4=CC(=O)C=CC4(C)[C@@]3(F)[C@@H](O)CC2(C)[C@@]1(O)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B11 mock treatment 168520.0 -8610.0 -0.59 167680.0 -8010.0 -0.6 -0.8368 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B12 mock treatment 169960.0 -7170.0 -0.49 166160.0 -9530.0 -0.71 -0.8474 -0.9835 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B13 mock treatment 169440.0 -7690.0 -0.52 170320.0 -5370.0 -0.4 -0.6535 -0.9911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B14 mock treatment 163440.0 -13700.0 -0.93 168760.0 -6930.0 -0.52 -1.0248 -0.961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B15 compound treatment 217200.0 40100.0 2.73 227880.0 52200.0 3.88 4.6782 0.9852 1940 HSCI1_000209 NSC(=S)N1CCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B16 compound treatment 159680.0 -17400.0 -1.19 160400.0 -15300.0 -1.14 -1.6461 -0.9998 1000071 HSCI1_000210 C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B17 compound treatment 181480.0 4350.0 0.3 179400.0 3710.0 0.28 0.4048 0.9993 3176212 HSCI1_000211 Nc1ncnc2n(cnc12)C3OC(CO)[C@H](O)[C@@H]3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B18 compound treatment 162400.0 -14700.0 -1.0 162960.0 -12700.0 -0.95 -1.3802 -0.9996 831767 HSCI1_000212 NCCCNCCCCNCCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B19 compound treatment 177280.0 150.0 0.01 165080.0 -10600.0 -0.79 -0.5513 -0.6979 3054778 HSCI1_000213 NC(=O)c1ncn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c1N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B20 compound treatment 166280.0 -10800.0 -0.74 169240.0 -6450.0 -0.48 -0.8627 -0.9781 2293 HSCI1_000214 CSC(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B21 compound treatment 213760.0 36600.0 2.5 210200.0 34500.0 2.57 3.5819 0.9999 1001920 HSCI1_000215 CNC[C@H](O)c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B22 compound treatment 164160.0 -13000.0 -0.88 161120.0 -14600.0 -1.08 -1.3922 -0.9949 3054779 HSCI1_000216 CN/C(=N\C)/NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B23 mock treatment 164440.0 -12700.0 -0.87 164960.0 -10700.0 -0.8 -1.1766 -0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 B24 mock treatment 161320.0 -15800.0 -1.08 162080.0 -13600.0 -1.01 -1.4786 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C01 mock treatment 170040.0 -7090.0 -0.48 163600.0 -12100.0 -0.9 -0.9782 -0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C02 mock treatment 166800.0 -10300.0 -0.7 165800.0 -9890.0 -0.74 -1.0186 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C03 compound treatment 173720.0 -3410.0 -0.23 171720.0 -3970.0 -0.3 -0.3735 -0.9929 2022 HSCI1_000217 CC1(C)C(C=C(Br)Br)C1C(=O)OC(C#N)c2cccc(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C04 compound treatment 184160.0 7030.0 0.48 175840.0 147.0 0.01 0.3466 0.723 3176214 HSCI1_000218 COc1ccc2c(cc(C)c3nnc(SCC(=O)Nc4cccc(c4)C(=O)C)n32)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C05 compound treatment 351600.0 174000.0 11.89 345680.0 170000.0 12.65 17.3569 0.9995 3054780 HSCI1_000219 CCCCc1c([nH]c2nccnc12)c3ccc(O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C06 compound treatment 177200.0 70.3 0.0 172440.0 -3250.0 -0.24 -0.1678 -0.693 3054781 HSCI1_000220 NC(=N)SCCc1ccc(OCc2ccc(cc2)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C07 compound treatment 273880.0 96800.0 6.6 275680.0 100000.0 7.44 9.9262 0.9982 360 HSCI1_000221 Oc1ccc(cc1)c2cc(=O)c3c(O)cc(O)cc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C08 compound treatment 295760.0 119000.0 8.09 274120.0 98400.0 7.33 10.8989 0.9988 2260 HSCI1_000222 Cc1cc(O)c2c(=O)c3c(O)cc(O)c4c5c(O)cc(O)c6c(=O)c7c(O)cc(CO)c8c1c2c(c34)c(c65)c78 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C09 compound treatment 173640.0 -3490.0 -0.24 170920.0 -4770.0 -0.36 -0.4194 -0.981 3054782 HSCI1_000223 O=c1cc(oc2c1ccc3ccccc32)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C10 compound treatment 182880.0 5750.0 0.39 183120.0 7430.0 0.55 0.6681 0.9858 3176215 HSCI1_000224 C1CCC(CC1)n2cnc3c(Nc4ccc(cc4)N5CCOCC5)nc(Oc6cccc7ccccc67)nc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C11 mock treatment 168320.0 -8810.0 -0.6 170120.0 -5570.0 -0.41 -0.718 -0.9837 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C12 mock treatment 176440.0 -690.0 -0.05 168360.0 -7330.0 -0.55 -0.4192 -0.7652 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C13 mock treatment 171320.0 -5810.0 -0.4 172440.0 -3250.0 -0.24 -0.4513 -0.9721 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C14 mock treatment 173960.0 -3170.0 -0.22 175520.0 -173.0 -0.01 -0.1619 -0.748 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C15 mock treatment 192880.0 15800.0 1.07 191400.0 15700.0 1.17 1.5859 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C16 mock treatment 166000.0 -11100.0 -0.76 168160.0 -7530.0 -0.56 -0.933 -0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C17 compound treatment 182840.0 5710.0 0.39 186840.0 11100.0 0.83 0.8619 0.9405 3176216 HSCI1_000225 CCCCCCCCCCCCCCCCC(=C)OOCC(COP(=O)(ON)O[C@@H]1[C@H](O)[C@H](O)[C@@H](OP(=O)(O)ON)[C@H](OP(=O)(O)ON)[C@H]1O)OOC(=C)CC/C=C/C/C=C/C\C=C\C\C=C\CCCCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C18 compound treatment 172040.0 -5090.0 -0.35 165560.0 -10100.0 -0.75 -0.7787 -0.9379 907140 HSCI1_000226 NCCCCNS(=O)(=O)c1ccc2ccccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C19 compound treatment 202320.0 25200.0 1.72 197040.0 21300.0 1.59 2.3378 0.9992 3054783 HSCI1_000227 Nc1nc2n(cnc2c(=O)[nH]1)C3OC(COP(=O)(O)OP(=S)(O)O)[C@H](O)[C@@H]3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C20 compound treatment 197640.0 20500.0 1.4 190840.0 15100.0 1.13 1.7859 0.9943 2081802 HSCI1_000228 CC[C@@]1(O)C(=O)OCc2c1cc3-c4nc5ccc(O)c(CN(C)C)c5cc4Cn3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C21 compound treatment 173760.0 -3370.0 -0.23 173600.0 -2090.0 -0.16 -0.2726 -0.9821 3176218 HSCI1_000229 Nc1nc2n(C3OC4COP(O)(O)OC4C3O)c(Br)nc2c(=O)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C22 compound treatment 200200.0 23100.0 1.57 205080.0 29400.0 2.19 2.6587 0.9869 3054784 HSCI1_000230 Nc1nc(Cl)nc2n(cnc12)C3C[C@@H](O)C(COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C23 compound treatment 162960.0 -14200.0 -0.97 166040.0 -9650.0 -0.72 -1.1911 -0.9894 1338 HSCI1_000231 CCCC(C(=O)OCCN(CC)CC)(c1ccccc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 C24 mock treatment 164520.0 -12600.0 -0.86 165360.0 -10300.0 -0.77 -1.1517 -0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D01 mock treatment 165560.0 -11600.0 -0.79 165400.0 -10300.0 -0.77 -1.0995 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D02 mock treatment 169440.0 -7690.0 -0.52 171040.0 -4650.0 -0.35 -0.6156 -0.9797 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D03 compound treatment 289320.0 112000.0 7.65 295080.0 119000.0 8.89 11.6916 0.9972 3176219 HSCI1_000232 O/N=C/1\C(=C/2\C(=O)Nc3cc(Br)ccc23)\Nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D04 compound treatment 229240.0 52100.0 3.55 219800.0 44100.0 3.28 4.8334 0.9992 3054785 HSCI1_000233 O=C1NC(=O)c2c1ccc(Nc3ccccc3)c2Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D05 compound treatment 179000.0 1870.0 0.13 179320.0 3630.0 0.27 0.281 0.9414 1277018 HSCI1_000234 COc1cc2ncnc(Nc3ccc(Oc4ccccc4)cc3)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D06 compound treatment 197760.0 20600.0 1.41 192320.0 16600.0 1.24 1.8696 0.998 1919 HSCI1_000235 CCCCCc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D07 compound treatment 169800.0 -7330.0 -0.5 175080.0 -613.0 -0.05 -0.3856 -0.7685 3176221 HSCI1_000236 C1C[C@H](N/C/2=N/CCCCCCCCCCC2)[C@@H](C1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D08 compound treatment 178040.0 910.0 0.06 174000.0 -1690.0 -0.13 -0.0452 -0.322 3054786 HSCI1_000237 OCC1OC([C@@H](O)[C@H]1O)n2cnc3cc(Cl)c(Cl)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D09 compound treatment 179880.0 2750.0 0.19 180240.0 4550.0 0.34 0.3719 0.9612 3176222 HSCI1_000238 COc1cc2ncnc(Nc3ccc(OCc4ccccc4)cc3)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D10 compound treatment 170880.0 -6250.0 -0.43 172680.0 -3010.0 -0.22 -0.4599 -0.9551 407 HSCI1_000239 [O-][N+](=O)c1cccc2c(Br)n[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D11 mock treatment 169120.0 -8010.0 -0.55 174040.0 -1650.0 -0.12 -0.4731 -0.8453 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D12 mock treatment 173680.0 -3450.0 -0.24 169760.0 -5930.0 -0.44 -0.4786 -0.9565 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D13 mock treatment 173640.0 -3490.0 -0.24 165840.0 -9850.0 -0.73 -0.6868 -0.8908 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D14 mock treatment 171440.0 -5690.0 -0.39 170600.0 -5090.0 -0.38 -0.5423 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D15 mock treatment 170760.0 -6370.0 -0.43 169000.0 -6690.0 -0.5 -0.6593 -0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D16 mock treatment 172080.0 -5050.0 -0.34 165560.0 -10100.0 -0.75 -0.7767 -0.9369 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D17 compound treatment 200640.0 23500.0 1.6 197520.0 21800.0 1.62 2.2821 1.0 3054787 HSCI1_000240 N/N=C(/N)\NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D18 compound treatment 169920.0 -7210.0 -0.49 179160.0 3470.0 0.26 -0.1651 -0.2975 907294 HSCI1_000241 CN(C)C(=N)NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D19 compound treatment 171560.0 -5570.0 -0.38 169400.0 -6290.0 -0.47 -0.5997 -0.9946 3176223 HSCI1_000242 CSC(=N)NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D20 compound treatment 171280.0 -5850.0 -0.4 170920.0 -4770.0 -0.36 -0.5332 -0.9983 3054789 HSCI1_000243 CNC(=N)NCCC[C@@H](N)C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D21 compound treatment 179760.0 2630.0 0.18 173960.0 -1730.0 -0.13 0.0356 0.1611 3176224 HSCI1_000244 OP(=O)(O)C(Cl)(Cl)P(=O)(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D22 compound treatment 175360.0 -1770.0 -0.12 170200.0 -5490.0 -0.41 -0.3744 -0.8783 3176225 HSCI1_000245 CNC(=N)NCCC[C@H](N)C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D23 compound treatment 168560.0 -8570.0 -0.58 164440.0 -11300.0 -0.84 -1.0054 -0.9845 2215 HSCI1_000246 CCCNC(=N)NCCCC(N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 D24 mock treatment 169160.0 -7970.0 -0.54 161720.0 -14000.0 -1.04 -1.1196 -0.9542 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E01 mock treatment 171600.0 -5530.0 -0.38 173760.0 -1930.0 -0.14 -0.3683 -0.9128 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E02 mock treatment 175640.0 -1490.0 -0.1 176040.0 347.0 0.03 -0.0536 -0.5113 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E03 mock treatment 184040.0 6910.0 0.47 179640.0 3950.0 0.29 0.5408 0.9741 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E04 mock treatment 186640.0 9510.0 0.65 177480.0 1790.0 0.13 0.5525 0.8347 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E05 compound treatment 277080.0 100000.0 6.81 269280.0 93600.0 6.97 9.7437 0.9999 3176226 HSCI1_000247 CCCCc1c([nH]c2nccnc12)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E06 compound treatment 172920.0 -4210.0 -0.29 172800.0 -2890.0 -0.22 -0.3552 -0.99 2371 HSCI1_000248 CCCCCCCCNC(=O)C(Cc1ccc(OCc2ccncc2)cc1)NC(=O)C3CCC(CN)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E07 compound treatment 230000.0 52900.0 3.6 236320.0 60600.0 4.51 5.7394 0.9938 1989 HSCI1_000249 Clc1[nH]c2ccccc2c1/C=C\3/C(=O)Nc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E08 compound treatment 179520.0 2390.0 0.16 175520.0 -173.0 -0.01 0.1061 0.6491 1416171 HSCI1_000250 OC(CN1CCNCC1)Cn2c3ccc(Br)cc3c4cc(Br)ccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E09 mock treatment 177520.0 390.0 0.03 177240.0 1550.0 0.12 0.1002 0.8482 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E10 mock treatment 183800.0 6670.0 0.45 176320.0 627.0 0.05 0.3545 0.7756 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E11 compound treatment 190160.0 13000.0 0.89 188880.0 13200.0 0.98 1.3222 0.9988 663 HSCI1_000251 Fc1ccc(cc1)c2nc3SCCn3c2c4ccncc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E12 compound treatment 184120.0 6990.0 0.48 183920.0 8230.0 0.61 0.7699 0.9923 1000089 HSCI1_000252 COC1C(C)OC(OC2CC(C)(O)C(C(=O)OC)c3cc4C(=O)c5c6OC7OC(C)(C(O)C(C7O)N(C)C)c6cc(O)c5C(=O)c4c(O)c23)C(OC)C1(C)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E13 compound treatment 205840.0 28700.0 1.96 191920.0 16200.0 1.21 2.238 0.9731 3054791 HSCI1_000253 Nc1nc2n(cnc2c(=O)[nH]1)C3OC4COP(O)(O)OC4C3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E14 compound treatment 184360.0 7230.0 0.49 180160.0 4470.0 0.33 0.5836 0.9816 3176276 HSCI1_000254 NCC[C@H](NC(=O)[C@@H](N)CCCNC(=N)N[N+](=O)[O-])C(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E15 mock treatment 168920.0 -8210.0 -0.56 171960.0 -3730.0 -0.28 -0.5923 -0.9478 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E16 mock treatment 181160.0 4030.0 0.27 178080.0 2390.0 0.18 0.3199 0.9777 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E17 mock treatment 176160.0 -970.0 -0.07 177840.0 2150.0 0.16 0.0662 0.383 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E18 mock treatment 179160.0 2030.0 0.14 179680.0 3990.0 0.3 0.3077 0.9398 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E19 compound treatment 191400.0 14300.0 0.97 181800.0 6110.0 0.45 1.0093 0.9399 1000095 HSCI1_000255 CC(O)C(O)[C@H]1CNc2nc(N)[nH]c(=O)c2N1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E20 compound treatment 176960.0 -170.0 -0.01 174440.0 -1250.0 -0.09 -0.0741 -0.7887 3054834 HSCI1_000256 NCCNC[C@@H](N)CCCNC(=N)N[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E21 compound treatment 200160.0 23000.0 1.57 198480.0 22800.0 1.7 2.3095 0.9993 423 HSCI1_000257 COC(=O)[C@@H](N)CCCNC(=N)N[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E22 compound treatment 178600.0 1470.0 0.1 172920.0 -2770.0 -0.21 -0.0751 -0.3272 2114444 HSCI1_000258 O=c1n(CCN2CCCCC2)c(=O)c3ccc4c5ccc6c(=O)n(CCN7CCCCC7)c(=O)c8ccc(c9ccc1c3c94)c5c86 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E23 compound treatment 173880.0 -3250.0 -0.22 173200.0 -2490.0 -0.19 -0.2879 -0.9961 832002 HSCI1_000259 CC(=N)NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 E24 mock treatment 166960.0 -10200.0 -0.69 166880.0 -8810.0 -0.66 -0.9541 -0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F01 mock treatment 172200.0 -4930.0 -0.34 169120.0 -6570.0 -0.49 -0.5836 -0.9832 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F02 mock treatment 180640.0 3510.0 0.24 171840.0 -3850.0 -0.29 -0.0336 -0.0899 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F03 mock treatment 180440.0 3310.0 0.23 174760.0 -933.0 -0.07 0.1105 0.4678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F04 mock treatment 181760.0 4630.0 0.32 174840.0 -853.0 -0.06 0.1783 0.5537 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F05 compound treatment 259520.0 82400.0 5.62 248040.0 72300.0 5.38 7.7793 0.9998 3176278 HSCI1_000260 CC(=O)O/N=C/1\C(=C/2\C(=O)Nc3cc(Br)ccc23)\Nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F06 compound treatment 179400.0 2270.0 0.15 177640.0 1950.0 0.14 0.2119 0.9995 1505 HSCI1_000261 CC(C)Cn1c(=O)n(C)c(=O)c2[nH]cnc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F07 compound treatment 280840.0 104000.0 7.07 288320.0 113000.0 8.38 10.927 0.9964 3054836 HSCI1_000262 COc1ccc(CNc2nc(nc3n(cnc23)C(C)C)N(CCO)CCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F08 compound treatment 180400.0 3270.0 0.22 180080.0 4390.0 0.33 0.3885 0.9827 1980 HSCI1_000263 CC1(C2CCC(O2)C1(C)C(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F09 mock treatment 178320.0 1190.0 0.08 177160.0 1470.0 0.11 0.1346 0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F10 mock treatment 184680.0 7550.0 0.51 182680.0 6990.0 0.52 0.7317 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F11 compound treatment 418080.0 241000.0 16.43 415840.0 240000.0 17.87 24.2542 0.9991 832084 HSCI1_000264 NS(=O)(=O)c1ccc(Nc2nc(OCC3CCCCC3)c4nc[nH]c4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F12 compound treatment 188400.0 11300.0 0.77 184560.0 8870.0 0.66 1.01 0.9971 445 HSCI1_000265 NC(=O)c1cccc(N)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F13 compound treatment 184280.0 7150.0 0.49 184960.0 9270.0 0.69 0.8324 0.9856 2194 HSCI1_000266 OS(=O)(=O)c1cc(c2c(NC(=O)c3cccc(c3)[N+](=O)[O-])ccc(c2c1)S(=O)(=O)O)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F14 compound treatment 184640.0 7510.0 0.51 180880.0 5190.0 0.39 0.635 0.9903 2025 HSCI1_000267 NCCCC(N)(C(F)F)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F15 mock treatment 179000.0 1870.0 0.13 178000.0 2310.0 0.17 0.2116 0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F16 mock treatment 178920.0 1790.0 0.12 179720.0 4030.0 0.3 0.2982 0.9216 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F17 mock treatment 178600.0 1470.0 0.1 177120.0 1430.0 0.11 0.146 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F18 mock treatment 172880.0 -4250.0 -0.29 176360.0 667.0 0.05 -0.1698 -0.5776 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F19 compound treatment 182880.0 5750.0 0.39 184160.0 8470.0 0.63 0.7228 0.9739 2259 HSCI1_000268 CN1CCc2cc3OCOc3cc2C(=O)Cc4ccc5OCOc5c4C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F20 compound treatment 180920.0 3790.0 0.26 177360.0 1670.0 0.12 0.2704 0.9435 2674 HSCI1_000269 N[C@@H](CCC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F21 compound treatment 177640.0 510.0 0.03 173200.0 -2490.0 -0.19 -0.1066 -0.5647 3176279 HSCI1_000270 CC[C@]1(O)C[C@H]2CN(C1)CCc3c([nH]c4ccccc34)[C@@](C2)(C(=O)OC)c5cc6c(cc5OC)N(C=O)[C@@H]7[C@@]86CCN9CC=C[C@@](CC)([C@H]98)[C@@H](OC(=O)C)[C@]7(O)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F22 compound treatment 190960.0 13800.0 0.94 183040.0 7350.0 0.55 1.0534 0.9664 2129 HSCI1_000271 OCC(O)C1OC(=O)C(=C1O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F23 compound treatment 176080.0 -1050.0 -0.07 175240.0 -453.0 -0.03 -0.0745 -0.9412 1000078 HSCI1_000272 COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 F24 mock treatment 169720.0 -7410.0 -0.51 165760.0 -9930.0 -0.74 -0.88 -0.9828 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G01 mock treatment 178760.0 1630.0 0.11 174280.0 -1410.0 -0.11 0.0042 0.0275 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G02 compound treatment 140760.0 -36400.0 -2.48 138360.0 -37300.0 -2.78 -3.7181 -0.9984 25 HSCI1_000273 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@@H](N)COP(=O)(O)OCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G03 mock treatment 191640.0 14500.0 0.99 184880.0 9190.0 0.68 1.183 0.9837 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G04 mock treatment 187760.0 10600.0 0.72 184840.0 9150.0 0.68 0.9938 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G05 mock treatment 192800.0 15700.0 1.07 196000.0 20300.0 1.51 1.8241 0.9856 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G06 mock treatment 181800.0 4670.0 0.32 186120.0 10400.0 0.78 0.7739 0.9226 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G07 compound treatment 187680.0 10600.0 0.72 307520.0 132000.0 9.81 7.4464 0.7569 3054838 HSCI1_000274 CC(C)(c1ccc(NS(=O)(=O)C(F)(F)F)cc1)c2ccc(cc2)C(C)(C)c3cccc(NS(=O)(=O)C(F)(F)F)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G08 compound treatment 186920.0 9790.0 0.67 190880.0 15200.0 1.13 1.2712 0.9684 546 HSCI1_000275 Cc1ncc2ccccc2c1C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G09 compound treatment 197840.0 20700.0 1.41 202000.0 26300.0 1.96 2.3829 0.9871 1947905 HSCI1_000276 Clc1ccc(CN2C(=O)C(=O)c3ccccc23)cc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G10 compound treatment 192120.0 15000.0 1.02 192320.0 16600.0 1.24 1.5977 0.9955 636 HSCI1_000277 C/C(=C(\C#N)/C(=O)Nc1cccc(F)c1)/O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G11 compound treatment 224680.0 47600.0 3.24 235040.0 59300.0 4.42 5.4156 0.9884 3176281 HSCI1_000278 COc1ccc(CNC(=O)Nc2ncc(s2)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G12 compound treatment 218200.0 41100.0 2.8 217440.0 41700.0 3.11 4.177 0.9987 3054840 HSCI1_000279 CC1OC(C[C@H]1O)n2cnc3c(N)ncnc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G13 compound treatment 195960.0 18800.0 1.28 198520.0 22800.0 1.7 2.1091 0.9905 2319 HSCI1_000280 CN(C)CC1Cc2ccccc2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G14 compound treatment 214480.0 37400.0 2.55 210360.0 34700.0 2.58 3.625 1.0 3176282 HSCI1_000281 N[C@@H](CCN/C(=N/O)/N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G15 compound treatment 182560.0 5430.0 0.37 183960.0 8270.0 0.62 0.6968 0.9705 2145 HSCI1_000282 NC(=N)NCCS 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G16 compound treatment 186680.0 9550.0 0.65 184720.0 9030.0 0.67 0.9355 0.9999 3583 HSCI1_000283 Cn1cc(NC(=O)c2cc(NC(=O)CNC(=N)N)cn2C)cc1C(=O)NCCC(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G17 mock treatment 184160.0 7030.0 0.48 183360.0 7670.0 0.57 0.7424 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G18 mock treatment 176520.0 -610.0 -0.04 179400.0 3710.0 0.28 0.1657 0.5939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G19 mock treatment 183200.0 6070.0 0.41 181600.0 5910.0 0.44 0.6035 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G20 mock treatment 182840.0 5710.0 0.39 183080.0 7390.0 0.55 0.664 0.9857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G21 compound treatment 214920.0 37800.0 2.58 202840.0 27100.0 2.02 3.2505 0.9928 1030173 HSCI1_000284 NC(=N)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G22 compound treatment 181320.0 4190.0 0.29 176120.0 427.0 0.03 0.2245 0.7809 3176283 HSCI1_000285 COc1cc(ccc1[n+]2nc(nn2c3ccc(cc3)[N+](=O)[O-])c4ccccc4)c5ccc(c(OC)c5)[n+]6nc(nn6c7ccc(cc7)[N+](=O)[O-])c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G23 compound treatment 180240.0 3110.0 0.21 173280.0 -2410.0 -0.18 0.0229 0.0825 469 HSCI1_000286 CCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 G24 mock treatment 173520.0 -3610.0 -0.25 169560.0 -6130.0 -0.46 -0.4968 -0.958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H01 mock treatment 174000.0 -3130.0 -0.21 173760.0 -1930.0 -0.14 -0.2526 -0.9816 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H02 compound treatment 176360.0 -770.0 -0.05 173240.0 -2450.0 -0.18 -0.1662 -0.8749 1594 HSCI1_000287 N[C@@H](CCCNC(=N)N[N+](=O)[O-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H03 mock treatment 181120.0 3990.0 0.27 185600.0 9910.0 0.74 0.7137 0.9082 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H04 mock treatment 188040.0 10900.0 0.74 181800.0 6110.0 0.45 0.8473 0.9721 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H05 mock treatment 183400.0 6270.0 0.43 183480.0 7790.0 0.58 0.7121 0.9888 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H06 mock treatment 183000.0 5870.0 0.4 184880.0 9190.0 0.68 0.7665 0.9675 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H07 compound treatment 193400.0 16300.0 1.11 193840.0 18100.0 1.35 1.7394 0.9952 3054842 HSCI1_000288 CSc1nc(c([nH]1)c2ccnc(NC(C)c3ccccc3)c2)c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H08 compound treatment 180680.0 3550.0 0.24 173040.0 -2650.0 -0.2 0.0315 0.1009 1961 HSCI1_000289 CC(C)(C)c1cc(O)c(cc1O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H09 compound treatment 323760.0 147000.0 10.0 323840.0 148000.0 11.03 14.8654 0.9988 572 HSCI1_000290 CN(C)CCCn1cc(C2=C(C(=O)NC2=O)c3c[nH]c4ccccc34)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H10 compound treatment 192400.0 15300.0 1.04 187480.0 11800.0 0.88 1.3565 0.9964 1907755 HSCI1_000291 COCc1nc2n(CC(C)C)c(=O)n(C)c(=O)c2[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H11 compound treatment 363720.0 187000.0 12.72 356320.0 181000.0 13.44 18.5012 0.9996 574 HSCI1_000292 NCCCn1cc(C2=C(C(=O)NC2=O)c3c[nH]c4ccccc34)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H12 compound treatment 219880.0 42800.0 2.91 214600.0 38900.0 2.9 4.1085 1.0 3176284 HSCI1_000293 COc1cc2C3CC[C@]4(C)[C@@H](O)CCC4C3CCc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H13 compound treatment 395200.0 218000.0 14.87 397000.0 221000.0 16.47 22.1597 0.9987 2195 HSCI1_000294 OS(=O)(=O)c1cc(c2c(NC(=O)c3cccc(NC(=O)Nc4cccc(c4)C(=O)Nc5ccc(c6cc(cc(c56)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O)c3)ccc(c2c1)S(=O)(=O)O)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H14 compound treatment 186280.0 9150.0 0.62 184240.0 8550.0 0.64 0.8909 1.0 1714 HSCI1_000295 CN(C)C(=N)NC(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H15 compound treatment 398280.0 221000.0 15.08 390320.0 215000.0 15.97 21.9566 0.9996 2197 HSCI1_000296 OS(=O)(=O)c1ccc(NC(=O)c2cc(NC(=O)Nc3cc(cc(c3)C(=O)Nc4ccc(cc4S(=O)(=O)O)S(=O)(=O)O)C(=O)Nc5ccc(cc5S(=O)(=O)O)S(=O)(=O)O)cc(c2)C(=O)Nc6ccc(cc6S(=O)(=O)O)S(=O)(=O)O)c(c1)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H16 compound treatment 187680.0 10600.0 0.72 185880.0 10200.0 0.76 1.0447 0.9997 3054849 HSCI1_000297 CCNC(=N)NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H17 mock treatment 185200.0 8070.0 0.55 182240.0 6550.0 0.49 0.7336 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H18 mock treatment 179120.0 1990.0 0.14 179400.0 3710.0 0.28 0.291 0.9466 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H19 mock treatment 179240.0 2110.0 0.14 183840.0 8150.0 0.61 0.5305 0.8513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H20 mock treatment 179720.0 2590.0 0.18 176680.0 987.0 0.07 0.1768 0.9244 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H21 compound treatment 236840.0 59700.0 4.07 225840.0 50100.0 3.73 5.5176 0.9991 3054896 HSCI1_000298 NC(=O)c1cn(C2OC(CO)[C@H](O)[C@@H]2O)c3ncnc(N)c13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H22 compound treatment 186440.0 9310.0 0.63 186040.0 10300.0 0.77 0.9934 0.9954 2063 HSCI1_000299 CCOC(=O)c1cnc2n(CC)ncc2c1NN=C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H23 compound treatment 215320.0 38200.0 2.6 212200.0 36500.0 2.72 3.7624 0.9998 606 HSCI1_000300 CNCCNS(=O)(=O)c1cccc2cnccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 H24 mock treatment 169600.0 -7530.0 -0.51 172080.0 -3610.0 -0.27 -0.5532 -0.9545 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I01 mock treatment 173800.0 -3330.0 -0.23 174440.0 -1250.0 -0.09 -0.2265 -0.9228 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I02 compound treatment 184520.0 7390.0 0.5 184600.0 8910.0 0.66 0.825 0.9908 662 HSCI1_000301 Cc1nc(c(o1)c2ccncc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I03 compound treatment 189600.0 12500.0 0.85 190200.0 14500.0 1.08 1.3646 0.993 3054901 HSCI1_000302 Clc1cc(Cl)c(NC(=O)Nc2ccncc2)c(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I04 compound treatment 393240.0 216000.0 14.73 384320.0 209000.0 15.53 21.3979 0.9997 2110413 HSCI1_000303 Cc1cc(C)c(/C=C/2\C(=O)Nc3ccccc23)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I05 mock treatment 192080.0 15000.0 1.02 186840.0 11100.0 0.83 1.3074 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I06 mock treatment 188320.0 11200.0 0.76 177720.0 2030.0 0.15 0.6461 0.8308 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I07 mock treatment 185560.0 8430.0 0.57 189800.0 14100.0 1.05 1.1488 0.9598 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I08 mock treatment 187240.0 10100.0 0.69 180080.0 4390.0 0.33 0.7183 0.9417 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I09 compound treatment 192320.0 15200.0 1.04 188920.0 13200.0 0.98 1.4284 0.9997 2023 HSCI1_000304 CCCCn1c(=O)n(CCCC)c2ncn(CC(=O)C)c2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I10 compound treatment 491200.0 314000.0 21.41 493960.0 318000.0 23.69 31.8905 0.9987 2196 HSCI1_000305 OS(=O)(=O)c1cc(c2c(NC(=O)c3ccc(NC(=O)c4ccc(NC(=O)Nc5ccc(cc5)C(=O)Nc6ccc(cc6)C(=O)Nc7ccc(c8cc(cc(c78)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O)cc4)cc3)ccc(c2c1)S(=O)(=O)O)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I11 compound treatment 234360.0 57200.0 3.9 237800.0 62100.0 4.62 6.0275 0.9964 3054905 HSCI1_000306 Oc1ccc(cc1O)C(=O)/C(=C/c2ccc3oc(=O)[nH]c3c2)/C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I12 compound treatment 188680.0 11600.0 0.79 188120.0 12400.0 0.92 1.2108 0.9968 3054907 HSCI1_000307 Cc1nc2cc3nc(cnc3cc2n1C)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I13 compound treatment 190920.0 13800.0 0.94 185480.0 9790.0 0.73 1.1799 0.992 3479224 HSCI1_000308 CC(=N)NCCCCC(N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I14 compound treatment 276080.0 99000.0 6.75 283560.0 108000.0 8.03 10.447 0.9963 2061 HSCI1_000309 Oc1cc(c2cc(ccc2c1N=Nc3ccc4ccccc4c3O)[N+](=O)[O-])S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I15 compound treatment 199120.0 22000.0 1.5 197040.0 21300.0 1.59 2.1835 0.9996 2087 HSCI1_000310 NC(CCC(=O)NC(CSN=O)C(=O)NCC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I16 compound treatment 183280.0 6150.0 0.42 181920.0 6230.0 0.46 0.6242 0.9988 1870 HSCI1_000311 NC(=N)SCCc1cccc(CCSC(=N)N)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I17 compound treatment 205360.0 28200.0 1.92 207160.0 31500.0 2.34 3.017 0.9953 2408 HSCI1_000312 NCCC(O)(P(=O)(O)O)P(=O)(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I18 compound treatment 180920.0 3790.0 0.26 175200.0 -493.0 -0.04 0.1568 0.6006 3054955 HSCI1_000313 Cc1ccc(cc1)S(=O)(=O)N[C@H](CCCCN)C(=O)CCl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I19 mock treatment 179840.0 2710.0 0.18 182480.0 6790.0 0.51 0.4878 0.907 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I20 mock treatment 180040.0 2910.0 0.2 180440.0 4750.0 0.35 0.3901 0.9628 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I21 mock treatment 188400.0 11300.0 0.77 182000.0 6310.0 0.47 0.8752 0.972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I22 mock treatment 182200.0 5070.0 0.35 176480.0 787.0 0.06 0.2858 0.8153 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I23 compound treatment 194280.0 17200.0 1.17 183920.0 8230.0 0.61 1.2597 0.9544 1956 HSCI1_000314 N[C@H](CSCCB(O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 I24 mock treatment 170440.0 -6690.0 -0.46 168000.0 -7690.0 -0.57 -0.7274 -0.9936 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J01 mock treatment 176600.0 -530.0 -0.04 176600.0 907.0 0.07 0.0222 0.2898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J02 compound treatment 262280.0 85200.0 5.81 266160.0 90500.0 6.73 8.866 0.9973 1005830 HSCI1_000315 Cc1cc(ccc1N=Nc2cc(c3ccccc3c2N)S(=O)(=O)O)c4ccc(N=Nc5cc(c6ccccc6c5N)S(=O)(=O)O)c(C)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J03 compound treatment 347040.0 170000.0 11.58 333880.0 158000.0 11.77 16.5161 1.0 573 HSCI1_000316 CN1CCCC1CCn2cc(C3=C(C(=O)NC3=O)c4c[nH]c5ccccc45)c6ccccc26 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J04 compound treatment 202600.0 25500.0 1.74 197840.0 22100.0 1.65 2.3934 0.9997 1038990 HSCI1_000317 FC(F)(F)c1ccc2Sc3ccccc3N(CCCN4CCN(CCCl)CC4)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J05 mock treatment 186800.0 9670.0 0.66 181920.0 6230.0 0.46 0.7939 0.9851 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J06 mock treatment 182360.0 5230.0 0.36 182040.0 6350.0 0.47 0.5862 0.9904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J07 mock treatment 186520.0 9390.0 0.64 183440.0 7750.0 0.58 0.8604 0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J08 mock treatment 189040.0 11900.0 0.81 183760.0 8070.0 0.6 0.9987 0.989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J09 compound treatment 324000.0 147000.0 10.01 322680.0 147000.0 10.94 14.816 0.999 3054961 HSCI1_000318 OCc1cc2ncnc(Nc3cc(Br)c(O)c(Br)c3)c2cc1CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J10 compound treatment 263880.0 86800.0 5.91 263880.0 88200.0 6.56 8.8232 0.9986 1979 HSCI1_000319 Clc1ccc(cc1)C(c2ccc(Cl)cc2)[n+]3ccn(CC(OCc4ccc(Cl)cc4Cl)c5ccc(Cl)cc5Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J11 compound treatment 253200.0 76100.0 5.19 246720.0 71000.0 5.29 7.4052 1.0 580 HSCI1_000320 Cn1cc(C2=C(C(=O)NC2=O)c3cn(CCCN)c4ccccc34)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J12 compound treatment 183000.0 5870.0 0.4 183120.0 7430.0 0.55 0.6738 0.9874 3054964 HSCI1_000321 CC(=O)O[C@H]1[C@@H](O)[C@H]2C(C)(C)CCC[C@]2(C)C3C(=O)C[C@@](C)(O[C@]13C)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J13 compound treatment 184760.0 7630.0 0.52 182760.0 7070.0 0.53 0.7397 1.0 907101 HSCI1_000322 NCCCCNS(=O)(=O)c1ccc2c(Cl)cccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J14 compound treatment 185760.0 8630.0 0.59 186280.0 10600.0 0.79 0.9732 0.9897 3176334 HSCI1_000323 CC(C)[C@@]1(C)[C@@H]([C@H](OO)c2ccc[nH]2)[C@]3(O)[C@]4(O)[C@@]1(C)[C@@]5(O)C[C@@]3(C)[C@@]6(O)CCC(=C)[C@@H](O)[C@]46O5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J15 compound treatment 491600.0 314000.0 21.44 489640.0 314000.0 23.37 31.6824 0.9991 3054966 HSCI1_000324 C[C@@H]1CNCCCN1S(=O)(=O)c2cccc3cncc(C)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J16 compound treatment 183840.0 6710.0 0.46 183040.0 7350.0 0.55 0.7101 0.9961 3176335 HSCI1_000325 CN1CCN(CCCC(=O)O[C@H]2[C@@H](O)[C@H]3C(C)(C)CC[C@H](O)[C@]3(C)[C@@]4(O)C(=O)C[C@@](C)(O[C@]24C)C=C)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J17 compound treatment 189440.0 12300.0 0.84 190160.0 14500.0 1.08 1.3548 0.9924 1049343 HSCI1_000326 CCC(C)C1NC(=O)C(NC(=O)c2c(N)c(=O)c(C)c3oc4c(C)ccc(C(=O)NC5C(C)OC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C6CCCN6C(=O)C(NC5=O)C(C)C)c4nc23)C(C)OC(=O)C(C(C)C)N(C)C(=O)CN(C)C(=O)C7CCCN7C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J18 compound treatment 176240.0 -890.0 -0.06 181480.0 5790.0 0.43 0.2616 0.6016 3054969 HSCI1_000327 C[C@@]12CCC(=O)C=C2CC[C@H]3[C@@H]4CC[C@H](C(=O)CO)[C@@]4(O)C[C@H](O)[C@@H]31 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J19 mock treatment 180880.0 3750.0 0.26 173840.0 -1850.0 -0.14 0.0833 0.2866 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J20 mock treatment 179000.0 1870.0 0.13 173800.0 -1890.0 -0.14 -0.0095 -0.0499 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J21 mock treatment 178120.0 990.0 0.07 175040.0 -653.0 -0.05 0.0134 0.1605 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J22 mock treatment 175520.0 -1610.0 -0.11 173080.0 -2610.0 -0.19 -0.2151 -0.9633 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J23 compound treatment 155520.0 -21600.0 -1.47 157880.0 -17800.0 -1.33 -1.9792 -0.9986 3054970 HSCI1_000328 NC(=NCCSSCCN=C(N)N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 J24 mock treatment 168360.0 -8770.0 -0.6 167880.0 -7810.0 -0.58 -0.834 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K01 mock treatment 175960.0 -1170.0 -0.08 181120.0 5430.0 0.4 0.2292 0.5567 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K02 compound treatment 191680.0 14600.0 0.99 193320.0 17600.0 1.31 1.6291 0.9905 637 HSCI1_000329 C/C(=C(\C#N)/C(=O)Nc1ccc(OC(F)(F)F)cc1)/O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K03 compound treatment 271040.0 93900.0 6.4 240560.0 64900.0 4.83 7.941 0.9903 391 HSCI1_000330 Clc1ccc2NC(=O)CSC(c3ccccc3Cl)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K04 compound treatment 198800.0 21700.0 1.48 195960.0 20300.0 1.51 2.1113 0.9999 3055003 HSCI1_000331 O=C1c2ccccc2-[n+]3ccc4c5ccccc5[nH]c4c13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K05 compound treatment 257200.0 80100.0 5.46 248680.0 73000.0 5.43 7.7012 1.0 3055004 HSCI1_000332 Fc1ccc(cc1)C(=O)/C=C/2\C(=O)Nc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K06 compound treatment 178000.0 870.0 0.06 172560.0 -3130.0 -0.23 -0.1229 -0.5109 3176336 HSCI1_000333 CC(C)(C)C(=O)Nc1ccc-2c(c1)C(=O)C(=O)c3ccccc32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K07 mock treatment 189160.0 12000.0 0.82 187400.0 11700.0 0.87 1.1961 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K08 mock treatment 187000.0 9870.0 0.67 183040.0 7350.0 0.55 0.8625 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K09 mock treatment 192640.0 15500.0 1.06 192960.0 17300.0 1.29 1.6564 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K10 mock treatment 187200.0 10100.0 0.69 187560.0 11900.0 0.88 1.11 0.9922 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K11 compound treatment 197160.0 20000.0 1.37 198320.0 22600.0 1.68 2.1564 0.9946 3055006 HSCI1_000334 COc1cccc(c1)c2cc(NCc3ccc4OCOc4c3)nc(N)n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K12 compound treatment 197520.0 20400.0 1.39 192200.0 16500.0 1.23 1.8517 0.9981 3176337 HSCI1_000335 COc1ccc(cc1)c2cnc3c(cnn3c2)c4ccsc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K13 compound treatment 198360.0 21200.0 1.45 192320.0 16600.0 1.24 1.8985 0.997 3055009 HSCI1_000336 CC1=C(O)C(=O)[C@H]2O[C@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K14 compound treatment 198080.0 21000.0 1.43 193080.0 17400.0 1.29 1.925 0.9988 1709 HSCI1_000337 NCCCC(O)(P(=O)(O)O)P(=O)(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K15 mock treatment 192440.0 15300.0 1.04 190000.0 14300.0 1.06 1.491 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K16 mock treatment 188320.0 11200.0 0.76 182920.0 7230.0 0.54 0.9198 0.9854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K17 compound treatment 179440.0 2310.0 0.16 187040.0 11300.0 0.84 0.7085 0.8248 3176338 HSCI1_000338 CCCCCCCCCCCCCCCCOCC(COCC(F)(F)F)OP(=O)(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K18 compound treatment 189160.0 12000.0 0.82 183240.0 7550.0 0.56 0.9771 0.9829 1932 HSCI1_000339 OP(=O)(O)Oc1cccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K19 compound treatment 178880.0 1750.0 0.12 180800.0 5110.0 0.38 0.3531 0.8865 95 HSCI1_000340 CCCCCC(O)/C=C/C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K20 compound treatment 172600.0 -4530.0 -0.31 169480.0 -6210.0 -0.46 -0.5454 -0.9807 3176339 HSCI1_000341 CC(C)[C@@H](C)/C=C/[C@@H](C)[C@H]1CC[C@H]2\C(=C\C=C/3\C[C@@H](O)C[C@H](O)C3=C)\CCC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K21 mock treatment 185200.0 8070.0 0.55 176360.0 667.0 0.05 0.4241 0.7678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K22 mock treatment 183440.0 6310.0 0.43 183960.0 8270.0 0.62 0.7393 0.9847 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K23 mock treatment 174440.0 -2690.0 -0.18 172840.0 -2850.0 -0.21 -0.2798 -0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 K24 mock treatment 173760.0 -3370.0 -0.23 168520.0 -7170.0 -0.53 -0.54 -0.929 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L01 mock treatment 171200.0 -5930.0 -0.4 173400.0 -2290.0 -0.17 -0.4066 -0.9265 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L02 compound treatment 201320.0 24200.0 1.65 190760.0 15100.0 1.12 1.9591 0.9823 594 HSCI1_000342 Cc1nc2sccn2c(=O)c1CCN3CCC(=C(c4ccccc4)c5ccc(F)cc5)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L03 compound treatment 489680.0 313000.0 21.31 490000.0 314000.0 23.39 31.6088 0.9989 581 HSCI1_000343 Cn1cc(C2=C(C(=O)NC2=O)c3c4CC(CN)CCn4c5ccccc35)c6ccccc16 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L04 compound treatment 332960.0 156000.0 10.62 318600.0 143000.0 10.64 15.0332 1.0 1002019 HSCI1_000344 COc1ccc2C3CC[C@]4(C)[C@H](CCC4C3CCc2c1)NCCCCCCN5C(=O)C=CC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L05 compound treatment 198320.0 21200.0 1.44 199720.0 24000.0 1.79 2.286 0.9944 3055016 HSCI1_000345 COc1cc2ncnc(N3CCN(CC3)C(=O)Nc4ccc(Oc5ccccc5)cc4)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L06 compound treatment 187480.0 10400.0 0.71 185600.0 9910.0 0.74 1.0203 0.9998 2348 HSCI1_000346 COc1ccc2C3CC[C@]4(C)[C@H](CCC4C3CCc2c1)NCCCCCCN5C(=O)CCC5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L07 mock treatment 181280.0 4150.0 0.28 188400.0 12700.0 0.95 0.8688 0.8801 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L08 mock treatment 185760.0 8630.0 0.59 186400.0 10700.0 0.8 0.9795 0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L09 mock treatment 187200.0 10100.0 0.69 187120.0 11400.0 0.85 1.0868 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L10 mock treatment 184000.0 6870.0 0.47 186360.0 10700.0 0.79 0.8926 0.9683 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L11 compound treatment 184680.0 7550.0 0.51 182160.0 6470.0 0.48 0.7043 0.9994 582 HSCI1_000347 CN(C)CC1CCn2c(C1)c(C3=C(C(=O)NC3=O)c4cn(C)c5ccccc45)c6ccccc26 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L12 compound treatment 203600.0 26500.0 1.8 198240.0 22500.0 1.68 2.4627 0.9993 595 HSCI1_000348 Fc1ccc(cc1)C(=C2CCN(CCn3c(=O)c4ccccc4[nH]c3=S)CC2)c5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L13 compound treatment 185120.0 7990.0 0.54 180280.0 4590.0 0.34 0.6266 0.9747 3176385 HSCI1_000349 NCC1OC(OC2C(N)CC(N)C(O)C2O[C@@H]3OC[C@H](COCC4OCC(O)C(O)C4N)[C@@H]3O)C(N)C(O)C1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L14 compound treatment 188520.0 11400.0 0.78 187320.0 11600.0 0.87 1.161 0.9985 3055065 HSCI1_000350 Nc1ncn([C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L15 mock treatment 187200.0 10100.0 0.69 182880.0 7190.0 0.53 0.8637 0.9924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L16 mock treatment 183680.0 6550.0 0.45 178400.0 2710.0 0.2 0.4582 0.9353 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L17 compound treatment 177560.0 430.0 0.03 179320.0 3630.0 0.27 0.2116 0.7794 372 HSCI1_000351 COc1ccc(CCN(C)CCCC(C#N)(C(C)C)c2cc(OC)c(OC)c(OC)c2)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L18 compound treatment 197040.0 19900.0 1.36 188440.0 12700.0 0.95 1.6307 0.9847 1367 HSCI1_000352 Cc1cc(O)ccc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L19 compound treatment 185760.0 8630.0 0.59 174280.0 -1410.0 -0.11 0.3417 0.5716 3055069 HSCI1_000353 CC/C(=C(\c1ccc(O)cc1)/c2ccc(OCCN(C)C)cc2)/c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L20 compound treatment 178560.0 1430.0 0.1 178760.0 3070.0 0.23 0.2303 0.9281 2237 HSCI1_000354 FS(=O)(=O)Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L21 mock treatment 178640.0 1510.0 0.1 175040.0 -653.0 -0.05 0.0384 0.3374 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L22 mock treatment 174280.0 -2850.0 -0.19 170760.0 -4930.0 -0.37 -0.397 -0.9557 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L23 mock treatment 187640.0 10500.0 0.72 173520.0 -2170.0 -0.16 0.3923 0.534 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 L24 mock treatment 168000.0 -9130.0 -0.62 164560.0 -11100.0 -0.83 -1.0261 -0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M01 mock treatment 175000.0 -2130.0 -0.15 176840.0 1150.0 0.09 -0.0423 -0.2513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M02 compound treatment 191480.0 14400.0 0.98 189920.0 14200.0 1.06 1.4405 0.9992 1900 HSCI1_000355 COc1ccc2ncnc(NCc3ccc4OCOc4c3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M03 compound treatment 364160.0 187000.0 12.75 366920.0 191000.0 14.23 19.0803 0.9985 3055072 HSCI1_000356 Cn1cc(/C=C/2\C(=O)Nc3ccc(cc23)S(=O)(=O)N)c4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M04 compound treatment 253240.0 76100.0 5.19 250920.0 75200.0 5.6 7.6282 0.9993 292 HSCI1_000357 O=C1NCc2c1c3c4ccccc4[nH]c3c5[nH]c6ccccc6c25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M05 compound treatment 416840.0 240000.0 16.34 415800.0 240000.0 17.87 24.1923 0.999 907290 HSCI1_000358 CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](O)[C@@]3(C)O[C@](C)(CC(=O)[C@@]32O)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M06 compound treatment 363520.0 186000.0 12.71 368880.0 193000.0 14.38 19.1525 0.9981 3055076 HSCI1_000359 NS(=O)(=O)c1ccc(N/C=C/2\C(=O)Nc3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M07 compound treatment 218960.0 41800.0 2.85 209640.0 33900.0 2.53 3.8031 0.9982 3055122 HSCI1_000360 OC(=O)c1ccc2c3nc4ccccc4n3c(=O)c5cccc1c52 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M08 compound treatment 388080.0 211000.0 14.38 390720.0 215000.0 16.0 21.4859 0.9986 3176387 HSCI1_000361 Nc1cccc(c1)c2cc3c(Oc4cccc(O)c4)ncnc3[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M09 mock treatment 314920.0 138000.0 9.39 325880.0 150000.0 11.18 14.5466 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M10 mock treatment 192640.0 15500.0 1.06 187080.0 11400.0 0.85 1.347 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M11 mock treatment 189800.0 12700.0 0.86 187720.0 12000.0 0.9 1.2437 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M12 mock treatment 186320.0 9190.0 0.63 188240.0 12500.0 0.93 1.1033 0.9812 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M13 mock treatment 189440.0 12300.0 0.84 191320.0 15600.0 1.16 1.4159 0.9872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M14 mock treatment 184840.0 7710.0 0.53 188440.0 12700.0 0.95 1.0425 0.9612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M15 compound treatment 239800.0 62700.0 4.27 244760.0 69100.0 5.14 6.6561 0.9958 2796 HSCI1_000362 CCCCCCCC/C=C\CCCCCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M16 compound treatment 203000.0 25900.0 1.76 198600.0 22900.0 1.7 2.4527 0.9999 3176388 HSCI1_000363 COC(=O)CC(O)(CCCC(C)(C)O)C(=O)O[C@H]1[C@@H]2c3cc4OCOc4cc3CCN5CCC[C@]25C=C1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M17 compound treatment 183840.0 6710.0 0.46 180520.0 4830.0 0.36 0.5775 0.9928 1000076 HSCI1_000364 CCCCCCCCCCCCCCCCCCOCC(COP(=O)(O)OCC[N+](C)(C)C)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M18 compound treatment 206680.0 29600.0 2.01 194320.0 18600.0 1.39 2.4048 0.9834 2058 HSCI1_000365 OC(=O)C1C(C2CCC1O2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M19 compound treatment 185480.0 8350.0 0.57 183840.0 8150.0 0.61 0.8313 0.9995 1000072 HSCI1_000366 CC(C)OP(=O)(F)OC(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M20 compound treatment 261080.0 84000.0 5.72 262680.0 87000.0 6.47 8.625 0.9981 3176389 HSCI1_000367 CC(=O)O[C@@H]1CC2[C@@]3(C)CCCC(C)(C)C3CC[C@@]2(C)C4CC=C(C=O)[C@H](C=O)[C@@]14C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M21 compound treatment 186280.0 9150.0 0.62 179520.0 3830.0 0.28 0.6425 0.9369 3176390 HSCI1_000368 CCCC(=O)OC1C(OC2COP(O)(O)OC12)n3cnc4c(=O)[nH]c(NOC(=C)CC)nc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M22 compound treatment 202600.0 25500.0 1.74 214880.0 39200.0 2.92 3.2902 0.9693 3055129 HSCI1_000369 CC#C[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CCC4=C3[C@H](C[C@@]21C)c5ccc(cc5)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M23 mock treatment 175600.0 -1530.0 -0.1 176560.0 867.0 0.06 -0.0281 -0.2295 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 M24 mock treatment 174720.0 -2410.0 -0.16 172240.0 -3450.0 -0.26 -0.2979 -0.9766 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N01 mock treatment 178000.0 870.0 0.06 179240.0 3550.0 0.26 0.2286 0.845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N02 compound treatment 443920.0 267000.0 18.19 436120.0 260000.0 19.38 26.5672 0.9995 600 HSCI1_000370 COC(=O)/C=C/c1cc(O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N03 compound treatment 205920.0 28800.0 1.96 198680.0 23000.0 1.71 2.5977 0.9977 630 HSCI1_000371 COc1ccc(cc1)S(=O)(=O)N(CCO)c2ccccc2CN(C)C/C=C/c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N04 compound treatment 199720.0 22600.0 1.54 200960.0 25300.0 1.88 2.4188 0.9951 2283 HSCI1_000372 CCCCCCCNS(=O)(=O)c1cccc2c(Cl)cccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N05 compound treatment 192720.0 15600.0 1.06 196480.0 20800.0 1.55 1.8455 0.9832 629 HSCI1_000373 COc1ccc(cc1)S(=O)(=O)Nc2ccccc2CN(C)C/C=C/c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N06 compound treatment 197240.0 20100.0 1.37 189440.0 13700.0 1.02 1.6929 0.9896 1884 HSCI1_000374 Cc1ccnc(N)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N07 compound treatment 204480.0 27400.0 1.86 204600.0 28900.0 2.15 2.8398 0.9975 1918023 HSCI1_000375 CC[n+]1c(/C=C/N(C)c2ccccc2)n(c3ccccc3)c4ccc(cc14)c5nc6ccccc6s5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N08 compound treatment 194240.0 17100.0 1.17 190040.0 14300.0 1.07 1.5799 0.999 2344 HSCI1_000376 FC(F)(F)C(=O)CC(=O)c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N09 mock treatment 196600.0 19500.0 1.33 191040.0 15300.0 1.14 1.7463 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N10 mock treatment 186320.0 9190.0 0.63 187240.0 11500.0 0.86 1.0507 0.9879 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N11 mock treatment 184760.0 7630.0 0.52 184880.0 9190.0 0.68 0.8513 0.9909 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N12 mock treatment 188760.0 11600.0 0.79 183240.0 7550.0 0.56 0.9578 0.9857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N13 mock treatment 184040.0 6910.0 0.47 184120.0 8430.0 0.63 0.7766 0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N14 mock treatment 184560.0 7430.0 0.51 185760.0 10100.0 0.75 0.888 0.9818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N15 compound treatment 186880.0 9750.0 0.66 186000.0 10300.0 0.77 1.0125 0.9975 1000048 HSCI1_000377 CC(C)COCC(CN(Cc1ccccc1)c2ccccc2)N3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N16 compound treatment 190240.0 13100.0 0.89 181640.0 5950.0 0.44 0.945 0.9474 2187 HSCI1_000378 O=C(NC1CCCCC1)NC2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N17 compound treatment 180280.0 3150.0 0.21 180600.0 4910.0 0.37 0.4101 0.968 2083 HSCI1_000379 CC(CCC(=O)NCC(=O)O)C1CCC2C3CCC4CC(O)CCC4(C)C3CC(O)C12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N18 compound treatment 177560.0 430.0 0.03 177760.0 2070.0 0.15 0.1295 0.8271 1934 HSCI1_000380 NNC(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N19 compound treatment 185200.0 8070.0 0.55 178280.0 2590.0 0.19 0.5252 0.901 30 HSCI1_000381 COC(=O)C1=C(C)NC(=C(C1c2ccccc2C(F)(F)F)[N+](=O)[O-])C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N20 compound treatment 268560.0 91400.0 6.23 278440.0 103000.0 7.65 9.815 0.9949 420 HSCI1_000382 CCN1C(=O)C=CC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N21 compound treatment 179160.0 2030.0 0.14 175400.0 -293.0 -0.02 0.0824 0.5883 3054850 HSCI1_000383 C[C@@]12C[C@H](O)[C@H]3[C@@H](CCC4=CC(=O)CC[C@]34C)[C@@H]2CC[C@@H]1C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N22 compound treatment 176840.0 -290.0 -0.02 173600.0 -2090.0 -0.16 -0.1241 -0.7904 2003 HSCI1_000384 CNC1CCc2cc(OC)c(OC)c(OC)c2-c3ccc(OC)c(=O)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N23 mock treatment 170160.0 -6970.0 -0.48 174440.0 -1250.0 -0.09 -0.402 -0.8301 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 N24 mock treatment 174600.0 -2530.0 -0.17 167600.0 -8090.0 -0.6 -0.5479 -0.8744 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O01 mock treatment 172240.0 -4890.0 -0.33 171920.0 -3770.0 -0.28 -0.4343 -0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O02 mock treatment 180360.0 3230.0 0.22 182160.0 6470.0 0.48 0.4961 0.9372 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O03 compound treatment 333640.0 157000.0 10.67 337240.0 162000.0 12.02 16.0469 0.9982 3054852 HSCI1_000385 O=C/1Nc2ccc(cc2\C1=C\c3ccc[nH]3)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O04 compound treatment 181880.0 4750.0 0.32 185160.0 9470.0 0.7 0.7272 0.9378 3176393 HSCI1_000386 Cn1nc(N)c2cn(C3OC(CO)C(O)C3O)c4ncnc1c24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O05 compound treatment 505440.0 328000.0 22.38 496640.0 321000.0 23.89 32.718 0.9995 3176394 HSCI1_000387 C1CCC(CC1)Nc2nc(Nc3ccc(cc3)N4CCOCC4)nc5[nH]cnc25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O06 compound treatment 318080.0 141000.0 9.61 324040.0 148000.0 11.04 14.6021 0.9976 575 HSCI1_000388 O=C1NC(=O)C(=C1c2c[nH]c3ccccc23)c4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O07 compound treatment 191960.0 14800.0 1.01 185440.0 9750.0 0.73 1.2279 0.9867 3176395 HSCI1_000389 CCCCN1C(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@@H](N2C1=O)c5ccc(OC)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O08 compound treatment 214120.0 37000.0 2.52 212160.0 36500.0 2.71 3.7024 0.9993 2116778 HSCI1_000390 CCOC(=O)c1cnc2oc3ccc(O)cc3c2c1c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O09 compound treatment 495600.0 318000.0 21.71 490520.0 315000.0 23.43 31.9215 0.9993 3176396 HSCI1_000391 CC(C)[C@H](CO)Nc1nc(Nc2cc(N)cc(Cl)c2)c3ncn(C(C)C)c3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O10 compound treatment 356520.0 179000.0 12.23 352040.0 176000.0 13.12 17.9288 0.9994 676 HSCI1_000392 COc1cc2ncnc(Nc3cccc(O)c3)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O11 mock treatment 188640.0 11500.0 0.78 179080.0 3390.0 0.25 0.7331 0.8895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O12 mock treatment 183840.0 6710.0 0.46 177520.0 1830.0 0.14 0.4196 0.8792 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O13 mock treatment 181360.0 4230.0 0.29 179040.0 3350.0 0.25 0.3801 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O14 mock treatment 182560.0 5430.0 0.37 186640.0 10900.0 0.81 0.8379 0.9363 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O15 compound treatment 180800.0 3670.0 0.25 182240.0 6550.0 0.49 0.5215 0.952 1398 HSCI1_000393 CC(C)CCCC(C)CCCC(C)CCCC1(C)CCc2c(C)c(OC(=O)C)c(C)c(C)c2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O16 compound treatment 213960.0 36800.0 2.51 210400.0 34700.0 2.58 3.6021 0.9999 2060355 HSCI1_000394 CC1=C(C=C)/C(=C/c2[nH]c(Cc3[nH]c(\C=C\4/NC(=O)C(=C4C)C=C)c(C)c3CCC(=O)O)c(CCC(=O)O)c2C)/NC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O17 compound treatment 204760.0 27600.0 1.88 200040.0 24300.0 1.81 2.6133 0.9998 1929 HSCI1_000395 Nc1cccc2c(=O)[nH]ccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O18 compound treatment 196280.0 19200.0 1.31 182080.0 6390.0 0.48 1.2593 0.9063 2286 HSCI1_000396 CCSC(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O19 compound treatment 170800.0 -6330.0 -0.43 172080.0 -3610.0 -0.27 -0.4953 -0.9741 23 HSCI1_000397 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@@H](N)COP(=O)(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O20 compound treatment 179240.0 2110.0 0.14 179320.0 3630.0 0.27 0.2926 0.9566 3054913 HSCI1_000398 Cc1ccc(cc1)S(=O)(=O)N[C@H](Cc2ccccc2)C(=O)CCl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O21 compound treatment 151160.0 -26000.0 -1.77 145520.0 -30200.0 -2.25 -2.8399 -0.9931 3176397 HSCI1_000399 CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2/C(=C/C=C/3\C[C@@H](O)C[C@H](O)C3=C)/CCC[C@@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O22 compound treatment 167600.0 -9530.0 -0.65 169280.0 -6410.0 -0.48 -0.7969 -0.9885 988 HSCI1_000400 COc1ccc2[nH]cc(CCNC(=O)C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O23 mock treatment 166960.0 -10200.0 -0.69 168960.0 -6730.0 -0.5 -0.8446 -0.9873 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 O24 mock treatment 165640.0 -11500.0 -0.78 164400.0 -11300.0 -0.84 -1.1482 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P01 mock treatment 174400.0 -2730.0 -0.19 175080.0 -613.0 -0.05 -0.1639 -0.8552 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P02 mock treatment 175440.0 -1690.0 -0.12 171720.0 -3970.0 -0.3 -0.2906 -0.9155 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P03 mock treatment 177360.0 230.0 0.02 177280.0 1590.0 0.12 0.0946 0.7941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P04 mock treatment 178600.0 1470.0 0.1 175440.0 -253.0 -0.02 0.0575 0.5642 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P05 mock treatment 184080.0 6950.0 0.47 179520.0 3830.0 0.28 0.5364 0.9703 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P06 mock treatment 181800.0 4670.0 0.32 178120.0 2430.0 0.18 0.3529 0.9639 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P07 mock treatment 176400.0 -730.0 -0.05 180440.0 4750.0 0.35 0.2146 0.6016 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P08 mock treatment 178920.0 1790.0 0.12 180800.0 5110.0 0.38 0.3551 0.8895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P09 mock treatment 179960.0 2830.0 0.19 179960.0 4270.0 0.32 0.361 0.9715 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P10 mock treatment 179880.0 2750.0 0.19 179320.0 3630.0 0.27 0.3234 0.9842 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P11 mock treatment 177720.0 590.0 0.04 175960.0 267.0 0.02 0.0425 0.9469 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P12 mock treatment 178040.0 910.0 0.06 176200.0 507.0 0.04 0.0705 0.9715 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P13 mock treatment 177800.0 670.0 0.05 174720.0 -973.0 -0.07 -0.0189 -0.2208 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P14 mock treatment 178480.0 1350.0 0.09 176320.0 627.0 0.05 0.0981 0.9503 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P15 mock treatment 175520.0 -1610.0 -0.11 181200.0 5510.0 0.41 0.2122 0.5001 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P16 mock treatment 176320.0 -810.0 -0.06 175680.0 -13.4 0.0 -0.0397 -0.7198 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P17 mock treatment 174640.0 -2490.0 -0.17 173200.0 -2490.0 -0.19 -0.2512 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P18 mock treatment 178320.0 1190.0 0.08 178600.0 2910.0 0.22 0.2104 0.9104 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P19 mock treatment 171880.0 -5250.0 -0.36 173960.0 -1730.0 -0.13 -0.3443 -0.905 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P20 mock treatment 170280.0 -6850.0 -0.47 172200.0 -3490.0 -0.26 -0.5141 -0.9618 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P21 mock treatment 171160.0 -5970.0 -0.41 166400.0 -9290.0 -0.69 -0.7769 -0.968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P22 mock treatment 167440.0 -9690.0 -0.66 170120.0 -5570.0 -0.41 -0.7604 -0.9749 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P23 mock treatment 169400.0 -7730.0 -0.53 170080.0 -5610.0 -0.42 -0.6681 -0.9934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2105 P24 mock treatment 164760.0 -12400.0 -0.84 161280.0 -14400.0 -1.07 -1.3549 -0.9929 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A01 compound treatment 173440.0 -4810.0 -0.33 164960.0 -13700.0 -1.02 -0.9536 -0.8895 3221174 PK04_130001 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N[C@@H]3[C@H](O)Cc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A02 compound treatment 164280.0 -14000.0 -0.95 168680.0 -9990.0 -0.74 -1.1994 -0.9925 3211805 PK04_130002 CO[C@H](CCO)[C@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A03 compound treatment 163840.0 -14400.0 -0.98 169760.0 -8910.0 -0.66 -1.1637 -0.9817 3221177 PK04_130003 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)NCc4ccccc4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A04 compound treatment 167680.0 -10600.0 -0.72 167720.0 -11000.0 -0.82 -1.086 -0.9981 3080218 PK04_130004 OCCC[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A05 compound treatment 202040.0 23800.0 1.62 166880.0 -11800.0 -0.88 0.5262 0.2853 3221180 PK04_130005 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccc(O)cc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A06 compound treatment 164320.0 -13900.0 -0.95 171240.0 -7430.0 -0.55 -1.0627 -0.9669 3211801 PK04_130006 CSc1ccc(NC(=O)O[C@H](CCCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A07 compound treatment 200880.0 22600.0 1.54 197400.0 18700.0 1.39 2.0765 0.9987 3221183 PK04_130007 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2O)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A08 compound treatment 187600.0 9350.0 0.64 185800.0 7130.0 0.53 0.8258 0.9958 3080220 PK04_130008 COc1ccc(NC(=O)O[C@@H](CC=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A09 compound treatment 201960.0 23700.0 1.62 184520.0 5850.0 0.44 1.4507 0.8666 3221185 PK04_130009 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccc(O)cc2)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A10 compound treatment 170640.0 -7610.0 -0.52 169960.0 -8710.0 -0.65 -0.8254 -0.9939 3080222 PK04_130010 CO[C@H](CCO)[C@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A11 compound treatment 194800.0 16600.0 1.13 185200.0 6530.0 0.49 1.1414 0.9291 3221188 PK04_130011 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccc(Cl)cc2)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A12 compound treatment 169680.0 -8570.0 -0.58 166400.0 -12300.0 -0.91 -1.059 -0.9767 3211814 PK04_130012 C[C@H](CCO)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A13 mock treatment 169600.0 -8650.0 -0.59 169960.0 -8710.0 -0.65 -0.8755 -0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A14 mock treatment 169360.0 -8890.0 -0.61 167080.0 -11600.0 -0.86 -1.0387 -0.9851 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A15 compound treatment 187960.0 9710.0 0.66 181760.0 3090.0 0.23 0.6306 0.8998 3221191 PK04_130013 OCCCCCCNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A16 compound treatment 182000.0 3750.0 0.26 181680.0 3010.0 0.22 0.339 0.9978 3080206 PK04_130014 CSc1ccc(NC(=O)O[C@H](CCCO)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A17 compound treatment 169720.0 -8530.0 -0.58 164080.0 -14600.0 -1.09 -1.1792 -0.9571 3221194 PK04_130015 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)N[C@@H]4[C@H](O)Cc5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A18 compound treatment 187000.0 8750.0 0.6 178160.0 -513.0 -0.04 0.3948 0.6605 3211690 PK04_130016 COc1ccc(NC(=O)O[C@H](CCCO)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A19 compound treatment 184160.0 5910.0 0.4 183080.0 4410.0 0.33 0.5169 0.9948 3221197 PK04_130017 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2F)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A20 compound treatment 166080.0 -12200.0 -0.83 162200.0 -16500.0 -1.23 -1.4536 -0.9819 3189020 PK04_130018 C[C@@H](C=C)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A21 compound treatment 172160.0 -6090.0 -0.42 166080.0 -12600.0 -0.94 -0.9563 -0.9329 2019329 PK04_130019 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N3CCCCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A22 compound treatment 173720.0 -4530.0 -0.31 173800.0 -4870.0 -0.36 -0.4748 -0.9968 3080190 PK04_130020 CO[C@@H](CCO)[C@@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A23 compound treatment 183560.0 5310.0 0.36 167040.0 -11600.0 -0.87 -0.3562 -0.3796 3221200 PK04_130021 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCCCC2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 A24 compound treatment 180360.0 2110.0 0.14 182680.0 4010.0 0.3 0.3126 0.9441 3211695 PK04_130022 CO[C@@H](CCO)[C@@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B01 compound treatment 166080.0 -12200.0 -0.83 166600.0 -12100.0 -0.9 -1.2221 -0.9992 3176327 PK04_130023 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B02 compound treatment 172960.0 -5290.0 -0.36 171760.0 -6910.0 -0.51 -0.6188 -0.9849 3221203 PK04_130024 C[C@@H]1[C@H]([C@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)O[C@@]14C(=O)N(c5ccccc54)c6ccccc6)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B03 compound treatment 183080.0 4830.0 0.33 186160.0 7490.0 0.56 0.6269 0.9685 3052745 PK04_130025 NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B04 compound treatment 179840.0 1590.0 0.11 172600.0 -6070.0 -0.45 -0.2429 -0.5227 3221205 PK04_130026 C[C@H]1[C@@H]([C@@H](CC(=O)N(CCO)Cc2ccccc2)O[C@]13C(=O)N(c4ccccc43)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B05 compound treatment 252440.0 74200.0 5.06 221920.0 43200.0 3.22 5.8526 0.9762 3176512 PK04_130027 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B06 compound treatment 168880.0 -9370.0 -0.64 170240.0 -8430.0 -0.63 -0.8955 -1.0 3221207 PK04_130028 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(C)c3ccccc32)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B07 compound treatment 223760.0 45500.0 3.1 217640.0 39000.0 2.9 4.2447 0.9994 3176123 PK04_130029 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B08 compound treatment 164200.0 -14000.0 -0.96 165960.0 -12700.0 -0.95 -1.3464 -1.0 3221209 PK04_130030 C[C@H]1[C@@H]([C@@H](CC(=O)N2CCC[C@H]2CO)O[C@]13C(=O)N(C)c4c3cc(C)cc4Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B09 compound treatment 171040.0 -7210.0 -0.49 170640.0 -8030.0 -0.6 -0.7703 -0.9953 3052645 PK04_130031 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B10 compound treatment 176080.0 -2170.0 -0.15 173520.0 -5150.0 -0.38 -0.3758 -0.9142 3221211 PK04_130032 C[C@@H]1[C@H]([C@H](CCn2cc(nn2)[C@H](O)c3ccccc3)O[C@@]14C(=O)N(C)c5ccccc54)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B11 compound treatment 172720.0 -5530.0 -0.38 170000.0 -8670.0 -0.65 -0.723 -0.9672 3052831 PK04_130033 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B12 compound treatment 193400.0 15200.0 1.03 194920.0 16200.0 1.21 1.5854 0.9969 3221213 PK04_130034 C[C@H]1[C@@H]([C@@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)O[C@]14C(=O)N(c5ccccc54)c6ccccc6)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B13 mock treatment 163080.0 -15200.0 -1.03 167520.0 -11200.0 -0.83 -1.3183 -0.9941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B14 mock treatment 169440.0 -8810.0 -0.6 170280.0 -8390.0 -0.62 -0.8664 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B15 compound treatment 177160.0 -1090.0 -0.07 174160.0 -4510.0 -0.34 -0.29 -0.8431 3176778 PK04_130035 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B16 compound treatment 179880.0 1630.0 0.11 184080.0 5410.0 0.4 0.3632 0.8699 3221214 PK04_130036 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(CC=C)c3ccccc32)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B17 compound treatment 177440.0 -810.0 -0.06 175320.0 -3350.0 -0.25 -0.2155 -0.8431 3176195 PK04_130037 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B18 compound treatment 170000.0 -8250.0 -0.56 168080.0 -10600.0 -0.79 -0.9552 -0.9863 3221216 PK04_130038 C[C@H]1[C@@H]([C@@H](CCn2cc(CCO)nn2)O[C@]13C(=O)N(CC=C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B19 compound treatment 183680.0 5430.0 0.37 177480.0 -1190.0 -0.09 0.199 0.5227 3052584 PK04_130039 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B20 compound treatment 167480.0 -10800.0 -0.73 161560.0 -17100.0 -1.27 -1.4198 -0.9658 3221218 PK04_130040 C[C@@H]1[C@H]([C@H](CC(=O)N2CCC[C@H]2CO)O[C@@]13C(=O)N(C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B21 compound treatment 197120.0 18900.0 1.29 163800.0 -14900.0 -1.11 0.127 0.0748 3176736 PK04_130041 CN(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B22 compound treatment 169840.0 -8410.0 -0.57 164520.0 -14200.0 -1.05 -1.1503 -0.9591 3221220 PK04_130042 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(C)c3c2cc(C)cc3Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B23 compound treatment 184680.0 6430.0 0.44 178560.0 -113.0 -0.01 0.304 0.6934 3052927 PK04_130043 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 B24 compound treatment 167000.0 -11200.0 -0.77 161920.0 -16800.0 -1.25 -1.424 -0.9728 3221222 PK04_130044 C[C@H]1[C@@H]([C@@H](CCn2cc(CCO)nn2)O[C@]13C(=O)N(c4ccccc43)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C01 compound treatment 170760.0 -7490.0 -0.51 169360.0 -9310.0 -0.69 -0.8512 -0.9887 3221224 PK04_130045 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)NCc3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C02 compound treatment 207920.0 29700.0 2.02 204240.0 25600.0 1.9 2.7759 0.9995 3211914 PK04_130046 COc1ccc(NC(=O)O[C@H]([C@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C03 compound treatment 171840.0 -6410.0 -0.44 170720.0 -7950.0 -0.59 -0.7276 -0.9889 3221227 PK04_130047 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCOCCOCCOCCOCC2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C04 compound treatment 172680.0 -5570.0 -0.38 170720.0 -7950.0 -0.59 -0.6871 -0.977 3211809 PK04_130048 CSc1ccc(NC(=O)O[C@@H]([C@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C05 compound treatment 198400.0 20200.0 1.37 190240.0 11600.0 0.86 1.5802 0.9747 2019446 PK04_130049 COC(CN(C)C(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2coc3ccccc3c2=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C06 compound treatment 174640.0 -3610.0 -0.25 174320.0 -4350.0 -0.32 -0.4031 -0.9908 3069417 PK04_130050 C[C@H](C=C)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C07 compound treatment 198920.0 20700.0 1.41 191160.0 12500.0 0.93 1.6536 0.9796 3221230 PK04_130051 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)Nc3ccc(O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C08 compound treatment 171520.0 -6730.0 -0.46 171640.0 -7030.0 -0.52 -0.6946 -0.9978 3080227 PK04_130052 CSc1ccc(NC(=O)O[C@H]([C@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C09 compound treatment 195040.0 16800.0 1.14 196320.0 17600.0 1.31 1.7382 0.9977 3221232 PK04_130053 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C10 compound treatment 180000.0 1750.0 0.12 177880.0 -793.0 -0.06 0.0426 0.3203 3080226 PK04_130054 COc1ccc(NC(=O)O[C@@H]([C@@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C11 mock treatment 172160.0 -6090.0 -0.42 173200.0 -5470.0 -0.41 -0.5816 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C12 mock treatment 169840.0 -8410.0 -0.57 172760.0 -5910.0 -0.44 -0.7166 -0.9915 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C13 compound treatment 172840.0 -5410.0 -0.37 175880.0 -2790.0 -0.21 -0.4078 -0.9632 3221235 PK04_130055 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)NCCCCCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C14 compound treatment 235280.0 57000.0 3.89 225240.0 46600.0 3.47 5.2001 0.9984 3080272 PK04_130056 OCCC[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C15 mock treatment 171920.0 -6330.0 -0.43 170560.0 -8110.0 -0.6 -0.7321 -0.9864 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C16 mock treatment 166520.0 -11700.0 -0.8 169080.0 -9590.0 -0.71 -1.0703 -0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C17 compound treatment 189760.0 11500.0 0.78 184640.0 5970.0 0.44 0.8689 0.9637 3221238 PK04_130057 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)Nc4ccc(O)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C18 compound treatment 235400.0 57200.0 3.9 231800.0 53100.0 3.95 5.5511 1.0 3080228 PK04_130058 OCCC[C@@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C19 compound treatment 195440.0 17200.0 1.17 193080.0 14400.0 1.07 1.5869 0.999 2019457 PK04_130059 Nc1ccccc1NC(=O)C2=C[C@@H](C[C@H](OCCCCO)O2)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C20 compound treatment 186320.0 8070.0 0.55 182280.0 3610.0 0.27 0.5789 0.9456 3080205 PK04_130060 OCCC[C@@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C21 compound treatment 231200.0 53000.0 3.61 213280.0 34600.0 2.58 4.3739 0.9863 3221241 PK04_130061 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N[C@@H]2[C@H](O)Cc3ccccc23)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C22 compound treatment 196320.0 18100.0 1.23 195560.0 16900.0 1.26 1.7599 1.0 3211908 PK04_130062 COc1ccc(NC(=O)O[C@@H]([C@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C23 compound treatment 165560.0 -12700.0 -0.87 165920.0 -12800.0 -0.95 -1.2829 -0.9989 2019323 PK04_130063 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)Nc3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 C24 compound treatment 165360.0 -12900.0 -0.88 160040.0 -18600.0 -1.39 -1.602 -0.9758 3211812 PK04_130064 C[C@@H](CCO)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D01 compound treatment 239400.0 61200.0 4.17 212640.0 34000.0 2.53 4.7356 0.9713 3175965 PK04_130065 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccc(I)cc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D02 compound treatment 183560.0 5310.0 0.36 178040.0 -633.0 -0.05 0.2227 0.6099 3221243 PK04_130066 COc1cc2c3N(C(=O)[C@@]42O[C@H](CCO)[C@H]([C@@H]4C)[Si](C)(C)F)C(C)(C)C=C(C)c3c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D03 compound treatment 179440.0 1190.0 0.08 177320.0 -1350.0 -0.1 -0.0138 -0.1069 3176379 PK04_130067 NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D04 compound treatment 175040.0 -3210.0 -0.22 168840.0 -9830.0 -0.73 -0.6722 -0.88 3221245 PK04_130068 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(C)c3ccccc32)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D05 compound treatment 250200.0 72000.0 4.91 256960.0 78300.0 5.83 7.5887 0.9963 3052839 PK04_130069 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D06 compound treatment 189760.0 11500.0 0.78 186120.0 7450.0 0.55 0.9468 0.9855 3221246 PK04_130070 C[C@@H]1[C@H]([C@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)O[C@@]14C(=O)N(C)c5c4cc(C)cc5Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D07 compound treatment 231600.0 53400.0 3.64 230200.0 51500.0 3.83 5.2837 0.9997 3176048 PK04_130071 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D08 compound treatment 172520.0 -5730.0 -0.39 174160.0 -4510.0 -0.34 -0.5137 -0.9972 3221248 PK04_130072 C[C@@H]1[C@H]([C@H](CC(=O)N2CCC[C@H]2CO)O[C@@]13C(=O)N(c4ccccc43)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D09 compound treatment 169360.0 -8890.0 -0.61 171040.0 -7630.0 -0.57 -0.8303 -0.9995 3175970 PK04_130073 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D10 compound treatment 181480.0 3230.0 0.22 177200.0 -1470.0 -0.11 0.0782 0.3179 3221250 PK04_130074 C[C@H]1[C@@H]([C@@H](CC(=O)N2CCC[C@H]2CO)O[C@]13C(=O)N(c4ccccc43)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D11 mock treatment 171040.0 -7210.0 -0.49 176280.0 -2390.0 -0.18 -0.4735 -0.9057 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D12 mock treatment 174760.0 -3490.0 -0.24 167520.0 -11200.0 -0.83 -0.7552 -0.8746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D13 compound treatment 178440.0 190.0 0.01 176480.0 -2190.0 -0.16 -0.1062 -0.6488 3176675 PK04_130075 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D14 compound treatment 178880.0 630.0 0.04 169440.0 -9230.0 -0.69 -0.4555 -0.6616 3221251 PK04_130076 C[C@@H]1[C@H]([C@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)O[C@@]14C(=O)N(C)c5ccccc54)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D15 mock treatment 167080.0 -11200.0 -0.76 169600.0 -9070.0 -0.68 -1.016 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D16 mock treatment 171600.0 -6650.0 -0.45 169960.0 -8710.0 -0.65 -0.7791 -0.9847 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D17 compound treatment 178000.0 -250.0 -0.02 172800.0 -5870.0 -0.44 -0.3211 -0.7341 3052531 PK04_130077 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D18 compound treatment 177080.0 -1170.0 -0.08 173920.0 -4750.0 -0.35 -0.3065 -0.8453 3221253 PK04_130078 C[C@H]1[C@@H]([C@@H](CCn2cc(CCO)nn2)O[C@]13C(=O)N(C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D19 compound treatment 195160.0 16900.0 1.15 197800.0 19100.0 1.42 1.8218 0.9945 3052793 PK04_130079 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D20 compound treatment 191000.0 12800.0 0.87 177360.0 -1310.0 -0.1 0.5456 0.6237 3221255 PK04_130080 C[C@H]1[C@@H]([C@@H](CCn2cc(nn2)[C@H](O)c3ccccc3)O[C@]14C(=O)N(C)c5ccccc54)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D21 compound treatment 265800.0 87600.0 5.97 218840.0 40200.0 2.99 6.3346 0.9489 3052828 PK04_130081 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D22 compound treatment 175320.0 -2930.0 -0.2 176800.0 -1870.0 -0.14 -0.2398 -0.9846 3221256 PK04_130082 C[C@@H]1[C@H]([C@H](CCn2cc(CCO)nn2)O[C@@]13C(=O)N(c4ccccc43)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D23 compound treatment 289720.0 111000.0 7.6 248480.0 69800.0 5.2 9.0476 0.9828 3052592 PK04_130083 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 D24 compound treatment 173440.0 -4810.0 -0.33 166560.0 -12100.0 -0.9 -0.8694 -0.9062 3221257 PK04_130084 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(C)c3c2cc(C)cc3Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E01 mock treatment 170640.0 -7610.0 -0.52 172280.0 -6390.0 -0.48 -0.7033 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E02 mock treatment 170200.0 -8050.0 -0.55 175040.0 -3630.0 -0.27 -0.5793 -0.9468 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E03 compound treatment 194000.0 15800.0 1.07 193960.0 15300.0 1.14 1.5638 0.9996 2019322 PK04_130085 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)Nc3ccccc3N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E04 compound treatment 198720.0 20500.0 1.4 197360.0 18700.0 1.39 1.9703 1.0 3080210 PK04_130086 CO[C@@H](CCO)[C@@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E05 compound treatment 208400.0 30200.0 2.06 203400.0 24700.0 1.84 2.7548 0.9985 3221259 PK04_130087 OCCCCCCNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E06 compound treatment 183320.0 5070.0 0.35 177640.0 -1030.0 -0.08 0.1901 0.5367 3211802 PK04_130088 OCCC[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E07 compound treatment 187920.0 9670.0 0.66 182680.0 4010.0 0.3 0.6771 0.9357 3221261 PK04_130089 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)NCc4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E08 compound treatment 200600.0 22400.0 1.52 195320.0 16600.0 1.24 1.9536 0.9947 3080219 PK04_130090 COc1ccc(NC(=O)O[C@H](CCCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E09 mock treatment 179760.0 1510.0 0.1 174120.0 -4550.0 -0.34 -0.1668 -0.471 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E10 mock treatment 177920.0 -330.0 -0.02 177800.0 -873.0 -0.06 -0.0618 -0.8993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E11 compound treatment 185760.0 7510.0 0.51 184360.0 5690.0 0.42 0.6614 0.9955 3221264 PK04_130091 COC(CN(C)C(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2cc(=O)n(c3ccccc3)n2C)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E12 compound treatment 199440.0 21200.0 1.44 193080.0 14400.0 1.07 1.7798 0.9892 3069920 PK04_130092 O[C@@H](CC=C)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E13 compound treatment 198960.0 20700.0 1.41 194160.0 15500.0 1.15 1.8135 0.9949 3221266 PK04_130093 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)Nc4ccccc4N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E14 compound treatment 200240.0 22000.0 1.5 196360.0 17700.0 1.32 1.9909 0.9979 3211678 PK04_130094 CO[C@H](CCO)[C@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E15 compound treatment 192240.0 14000.0 0.95 188600.0 9930.0 0.74 1.1969 0.992 3221269 PK04_130095 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)N4CCOCCOCCOCCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E16 compound treatment 292880.0 115000.0 7.82 283320.0 105000.0 7.79 11.0335 1.0 3211906 PK04_130096 CSc1ccc(NC(=O)O[C@@H]([C@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E17 mock treatment 179880.0 1630.0 0.11 178680.0 6.82 0.0 0.079 0.7103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E18 mock treatment 184360.0 6110.0 0.42 180600.0 1930.0 0.14 0.396 0.8988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E19 compound treatment 212880.0 34600.0 2.36 200000.0 21300.0 1.59 2.7919 0.9813 2019458 PK04_130097 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2O)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E20 compound treatment 206400.0 28200.0 1.92 192480.0 13800.0 1.03 2.0837 0.9571 3211804 PK04_130098 COc1ccc(NC(=O)O[C@@H](CCCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E21 compound treatment 244880.0 66600.0 4.54 228000.0 49300.0 3.67 5.8081 0.9944 3221271 PK04_130099 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2F)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E22 compound treatment 194160.0 15900.0 1.08 185520.0 6850.0 0.51 1.1273 0.9407 3211680 PK04_130100 CO[C@@H](CCO)[C@@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E23 compound treatment 207200.0 29000.0 1.97 194960.0 16300.0 1.21 2.2528 0.9726 2019464 PK04_130101 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCCCC2)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 E24 compound treatment 212040.0 33800.0 2.3 202800.0 24100.0 1.8 2.8987 0.9924 3211909 PK04_130102 CSc1ccc(NC(=O)O[C@H]([C@@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F01 mock treatment 169880.0 -8370.0 -0.57 171200.0 -7470.0 -0.56 -0.7968 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F02 mock treatment 174280.0 -3970.0 -0.27 170400.0 -8270.0 -0.62 -0.6268 -0.9319 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F03 compound treatment 185880.0 7630.0 0.52 184120.0 5450.0 0.41 0.6545 0.9924 3176785 PK04_130103 NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F04 compound treatment 199520.0 21300.0 1.45 192040.0 13400.0 0.99 1.7289 0.9831 3221273 PK04_130104 C[C@H]1[C@@H]([C@@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)O[C@]14C(=O)N(C)c5c4cc(C)cc5Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F05 compound treatment 243040.0 64800.0 4.42 236240.0 57600.0 4.28 6.1531 0.9999 3176500 PK04_130105 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F06 compound treatment 181640.0 3390.0 0.23 182960.0 4290.0 0.32 0.3891 0.9875 3221274 PK04_130106 C[C@@H]1[C@H]([C@H](CCn2cc(CCO)nn2)O[C@@]13C(=O)N(CC=C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F07 compound treatment 196120.0 17900.0 1.22 207160.0 28500.0 2.12 2.3607 0.9654 3052886 PK04_130107 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F08 compound treatment 186280.0 8030.0 0.55 178600.0 -73.2 -0.01 0.3833 0.7 3221275 PK04_130108 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(c3ccccc32)c4ccccc4)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F09 mock treatment 177760.0 -490.0 -0.03 170800.0 -7870.0 -0.59 -0.4379 -0.7462 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F10 mock treatment 185680.0 7430.0 0.51 175200.0 -3470.0 -0.26 0.1754 0.3085 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F11 compound treatment 196280.0 18000.0 1.23 188240.0 9570.0 0.71 1.3727 0.9663 3052654 PK04_130109 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F12 compound treatment 185440.0 7190.0 0.49 184120.0 5450.0 0.41 0.6333 0.9955 3221277 PK04_130110 C[C@H]1[C@@H]([C@@H](CC(=O)N(CCO)Cc2ccccc2)O[C@]13C(=O)N(C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F13 compound treatment 188560.0 10300.0 0.7 183080.0 4410.0 0.33 0.729 0.9398 3052647 PK04_130111 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F14 compound treatment 203720.0 25500.0 1.74 198360.0 19700.0 1.47 2.264 0.9964 3221279 PK04_130112 C[C@H]1[C@@H]([C@@H](CC(=O)N2Cc3ccccc3C[C@H]2CO)O[C@]14C(=O)N(C)c5ccccc54)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F15 compound treatment 193720.0 15500.0 1.05 190760.0 12100.0 0.9 1.3819 0.9969 3176113 PK04_130113 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F16 compound treatment 189560.0 11300.0 0.77 193840.0 15200.0 1.13 1.3435 0.9827 3221280 PK04_130114 C[C@H]1[C@@H]([C@@H](CCn2cc(nn2)[C@H](O)c3ccccc3)O[C@]14C(=O)N(CC=C)c5ccccc54)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F17 mock treatment 174640.0 -3610.0 -0.25 180160.0 1490.0 0.11 -0.0958 -0.3549 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F18 mock treatment 180640.0 2390.0 0.16 181800.0 3130.0 0.23 0.2798 0.9848 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F19 compound treatment 187320.0 9070.0 0.62 185760.0 7090.0 0.53 0.8102 0.9969 3052888 PK04_130115 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F20 compound treatment 195600.0 17400.0 1.18 185200.0 6530.0 0.49 1.1799 0.9227 3221282 PK04_130116 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(c3ccccc32)c4ccccc4)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F21 compound treatment 252280.0 74000.0 5.05 249000.0 70300.0 5.23 7.27 0.9998 3176499 PK04_130117 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F22 compound treatment 181640.0 3390.0 0.23 188600.0 9930.0 0.74 0.6859 0.886 3221283 PK04_130118 C[C@@H]1[C@H]([C@H](CC(=O)N(CCO)Cc2ccccc2)O[C@@]13C(=O)N(C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F23 compound treatment 247000.0 68800.0 4.69 246920.0 68200.0 5.08 6.906 0.9992 3175968 PK04_130119 CC(=O)NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 F24 compound treatment 191000.0 12800.0 0.87 185720.0 7050.0 0.52 0.9855 0.9707 3221284 PK04_130120 C[C@@H]1[C@H]([C@H](CC(=O)N2CCC[C@H]2CO)O[C@@]13C(=O)N(C)c4c3cc(C)cc4Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G01 compound treatment 180640.0 2390.0 0.16 182320.0 3650.0 0.27 0.3072 0.9702 2019328 PK04_130121 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N3CCOCCOCCOCCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G02 compound treatment 285520.0 107000.0 7.31 276920.0 98200.0 7.31 10.3418 1.0 3211907 PK04_130122 COc1ccc(NC(=O)O[C@@H]([C@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G03 mock treatment 179600.0 1350.0 0.09 186920.0 8250.0 0.61 0.4991 0.8042 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G04 mock treatment 183720.0 5470.0 0.37 181040.0 2370.0 0.18 0.3883 0.9414 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G05 compound treatment 185640.0 7390.0 0.5 181840.0 3170.0 0.24 0.5229 0.9401 3221285 PK04_130123 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)NCCCCCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G06 compound treatment 206920.0 28700.0 1.95 204720.0 26000.0 1.94 2.7529 1.0 3211815 PK04_130124 COc1ccc(NC(=O)O[C@H]([C@H](C)C=C)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G07 compound treatment 187920.0 9670.0 0.66 179920.0 1250.0 0.09 0.5318 0.7988 3221287 PK04_130125 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)NCc3ccccc3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G08 compound treatment 200160.0 21900.0 1.49 195760.0 17100.0 1.27 1.9555 0.9968 3211803 PK04_130126 CSc1ccc(NC(=O)O[C@@H](CCCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G09 compound treatment 190720.0 12500.0 0.85 189880.0 11200.0 0.83 1.191 1.0 3221289 PK04_130127 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)N4CCCCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G10 compound treatment 185440.0 7190.0 0.49 185280.0 6610.0 0.49 0.6943 1.0 3211807 PK04_130128 CO[C@@H](CCO)[C@@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G11 compound treatment 193240.0 15000.0 1.02 189640.0 11000.0 0.82 1.2998 0.9938 2019311 PK04_130129 COC(CN(C)C(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccc(cc2)C(=O)OC)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G12 compound treatment 224400.0 46200.0 3.15 221080.0 42400.0 3.16 4.4566 1.0 3211818 PK04_130130 COc1ccc(NC(=O)O[C@H](CCCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G13 compound treatment 207560.0 29300.0 2.0 198200.0 19500.0 1.45 2.4407 0.9878 3221292 PK04_130131 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)Nc4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G14 compound treatment 206040.0 27800.0 1.89 208640.0 30000.0 2.23 2.9168 0.9967 3080207 PK04_130132 OCCC[C@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G15 compound treatment 195080.0 16800.0 1.15 193000.0 14300.0 1.07 1.5654 0.9993 2019470 PK04_130133 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G16 compound treatment 196760.0 18500.0 1.26 193120.0 14400.0 1.08 1.6527 0.9968 3080225 PK04_130134 COc1ccc(NC(=O)O[C@H]([C@@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G17 compound treatment 213160.0 34900.0 2.38 203440.0 24800.0 1.84 2.9864 0.992 3221294 PK04_130135 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N[C@@H]2[C@H](O)Cc3ccccc23)c4coc5ccccc5c4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G18 compound treatment 186920.0 8670.0 0.59 189360.0 10700.0 0.8 0.9804 0.9893 3211806 PK04_130136 CO[C@@H](CCO)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G19 mock treatment 185160.0 6910.0 0.47 185200.0 6530.0 0.49 0.6766 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G20 mock treatment 186120.0 7870.0 0.54 180760.0 2090.0 0.16 0.4892 0.8758 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G21 compound treatment 194440.0 16200.0 1.1 191560.0 12900.0 0.96 1.4587 0.9975 2019463 PK04_130137 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCOCCOCCOCCOCC2)c3coc4ccccc4c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G22 compound treatment 220400.0 42200.0 2.87 214880.0 36200.0 2.69 3.9375 0.9995 3080280 PK04_130138 COc1ccc(NC(=O)O[C@H]([C@@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G23 compound treatment 185040.0 6790.0 0.46 180320.0 1650.0 0.12 0.414 0.8645 3221297 PK04_130139 Cn1c(cc(=O)n1c2ccccc2)[C@@H]3C[C@H](OCCCCO)OC(=C3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 G24 compound treatment 201840.0 23600.0 1.61 194400.0 15700.0 1.17 1.9649 0.9878 3211912 PK04_130140 C[C@H](CCO)[C@@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H01 compound treatment 192720.0 14500.0 0.99 188080.0 9410.0 0.7 1.1927 0.9859 3052931 PK04_130141 NCCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H02 compound treatment 187760.0 9510.0 0.65 182360.0 3690.0 0.27 0.6525 0.9268 3221300 PK04_130142 C[C@@H]1[C@H]([C@H](CCn2cc(CCO)nn2)O[C@@]13C(=O)N(C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H03 mock treatment 178480.0 230.0 0.02 177760.0 -913.0 -0.07 -0.0369 -0.5297 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H04 mock treatment 182040.0 3790.0 0.26 182840.0 4170.0 0.31 0.402 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H05 compound treatment 187440.0 9190.0 0.63 178680.0 6.82 0.0 0.4434 0.7077 3176330 PK04_130143 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H06 compound treatment 203680.0 25400.0 1.73 201280.0 22600.0 1.68 2.4157 0.9999 3221301 PK04_130144 C[C@@H]1[C@H]([C@H](CC(=O)N(CCO)Cc2ccccc2)O[C@@]13C(=O)N(c4ccccc43)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H07 compound treatment 287400.0 109000.0 7.44 290440.0 112000.0 8.32 11.144 0.9985 3176685 PK04_130145 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H08 compound treatment 188720.0 10500.0 0.71 184960.0 6290.0 0.47 0.8356 0.979 3221302 PK04_130146 C[C@H]1[C@@H]([C@@H](CC(=O)N2CCC[C@H]2CO)O[C@]13C(=O)N(C)c4ccccc43)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H09 compound treatment 190440.0 12200.0 0.83 185640.0 6970.0 0.52 0.9543 0.9742 3052879 PK04_130147 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H10 compound treatment 182320.0 4070.0 0.28 178760.0 86.8 0.01 0.2008 0.7234 3221303 PK04_130148 C[C@H]1[C@@H]([C@@H](CC(=O)N(CCO)Cc2ccccc2)O[C@]13C(=O)N(C)c4c3cc(C)cc4Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H11 compound treatment 191360.0 13100.0 0.89 189800.0 11100.0 0.83 1.2176 0.9993 3176775 PK04_130149 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H12 compound treatment 185000.0 6750.0 0.46 184320.0 5650.0 0.42 0.6226 0.999 3221305 PK04_130150 COc1cc2c3N(C(=O)[C@]42O[C@@H](CCO)[C@@H]([C@H]4C)[Si](C)(C)O)C(C)(C)C=C(C)c3c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H13 compound treatment 191640.0 13400.0 0.91 187560.0 8890.0 0.66 1.1132 0.9875 3052783 PK04_130151 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H14 compound treatment 201600.0 23400.0 1.59 200840.0 22200.0 1.65 2.2923 0.9998 3221307 PK04_130152 C[C@@H]1[C@H]([C@H](CCn2cc(nn2)[C@H](O)c3ccccc3)O[C@@]14C(=O)N(CC=C)c5ccccc54)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H15 compound treatment 197680.0 19400.0 1.32 189040.0 10400.0 0.77 1.4823 0.9669 3176626 PK04_130153 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H16 compound treatment 201680.0 23400.0 1.6 197240.0 18600.0 1.38 2.1067 0.9974 3221308 PK04_130154 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccccc32)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H17 compound treatment 216600.0 38400.0 2.61 213800.0 35100.0 2.61 3.6975 1.0 3176501 PK04_130155 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H18 compound treatment 178240.0 -9.55 0.0 182360.0 3690.0 0.27 0.1936 0.7054 3221309 PK04_130156 C[C@@H]1[C@H]([C@H](CC(=O)N(CCO)Cc2ccccc2)O[C@@]13C(=O)N(C)c4c3cc(C)cc4Br)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H19 mock treatment 178640.0 390.0 0.03 183360.0 4690.0 0.35 0.2655 0.7589 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H20 mock treatment 182280.0 4030.0 0.27 183920.0 5250.0 0.39 0.4704 0.9852 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H21 compound treatment 181160.0 2910.0 0.2 180000.0 1330.0 0.1 0.2101 0.9481 3052741 PK04_130157 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H22 compound treatment 203000.0 24800.0 1.69 205000.0 26300.0 1.96 2.5787 0.9972 3221310 PK04_130158 C[C@@H]1[C@H]([C@H](CCn2cc(nn2)[C@H](O)c3ccccc3)O[C@@]14C(=O)N(c5ccccc54)c6ccccc6)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H23 compound treatment 243320.0 65100.0 4.44 242840.0 64200.0 4.78 6.5139 0.9993 3176203 PK04_130159 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 H24 compound treatment 181160.0 2910.0 0.2 168760.0 -9910.0 -0.74 -0.3814 -0.4992 3221312 PK04_130160 C[C@H]1[C@@H]([C@@H](CCn2cc(nn2)[C@H](O)c3ccccc3)O[C@]14C(=O)N(c5ccccc54)c6ccccc6)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I01 compound treatment 198520.0 20300.0 1.38 202520.0 23800.0 1.77 2.2322 0.9923 3221313 PK04_130161 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccc(Cl)cc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I02 compound treatment 195840.0 17600.0 1.2 194160.0 15500.0 1.15 1.663 0.9998 3080209 PK04_130162 CO[C@H](CCO)[C@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I03 compound treatment 223680.0 45400.0 3.1 212240.0 33600.0 2.5 3.9567 0.9943 3221314 PK04_130163 Nc1ccccc1NC(=O)C2=C[C@@H](C[C@H](OCCCCO)O2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I04 compound treatment 198680.0 20400.0 1.39 193960.0 15300.0 1.14 1.7894 0.995 3069956 PK04_130164 CO[C@@H](C=C)[C@@H](O)c1ccc(OC)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I05 mock treatment 188760.0 10500.0 0.72 185320.0 6650.0 0.49 0.8565 0.9836 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I06 mock treatment 188280.0 10000.0 0.68 182120.0 3450.0 0.26 0.6649 0.9104 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I07 compound treatment 217360.0 39100.0 2.67 218240.0 39600.0 2.94 3.9678 0.9988 3221316 PK04_130165 COC(CN(C)C(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2cccs2)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I08 compound treatment 203920.0 25700.0 1.75 199000.0 20300.0 1.51 2.3073 0.9974 3211693 PK04_130166 CO[C@H](CCO)[C@H](O)c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I09 compound treatment 190520.0 12300.0 0.84 187480.0 8810.0 0.66 1.055 0.9927 2019335 PK04_130167 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I10 compound treatment 219520.0 41300.0 2.81 213120.0 34400.0 2.56 3.8024 0.9989 3080278 PK04_130168 CSc1ccc(NC(=O)O[C@@H]([C@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I11 compound treatment 207920.0 29700.0 2.02 194600.0 15900.0 1.19 2.2686 0.9676 3221318 PK04_130169 COc1cc2c[n+](Cc3cc4OCOc4cc3Br)ccc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I12 compound treatment 216200.0 38000.0 2.59 213680.0 35000.0 2.61 3.6719 1.0 3211911 PK04_130170 COc1ccc(NC(=O)O[C@@H]([C@@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I13 compound treatment 192840.0 14600.0 0.99 189920.0 11200.0 0.84 1.2953 0.9963 3221319 PK04_130171 COc1cc2c[n+](Cc3sc4ccccc4c3Cl)ccc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I14 compound treatment 198960.0 20700.0 1.41 197760.0 19100.0 1.42 2.0029 1.0 3080208 PK04_130172 COc1ccc(NC(=O)O[C@@H](CCCO)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I15 compound treatment 191560.0 13300.0 0.91 189840.0 11200.0 0.83 1.2294 0.999 3221320 PK04_130173 COc1cc2c[n+](Cc3ccc(o3)[N+](=O)[O-])ccc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I16 compound treatment 185360.0 7110.0 0.48 186520.0 7850.0 0.58 0.7557 0.9957 3080223 PK04_130174 CO[C@@H](CCO)[C@@H](OC(=O)Nc1ccc(OC)cc1)c2ccc(OCCO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I17 compound treatment 185040.0 6790.0 0.46 187280.0 8610.0 0.64 0.7803 0.9873 3221321 PK04_130175 COc1cc2c[n+](Cc3cccc(OC(F)(F)F)c3)ccc2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I18 compound treatment 310880.0 133000.0 9.04 299440.0 121000.0 8.99 12.7496 1.0 3080282 PK04_130176 CSc1ccc(NC(=O)O[C@H]([C@H](C)C=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I19 compound treatment 196000.0 17800.0 1.21 198320.0 19600.0 1.46 1.8897 0.9956 3221322 PK04_130177 COP(=O)(OC)/N=C\1/CC(=CC(N1Cc2cccc(OC(F)(F)F)c2)c3cccs3)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I20 compound treatment 198880.0 20600.0 1.41 194800.0 16100.0 1.2 1.8433 0.9969 3211594 PK04_130178 CO[C@H](C=C)[C@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I21 mock treatment 178280.0 30.5 0.0 179040.0 367.0 0.03 0.0208 0.7587 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I22 mock treatment 178880.0 630.0 0.04 177400.0 -1270.0 -0.09 -0.0366 -0.3519 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I23 compound treatment 233560.0 55300.0 3.77 235960.0 57300.0 4.26 5.6813 0.9981 3221324 PK04_130179 COP(=O)(OC)/N=C\1/CC(=CC(N1Cc2cc3OCOc3cc2Br)c4cccs4)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 I24 compound treatment 174120.0 -4130.0 -0.28 173640.0 -5030.0 -0.37 -0.464 -0.9901 3211811 PK04_130180 CSc1ccc(NC(=O)O[C@H]([C@@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J01 compound treatment 185200.0 6950.0 0.47 179040.0 367.0 0.03 0.3544 0.7466 3176788 PK04_130181 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J02 compound treatment 206840.0 28600.0 1.95 209560.0 30900.0 2.3 3.0038 0.9966 3221326 PK04_130182 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5CCOC5=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J03 compound treatment 197800.0 19600.0 1.33 197640.0 19000.0 1.41 1.9407 0.9996 3176789 PK04_130183 NCCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J04 compound treatment 190680.0 12400.0 0.85 188400.0 9730.0 0.72 1.1112 0.9969 3221328 PK04_130184 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(c3)N(C=O)c4ccccc4)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J05 mock treatment 186240.0 7990.0 0.54 181400.0 2730.0 0.2 0.5287 0.9095 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J06 mock treatment 184520.0 6270.0 0.43 188880.0 10200.0 0.76 0.8395 0.963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J07 compound treatment 285040.0 107000.0 7.28 277440.0 98800.0 7.35 10.3461 1.0 3052827 PK04_130185 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J08 compound treatment 202720.0 24500.0 1.67 205400.0 26700.0 1.99 2.5863 0.9962 3221330 PK04_130186 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccc(cc32)N4CCOC4=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J09 compound treatment 199920.0 21700.0 1.48 206640.0 28000.0 2.08 2.5165 0.9859 3052794 PK04_130187 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J10 compound treatment 191760.0 13500.0 0.92 192480.0 13800.0 1.03 1.3779 0.9985 3221332 PK04_130188 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(CC=C)c3ccc(cc32)N4C(=O)c5cccc6cccc4c56)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J11 compound treatment 194680.0 16400.0 1.12 192640.0 14000.0 1.04 1.5271 0.9993 3176437 PK04_130189 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J12 compound treatment 198960.0 20700.0 1.41 201840.0 23200.0 1.72 2.2176 0.9951 3221334 PK04_130190 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(CC=C)c3ccc(cc32)N4CCOC4=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J13 compound treatment 187680.0 9430.0 0.64 186800.0 8130.0 0.6 0.8823 0.9995 3176038 PK04_130191 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J14 compound treatment 206800.0 28600.0 1.95 205360.0 26700.0 1.99 2.7808 0.9999 3221335 PK04_130192 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(c3)N4CCC4=O)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J15 compound treatment 188120.0 9870.0 0.67 186760.0 8090.0 0.6 0.9014 0.9985 3052796 PK04_130193 Oc1ccc(cc1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@H](Cc4ccccc4)NC3=O)C(=O)NCc5ccc(F)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J16 compound treatment 200240.0 22000.0 1.5 194920.0 16200.0 1.21 1.9152 0.9943 3221337 PK04_130194 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5CCCCC5=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J17 compound treatment 183040.0 4790.0 0.33 185680.0 7010.0 0.52 0.5997 0.9746 3176331 PK04_130195 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J18 compound treatment 183160.0 4910.0 0.33 184440.0 5770.0 0.43 0.5402 0.9924 3221339 PK04_130196 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5CCC5=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J19 compound treatment 200240.0 22000.0 1.5 203640.0 25000.0 1.86 2.3741 0.9943 3176671 PK04_130197 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J20 compound treatment 207920.0 29700.0 2.02 215320.0 36600.0 2.73 3.359 0.9892 3221341 PK04_130198 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(c3)N4C(=O)c5ccccc5Oc6ccccc46)c7ccccc72)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J21 mock treatment 172920.0 -5330.0 -0.36 177600.0 -1070.0 -0.08 -0.3134 -0.8424 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J22 mock treatment 171600.0 -6650.0 -0.45 179280.0 607.0 0.05 -0.2886 -0.6335 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J23 compound treatment 247400.0 69200.0 4.71 263200.0 84500.0 6.29 7.7821 0.9899 3176271 PK04_130199 OCCOc1cccc(c1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 J24 compound treatment 186760.0 8510.0 0.58 175760.0 -2910.0 -0.22 0.257 0.4149 3221343 PK04_130200 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccc(cc32)N4C(=O)c5ccccc5Oc6ccccc46)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K01 compound treatment 209280.0 31000.0 2.12 207200.0 28500.0 2.12 2.9972 1.0 3221345 PK04_130201 COP(=O)(OC)/N=C\1/CC(=CC(N1Cc2cccc(OC(F)(F)F)c2)c3cccs3)c4ccc(CO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K02 compound treatment 213840.0 35600.0 2.43 213800.0 35100.0 2.61 3.5644 0.9993 3211905 PK04_130202 C[C@H](CCO)[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K03 compound treatment 277640.0 99400.0 6.78 285800.0 107000.0 7.97 10.4293 0.9967 3221347 PK04_130203 COc1ccc(CN2CCc3cc(OC)c(O)cc3C2C#Cc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K04 compound treatment 194120.0 15900.0 1.08 194400.0 15700.0 1.17 1.5928 0.9992 3211691 PK04_130204 CSc1ccc(NC(=O)O[C@@H](CCCO)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K05 compound treatment 276440.0 98200.0 6.69 276640.0 98000.0 7.29 9.8894 0.9991 3221348 PK04_130205 COc1cc2CCN(C)C(C#Cc3ccccc3)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K06 compound treatment 194400.0 16200.0 1.1 190720.0 12000.0 0.9 1.4126 0.9948 3211813 PK04_130206 CSc1ccc(NC(=O)O[C@@H]([C@@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K07 mock treatment 189240.0 11000.0 0.75 191840.0 13200.0 0.98 1.2228 0.9912 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K08 mock treatment 188360.0 10100.0 0.69 182720.0 4050.0 0.3 0.7004 0.9311 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K09 compound treatment 296880.0 119000.0 8.09 301320.0 123000.0 9.13 12.1736 0.9982 3221349 PK04_130207 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C#Cc4ccccc4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K10 compound treatment 377000.0 199000.0 13.55 358640.0 180000.0 13.39 19.0527 1.0 3211817 PK04_130208 CSc1ccc(NC(=O)O[C@H](CC=C)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K11 compound treatment 297720.0 119000.0 8.15 296000.0 117000.0 8.73 11.9341 0.9994 3221350 PK04_130209 COCC#CC1N(Cc2ccc(OC)cc2)CCc3cc(OC)c(O)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K12 compound treatment 226800.0 48600.0 3.31 223560.0 44900.0 3.34 4.7028 1.0 3080279 PK04_130210 C[C@@H](CCO)[C@@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K13 compound treatment 230560.0 52300.0 3.57 227760.0 49100.0 3.65 5.1051 0.9999 3221351 PK04_130211 COCC#CC1N(C)CCc2cc(OC)c(O)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K14 compound treatment 195600.0 17400.0 1.18 204080.0 25400.0 1.89 2.1735 0.9745 3080188 PK04_130212 CO[C@H](CCO)[C@H](O)c1ccc(OC)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K15 mock treatment 187520.0 9270.0 0.63 189400.0 10700.0 0.8 1.0114 0.9933 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K16 mock treatment 187320.0 9070.0 0.62 184280.0 5610.0 0.42 0.7323 0.9817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K17 compound treatment 286600.0 108000.0 7.39 280400.0 102000.0 7.57 10.5771 0.9999 3221353 PK04_130213 COCC#CC1N(Cc2ccc(o2)[N+](=O)[O-])CCc3cc(OC)c(O)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K18 compound treatment 184680.0 6430.0 0.44 179240.0 567.0 0.04 0.3398 0.7716 3080221 PK04_130214 CO[C@H](CCO)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K19 compound treatment 281720.0 103000.0 7.05 282880.0 104000.0 7.76 10.4723 0.9989 3221354 PK04_130215 COc1ccc(CN2CCc3cc(OC)c(O)cc3C2C#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K20 compound treatment 197880.0 19600.0 1.34 191120.0 12400.0 0.93 1.6014 0.9839 3211696 PK04_130216 CO[C@@H](CCO)[C@@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K21 compound treatment 308000.0 130000.0 8.85 323360.0 145000.0 10.77 13.8696 0.9952 3221356 PK04_130217 COc1cc2CCN(C)C(C#C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K22 compound treatment 183840.0 5590.0 0.38 187640.0 8970.0 0.67 0.7414 0.9647 3211816 PK04_130218 COc1ccc(NC(=O)O[C@H]([C@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K23 mock treatment 172880.0 -5370.0 -0.37 173120.0 -5550.0 -0.41 -0.5511 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 K24 mock treatment 165400.0 -12800.0 -0.88 166040.0 -12600.0 -0.94 -1.2843 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L01 compound treatment 179320.0 1070.0 0.07 175560.0 -3110.0 -0.23 -0.1122 -0.462 3176382 PK04_130219 CN(C)CCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L02 compound treatment 225640.0 47400.0 3.23 221400.0 42700.0 3.18 4.5332 1.0 3221357 PK04_130220 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(CC=C)c3ccc(cc32)N4CCCCC4=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L03 compound treatment 188920.0 10700.0 0.73 191840.0 13200.0 0.98 1.2073 0.9892 3176383 PK04_130221 NCCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L04 compound treatment 220600.0 42400.0 2.89 221240.0 42600.0 3.17 4.2818 0.9989 3221359 PK04_130222 C[C@H](O)C(=O)Nc1ccc2N(CC=C)C(=O)[C@]3(O[C@H](CCO)[C@H]([C@@H]3C)[Si](C)(C)F)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L05 compound treatment 269520.0 91300.0 6.22 275240.0 96600.0 7.19 9.4821 0.9974 3052642 PK04_130223 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)[C@@H]4CCCN4C3=O)C(=O)OCCOc5ccc(cc5)[C@H]6N7[C@@H]([C@@H](C(=O)OCC=C)[C@]68C(=O)Nc9ccccc98)C(=O)O[C@@H]([C@@H]7c%10ccccc%10)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L06 compound treatment 207360.0 29100.0 1.98 201560.0 22900.0 1.7 2.6078 0.9971 3221361 PK04_130224 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccc(cc32)N4CCC4=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L07 mock treatment 184000.0 5750.0 0.39 180000.0 1330.0 0.1 0.347 0.8584 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L08 mock treatment 185800.0 7550.0 0.51 184240.0 5570.0 0.41 0.657 0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L09 compound treatment 201440.0 23200.0 1.58 202240.0 23600.0 1.75 2.3582 0.9987 3176673 PK04_130225 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L10 compound treatment 212000.0 33800.0 2.3 205200.0 26500.0 1.97 3.0231 0.9971 3221363 PK04_130226 COc1ccc(cc1)C(=O)Nc2cccc(CN3C(=O)[C@]4(O[C@H](CCO)[C@H]([C@@H]4C)[Si](C)(C)F)c5ccccc35)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L11 compound treatment 189960.0 11700.0 0.8 188400.0 9730.0 0.72 1.0764 0.9988 3052529 PK04_130227 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L12 compound treatment 203280.0 25000.0 1.71 201400.0 22700.0 1.69 2.4027 1.0 3221365 PK04_130228 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3cccc(c3)N(C=O)c4ccccc4)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L13 compound treatment 189400.0 11200.0 0.76 188760.0 10100.0 0.75 1.0684 1.0 3052693 PK04_130229 CN(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L14 compound treatment 207960.0 29700.0 2.03 206160.0 27500.0 2.05 2.8789 1.0 3221366 PK04_130230 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccccc3)c4ccc(NC(=O)C)cc42)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L15 mock treatment 179560.0 1310.0 0.09 179720.0 1050.0 0.08 0.1183 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L16 mock treatment 182800.0 4550.0 0.31 179440.0 767.0 0.06 0.2597 0.8234 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L17 compound treatment 196200.0 18000.0 1.22 199760.0 21100.0 1.57 1.9751 0.9924 3176205 PK04_130231 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L18 compound treatment 209080.0 30800.0 2.1 206640.0 28000.0 2.08 2.9581 1.0 3221368 PK04_130232 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(c3)N4CCOC4=O)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L19 compound treatment 192600.0 14400.0 0.98 191400.0 12700.0 0.95 1.3616 0.9999 3176125 PK04_130233 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L20 compound treatment 217840.0 39600.0 2.7 215680.0 37000.0 2.75 3.8562 0.9999 3221370 PK04_130234 COc1ccc(cc1)C(=O)Nc2ccc3N(CC=C)C(=O)[C@@]4(O[C@@H](CCO)[C@@H]([C@H]4C)[Si](C)(C)F)c3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L21 compound treatment 297680.0 119000.0 8.14 295160.0 116000.0 8.67 11.888 0.9995 3052877 PK04_130235 Oc1ccc(cc1)[C@H]2[C@H](C[C@@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L22 compound treatment 215760.0 37500.0 2.56 213880.0 35200.0 2.62 3.6612 0.9999 3221372 PK04_130236 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccc(NC(=O)C)cc32)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L23 mock treatment 166000.0 -12200.0 -0.84 169720.0 -8950.0 -0.67 -1.0617 -0.9937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 L24 mock treatment 172840.0 -5410.0 -0.37 167880.0 -10800.0 -0.8 -0.8288 -0.9376 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M01 compound treatment 302080.0 124000.0 8.44 295320.0 117000.0 8.68 12.1085 0.9999 3221374 PK04_130237 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C#C)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M02 compound treatment 184080.0 5830.0 0.4 185160.0 6490.0 0.48 0.6225 0.9953 3211810 PK04_130238 C[C@@H](CCO)[C@@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M03 compound treatment 193400.0 15200.0 1.03 189240.0 10600.0 0.79 1.2865 0.9909 3221375 PK04_130239 CC(C)C(=C=CC[C@@H](O)c1ccc(OCCO)cc1)C[C@@H](O)c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M04 compound treatment 203080.0 24800.0 1.69 195520.0 16800.0 1.25 2.0836 0.9891 3080224 PK04_130240 COc1ccc(NC(=O)O[C@@H]([C@H](C)CCO)c2ccc(OCCO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M05 compound treatment 199600.0 21400.0 1.46 195000.0 16300.0 1.22 1.8885 0.996 3221376 PK04_130241 COCC(=C=CC[C@@H](O)c1ccc(OCCO)cc1)C[C@@H](O)c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M06 compound treatment 239360.0 61100.0 4.17 234840.0 56200.0 4.18 5.902 1.0 3211820 PK04_130242 COc1ccc(NC(=O)O[C@@H](CCCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M07 compound treatment 196040.0 17800.0 1.21 195320.0 16600.0 1.24 1.7337 0.9999 3221377 PK04_130243 CCCCC(=C=CC[C@@H](O)c1cccc(OCCO)c1)C[C@@H](O)c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M08 compound treatment 204960.0 26700.0 1.82 200520.0 21800.0 1.63 2.4374 0.9984 3211694 PK04_130244 CO[C@H](CCO)[C@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M09 mock treatment 188600.0 10400.0 0.71 188240.0 9570.0 0.71 1.0025 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M10 mock treatment 192240.0 14000.0 0.95 182480.0 3810.0 0.28 0.8748 0.8792 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M11 compound treatment 195360.0 17100.0 1.17 191520.0 12800.0 0.96 1.501 0.9951 3221378 PK04_130245 CC(C)C(=C=CC[C@@H](O)c1cccc(OCCO)c1)C[C@@H](O)c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M12 compound treatment 204160.0 25900.0 1.77 204120.0 25400.0 1.89 2.5883 0.9994 3080189 PK04_130246 CO[C@H](CCO)[C@H](OC(=O)Nc1ccc(SC)cc1)c2ccc(OC)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M13 mock treatment 186720.0 8470.0 0.58 193640.0 15000.0 1.11 1.196 0.9532 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M14 mock treatment 183000.0 4750.0 0.32 187200.0 8530.0 0.63 0.6778 0.9513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M15 compound treatment 194480.0 16200.0 1.11 196560.0 17900.0 1.33 1.7238 0.9958 3221379 PK04_130247 COCC(=C=CC[C@@H](O)c1cccc(OCCO)c1)C[C@@H](O)c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M16 compound treatment 198480.0 20200.0 1.38 197920.0 19200.0 1.43 1.9882 0.9998 3211679 PK04_130248 CO[C@@H](CCO)[C@@H](O)c1ccc(OC)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M17 compound treatment 184920.0 6670.0 0.45 186480.0 7810.0 0.58 0.7324 0.9927 3221380 PK04_130249 CCCCC(=C=CC[C@@H](O)c1ccccc1OCCO)C[C@@H](O)c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M18 compound treatment 188120.0 9870.0 0.67 190520.0 11800.0 0.88 1.0993 0.9911 3211808 PK04_130250 C[C@H](CCO)[C@H](O)c1ccc(OCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M19 mock treatment 185120.0 6870.0 0.47 185200.0 6530.0 0.49 0.6747 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M20 compound treatment 231960.0 53700.0 3.66 228520.0 49800.0 3.71 5.2126 1.0 3080271 PK04_130251 CSc1ccc(NC(=O)O[C@H](CCCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M21 mock treatment 185400.0 7150.0 0.49 183480.0 4810.0 0.36 0.5977 0.9884 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M22 compound treatment 211160.0 32900.0 2.24 211800.0 33100.0 2.47 3.3299 0.9989 3211910 PK04_130252 C[C@@H](CCO)[C@H](O)c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M23 mock treatment 173160.0 -5090.0 -0.35 182200.0 3530.0 0.26 -0.0597 -0.1373 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 M24 compound treatment 215840.0 37600.0 2.56 217760.0 39100.0 2.91 3.8692 0.998 3211692 PK04_130253 COc1ccc(NC(=O)O[C@@H](CC=C)c2ccc(O)c(F)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N01 compound treatment 188760.0 10500.0 0.72 189160.0 10500.0 0.78 1.0586 0.9991 3176433 PK04_130254 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N02 compound treatment 204400.0 26200.0 1.78 208040.0 29400.0 2.19 2.8062 0.9949 3221382 PK04_130255 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5CCCCC5=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N03 compound treatment 230680.0 52400.0 3.57 235720.0 57000.0 4.25 5.5298 0.9963 3175967 PK04_130256 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N04 compound treatment 195320.0 17100.0 1.16 189440.0 10800.0 0.8 1.3896 0.9834 3221383 PK04_130257 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5C(=O)c6ccccc6Oc7ccccc57)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N05 compound treatment 250680.0 72400.0 4.94 242160.0 63500.0 4.73 6.8329 0.9998 3052653 PK04_130258 OCCOc1cccc(c1)[C@@H]2[C@@H](C[C@H]3N2C(=O)CNC3=O)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N06 compound treatment 203000.0 24800.0 1.69 203160.0 24500.0 1.82 2.4819 0.9993 3221385 PK04_130259 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(CC=C)c3ccc(cc32)N4C(=O)c5cccc6cccc4c56)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N07 compound treatment 204120.0 25900.0 1.76 202760.0 24100.0 1.79 2.5148 1.0 3052758 PK04_130260 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N08 compound treatment 213840.0 35600.0 2.43 214080.0 35400.0 2.64 3.5791 0.9992 3221386 PK04_130261 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3ccc(cc3)N4CCCCC4=O)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N09 mock treatment 186840.0 8590.0 0.59 185080.0 6410.0 0.48 0.7513 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N10 mock treatment 189880.0 11600.0 0.79 183320.0 4650.0 0.35 0.8052 0.9308 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N11 compound treatment 193600.0 15400.0 1.05 188920.0 10200.0 0.76 1.2793 0.9879 3176332 PK04_130262 CN(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N12 compound treatment 208640.0 30400.0 2.07 212200.0 33500.0 2.5 3.2295 0.9957 3221388 PK04_130263 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3ccccc3)c4ccc(NC(=O)C)cc42)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N13 mock treatment 186480.0 8230.0 0.56 190960.0 12300.0 0.91 1.0434 0.9725 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N14 mock treatment 185840.0 7590.0 0.52 187000.0 8330.0 0.62 0.8041 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N15 compound treatment 195480.0 17200.0 1.17 196280.0 17600.0 1.31 1.7573 0.9985 3176440 PK04_130264 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCc4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N16 compound treatment 181720.0 3470.0 0.24 179560.0 887.0 0.07 0.214 0.8711 3221389 PK04_130265 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3cccc(c3)N4C(=O)c5cccc6cccc4c56)c7ccccc72)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N17 compound treatment 196600.0 18400.0 1.25 195240.0 16600.0 1.23 1.7565 1.0 3174818 PK04_130266 CN(C)CCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3cccc(OCCO)c3)C(=O)[C@H](CCCCNC(=O)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N18 compound treatment 219360.0 41100.0 2.8 217000.0 38300.0 2.85 3.9989 1.0 3221391 PK04_130267 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5CCOC5=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N19 compound treatment 190200.0 12000.0 0.81 190760.0 12100.0 0.9 1.2122 0.9988 3052539 PK04_130268 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)NCCCCCCN(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N20 compound treatment 202680.0 24400.0 1.67 197520.0 18800.0 1.4 2.1696 0.9963 3221392 PK04_130269 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N(C=O)c5ccccc5)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N21 compound treatment 246680.0 68400.0 4.67 260800.0 82100.0 6.11 7.6211 0.9911 3052582 PK04_130270 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N22 compound treatment 176000.0 -2250.0 -0.15 184200.0 5530.0 0.41 0.1824 0.4155 3221394 PK04_130271 C[C@H](O)C(=O)Nc1ccc(CN2C(=O)[C@@]3(O[C@@H](CCO)[C@@H]([C@H]3C)[Si](C)(C)F)c4ccccc24)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N23 compound treatment 254920.0 76700.0 5.23 240000.0 61300.0 4.56 6.9236 0.9977 3052791 PK04_130272 CC(C)C[C@@H]1NC(=O)[C@@H]2C[C@@H]([C@@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 N24 compound treatment 184680.0 6430.0 0.44 183240.0 4570.0 0.34 0.5503 0.9921 3221396 PK04_130273 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(NC(=O)C)c3)c4ccccc42)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O01 mock treatment 173360.0 -4890.0 -0.33 181400.0 2730.0 0.2 -0.0922 -0.2363 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O02 compound treatment 202120.0 23900.0 1.63 206520.0 27800.0 2.07 2.6163 0.9928 3211913 PK04_130274 CSc1ccc(NC(=O)O[C@H]([C@H](C)CCO)c2ccc(O)c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O03 mock treatment 176840.0 -1410.0 -0.1 180120.0 1450.0 0.11 0.0082 0.0568 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O04 mock treatment 176920.0 -1330.0 -0.09 181760.0 3090.0 0.23 0.0984 0.3982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O05 mock treatment 184080.0 5830.0 0.4 183280.0 4610.0 0.34 0.5235 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O06 mock treatment 176880.0 -1370.0 -0.09 186800.0 8130.0 0.6 0.3617 0.591 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O07 mock treatment 183040.0 4790.0 0.33 183280.0 4610.0 0.34 0.4734 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O08 mock treatment 182200.0 3950.0 0.27 177120.0 -1550.0 -0.12 0.1087 0.3709 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O09 mock treatment 184320.0 6070.0 0.41 175360.0 -3310.0 -0.25 0.1183 0.2455 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O10 mock treatment 177520.0 -730.0 -0.05 179840.0 1170.0 0.09 0.0262 0.2622 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O11 mock treatment 179080.0 830.0 0.06 180920.0 2250.0 0.17 0.1583 0.8965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O12 mock treatment 174920.0 -3330.0 -0.23 180840.0 2170.0 0.16 -0.0465 -0.1669 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O13 mock treatment 181720.0 3470.0 0.24 187560.0 8890.0 0.66 0.635 0.904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O14 mock treatment 178560.0 310.0 0.02 177880.0 -793.0 -0.06 -0.0268 -0.427 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O15 mock treatment 179000.0 750.0 0.05 177880.0 -793.0 -0.06 -0.0056 -0.0712 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O16 mock treatment 178200.0 -49.5 0.0 178600.0 -73.2 -0.01 -0.0062 -0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O17 mock treatment 173040.0 -5210.0 -0.36 176720.0 -1950.0 -0.15 -0.3539 -0.9223 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O18 mock treatment 176760.0 -1490.0 -0.1 179040.0 367.0 0.03 -0.0525 -0.4993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O19 mock treatment 170720.0 -7530.0 -0.51 175120.0 -3550.0 -0.26 -0.55 -0.9524 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O20 mock treatment 171360.0 -6890.0 -0.47 174560.0 -4110.0 -0.31 -0.5486 -0.9785 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O21 mock treatment 175960.0 -2290.0 -0.16 172920.0 -5750.0 -0.43 -0.4132 -0.9065 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O22 mock treatment 166600.0 -11600.0 -0.79 172120.0 -6550.0 -0.49 -0.9065 -0.9726 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O23 mock treatment 168320.0 -9930.0 -0.68 173600.0 -5070.0 -0.38 -0.7457 -0.962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 O24 mock treatment 166680.0 -11600.0 -0.79 171560.0 -7110.0 -0.53 -0.9321 -0.9812 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P01 compound treatment 180800.0 2550.0 0.17 180840.0 2170.0 0.16 0.237 0.9993 3175838 PK04_130275 NCCCCCNC(=O)[C@H]1C[C@@H]2N([C@H]1c3ccc(O)cc3)C(=O)[C@H](CCCCN)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P02 compound treatment 187440.0 9190.0 0.63 187200.0 8530.0 0.63 0.8918 1.0 3221398 PK04_130276 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccc(cc3)N4CCCCC4=O)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P03 compound treatment 160160.0 -18100.0 -1.23 157960.0 -20700.0 -1.54 -1.9622 -0.9939 3052740 PK04_130277 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3cccc(OCCO)c3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P04 compound treatment 180200.0 1950.0 0.13 182000.0 3330.0 0.25 0.2691 0.9575 3221399 PK04_130278 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3cccc(NC(=O)C)c3)c4ccccc42)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P05 compound treatment 181240.0 2990.0 0.2 183880.0 5210.0 0.39 0.4182 0.955 3176784 PK04_130279 C[N+](C)(C)CCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)OCCOc4ccc(cc4)[C@H]5N6[C@@H]([C@@H](C(=O)OCC=C)[C@]57C(=O)Nc8ccccc87)C(=O)O[C@@H]([C@@H]6c9ccccc9)c%10ccccc%10 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P06 compound treatment 185640.0 7390.0 0.5 187800.0 9130.0 0.68 0.8366 0.9892 3221400 PK04_130280 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5C(=O)c6ccccc6Oc7ccccc57)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P07 compound treatment 204600.0 26400.0 1.8 201360.0 22700.0 1.69 2.4643 0.9995 3052752 PK04_130281 CC(=O)NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P08 compound treatment 182640.0 4390.0 0.3 182320.0 3650.0 0.27 0.4036 0.9988 3221401 PK04_130282 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3ccccc3)c4ccc(cc42)N5CCC5=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P09 compound treatment 209480.0 31200.0 2.13 205160.0 26500.0 1.97 2.8995 0.9993 3052788 PK04_130283 CC(C)C[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)NCCCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P10 compound treatment 168800.0 -9450.0 -0.64 173720.0 -4950.0 -0.37 -0.7162 -0.9649 3221402 PK04_130284 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(Cc3cccc(c3)N4CCCCC4=O)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P11 mock treatment 178040.0 -210.0 -0.01 175640.0 -3030.0 -0.23 -0.1697 -0.7504 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P12 mock treatment 179280.0 1030.0 0.07 177400.0 -1270.0 -0.09 -0.0173 -0.1469 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P13 compound treatment 193160.0 14900.0 1.02 191920.0 13200.0 0.99 1.416 0.9999 3052846 PK04_130285 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)CNC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P14 compound treatment 212960.0 34700.0 2.37 211840.0 33200.0 2.47 3.4188 0.9998 3221404 PK04_130286 C[C@H](O)C(=O)Nc1cccc(CN2C(=O)[C@]3(O[C@H](CCO)[C@H]([C@@H]3C)[Si](C)(C)F)c4ccccc24)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P15 compound treatment 208840.0 30600.0 2.09 206240.0 27600.0 2.05 2.9255 1.0 3052836 PK04_130287 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@@H]4CCCN4C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P16 compound treatment 171320.0 -6930.0 -0.47 174480.0 -4190.0 -0.31 -0.5547 -0.9797 3221406 PK04_130288 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(c3)N4CCCCC4=O)c5ccccc52)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P17 compound treatment 196240.0 18000.0 1.23 198120.0 19400.0 1.45 1.8907 0.9966 3176730 PK04_130289 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P18 compound treatment 188080.0 9830.0 0.67 187240.0 8570.0 0.64 0.9248 0.9997 3221407 PK04_130290 C[C@H](O)C(=O)Nc1ccc(CN2C(=O)[C@]3(O[C@H](CCO)[C@H]([C@@H]3C)[Si](C)(C)F)c4ccccc24)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P19 compound treatment 188280.0 10000.0 0.68 190440.0 11800.0 0.88 1.1028 0.9925 3052799 PK04_130291 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P20 compound treatment 192800.0 14600.0 0.99 190120.0 11400.0 0.85 1.3039 0.9971 3221408 PK04_130292 COc1ccc(cc1)C(=O)Nc2ccc(CN3C(=O)[C@]4(O[C@H](CCO)[C@H]([C@@H]4C)[Si](C)(C)F)c5ccccc35)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P21 compound treatment 195400.0 17200.0 1.17 196920.0 18200.0 1.36 1.7871 0.9972 3176730 PK04_130293 C[N+](C)(C)CCCCNC(=O)[C@@H]1C[C@H]2N([C@@H]1c3ccc(O)cc3)C(=O)[C@H](CCCC[N+](C)(C)C)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P22 compound treatment 208720.0 30500.0 2.08 179720.0 1050.0 0.08 1.524 0.7331 3221410 PK04_130294 C[C@@H]1[C@H]([C@H](CCO)O[C@@]12C(=O)N(CC=C)c3ccc(cc32)N4CCC4=O)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P23 compound treatment 175560.0 -2690.0 -0.18 177600.0 -1070.0 -0.08 -0.1861 -0.9307 3176786 PK04_130295 NCCCC[C@@H]1NC(=O)[C@H]2C[C@H]([C@H](N2C1=O)c3ccc(O)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2130 P24 compound treatment 177680.0 -570.0 -0.04 168520.0 -10200.0 -0.76 -0.5618 -0.7425 3221411 PK04_130296 C[C@H]1[C@@H]([C@@H](CCO)O[C@]12C(=O)N(Cc3cccc(c3)N4C(=O)COc5ccccc45)c6ccccc62)[Si](C)(C)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A01 compound treatment 160680.0 -16600.0 -1.13 163000.0 -13400.0 -1.0 -1.5068 -0.998 3237406 Sulf1.1-A_000001 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A02 compound treatment 170960.0 -6340.0 -0.43 174560.0 -1850.0 -0.14 -0.4028 -0.8882 3237380 Sulf1.1-A_000002 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3ccc(Cl)cc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A03 compound treatment 166520.0 -10800.0 -0.73 169480.0 -6930.0 -0.52 -0.8842 -0.985 3237177 Sulf1.1-A_000003 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc(cc3)c4ccccc4)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A04 compound treatment 177720.0 421.0 0.03 179200.0 2790.0 0.21 0.1673 0.7971 3237394 Sulf1.1-A_000004 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A05 compound treatment 180240.0 2940.0 0.2 178000.0 1590.0 0.12 0.2256 0.9686 3237332 Sulf1.1-A_000005 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A06 compound treatment 175160.0 -2140.0 -0.15 174800.0 -1610.0 -0.12 -0.1877 -0.9951 3237396 Sulf1.1-A_000006 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc(Cl)cc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A07 compound treatment 175800.0 -1500.0 -0.1 173160.0 -3250.0 -0.24 -0.2431 -0.9267 3237257 Sulf1.1-A_000007 Cc1ccc(cc1)S(=O)(=O)NC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A08 compound treatment 167800.0 -9500.0 -0.65 170720.0 -5690.0 -0.42 -0.7572 -0.9787 3237153 Sulf1.1-A_000008 OCCOc1ccc(CN2CC[C@@H](C2)N3C(=O)c4ccccc4C3=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A09 compound treatment 184040.0 6740.0 0.46 172840.0 -3570.0 -0.27 0.1372 0.2586 3237428 Sulf1.1-A_000009 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A10 compound treatment 189200.0 11900.0 0.81 185920.0 9510.0 0.71 1.0744 0.9977 3237318 Sulf1.1-A_000010 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3cccc4cccnc34)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A11 compound treatment 168760.0 -8540.0 -0.58 164720.0 -11700.0 -0.87 -1.0267 -0.9809 3237197 Sulf1.1-A_000011 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A12 compound treatment 185400.0 8100.0 0.55 183480.0 7070.0 0.53 0.7628 0.9997 3237446 Sulf1.1-A_000012 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3ccc(Cl)c(Cl)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A13 mock treatment 164320.0 -13000.0 -0.88 169080.0 -7330.0 -0.55 -1.0113 -0.973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A14 mock treatment 164840.0 -12500.0 -0.85 164400.0 -12000.0 -0.89 -1.2325 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A15 compound treatment 167880.0 -9420.0 -0.64 161880.0 -14500.0 -1.08 -1.2186 -0.9691 3237240 Sulf1.1-A_000013 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3cccc(F)c3)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A16 compound treatment 183600.0 6300.0 0.43 181200.0 4790.0 0.36 0.556 0.9957 3237246 Sulf1.1-A_000014 COc1ccc(cc1)S(=O)(=O)NC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A17 compound treatment 172040.0 -5260.0 -0.36 169560.0 -6850.0 -0.51 -0.6139 -0.9852 3237241 Sulf1.1-A_000015 CC(C)S(=O)(=O)NCC1CCN(Cc2ccc(OCCO)cc2)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A18 compound treatment 161600.0 -15700.0 -1.07 164920.0 -11500.0 -0.85 -1.3614 -0.9938 3237449 Sulf1.1-A_000016 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A19 compound treatment 173160.0 -4140.0 -0.28 174880.0 -1530.0 -0.11 -0.2799 -0.92 3237371 Sulf1.1-A_000017 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3cccc4cccnc34)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A20 compound treatment 166640.0 -10700.0 -0.73 164640.0 -11800.0 -0.88 -1.1331 -0.9957 3237416 Sulf1.1-A_000018 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cccc(F)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A21 compound treatment 168440.0 -8860.0 -0.6 165720.0 -10700.0 -0.8 -0.9895 -0.9908 3237365 Sulf1.1-A_000019 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3ccc(Cl)cc3)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A22 compound treatment 165120.0 -12200.0 -0.83 163520.0 -12900.0 -0.96 -1.2653 -0.9974 3237151 Sulf1.1-A_000020 OCCOc1ccc(CN2CC[C@H](C2)N3C(=O)c4ccccc4C3=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A23 compound treatment 167440.0 -9860.0 -0.67 169360.0 -7050.0 -0.52 -0.8462 -0.9925 3237460 Sulf1.1-A_000021 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 A24 compound treatment 170160.0 -7140.0 -0.49 162280.0 -14100.0 -1.05 -1.0876 -0.9387 3237391 Sulf1.1-A_000022 CC(C)S(=O)(=O)NC1CCN(Cc2cccc(OCCO)c2)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B01 compound treatment 180960.0 3660.0 0.25 178760.0 2350.0 0.18 0.3003 0.985 3237454 Sulf1.1-A_000023 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B02 mock treatment 162760.0 -14500.0 -0.99 156480.0 -19900.0 -1.48 -1.7496 -0.9808 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B03 compound treatment 188800.0 11500.0 0.78 187160.0 10800.0 0.8 1.1203 0.9999 3237356 Sulf1.1-A_000024 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cccc(F)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B04 mock treatment 163040.0 -14300.0 -0.97 164720.0 -11700.0 -0.87 -1.3025 -0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B05 compound treatment 167600.0 -9700.0 -0.66 163560.0 -12800.0 -0.96 -1.1437 -0.9838 3237374 Sulf1.1-A_000025 Cc1nc(cn1C)S(=O)(=O)NCC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B06 mock treatment 166040.0 -11300.0 -0.77 165440.0 -11000.0 -0.82 -1.1199 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B07 compound treatment 173080.0 -4220.0 -0.29 170320.0 -6090.0 -0.45 -0.5237 -0.976 3237437 Sulf1.1-A_000026 Cc1ccc(cc1)S(=O)(=O)N[C@@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B08 mock treatment 164120.0 -13200.0 -0.9 162520.0 -13900.0 -1.03 -1.3662 -0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B09 compound treatment 161920.0 -15400.0 -1.05 160480.0 -15900.0 -1.19 -1.5796 -0.9981 3237320 Sulf1.1-A_000027 Cc1ccccc1S(=O)(=O)NC[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B10 mock treatment 170040.0 -7260.0 -0.49 166560.0 -9850.0 -0.73 -0.8682 -0.9817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B11 compound treatment 218720.0 41400.0 2.82 209360.0 33000.0 2.45 3.7311 0.9975 3237427 Sulf1.1-A_000028 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B12 mock treatment 164480.0 -12800.0 -0.87 166440.0 -9970.0 -0.74 -1.1425 -0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B13 mock treatment 165080.0 -12200.0 -0.83 167280.0 -9130.0 -0.68 -1.0694 -0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B14 mock treatment 168680.0 -8620.0 -0.59 166280.0 -10100.0 -0.75 -0.9485 -0.9924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B15 compound treatment 166800.0 -10500.0 -0.72 163760.0 -12600.0 -0.94 -1.1717 -0.9909 3237372 Sulf1.1-A_000029 Cc1ccccc1S(=O)(=O)NCC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B16 mock treatment 168120.0 -9180.0 -0.63 162720.0 -13700.0 -1.02 -1.1628 -0.9726 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B17 compound treatment 173400.0 -3900.0 -0.27 170200.0 -6210.0 -0.46 -0.5146 -0.9656 3237289 Sulf1.1-A_000030 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B18 mock treatment 166320.0 -11000.0 -0.75 165080.0 -11300.0 -0.84 -1.1254 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B19 compound treatment 167360.0 -9940.0 -0.68 165000.0 -11400.0 -0.85 -1.0795 -0.9938 3237235 Sulf1.1-A_000031 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3ccc(Cl)c(Cl)c3)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B20 mock treatment 164560.0 -12700.0 -0.87 167920.0 -8490.0 -0.63 -1.0608 -0.9878 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B21 compound treatment 168160.0 -9140.0 -0.62 170400.0 -6010.0 -0.45 -0.7567 -0.9867 3237435 Sulf1.1-A_000032 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3cccc(F)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B22 mock treatment 162400.0 -14900.0 -1.02 163280.0 -13100.0 -0.98 -1.4091 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B23 compound treatment 170280.0 -7020.0 -0.48 162680.0 -13700.0 -1.02 -1.0608 -0.9403 3237254 Sulf1.1-A_000033 Cc1nc(cn1C)S(=O)(=O)NC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 B24 mock treatment 165400.0 -11900.0 -0.81 155840.0 -20600.0 -1.53 -1.656 -0.9559 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C01 compound treatment 175160.0 -2140.0 -0.15 174880.0 -1530.0 -0.11 -0.1835 -0.9924 3237301 Sulf1.1-A_000034 CC(C)S(=O)(=O)N[C@@H]1CCN(Cc2ccc(OCCO)cc2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C02 compound treatment 183280.0 5980.0 0.41 180240.0 3830.0 0.29 0.4901 0.9847 3237158 Sulf1.1-A_000035 OCCOc1ccc(CN2CCC[C@@H](CN3C(=O)c4ccccc4C3=O)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C03 compound treatment 179080.0 1780.0 0.12 178560.0 2150.0 0.16 0.1992 0.9906 3237256 Sulf1.1-A_000036 CC(C)S(=O)(=O)NC1CCN(Cc2ccc(OCCO)cc2)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C04 compound treatment 188000.0 10700.0 0.73 183440.0 7030.0 0.52 0.886 0.9867 3237156 Sulf1.1-A_000037 OCCOc1ccc(CN2CCC[C@H](C2)N3C(=O)c4ccccc4C3=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C05 compound treatment 180840.0 3540.0 0.24 179600.0 3190.0 0.24 0.3387 1.0 3237312 Sulf1.1-A_000038 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc(cc3)c4ccccc4)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C06 compound treatment 189880.0 12600.0 0.86 181960.0 5550.0 0.41 0.8987 0.944 3237455 Sulf1.1-A_000039 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3ccccc3[N+](=O)[O-])c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C07 compound treatment 176200.0 -1100.0 -0.07 174880.0 -1530.0 -0.11 -0.1333 -0.9796 3237443 Sulf1.1-A_000040 Cc1ccc(F)cc1S(=O)(=O)N2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C08 compound treatment 182600.0 5300.0 0.36 181440.0 5030.0 0.37 0.5204 0.9998 3237464 Sulf1.1-A_000041 Cc1ccccc1S(=O)(=O)N2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C09 compound treatment 196160.0 18900.0 1.29 193400.0 17000.0 1.26 1.8036 1.0 3237452 Sulf1.1-A_000042 CC(C)S(=O)(=O)N1CCN(Cc2ccc(OCCO)cc2)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C10 compound treatment 181200.0 3900.0 0.27 182560.0 6150.0 0.46 0.5119 0.9666 3237191 Sulf1.1-A_000043 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3cccc(F)c3)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C11 mock treatment 166960.0 -10300.0 -0.7 171240.0 -5170.0 -0.38 -0.7704 -0.9594 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C12 mock treatment 171000.0 -6300.0 -0.43 174080.0 -2330.0 -0.17 -0.4261 -0.9202 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C13 compound treatment 179560.0 2260.0 0.15 174720.0 -1690.0 -0.13 0.0202 0.1017 3237189 Sulf1.1-A_000044 Cc1nc(cn1C)S(=O)(=O)NC[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C14 compound treatment 169560.0 -7740.0 -0.53 178640.0 2230.0 0.17 -0.2556 -0.462 3237360 Sulf1.1-A_000045 Cc1ccc(cc1)S(=O)(=O)N[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C15 mock treatment 163920.0 -13400.0 -0.91 170360.0 -6050.0 -0.45 -0.9632 -0.947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C16 mock treatment 166880.0 -10400.0 -0.71 172520.0 -3890.0 -0.29 -0.7068 -0.9216 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C17 compound treatment 180240.0 2940.0 0.2 180800.0 4390.0 0.33 0.373 0.9724 3237358 Sulf1.1-A_000046 CC(C)S(=O)(=O)N[C@@H]1CCCN(Cc2cccc(OCCO)c2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C18 compound treatment 165480.0 -11800.0 -0.81 167800.0 -8610.0 -0.64 -1.0227 -0.9935 3237390 Sulf1.1-A_000047 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3cccc(F)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C19 compound treatment 169840.0 -7460.0 -0.51 175880.0 -527.0 -0.04 -0.3873 -0.7594 3237243 Sulf1.1-A_000048 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C20 compound treatment 171080.0 -6220.0 -0.42 168040.0 -8370.0 -0.62 -0.7401 -0.9825 3237467 Sulf1.1-A_000049 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3cccc(F)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C21 compound treatment 170760.0 -6540.0 -0.45 173760.0 -2650.0 -0.2 -0.4545 -0.9326 3237185 Sulf1.1-A_000050 Cc1ccccc1S(=O)(=O)NC[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C22 compound treatment 176040.0 -1260.0 -0.09 170000.0 -6410.0 -0.48 -0.3979 -0.8212 3237163 Sulf1.1-A_000051 OCCOc1cccc(CN2CCC(CC2)N3C(=O)c4ccccc4C3=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C23 compound treatment 163200.0 -14100.0 -0.96 160600.0 -15800.0 -1.18 -1.5116 -0.995 3237285 Sulf1.1-A_000052 Cc1ccc(cc1)S(=O)(=O)N[C@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 C24 compound treatment 171880.0 -5420.0 -0.37 162480.0 -13900.0 -1.04 -0.9942 -0.9035 3237265 Sulf1.1-A_000053 Cc1ccc(F)cc1S(=O)(=O)N[C@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D01 compound treatment 177360.0 60.8 0.0 179120.0 2710.0 0.2 0.1457 0.7215 3237408 Sulf1.1-A_000054 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cccc4cccnc34)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D02 mock treatment 171200.0 -6100.0 -0.42 166440.0 -9970.0 -0.74 -0.8186 -0.9626 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D03 compound treatment 181920.0 4620.0 0.32 179640.0 3230.0 0.24 0.3929 0.9912 3237375 Sulf1.1-A_000055 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3cccc(F)c3)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D04 mock treatment 175160.0 -2140.0 -0.15 171840.0 -4570.0 -0.34 -0.3435 -0.9286 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D05 compound treatment 203080.0 25800.0 1.76 200920.0 24500.0 1.82 2.5329 0.9998 3237458 Sulf1.1-A_000056 COc1ccc(cc1)S(=O)(=O)N2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D06 mock treatment 170760.0 -6540.0 -0.45 173400.0 -3010.0 -0.22 -0.4735 -0.9492 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D07 compound treatment 192280.0 15000.0 1.02 190280.0 13900.0 1.03 1.4523 1.0 3237247 Sulf1.1-A_000057 Cc1ccc(F)cc1S(=O)(=O)NC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D08 mock treatment 169040.0 -8260.0 -0.56 168960.0 -7450.0 -0.55 -0.7901 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D09 compound treatment 175240.0 -2060.0 -0.14 169840.0 -6570.0 -0.49 -0.4449 -0.8748 3237279 Sulf1.1-A_000058 Cc1nc(cn1C)S(=O)(=O)N[C@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D10 mock treatment 172120.0 -5180.0 -0.35 171480.0 -4930.0 -0.37 -0.509 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D11 mock treatment 174120.0 -3180.0 -0.22 171360.0 -5050.0 -0.38 -0.4189 -0.9659 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D12 mock treatment 173920.0 -3380.0 -0.23 166720.0 -9690.0 -0.72 -0.6727 -0.8888 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D13 compound treatment 188360.0 11100.0 0.75 187440.0 11000.0 0.82 1.1139 0.9991 3237383 Sulf1.1-A_000059 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D14 mock treatment 170000.0 -7300.0 -0.5 167920.0 -8490.0 -0.63 -0.7985 -0.993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D15 mock treatment 169040.0 -8260.0 -0.56 171080.0 -5330.0 -0.4 -0.6785 -0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D16 mock treatment 175400.0 -1900.0 -0.13 171520.0 -4890.0 -0.36 -0.3487 -0.9033 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D17 compound treatment 185320.0 8020.0 0.55 176680.0 273.0 0.02 0.401 0.7329 3237175 Sulf1.1-A_000060 Cc1ccc(F)cc1S(=O)(=O)NC[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D18 mock treatment 167160.0 -10100.0 -0.69 170120.0 -6290.0 -0.47 -0.8197 -0.9819 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D19 compound treatment 180880.0 3580.0 0.24 187280.0 10900.0 0.81 0.7449 0.8812 3237205 Sulf1.1-A_000061 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D20 mock treatment 171920.0 -5380.0 -0.37 175960.0 -447.0 -0.03 -0.2828 -0.7681 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D21 compound treatment 175440.0 -1860.0 -0.13 180720.0 4310.0 0.32 0.1374 0.398 3237238 Sulf1.1-A_000062 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3ccc4ccccc4c3)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D22 mock treatment 167400.0 -9900.0 -0.67 167640.0 -8770.0 -0.65 -0.9386 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D23 compound treatment 184080.0 6780.0 0.46 188440.0 12000.0 0.9 0.9602 0.9527 3237342 Sulf1.1-A_000063 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 D24 mock treatment 160120.0 -17200.0 -1.17 165520.0 -10900.0 -0.81 -1.4011 -0.9838 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E01 mock treatment 180520.0 3220.0 0.22 176560.0 153.0 0.01 0.1633 0.7428 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E02 mock treatment 173920.0 -3380.0 -0.23 171400.0 -5010.0 -0.37 -0.4264 -0.9733 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E03 compound treatment 183200.0 5900.0 0.4 178800.0 2390.0 0.18 0.4104 0.9328 3237456 Sulf1.1-A_000064 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E04 compound treatment 197000.0 19700.0 1.34 196000.0 19600.0 1.46 1.9809 0.9992 3237281 Sulf1.1-A_000065 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cccc(F)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E05 compound treatment 229240.0 51900.0 3.54 230040.0 53600.0 3.99 5.3266 0.9982 3237430 Sulf1.1-A_000066 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E06 compound treatment 186400.0 9100.0 0.62 193160.0 16800.0 1.25 1.3204 0.9481 3237248 Sulf1.1-A_000067 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E07 compound treatment 184200.0 6900.0 0.47 181560.0 5150.0 0.38 0.6039 0.9949 3237392 Sulf1.1-A_000068 Cc1ccc(cc1)S(=O)(=O)NC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E08 compound treatment 185320.0 8020.0 0.55 185120.0 8710.0 0.65 0.8452 0.9964 3237369 Sulf1.1-A_000069 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3cc(Cl)ccc3Cl)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E09 mock treatment 177960.0 661.0 0.05 178320.0 1910.0 0.14 0.1325 0.8875 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E10 mock treatment 176720.0 -579.0 -0.04 178440.0 2030.0 0.15 0.0791 0.5056 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E11 compound treatment 186840.0 9540.0 0.65 189480.0 13100.0 0.97 1.148 0.9808 3237294 Sulf1.1-A_000070 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3cc(Cl)ccc3Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E12 compound treatment 201400.0 24100.0 1.64 201360.0 25000.0 1.86 2.4751 0.9981 3237436 Sulf1.1-A_000071 CC(C)S(=O)(=O)N[C@@H]1CCN(Cc2cccc(OCCO)c2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E13 compound treatment 210520.0 33200.0 2.26 207280.0 30900.0 2.3 3.2263 1.0 3237379 Sulf1.1-A_000072 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E14 compound treatment 190920.0 13600.0 0.93 184560.0 8150.0 0.61 1.0857 0.9787 3237253 Sulf1.1-A_000073 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3ccc4ccccc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E15 compound treatment 146600.0 -30700.0 -2.09 149080.0 -27300.0 -2.03 -2.9181 -0.9999 3237322 Sulf1.1-A_000074 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc4ccccc4c3)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E16 compound treatment 191000.0 13700.0 0.93 187160.0 10800.0 0.8 1.2264 0.997 3237219 Sulf1.1-A_000075 Cc1nc(cn1C)S(=O)(=O)N[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E17 mock treatment 183920.0 6620.0 0.45 177960.0 1550.0 0.12 0.4009 0.8604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E18 mock treatment 174800.0 -2500.0 -0.17 171720.0 -4690.0 -0.35 -0.3671 -0.9457 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E19 compound treatment 187360.0 10100.0 0.69 190120.0 13700.0 1.02 1.2067 0.9813 3237298 Sulf1.1-A_000076 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc4ccccc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E20 compound treatment 209120.0 31800.0 2.17 208280.0 31900.0 2.37 3.2114 0.999 3237439 Sulf1.1-A_000077 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3ccccc3[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E21 compound treatment 179240.0 1940.0 0.13 186560.0 10200.0 0.76 0.6279 0.8185 3237225 Sulf1.1-A_000078 Cc1ccc(cc1)S(=O)(=O)N[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E22 compound treatment 196720.0 19400.0 1.32 192120.0 15700.0 1.17 1.7632 0.9981 3237306 Sulf1.1-A_000079 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc(Cl)cc3)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E23 compound treatment 178920.0 1620.0 0.11 181000.0 4590.0 0.34 0.3199 0.8903 3237420 Sulf1.1-A_000080 Cc1ccc(cc1)S(=O)(=O)N[C@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 E24 compound treatment 174920.0 -2380.0 -0.16 176760.0 353.0 0.03 -0.0961 -0.5849 3237469 Sulf1.1-A_000081 Cc1ccc(cc1)S(=O)(=O)N2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F01 mock treatment 171480.0 -5820.0 -0.4 176400.0 -6.79 0.0 -0.2809 -0.708 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F02 mock treatment 170400.0 -6900.0 -0.47 177320.0 913.0 0.07 -0.2845 -0.5987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F03 compound treatment 202800.0 25500.0 1.74 190840.0 14400.0 1.07 1.9889 0.9732 3237364 Sulf1.1-A_000082 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3ccccc3)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F04 mock treatment 183280.0 5980.0 0.41 173320.0 -3090.0 -0.23 0.1259 0.2689 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F05 compound treatment 213960.0 36700.0 2.5 223640.0 47200.0 3.52 4.2531 0.986 3237352 Sulf1.1-A_000083 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc4ccccc4c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F06 mock treatment 177880.0 581.0 0.04 177520.0 1110.0 0.08 0.0866 0.9429 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F07 compound treatment 186200.0 8900.0 0.61 185160.0 8750.0 0.65 0.8898 0.9994 3237271 Sulf1.1-A_000084 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F08 mock treatment 180400.0 3100.0 0.21 182040.0 5630.0 0.42 0.4459 0.9497 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F09 mock treatment 180960.0 3660.0 0.25 174520.0 -1890.0 -0.14 0.0772 0.2695 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F10 mock treatment 185240.0 7940.0 0.54 177040.0 633.0 0.05 0.4161 0.7658 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F11 compound treatment 249680.0 72400.0 4.93 246160.0 69800.0 5.19 7.1603 0.9997 3237444 Sulf1.1-A_000085 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F12 mock treatment 178560.0 1260.0 0.09 178320.0 1910.0 0.14 0.1615 0.9708 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F13 compound treatment 174080.0 -3220.0 -0.22 168440.0 -7970.0 -0.59 -0.5745 -0.9086 3237438 Sulf1.1-A_000086 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F14 mock treatment 177800.0 501.0 0.03 177600.0 1190.0 0.09 0.0869 0.9137 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F15 compound treatment 169120.0 -8180.0 -0.56 163760.0 -12600.0 -0.94 -1.0599 -0.9688 3237422 Sulf1.1-A_000087 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F16 mock treatment 180560.0 3260.0 0.22 175520.0 -887.0 -0.07 0.1105 0.4766 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F17 mock treatment 178040.0 741.0 0.05 177640.0 1230.0 0.09 0.1006 0.9604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F18 mock treatment 179360.0 2060.0 0.14 180920.0 4510.0 0.34 0.3369 0.9252 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F19 compound treatment 179000.0 1700.0 0.12 173600.0 -2810.0 -0.21 -0.0657 -0.2751 3237453 Sulf1.1-A_000088 Cc1ccc(cc1)S(=O)(=O)N2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F20 mock treatment 181200.0 3900.0 0.27 176160.0 -247.0 -0.02 0.1751 0.6567 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F21 compound treatment 181720.0 4420.0 0.3 182400.0 5990.0 0.45 0.5285 0.9818 3237203 Sulf1.1-A_000089 COc1ccc(cc1)S(=O)(=O)N[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F22 mock treatment 167760.0 -9540.0 -0.65 171520.0 -4890.0 -0.36 -0.7171 -0.9623 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F23 compound treatment 178680.0 1380.0 0.09 180160.0 3750.0 0.28 0.2641 0.8959 3237326 Sulf1.1-A_000090 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3cccc(F)c3)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 F24 mock treatment 168720.0 -8580.0 -0.58 171560.0 -4850.0 -0.36 -0.6687 -0.973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G01 compound treatment 211280.0 34000.0 2.32 202920.0 26500.0 1.97 3.0335 0.9968 3237230 Sulf1.1-A_000091 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3ccc(Cl)cc3)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G02 compound treatment 179880.0 2580.0 0.18 181280.0 4870.0 0.36 0.3809 0.9448 3237376 Sulf1.1-A_000092 CC(C)S(=O)(=O)NCC1CCN(Cc2cccc(OCCO)c2)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G03 mock treatment 176440.0 -859.0 -0.06 177480.0 1070.0 0.08 0.0151 0.152 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G04 mock treatment 179560.0 2260.0 0.15 178680.0 2270.0 0.17 0.2286 0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G05 compound treatment 194920.0 17600.0 1.2 188040.0 11600.0 0.87 1.4617 0.9871 3237466 Sulf1.1-A_000093 Cc1nc(cn1C)S(=O)(=O)N2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G06 compound treatment 205080.0 27800.0 1.89 203320.0 26900.0 2.0 2.7556 0.9996 3237165 Sulf1.1-A_000094 OCCOc1cccc(CN2CCC[C@H](C2)N3C(=O)c4ccccc4C3=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G07 compound treatment 208800.0 31500.0 2.15 206920.0 30500.0 2.27 3.1244 0.9996 3237290 Sulf1.1-A_000095 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc(Cl)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G08 compound treatment 214000.0 36700.0 2.5 201720.0 25300.0 1.88 3.1015 0.9902 3237199 Sulf1.1-A_000096 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G09 compound treatment 226440.0 49100.0 3.35 219920.0 43500.0 3.24 4.659 0.9999 3237213 Sulf1.1-A_000097 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cccc4cccnc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G10 compound treatment 153560.0 -23700.0 -1.62 151440.0 -25000.0 -1.86 -2.4584 -0.9976 3237354 Sulf1.1-A_000098 Cc1nc(cn1C)S(=O)(=O)N[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G11 compound treatment 178360.0 1060.0 0.07 168880.0 -7530.0 -0.56 -0.345 -0.6108 3237348 Sulf1.1-A_000099 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cccc4cccnc34)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G12 compound treatment 211440.0 34100.0 2.33 206520.0 30100.0 2.24 3.2307 0.9998 3237154 Sulf1.1-A_000100 OCCOc1ccc(CN2CCC(CC2)N3C(=O)c4ccccc4C3=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G13 compound treatment 220560.0 43300.0 2.95 216960.0 40600.0 3.02 4.2198 0.9999 3237231 Sulf1.1-A_000101 COc1ccc(cc1)S(=O)(=O)NCC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G14 compound treatment 181920.0 4620.0 0.32 183800.0 7390.0 0.55 0.6118 0.965 3237160 Sulf1.1-A_000102 OCCOc1cccc(CN2CC[C@H](C2)N3C(=O)c4ccccc4C3=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G15 compound treatment 186320.0 9020.0 0.62 188080.0 11700.0 0.87 1.0492 0.9857 3237336 Sulf1.1-A_000103 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc(Cl)cc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G16 compound treatment 191600.0 14300.0 0.97 183760.0 7350.0 0.55 1.0764 0.9627 3237258 Sulf1.1-A_000104 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G17 compound treatment 195960.0 18700.0 1.27 198600.0 22200.0 1.65 2.0676 0.9917 3237440 Sulf1.1-A_000105 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G18 compound treatment 211280.0 34000.0 2.32 201600.0 25200.0 1.88 2.964 0.9945 3237173 Sulf1.1-A_000106 COc1ccc(cc1)S(=O)(=O)NC[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G19 mock treatment 179800.0 2500.0 0.17 182360.0 5950.0 0.44 0.4339 0.9139 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G20 mock treatment 182040.0 4740.0 0.32 178360.0 1950.0 0.15 0.3313 0.9349 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G21 compound treatment 181920.0 4620.0 0.32 177040.0 633.0 0.05 0.2561 0.8039 3237368 Sulf1.1-A_000107 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3ccc(cc3)c4ccccc4)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G22 compound treatment 196720.0 19400.0 1.32 201600.0 25200.0 1.88 2.2621 0.9855 3237402 Sulf1.1-A_000108 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G23 compound treatment 170400.0 -6900.0 -0.47 172560.0 -3850.0 -0.29 -0.535 -0.9717 3237211 Sulf1.1-A_000109 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 G24 compound treatment 190520.0 13200.0 0.9 187840.0 11400.0 0.85 1.2391 0.9996 3237251 Sulf1.1-A_000110 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3cccc4cccnc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H01 compound treatment 194280.0 17000.0 1.16 188040.0 11600.0 0.87 1.4308 0.9898 3237316 Sulf1.1-A_000111 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc(Cl)c(Cl)c3)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H02 mock treatment 175600.0 -1700.0 -0.12 173120.0 -3290.0 -0.24 -0.2549 -0.9417 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H03 mock treatment 182120.0 4820.0 0.33 180680.0 4270.0 0.32 0.4573 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H04 mock treatment 180960.0 3660.0 0.25 179400.0 2990.0 0.22 0.334 0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H05 compound treatment 170560.0 -6740.0 -0.46 162840.0 -13600.0 -1.01 -1.0389 -0.9365 3237215 Sulf1.1-A_000112 Cc1ccccc1S(=O)(=O)N[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H06 mock treatment 178800.0 1500.0 0.1 179200.0 2790.0 0.21 0.2193 0.9467 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H07 compound treatment 207120.0 29800.0 2.03 204360.0 28000.0 2.08 2.9087 0.9999 3237447 Sulf1.1-A_000113 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3cccc4cccnc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H08 mock treatment 185640.0 8340.0 0.57 182400.0 5990.0 0.45 0.7175 0.9928 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H09 compound treatment 161560.0 -15700.0 -1.07 155560.0 -20800.0 -1.55 -1.8559 -0.9838 3237209 Sulf1.1-A_000114 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cc(Cl)ccc3Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H10 mock treatment 181160.0 3860.0 0.26 184080.0 7670.0 0.57 0.5899 0.9382 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H11 compound treatment 219800.0 42500.0 2.9 209160.0 32800.0 2.44 3.7726 0.9963 3237245 Sulf1.1-A_000115 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3ccc(Cl)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H12 mock treatment 186360.0 9060.0 0.62 177120.0 713.0 0.05 0.4743 0.765 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H13 compound treatment 215040.0 37700.0 2.57 204800.0 28400.0 2.11 3.3137 0.9952 3237367 Sulf1.1-A_000116 Cc1ccc(F)cc1S(=O)(=O)NCC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H14 mock treatment 183440.0 6140.0 0.42 188920.0 12500.0 0.93 0.9546 0.9349 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H15 compound treatment 205800.0 28500.0 1.94 207840.0 31400.0 2.34 3.0282 0.9957 3237250 Sulf1.1-A_000117 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H16 mock treatment 185680.0 8380.0 0.57 178120.0 1710.0 0.13 0.4942 0.8441 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H17 compound treatment 192440.0 15100.0 1.03 185120.0 8710.0 0.65 1.1885 0.9749 3237195 Sulf1.1-A_000118 Cc1ccc(cc1)S(=O)(=O)NC[C@@H]2CCCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H18 mock treatment 183200.0 5900.0 0.4 182160.0 5750.0 0.43 0.5872 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H19 mock treatment 185880.0 8580.0 0.59 176680.0 273.0 0.02 0.428 0.7312 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H20 mock treatment 174840.0 -2460.0 -0.17 177480.0 1070.0 0.08 -0.0621 -0.3342 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H21 compound treatment 193280.0 16000.0 1.09 186680.0 10300.0 0.76 1.3111 0.985 3237330 Sulf1.1-A_000119 Cc1ccc(cc1)S(=O)(=O)NC[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H22 mock treatment 180240.0 2940.0 0.2 174560.0 -1850.0 -0.14 0.0446 0.1834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H23 compound treatment 158880.0 -18400.0 -1.26 160960.0 -15400.0 -1.15 -1.7009 -0.999 3237275 Sulf1.1-A_000120 Cc1ccccc1S(=O)(=O)N[C@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 H24 mock treatment 169280.0 -8020.0 -0.55 165240.0 -11200.0 -0.83 -0.9743 -0.9794 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I01 compound treatment 195040.0 17700.0 1.21 189680.0 13300.0 0.99 1.5538 0.995 3237314 Sulf1.1-A_000121 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3cc(Cl)ccc3Cl)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I02 compound treatment 191560.0 14300.0 0.97 193400.0 17000.0 1.26 1.5818 0.9916 3237346 Sulf1.1-A_000122 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I03 compound treatment 197960.0 20700.0 1.41 193280.0 16900.0 1.26 1.884 0.9984 3237404 Sulf1.1-A_000123 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cc(Cl)ccc3Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I04 compound treatment 196520.0 19200.0 1.31 198360.0 22000.0 1.63 2.0819 0.994 3237340 Sulf1.1-A_000124 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I05 mock treatment 179520.0 2220.0 0.15 181720.0 5310.0 0.4 0.3867 0.9132 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I06 mock treatment 182000.0 4700.0 0.32 181160.0 4750.0 0.35 0.4768 0.9988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I07 compound treatment 197880.0 20600.0 1.4 196280.0 19900.0 1.48 2.038 0.9997 3237334 Sulf1.1-A_000125 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I08 compound treatment 200880.0 23600.0 1.61 195160.0 18800.0 1.4 2.1237 0.9975 3237162 Sulf1.1-A_000126 OCCOc1cccc(CN2CC[C@@H](C2)N3C(=O)c4ccccc4C3=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I09 compound treatment 229960.0 52700.0 3.59 225960.0 49600.0 3.69 5.1466 0.9999 3237468 Sulf1.1-A_000127 CC(C)S(=O)(=O)N1CCN(Cc2cccc(OCCO)c2)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I10 compound treatment 196000.0 18700.0 1.27 187680.0 11300.0 0.84 1.4948 0.9794 3237295 Sulf1.1-A_000128 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I11 compound treatment 186400.0 9100.0 0.62 191920.0 15500.0 1.15 1.2552 0.9576 3237424 Sulf1.1-A_000129 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I12 compound treatment 221920.0 44600.0 3.04 219160.0 42800.0 3.18 4.4011 0.9997 3237287 Sulf1.1-A_000130 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I13 compound treatment 232480.0 55200.0 3.76 219000.0 42600.0 3.17 4.9018 0.9964 3237269 Sulf1.1-A_000131 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cc(Cl)ccc3Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I14 compound treatment 188080.0 10800.0 0.73 193080.0 16700.0 1.24 1.3972 0.9687 3237155 Sulf1.1-A_000132 OCCOc1ccc(CN2CCC(CN3C(=O)c4ccccc4C3=O)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I15 compound treatment 201240.0 23900.0 1.63 200400.0 24000.0 1.79 2.4169 0.999 3237463 Sulf1.1-A_000133 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3cccc4cccnc34)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I16 compound treatment 196960.0 19700.0 1.34 195360.0 19000.0 1.41 1.9453 0.9997 3237410 Sulf1.1-A_000134 Cc1ccccc1S(=O)(=O)N[C@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I17 compound treatment 206760.0 29500.0 2.01 200480.0 24100.0 1.79 2.6872 0.9984 3237385 Sulf1.1-A_000135 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3ccc(Cl)c(Cl)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I18 compound treatment 192960.0 15700.0 1.07 193320.0 16900.0 1.26 1.6451 0.9966 3237167 Sulf1.1-A_000136 OCCOc1cccc(CN2CCC[C@@H](CN3C(=O)c4ccccc4C3=O)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I19 compound treatment 200600.0 23300.0 1.59 197000.0 20600.0 1.53 2.2071 0.9998 3237450 Sulf1.1-A_000137 Cc1nc(cn1C)S(=O)(=O)N2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I20 compound treatment 192120.0 14800.0 1.01 194560.0 18200.0 1.35 1.6698 0.9898 3237221 Sulf1.1-A_000138 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cccc(F)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I21 mock treatment 175640.0 -1660.0 -0.11 176520.0 113.0 0.01 -0.074 -0.6526 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I22 mock treatment 171440.0 -5860.0 -0.4 175240.0 -1170.0 -0.09 -0.3439 -0.8412 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I23 compound treatment 184600.0 7300.0 0.5 185240.0 8830.0 0.66 0.8168 0.9906 3237187 Sulf1.1-A_000139 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc4ccccc4c3)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 I24 compound treatment 168800.0 -8500.0 -0.58 167200.0 -9210.0 -0.69 -0.8943 -0.9965 3237393 Sulf1.1-A_000140 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J01 compound treatment 190240.0 12900.0 0.88 190320.0 13900.0 1.04 1.3561 0.9968 3237433 Sulf1.1-A_000141 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc4ccccc4c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J02 mock treatment 177120.0 -179.0 -0.01 176000.0 -407.0 -0.03 -0.03 -0.9204 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J03 compound treatment 217600.0 40300.0 2.75 204200.0 27800.0 2.07 3.4055 0.9902 3237382 Sulf1.1-A_000142 Cc1ccc(F)cc1S(=O)(=O)NC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J04 mock treatment 184320.0 7020.0 0.48 181240.0 4830.0 0.36 0.5928 0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J05 mock treatment 180520.0 3220.0 0.22 179520.0 3110.0 0.23 0.3191 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J06 mock treatment 177880.0 581.0 0.04 186800.0 10400.0 0.77 0.575 0.7423 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J07 compound treatment 210240.0 32900.0 2.25 211040.0 34600.0 2.58 3.4107 0.9976 3237388 Sulf1.1-A_000143 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3ccc4ccccc4c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J08 mock treatment 185840.0 8540.0 0.58 182280.0 5870.0 0.44 0.7208 0.99 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J09 compound treatment 201560.0 24300.0 1.65 198760.0 22400.0 1.66 2.346 1.0 3237381 Sulf1.1-A_000144 COc1ccc(cc1)S(=O)(=O)NC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J10 mock treatment 187520.0 10200.0 0.7 183720.0 7310.0 0.54 0.8776 0.9925 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J11 compound treatment 219640.0 42300.0 2.89 211160.0 34800.0 2.59 3.8702 0.9985 3237373 Sulf1.1-A_000145 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3ccc4ccccc4c3)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J12 mock treatment 187200.0 9900.0 0.68 190480.0 14100.0 1.05 1.2179 0.9774 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J13 compound treatment 203480.0 26200.0 1.78 198760.0 22400.0 1.66 2.4385 0.9994 3237412 Sulf1.1-A_000146 OCCOc1cccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc4ccccc4c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J14 mock treatment 182320.0 5020.0 0.34 180920.0 4510.0 0.34 0.4796 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J15 compound treatment 160600.0 -16700.0 -1.14 154680.0 -21700.0 -1.62 -1.9485 -0.9853 3237344 Sulf1.1-A_000147 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cc(Cl)ccc3Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J16 mock treatment 188640.0 11300.0 0.77 192800.0 16400.0 1.22 1.4095 0.9758 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J17 compound treatment 215520.0 38200.0 2.61 215320.0 38900.0 2.9 3.8905 0.9986 3237448 Sulf1.1-A_000148 Cc1ccccc1S(=O)(=O)N2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J18 mock treatment 181720.0 4420.0 0.3 178320.0 1910.0 0.14 0.3138 0.9414 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J19 compound treatment 183320.0 6020.0 0.41 180960.0 4550.0 0.34 0.5299 0.9955 3237362 Sulf1.1-A_000149 OCCOc1cccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J20 mock treatment 175400.0 -1900.0 -0.13 180440.0 4030.0 0.3 0.1207 0.3692 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J21 mock treatment 173200.0 -4100.0 -0.28 178640.0 2230.0 0.17 -0.0801 -0.2463 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J22 mock treatment 172120.0 -5180.0 -0.35 175720.0 -687.0 -0.05 -0.2858 -0.8011 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J23 compound treatment 175360.0 -1940.0 -0.13 181120.0 4710.0 0.35 0.1546 0.4123 3237283 Sulf1.1-A_000150 CC(C)S(=O)(=O)N[C@H]1CCN(Cc2ccc(OCCO)cc2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 J24 mock treatment 166920.0 -10400.0 -0.71 167080.0 -9330.0 -0.69 -0.9912 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K01 compound treatment 198480.0 21200.0 1.44 202800.0 26400.0 1.96 2.4101 0.9885 3237445 Sulf1.1-A_000151 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3cc(Cl)ccc3Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K02 compound treatment 205000.0 27700.0 1.89 203000.0 26600.0 1.98 2.7349 0.9997 3237164 Sulf1.1-A_000152 OCCOc1cccc(CN2CCC(CN3C(=O)c4ccccc4C3=O)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K03 compound treatment 211080.0 33800.0 2.3 202400.0 26000.0 1.93 2.9965 0.9962 3237239 Sulf1.1-A_000153 Cc1nc(cn1C)S(=O)(=O)NCC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K04 compound treatment 203400.0 26100.0 1.78 201920.0 25500.0 1.9 2.601 0.9995 3237465 Sulf1.1-A_000154 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K05 compound treatment 194080.0 16800.0 1.14 187720.0 11300.0 0.84 1.4044 0.9886 3237233 Sulf1.1-A_000155 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3ccc(cc3)c4ccccc4)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K06 compound treatment 193400.0 16100.0 1.1 189720.0 13300.0 0.99 1.4768 0.9987 3237201 Sulf1.1-A_000156 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc(Cl)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K07 mock treatment 183240.0 5940.0 0.41 185000.0 8590.0 0.64 0.7386 0.9757 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K08 mock treatment 187240.0 9940.0 0.68 179720.0 3310.0 0.25 0.6536 0.9063 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K09 compound treatment 219800.0 42500.0 2.9 217800.0 41400.0 3.08 4.2273 0.9995 3237297 Sulf1.1-A_000157 Cc1ccccc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K10 compound treatment 196040.0 18700.0 1.28 196720.0 20300.0 1.51 1.9725 0.9965 3237183 Sulf1.1-A_000158 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3cccc4cccnc34)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K11 compound treatment 225040.0 47700.0 3.25 211440.0 35000.0 2.61 4.1452 0.994 3237171 Sulf1.1-A_000159 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc(Cl)cc3)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K12 compound treatment 195640.0 18300.0 1.25 189360.0 13000.0 0.96 1.5659 0.9917 3237418 Sulf1.1-A_000160 CC(C)S(=O)(=O)N[C@H]1CCN(Cc2cccc(OCCO)c2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K13 compound treatment 159400.0 -17900.0 -1.22 153520.0 -22900.0 -1.7 -2.0674 -0.9866 3237386 Sulf1.1-A_000161 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3cccc4cccnc34)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K14 compound treatment 192000.0 14700.0 1.0 184760.0 8350.0 0.62 1.1483 0.9736 3237261 Sulf1.1-A_000162 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc(Cl)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K15 mock treatment 184200.0 6900.0 0.47 180880.0 4470.0 0.33 0.5681 0.9857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K16 mock treatment 176480.0 -819.0 -0.06 184960.0 8550.0 0.64 0.4106 0.6426 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K17 compound treatment 199600.0 22300.0 1.52 193880.0 17500.0 1.3 1.9947 0.997 3237223 Sulf1.1-A_000163 CC(C)S(=O)(=O)N[C@@H]1CCCN(Cc2ccc(OCCO)cc2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K18 compound treatment 177560.0 261.0 0.02 173840.0 -2570.0 -0.19 -0.1225 -0.6385 3237441 Sulf1.1-A_000164 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3ccc(Cl)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K19 compound treatment 195320.0 18000.0 1.23 199000.0 22600.0 1.68 2.0578 0.9881 3237400 Sulf1.1-A_000165 Cc1ccc(F)cc1S(=O)(=O)N[C@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K20 compound treatment 188160.0 10900.0 0.74 202720.0 26300.0 1.96 1.9084 0.9115 3237398 Sulf1.1-A_000166 COc1ccc(cc1)S(=O)(=O)N[C@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K21 compound treatment 193280.0 16000.0 1.09 189800.0 13400.0 1.0 1.4753 0.999 3237299 Sulf1.1-A_000167 Cc1nc(cn1C)S(=O)(=O)N[C@@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K22 compound treatment 188760.0 11500.0 0.78 189360.0 13000.0 0.96 1.2342 0.9946 3237277 Sulf1.1-A_000168 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc4ccccc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K23 mock treatment 175960.0 -1340.0 -0.09 175880.0 -527.0 -0.04 -0.0923 -0.9287 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 K24 mock treatment 168000.0 -9300.0 -0.63 171240.0 -5170.0 -0.38 -0.7202 -0.9713 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L01 compound treatment 179480.0 2180.0 0.15 180120.0 3710.0 0.28 0.3005 0.9577 3237324 Sulf1.1-A_000169 Cc1nc(cn1C)S(=O)(=O)NC[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L02 mock treatment 175520.0 -1780.0 -0.12 181120.0 4710.0 0.35 0.1623 0.4372 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L03 compound treatment 184600.0 7300.0 0.5 179040.0 2630.0 0.2 0.4905 0.917 3237179 Sulf1.1-A_000170 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3cc(Cl)ccc3Cl)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L04 mock treatment 179440.0 2140.0 0.15 180600.0 4190.0 0.31 0.3239 0.9401 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L05 compound treatment 190480.0 13200.0 0.9 180280.0 3870.0 0.29 0.8393 0.8893 3237242 Sulf1.1-A_000171 Cc1ccc(cc1)S(=O)(=O)NCC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L06 mock treatment 182240.0 4940.0 0.34 185720.0 9310.0 0.69 0.7283 0.9451 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L07 mock treatment 186400.0 9100.0 0.62 178320.0 1910.0 0.14 0.5394 0.8474 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L08 mock treatment 183480.0 6180.0 0.42 181520.0 5110.0 0.38 0.5671 0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L09 compound treatment 199920.0 22600.0 1.54 197120.0 20700.0 1.54 2.1806 1.0 3237293 Sulf1.1-A_000172 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L10 mock treatment 184360.0 7060.0 0.48 181640.0 5230.0 0.39 0.6158 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L11 compound treatment 201920.0 24600.0 1.68 195680.0 19300.0 1.43 2.2012 0.9969 3237255 Sulf1.1-A_000173 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3cccc(F)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L12 mock treatment 191800.0 14500.0 0.99 183760.0 7350.0 0.55 1.086 0.9611 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L13 compound treatment 197040.0 19700.0 1.35 189200.0 12800.0 0.95 1.6249 0.9856 3237296 Sulf1.1-A_000174 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3cccc4cccnc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L14 mock treatment 183160.0 5860.0 0.4 188000.0 11600.0 0.86 0.8927 0.9388 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L15 mock treatment 181480.0 4180.0 0.29 183480.0 7070.0 0.53 0.5738 0.9585 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L16 mock treatment 185920.0 8620.0 0.59 190240.0 13800.0 1.03 1.1436 0.9647 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L17 compound treatment 192120.0 14800.0 1.01 188080.0 11700.0 0.87 1.3288 0.9972 3237338 Sulf1.1-A_000175 COc1ccc(cc1)S(=O)(=O)N[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L18 mock treatment 175920.0 -1380.0 -0.09 178240.0 1830.0 0.14 0.03 0.181 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L19 compound treatment 191480.0 14200.0 0.97 193640.0 17200.0 1.28 1.5906 0.9903 3237459 Sulf1.1-A_000176 Cc1ccc(F)cc1S(=O)(=O)N2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L20 mock treatment 179240.0 1940.0 0.13 177520.0 1110.0 0.08 0.1521 0.9746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L21 compound treatment 195120.0 17800.0 1.21 186320.0 9910.0 0.74 1.3808 0.9714 3237267 Sulf1.1-A_000177 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L22 mock treatment 177240.0 -59.3 0.0 173720.0 -2690.0 -0.2 -0.1443 -0.7212 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L23 mock treatment 168040.0 -9260.0 -0.63 170000.0 -6410.0 -0.48 -0.7835 -0.9904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 L24 mock treatment 164880.0 -12400.0 -0.85 166640.0 -9770.0 -0.73 -1.1127 -0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M01 compound treatment 189200.0 11900.0 0.81 188360.0 12000.0 0.89 1.2028 0.9989 3237244 Sulf1.1-A_000178 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M02 compound treatment 209800.0 32500.0 2.22 201360.0 25000.0 1.86 2.88 0.9961 3237308 Sulf1.1-A_000179 COc1ccc(cc1)S(=O)(=O)NC[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M03 compound treatment 197480.0 20200.0 1.38 191640.0 15200.0 1.13 1.7746 0.9954 3237252 Sulf1.1-A_000180 Cc1ccccc1S(=O)(=O)NC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M04 compound treatment 213840.0 36500.0 2.49 204840.0 28400.0 2.12 3.2579 0.9967 3237470 Sulf1.1-A_000181 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M05 compound treatment 197920.0 20600.0 1.41 191880.0 15500.0 1.15 1.8084 0.9951 3237431 Sulf1.1-A_000182 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3cccc4cccnc34)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M06 compound treatment 204320.0 27000.0 1.84 206000.0 29600.0 2.2 2.86 0.9961 3237350 Sulf1.1-A_000183 Cc1ccccc1S(=O)(=O)N[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M07 compound treatment 194160.0 16900.0 1.15 194600.0 18200.0 1.35 1.7703 0.9967 3237259 Sulf1.1-A_000184 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M08 compound treatment 207120.0 29800.0 2.03 200040.0 23600.0 1.76 2.6814 0.9974 3237378 Sulf1.1-A_000185 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M09 mock treatment 187960.0 10700.0 0.73 183720.0 7310.0 0.54 0.8988 0.9898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M10 mock treatment 187840.0 10500.0 0.72 182800.0 6390.0 0.48 0.8446 0.98 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M11 compound treatment 197880.0 20600.0 1.4 207120.0 30700.0 2.29 2.6085 0.9725 3237227 Sulf1.1-A_000186 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M12 compound treatment 216080.0 38800.0 2.64 209320.0 32900.0 2.45 3.6017 0.9993 3237234 Sulf1.1-A_000187 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3cc(Cl)ccc3Cl)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M13 mock treatment 189840.0 12500.0 0.85 186520.0 10100.0 0.75 1.1368 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M14 mock treatment 205360.0 28100.0 1.91 204400.0 28000.0 2.08 2.826 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M15 compound treatment 212120.0 34800.0 2.37 208360.0 32000.0 2.38 3.3603 1.0 3237462 Sulf1.1-A_000188 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3ccc(Cl)c(Cl)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M16 compound treatment 201520.0 24200.0 1.65 195720.0 19300.0 1.44 2.1841 0.9976 3237169 Sulf1.1-A_000189 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccccc3)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M17 compound treatment 192800.0 15500.0 1.06 194640.0 18200.0 1.36 1.7068 0.9924 3237377 Sulf1.1-A_000190 Cc1ccc(cc1)S(=O)(=O)NCC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M18 compound treatment 198440.0 21100.0 1.44 207920.0 31500.0 2.35 2.6776 0.9727 3237217 Sulf1.1-A_000191 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc4ccccc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M19 compound treatment 198320.0 21000.0 1.43 199800.0 23400.0 1.74 2.2445 0.9953 3237291 Sulf1.1-A_000192 COc1ccc(cc1)S(=O)(=O)N[C@@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M20 compound treatment 193680.0 16400.0 1.12 191440.0 15000.0 1.12 1.5809 1.0 3237442 Sulf1.1-A_000193 COc1ccc(cc1)S(=O)(=O)N2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M21 compound treatment 185400.0 8100.0 0.55 185520.0 9110.0 0.68 0.8701 0.9948 3237302 Sulf1.1-A_000194 Cc1ccc(cc1)S(=O)(=O)N[C@@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M22 compound treatment 185800.0 8500.0 0.58 187400.0 11000.0 0.82 0.9884 0.9857 3237370 Sulf1.1-A_000195 OCCOc1cccc(CN2CCC(CNS(=O)(=O)c3ccc(Cl)c(Cl)c3)CC2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M23 compound treatment 176040.0 -1260.0 -0.09 184840.0 8430.0 0.63 0.3831 0.6048 3237303 Sulf1.1-A_000196 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 M24 compound treatment 185000.0 7700.0 0.53 185680.0 9270.0 0.69 0.8593 0.9909 3237229 Sulf1.1-A_000197 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3ccccc3)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N01 compound treatment 185600.0 8300.0 0.57 181760.0 5350.0 0.4 0.6819 0.9852 3237387 Sulf1.1-A_000198 Cc1ccccc1S(=O)(=O)NC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N02 mock treatment 177440.0 141.0 0.01 183400.0 6990.0 0.52 0.3748 0.72 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N03 compound treatment 216720.0 39400.0 2.69 208800.0 32400.0 2.41 3.6052 0.9985 3237207 Sulf1.1-A_000199 OCCOc1ccc(CN2CCC[C@H](C2)NS(=O)(=O)c3ccc(cc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N04 mock treatment 184600.0 7300.0 0.5 182320.0 5910.0 0.44 0.6632 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N05 compound treatment 183680.0 6380.0 0.44 175880.0 -527.0 -0.04 0.2799 0.6408 3237249 Sulf1.1-A_000200 OCCOc1ccc(CN2CCC(CC2)NS(=O)(=O)c3cc(Cl)ccc3Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N06 mock treatment 188080.0 10800.0 0.73 183320.0 6910.0 0.51 0.8835 0.9848 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N07 compound treatment 198520.0 21200.0 1.45 194040.0 17600.0 1.31 1.951 0.9988 3237236 Sulf1.1-A_000201 OCCOc1ccc(CN2CCC(CNS(=O)(=O)c3cccc4cccnc34)CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N08 mock treatment 187160.0 9860.0 0.67 181760.0 5350.0 0.4 0.7571 0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N09 mock treatment 188160.0 10900.0 0.74 178760.0 2350.0 0.18 0.6474 0.8509 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N10 mock treatment 190480.0 13200.0 0.9 184600.0 8190.0 0.61 1.0666 0.9822 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N11 mock treatment 192040.0 14700.0 1.0 195000.0 18600.0 1.38 1.6891 0.9877 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N12 mock treatment 189600.0 12300.0 0.84 186880.0 10500.0 0.78 1.1442 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N13 mock treatment 189520.0 12200.0 0.83 185800.0 9390.0 0.7 1.0835 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N14 mock treatment 188120.0 10800.0 0.74 181960.0 5550.0 0.41 0.8139 0.9625 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N15 mock treatment 188920.0 11600.0 0.79 181520.0 5110.0 0.38 0.8293 0.9436 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N16 mock treatment 184360.0 7060.0 0.48 188960.0 12600.0 0.93 1.001 0.9524 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N17 mock treatment 181200.0 3900.0 0.27 180600.0 4190.0 0.31 0.4087 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N18 mock treatment 181720.0 4420.0 0.3 181400.0 4990.0 0.37 0.4759 0.9946 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N19 mock treatment 178400.0 1100.0 0.08 177040.0 633.0 0.05 0.0864 0.9749 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N20 mock treatment 177680.0 381.0 0.03 175400.0 -1010.0 -0.07 -0.0346 -0.4367 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N21 mock treatment 176680.0 -619.0 -0.04 178040.0 1630.0 0.12 0.0561 0.436 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N22 mock treatment 175880.0 -1420.0 -0.1 170880.0 -5530.0 -0.41 -0.3593 -0.8502 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N23 mock treatment 172240.0 -5060.0 -0.34 174040.0 -2370.0 -0.18 -0.3685 -0.9513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 N24 mock treatment 170320.0 -6980.0 -0.48 170480.0 -5930.0 -0.44 -0.6484 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O01 compound treatment 220040.0 42700.0 2.91 233120.0 56700.0 4.22 5.0452 0.9836 3237273 Sulf1.1-A_000202 OCCOc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cccc4cccnc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O02 compound treatment 183880.0 6580.0 0.45 174080.0 -2330.0 -0.17 0.1948 0.405 3237426 Sulf1.1-A_000203 COc1ccc(cc1)S(=O)(=O)N[C@@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O03 compound treatment 198880.0 21600.0 1.47 190840.0 14400.0 1.07 1.8 0.9881 3237429 Sulf1.1-A_000204 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3cc(Cl)ccc3Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O04 compound treatment 197000.0 19700.0 1.34 182160.0 5750.0 0.43 1.2525 0.8885 3237432 Sulf1.1-A_000205 Cc1ccccc1S(=O)(=O)N[C@@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O05 compound treatment 192560.0 15300.0 1.04 194520.0 18100.0 1.35 1.689 0.9918 3237425 Sulf1.1-A_000206 OCCOc1cccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccc(Cl)cc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O06 compound treatment 218880.0 41600.0 2.83 209240.0 32800.0 2.44 3.7325 0.9973 3237304 Sulf1.1-A_000207 OCCOc1cccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccccc3)C2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O07 compound treatment 189840.0 12500.0 0.85 177440.0 1030.0 0.08 0.6589 0.7676 3237232 Sulf1.1-A_000208 Cc1ccc(F)cc1S(=O)(=O)NCC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O08 compound treatment 217040.0 39700.0 2.71 209840.0 33400.0 2.49 3.6754 0.9991 3237328 Sulf1.1-A_000209 CC(C)S(=O)(=O)NC[C@@H]1CCCN(Cc2cccc(OCCO)c2)C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O09 compound treatment 188520.0 11200.0 0.76 180480.0 4070.0 0.3 0.7553 0.9179 3237366 Sulf1.1-A_000210 COc1ccc(cc1)S(=O)(=O)NCC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O10 compound treatment 195640.0 18300.0 1.25 189240.0 12800.0 0.96 1.5596 0.9912 3237292 Sulf1.1-A_000211 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O11 mock treatment 181680.0 4380.0 0.3 178320.0 1910.0 0.14 0.3119 0.9426 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O12 mock treatment 182040.0 4740.0 0.32 179000.0 2590.0 0.19 0.365 0.9696 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O13 compound treatment 203920.0 26600.0 1.81 200200.0 23800.0 1.77 2.5355 0.9999 3237389 Sulf1.1-A_000212 Cc1nc(cn1C)S(=O)(=O)NC2CCN(Cc3cccc(OCCO)c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O14 compound treatment 208120.0 30800.0 2.1 211360.0 35000.0 2.6 3.3253 0.9944 3237457 Sulf1.1-A_000213 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3ccc(Cl)cc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O15 compound treatment 197840.0 20500.0 1.4 197840.0 21400.0 1.6 2.1182 0.9979 3237181 Sulf1.1-A_000214 OCCOc1ccc(CN2CCC[C@@H](CNS(=O)(=O)c3ccc(Cl)c(Cl)c3)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O16 compound treatment 189080.0 11800.0 0.8 190040.0 13600.0 1.01 1.2854 0.9933 3237310 Sulf1.1-A_000215 Cc1ccc(F)cc1S(=O)(=O)NC[C@@H]2CCCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O17 compound treatment 188840.0 11500.0 0.79 183560.0 7150.0 0.53 0.9328 0.9819 3237451 Sulf1.1-A_000216 OCCOc1ccc(CN2CCN(CC2)S(=O)(=O)c3cccc(F)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O18 compound treatment 193160.0 15900.0 1.08 193760.0 17400.0 1.29 1.6779 0.9961 3237434 Sulf1.1-A_000217 Cc1nc(cn1C)S(=O)(=O)N[C@@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O19 compound treatment 181840.0 4540.0 0.31 181480.0 5070.0 0.38 0.4859 0.9951 3237263 Sulf1.1-A_000218 COc1ccc(cc1)S(=O)(=O)N[C@H]2CCN(Cc3ccc(OCCO)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O20 compound treatment 205480.0 28200.0 1.92 207360.0 31000.0 2.3 2.9875 0.9959 3237300 Sulf1.1-A_000219 OCCOc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3cccc(F)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O21 compound treatment 188560.0 11300.0 0.77 184600.0 8190.0 0.61 0.9741 0.9935 3237461 Sulf1.1-A_000220 OCCOc1cccc(CN2CCN(CC2)S(=O)(=O)c3cc(Cl)ccc3Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O22 compound treatment 190240.0 12900.0 0.88 186800.0 10400.0 0.77 1.1708 0.9979 3237237 Sulf1.1-A_000221 Cc1ccccc1S(=O)(=O)NCC2CCN(Cc3ccc(OCCO)cc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O23 compound treatment 179640.0 2340.0 0.16 185960.0 9550.0 0.71 0.6156 0.8448 3237384 Sulf1.1-A_000222 OCCOc1cccc(CN2CCC(CC2)NS(=O)(=O)c3cc(Cl)ccc3Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 O24 compound treatment 192480.0 15200.0 1.03 198240.0 21800.0 1.62 1.8809 0.9763 3237414 Sulf1.1-A_000223 Cc1nc(cn1C)S(=O)(=O)N[C@H]2CCN(Cc3cccc(OCCO)c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P01 mock treatment 176960.0 -339.0 -0.02 179920.0 3510.0 0.26 0.1685 0.6421 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P02 mock treatment 176840.0 -459.0 -0.03 176680.0 273.0 0.02 -0.0078 -0.2079 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P03 mock treatment 179160.0 1860.0 0.13 177840.0 1430.0 0.11 0.1651 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P04 mock treatment 182200.0 4900.0 0.33 172760.0 -3650.0 -0.27 0.0443 0.103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P05 mock treatment 180280.0 2980.0 0.2 177920.0 1510.0 0.11 0.2233 0.9612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P06 mock treatment 180760.0 3460.0 0.24 175720.0 -687.0 -0.05 0.1307 0.5414 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P07 mock treatment 180800.0 3500.0 0.24 178160.0 1750.0 0.13 0.261 0.9596 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P08 mock treatment 178440.0 1140.0 0.08 178960.0 2550.0 0.19 0.1894 0.9223 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P09 mock treatment 186080.0 8780.0 0.6 175160.0 -1250.0 -0.09 0.3577 0.5904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P10 mock treatment 182160.0 4860.0 0.33 176120.0 -287.0 -0.02 0.2192 0.6602 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P11 mock treatment 180280.0 2980.0 0.2 176360.0 -46.8 0.0 0.1412 0.6949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P12 mock treatment 179760.0 2460.0 0.17 175960.0 -447.0 -0.03 0.0951 0.5561 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P13 mock treatment 178360.0 1060.0 0.07 178400.0 1990.0 0.15 0.156 0.9455 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P14 mock treatment 179400.0 2100.0 0.14 177200.0 793.0 0.06 0.143 0.9232 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P15 mock treatment 181000.0 3700.0 0.25 176240.0 -167.0 -0.01 0.1696 0.6715 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P16 mock treatment 180320.0 3020.0 0.21 170200.0 -6210.0 -0.46 -0.181 -0.3579 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P17 mock treatment 176680.0 -619.0 -0.04 174720.0 -1690.0 -0.13 -0.1186 -0.8956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P18 mock treatment 171320.0 -5980.0 -0.41 175400.0 -1010.0 -0.07 -0.3412 -0.8233 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P19 mock treatment 175280.0 -2020.0 -0.14 176120.0 -287.0 -0.02 -0.1124 -0.8071 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P20 mock treatment 171880.0 -5420.0 -0.37 169960.0 -6450.0 -0.48 -0.6005 -0.9917 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P21 mock treatment 171560.0 -5740.0 -0.39 169040.0 -7370.0 -0.55 -0.6644 -0.9863 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P22 mock treatment 170560.0 -6740.0 -0.46 171080.0 -5330.0 -0.4 -0.6052 -0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P23 mock treatment 171160.0 -6140.0 -0.42 166200.0 -10200.0 -0.76 -0.8331 -0.9606 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2168 P24 mock treatment 164280.0 -13000.0 -0.89 169040.0 -7370.0 -0.55 -1.0153 -0.9732 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A01 compound treatment 186840.0 11000.0 0.75 185520.0 10100.0 0.75 1.064 1.0 1952677 BCB03_000001 CCCCCCC#Cc1c(C(CC(=O)C)c2ccccc2)c(=O)oc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A02 compound treatment 161000.0 -14800.0 -1.01 162200.0 -13200.0 -0.98 -1.409 -0.9999 3092787 BCB03_000002 CC(C)OC(=O)/C=C\1/C[C@H](O[C@H](O1)c2cccc(c2)C(F)(F)F)c3cccc(c3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A03 compound treatment 165480.0 -10300.0 -0.71 165840.0 -9550.0 -0.71 -1.0015 -1.0 1952679 BCB03_000003 Clc1ccc2oc(=O)cc(Sc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A04 compound treatment 166840.0 -8990.0 -0.61 165000.0 -10400.0 -0.77 -0.9801 -0.9933 3092788 BCB03_000004 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccccc2C(F)(F)F)c3ccccc3C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A05 compound treatment 168840.0 -6990.0 -0.48 162320.0 -13100.0 -0.97 -1.0248 -0.946 1952690 BCB03_000005 COC(=O)CC(C(=O)OC)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A06 compound treatment 164960.0 -10900.0 -0.74 162160.0 -13200.0 -0.98 -1.2202 -0.9902 3001175 BCB03_000006 CON(C)C(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(Cl)c2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A07 compound treatment 168600.0 -7230.0 -0.49 169160.0 -6230.0 -0.46 -0.6764 -0.9995 1952707 BCB03_000007 CCCCSc1cc(=O)oc2cc(OC)ccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A08 compound treatment 162640.0 -13200.0 -0.9 165360.0 -10000.0 -0.75 -1.1637 -0.9957 3001176 BCB03_000008 CC(C)OC(=O)CC(=O)CC(O)c1ccc(cc1)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A09 compound treatment 168640.0 -7190.0 -0.49 166840.0 -8550.0 -0.64 -0.7965 -0.9916 1952793 BCB03_000009 FC(F)(F)c1ccc(cc1)C(=O)Oc2ccccc2C#Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A10 compound treatment 162360.0 -13500.0 -0.92 163800.0 -11600.0 -0.86 -1.2593 -0.9995 3001249 BCB03_000010 CC(C)OC(=O)CC(=O)CC(O)c1cccc(c1)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A11 compound treatment 157000.0 -18800.0 -1.28 158520.0 -16900.0 -1.26 -1.7955 -0.9999 1952795 BCB03_000011 COC(=O)/C=C/c1cc(OC)cc(C#Cc2ccc(Oc3ccccc3)c(OC)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A12 compound treatment 165320.0 -10500.0 -0.72 166040.0 -9350.0 -0.7 -0.9987 -0.9999 3001250 BCB03_000012 CC(C)OC(=O)CC(=O)CC(O)c1cccc(C#N)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A13 mock treatment 163440.0 -12400.0 -0.84 164600.0 -10800.0 -0.8 -1.1651 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A14 mock treatment 162720.0 -13100.0 -0.89 166240.0 -9150.0 -0.68 -1.1135 -0.991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A15 compound treatment 156240.0 -19600.0 -1.34 159080.0 -16300.0 -1.21 -1.8027 -0.9989 1952801 BCB03_000013 Oc1ccccc1C#Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A16 compound treatment 165400.0 -10400.0 -0.71 162880.0 -12500.0 -0.93 -1.1611 -0.9911 3001251 BCB03_000014 CC(C)OC(=O)CC(=O)CC(O)c1ccc(C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A17 compound treatment 166560.0 -9270.0 -0.63 174600.0 -792.0 -0.06 -0.4884 -0.7697 1952761 BCB03_000015 COc1ccc(cc1)C(=C2C(=O)Oc3ccccc23)c4ccc(OC)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A18 compound treatment 194000.0 18200.0 1.24 194520.0 19100.0 1.42 1.8828 0.9976 3001252 BCB03_000016 COC(=O)C1=CCC(CC1)(C=C)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A19 compound treatment 174040.0 -1790.0 -0.12 168800.0 -6590.0 -0.49 -0.433 -0.8566 1952804 BCB03_000017 COc1cc(CO[Si](C)(C)C(C)(C)C)cc(C#CC2(O)CCCCC2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A20 compound treatment 180280.0 4450.0 0.3 177400.0 2010.0 0.15 0.3204 0.9467 3001253 BCB03_000018 COC(=O)/C=C(/CC(O)c1cccc(Cl)c1)\OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A21 compound treatment 173760.0 -2070.0 -0.14 172800.0 -2590.0 -0.19 -0.236 -0.9881 1952805 BCB03_000019 CC(C)(C)[Si](C)(C)OCCNC(=O)c1cc(cc2c(coc12)C(O)(c3ccccc3)c4ccccc4)c5cc(I)cc(I)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A22 compound treatment 167600.0 -8230.0 -0.56 163480.0 -11900.0 -0.89 -1.0235 -0.9756 3001254 BCB03_000020 OC(C/C(=C/C(=O)OCCF)/OCCF)c1cccc(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A23 compound treatment 206520.0 30700.0 2.09 205000.0 29600.0 2.2 3.0379 0.9997 1952808 BCB03_000021 CCCCCc1cc2ccccc2o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 A24 compound treatment 166600.0 -9230.0 -0.63 165800.0 -9590.0 -0.71 -0.9496 -0.998 3001255 BCB03_000022 CCO/C(=C\C(=O)OC)/CC(O)c1cccc(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B01 compound treatment 171720.0 -4110.0 -0.28 163880.0 -11500.0 -0.86 -0.8038 -0.8918 3000770 BCB03_000023 Cc1ccc(cc1)S(=O)(=O)N2C[C@H]([C@@H](C[C@H]2c3ccccc3)Sc4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B02 compound treatment 253240.0 77400.0 5.28 244480.0 69100.0 5.14 7.3679 0.9999 3070361 BCB03_000024 CN1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3c5ccc(CO)cc5)c6cccs6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B03 compound treatment 160320.0 -15500.0 -1.06 165440.0 -9950.0 -0.74 -1.2713 -0.9849 3000771 BCB03_000025 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B04 compound treatment 200480.0 24700.0 1.68 202240.0 26800.0 2.0 2.6015 0.9963 3189527 BCB03_000026 OCCCC1=CC(C2CC2)N(Cc3cccc(OC(F)(F)F)c3)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B05 compound treatment 169800.0 -6030.0 -0.41 170040.0 -5350.0 -0.4 -0.5722 -0.9999 3092495 BCB03_000027 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(F)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B06 compound treatment 254560.0 78700.0 5.37 244480.0 69100.0 5.14 7.4316 0.9998 3189528 BCB03_000028 OCc1ccc(cc1)C2=CC(C3CC3)N(Cc4sc5ccccc5c4Cl)/C(=N\P(=O)(Oc6ccccc6)Oc7ccccc7)/C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B07 compound treatment 165920.0 -9910.0 -0.68 168240.0 -7150.0 -0.53 -0.854 -0.9931 3092496 BCB03_000029 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(OC)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B08 compound treatment 177600.0 1770.0 0.12 174080.0 -1310.0 -0.1 0.0165 0.1059 3189529 BCB03_000030 CN1C(=O)C2C(C3C(C4CC4)N(C)C2C=C3c5ccc(CO)cc5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B09 compound treatment 165520.0 -10300.0 -0.7 167440.0 -7950.0 -0.59 -0.9154 -0.9964 3000773 BCB03_000031 CCOC(=O)C1=C[C@H](N([C@H]1c2cccc(Cl)c2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B10 compound treatment 165000.0 -10800.0 -0.74 167240.0 -8150.0 -0.61 -0.9509 -0.9953 3070364 BCB03_000032 CN1C(=O)C2C(C3C(N(C)C2C=C3CCCO)c4ccc(CN5CCCC5)cc4)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B11 compound treatment 172280.0 -3550.0 -0.24 175480.0 88.0 0.01 -0.1663 -0.6877 3000774 BCB03_000033 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2Cl)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B12 compound treatment 189360.0 13500.0 0.92 183760.0 8370.0 0.62 1.0928 0.9817 3189532 BCB03_000034 CN/1C(C=C(CCCO)C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B13 mock treatment 169200.0 -6630.0 -0.45 167520.0 -7870.0 -0.59 -0.7337 -0.9918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B14 mock treatment 161440.0 -14400.0 -0.98 161000.0 -14400.0 -1.07 -1.451 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B15 compound treatment 162960.0 -12900.0 -0.88 159200.0 -16200.0 -1.21 -1.4724 -0.9878 3000775 BCB03_000035 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(C)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B16 compound treatment 174640.0 -1190.0 -0.08 184000.0 8610.0 0.64 0.3958 0.613 3189533 BCB03_000036 CC1C=C(CCCO)C/C(=N/P(=O)(Oc2ccccc2)Oc3ccccc3)/N1Cc4cccc(OC(F)(F)F)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B17 compound treatment 162480.0 -13300.0 -0.91 164040.0 -11400.0 -0.84 -1.2408 -0.9993 3092507 BCB03_000037 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(OC)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B18 compound treatment 169120.0 -6710.0 -0.46 168920.0 -6470.0 -0.48 -0.6639 -0.9997 3189534 BCB03_000038 CN1C(=O)C2C(C3C(N(Cc4sc5ccccc5c4Cl)C2C=C3CCCO)c6ccc(CN7CCCC7)cc6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B19 compound treatment 164840.0 -11000.0 -0.75 165280.0 -10100.0 -0.75 -1.0618 -1.0 3092508 BCB03_000039 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B20 compound treatment 167320.0 -8510.0 -0.58 166600.0 -8790.0 -0.65 -0.8728 -0.9982 3070367 BCB03_000040 CC1C2C3C(C(C=C2CCCO)N1Cc4cccc(OC(F)(F)F)c4)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B21 compound treatment 161080.0 -14700.0 -1.01 160200.0 -15200.0 -1.13 -1.5104 -0.9983 3000857 BCB03_000041 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(F)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B22 compound treatment 190120.0 14300.0 0.97 188560.0 13200.0 0.98 1.3821 1.0 3189537 BCB03_000042 CN1C(=O)C2C(C3C(N(C)C2C=C3c4ccc(CO)cc4)c5cccs5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B23 compound treatment 161760.0 -14100.0 -0.96 163720.0 -11700.0 -0.87 -1.2924 -0.9988 3000858 BCB03_000043 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(Cl)c(Cl)c2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 B24 compound treatment 182440.0 6610.0 0.45 187600.0 12200.0 0.91 0.9613 0.9477 3189538 BCB03_000044 CN1C(=O)C2C(C3C(C4CC4)N(Cc5sc6ccccc6c5Cl)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C01 compound treatment 165840.0 -9990.0 -0.68 165040.0 -10400.0 -0.77 -1.0262 -0.9981 1952809 BCB03_000045 CC(=O)Oc1ccccc1C#Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C02 compound treatment 170720.0 -5110.0 -0.35 166080.0 -9310.0 -0.69 -0.7362 -0.9493 3092872 BCB03_000046 FCCOC(=O)C1=CCC(O1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C03 compound treatment 177720.0 1890.0 0.13 183720.0 8330.0 0.62 0.5296 0.8364 1952811 BCB03_000047 CC(C)(C)[Si](C)(C)Oc1ccc(C#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C04 compound treatment 176200.0 374.0 0.03 174080.0 -1310.0 -0.1 -0.051 -0.5058 3000746 BCB03_000048 CC(C)OC(=O)C1=CCC(O1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C05 compound treatment 253720.0 77900.0 5.31 272520.0 97100.0 7.23 8.8667 0.9885 1952813 BCB03_000049 OCCCC#Cc1cc(O)cc(Cl)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C06 compound treatment 171640.0 -4190.0 -0.29 174800.0 -592.0 -0.04 -0.233 -0.8067 3000748 BCB03_000050 CCOC(=O)C1=CCC(O1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C07 compound treatment 172280.0 -3550.0 -0.24 175160.0 -232.0 -0.02 -0.1832 -0.7557 1952814 BCB03_000051 CC(=O)Cc1c(Cl)cc(cc1I)C(=O)NCCO[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C08 compound treatment 176200.0 374.0 0.03 170640.0 -4750.0 -0.35 -0.2321 -0.6545 3000750 BCB03_000052 COC(=O)C1=CCC(O1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C09 compound treatment 170680.0 -5150.0 -0.35 171320.0 -4070.0 -0.3 -0.4624 -0.9973 1952821 BCB03_000053 CC(C)(C)[Si](C)(C)COCNC(=O)C1CC2C3C(OC2C(Cl)C1)C4(CCCC4)OC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C10 compound treatment 168960.0 -6870.0 -0.47 171920.0 -3470.0 -0.26 -0.5137 -0.9608 2065163 BCB03_000054 CCOC(=O)/C=C/c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C11 mock treatment 164560.0 -11300.0 -0.77 171800.0 -3590.0 -0.27 -0.7322 -0.9002 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C12 mock treatment 170040.0 -5790.0 -0.39 170440.0 -4950.0 -0.37 -0.5396 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C13 compound treatment 206640.0 30800.0 2.1 201760.0 26400.0 1.96 2.8732 0.9994 1952823 BCB03_000055 C#Cc1ccccc1Oc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C14 compound treatment 168640.0 -7190.0 -0.49 173840.0 -1550.0 -0.12 -0.4281 -0.8505 3000752 BCB03_000056 CCOC(=O)/C=C/c1cc(F)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C15 mock treatment 169880.0 -5950.0 -0.41 167360.0 -8030.0 -0.6 -0.7094 -0.9821 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C16 mock treatment 168840.0 -6990.0 -0.48 168280.0 -7110.0 -0.53 -0.7111 -0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C17 compound treatment 164640.0 -11200.0 -0.76 169520.0 -5870.0 -0.44 -0.8483 -0.9651 1952825 BCB03_000057 CCCC(C)(O)C#Cc1cc(cc(C(=O)NCCO[Si](C)(C)C(C)(C)C)c1OC(=O)C)c2cc(F)cc(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C18 compound treatment 175440.0 -386.0 -0.03 166680.0 -8710.0 -0.65 -0.4771 -0.7352 3000753 BCB03_000058 CCOC(=O)/C=C/c1cc(ccc1O)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C19 compound treatment 179880.0 4050.0 0.28 173800.0 -1590.0 -0.12 0.1116 0.3713 1952828 BCB03_000059 CCc1cc(OC)c(O)c(C#CC(O)c2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C20 compound treatment 192720.0 16900.0 1.15 190000.0 14600.0 1.09 1.5832 0.9996 3000754 BCB03_000060 CCOC(=O)/C=C/c1cccc(OC)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C21 compound treatment 194760.0 18900.0 1.29 196680.0 21300.0 1.58 2.0331 0.9948 1952829 BCB03_000061 O=C(/C(=C\c1ccccc1)/c2cccc(c2)S(=O)=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C22 compound treatment 181760.0 5930.0 0.4 179520.0 4130.0 0.31 0.5033 0.9908 3000755 BCB03_000062 CCOC(=O)/C=C/c1cccc(C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C23 compound treatment 163560.0 -12300.0 -0.84 161120.0 -14300.0 -1.06 -1.3424 -0.993 1952832 BCB03_000063 CCc1cc(OC)c(O)c(C#CC(C)(O)C=C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 C24 compound treatment 162000.0 -13800.0 -0.94 162480.0 -12900.0 -0.96 -1.3461 -1.0 3000762 BCB03_000064 CCOC(=O)/C=C/c1ccccc1OC(=O)C#CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D01 compound treatment 166600.0 -9230.0 -0.63 162720.0 -12700.0 -0.94 -1.1117 -0.9806 3000859 BCB03_000065 CCOC(=O)C1=C[C@H](N([C@H]1c2cccc(Cl)c2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D02 compound treatment 157600.0 -18200.0 -1.24 152520.0 -22900.0 -1.7 -2.0824 -0.988 3189665 BCB03_000066 OCCCC1=CC(N(Cc2cccc(OC(F)(F)F)c2)/C(=N\P(=O)(Oc3ccccc3)Oc4ccccc4)/C1)c5ccc(CN6CCCC6)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D03 compound treatment 172360.0 -3470.0 -0.24 163160.0 -12200.0 -0.91 -0.8109 -0.8621 3092513 BCB03_000067 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2Cl)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D04 compound treatment 219480.0 43700.0 2.98 211680.0 36300.0 2.7 4.0142 0.9988 3189666 BCB03_000068 OCCCC1=CC(C2CC2)N(Cc3cc4OCOc4cc3Br)/C(=N\P(=O)(Oc5ccccc5)Oc6ccccc6)/C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D05 compound treatment 178840.0 3010.0 0.21 175000.0 -392.0 -0.03 0.1246 0.6007 3092514 BCB03_000069 CCOC(=O)C1=C[C@H](N([C@H]1c2cccc3ccccc23)S(=O)(=O)c4ccc(C)cc4)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D06 compound treatment 162720.0 -13100.0 -0.89 164040.0 -11400.0 -0.84 -1.2293 -0.9996 3189668 BCB03_000070 OCCCC1=CC(N(Cc2sc3ccccc3c2Cl)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C1)c6ccc(CN7CCCC7)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D07 compound treatment 167160.0 -8670.0 -0.59 166560.0 -8830.0 -0.66 -0.8826 -0.9986 3000861 BCB03_000071 CCOC(=O)C1=C[C@@H](C(C)C)N([C@H]1c2ccc(cc2)C(F)(F)F)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D08 compound treatment 216280.0 40500.0 2.76 208640.0 33200.0 2.47 3.7 0.9985 3189669 BCB03_000072 CN1C(=O)C2C(C3C(C4CC4)N(Cc5cc6OCOc6cc5Br)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D09 compound treatment 167120.0 -8710.0 -0.59 161520.0 -13900.0 -1.03 -1.1498 -0.9655 3092596 BCB03_000073 CCOC(=O)C1=C[C@@H](C(C)C)N([C@H]1c2ccc(cc2)C(C)C)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D10 compound treatment 188960.0 13100.0 0.9 187760.0 12400.0 0.92 1.284 0.9999 3189670 BCB03_000074 NC(=O)N1C(=O)C2C(C3C(N(Cc4cc5OCOc5cc4Br)C2C=C3CCCO)c6ccc(CN7CCCC7)cc6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D11 mock treatment 169600.0 -6230.0 -0.42 167800.0 -7590.0 -0.57 -0.6997 -0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D12 mock treatment 166120.0 -9710.0 -0.66 167040.0 -8350.0 -0.62 -0.9075 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D13 compound treatment 165600.0 -10200.0 -0.7 166080.0 -9310.0 -0.69 -0.9831 -1.0 3000869 BCB03_000075 CCOC(=O)C1=C[C@@H](C(C)C)N([C@H]1c2ccccc2F)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D14 compound treatment 184560.0 8730.0 0.6 181240.0 5850.0 0.44 0.7288 0.9881 3070434 BCB03_000076 NC(=O)N1C(=O)C2C(C3C(N(Cc4sc5ccccc5c4Cl)C2C=C3CCCO)c6ccc(CN7CCCC7)cc6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D15 mock treatment 171600.0 -4230.0 -0.29 166200.0 -9190.0 -0.68 -0.6875 -0.9261 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D16 mock treatment 165040.0 -10800.0 -0.74 167720.0 -7670.0 -0.57 -0.9238 -0.9922 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D17 compound treatment 169480.0 -6350.0 -0.43 169040.0 -6350.0 -0.47 -0.6402 -0.999 3000870 BCB03_000077 CCOC(=O)C1=C[C@@H](CC)N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D18 compound treatment 217160.0 41300.0 2.82 218040.0 42600.0 3.17 4.2371 0.9982 3189673 BCB03_000078 NC(=O)N1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5cccs5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D19 compound treatment 169280.0 -6550.0 -0.45 168560.0 -6830.0 -0.51 -0.6751 -0.9979 3092599 BCB03_000079 CCOC(=O)C1=CCN(C1c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D20 compound treatment 192160.0 16300.0 1.11 183080.0 7690.0 0.57 1.192 0.9521 3189674 BCB03_000080 OCc1ccc(cc1)C2=CC(N(Cc3cccc(OC(F)(F)F)c3)CC2)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D21 compound treatment 171520.0 -4310.0 -0.29 163480.0 -11900.0 -0.89 -0.8345 -0.8936 3092600 BCB03_000081 CCC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccccc3)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D22 compound treatment 277480.0 102000.0 6.93 280520.0 105000.0 7.82 10.4332 0.9982 3070436 BCB03_000082 NC(=O)N1C(=O)C2C(C3C(C4CC4)N(Cc5sc6ccccc6c5Cl)C2C=C3c7ccc(CO)cc7)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D23 compound treatment 167000.0 -8830.0 -0.6 164920.0 -10500.0 -0.78 -0.9766 -0.9918 3092601 BCB03_000083 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 D24 compound treatment 162280.0 -13500.0 -0.92 164720.0 -10700.0 -0.79 -1.2147 -0.9972 3070437 BCB03_000084 CN1CCC(=CC1C2CC2)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E01 mock treatment 171720.0 -4110.0 -0.28 173000.0 -2390.0 -0.18 -0.3239 -0.9761 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E02 mock treatment 166320.0 -9510.0 -0.65 174080.0 -1310.0 -0.1 -0.5273 -0.8046 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E03 mock treatment 175520.0 -306.0 -0.02 175760.0 368.0 0.03 0.0046 0.1333 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E04 compound treatment 174840.0 -986.0 -0.07 179720.0 4330.0 0.32 0.1802 0.5477 3093836 BCB03_000085 CCOC(=O)[C@H]1CC=C2[C@@H]1c3ccccc3OC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E05 compound treatment 187800.0 12000.0 0.82 192480.0 17100.0 1.27 1.4765 0.977 1952837 BCB03_000086 COCCNC(=O)c1ccc(c(C#CC(C)(O)CC(C)C)c1O)c2cc(F)cc(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E06 compound treatment 180520.0 4690.0 0.32 179360.0 3970.0 0.3 0.4351 0.9992 3000764 BCB03_000087 CCOC(=O)[C@H]1CC=C2[C@@H]1c3cc(Br)ccc3OC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E07 compound treatment 175960.0 134.0 0.01 179920.0 4530.0 0.34 0.2447 0.7259 1952838 BCB03_000088 COc1cc(CO[Si](C)(C)C(C)(C)C)cc(C#CC2(O)CCC3C2CC4Cc5cc(O)ccc5C43)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E08 compound treatment 178560.0 2730.0 0.19 177040.0 1650.0 0.12 0.2185 0.9794 3000765 BCB03_000089 CCOC(=O)/C=C/c1cc(Br)ccc1OC(=O)C#CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E09 mock treatment 176120.0 294.0 0.02 172240.0 -3150.0 -0.23 -0.1517 -0.6444 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E10 mock treatment 180640.0 4810.0 0.33 175360.0 -32.0 0.0 0.2304 0.702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E11 compound treatment 175440.0 -386.0 -0.03 173280.0 -2110.0 -0.16 -0.1298 -0.8143 1952839 BCB03_000090 Oc1ccccc1C#CC#Cc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E12 compound treatment 178400.0 2570.0 0.18 178840.0 3450.0 0.26 0.3055 0.9828 3000766 BCB03_000091 O=c1oc2ccccc2cc1C#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E13 compound treatment 189280.0 13500.0 0.92 189480.0 14100.0 1.05 1.39 0.9978 1952842 BCB03_000092 COC(=O)Cc1cc(cc(I)c1O)c2cc(F)cc(I)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E14 compound treatment 177320.0 1490.0 0.1 180120.0 4730.0 0.35 0.3208 0.8758 3000767 BCB03_000093 Cn1c2C3NC(C(=O)c2c4ccccc14)C(C)(C=C3)C(=O)OCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E15 compound treatment 173600.0 -2230.0 -0.15 174120.0 -1270.0 -0.09 -0.1743 -0.9742 2065685 BCB03_000094 CCOCOc1cc(O)c(C(=O)/C=C/c2ccccc2)c(OCOCC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E16 compound treatment 194760.0 18900.0 1.29 193320.0 17900.0 1.33 1.8563 0.9999 3000768 BCB03_000095 [O-][N+](=O)c1ccccc1S(=O)(=O)N2C3CC=C(C2C(=O)c4c3[nH]c5ccccc45)C(=O)OCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E17 mock treatment 172840.0 -2990.0 -0.2 175720.0 328.0 0.02 -0.1267 -0.6179 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E18 mock treatment 174160.0 -1670.0 -0.11 177400.0 2010.0 0.15 0.0253 0.135 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E19 compound treatment 184640.0 8810.0 0.6 180120.0 4730.0 0.35 0.6737 0.9675 2065729 BCB03_000096 CCOCOc1cc(OCOCC)c2C(=O)CC(Oc2c1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E20 compound treatment 185480.0 9650.0 0.66 188840.0 13400.0 1.0 1.1731 0.9793 3093843 BCB03_000097 CCOC(=O)C1=CC[C@@H]2[C@H]1C(=O)N(C2=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E21 compound treatment 187880.0 12100.0 0.82 190200.0 14800.0 1.1 1.3604 0.9895 1952773 BCB03_000098 CCCNC(=O)c1cc(cc2c3C(=O)OC4(CCCC4)c3oc12)c5cc(F)cc(F)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E22 compound treatment 173800.0 -2030.0 -0.14 175920.0 528.0 0.04 -0.0699 -0.4867 3000776 BCB03_000099 CCOC(=O)C1=CC[C@@H]2[C@H]1C(=O)N(CC)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E23 compound treatment 175720.0 -106.0 -0.01 179960.0 4570.0 0.34 0.2353 0.6919 1952780 BCB03_000100 COc1cccc(c1)c2c(oc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 E24 compound treatment 166480.0 -9350.0 -0.64 168200.0 -7190.0 -0.54 -0.8291 -0.9962 3000848 BCB03_000101 CCOC(=O)[C@H]1[C@H](C[C@@H]2[C@H]1C(=O)N(CC)C2=O)Sc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F01 mock treatment 167560.0 -8270.0 -0.56 169200.0 -6190.0 -0.46 -0.7244 -0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F02 mock treatment 172440.0 -3390.0 -0.23 169560.0 -5830.0 -0.43 -0.4702 -0.9563 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F03 compound treatment 178960.0 3130.0 0.21 175480.0 88.0 0.01 0.1557 0.7284 3000874 BCB03_000102 Cc1ccc(cc1)[C@@H]2N(CC=C2C(=O)O)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F04 compound treatment 175600.0 -226.0 -0.02 179800.0 4410.0 0.33 0.2211 0.6731 3187712 BCB03_000103 OCCCC1=CC(N(Cc2cc3OCOc3cc2Br)CC1)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F05 compound treatment 178280.0 2450.0 0.17 181720.0 6330.0 0.47 0.4513 0.903 3092602 BCB03_000104 C[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F06 compound treatment 180640.0 4810.0 0.33 186240.0 10800.0 0.81 0.803 0.9213 3187713 BCB03_000105 CN1C(C2CC2)C3C4C(C1C=C3c5ccc(CO)cc5)C(=O)N(C(=O)N)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F07 compound treatment 178080.0 2250.0 0.15 173640.0 -1750.0 -0.13 0.0164 0.0816 3092680 BCB03_000106 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F08 compound treatment 214480.0 38700.0 2.64 225040.0 49600.0 3.7 4.4763 0.9863 3187714 BCB03_000107 OCCCC1=CC(C2CC2)N(Cc3cc4OCOc4cc3Br)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F09 mock treatment 171640.0 -4190.0 -0.29 181400.0 6010.0 0.45 0.1144 0.2156 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F10 mock treatment 174640.0 -1190.0 -0.08 176680.0 1290.0 0.1 0.0106 0.0844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F11 compound treatment 182520.0 6690.0 0.46 181240.0 5850.0 0.44 0.6305 0.9997 3092681 BCB03_000108 CCC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F12 compound treatment 190200.0 14400.0 0.98 181560.0 6170.0 0.46 1.0175 0.9403 3070498 BCB03_000109 CC1C=C(CCCO)CCN1Cc2cccc(OC(F)(F)F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F13 compound treatment 182640.0 6810.0 0.46 176000.0 608.0 0.05 0.3605 0.7723 3000959 BCB03_000110 CC(C)[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F14 compound treatment 208480.0 32700.0 2.23 204800.0 29400.0 2.19 3.1219 1.0 3070499 BCB03_000111 CN1CCC(=CC1c2cccs2)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F15 compound treatment 182800.0 6970.0 0.48 178720.0 3330.0 0.25 0.5113 0.9538 3092683 BCB03_000112 Cc1ccc(cc1)[C@@H]2N([C@@H](C=C2C(=O)O)C(C)(C)C)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F16 compound treatment 194480.0 18700.0 1.27 185360.0 9970.0 0.74 1.4238 0.9671 3187718 BCB03_000113 CN1C(C2C3C(C1C=C2CCCO)C(=O)N(C(=O)N)C3=O)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F17 mock treatment 182200.0 6370.0 0.43 174320.0 -1070.0 -0.08 0.2508 0.5678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F18 mock treatment 172400.0 -3430.0 -0.23 172680.0 -2710.0 -0.2 -0.3079 -0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F19 compound treatment 181520.0 5690.0 0.39 179680.0 4290.0 0.32 0.5001 0.9953 3092684 BCB03_000114 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F20 compound treatment 186960.0 11100.0 0.76 188840.0 13400.0 1.0 1.2445 0.9907 3187719 BCB03_000115 OCCCC1=CC(N(Cc2sc3ccccc3c2Cl)CC1)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F21 compound treatment 174080.0 -1750.0 -0.12 173200.0 -2190.0 -0.16 -0.1996 -0.988 3000962 BCB03_000116 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C#N)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F22 compound treatment 253080.0 77300.0 5.27 250720.0 75300.0 5.61 7.6886 0.9995 3187720 BCB03_000117 OCc1ccc(cc1)C2=CC(C3CC3)N(Cc4sc5ccccc5c4Cl)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F23 compound treatment 170440.0 -5390.0 -0.37 169840.0 -5550.0 -0.41 -0.5519 -0.9983 3092686 BCB03_000118 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(OC)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 F24 compound treatment 183280.0 7450.0 0.51 176480.0 1090.0 0.08 0.4166 0.8096 3070502 BCB03_000119 CN1C(C2C3C(C1C=C2c4ccc(CO)cc4)C(=O)N(C(=O)N)C3=O)c5cccs5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G01 compound treatment 171240.0 -4590.0 -0.31 176160.0 768.0 0.06 -0.1807 -0.5684 3107406 BCB03_000120 COC(=O)/C=C/c1cc(OC)c2oc(c(C)c2c1)c3ccccc3.c1ccsc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G02 compound treatment 184640.0 8810.0 0.6 189240.0 13800.0 1.03 1.1537 0.967 3000850 BCB03_000121 OC(=O)C1=CC[C@@H]2[C@H]1C(=O)N(C2=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G03 mock treatment 184600.0 8770.0 0.6 180320.0 4930.0 0.37 0.6823 0.9724 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G04 mock treatment 180520.0 4690.0 0.32 186520.0 11100.0 0.83 0.8119 0.9144 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G05 compound treatment 174400.0 -1430.0 -0.1 178480.0 3090.0 0.23 0.0937 0.3757 1952785 BCB03_000122 CCc1cc(OC)c2oc(c(C(=O)c3ccccc3)c2c1)c4ccc(Oc5ccccc5)c(OC)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G06 compound treatment 182280.0 6450.0 0.44 186960.0 11600.0 0.86 0.9199 0.9514 3092501 BCB03_000123 OC(=O)[C@H]1[C@H](C[C@@H]2[C@H]1C(=O)N(C2=O)c3ccccc3)Sc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G07 compound treatment 189080.0 13300.0 0.9 190360.0 15000.0 1.11 1.4267 0.9946 1952788 BCB03_000124 CCc1cc(OC)c2oc(c(C(=O)c3ccc(OC)cc3)c2c1)c4ccc(Oc5ccccc5)c(OC)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G08 compound treatment 182000.0 6170.0 0.42 180240.0 4850.0 0.36 0.5528 0.9971 3092502 BCB03_000125 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G09 compound treatment 199560.0 23700.0 1.62 202120.0 26700.0 1.99 2.5508 0.9947 2065776 BCB03_000126 Cc1ccc(SC2(CC(=O)N(Cc3ccccc3)C2c4ccccc4I)C(=O)NCc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G10 compound treatment 188440.0 12600.0 0.86 188160.0 12800.0 0.95 1.28 0.9988 3000853 BCB03_000127 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G11 compound treatment 210280.0 34500.0 2.35 202640.0 27200.0 2.03 3.0949 0.9973 1034979 BCB03_000128 c1c(cn2ccccc12)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G12 compound treatment 187960.0 12100.0 0.83 182440.0 7050.0 0.52 0.9559 0.9758 3000854 BCB03_000129 CCOC(=O)C1=CC[C@H](N([C@H]1c2cccc(OC)c2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G13 compound treatment 182840.0 7010.0 0.48 181040.0 5650.0 0.42 0.6354 0.9979 2065809 BCB03_000130 COC(=O)Cc1cn[nH]c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G14 compound treatment 195360.0 19500.0 1.33 185800.0 10400.0 0.77 1.4894 0.9668 3000855 BCB03_000131 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G15 compound treatment 181600.0 5770.0 0.39 182640.0 7250.0 0.54 0.6598 0.988 2065826 BCB03_000132 CC(C(=O)O)c1ccccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G16 compound treatment 191960.0 16100.0 1.1 185280.0 9890.0 0.74 1.2982 0.9809 3000862 BCB03_000133 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2C)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G17 compound treatment 176920.0 1090.0 0.07 181080.0 5690.0 0.42 0.3521 0.819 2065840 BCB03_000134 CCOC(=O)CC(CC(=O)OCC)(C(=O)OCC)c1cccnc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G18 compound treatment 182520.0 6690.0 0.46 184400.0 9010.0 0.67 0.7968 0.9824 3000863 BCB03_000135 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)C[Si](C)(C)C)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G19 mock treatment 180720.0 4890.0 0.33 175640.0 248.0 0.02 0.249 0.7451 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G20 mock treatment 177600.0 1770.0 0.12 180960.0 5570.0 0.41 0.3785 0.8769 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G21 compound treatment 178120.0 2290.0 0.16 171880.0 -3510.0 -0.26 -0.0743 -0.2438 2065855 BCB03_000136 CCOC(=O)CC(C(=O)OCC)c1cccnc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G22 compound treatment 181160.0 5330.0 0.36 182920.0 7530.0 0.56 0.6533 0.9781 3092589 BCB03_000137 CCOC(=O)C1=CC[C@H](N([C@H]1/C=C/c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G23 compound treatment 209200.0 33400.0 2.28 207920.0 32500.0 2.42 3.3208 0.9995 2065872 BCB03_000138 CCOC(=O)/C(=C/1\NSc2ccccc12)/C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 G24 compound treatment 174280.0 -1550.0 -0.11 178320.0 2930.0 0.22 0.0795 0.3286 3092590 BCB03_000139 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)c4cccc(Cl)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H01 compound treatment 177920.0 2090.0 0.14 173520.0 -1870.0 -0.14 0.0024 0.0121 3092687 BCB03_000140 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3cccc(Cl)c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H02 compound treatment 194520.0 18700.0 1.27 189520.0 14100.0 1.05 1.6447 0.9954 3187850 BCB03_000141 OCCCC1=CC(C2CC2)N(Cc3cccc(OC(F)(F)F)c3)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H03 mock treatment 174280.0 -1550.0 -0.11 185840.0 10400.0 0.78 0.4753 0.6057 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H04 mock treatment 177200.0 1370.0 0.09 180040.0 4650.0 0.35 0.3108 0.8673 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H05 compound treatment 180960.0 5130.0 0.35 181680.0 6290.0 0.47 0.5784 0.9898 3092697 BCB03_000142 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H06 compound treatment 186840.0 11000.0 0.75 186760.0 11400.0 0.85 1.1292 0.9982 3187852 BCB03_000143 CN1C(C2C3C(C1C=C2CCCO)C(=O)N(C(=O)N)C3=O)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H07 compound treatment 189640.0 13800.0 0.94 193360.0 18000.0 1.34 1.6115 0.9853 3092698 BCB03_000144 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccco3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H08 compound treatment 180040.0 4210.0 0.29 178600.0 3210.0 0.24 0.372 0.9958 3187853 BCB03_000145 CC1C2C3C(C(C=C2CCCO)N1Cc4cccc(OC(F)(F)F)c4)C(=O)N(C(=O)N)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H09 compound treatment 179560.0 3730.0 0.25 182680.0 7290.0 0.54 0.5635 0.9405 3092699 BCB03_000146 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3cccc4ccccc34)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H10 compound treatment 198560.0 22700.0 1.55 195720.0 20300.0 1.51 2.1658 0.9999 3070552 BCB03_000147 OCCCC1=CC(C2CC2)N(Cc3sc4ccccc4c3Cl)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H11 compound treatment 185560.0 9730.0 0.66 180720.0 5330.0 0.4 0.7496 0.9697 3092700 BCB03_000148 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(Br)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H12 compound treatment 201400.0 25600.0 1.74 199080.0 23700.0 1.76 2.4795 1.0 3070553 BCB03_000149 CN1CCC(=CC1c2cccs2)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H13 compound treatment 193680.0 17900.0 1.22 182640.0 7250.0 0.54 1.2421 0.933 3000975 BCB03_000150 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(cc3)C(C)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H14 compound treatment 214240.0 38400.0 2.62 207200.0 31800.0 2.37 3.5258 0.9987 3187856 BCB03_000151 OCCCC1=CC(N(Cc2cccc(OC(F)(F)F)c2)CC1)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H15 compound treatment 183600.0 7770.0 0.53 187560.0 12200.0 0.91 1.0151 0.9674 3000976 BCB03_000152 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](C=C([C@@H]2c3ccccc3)C(=O)O)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H16 compound treatment 194480.0 18700.0 1.27 184520.0 9130.0 0.68 1.3796 0.9569 3187857 BCB03_000153 NC(=O)N1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5ccc(CN6CCCC6)cc5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H17 compound treatment 182960.0 7130.0 0.49 184000.0 8610.0 0.64 0.7969 0.9908 3092773 BCB03_000154 CC(C)[C@@H]1[C@@H](Sc2ccccc2)[C@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H18 compound treatment 249320.0 73500.0 5.01 248760.0 73400.0 5.46 7.4042 0.9991 3070555 BCB03_000155 OCc1ccc(cc1)C2=CC(C3CC3)N(Cc4cc5OCOc5cc4Br)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H19 mock treatment 177960.0 2130.0 0.15 177880.0 2490.0 0.19 0.2338 0.9929 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H20 mock treatment 174960.0 -866.0 -0.06 175280.0 -112.0 -0.01 -0.0477 -0.799 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H21 compound treatment 188120.0 12300.0 0.84 181640.0 6250.0 0.47 0.9215 0.9614 3092774 BCB03_000156 CC[C@@H]1C(Sc2ccccc2)C([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H22 compound treatment 227880.0 52100.0 3.55 228480.0 53100.0 3.95 5.3033 0.9986 3070556 BCB03_000157 NC(=O)N1C(=O)C2C(C3C(C4CC4)N(Cc5sc6ccccc6c5Cl)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H23 compound treatment 225000.0 49200.0 3.35 221480.0 46100.0 3.43 4.7961 0.9999 3092783 BCB03_000158 CCC[C@@H]1[C@@H](Sc2ccccc2)[C@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 H24 compound treatment 221640.0 45800.0 3.12 211400.0 36000.0 2.68 4.1036 0.9971 3070597 BCB03_000159 NC(=O)N1C(=O)C2C(C3C(C4CC4)N(Cc5cc6OCOc6cc5Br)C2C=C3c7ccc(CO)cc7)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I01 compound treatment 177920.0 2090.0 0.14 182240.0 6850.0 0.51 0.4613 0.8716 2065633 BCB03_000160 CCOC(=O)CC(C#N)(C(=O)OCC)c1nsc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I02 compound treatment 180600.0 4770.0 0.33 175000.0 -392.0 -0.03 0.2095 0.6411 3000865 BCB03_000161 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2I)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I03 compound treatment 177760.0 1930.0 0.13 178240.0 2850.0 0.21 0.2431 0.9739 2065650 BCB03_000162 [O-][N+](=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I04 compound treatment 184520.0 8690.0 0.59 184400.0 9010.0 0.67 0.8932 0.9981 3000866 BCB03_000163 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I05 mock treatment 182480.0 6650.0 0.45 179120.0 3730.0 0.28 0.517 0.9722 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I06 mock treatment 182160.0 6330.0 0.43 175920.0 528.0 0.04 0.3331 0.7683 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I07 compound treatment 187760.0 11900.0 0.81 183640.0 8250.0 0.61 1.0094 0.9904 1065064 BCB03_000164 [O-][N+](=O)c1ccc(CBr)c(I)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I08 compound treatment 183920.0 8090.0 0.55 180920.0 5530.0 0.41 0.6811 0.9895 3000867 BCB03_000165 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I09 compound treatment 183680.0 7850.0 0.54 179120.0 3730.0 0.28 0.5748 0.9532 2065874 BCB03_000166 COC(=O)C(C(=O)OC)c1ccc(cc1I)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I10 compound treatment 201840.0 26000.0 1.77 197360.0 22000.0 1.64 2.4102 0.9992 3092595 BCB03_000167 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(SC)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(OCc5ccccc5)c(OC)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I11 compound treatment 221680.0 45900.0 3.13 252600.0 77200.0 5.75 6.2738 0.9591 BCB03_000168 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I12 compound treatment 194040.0 18200.0 1.24 199080.0 23700.0 1.76 2.1247 0.9853 3000949 BCB03_000169 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(cc2)[N+](=O)[O-])S(=O)(=O)c3ccc(C)cc3)c4cccc(Br)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I13 compound treatment 207240.0 31400.0 2.14 194760.0 19400.0 1.44 2.5337 0.9814 3107360 BCB03_000170 Cc1ccc(cc1)S(=O)(=O)O.Cc1cc(=O)oc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I14 compound treatment 186240.0 10400.0 0.71 183240.0 7850.0 0.58 0.915 0.9953 3000951 BCB03_000171 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I15 compound treatment 191280.0 15500.0 1.05 189400.0 14000.0 1.04 1.4822 1.0 1952728 BCB03_000172 Cc1ccc2oc(=O)cc(c3cccs3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I16 compound treatment 183080.0 7250.0 0.49 181840.0 6450.0 0.48 0.689 0.9999 3000952 BCB03_000173 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3cccc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I17 compound treatment 177080.0 1250.0 0.09 179800.0 4410.0 0.33 0.2924 0.8625 1952730 BCB03_000174 O=c1cc(Cc2ccccc2)c3ccccc3o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I18 compound treatment 182920.0 7090.0 0.48 180360.0 4970.0 0.37 0.6034 0.9912 3092606 BCB03_000175 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(F)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I19 compound treatment 183600.0 7770.0 0.53 185960.0 10600.0 0.79 0.9309 0.9815 1952746 BCB03_000176 Cc1ccc(cc1)c2cc(=O)oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I20 compound treatment 181320.0 5490.0 0.37 180960.0 5570.0 0.41 0.5579 0.9987 3092607 BCB03_000177 CCOC(=O)[C@@H]1N([C@@H](CC=C1C(=O)OCC)c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I21 mock treatment 173960.0 -1870.0 -0.13 169360.0 -6030.0 -0.45 -0.4074 -0.8731 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I22 mock treatment 176400.0 574.0 0.04 171760.0 -3630.0 -0.27 -0.1635 -0.5986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I23 compound treatment 176280.0 454.0 0.03 174480.0 -912.0 -0.07 -0.0261 -0.3504 3005760 BCB03_000178 CCOP(=O)(O)OCC.Cc1cc(=O)oc2ccc(Cl)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 I24 compound treatment 170160.0 -5670.0 -0.39 167000.0 -8390.0 -0.62 -0.7148 -0.9733 3000954 BCB03_000179 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(OC)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J01 compound treatment 175920.0 93.5 0.01 172360.0 -3030.0 -0.23 -0.1551 -0.6868 3092784 BCB03_000180 CCS[C@@H]1[C@@H](CC)N([C@H]([C@@H]1C(=O)O)c2ccc(C)cc2)S(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J02 compound treatment 250320.0 74500.0 5.08 247520.0 72100.0 5.37 7.3871 0.9996 3187985 BCB03_000181 NC(=O)N1C(=O)C2C(C3C(N(Cc4cc5OCOc5cc4Br)C2C=C3CCCO)c6cccs6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J03 compound treatment 182560.0 6730.0 0.46 177960.0 2570.0 0.19 0.4598 0.9246 3092785 BCB03_000182 CCOC1=C2C(N(CC2C3C(C1)C(=O)N(C3=O)c4ccccc4)S(=O)(=O)c5ccc(C)cc5)c6ccc(C)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J04 compound treatment 202160.0 26300.0 1.8 203680.0 28300.0 2.11 2.7582 0.9969 3187986 BCB03_000183 CN1CCC(=CC1c2ccc(CN3CCCC3)cc2)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J05 mock treatment 185600.0 9770.0 0.67 179920.0 4530.0 0.34 0.7095 0.9501 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J06 mock treatment 183440.0 7610.0 0.52 185680.0 10300.0 0.77 0.9085 0.9821 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J07 compound treatment 194720.0 18900.0 1.29 187760.0 12400.0 0.92 1.5617 0.9864 3001173 BCB03_000184 CCOC1=C2C(N(CC2n3n(C1)c(=O)n(c4ccccc4)c3=O)S(=O)(=O)c5ccc(C)cc5)c6ccc(C)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J08 compound treatment 180920.0 5090.0 0.35 183320.0 7930.0 0.59 0.6628 0.9681 3070607 BCB03_000185 OCCCC1=CC(N(Cc2cccc(OC(F)(F)F)c2)CC1)c3ccc(CN4CCCC4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J09 compound treatment 194360.0 18500.0 1.26 198520.0 23100.0 1.72 2.1106 0.9884 3001174 BCB03_000186 Cc1ccc(cc1)C2C3C(CN2S(=O)(=O)c4ccc(C)cc4)C5C(CC3=O)C(=O)N(C5=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J10 compound treatment 246000.0 70200.0 4.78 245480.0 70100.0 5.22 7.0715 0.9991 3070608 BCB03_000187 OCCCC1=CC(N(Cc2cc3OCOc3cc2Br)CC1)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J11 compound treatment 186520.0 10700.0 0.73 184200.0 8810.0 0.66 0.9791 0.9986 3092789 BCB03_000188 CCN1C(=O)C2CC(=O)C3C(N(CC3C2C1=O)S(=O)(=O)c4ccc(C)cc4)c5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J12 compound treatment 205560.0 29700.0 2.03 203640.0 28200.0 2.1 2.92 0.9998 3070609 BCB03_000189 CN1CCC(=CC1C2CC2)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J13 compound treatment 186320.0 10500.0 0.72 186840.0 11400.0 0.85 1.1084 0.9962 3092790 BCB03_000190 CC[C@@H]1[C@@H]2[C@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)CC5C2C(=O)N(CC)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J14 compound treatment 218960.0 43100.0 2.94 222280.0 46900.0 3.49 4.547 0.9964 3187991 BCB03_000191 NC(=O)N1C(=O)C2C(C3C(C4CC4)N(Cc5cc6OCOc6cc5Br)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J15 compound treatment 183000.0 7170.0 0.49 183440.0 8050.0 0.6 0.7694 0.9949 3092866 BCB03_000192 CC[C@@H]1[C@H]2[C@@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)CC5C2C(=O)N(CC)C5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J16 compound treatment 194160.0 18300.0 1.25 190640.0 15200.0 1.13 1.6863 0.9988 3187992 BCB03_000193 NC(=O)N1C(=O)C2C(C3C(C4CC4)N(Cc5cccc(OC(F)(F)F)c5)C2C=C3CCCO)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J17 compound treatment 179000.0 3170.0 0.22 177760.0 2370.0 0.18 0.2776 0.9948 3092867 BCB03_000194 CCOC(=O)C1=CC[C@H](N([C@H]1CC)S(=O)(=O)c2ccc(C)cc2)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J18 compound treatment 184200.0 8370.0 0.57 182760.0 7370.0 0.55 0.7914 0.9998 3187993 BCB03_000195 CN1C(C2CC2)C3C4C(C1C=C3CCCO)C(=O)N(C(=O)N)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J19 compound treatment 181040.0 5210.0 0.36 179680.0 4290.0 0.32 0.477 0.9986 3092868 BCB03_000196 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J20 compound treatment 201920.0 26100.0 1.78 175800.0 408.0 0.03 1.2794 0.7191 3187994 BCB03_000197 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J21 mock treatment 174040.0 -1790.0 -0.12 173160.0 -2230.0 -0.17 -0.2036 -0.9884 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J22 mock treatment 169560.0 -6270.0 -0.43 166520.0 -8870.0 -0.66 -0.769 -0.9778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J23 compound treatment 180800.0 4970.0 0.34 176240.0 848.0 0.06 0.2844 0.8246 3092869 BCB03_000198 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 J24 compound treatment 187320.0 11500.0 0.78 177960.0 2570.0 0.19 0.6892 0.8545 3070656 BCB03_000199 CN1C=C(C(=O)OCCS(=O)(=O)C)C(=CC(=CC1c2cccs2)CCCO)C(=O)OCCS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K01 compound treatment 174120.0 -1710.0 -0.12 178240.0 2850.0 0.21 0.0676 0.2796 3005761 BCB03_000200 Cc1ccc(cc1)S(=O)(=O)O.Cc1cc(=O)oc2ccc(Cl)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K02 compound treatment 184320.0 8490.0 0.58 181320.0 5930.0 0.44 0.7214 0.991 3000955 BCB03_000201 CCOC(=O)C1=CC[C@H](N([C@H]1C)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K03 compound treatment 182440.0 6610.0 0.45 180840.0 5450.0 0.41 0.6055 0.9986 1952748 BCB03_000202 O=Cc1cccc(c1)c2cc(=O)oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K04 compound treatment 188840.0 13000.0 0.89 188880.0 13500.0 1.0 1.3372 0.9981 3092688 BCB03_000203 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccncc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K05 compound treatment 177600.0 1770.0 0.12 177280.0 1890.0 0.14 0.1849 0.9972 1107217 BCB03_000204 Cc1cccnc1I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K06 compound treatment 184640.0 8810.0 0.6 186000.0 10600.0 0.79 0.9832 0.9909 3000965 BCB03_000205 CCOC(=O)C1=CC[C@H](N([C@H]1C=C(C)C)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K07 mock treatment 187600.0 11800.0 0.8 179520.0 4130.0 0.31 0.7848 0.9132 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K08 mock treatment 181760.0 5930.0 0.4 179520.0 4130.0 0.31 0.5033 0.9908 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K09 compound treatment 188400.0 12600.0 0.86 181400.0 6010.0 0.45 0.9223 0.954 3005761 BCB03_000206 Cc1ccc(cc1)S(=O)(=O)O.Cc1cc(=O)oc2ccc(Cl)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K10 compound treatment 199680.0 23900.0 1.63 193520.0 18100.0 1.35 2.104 0.9957 3000966 BCB03_000207 CCOC(=O)C1=CC[C@H](N([C@H]1C#N)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K11 compound treatment 210120.0 34300.0 2.34 213640.0 38200.0 2.85 3.6661 0.9952 1952755 BCB03_000208 C=C(c1ccccc1)c2cc(=O)oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K12 compound treatment 187240.0 11400.0 0.78 184080.0 8690.0 0.65 1.0075 0.9958 3092692 BCB03_000209 CCOC(=O)C1=CC[C@H](N([C@H]1c2cccc(OC)c2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K13 compound treatment 180320.0 4490.0 0.31 177880.0 2490.0 0.19 0.3476 0.9709 1952760 BCB03_000210 CC(C)(C)[Si](C)(C)OCCNC(=O)c1cc(c2cc(F)cc(F)c2)c3oc4c(C(=O)OC4(c5ccccc5)c6ccccc6)c3c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K14 compound treatment 183600.0 7770.0 0.53 177880.0 2490.0 0.19 0.5057 0.9008 3092693 BCB03_000211 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K15 mock treatment 183760.0 7930.0 0.54 181240.0 5850.0 0.44 0.6902 0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K16 mock treatment 179640.0 3810.0 0.26 174360.0 -1030.0 -0.08 0.1295 0.4778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K17 compound treatment 174000.0 -1830.0 -0.12 178880.0 3490.0 0.26 0.0955 0.3317 1952770 BCB03_000212 O=C/1Oc2ccccc2C\C1=C(/c3ccccc3)\c4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K18 compound treatment 179240.0 3410.0 0.23 182000.0 6610.0 0.49 0.5123 0.9416 3000969 BCB03_000213 CCOC(=O)C1=CC[C@H](N([C@H]1C=C)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K19 compound treatment 192000.0 16200.0 1.1 188840.0 13400.0 1.0 1.4874 0.9988 3000871 BCB03_000214 O=c1cccc(o1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K20 compound treatment 191040.0 15200.0 1.04 191040.0 15600.0 1.16 1.5569 0.9983 3001047 BCB03_000215 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(c(OC)c4)c5ccc(OCc6ccccc6)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K21 compound treatment 192760.0 16900.0 1.15 189760.0 14400.0 1.07 1.5725 0.9993 3000872 BCB03_000216 COc1cccc(c1)c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K22 compound treatment 182560.0 6730.0 0.46 177520.0 2130.0 0.16 0.4366 0.8991 3001048 BCB03_000217 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K23 mock treatment 177200.0 1370.0 0.09 175680.0 288.0 0.02 0.0814 0.8471 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 K24 mock treatment 174400.0 -1430.0 -0.1 166040.0 -9350.0 -0.7 -0.5609 -0.7982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L01 compound treatment 176520.0 694.0 0.05 178240.0 2850.0 0.21 0.1833 0.8441 3092870 BCB03_000218 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L02 compound treatment 268560.0 92700.0 6.32 264640.0 89200.0 6.64 9.1675 0.9997 3188115 BCB03_000219 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L03 compound treatment 179600.0 3770.0 0.26 181920.0 6530.0 0.49 0.5255 0.9558 3092871 BCB03_000220 CCOC(=O)C1=CC[C@H](N([C@H]1c2cccc(Br)c2)S(=O)(=O)c3ccc(C)cc3)c4ccc(OCC=C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L04 compound treatment 194880.0 19100.0 1.3 191680.0 16300.0 1.21 1.7757 0.9994 3188116 BCB03_000221 CC1C=C(CCCO)C=C(C(=O)OCCS(=O)(=O)C)C(=CN1Cc2cccc(OC(F)(F)F)c2)C(=O)OCCS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L05 compound treatment 190240.0 14400.0 0.98 183440.0 8050.0 0.6 1.1184 0.9718 3092774 BCB03_000222 CC[C@@H]1C(Sc2ccccc2)C([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L06 compound treatment 229360.0 53500.0 3.65 225680.0 50300.0 3.74 5.2273 0.9999 3188117 BCB03_000223 CS(=O)(=O)CCOC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L07 mock treatment 181320.0 5490.0 0.37 179160.0 3770.0 0.28 0.4631 0.9898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L08 mock treatment 175760.0 -66.5 0.0 181920.0 6530.0 0.49 0.3404 0.7005 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L09 compound treatment 193840.0 18000.0 1.23 182080.0 6690.0 0.5 1.2204 0.9209 3187870 BCB03_000224 COC(=O)C[C@H]1O[C@@H](CCc2ccccc2)[C@@H](C)[C@@H]1[Si](C)(C)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L10 compound treatment 236800.0 61000.0 4.16 221600.0 46200.0 3.44 5.3713 0.9956 3188119 BCB03_000225 CS(=O)(=O)CCOC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L11 compound treatment 190840.0 15000.0 1.02 192640.0 17200.0 1.28 1.6315 0.9937 3071511 BCB03_000226 COC(=O)C[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)c3ccc(OC)cc3)C(=O)N(Cc4ccccc4)c5ccc(I)cc52 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L12 compound treatment 222080.0 46300.0 3.15 216320.0 40900.0 3.05 4.3838 0.9999 3188120 BCB03_000227 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L13 compound treatment 181120.0 5290.0 0.36 183720.0 8330.0 0.62 0.6935 0.9669 3187872 BCB03_000228 COC(=O)C[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)c3ccc(OC)cc3)C(=O)N(Cc4ccccc4)c5ccc(NC(=O)C)cc52 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L14 compound treatment 239600.0 63800.0 4.35 236880.0 61500.0 4.58 6.3104 0.9997 3188122 BCB03_000229 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(C=C1C(=O)OCCS(=O)(=O)C)c3ccc(CO)cc3)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L15 mock treatment 184240.0 8410.0 0.57 176360.0 968.0 0.07 0.4565 0.7897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L16 mock treatment 176840.0 1010.0 0.07 175640.0 248.0 0.02 0.0619 0.8656 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L17 compound treatment 190280.0 14500.0 0.99 189360.0 14000.0 1.04 1.4319 0.9996 3414061 BCB03_000230 COC(=O)C[C@@H]1C[C@H](C)[C@]2(O1)C(=O)N(Cc3ccccc3)c4ccc(NC(=O)C)cc42 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L18 compound treatment 228120.0 52300.0 3.57 216920.0 41500.0 3.09 4.7065 0.9975 3188123 BCB03_000231 CN1C=C(C(=O)OCCS(=O)(=O)C)C(=CC(=CC1c2cccs2)c3ccc(CO)cc3)C(=O)OCCS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L19 compound treatment 200200.0 24400.0 1.66 195920.0 20500.0 1.53 2.2554 0.9991 3071513 BCB03_000232 CC(C)[Si](OCC[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)O)C(=O)N(Cc3ccccc3)c4ccccc42)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L20 compound treatment 264120.0 88300.0 6.02 257200.0 81800.0 6.09 8.5619 1.0 3188124 BCB03_000233 CS(=O)(=O)CCOC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(C=C1C(=O)OCCS(=O)(=O)C)c4ccc(CO)cc4)C5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L21 compound treatment 201640.0 25800.0 1.76 194600.0 19200.0 1.43 2.2553 0.9947 3071514 BCB03_000234 COc1ccc(cc1)[Si](C)(C)[C@H]2[C@H](C)[C@]3(O[C@@H]2CCO)C(=O)N(Cc4ccccc4)c5ccccc53 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L22 compound treatment 218320.0 42500.0 2.9 215880.0 40500.0 3.01 4.1793 0.9998 3188125 BCB03_000235 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)c4ccc(CN5CCCC5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L23 mock treatment 168760.0 -7070.0 -0.48 168960.0 -6430.0 -0.48 -0.6792 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 L24 mock treatment 168560.0 -7270.0 -0.5 163800.0 -11600.0 -0.86 -0.9604 -0.9653 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M01 compound treatment 179400.0 3570.0 0.24 183920.0 8530.0 0.63 0.6211 0.9135 1984103 BCB03_000236 Cc1ccc(cc1)c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M02 compound treatment 187000.0 11200.0 0.76 190280.0 14900.0 1.11 1.3222 0.9833 3001049 BCB03_000237 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M03 compound treatment 186600.0 10800.0 0.73 190200.0 14800.0 1.1 1.2987 0.9806 3000873 BCB03_000238 Clc1cccc(c1)c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M04 compound treatment 185160.0 9330.0 0.64 189600.0 14200.0 1.06 1.1977 0.9705 3092778 BCB03_000239 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(CC)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M05 compound treatment 185120.0 9290.0 0.63 182600.0 7210.0 0.54 0.8274 0.9966 3000875 BCB03_000240 Clc1ccccc1c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M06 compound treatment 209080.0 33300.0 2.27 203560.0 28200.0 2.1 3.0855 0.9992 3001168 BCB03_000241 CCOC(=O)C1=C(N([C@@H](CC1)c2ccccc2)S(=O)(=O)CC[Si](C)(C)C)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M07 compound treatment 187920.0 12100.0 0.82 190600.0 15200.0 1.13 1.3834 0.9879 3000956 BCB03_000242 CCCc1cccc(=O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M08 compound treatment 190440.0 14600.0 1.0 196240.0 20800.0 1.55 1.8017 0.9771 3092780 BCB03_000243 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(OC)cc2)S(=O)(=O)c3ccc(C)cc3)c4cc(Cl)ccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M09 mock treatment 179640.0 3810.0 0.26 184080.0 8690.0 0.65 0.6411 0.9199 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M10 mock treatment 185440.0 9610.0 0.66 188080.0 12700.0 0.94 1.1312 0.9841 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M11 compound treatment 184760.0 8930.0 0.61 183920.0 8530.0 0.63 0.8795 0.9998 3000957 BCB03_000244 Fc1ccc(cc1)c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M12 compound treatment 183720.0 7890.0 0.54 191200.0 15800.0 1.18 1.2125 0.9372 3092781 BCB03_000245 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M13 mock treatment 187640.0 11800.0 0.81 183880.0 8490.0 0.63 1.0162 0.9928 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M14 mock treatment 180520.0 4690.0 0.32 182840.0 7450.0 0.55 0.6182 0.9659 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M15 compound treatment 188600.0 12800.0 0.87 188120.0 12700.0 0.95 1.2856 0.9991 3000958 BCB03_000246 O=c1cccc(o1)c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M16 compound treatment 208640.0 32800.0 2.24 213880.0 38500.0 2.86 3.6074 0.9925 3001177 BCB03_000247 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccco3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M17 compound treatment 181960.0 6130.0 0.42 185400.0 10000.0 0.74 0.8224 0.9627 3092682 BCB03_000248 FC(F)(F)c1ccc(cc1)c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M18 compound treatment 193320.0 17500.0 1.19 194960.0 19600.0 1.46 1.8732 0.9951 3001178 BCB03_000249 CCOC(=O)C1=CC[C@H](N([C@@H]1C#N)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M19 compound treatment 183480.0 7650.0 0.52 190320.0 14900.0 1.11 1.1546 0.9406 3000960 BCB03_000250 FC(F)(F)c1ccccc1c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M20 compound treatment 186160.0 10300.0 0.7 186880.0 11500.0 0.86 1.1028 0.9954 3001179 BCB03_000251 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)CC[Si](C)(C)C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M21 compound treatment 195440.0 19600.0 1.34 197880.0 22500.0 1.67 2.129 0.9938 3000961 BCB03_000252 O=c1cccc(o1)c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M22 compound treatment 215400.0 39600.0 2.7 201400.0 26000.0 1.94 3.2765 0.9867 3001245 BCB03_000253 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3cccn3C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M23 compound treatment 178840.0 3010.0 0.21 179800.0 4410.0 0.33 0.3773 0.9746 3092685 BCB03_000254 O=c1cccc(o1)c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 M24 compound treatment 188000.0 12200.0 0.83 184320.0 8930.0 0.66 1.0567 0.9939 3001246 BCB03_000255 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N01 compound treatment 198680.0 22900.0 1.56 193800.0 18400.0 1.37 2.0705 0.9979 3071515 BCB03_000256 COC(=O)C[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)c3ccc(C)cc3)C(=O)N(C)c4ccccc42 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N02 compound treatment 185560.0 9730.0 0.66 183440.0 8050.0 0.6 0.8928 0.9987 3188247 BCB03_000257 CN1C=C(C(=O)OCCS(=O)(=O)C)C(=CC(=CC1C2CC2)CCCO)C(=O)OCCS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N03 compound treatment 195120.0 19300.0 1.32 197600.0 22200.0 1.65 2.0989 0.9936 3071516 BCB03_000258 COC(=O)C[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)c3ccc(OC)cc3)C(=O)N(C)c4ccccc42 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N04 compound treatment 229120.0 53300.0 3.63 225880.0 50500.0 3.76 5.2263 0.9999 3188248 BCB03_000259 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N05 compound treatment 187880.0 12100.0 0.82 194560.0 19200.0 1.43 1.5899 0.9657 3414062 BCB03_000260 COC(=O)C[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)c3ccccc3)C(=O)N(C)c4ccccc42 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N06 compound treatment 291440.0 116000.0 7.88 276120.0 101000.0 7.5 10.8746 0.9997 3188250 BCB03_000261 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(C=C1C(=O)OCCS(=O)(=O)C)c4ccc(CO)cc4)C5CC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N07 compound treatment 182280.0 6450.0 0.44 185560.0 10200.0 0.76 0.8462 0.9667 3188927 BCB03_000262 COC(=O)C[C@H]1O[C@@]2([C@@H](C)[C@@H]1[Si](C)(C)F)C(=O)N(C)c3ccccc32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N08 compound treatment 189680.0 13900.0 0.94 190800.0 15400.0 1.15 1.4787 0.9954 3188251 BCB03_000263 CS(=O)(=O)CCOC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OCCS(=O)(=O)C)c3ccc(CN4CCCC4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N09 mock treatment 183480.0 7650.0 0.52 183160.0 7770.0 0.58 0.7778 0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N10 mock treatment 183920.0 8090.0 0.55 182160.0 6770.0 0.5 0.7464 0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N11 compound treatment 185640.0 9810.0 0.67 184800.0 9410.0 0.7 0.9682 0.9997 3071435 BCB03_000264 COC(=O)C[C@H]1O[C@@]2(C[C@@H]1[Si](C)(C)C)C(=O)N(C)c3ccccc32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N12 compound treatment 200920.0 25100.0 1.71 208160.0 32800.0 2.44 2.9342 0.985 3188252 BCB03_000265 CN1C=C(C(=O)OCCS(=O)(=O)C)C(=CC(=CC1C2CC2)c3ccc(CO)cc3)C(=O)OCCS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N13 mock treatment 181760.0 5930.0 0.4 181960.0 6570.0 0.49 0.6317 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N14 mock treatment 185120.0 9290.0 0.63 184520.0 9130.0 0.68 0.9284 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N15 compound treatment 182440.0 6610.0 0.45 177200.0 1810.0 0.13 0.414 0.8798 3188929 BCB03_000266 COC(=O)C/C=C/C[C@]1(O)C(=O)N(C)c2ccccc21 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N16 compound treatment 218880.0 43100.0 2.94 203240.0 27800.0 2.07 3.5411 0.9855 3188253 BCB03_000267 COP(=O)(OC)/N=C\1/CC(=CC(N1C)c2cccs2)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N17 compound treatment 193240.0 17400.0 1.19 191880.0 16500.0 1.23 1.7072 0.9999 3188930 BCB03_000268 COc1ccc(cc1)[Si](C)(C)[C@H](CCn2cc(CCO[Si](C(C)C)(C(C)C)C(C)C)nn2)/C=C/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N18 compound treatment 186520.0 10700.0 0.73 183120.0 7730.0 0.58 0.9222 0.9931 3188254 BCB03_000269 CN1C=C(C(=O)OCCS(=O)(=O)C)C(=CC(=CC1c2ccc(CN3CCCC3)cc2)CCCO)C(=O)OCCS(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N19 compound treatment 188200.0 12400.0 0.84 184600.0 9210.0 0.69 1.0811 0.9947 3071465 BCB03_000270 CCCCNC(=O)c1ccc(C#CC(C)(C)C)c(OC(=O)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N20 compound treatment 226760.0 50900.0 3.47 223680.0 48300.0 3.59 4.9967 0.9999 3188255 BCB03_000271 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1Cc3sc4ccccc4c3Cl)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N21 compound treatment 184800.0 8970.0 0.61 175760.0 368.0 0.03 0.452 0.738 1952196 BCB03_000272 CCCCNC(=O)c1ccc(C#C[Si](C)(C)C)c(OC(=O)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N22 compound treatment 182160.0 6330.0 0.43 176280.0 888.0 0.07 0.3521 0.806 3188256 BCB03_000273 COP(=O)(OC)/N=C\1/CC(=CC(N1Cc2sc3ccccc3c2Cl)c4ccc(CN5CCCC5)cc4)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N23 compound treatment 181840.0 6010.0 0.41 180560.0 5170.0 0.38 0.5619 0.9995 3071510 BCB03_000274 CCCCNC(=O)c1ccc(C#C[Si](C(C)C)(C(C)C)C(C)C)c(OC(=O)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 N24 compound treatment 181600.0 5770.0 0.39 179080.0 3690.0 0.27 0.4724 0.9845 3188257 BCB03_000275 COP(=O)(OC)/N=C\1/CC(=CC(N1C)c2cccs2)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O01 compound treatment 219600.0 43800.0 2.98 212680.0 37300.0 2.78 4.0726 0.9993 3000963 BCB03_000276 O=c1cccc(CCc2ccccc2)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O02 compound treatment 182800.0 6970.0 0.48 186440.0 11000.0 0.82 0.9176 0.9661 3001247 BCB03_000277 CCOC(=O)C1=CCC(NC1)c2cc3ccccc3[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O03 compound treatment 184680.0 8850.0 0.6 186920.0 11500.0 0.86 1.0335 0.9852 3000971 BCB03_000278 [O-][N+](=O)c1ccc(cc1)c2cccc(=O)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O04 compound treatment 183760.0 7930.0 0.54 186600.0 11200.0 0.83 0.9723 0.978 3001248 BCB03_000279 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccccc2[N+](=O)[O-])c3cc4ccccc4[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O05 compound treatment 174200.0 -1630.0 -0.11 180640.0 5250.0 0.39 0.1978 0.4871 3000972 BCB03_000280 O=c1cccc(/C=C/c2ccccc2)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O06 compound treatment 181760.0 5930.0 0.4 184600.0 9210.0 0.69 0.7706 0.9684 3000756 BCB03_000281 CCOC(=O)C1=CCC(N(CCN2CC(=CCC2c3cc4ccccc4[nH]3)C(=O)OCC)C1)c5cc6ccccc6[nH]5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O07 compound treatment 194080.0 18300.0 1.24 196360.0 21000.0 1.56 1.9835 0.9937 3000973 BCB03_000282 O=c1cccc(o1)c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O08 compound treatment 183800.0 7970.0 0.54 181520.0 6130.0 0.46 0.7069 0.9962 3000757 BCB03_000283 CC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O09 compound treatment 180720.0 4890.0 0.33 178840.0 3450.0 0.26 0.4174 0.9916 3000974 BCB03_000284 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(Cl)c2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O10 compound treatment 217400.0 41600.0 2.83 214880.0 39500.0 2.94 4.0824 0.9998 3093828 BCB03_000285 Cc1ccc(cc1)[C@@H]2C[C@@H](Sc3ccccc3)[C@@H](CN2S(=O)(=O)c4ccc(C)cc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O11 mock treatment 175080.0 -746.0 -0.05 172880.0 -2510.0 -0.19 -0.1682 -0.868 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O12 mock treatment 181840.0 6010.0 0.41 183320.0 7930.0 0.59 0.7071 0.9842 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O13 compound treatment 190520.0 14700.0 1.0 185640.0 10200.0 0.76 1.2477 0.9909 3092701 BCB03_000286 CCOC(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(c2)[N+](=O)[O-])c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O14 compound treatment 178800.0 2970.0 0.2 175040.0 -352.0 -0.03 0.1248 0.6106 3093829 BCB03_000287 Cc1ccc(cc1)C2CC=C(CN2S(=O)(=O)c3ccc(C)cc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O15 compound treatment 185000.0 9170.0 0.63 182480.0 7090.0 0.53 0.8153 0.9964 3092771 BCB03_000288 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccccn2)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O16 compound treatment 182360.0 6530.0 0.45 179080.0 3690.0 0.27 0.5091 0.9729 3093830 BCB03_000289 Cc1ccc(cc1)S(=O)(=O)N2CC(=CCC2c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O17 compound treatment 176200.0 374.0 0.03 176720.0 1330.0 0.1 0.0879 0.8612 3092772 BCB03_000290 COC(=O)c1cccc(c1)[C@@H]2C/C(=C\C(=O)OC(C)C)/O[C@@H](O2)c3cccc(c3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O18 compound treatment 185000.0 9170.0 0.63 188120.0 12700.0 0.95 1.1121 0.9797 3000760 BCB03_000291 Cc1ccc(cc1)[C@@H]2CC=C([C@@H](N2S(=O)(=O)c3ccc(C)cc3)c4ccccc4)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O19 compound treatment 192200.0 16400.0 1.12 192960.0 17600.0 1.31 1.7139 0.9969 3000977 BCB03_000292 CC(C)OC(=O)/C=C\1/C[C@H](O[C@H](O1)c2ccc(C#N)cc2)c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O20 compound treatment 180520.0 4690.0 0.32 180480.0 5090.0 0.38 0.494 0.9965 3093833 BCB03_000293 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](CC=C([C@@H]2c3ccccc3)C(=O)O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O21 compound treatment 185040.0 9210.0 0.63 177440.0 2050.0 0.15 0.552 0.8539 3092782 BCB03_000294 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccc(cc2)C(F)(F)F)c3ccc(cc3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O22 compound treatment 172800.0 -3030.0 -0.21 169160.0 -6230.0 -0.46 -0.4739 -0.9335 3093834 BCB03_000295 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](CC=C([C@@H]2c3ccccc3)C(=O)O)c4ccc(C#N)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O23 compound treatment 166440.0 -9390.0 -0.64 165600.0 -9790.0 -0.73 -0.9678 -0.9979 3092786 BCB03_000296 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(c2)C(F)(F)F)c3cccc(c3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 O24 compound treatment 171160.0 -4670.0 -0.32 167600.0 -7790.0 -0.58 -0.635 -0.96 3093844 BCB03_000297 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](CC=C([C@@H]2c3ccccc3)C(=O)O)c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P01 compound treatment 210480.0 34700.0 2.36 209800.0 34400.0 2.56 3.4814 0.9992 3071725 BCB03_000298 COC(=O)[C@H](Cc1ccc(O)cc1)N[C@@H](/C=C/C2CC2)[C@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P02 compound treatment 192080.0 16300.0 1.11 193440.0 18000.0 1.34 1.7334 0.9954 3188381 BCB03_000299 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1C)c3ccc(CO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P03 compound treatment 199600.0 23800.0 1.62 201600.0 26200.0 1.95 2.5254 0.9958 3188399 BCB03_000300 COC(=O)[C@H](Cc1ccc(O)cc1)N(CC#C)[C@@H](/C=C/C2CC2)[C@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P04 compound treatment 217040.0 41200.0 2.81 220440.0 45000.0 3.35 4.3576 0.9961 3070118 BCB03_000301 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1Cc3cc4OCOc4cc3Br)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P05 compound treatment 190800.0 15000.0 1.02 198200.0 22800.0 1.7 1.9222 0.9704 3188400 BCB03_000302 COC(=O)[C@H](Cc1ccc(OCC#C)cc1)N(CC#C)[C@@H](/C=C/C2CC2)[C@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P06 compound treatment 182920.0 7090.0 0.48 184360.0 8970.0 0.67 0.8139 0.9875 3070119 BCB03_000303 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1Cc3cccc(OC(F)(F)F)c3)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P07 compound treatment 202880.0 27100.0 1.84 194160.0 18800.0 1.4 2.2919 0.9906 3188401 BCB03_000304 Oc1ccc(C[C@@H]2N(CC#C)[C@@H](/C=C/C3CC3)[C@@H](Cc4ccccc4)OC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P08 compound treatment 180160.0 4330.0 0.3 182200.0 6810.0 0.51 0.5672 0.967 3188385 BCB03_000305 COP(=O)(OC)/N=C\1/CC(=CC(N1Cc2cccc(OC(F)(F)F)c2)c3ccc(CN4CCCC4)cc3)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P09 compound treatment 189760.0 13900.0 0.95 191200.0 15800.0 1.18 1.5037 0.9944 3188402 BCB03_000306 O=C1O[C@H](Cc2ccccc2)[C@H](/C=C/C3CC3)N(CC#C)[C@H]1Cc4ccc(OCC#C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P10 compound treatment 232600.0 56800.0 3.87 224840.0 49400.0 3.68 5.3393 0.9997 3188386 BCB03_000307 NC(=O)N1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3c5ccc(CO)cc5)c6cccs6)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P11 mock treatment 171080.0 -4750.0 -0.32 177760.0 2370.0 0.18 -0.1042 -0.2828 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P12 mock treatment 177200.0 1370.0 0.09 176320.0 928.0 0.07 0.1151 0.9888 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P13 compound treatment 219840.0 44000.0 3.0 218400.0 43000.0 3.2 4.3852 0.9995 3070937 BCB03_000308 COC(=O)[C@H](Cc1ccc(O)cc1)N2CC3=CCCC=C[C@@H]3[C@H]2[C@H](O)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P14 compound treatment 182360.0 6530.0 0.45 180800.0 5410.0 0.4 0.5996 0.9987 3188387 BCB03_000309 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1C)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P15 compound treatment 221280.0 45500.0 3.1 224320.0 48900.0 3.64 4.7662 0.9968 3188528 BCB03_000310 Oc1ccc(C[C@@H]2N3CC4=CCCC=C[C@@H]4[C@H]3[C@@H](Cc5ccccc5)OC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P16 compound treatment 180960.0 5130.0 0.35 184400.0 9010.0 0.67 0.7216 0.9541 3070122 BCB03_000311 COP(=O)(OC)/N=C\1/CC(=CC(N1C)c2ccc(CN3CCCC3)cc2)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P17 compound treatment 176080.0 254.0 0.02 178200.0 2810.0 0.21 0.16 0.763 3188529 BCB03_000312 COC(=O)[C@H](Cc1ccccc1)N[C@@H](/C=C/C2CC2)[C@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P18 compound treatment 236600.0 60800.0 4.14 240440.0 65000.0 4.84 6.3531 0.997 3188390 BCB03_000313 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1Cc3cc4OCOc4cc3Br)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P19 compound treatment 195160.0 19300.0 1.32 193960.0 18600.0 1.38 1.9092 0.9997 3188530 BCB03_000314 COC(=O)[C@H](Cc1ccccc1)N(CC#C)[C@@H](/C=C/C2CC2)[C@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P20 compound treatment 170560.0 -5270.0 -0.36 175200.0 -192.0 -0.01 -0.264 -0.7347 3188503 BCB03_000315 COP(=O)(OC)/N=C\1/CC(=CC(C)N1Cc2cccc(OC(F)(F)F)c2)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P21 compound treatment 197640.0 21800.0 1.49 194600.0 19200.0 1.43 2.0625 0.9998 3070940 BCB03_000316 COC(=O)[C@H](Cc1ccccc1)N2CC(=C[C@H]2[C@H](O)Cc3ccccc3)/C=C/C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P22 compound treatment 186080.0 10300.0 0.7 180840.0 5450.0 0.41 0.781 0.9664 3070124 BCB03_000317 COP(=O)(OC)/N=C\1/CC(=CC(N1Cc2cc3OCOc3cc2Br)c4ccc(CN5CCCC5)cc4)CCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P23 compound treatment 170680.0 -5150.0 -0.35 172920.0 -2470.0 -0.18 -0.3782 -0.9546 3188533 BCB03_000318 O=C1O[C@@H](Cc2ccccc2)[C@@H](/C=C/C3CC3)N(CC#C)[C@H]1Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2281 P24 compound treatment 206760.0 30900.0 2.11 221080.0 45700.0 3.4 3.8957 0.9736 3188506 BCB03_000319 COP(=O)(OC)/N=C\1/CC(=CC(C2CC2)N1Cc3sc4ccccc4c3Cl)c5ccc(CO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A01 compound treatment 181200.0 5320.0 0.36 180960.0 5990.0 0.45 0.572 0.9947 3188507 BCB03_000320 CCCCCCc1nc(cc2CO[Si](C(C)C)(C(C)C)c21)c3ccc(o3)c4ccc(Cl)c(Cl)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A02 compound treatment 164720.0 -11200.0 -0.76 168680.0 -6290.0 -0.47 -0.8688 -0.9727 3071186 BCB03_000321 COc1ccc(cc1)[C@H]2OC[C@@H]3CCC(=O)N23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A03 compound treatment 162640.0 -13200.0 -0.9 160600.0 -14400.0 -1.07 -1.3943 -0.9965 3070126 BCB03_000322 CCCCCCc1nc(cc2CO[Si](C(C)C)(C(C)C)c21)c3cc(C)c(OC)c(C)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A04 compound treatment 168080.0 -7800.0 -0.53 167400.0 -7570.0 -0.56 -0.7742 -0.9996 3071252 BCB03_000323 COc1cccc(C[C@H]2C[C@@H](CO)NC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A05 compound treatment 163360.0 -12500.0 -0.85 162960.0 -12000.0 -0.89 -1.2354 -0.9997 3070127 BCB03_000324 CCCCCCc1nc(cc2CO[Si](C(C)C)(C(C)C)c21)c3ccc(OC)nc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A06 compound treatment 177440.0 1560.0 0.11 162720.0 -12200.0 -0.91 -0.5692 -0.6203 3071181 BCB03_000325 COc1cccc(C[C@H]2C[C@@H](CO[Si](C(C)C)(C(C)C)C(C)C)N3C(=O)[C@]4(O[C@@]23[C@H]5[C@@H]4C(=O)N(C)C5=O)C(=O)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A07 compound treatment 171200.0 -4680.0 -0.32 169520.0 -5450.0 -0.41 -0.5122 -0.993 3070128 BCB03_000326 CCCCCCc1nc(Cc2cc(OC)c(OC)c(OC)c2)cc3CO[Si](C(C)C)(C(C)C)c31 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A08 compound treatment 176440.0 561.0 0.04 171720.0 -3250.0 -0.24 -0.1438 -0.5879 3189172 BCB03_000327 COc1cccc(C[C@H]2C[C@@H](CO[Si](C(C)C)(C(C)C)C(C)C)N3C(=O)[C@@]4(O[C@]23[C@@H]5[C@H]4C(=O)N(C)C5=O)C(=O)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A09 compound treatment 161840.0 -14000.0 -0.96 159120.0 -15800.0 -1.18 -1.5107 -0.9946 3070129 BCB03_000328 CCCCCCc1nc(cc2CO[Si](C(C)C)(C(C)C)c21)C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A10 compound treatment 160600.0 -15300.0 -1.04 163720.0 -11200.0 -0.84 -1.3284 -0.9941 3071185 BCB03_000329 COc1ccc(cc1)[C@H]2OC[C@@H]3CC4(CC=CC4)C(=O)N23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A11 compound treatment 186520.0 10600.0 0.73 192240.0 17300.0 1.29 1.4221 0.9633 3188514 BCB03_000330 CCCCCCc1nc(c2ccc(o2)c3ccc(Cl)c(Cl)c3)c(C)c4CO[Si](C(C)C)(C(C)C)c41 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A12 compound treatment 173520.0 -2360.0 -0.16 172320.0 -2650.0 -0.2 -0.253 -0.995 3189173 BCB03_000331 NC(=N)NCc1cn(CCc2c[nH]c3ccccc23)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A13 mock treatment 168840.0 -7040.0 -0.48 169160.0 -5810.0 -0.43 -0.6449 -0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A14 mock treatment 166520.0 -9360.0 -0.64 166800.0 -8170.0 -0.61 -0.8809 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A15 compound treatment 162640.0 -13200.0 -0.9 164400.0 -10600.0 -0.79 -1.1943 -0.9976 3070178 BCB03_000332 CCCCCCc1nc(c(C)c2CO[Si](C(C)C)(C(C)C)c21)c3cc(C)c(OC)c(C)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A16 compound treatment 166600.0 -9280.0 -0.63 163320.0 -11600.0 -0.87 -1.0602 -0.988 3071253 BCB03_000333 COC(=O)c1c(CC[C@@H](CO)NC(=O)N(C)Cc2ccccc2)oc(C(=O)OCC=C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A17 compound treatment 162520.0 -13400.0 -0.91 154920.0 -20000.0 -1.49 -1.699 -0.972 3070179 BCB03_000334 CCCCCCc1nc(c(C)c2CO[Si](C(C)C)(C(C)C)c21)c3ccc(OC)nc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A18 compound treatment 167320.0 -8560.0 -0.58 163840.0 -11100.0 -0.83 -0.9982 -0.9853 3071184 BCB03_000335 COc1ccc(cc1)[C@H]2OC[C@@H]3C[C@@H](Cc4ccccc4)C(=O)N23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A19 compound treatment 171960.0 -3920.0 -0.27 167120.0 -7850.0 -0.58 -0.6018 -0.9372 3070180 BCB03_000336 CCCCCCc1nc(Cc2cc(OC)c(OC)c(OC)c2)c(C)c3CO[Si](C(C)C)(C(C)C)c31 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A20 compound treatment 167920.0 -7960.0 -0.54 164440.0 -10500.0 -0.78 -0.9377 -0.9839 3071183 BCB03_000337 COc1ccc(cc1)[C@H]2OC[C@@H]3C[C@H](Cc4ccccc4)C(=O)N23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A21 compound treatment 164080.0 -11800.0 -0.8 163640.0 -11300.0 -0.84 -1.1649 -0.9997 3070181 BCB03_000338 CCCCCCc1nc(C2CC2)c(C)c3CO[Si](C(C)C)(C(C)C)c31 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A22 compound treatment 164520.0 -11400.0 -0.77 161480.0 -13500.0 -1.0 -1.2573 -0.9918 3189417 BCB03_000339 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@@H](Cc3ccccc3)Cn4cc(COC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A23 compound treatment 167360.0 -8520.0 -0.58 162120.0 -12800.0 -0.96 -1.0867 -0.9715 3188651 BCB03_000340 CCCCCCc1nc(cc2[C@@H](O[Si](C(C)C)(C(C)C)c21)c3ccccc3)c4ccc(o4)c5ccc(Cl)c(Cl)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 A24 compound treatment 164320.0 -11600.0 -0.79 160880.0 -14100.0 -1.05 -1.2986 -0.9901 3070196 BCB03_000341 CC(C)[C@@H](C(=O)O)n1cc(nn1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B01 compound treatment 176520.0 641.0 0.04 177880.0 2910.0 0.22 0.1843 0.8328 3188662 BCB03_000342 COC(=O)[C@H](Cc1ccccc1)N2CC(=C[C@@H]2[C@@H](O)Cc3ccccc3)/C=C/C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B02 compound treatment 257160.0 81300.0 5.54 244440.0 69500.0 5.17 7.5747 0.9994 3071724 BCB03_000343 BrC1=C[C@]23COC[C@H]3C[C@@H]1[C@]4(CO4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B03 compound treatment 191840.0 16000.0 1.09 199760.0 24800.0 1.85 2.0743 0.9683 3188663 BCB03_000344 COC(=O)[C@H](Cc1ccccc1)N2CC(=C)[C@@H](/C=C/C=C)[C@@H]2[C@@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B04 compound treatment 163560.0 -12300.0 -0.84 165200.0 -9770.0 -0.73 -1.1078 -0.9974 3071727 BCB03_000345 C[C@]12COC[C@@]2(C=C(Br)[C@@H]3C1)C(=O)[C@@]43CO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B05 compound treatment 172000.0 -3880.0 -0.26 170840.0 -4130.0 -0.31 -0.4041 -0.9972 3070955 BCB03_000346 COC(=O)[C@H](Cc1ccccc1)N2CC(C)(OC)O[C@@H](Cc3ccccc3)[C@H]2/C=C/C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B06 compound treatment 167400.0 -8480.0 -0.58 164120.0 -10800.0 -0.81 -0.9796 -0.9866 3071766 BCB03_000347 CCCCC[C@H]1OC[C@@]2(C=C(Br)[C@@H]3CC12)C(=O)[C@@]43CO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B07 compound treatment 175880.0 0.635 0.0 174840.0 -126.0 -0.01 -0.0066 -0.7038 3188666 BCB03_000348 COC(=O)[C@H](Cc1ccccc1)N2CC3=C[C@@H](C4CC4)n5n([C@H]3[C@@H]2[C@@H](O)Cc6ccccc6)c(=O)n(C)c5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B08 compound treatment 167640.0 -8240.0 -0.56 163200.0 -11800.0 -0.88 -1.0164 -0.977 3071767 BCB03_000349 CC1(C)OC[C@@]2(C=C(Br)[C@@H]3C[C@H]12)C(=O)[C@@]43CO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B09 compound treatment 169320.0 -6560.0 -0.45 164840.0 -10100.0 -0.75 -0.8491 -0.9689 3188667 BCB03_000350 O[C@@H](Cc1ccccc1)[C@@H](/C=C/C2CC2)N(CC#Cc3ccccc3)Cc4ccccc4Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B10 compound treatment 169120.0 -6760.0 -0.46 164840.0 -10100.0 -0.75 -0.8588 -0.9721 3071770 BCB03_000351 BrC1=C[C@]23COCC[C@H]3C[C@@H]1[C@@]4(CO4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B11 compound treatment 168320.0 -7560.0 -0.52 168080.0 -6890.0 -0.51 -0.7268 -1.0 3188668 BCB03_000352 CCC#CCN(Cc1ccccc1Br)[C@H](/C=C/c2ccccc2)[C@@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B12 compound treatment 219640.0 43800.0 2.98 221240.0 46300.0 3.44 4.5449 0.9974 3071774 BCB03_000353 C=CCC1=C[C@H]2[C@H]([C@H]3C=C[C@]2(CC=C)C(=O)[C@@]43CO4)[C@@]5(CO5)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B13 mock treatment 165720.0 -10200.0 -0.69 160480.0 -14500.0 -1.08 -1.2521 -0.9771 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B14 mock treatment 163640.0 -12200.0 -0.83 160600.0 -14400.0 -1.07 -1.3461 -0.9925 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B15 compound treatment 163640.0 -12200.0 -0.83 159880.0 -15100.0 -1.12 -1.384 -0.9893 3070996 BCB03_000354 O[C@@H](Cc1ccccc1)[C@@H](/C=C/c2ccccc2)N(CC#C)Cc3ccccc3Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B16 compound treatment 201880.0 26000.0 1.77 196880.0 21900.0 1.63 2.4067 0.9991 3188527 BCB03_000355 CC1=C[C@]2(CO)C(=O)[C@]3(CO3)[C@H]1[C@@H]4[C@@]5(CO5)C(=O)C(=C[C@@]42C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B17 compound treatment 170840.0 -5040.0 -0.34 162440.0 -12500.0 -0.93 -0.9021 -0.908 3070997 BCB03_000356 CCCC/C=C/[C@H]([C@@H](O)Cc1ccccc1)N(CC#Cc2ccccc2)Cc3ccccc3Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B18 compound treatment 165120.0 -10800.0 -0.73 166800.0 -8170.0 -0.61 -0.9484 -0.9956 3070938 BCB03_000357 CC(C)Cc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3cc(F)ccc3C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B19 compound treatment 168160.0 -7720.0 -0.53 163040.0 -11900.0 -0.89 -0.9998 -0.9689 3071055 BCB03_000358 CCC#CCN(Cc1ccccc1Br)[C@H](/C=C/C2CC2)[C@@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B20 compound treatment 176920.0 1040.0 0.07 165600.0 -9370.0 -0.7 -0.4427 -0.6319 3070939 BCB03_000359 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc(cc3)c4ccccc4)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B21 compound treatment 179200.0 3320.0 0.23 181320.0 6350.0 0.47 0.4945 0.9431 3188794 BCB03_000360 O[C@@H](Cc1ccccc1)[C@H](NCc2cccc(Cl)c2)/C=C/C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B22 compound treatment 170080.0 -5800.0 -0.4 170560.0 -4410.0 -0.33 -0.5114 -0.9957 3188531 BCB03_000361 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc(Oc4ccccc4)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B23 compound treatment 160120.0 -15800.0 -1.07 162880.0 -12100.0 -0.9 -1.3958 -0.9961 3188796 BCB03_000362 O[C@@H](Cc1ccccc1)[C@@H](/C=C/C2CC2)N(CC#Cc3ccccc3)Cc4cccc(Cl)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 B24 compound treatment 160240.0 -15600.0 -1.07 145720.0 -29200.0 -2.18 -2.2931 -0.9461 3188532 BCB03_000363 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc(cc3)C(F)(F)F)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C01 compound treatment 164600.0 -11300.0 -0.77 166960.0 -8010.0 -0.6 -0.9651 -0.992 3070235 BCB03_000364 CCCCCCc1nc(cc2[C@@H](O[Si](C(C)C)(C(C)C)c21)c3ccccc3)c4cc(C)c(OC)c(C)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C02 compound treatment 163160.0 -12700.0 -0.87 168920.0 -6050.0 -0.45 -0.9314 -0.9533 3189039 BCB03_000365 OC(=O)[C@H](Cc1ccccc1)n2cc(nn2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C03 compound treatment 158520.0 -17400.0 -1.18 168560.0 -6410.0 -0.48 -1.174 -0.9201 3070236 BCB03_000366 CCCCCCc1nc(cc2[C@@H](O[Si](C(C)C)(C(C)C)c21)c3ccccc3)c4ccc(OC)nc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C04 compound treatment 200680.0 24800.0 1.69 201920.0 27000.0 2.01 2.6141 0.9964 3070086 BCB03_000367 N[C@@H](Cc1ccccc1)C(=O)NCc2cn(CCCNC(=N)N)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C05 compound treatment 177560.0 1680.0 0.11 173080.0 -1890.0 -0.14 -0.0182 -0.1006 3188655 BCB03_000368 CCCCCCc1nc(Cc2cc(OC)c(OC)c(OC)c2)cc3[C@@H](O[Si](C(C)C)(C(C)C)c31)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C06 compound treatment 168880.0 -7000.0 -0.48 168360.0 -6610.0 -0.49 -0.6851 -0.9999 3070191 BCB03_000369 N[C@@H](Cc1ccccc1)C(=O)NCc2cn(Cc3ccccc3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C07 compound treatment 167880.0 -8000.0 -0.55 163200.0 -11800.0 -0.88 -1.0048 -0.974 3188656 BCB03_000370 CCCCCCc1nc(cc2[C@@H](O[Si](C(C)C)(C(C)C)c21)c3ccccc3)C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C08 compound treatment 168320.0 -7560.0 -0.52 170600.0 -4370.0 -0.32 -0.5942 -0.9753 3071180 BCB03_000371 OC(=O)[C@H](Cc1ccccc1)n2cc(nn2)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C09 compound treatment 169600.0 -6280.0 -0.43 168920.0 -6050.0 -0.45 -0.6209 -0.9997 3188772 BCB03_000372 CCCCCCc1nc(CCCc2cc3[C@@H](O[Si](C(C)C)(C(C)C)c3c(CCCCCC)n2)c4ccccc4)cc5[C@@H](O[Si](C(C)C)(C(C)C)c51)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C10 compound treatment 166680.0 -9200.0 -0.63 167880.0 -7090.0 -0.53 -0.8164 -0.9963 3070134 BCB03_000373 OC(=O)[C@H](Cc1ccccc1)n2cc(nn2)C3(O)CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C11 mock treatment 166040.0 -9840.0 -0.67 168680.0 -6290.0 -0.47 -0.8051 -0.9845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C12 mock treatment 175760.0 -119.0 -0.01 174800.0 -166.0 -0.01 -0.0145 -0.9796 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C13 compound treatment 174160.0 -1720.0 -0.12 166760.0 -8210.0 -0.61 -0.5147 -0.8277 3070242 BCB03_000374 CC(C)[Si]1(OCc2cc(nc(c21)c3ccccc3)c4ccc(o4)c5ccc(Cl)c(Cl)c5)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C14 compound treatment 165240.0 -10600.0 -0.73 173760.0 -1210.0 -0.09 -0.5764 -0.7886 3070089 BCB03_000375 CC(C)[C@@H](C(=O)O)n1cc(nn1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C15 mock treatment 162000.0 -13900.0 -0.95 168560.0 -6410.0 -0.48 -1.0062 -0.9496 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C16 mock treatment 165040.0 -10800.0 -0.74 167600.0 -7370.0 -0.55 -0.9102 -0.9892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C17 compound treatment 164320.0 -11600.0 -0.79 159840.0 -15100.0 -1.13 -1.3533 -0.9848 3070245 BCB03_000376 COc1c(C)cc(cc1C)c2cc3CO[Si](C(C)C)(C(C)C)c3c(n2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C18 compound treatment 171200.0 -4680.0 -0.32 168400.0 -6570.0 -0.49 -0.5711 -0.9786 3071179 BCB03_000377 CC(C)[C@@H](C(=O)O)n1cc(nn1)C2(O)CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C19 compound treatment 170400.0 -5480.0 -0.37 166640.0 -8330.0 -0.62 -0.7023 -0.9706 3070527 BCB03_000378 COc1cc(Cc2cc3CO[Si](C(C)C)(C(C)C)c3c(n2)c4ccccc4)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C20 compound treatment 165080.0 -10800.0 -0.74 166680.0 -8290.0 -0.62 -0.9567 -0.9961 3414058 BCB03_000379 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N(C)Cc3cn(C[C@H](Cc4ccccc4)NC2=O)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C21 compound treatment 176080.0 201.0 0.01 164600.0 -10400.0 -0.77 -0.5359 -0.6945 3070530 BCB03_000380 CC(C)[Si]1(OCc2cc(nc(c21)c3ccccc3)C4CC4)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C22 compound treatment 194960.0 19100.0 1.3 179640.0 4670.0 0.35 1.1658 0.8658 3189555 BCB03_000381 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N(Cc3ccccc3)Cc4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C23 compound treatment 168000.0 -7880.0 -0.54 157480.0 -17500.0 -1.3 -1.3001 -0.9234 3070081 BCB03_000382 CC(C)[Si]1(OCc2c1c(nc(c3ccc(o3)c4ccc(Cl)c(Cl)c4)c2C)c5ccccc5)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 C24 compound treatment 175320.0 -559.0 -0.04 172600.0 -2370.0 -0.18 -0.1515 -0.8408 3189558 BCB03_000383 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N(Cc3ccccc3)Cc4cnnn4C[C@@H](Cc5ccccc5)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D01 compound treatment 198600.0 22700.0 1.55 196880.0 21900.0 1.63 2.2486 0.9997 3071060 BCB03_000384 O[C@@H](Cc1ccccc1)[C@H](NCc2ccccc2Br)/C=C/c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D02 compound treatment 158920.0 -17000.0 -1.16 164640.0 -10300.0 -0.77 -1.361 -0.9803 3070941 BCB03_000385 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc4[nH]ccc4c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D03 compound treatment 213680.0 37800.0 2.58 213080.0 38100.0 2.84 3.8282 0.9989 3188797 BCB03_000386 O[C@@H](Cc1ccccc1)[C@H]2C3C=CCCC=C3CN2Cc4cccc(Cl)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D04 compound treatment 163960.0 -11900.0 -0.81 169280.0 -5690.0 -0.42 -0.8738 -0.9538 3070942 BCB03_000387 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3cccc4[nH]ccc34)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D05 compound treatment 166440.0 -9440.0 -0.64 174840.0 -126.0 -0.01 -0.4617 -0.7173 3188798 BCB03_000388 COC1(C)CN(Cc2ccccc2Br)[C@H](/C=C/c3ccccc3)[C@H](Cc4ccccc4)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D06 compound treatment 168560.0 -7320.0 -0.5 171200.0 -3770.0 -0.28 -0.551 -0.9628 3070943 BCB03_000389 CC(C)Oc1ccc(cc1)C(=O)N2CC[C@H](C2)NS(=O)(=O)c3cc(F)ccc3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D07 compound treatment 200400.0 24500.0 1.67 192840.0 17900.0 1.33 2.1228 0.9936 3188799 BCB03_000390 CN1C(=O)C2C3[C@H]([C@@H](O)Cc4ccccc4)N(Cc5cccc(Cl)c5)CC3=CC(C6CC6)C2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D08 compound treatment 169880.0 -6000.0 -0.41 165840.0 -9130.0 -0.68 -0.7695 -0.9705 3188537 BCB03_000391 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc(Br)cc3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D09 compound treatment 169920.0 -5960.0 -0.41 175560.0 594.0 0.04 -0.256 -0.6264 3071066 BCB03_000392 O[C@@H](Cc1ccccc1)[C@H](N(CC#C)CC2=CCCCC2)c3ccccc3Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D10 compound treatment 165400.0 -10500.0 -0.71 168040.0 -6930.0 -0.52 -0.8697 -0.9872 3070952 BCB03_000393 CC(C)Cc1ccc(CN2CC[C@@H](N)C2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D11 mock treatment 168640.0 -7240.0 -0.49 164960.0 -10000.0 -0.74 -0.8756 -0.98 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D12 mock treatment 174000.0 -1880.0 -0.13 170520.0 -4450.0 -0.33 -0.3246 -0.9147 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D13 compound treatment 176280.0 401.0 0.03 177440.0 2470.0 0.18 0.1495 0.8032 3071068 BCB03_000394 O=C(Cc1ccccc1)[C@H]2C3C=CCCC(=C3CN2Cc4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D14 compound treatment 168720.0 -7160.0 -0.49 169920.0 -5050.0 -0.38 -0.6107 -0.9916 3070953 BCB03_000395 CC(C)Cc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D15 mock treatment 164160.0 -11700.0 -0.8 166240.0 -8730.0 -0.65 -1.0242 -0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D16 mock treatment 169760.0 -6120.0 -0.42 163320.0 -11600.0 -0.87 -0.9079 -0.9438 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D17 compound treatment 219760.0 43900.0 2.99 201200.0 26200.0 1.95 3.4961 0.9786 3071112 BCB03_000396 O[C@@H](Cc1ccccc1)[C@H]2C3C=CCCC(=C3CN2Cc4cccc(Cl)c4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D18 compound treatment 169760.0 -6120.0 -0.42 166200.0 -8770.0 -0.65 -0.7563 -0.9767 3070954 BCB03_000397 CC(C)Cc1ccc(CN2CC[C@H](C2)NC(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D19 compound treatment 195000.0 19100.0 1.3 200040.0 25100.0 1.87 2.2414 0.9846 3188804 BCB03_000398 Clc1cccc(CN2CC3=CCCC=CC3[C@@H]2[C@H](Cc4ccccc4)OC(=O)C=C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D20 compound treatment 166400.0 -9480.0 -0.65 172440.0 -2530.0 -0.19 -0.5899 -0.8765 3188664 BCB03_000399 CC(C)Cc1ccc(CN2CC[C@H](C2)NC(=O)Nc3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D21 compound treatment 222640.0 46800.0 3.19 224640.0 49700.0 3.7 4.8685 0.9973 3071454 BCB03_000400 CCC1=C2CN(Cc3ccccc3Br)[C@@H]([C@@H](O)Cc4ccccc4)C2C=CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D22 compound treatment 164720.0 -11200.0 -0.76 170320.0 -4650.0 -0.35 -0.7825 -0.9363 3188665 BCB03_000401 CC(C)Oc1ccc(CN2CC[C@H](C2)NS(=O)(=O)c3cc(F)ccc3C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D23 compound treatment 193400.0 17500.0 1.19 190280.0 15300.0 1.14 1.6506 0.9997 3071455 BCB03_000402 CCC1=C2CN(Cc3ccccc3)[C@H](C2C=CCC1)C(=O)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 D24 compound treatment 162200.0 -13700.0 -0.93 155960.0 -19000.0 -1.41 -1.6597 -0.9796 3070994 BCB03_000403 CC(C)Oc1ccc(CN2CC[C@@H](C2)NS(=O)(=O)c3cc(F)ccc3C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E01 mock treatment 171760.0 -4120.0 -0.28 169840.0 -5130.0 -0.38 -0.4683 -0.9887 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E02 mock treatment 174240.0 -1640.0 -0.11 170080.0 -4890.0 -0.36 -0.3362 -0.8836 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E03 compound treatment 171800.0 -4080.0 -0.28 173720.0 -1250.0 -0.09 -0.2622 -0.8944 3189040 BCB03_000404 COc1c(C)cc(cc1C)c2nc(c3c(CO[Si]3(C(C)C)C(C)C)c2C)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E04 compound treatment 177120.0 1240.0 0.08 169200.0 -5770.0 -0.43 -0.2436 -0.557 3189560 BCB03_000405 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N(Cc3ccccc3)Cc4cn(C[C@@H]5CCCN5C2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E05 compound treatment 181120.0 5240.0 0.36 172720.0 -2250.0 -0.17 0.1345 0.3409 3189041 BCB03_000406 COc1ccc(cn1)c2nc(c3c(CO[Si]3(C(C)C)C(C)C)c2C)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E06 compound treatment 178360.0 2480.0 0.17 175440.0 474.0 0.04 0.1445 0.8367 3189559 BCB03_000407 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N(Cc3ccccc3)Cc4cnnn4C[C@@H]5CCCN5C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E07 compound treatment 208280.0 32400.0 2.21 206520.0 31600.0 2.35 3.2226 0.9995 3189042 BCB03_000408 CC(C)[Si]1(O[C@H](c2cc(nc(c21)c3ccccc3)c4ccc(o4)c5ccc(Cl)c(Cl)c5)c6ccccc6)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E08 compound treatment 176480.0 601.0 0.04 174200.0 -766.0 -0.06 -0.0113 -0.1616 3189043 BCB03_000409 N[C@@H](Cc1ccccc1)Cn2cc(nn2)C3(O)CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E09 mock treatment 175960.0 80.6 0.01 177360.0 2390.0 0.18 0.1299 0.7286 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E10 mock treatment 175960.0 80.6 0.01 174560.0 -406.0 -0.03 -0.0175 -0.569 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E11 compound treatment 175320.0 -559.0 -0.04 171280.0 -3690.0 -0.27 -0.2209 -0.7977 3070137 BCB03_000410 COc1c(C)cc(cc1C)c2cc3[C@@H](O[Si](C(C)C)(C(C)C)c3c(n2)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E12 compound treatment 182320.0 6440.0 0.44 178720.0 3750.0 0.28 0.5081 0.9762 3070143 BCB03_000411 N[C@@H](Cc1ccccc1)Cn2cc(nn2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E13 compound treatment 188000.0 12100.0 0.83 184800.0 9830.0 0.73 1.1019 0.9982 3189044 BCB03_000412 COc1ccc(cn1)c2cc3[C@@H](O[Si](C(C)C)(C(C)C)c3c(n2)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E14 compound treatment 176480.0 601.0 0.04 180480.0 5510.0 0.41 0.3192 0.7738 3189695 BCB03_000413 COC(=O)c1nc2oc1CC[C@@H](CO)NC(=O)N(C)Cc3cn(C[C@H](Cc4ccccc4)NC2=O)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E15 compound treatment 185760.0 9880.0 0.67 192240.0 17300.0 1.29 1.3854 0.9545 3189045 BCB03_000414 CC(C)[Si]1(O[C@H](c2cc(nc(c21)c3ccccc3)C4CC4)c5ccccc5)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E16 compound treatment 175360.0 -519.0 -0.04 176440.0 1470.0 0.11 0.0526 0.4558 3071393 BCB03_000415 COC(=O)c1nc2oc1CC[C@@H](CO)NC(=O)N(C)Cc3cnnn3C[C@H](Cc4ccccc4)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E17 mock treatment 175240.0 -639.0 -0.04 175720.0 754.0 0.06 0.0089 0.1248 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E18 mock treatment 176240.0 361.0 0.02 170880.0 -4090.0 -0.3 -0.1976 -0.6478 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E19 compound treatment 184240.0 8360.0 0.57 189000.0 14000.0 1.04 1.1416 0.9594 3189046 BCB03_000416 CC(C)[Si]1(OCc2cc(nc(CCc3ccccc3)c21)c4ccc(o4)c5ccc(Cl)c(Cl)c5)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E20 compound treatment 173440.0 -2440.0 -0.17 174240.0 -726.0 -0.05 -0.1558 -0.8909 3071396 BCB03_000417 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cn(C[C@H](C)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E21 compound treatment 169400.0 -6480.0 -0.44 175160.0 194.0 0.01 -0.3021 -0.6836 3189047 BCB03_000418 COc1c(C)cc(cc1C)c2cc3CO[Si](C(C)C)(C(C)C)c3c(CCc4ccccc4)n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E22 compound treatment 171160.0 -4720.0 -0.32 179320.0 4350.0 0.32 0.0016 0.0036 3187595 BCB03_000419 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cn(C[C@@H](NC2=O)C(C)C)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E23 compound treatment 169360.0 -6520.0 -0.44 168440.0 -6530.0 -0.49 -0.6577 -0.999 3189169 BCB03_000420 COc1ccc(cn1)c2cc3CO[Si](C(C)C)(C(C)C)c3c(CCc4ccccc4)n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 E24 compound treatment 182520.0 6640.0 0.45 179640.0 4670.0 0.35 0.5661 0.9915 3187594 BCB03_000421 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F01 mock treatment 174600.0 -1280.0 -0.09 166160.0 -8810.0 -0.66 -0.5251 -0.7942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F02 mock treatment 169920.0 -5960.0 -0.41 173840.0 -1130.0 -0.08 -0.3465 -0.8353 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F03 compound treatment 178760.0 2880.0 0.2 179920.0 4950.0 0.37 0.3996 0.9565 3071456 BCB03_000422 C/C=C\[C@@H](NCc1ccccc1Br)[C@@H](O)Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F04 compound treatment 177840.0 1960.0 0.13 180080.0 5110.0 0.38 0.3637 0.9015 3070995 BCB03_000423 Cc1ccc(F)cc1S(=O)(=O)N[C@@H]2CCN(Cc3ccc4OCOc4c3)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F05 compound treatment 184240.0 8360.0 0.57 171280.0 -3690.0 -0.27 0.2091 0.3305 3071457 BCB03_000424 CC(=CCN[C@H](CO)c1ccccc1)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F06 compound treatment 190720.0 14800.0 1.01 194200.0 19200.0 1.43 1.7277 0.9856 2133134 BCB03_000425 CCCCC(=O)N(CCN1CCOCC1)[C@@H]2CC(=C[C@H](Oc3c(I)cc(CO)cc3OC)[C@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F07 compound treatment 180120.0 4240.0 0.29 169400.0 -5570.0 -0.41 -0.0885 -0.1751 3071458 BCB03_000426 CC(=CCN(CC#C)[C@H](CO)c1ccccc1)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F08 compound treatment 174360.0 -1520.0 -0.1 171840.0 -3130.0 -0.23 -0.2377 -0.9336 2133147 BCB03_000427 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(CCN3CCOCC3)C(=O)C4CCCO4)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F09 mock treatment 176320.0 441.0 0.03 170280.0 -4690.0 -0.35 -0.2254 -0.6438 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F10 mock treatment 175720.0 -159.0 -0.01 174280.0 -686.0 -0.05 -0.0438 -0.8388 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F11 compound treatment 205400.0 29500.0 2.01 208160.0 33200.0 2.47 3.1701 0.9948 3187737 BCB03_000428 CC(=CCN(CC#Cc1ccccc1)[C@H](CO)c2ccccc2)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F12 compound treatment 228400.0 52500.0 3.58 215600.0 40600.0 3.02 4.6704 0.9965 3188671 BCB03_000429 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H](NCCc3c[nH]c4ccccc34)[C@@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F13 compound treatment 221320.0 45400.0 3.1 228080.0 53100.0 3.95 4.9859 0.9927 3071460 BCB03_000430 O=C1OC[C@@H](c2ccccc2)n3cc(/C=C/c4ccccc4)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F14 compound treatment 196000.0 20100.0 1.37 194800.0 19800.0 1.48 2.0138 0.9993 2129060 BCB03_000431 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H](NCC3CCCCC3)[C@@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F15 compound treatment 177880.0 2000.0 0.14 178640.0 3670.0 0.27 0.2898 0.9484 3071461 BCB03_000432 CC(=C)C/1CN([C@H](CO)c2ccccc2)C(=O)\C1=C/c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F16 compound treatment 197240.0 21400.0 1.46 198240.0 23300.0 1.73 2.2546 0.9963 2129057 BCB03_000433 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H](NC[C@@H]3CCCO3)[C@@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F17 mock treatment 176280.0 401.0 0.03 172920.0 -2050.0 -0.15 -0.0883 -0.5711 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F18 mock treatment 176040.0 161.0 0.01 174480.0 -486.0 -0.04 -0.0178 -0.4717 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F19 compound treatment 189040.0 13200.0 0.9 186440.0 11500.0 0.85 1.2383 0.9997 3071462 BCB03_000434 OCC(/C=C/c1ccccc1)N(CC#C)C(C(=O)O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F20 compound treatment 212680.0 36800.0 2.51 218600.0 43600.0 3.25 4.0705 0.9919 2129061 BCB03_000435 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H](NC3CCCCCC3)[C@@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F21 compound treatment 191840.0 16000.0 1.09 188760.0 13800.0 1.03 1.4954 0.9996 3071463 BCB03_000436 C/C=C/CN([C@H](CO[Si](C)(C)C(C)(C)C)c1ccccc1)C(=O)C#Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F22 compound treatment 217200.0 41300.0 2.82 223560.0 48600.0 3.62 4.5494 0.9924 2129067 BCB03_000437 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H](NCc3ccccc3F)[C@@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F23 compound treatment 184280.0 8400.0 0.57 182360.0 7390.0 0.55 0.7941 0.9998 3071464 BCB03_000438 O=C1OC[C@H](N(CC#C)C1/C=C/c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 F24 compound treatment 241520.0 65600.0 4.48 241560.0 66600.0 4.96 6.6691 0.9987 2129068 BCB03_000439 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H](NCc3ccc(F)cc3)[C@@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G01 compound treatment 190280.0 14400.0 0.98 188120.0 13200.0 0.98 1.3865 1.0 3189170 BCB03_000440 COc1cc(Cc2cc3CO[Si](C(C)C)(C(C)C)c3c(CCc4ccccc4)n2)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G02 compound treatment 186400.0 10500.0 0.72 184880.0 9910.0 0.74 1.0289 0.9999 3187594 BCB03_000441 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G03 mock treatment 177240.0 1360.0 0.09 176880.0 1910.0 0.14 0.1663 0.9784 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G04 mock treatment 186160.0 10300.0 0.7 185560.0 10600.0 0.79 1.0532 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G05 compound treatment 173720.0 -2160.0 -0.15 174640.0 -326.0 -0.02 -0.1212 -0.8126 3189171 BCB03_000442 CC(C)[Si]1(OCc2cc(nc(CCc3ccccc3)c21)C4CC4)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G06 compound treatment 185000.0 9120.0 0.62 181120.0 6150.0 0.46 0.7636 0.9887 3187597 BCB03_000443 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cnnn4C[C@@H](NC2=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G07 compound treatment 179080.0 3200.0 0.22 181760.0 6790.0 0.51 0.5119 0.9294 3071182 BCB03_000444 CC(C)[Si]1(OCc2cc(CCCc3cc4CO[Si](C(C)C)(C(C)C)c4c(CCc5ccccc5)n3)nc(CCc6ccccc6)c21)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G08 compound treatment 178840.0 2960.0 0.2 180840.0 5870.0 0.44 0.4519 0.9384 3189696 BCB03_000445 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G09 compound treatment 202280.0 26400.0 1.8 200320.0 25400.0 1.89 2.6071 0.9997 3189286 BCB03_000446 CC(C)[Si]1(O[C@H](c2cc(nc(CCc3ccccc3)c21)c4ccc(o4)c5ccc(Cl)c(Cl)c5)c6ccccc6)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G10 compound treatment 188560.0 12700.0 0.86 186000.0 11000.0 0.82 1.192 0.9997 3187593 BCB03_000447 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)NC3(CCCCC3)c4cnnn4C[C@@H](Cc5ccccc5)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G11 compound treatment 214680.0 38800.0 2.65 208640.0 33700.0 2.51 3.6427 0.9996 3189287 BCB03_000448 COc1c(C)cc(cc1C)c2cc3[C@@H](O[Si](C(C)C)(C(C)C)c3c(CCc4ccccc4)n2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G12 compound treatment 185400.0 9520.0 0.65 184200.0 9230.0 0.69 0.945 0.9996 3414059 BCB03_000449 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@@H](Cc3ccccc3)Cn4cc(CN(Cc5ccccc5)C2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G13 compound treatment 185640.0 9760.0 0.67 189400.0 14400.0 1.07 1.2302 0.9735 3189288 BCB03_000450 COc1ccc(cn1)c2cc3[C@@H](O[Si](C(C)C)(C(C)C)c3c(CCc4ccccc4)n2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G14 compound treatment 178840.0 2960.0 0.2 183960.0 8990.0 0.67 0.6161 0.8811 3414060 BCB03_000451 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@@H](Cc3ccccc3)Cn4cc(nn4)C5(CCCCC5)NC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G15 compound treatment 193880.0 18000.0 1.23 201800.0 26800.0 2.0 2.28 0.9727 3189289 BCB03_000452 COc1cc(Cc2cc3[C@@H](O[Si](C(C)C)(C(C)C)c3c(CCc4ccccc4)n2)c5ccccc5)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G16 compound treatment 177080.0 1200.0 0.08 179080.0 4110.0 0.31 0.2744 0.8657 3189561 BCB03_000453 CN1Cc2cn(C[C@H](Cc3ccccc3)NC(=O)c4cc(c(CC[C@@H](CO)NC1=O)o4)S(=O)(=O)c5ccc(C)cc5)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G17 compound treatment 180320.0 4440.0 0.3 176360.0 1390.0 0.1 0.2875 0.8982 3189171 BCB03_000454 CC(C)[Si]1(OCc2cc(nc(CCc3ccccc3)c21)C4CC4)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G18 compound treatment 186240.0 10400.0 0.71 183040.0 8070.0 0.6 0.9244 0.9968 3189290 BCB03_000455 COc1ccc(cc1)[C@H]2OC[C@@H]3CC(CC=C)(CC=C)C(=O)N23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G19 mock treatment 184040.0 8160.0 0.56 180280.0 5310.0 0.4 0.6731 0.986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G20 mock treatment 183720.0 7840.0 0.53 179160.0 4190.0 0.31 0.5987 0.9672 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G21 compound treatment 178160.0 2280.0 0.16 173560.0 -1410.0 -0.1 0.036 0.1919 3071182 BCB03_000456 CC(C)[Si]1(OCc2cc(CCCc3cc4CO[Si](C(C)C)(C(C)C)c4c(CCc5ccccc5)n3)nc(CCc6ccccc6)c21)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G22 compound treatment 185680.0 9800.0 0.67 183200.0 8230.0 0.61 0.9058 0.9991 3071255 BCB03_000457 NC(=N)NCC#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G23 compound treatment 178840.0 2960.0 0.2 175960.0 994.0 0.07 0.1951 0.9073 3188910 BCB03_000458 CC(C)[Si]1(OCc2cc(nc(c21)c3ccc(Oc4ccccc4)cc3)c5ccc(o5)c6ccc(Cl)c(Cl)c6)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 G24 compound treatment 178040.0 2160.0 0.15 174080.0 -886.0 -0.07 0.0575 0.3566 3189419 BCB03_000459 OC(=O)CCC(=O)N[C@@H](Cc1ccccc1)C(=O)NCC#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H01 compound treatment 198640.0 22800.0 1.55 188560.0 13600.0 1.01 1.8127 0.9785 3071464 BCB03_000460 O=C1OC[C@H](N(CC#C)C1/C=C/c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H02 compound treatment 182360.0 6480.0 0.44 180000.0 5030.0 0.37 0.5774 0.9966 3071064 BCB03_000461 CCCC(=O)N(CCc1c[nH]c2ccccc12)[C@@H]3CC(=C[C@H](Oc4c(I)cc(CO)cc4OC)[C@H]3O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H03 mock treatment 178800.0 2920.0 0.2 176280.0 1310.0 0.1 0.21 0.9464 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H04 mock treatment 181880.0 6000.0 0.41 177240.0 2270.0 0.17 0.409 0.9237 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H05 compound treatment 185600.0 9720.0 0.66 179120.0 4150.0 0.31 0.6872 0.9398 3071517 BCB03_000462 CC(=C)C1C(=C)CN([C@H](CO)c2ccccc2)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H06 compound treatment 176960.0 1080.0 0.07 182320.0 7350.0 0.55 0.4391 0.7951 2133032 BCB03_000463 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(CC3CCCCC3)C(=O)c4ccc(cc4)C(F)(F)F)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H07 compound treatment 177400.0 1520.0 0.1 179440.0 4470.0 0.33 0.3088 0.8853 3187880 BCB03_000464 CC(C)(C)OC(=O)N(CC#C)[C@H](CO)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H08 compound treatment 178000.0 2120.0 0.14 181520.0 6550.0 0.49 0.4472 0.8789 2133035 BCB03_000465 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(CC3CCCCC3)C(=O)c4cc5ccccc5oc4=O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H09 compound treatment 217600.0 41700.0 2.84 208480.0 33500.0 2.49 3.7751 0.9979 3071519 BCB03_000466 CC(=CCN([C@H](CO)c1ccccc1)C(=O)C#Cc2ccccc2)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H10 compound treatment 180640.0 4760.0 0.32 180160.0 5190.0 0.39 0.5029 0.9962 2133267 BCB03_000467 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(Cc3ccc(F)cc3)C(=O)C4CCCO4)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H11 compound treatment 183760.0 7880.0 0.54 182120.0 7150.0 0.53 0.7564 1.0 3071520 BCB03_000468 OC[C@@H](N(C/C=C/c1ccccc1)CC#C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H12 compound treatment 201480.0 25600.0 1.75 194280.0 19300.0 1.44 2.2506 0.9954 2133153 BCB03_000469 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(CCN3CCOCC3)C(=O)C4CCOC4)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H13 compound treatment 180800.0 4920.0 0.34 183040.0 8070.0 0.6 0.6621 0.9621 3071521 BCB03_000470 CC(C)(C)[Si](C)(C)OC[C@@H](N(C/C=C/c1ccccc1)CC#C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H14 compound treatment 198720.0 22800.0 1.56 197080.0 22100.0 1.65 2.2649 0.9996 2132929 BCB03_000471 CC/C=C/C(=O)N(C[C@@H]1CCCO1)[C@@H]2CC(=C[C@H](Oc3c(I)cc(CO)cc3OC)[C@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H15 compound treatment 222960.0 47100.0 3.21 225640.0 50700.0 3.77 4.9366 0.9968 3071522 BCB03_000472 O=C1OC[C@H](N2CC(=CC21)/C=C/c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H16 compound treatment 204360.0 28500.0 1.94 200520.0 25600.0 1.9 2.7179 0.9999 2133065 BCB03_000473 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(C3CCCCCC3)C(=O)c4cc5ccccc5oc4=O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H17 compound treatment 194880.0 19000.0 1.3 195360.0 20400.0 1.52 1.9893 0.9969 3071523 BCB03_000474 OCC(/C=C/c1ccccc1)N(CC#C)Cc2ccccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H18 compound treatment 364960.0 189000.0 12.89 349440.0 174000.0 12.99 18.2975 1.0 2133224 BCB03_000475 CCCCC(=O)N(Cc1ccccc1F)[C@@H]2CC(=C[C@H](Oc3c(I)cc(CO)cc3OC)[C@H]2O)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H19 mock treatment 182720.0 6840.0 0.47 181400.0 6430.0 0.48 0.6684 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H20 mock treatment 181240.0 5360.0 0.37 177920.0 2950.0 0.22 0.4139 0.9704 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H21 compound treatment 205040.0 29200.0 1.99 203360.0 28400.0 2.11 2.9001 0.9995 3071524 BCB03_000476 OCC1C=C(CN1Cc2ccccc2Br)/C=C/c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H22 compound treatment 417640.0 242000.0 16.48 408120.0 233000.0 17.35 23.9253 0.9997 2133510 BCB03_000477 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@H]([C@@H]2O)N(CCc3cccc(F)c3)C(=O)CCC4CCCC4)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H23 compound treatment 176280.0 401.0 0.03 170840.0 -4130.0 -0.31 -0.1978 -0.6417 3414064 BCB03_000478 O=S1(=O)N2CCC[C@@H]2[C@@H](Oc3ccccc31)C#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 H24 compound treatment 245400.0 69500.0 4.74 226400.0 51400.0 3.83 6.0583 0.9944 2128988 BCB03_000479 COc1cc(CO)cc(I)c1O[C@H]2C=C(C[C@@H]3O[C@@H]32)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I01 compound treatment 175000.0 -879.0 -0.06 168840.0 -6130.0 -0.46 -0.3648 -0.7933 3070742 BCB03_000480 COc1c(C)cc(cc1C)c2cc3CO[Si](C(C)C)(C(C)C)c3c(n2)c4ccc(Oc5ccccc5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I02 compound treatment 177800.0 1920.0 0.13 178400.0 3430.0 0.26 0.2733 0.9517 3189420 BCB03_000481 COc1ccc(cc1)[C@H]2OC[C@@H]3C[C@](Cc4ccccc4)(C(=O)OCC=C)C(=O)N23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I03 compound treatment 182480.0 6600.0 0.45 182280.0 7310.0 0.54 0.7031 0.9955 3070750 BCB03_000482 COc1ccc(cn1)c2cc3CO[Si](C(C)C)(C(C)C)c3c(n2)c4ccc(Oc5ccccc5)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I04 compound treatment 178240.0 2360.0 0.16 183280.0 8310.0 0.62 0.5514 0.8623 1035256 BCB03_000483 C#CCNCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I05 mock treatment 180720.0 4840.0 0.33 179560.0 4590.0 0.34 0.4751 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I06 mock treatment 181360.0 5480.0 0.37 178080.0 3110.0 0.23 0.4281 0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I07 compound treatment 176960.0 1080.0 0.07 179160.0 4190.0 0.31 0.2728 0.8506 3188915 BCB03_000484 CC(C)[Si]1(OCc2cc(nc(c21)c3ccc(Oc4ccccc4)cc3)C5CC5)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I08 compound treatment 184520.0 8640.0 0.59 179600.0 4630.0 0.34 0.6604 0.9675 3071258 BCB03_000485 CC(C)[C@H](N=[N+]=[N-])C(=O)N[C@@H](Cc1ccccc1)C(=O)NCC#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I09 compound treatment 176800.0 921.0 0.06 180560.0 5590.0 0.42 0.3388 0.8046 3070808 BCB03_000486 CC(C)[Si]1(O[C@H](c2cc(nc(c21)c3ccc(Oc4ccccc4)cc3)C5CC5)c6ccccc6)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I10 compound treatment 181560.0 5680.0 0.39 180480.0 5510.0 0.41 0.5641 0.9996 3189550 BCB03_000487 COc1cccc(C[C@]2(C[C@@H](CO)NC2=O)C(=O)OCc3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I11 compound treatment 188280.0 12400.0 0.85 180200.0 5230.0 0.39 0.8733 0.9381 3070078 BCB03_000488 CC[C@@H]1O[Si](C(C)C)(C(C)C)c2c1cc(nc2c3ccc(Oc4ccccc4)cc3)c5cc(C)c(OC)c(C)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I12 compound treatment 183200.0 7320.0 0.5 177360.0 2390.0 0.18 0.4789 0.9037 3189551 BCB03_000489 COc1cccc(C[C@@]2(C[C@@H](CO)NC2=O)C(=O)OCc3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I13 compound treatment 188000.0 12100.0 0.83 188960.0 14000.0 1.04 1.3208 0.9934 3070690 BCB03_000490 CCCCCCc1nc(cc2CO[Si](C(C)C)(C(C)C)c21)C(=C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I14 compound treatment 182720.0 6840.0 0.47 181280.0 6310.0 0.47 0.6621 1.0 3071267 BCB03_000491 CN(C)S(=O)(=O)NCC#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I15 compound treatment 187200.0 11300.0 0.77 191240.0 16300.0 1.21 1.4022 0.9763 3071259 BCB03_000492 CC(C)[Si](O[C@@H](c1cn(Cc2ccccc2)nn1)c3ccccc3)(C#Cc4ccccc4)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I16 compound treatment 194280.0 18400.0 1.25 194240.0 19300.0 1.43 1.9014 0.9978 3189556 BCB03_000493 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N(Cc3ccccc3)Cc4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I17 compound treatment 185000.0 9120.0 0.62 186000.0 11000.0 0.82 1.0204 0.9906 3071266 BCB03_000494 CC(C)[Si](O[C@@H](c1cn(Cc2ccccc2)nn1)c3ccccc3)(C#CCCc4ccccc4)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I18 compound treatment 182160.0 6280.0 0.43 180880.0 5910.0 0.44 0.614 0.9999 3188911 BCB03_000495 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@H](Cc3ccccc3)Cn4cc(CN(C)C2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I19 compound treatment 186880.0 11000.0 0.75 187520.0 12600.0 0.93 1.191 0.9941 3189415 BCB03_000496 CCCCCCC#C[Si](O[C@@H](C#C)c1ccccc1)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I20 compound treatment 177720.0 1840.0 0.13 177560.0 2590.0 0.19 0.2253 0.9782 3188912 BCB03_000497 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@H](C)Cn3cc(CN(C)C2=O)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I21 mock treatment 174160.0 -1720.0 -0.12 176680.0 1710.0 0.13 0.0073 0.0423 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I22 mock treatment 176120.0 241.0 0.02 173800.0 -1170.0 -0.09 -0.0497 -0.5634 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I23 compound treatment 178800.0 2920.0 0.2 177720.0 2750.0 0.2 0.2858 0.9999 3189416 BCB03_000498 CCCCCCC#C[Si](OCC#CC)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 I24 compound treatment 168760.0 -7120.0 -0.49 168840.0 -6130.0 -0.46 -0.6656 -0.9995 3188913 BCB03_000499 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@@H](Cc3ccccc3)Cn4cc(CN(C)C2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J01 compound treatment 176840.0 961.0 0.07 172400.0 -2570.0 -0.19 -0.0887 -0.4395 3071594 BCB03_000500 O=S1(=O)N2CCC[C@H]2[C@H](Oc3ccccc31)C#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J02 compound treatment 183960.0 8080.0 0.55 180320.0 5350.0 0.4 0.6713 0.9874 3187871 BCB03_000501 OCCNC(=O)C1=C[C@H](Oc2ccccc2I)[C@@H](O)[C@@H](C1)N(Cc3ccco3)C(=O)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J03 compound treatment 191280.0 15400.0 1.05 188080.0 13100.0 0.98 1.4326 0.9993 3071530 BCB03_000502 CCOC(=O)[C@H]1C[C@H]2O[C@]32C[C@H]1C(=O)N4CCCC4[C@@H]3O[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J04 compound treatment 284640.0 109000.0 7.41 271640.0 96700.0 7.2 10.3309 0.9999 2129008 BCB03_000503 OCCNC(=O)C1=C[C@H](Oc2ccccc2I)[C@@H](O)[C@@H](C1)NCc3ccc(F)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J05 mock treatment 177120.0 1240.0 0.08 179480.0 4510.0 0.34 0.2974 0.8583 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J06 mock treatment 177000.0 1120.0 0.08 180160.0 5190.0 0.39 0.3274 0.8308 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J07 compound treatment 246040.0 70200.0 4.78 236560.0 61600.0 4.58 6.6239 0.9998 3071528 BCB03_000504 CCOC(=O)[C@H]1CC=C2CC1C(=O)N3CCC[C@@H]3[C@@H]2O[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J08 compound treatment 217760.0 41900.0 2.86 208920.0 34000.0 2.53 3.8059 0.9981 3187877 BCB03_000505 CC(C)C[C@@H]1NC(=O)[C@@]2(C3[C@H](Cc4ccccc4)NC2=O)C(/C=C/CC\C=C\CNC(=O)[C@@H](C)NC1=O)[C@@H]5O[C@]5(C)[C@H]3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J09 compound treatment 197520.0 21600.0 1.48 189480.0 14500.0 1.08 1.8071 0.9883 3071529 BCB03_000506 CCOC(=O)[C@@H]1CC2O[C@@]32C[C@@H]1C(=O)N4CCC[C@@H]4[C@H]3O[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J10 compound treatment 276360.0 100000.0 6.85 265800.0 90800.0 6.76 9.6244 1.0 3188005 BCB03_000507 CC(C)C[C@@H]1NC(=O)C(NC(=O)[C@@]2(C3[C@H](Cc4ccccc4)NC2=O)C(/C=C/CC\C=C\CNC1=O)[C@@H]5O[C@]5(C)[C@H]3C)[C@@H](C)OCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J11 compound treatment 192240.0 16400.0 1.12 191560.0 16600.0 1.24 1.662 0.9987 3071527 BCB03_000508 CCOC(=O)[C@@H]1CC=C2CC1C(=O)N3CCC[C@@H]3[C@H]2O[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J12 compound treatment 278080.0 102000.0 6.97 273240.0 98300.0 7.31 10.0989 0.9997 3188007 BCB03_000509 CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@@]2(C3[C@H](Cc4ccccc4)NC2=O)C(/C=C/CC\C=C\CNC1=O)[C@@H]5O[C@]5(C)[C@H]3C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J13 compound treatment 229960.0 54100.0 3.69 222640.0 47700.0 3.55 5.1161 0.9998 3071654 BCB03_000510 [O-][N+](=O)c1ccccc1S(=O)(=O)N2CCC[C@@H]2[C@H]3OCC=C3C(=C)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J14 compound treatment 218760.0 42900.0 2.92 221240.0 46300.0 3.44 4.5025 0.9967 3188008 BCB03_000511 C[C@H]1C2[C@H](Cc3ccccc3)NC(=O)[C@@]24C(/C=C/CC\C=C\CNC(=O)[C@@H]5CCCN5C(=O)[C@H](Cc6ccccc6)NC4=O)[C@@H]7O[C@@]71C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J15 compound treatment 210440.0 34600.0 2.36 199400.0 24400.0 1.82 2.952 0.9918 3071597 BCB03_000512 Cc1ccc(cc1)S(=O)(=O)NC/C=C\C(=C)[C@H](O)[C@H]2CCCN2S(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J16 compound treatment 221760.0 45900.0 3.13 219600.0 44600.0 3.32 4.5608 0.9995 3188142 BCB03_000513 C[C@@H](OCc1ccccc1)C2NC(=O)[C@@]3(C4[C@H](Cc5ccccc5)NC3=O)C(/C=C/C\C=C/CNC(=O)[C@@H](C)NC2=O)[C@@H]6O[C@]6(C)[C@H]4C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J17 compound treatment 195160.0 19300.0 1.31 194760.0 19800.0 1.47 1.9712 0.9984 3071598 BCB03_000514 Cc1ccc(cc1)S(=O)(=O)NC/C=C/C(=C)[C@H](O)[C@H]2CCCN2S(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J18 compound treatment 217080.0 41200.0 2.81 222920.0 48000.0 3.57 4.5099 0.993 3188271 BCB03_000515 CC(C)C[C@H]1NC(=O)CNC(=O)[C@@]2(C3[C@H](Cc4ccccc4)NC2=O)C(/C=C/C\C=C/CNC1=O)[C@@H]5O[C@]5(C)[C@H]3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J19 compound treatment 191600.0 15700.0 1.07 192080.0 17100.0 1.27 1.6586 0.9963 3188138 BCB03_000516 Cc1ccc(cc1)S(=O)(=O)N(CCC=C)CC#C[C@H]2Oc3ccccc3S(=O)(=O)N4CCC[C@@H]24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J20 compound treatment 265080.0 89200.0 6.08 274200.0 99200.0 7.39 9.5227 0.9953 3188272 BCB03_000517 CC(C)C[C@H]1NC(=O)C(NC(=O)[C@@]2(C3[C@H](Cc4ccccc4)NC2=O)C(/C=C/C\C=C/CNC1=O)[C@@H]5O[C@]5(C)[C@H]3C)[C@@H](C)OCc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J21 mock treatment 173960.0 -1920.0 -0.13 175480.0 514.0 0.04 -0.0655 -0.4802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J22 mock treatment 168720.0 -7160.0 -0.49 171680.0 -3290.0 -0.24 -0.5181 -0.9489 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J23 compound treatment 187000.0 11100.0 0.76 186240.0 11300.0 0.84 1.1294 0.9987 3071656 BCB03_000518 CN1C(=C)C2CC3C4C(C5CO[C@H]([C@H]6CCCN6S(=O)(=O)c7ccccc7[N+](=O)[O-])C5=C3CC2C1=O)C(=O)N(C)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 J24 compound treatment 235360.0 59500.0 4.06 247520.0 72600.0 5.4 6.6858 0.99 3188275 BCB03_000519 CC(C)C[C@H]1NC(=O)[C@H](C)NC(=O)[C@@]2(C3[C@H](Cc4ccccc4)NC2=O)C(/C=C/C\C=C/CNC1=O)[C@@H]5O[C@]5(C)[C@H]3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K01 compound treatment 204600.0 28700.0 1.96 201240.0 26300.0 1.96 2.7673 1.0 3071254 BCB03_000520 CC(C)[Si](O[C@@H](C#C)c1ccccc1)(C#Cc2ccccc2)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K02 compound treatment 197280.0 21400.0 1.46 198000.0 23000.0 1.71 2.2439 0.9968 3220747 BCB03_000521 COC(=O)c1c(CC[C@@H](CO)NC(=O)N2CCCC2)oc(C(=O)Cc3ccccc3)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K03 compound treatment 176560.0 681.0 0.05 176400.0 1430.0 0.11 0.1083 0.9304 3189418 BCB03_000522 CC#CCO[Si](C#Cc1ccccc1)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K04 compound treatment 196640.0 20800.0 1.42 196000.0 21000.0 1.57 2.1078 0.9987 3220749 BCB03_000523 COC(=O)c1c(CC[C@@H](CO)NC(=O)NCC(C)C)oc(C(=O)Cc2ccccc2)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K05 compound treatment 206760.0 30900.0 2.11 196480.0 21500.0 1.6 2.621 0.9909 3071256 BCB03_000524 CC(C)[Si](O[C@@H](C#C)c1ccccc1)(C#Cc2ccc(Oc3ccccc3)cc2)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K06 compound treatment 230160.0 54300.0 3.7 222520.0 47600.0 3.54 5.1195 0.9998 3220751 BCB03_000525 COC(=O)c1c(CC[C@@H](CO)NC(=O)Nc2ccc(OC)cc2)oc(C(=O)Cc3ccccc3)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K07 mock treatment 182400.0 6520.0 0.44 185080.0 10100.0 0.75 0.8466 0.9684 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K08 mock treatment 181600.0 5720.0 0.39 177720.0 2750.0 0.2 0.4207 0.9549 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K09 compound treatment 200600.0 24700.0 1.69 194920.0 20000.0 1.49 2.2419 0.998 3071257 BCB03_000526 CC[C@@H](O[Si](C#Cc1ccc(Oc2ccccc2)cc1)(C(C)C)C(C)C)C#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K10 compound treatment 185480.0 9600.0 0.65 182240.0 7270.0 0.54 0.8457 0.9956 3220772 BCB03_000527 COC(=O)c1c(CC[C@@H](CO)NC(=O)NCCc2c[nH]c3ccccc23)oc(C(=O)Cc4ccccc4)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K11 compound treatment 186200.0 10300.0 0.7 180040.0 5070.0 0.38 0.7646 0.9574 3189421 BCB03_000528 CC(C)[Si](Oc1ccccc1Br)(C#CCCCC#N)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K12 compound treatment 189600.0 13700.0 0.94 192040.0 17100.0 1.27 1.56 0.9886 3220775 BCB03_000529 COC(=O)c1c(CC[C@@H](CO)NC(=O)Nc2nc[nH]n2)oc(C(=O)Cc3ccccc3)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K13 compound treatment 182320.0 6440.0 0.44 189360.0 14400.0 1.07 1.068 0.9225 3189422 BCB03_000530 CC[C@@H](O[Si](C#CCCCC#N)(C(C)C)C(C)C)C#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K14 compound treatment 186400.0 10500.0 0.72 190520.0 15600.0 1.16 1.3258 0.9735 3220649 BCB03_000531 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](Cc2ccccc2)Cn3cc(nn3)C4(O)CCCCC4)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K15 mock treatment 181560.0 5680.0 0.39 181360.0 6390.0 0.48 0.6104 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K16 mock treatment 179600.0 3720.0 0.25 177040.0 2070.0 0.15 0.2885 0.9717 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K17 compound treatment 198240.0 22400.0 1.52 196280.0 21300.0 1.59 2.1997 0.9998 3189552 BCB03_000532 CC(C)[Si](O[C@@H](c1cn(Cc2ccccc2)nn1)c3ccccc3)(C#C[Si](C(C)C)(C(C)C)C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K18 compound treatment 174800.0 -1080.0 -0.07 176480.0 1510.0 0.11 0.0277 0.2055 3220651 BCB03_000533 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](Cc2ccccc2)Cn3cc(nn3)c4cncn4C)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K19 compound treatment 199240.0 23400.0 1.59 201840.0 26900.0 2.0 2.5405 0.9936 3189553 BCB03_000534 CC[C@@H](O[Si](C#C[Si](C(C)C)(C(C)C)C(C)C)(C(C)C)C(C)C)c1cn(nn1)[C@H](CO)Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K20 compound treatment 177240.0 1360.0 0.09 181400.0 6430.0 0.48 0.4042 0.8287 3220653 BCB03_000535 CCCCc1cn(C[C@H](Cc2ccccc2)NC(=O)N[C@H](CO)CCc3oc(C(=O)C)c(C(=O)OC)c3C(=O)OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K21 compound treatment 189600.0 13700.0 0.94 192520.0 17600.0 1.31 1.5853 0.9866 3189554 BCB03_000536 CC[C@@H](O[Si](C#C[Si](C(C)C)(C(C)C)C(C)C)(C(C)C)C(C)C)c1cn(Cc2cccc(Cl)c2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K22 compound treatment 175600.0 -279.0 -0.02 174600.0 -366.0 -0.03 -0.0327 -0.9848 3220655 BCB03_000537 CCOC(=O)c1cn(C[C@H](Cc2ccccc2)NC(=O)N[C@H](CO)CCc3oc(C(=O)C)c(C(=O)OC)c3C(=O)OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K23 mock treatment 170240.0 -5640.0 -0.38 164240.0 -10700.0 -0.8 -0.8363 -0.9439 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 K24 mock treatment 167640.0 -8240.0 -0.56 172120.0 -2850.0 -0.21 -0.547 -0.9111 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L01 compound treatment 198160.0 22300.0 1.52 195120.0 20200.0 1.5 2.1348 1.0 3071655 BCB03_000538 CN1C(=O)C2CC=C(CC2C1=O)C3=CCO[C@@H]3[C@H]4CCCN4S(=O)(=O)c5ccccc5[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L02 compound treatment 190040.0 14200.0 0.97 191360.0 16400.0 1.22 1.5455 0.9933 3188392 BCB03_000539 C[C@H]1C2[C@H](Cc3ccccc3)NC(=O)[C@@]24C(/C=C/C\C=C/CNC(=O)[C@@H]5CCCN5C(=O)CNC4=O)[C@@H]6O[C@@]61C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L03 compound treatment 184960.0 9080.0 0.62 176040.0 1070.0 0.08 0.4943 0.7919 3188141 BCB03_000540 C=CC(=C)[C@H]1Oc2ccccc2S(=O)(=O)N3CCC[C@@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L04 compound treatment 185600.0 9720.0 0.66 181480.0 6510.0 0.48 0.8114 0.9882 3188274 BCB03_000541 CC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2[C@H]4[C@@H](C1)C(=O)N(Cc5ccccc5)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L05 compound treatment 183520.0 7640.0 0.52 179520.0 4550.0 0.34 0.608 0.9783 3071592 BCB03_000542 CN1C(=O)C2CC=C(CC2C1=O)[C@H]3Oc4ccccc4S(=O)(=O)N5CCC[C@@H]35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L06 compound treatment 183920.0 8040.0 0.55 189600.0 14600.0 1.09 1.1578 0.9495 3070931 BCB03_000543 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)C)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L07 mock treatment 180800.0 4920.0 0.34 177920.0 2950.0 0.22 0.3927 0.979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L08 mock treatment 180480.0 4600.0 0.31 175440.0 474.0 0.04 0.2467 0.7818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L09 compound treatment 184680.0 8800.0 0.6 180560.0 5590.0 0.42 0.7187 0.9841 3071592 BCB03_000544 CN1C(=O)C2CC=C(CC2C1=O)[C@H]3Oc4ccccc4S(=O)(=O)N5CCC[C@@H]35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L10 compound treatment 199840.0 24000.0 1.63 193120.0 18200.0 1.35 2.1105 0.9956 3070933 BCB03_000545 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)COC)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L11 compound treatment 230040.0 54200.0 3.69 221840.0 46900.0 3.49 5.0779 0.9996 3071581 BCB03_000546 O=C1C2CC=C(CC2C(=O)c3ccccc13)[C@H]4Oc5ccccc5S(=O)(=O)N6CCC[C@@H]46 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L12 compound treatment 195320.0 19400.0 1.33 193160.0 18200.0 1.35 1.8947 0.9999 3188523 BCB03_000547 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)COc4ccccc4)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L13 compound treatment 255360.0 79500.0 5.42 253360.0 78400.0 5.83 7.9573 0.9993 3071582 BCB03_000548 O=C1c2ccccc2C(=O)c3cc(ccc13)[C@H]4Oc5ccccc5S(=O)(=O)N6CCC[C@@H]46 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L14 compound treatment 202000.0 26100.0 1.78 200600.0 25600.0 1.91 2.6083 0.9994 3188524 BCB03_000549 CC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2n4n(C1)c(=O)n(c5ccccc5)c4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L15 mock treatment 181920.0 6040.0 0.41 183880.0 8910.0 0.66 0.7603 0.9737 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L16 mock treatment 178680.0 2800.0 0.19 178360.0 3390.0 0.25 0.3136 0.9905 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L17 compound treatment 175440.0 -439.0 -0.03 175520.0 554.0 0.04 0.008 0.1567 3071529 BCB03_000550 CCOC(=O)[C@@H]1CC2O[C@@]32C[C@@H]1C(=O)N4CCC[C@@H]4[C@H]3O[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L18 compound treatment 197120.0 21200.0 1.45 196440.0 21500.0 1.6 2.1541 0.9988 3188525 BCB03_000551 COCC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2n4n(C1)c(=O)n(c5ccccc5)c4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L19 compound treatment 174360.0 -1520.0 -0.1 177920.0 2950.0 0.22 0.0822 0.3383 3071527 BCB03_000552 CCOC(=O)[C@@H]1CC=C2CC1C(=O)N3CCC[C@@H]3[C@H]2O[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L20 compound treatment 217600.0 41700.0 2.84 214200.0 39200.0 2.92 4.0761 0.9999 3188526 BCB03_000553 OB1C[C@H]2C(=C(COc3ccccc3)Cn4n2c(=O)n(c5ccccc5)c4=O)[C@@H](CCc6ccccc6)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L21 compound treatment 267440.0 91600.0 6.24 266520.0 91600.0 6.81 9.2323 0.999 3071531 BCB03_000554 CCOC(=O)[C@@H]1[C@@H]2CN(CCC2=C[C@@H]3[C@@H](O[Si](C(C)C)(C(C)C)C(C)C)[C@@H]4CCCN4C(=O)[C@@H]13)S(=O)(=O)c5ccc(C)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L22 compound treatment 180280.0 4400.0 0.3 177400.0 2430.0 0.18 0.3403 0.9708 3188538 BCB03_000555 CCCC[C@H]1OB(O)C[C@H]2C1=C(C)Cn3n2c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L23 mock treatment 171360.0 -4520.0 -0.31 175000.0 34.3 0.0 -0.2161 -0.7012 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 L24 mock treatment 168360.0 -7520.0 -0.51 169600.0 -5370.0 -0.4 -0.6449 -0.9924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M01 compound treatment 181680.0 5800.0 0.4 170400.0 -4570.0 -0.34 0.0394 0.0755 3071269 BCB03_000556 CC[C@@H](O[Si](C#C[Si](C(C)C)(C(C)C)C(C)C)(C(C)C)C(C)C)c1cn(nn1)[C@H](C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M02 compound treatment 182440.0 6560.0 0.45 175360.0 394.0 0.03 0.337 0.7519 3220657 BCB03_000557 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](C)Cn2cc(nn2)c3ccccn3)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M03 compound treatment 186360.0 10500.0 0.71 184360.0 9390.0 0.7 0.9997 0.9999 3189557 BCB03_000558 CCCC#C[Si](O[C@H](CC)c1cn(Cc2ccccc2)nn1)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M04 compound treatment 203080.0 27200.0 1.85 199560.0 24600.0 1.83 2.6056 1.0 3220659 BCB03_000559 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](C)Cn2cc(nn2)C3(O)CCCCC3)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M05 compound treatment 185200.0 9320.0 0.64 182960.0 7990.0 0.59 0.8701 0.9995 3071329 BCB03_000560 CCCC#C[Si](O[C@H](CC)c1cn(nn1)[C@H](CO)Cc2ccccc2)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M06 compound treatment 185640.0 9760.0 0.67 182480.0 7510.0 0.56 0.866 0.9963 3220661 BCB03_000561 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](C)Cn2cc(nn2)C3(O)CCCC3)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M07 compound treatment 183200.0 7320.0 0.5 183040.0 8070.0 0.6 0.7778 0.9957 3071331 BCB03_000562 CCCC#C[Si](O[C@H](CC)c1cn(nn1)[C@H](C)c2ccccc2)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M08 compound treatment 186360.0 10500.0 0.71 182640.0 7670.0 0.57 0.9091 0.9938 3220665 BCB03_000563 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@H](Cn2cc(Cc3ccccc3)nn2)C(C)C)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M09 mock treatment 180880.0 5000.0 0.34 179520.0 4550.0 0.34 0.4808 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M10 mock treatment 206560.0 30700.0 2.09 200560.0 25600.0 1.9 2.826 0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M11 compound treatment 200440.0 24600.0 1.67 208320.0 33400.0 2.48 2.9394 0.9816 3071332 BCB03_000564 CCCCCCC#C[Si](O[C@@H](c1cn(Cc2ccccc2)nn1)c3ccccc3)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M12 compound treatment 208040.0 32200.0 2.19 206880.0 31900.0 2.38 3.23 0.9992 3220667 BCB03_000565 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@H](Cn2cc(nn2)C3(O)CCCCC3)C(C)C)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M13 mock treatment 184720.0 8840.0 0.6 188760.0 13800.0 1.03 1.1522 0.9678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M14 mock treatment 179080.0 3200.0 0.22 182680.0 7710.0 0.57 0.5603 0.9122 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M15 compound treatment 189160.0 13300.0 0.91 197920.0 23000.0 1.71 1.8483 0.9559 3189692 BCB03_000566 CCCCCCC#C[Si](O[C@@H](c1cn(nn1)[C@H](CO)Cc2ccccc2)c3ccccc3)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M16 compound treatment 175440.0 -439.0 -0.03 175400.0 434.0 0.03 0.0017 0.038 3220669 BCB03_000567 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@H](Cn2cc(nn2)c3cncn3C)C(C)C)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M17 compound treatment 196080.0 20200.0 1.38 188800.0 13800.0 1.03 1.7019 0.9897 3189693 BCB03_000568 CCCCCCC#C[Si](O[C@@H](c1cn(Cc2cccc(Cl)c2)nn1)c3ccccc3)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M18 compound treatment 181960.0 6080.0 0.41 183920.0 8950.0 0.67 0.7644 0.9739 3414054 BCB03_000569 COC(=O)c1c(CC[C@@H](CO)NC(=O)N2CCC[C@H]2Cn3cc(nn3)c4ccccn4)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M19 compound treatment 196440.0 20600.0 1.4 192000.0 17000.0 1.27 1.8877 0.9987 3189694 BCB03_000570 CCCCCCC#C[Si](O[C@@H](c1cn(nn1)[C@H](C)c2ccccc2)c3ccccc3)(C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M20 compound treatment 178840.0 2960.0 0.2 179000.0 4030.0 0.3 0.355 0.9813 3414055 BCB03_000571 COC(=O)c1c(CC[C@@H](CO)NC(=O)N2CCC[C@H]2Cn3cc(Cc4ccccc4)nn3)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M21 compound treatment 183080.0 7200.0 0.49 176200.0 1230.0 0.09 0.4121 0.8251 3071395 BCB03_000572 CC(C)[Si](O[C@@H](c1cn(Cc2ccccc2)nn1)c3ccccc3)(C#CCCCC#N)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M22 compound treatment 169640.0 -6240.0 -0.43 171960.0 -3010.0 -0.22 -0.459 -0.955 3414056 BCB03_000573 COC(=O)c1c(CC[C@@H](CO)NC(=O)N2CCC[C@H]2Cn3cc(nn3)C4(O)CCCCC4)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M23 compound treatment 179720.0 3840.0 0.26 184520.0 9550.0 0.71 0.688 0.9079 3189697 BCB03_000574 CC(C)[Si](O[C@@H](c1cn(nn1)[C@H](CO)Cc2ccccc2)c3ccccc3)(C#CCCCC#N)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 M24 compound treatment 167280.0 -8600.0 -0.59 167160.0 -7810.0 -0.58 -0.8254 -1.0 3414057 BCB03_000575 CCCCc1cn(C[C@@H]2CCCN2C(=O)N[C@H](CO)CCc3oc(C(=O)C)c(C(=O)OC)c3C(=O)OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N01 compound treatment 180360.0 4480.0 0.31 177640.0 2670.0 0.2 0.3567 0.9785 3071585 BCB03_000576 OCCOCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N02 compound treatment 186440.0 10600.0 0.72 186320.0 11400.0 0.85 1.1067 0.9968 3215882 BCB03_000577 CCCC[C@H]1OB(O)C[C@H]2C1=C(COC)Cn3n2c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N03 compound treatment 184800.0 8920.0 0.61 182840.0 7870.0 0.59 0.8445 0.9998 3188130 BCB03_000578 OCCCCCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N04 compound treatment 204520.0 28600.0 1.95 202880.0 27900.0 2.08 2.8498 0.9995 3215880 BCB03_000579 CCCC[C@H]1OB(O)C[C@H]2C1=C(COc3ccccc3)Cn4n2c(=O)n(c5ccccc5)c4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N05 compound treatment 185720.0 9840.0 0.67 183760.0 8790.0 0.65 0.9372 0.9999 3071587 BCB03_000580 OCCCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N06 compound treatment 355480.0 180000.0 12.24 359840.0 185000.0 13.76 18.3878 0.9983 3188542 BCB03_000581 CC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2[C@H]4[C@@H](C1)C(=O)C=CC4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N07 compound treatment 183800.0 7920.0 0.54 182760.0 7790.0 0.58 0.792 0.9994 3071588 BCB03_000582 BrC1=C[C@H]2[C@H](C[C@@H]1[C@@]3(CO3)C2=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N08 compound treatment 183680.0 7800.0 0.53 179720.0 4750.0 0.35 0.6263 0.9804 3071661 BCB03_000583 COCC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2[C@H]4[C@@H](C1)C(=O)N(Cc5ccccc5)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N09 mock treatment 186240.0 10400.0 0.71 181640.0 6670.0 0.5 0.8507 0.9852 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N10 mock treatment 184280.0 8400.0 0.57 180280.0 5310.0 0.4 0.6847 0.9837 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N11 compound treatment 211560.0 35700.0 2.43 212480.0 37500.0 2.79 3.6944 0.9976 3071589 BCB03_000584 Cc1cccc(c1)[C@H]2C[C@H]3C(=C[C@@H]2C(=O)[C@@]43CO4)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N12 compound treatment 384920.0 209000.0 14.25 383360.0 208000.0 15.51 21.0448 0.9991 3188543 BCB03_000585 COCC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2[C@H]4[C@@H](C1)C(=O)C=CC4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N13 mock treatment 180920.0 5040.0 0.34 184280.0 9310.0 0.69 0.7332 0.9476 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N14 mock treatment 181840.0 5960.0 0.41 180760.0 5790.0 0.43 0.5923 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N15 compound treatment 205720.0 29800.0 2.03 201040.0 26100.0 1.94 2.8108 0.9997 3071590 BCB03_000586 COc1ccc(cc1)[C@H]2C[C@H]3C(=C[C@@H]2C(=O)[C@@]43CO4)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N16 compound treatment 318320.0 142000.0 9.71 321120.0 146000.0 10.88 14.5586 0.9984 3070948 BCB03_000587 OB1C[C@@H]2[C@H]3[C@@H](CC(=C2[C@@H](CCc4ccccc4)O1)COc5ccccc5)C(=O)C=CC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N17 compound treatment 186200.0 10300.0 0.7 184600.0 9630.0 0.72 1.0046 1.0 3071591 BCB03_000588 CO[C@@]1(C=C(Br)[C@@H]2C[C@@H]1c3ccccc3)C(=O)[C@@]42CO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N18 compound treatment 388400.0 213000.0 14.49 384080.0 209000.0 15.56 21.2505 0.9994 3070949 BCB03_000589 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)C)C(=O)C=CC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N19 compound treatment 187520.0 11600.0 0.79 188760.0 13800.0 1.03 1.2871 0.9919 3188261 BCB03_000590 CO[C@@]1(C=C(Br)[C@@H]2C[C@@H]1c3cccc(C)c3)C(=O)[C@@]42CO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N20 compound treatment 334360.0 158000.0 10.8 325920.0 151000.0 11.24 15.5845 0.9998 3070950 BCB03_000591 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)COC)C(=O)C=CC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N21 compound treatment 182400.0 6520.0 0.44 180280.0 5310.0 0.4 0.594 0.9983 3071600 BCB03_000592 COc1ccc(cc1)[C@H]2C[C@H]3C(=C[C@]2(OC)C(=O)[C@@]43CO4)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N22 compound treatment 299920.0 124000.0 8.46 306600.0 132000.0 9.8 12.9074 0.9973 3070951 BCB03_000593 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)COc4ccccc4)C(=O)C=CC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N23 compound treatment 171960.0 -3920.0 -0.27 171560.0 -3410.0 -0.25 -0.3682 -0.9997 3071601 BCB03_000594 OCCOCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 N24 compound treatment 196160.0 20300.0 1.38 202240.0 27300.0 2.03 2.4131 0.9825 3071664 BCB03_000595 OB1C[C@@H]2[C@H]3[C@@H](CC(=C2[C@@H](CCc4ccccc4)O1)COc5ccccc5)C(=O)N(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O01 compound treatment 191000.0 15100.0 1.03 187680.0 12700.0 0.95 1.3981 0.9991 3187592 BCB03_000596 CC(C)[Si](O[C@@H](c1cn(Cc2cccc(Cl)c2)nn1)c3ccccc3)(C#CCCCC#N)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O02 compound treatment 176360.0 481.0 0.03 173720.0 -1250.0 -0.09 -0.0424 -0.4311 3220705 BCB03_000597 CCc1oc(CC[C@@H](CO)NC(=O)NCCn2cc(nn2)C3(O)CCCCC3)c(C(=O)OC)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O03 compound treatment 186200.0 10300.0 0.7 186640.0 11700.0 0.87 1.1119 0.9945 3071397 BCB03_000598 CC(C)[Si](O[C@@H](c1cn(nn1)[C@H](C)c2ccccc2)c3ccccc3)(C#CCCCC#N)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O04 compound treatment 180600.0 4720.0 0.32 173280.0 -1690.0 -0.13 0.1389 0.402 3220708 BCB03_000599 COC(=O)c1c(CC[C@@H](CO)NC(=O)NCCn2cc(nn2)C3(O)CCCC3)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O05 compound treatment 189640.0 13800.0 0.94 188880.0 13900.0 1.04 1.3957 0.9988 3071398 BCB03_000600 CC(C)[Si](O[C@H](C)c1cn(Cc2ccccc2)nn1)(C#C[Si](C(C)C)(C(C)C)C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O06 compound treatment 181880.0 6000.0 0.41 184920.0 9950.0 0.74 0.8132 0.9608 3220711 BCB03_000601 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@H](Cc2ccccc2)Cn3cc(nn3)c4ccccn4)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O07 compound treatment 197560.0 21700.0 1.48 200280.0 25300.0 1.88 2.3774 0.9928 3071399 BCB03_000602 CC(C)[Si](O[C@H](C)c1cn(nn1)[C@H](CO)Cc2ccccc2)(C#C[Si](C(C)C)(C(C)C)C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O08 compound treatment 185840.0 9960.0 0.68 184720.0 9750.0 0.73 0.9935 0.9994 3220713 BCB03_000603 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@H](Cc2ccccc2)Cn3cc(nn3)c4ccccc4N)oc(C(=O)C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O09 compound treatment 194400.0 18500.0 1.26 194520.0 19600.0 1.46 1.9219 0.9975 3187596 BCB03_000604 CC(C)[Si](O[C@H](C)c1cn(Cc2cccc(Cl)c2)nn1)(C#C[Si](C(C)C)(C(C)C)C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O10 compound treatment 178280.0 2400.0 0.16 177480.0 2510.0 0.19 0.2481 0.9978 3220715 BCB03_000605 COC(=O)c1cn(C[C@@H](Cc2ccccc2)NC(=O)N[C@H](CO)CCc3oc(C(=O)C)c(C(=O)OC)c3C(=O)OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O11 mock treatment 177680.0 1800.0 0.12 175560.0 594.0 0.04 0.1181 0.9049 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O12 mock treatment 177480.0 1600.0 0.11 180280.0 5310.0 0.4 0.3568 0.8697 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O13 compound treatment 193240.0 17400.0 1.18 200400.0 25400.0 1.89 2.1755 0.9744 3071400 BCB03_000606 CC(C)[Si](O[C@H](C)c1cn(nn1)[C@H](C)c2ccccc2)(C#C[Si](C(C)C)(C(C)C)C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O14 compound treatment 176920.0 1040.0 0.07 173040.0 -1930.0 -0.14 -0.0512 -0.32 3220717 BCB03_000607 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](Cc2ccccc2)Cn3cc(nn3)c4ccccc4)oc(C(=O)N5CCOCC5)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O15 compound treatment 180960.0 5080.0 0.35 177560.0 2590.0 0.19 0.3815 0.9619 3070694 BCB03_000608 COc1ccc(cn1)c2cc3CO[Si](C(C)C)(C(C)C)c3c(Cc4ccccc4)n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O16 compound treatment 176040.0 161.0 0.01 179480.0 4510.0 0.34 0.2453 0.7298 3220739 BCB03_000609 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](Cc2ccccc2)Cn3cc(nn3)c4ccccn4)oc(C(=O)N5CCOCC5)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O17 compound treatment 184360.0 8480.0 0.58 179520.0 4550.0 0.34 0.6485 0.9676 3070746 BCB03_000610 COc1c(C)cc(cc1C)c2cc3CO[Si](C(C)C)(C(C)C)c3c(Cc4ccccc4)n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O18 compound treatment 177840.0 1960.0 0.13 180200.0 5230.0 0.39 0.37 0.8983 3220741 BCB03_000611 COC(=O)c1c(CC[C@@H](CO)NC(=O)N[C@@H](Cc2ccccc2)Cn3cc(nn3)C4(O)CCCC4)oc(C(=O)N5CCOCC5)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O19 compound treatment 185400.0 9520.0 0.65 192120.0 17200.0 1.28 1.3618 0.9508 3188534 BCB03_000612 COC(=O)[C@H](Cc1ccccc1)N2CC3=CCCC=C[C@@H]3[C@H]2[C@H](O)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O20 compound treatment 178840.0 2960.0 0.2 180320.0 5350.0 0.4 0.4245 0.9503 3220743 BCB03_000613 COCc1cn(C[C@H](Cc2ccccc2)NC(=O)N[C@H](CO)CCc3oc(C(=O)N4CCOCC4)c(C(=O)OC)c3C(=O)OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O21 compound treatment 177840.0 1960.0 0.13 180480.0 5510.0 0.41 0.3847 0.8913 3188535 BCB03_000614 COC(=O)[C@H](Cc1ccccc1)N2CC(=C)[C@H](/C=C/C=C)[C@H]2[C@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O22 compound treatment 169120.0 -6760.0 -0.46 173080.0 -1890.0 -0.14 -0.4251 -0.8824 3188660 BCB03_000615 COC(=O)[C@H](Cc1ccccc1)N[C@H](/C=C/C2CC2)[C@@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O23 compound treatment 175720.0 -159.0 -0.01 178800.0 3830.0 0.29 0.1941 0.6797 3188536 BCB03_000616 O=C1O[C@H](Cc2ccccc2)[C@H](/C=C/C3CC3)N(CC#C)[C@H]1Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 O24 compound treatment 181040.0 5160.0 0.35 192680.0 17700.0 1.32 1.181 0.8655 3188661 BCB03_000617 COC(=O)[C@H](Cc1ccccc1)N(CC#C)[C@H](/C=C/C2CC2)[C@@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P01 compound treatment 181760.0 5880.0 0.4 182880.0 7910.0 0.59 0.7 0.9824 3071602 BCB03_000618 OCCCCCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P02 compound treatment 178440.0 2560.0 0.17 176640.0 1670.0 0.12 0.2116 0.9863 3071666 BCB03_000619 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)C)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P03 compound treatment 182520.0 6640.0 0.45 176440.0 1470.0 0.11 0.3977 0.8538 3071603 BCB03_000620 OCCCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P04 compound treatment 187400.0 11500.0 0.79 180760.0 5790.0 0.43 0.8603 0.9601 3071711 BCB03_000621 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)COC)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P05 compound treatment 201520.0 25600.0 1.75 197440.0 22500.0 1.67 2.4189 0.9998 3071604 BCB03_000622 CCCCO[C@H]1C[C@H]2C(=C[C@@H]1C(=O)[C@@]32CO3)I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P06 compound treatment 203480.0 27600.0 1.88 205760.0 30800.0 2.29 2.9512 0.9952 3071776 BCB03_000623 CCCC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)COc4ccccc4)C(=O)N(Cc5ccccc5)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P07 compound treatment 216200.0 40300.0 2.75 213880.0 38900.0 2.9 3.9918 0.9997 3071651 BCB03_000624 IC1=C[C@H]2[C@H](C[C@@H]1[C@@]3(CO3)C2=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P08 compound treatment 177880.0 2000.0 0.14 179560.0 4590.0 0.34 0.3382 0.9188 3188405 BCB03_000625 CN1C(=O)[C@@H]2CC(=C3[C@@H](CCc4ccccc4)OB(O)C[C@@H]3[C@@H]2C1=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P09 compound treatment 206560.0 30700.0 2.09 203480.0 28500.0 2.12 2.9797 1.0 3071652 BCB03_000626 Cc1cccc(c1)[C@H]2C[C@H]3C(=C[C@@H]2C(=O)[C@@]43CO4)I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P10 compound treatment 194680.0 18800.0 1.28 195000.0 20000.0 1.49 1.9607 0.9972 3070929 BCB03_000627 COCC1=C2[C@@H](CCc3ccccc3)OB(O)C[C@@H]2[C@H]4[C@@H](C1)C(=O)N(C)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P11 mock treatment 172480.0 -3400.0 -0.23 172920.0 -2050.0 -0.15 -0.2715 -0.9792 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P12 mock treatment 176800.0 921.0 0.06 176640.0 1670.0 0.12 0.1325 0.9496 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P13 compound treatment 188520.0 12600.0 0.86 186400.0 11400.0 0.85 1.2111 1.0 3071653 BCB03_000628 COc1ccc(cc1)[C@H]2C[C@H]3C(=C[C@@H]2C(=O)[C@@]43CO4)I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P14 compound treatment 184800.0 8920.0 0.61 184520.0 9550.0 0.71 0.9329 0.997 3188406 BCB03_000629 CN1C(=O)[C@@H]2CC(=C3[C@@H](CCc4ccccc4)OB(O)C[C@@H]3[C@@H]2C1=O)COc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P15 compound treatment 181560.0 5680.0 0.39 178160.0 3190.0 0.24 0.442 0.9725 3188268 BCB03_000630 CCCCO[C@H]1C[C@H]2C(=C[C@]1(CO)C(=O)[C@@]32CO3)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P16 compound treatment 174800.0 -1080.0 -0.07 177680.0 2710.0 0.2 0.0908 0.4224 3070998 BCB03_000631 CC1=C([C@H](O)CCc2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P17 compound treatment 177000.0 1120.0 0.08 174160.0 -806.0 -0.06 0.0116 0.1197 3071714 BCB03_000632 OC[C@@]1(C=C(Br)[C@@H]2C[C@@H]1c3ccccc3)C(=O)[C@@]42CO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P18 compound treatment 174920.0 -959.0 -0.07 175880.0 914.0 0.07 0.0019 0.0198 3188793 BCB03_000633 CCCC[C@@H](O)C1=C(C)C[C@@H]2[C@H]([C@H]1CO)C(=O)N(C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P19 compound treatment 183000.0 7120.0 0.49 181240.0 6270.0 0.47 0.6735 0.9998 3071715 BCB03_000634 Cc1cccc(c1)[C@H]2C[C@H]3C(=C[C@]2(CO)C(=O)[C@@]43CO4)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P20 compound treatment 174520.0 -1360.0 -0.09 170440.0 -4530.0 -0.34 -0.3037 -0.8694 3071118 BCB03_000635 CCCC[C@@H](O)C1=C(COC)C[C@@H]2[C@H]([C@H]1CO)C(=O)N(C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P21 compound treatment 175520.0 -359.0 -0.02 175920.0 954.0 0.07 0.0329 0.4379 3071717 BCB03_000636 COc1ccc(cc1)[C@H]2C[C@H]3C(=C[C@]2(CO)C(=O)[C@@]43CO4)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P22 compound treatment 173360.0 -2520.0 -0.17 174000.0 -966.0 -0.07 -0.1723 -0.9253 3071120 BCB03_000637 CCCC[C@@H](O)C1=C(COc2ccccc2)C[C@@H]3[C@H]([C@H]1CO)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P23 compound treatment 263280.0 87400.0 5.96 257120.0 82200.0 6.11 8.537 0.9999 3071720 BCB03_000638 BrC1=C[C@]23COC[C@H]3C[C@@H]1[C@@]4(CO4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2282 P24 compound treatment 172520.0 -3360.0 -0.23 171960.0 -3010.0 -0.22 -0.3201 -0.9999 3188808 BCB03_000639 CC1=C([C@H](O)CCc2ccccc2)[C@H](CO)n3n(C1)c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A01 compound treatment 179680.0 5360.0 0.37 175200.0 1310.0 0.1 0.3274 0.866 3188923 BCB03_000640 COCC1=C([C@H](O)CCc2ccccc2)[C@H](CO)n3n(C1)c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A02 compound treatment 171640.0 -2680.0 -0.18 170320.0 -3570.0 -0.27 -0.317 -0.9835 3563114 BCB03_000641 COC(=O)C1=CN(Cc2ccc(OC)cc2)C(C)c3ccccc3C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A03 compound treatment 186480.0 12200.0 0.83 172280.0 -1610.0 -0.12 0.5015 0.599 3071127 BCB03_000642 OC[C@H]1C(=C(COc2ccccc2)Cn3n1c(=O)n(c4ccccc4)c3=O)[C@H](O)CCc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A04 compound treatment 172120.0 -2200.0 -0.15 164680.0 -9210.0 -0.69 -0.5907 -0.8422 3563115 BCB03_000643 CCOC(=O)C1=C2C(ON1)N(Cc3ccc(OC)cc3)C(C)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A05 compound treatment 165440.0 -8880.0 -0.61 163080.0 -10800.0 -0.8 -0.9969 -0.9902 3071425 BCB03_000644 CCCC[C@@H](O)C1=C(C)Cn2n([C@H]1CO)c(=O)n(c3ccccc3)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A06 compound treatment 194360.0 20000.0 1.37 195000.0 21100.0 1.57 2.0771 0.9976 3563116 BCB03_000645 COc1ccc(CN/2C(C)c3ccccc3C\C2=N\P(=O)(Oc4ccccc4)Oc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A07 compound treatment 166600.0 -7720.0 -0.53 165640.0 -8250.0 -0.61 -0.8063 -0.9971 3215868 BCB03_000646 CCCC[C@@H](O)C1=C(COC)Cn2n([C@H]1CO)c(=O)n(c3ccccc3)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A08 compound treatment 171320.0 -3000.0 -0.2 167840.0 -6050.0 -0.45 -0.463 -0.9365 3563118 BCB03_000647 COc1ccc(CN2CCc3ccccc3C2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A09 compound treatment 163200.0 -11100.0 -0.76 162080.0 -11800.0 -0.88 -1.1576 -0.9973 3215866 BCB03_000648 CCCC[C@@H](O)C1=C(COc2ccccc2)Cn3n([C@H]1CO)c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A10 compound treatment 169680.0 -4640.0 -0.32 166880.0 -7010.0 -0.52 -0.5926 -0.9714 3563119 BCB03_000649 COC(=O)C1=CN(Cc2ccc(OC)cc2)C(C=C)c3ccccc3C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A11 compound treatment 164520.0 -9800.0 -0.67 164960.0 -8930.0 -0.66 -0.9424 -1.0 3070999 BCB03_000650 COCC1=C([C@H](O)CCc2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A12 compound treatment 184760.0 10400.0 0.71 176120.0 2230.0 0.17 0.6207 0.8495 3563120 BCB03_000651 CCOC(=O)C1=C2C(ON1)N(Cc3ccc(OC)cc3)C(C=C)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A13 mock treatment 166280.0 -8040.0 -0.55 159160.0 -14700.0 -1.1 -1.1627 -0.9488 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A14 mock treatment 161560.0 -12800.0 -0.87 164640.0 -9250.0 -0.69 -1.1019 -0.9932 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A15 compound treatment 195080.0 20800.0 1.42 185720.0 11800.0 0.88 1.6234 0.974 3071000 BCB03_000652 OC[C@@H]1[C@H]2[C@@H](CC(=C1[C@H](O)CCc3ccccc3)COc4ccccc4)C(=O)N(Cc5ccccc5)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A16 compound treatment 210800.0 36500.0 2.49 195200.0 21300.0 1.59 2.8802 0.9764 3563121 BCB03_000653 COc1ccc(CN/2C(C=C)c3ccccc3C\C2=N\P(=O)(Oc4ccccc4)Oc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A17 compound treatment 166320.0 -8000.0 -0.55 167040.0 -6850.0 -0.51 -0.7461 -0.9994 3188676 BCB03_000654 CCCC[C@@H](O)C1=C(C)C[C@@H]2[C@H]([C@H]1CO)C(=O)N(Cc3ccccc3)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A18 compound treatment 175200.0 876.0 0.06 178320.0 4430.0 0.33 0.2756 0.8217 3563123 BCB03_000655 COc1ccc(CN2CCc3ccccc3C2C=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A19 compound treatment 169680.0 -4640.0 -0.32 166760.0 -7130.0 -0.53 -0.5989 -0.9696 3188677 BCB03_000656 CCCC[C@@H](O)C1=C(COC)C[C@@H]2[C@H]([C@H]1CO)C(=O)N(Cc3ccccc3)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A20 compound treatment 178040.0 3720.0 0.25 173560.0 -325.0 -0.02 0.162 0.6366 3563124 BCB03_000657 COC(=O)C1=CN(Cc2ccc(OC)cc2)C(C3CC3)c4ccccc4C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A21 compound treatment 193080.0 18800.0 1.28 182080.0 8190.0 0.61 1.3355 0.9426 3188788 BCB03_000658 CCCC[C@@H](O)C1=C(COc2ccccc2)C[C@@H]3[C@H]([C@H]1CO)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A22 compound treatment 167160.0 -7160.0 -0.49 166080.0 -7810.0 -0.58 -0.7561 -0.9963 3563125 BCB03_000659 CCOC(=O)C1=C2C(ON1)N(Cc3ccc(OC)cc3)C(C4CC4)c5ccccc25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A23 compound treatment 172120.0 -2200.0 -0.15 164160.0 -9730.0 -0.72 -0.6181 -0.8361 3071005 BCB03_000660 CN1C(=O)[C@@H]2CC(=C([C@H](O)CCc3ccccc3)[C@H](CO)[C@@H]2C1=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 A24 compound treatment 211120.0 36800.0 2.51 202880.0 29000.0 2.16 3.2998 0.9972 3563121 BCB03_000661 COc1ccc(CN/2C(C=C)c3ccccc3C\C2=N\P(=O)(Oc4ccccc4)Oc5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B01 compound treatment 176320.0 2000.0 0.14 165040.0 -8850.0 -0.66 -0.3693 -0.5493 3216005 BCB03_000662 CN1C(=O)[C@@H]2C[C@]/3(C)OC[C@H]([C@@H]2C1=O)\C3=C/c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B02 compound treatment 172720.0 -1600.0 -0.11 175880.0 1990.0 0.15 0.0277 0.15 3614372 BCB03_000663 CCCNc1ncnc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B03 compound treatment 190160.0 15800.0 1.08 186800.0 12900.0 0.96 1.4431 0.9983 3216013 BCB03_000664 CN1C(=O)[C@@H]2C[C@]/3(COc4ccccc4)OC[C@H]([C@@H]2C1=O)\C3=C/c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B04 compound treatment 158880.0 -15400.0 -1.05 157840.0 -16000.0 -1.19 -1.589 -0.998 3614373 BCB03_000665 CC(C)(C)OC(=O)NCCOCCOCCNc1ncnc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B05 compound treatment 196920.0 22600.0 1.54 177000.0 3110.0 0.23 1.2532 0.8045 3614374 BCB03_000666 C[C@]1(C[C@@H]2[C@H]([C@H]/3CO1)C(=O)N(Cc4ccccc4)C2=O)\C3=C\c5cccc(COC(=O)NCc6cccc(Cl)c6)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B06 compound treatment 208960.0 34600.0 2.36 200560.0 26700.0 1.99 3.0736 0.9963 3614376 BCB03_000667 CC(C)(C)OC(=O)NCCOCCOCCNC(=O)c1ccc(NC(=S)Nc2ccc(Nc3ccccc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B07 compound treatment 187360.0 13000.0 0.89 182160.0 8270.0 0.62 1.0639 0.9839 3614378 BCB03_000668 C[C@]1(C[C@@H]2[C@H]([C@H]/3CO1)C(=O)N(Cc4ccccc4)C2=O)\C3=C\c5cccc(COC(=O)NCC#C)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B08 compound treatment 180000.0 5680.0 0.39 174160.0 275.0 0.02 0.2881 0.7434 3614380 BCB03_000669 Oc1ccc2ncnc(NCc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B09 compound treatment 217360.0 43000.0 2.93 213480.0 39600.0 2.95 4.1585 1.0 3614381 BCB03_000670 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)c4cn(C[C@@H](Cc5ccccc5)NC(=O)c6oc(CC[C@H](CO)NC(=O)N[C@H](Cc7ccccc7)c8cn(C[C@@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B10 compound treatment 228760.0 54400.0 3.71 224520.0 50600.0 3.77 5.2891 1.0 3614383 BCB03_000671 ONC(=O)/C=C/c1ccc(OCCc2cccs2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B11 compound treatment 276880.0 103000.0 6.99 280760.0 107000.0 7.95 10.5686 0.9979 3614385 BCB03_000672 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)c4cn(C[C@@H](Cc5ccccc5)NC(=O)c6oc(CC[C@H](CO)NC(=O)N[C@@H](Cc7ccccc7)c8cn(C[C@@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B12 compound treatment 254600.0 80300.0 5.47 259920.0 86000.0 6.4 8.3978 0.9969 3614386 BCB03_000673 ONC(=O)/C=C/c1ccc(OCc2ccc-3c(Cc4ccccc43)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B13 mock treatment 167720.0 -6600.0 -0.45 164400.0 -9490.0 -0.71 -0.8176 -0.9764 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B14 mock treatment 165720.0 -8600.0 -0.59 166720.0 -7170.0 -0.53 -0.7919 -0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B15 compound treatment 302400.0 128000.0 8.73 290680.0 117000.0 8.69 12.321 1.0 3614388 BCB03_000674 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@H](Cc3ccccc3)c4cn(C[C@H](Cc5ccccc5)NC(=O)c6oc(CC[C@@H](CO)NC(=O)N[C@H](Cc7ccccc7)c8cn(C[C@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B16 compound treatment 238600.0 64300.0 4.38 221040.0 47200.0 3.51 5.5803 0.9939 3614389 BCB03_000675 ONC(=O)/C=C/c1ccc(OCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B17 compound treatment 290640.0 116000.0 7.93 275720.0 102000.0 7.58 10.9667 0.9997 3614391 BCB03_000676 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@@H](Cc3ccccc3)c4cn(C[C@H](Cc5ccccc5)NC(=O)c6oc(CC[C@@H](CO)NC(=O)N[C@@H](Cc7ccccc7)c8cn(C[C@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B18 compound treatment 255360.0 81000.0 5.52 262320.0 88400.0 6.58 8.5607 0.9962 3614392 BCB03_000677 ONC(=O)/C=C/c1ccc(OCc2ccc(Cl)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B19 compound treatment 191640.0 17300.0 1.18 183360.0 9470.0 0.71 1.3334 0.9697 3556401 BCB03_000678 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)c4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B20 compound treatment 214520.0 40200.0 2.74 205520.0 31600.0 2.35 3.6026 0.9971 3614394 BCB03_000679 Nc1cccc(COc2ccc(/C=C/C(=O)NO)cc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B21 compound treatment 175640.0 1320.0 0.09 161920.0 -12000.0 -0.89 -0.5663 -0.6327 3556405 BCB03_000680 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)c4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B22 compound treatment 236360.0 62000.0 4.23 217560.0 43700.0 3.25 5.2892 0.9915 3614396 BCB03_000681 ONC(=O)/C=C/c1ccc(OCCCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B23 compound treatment 189520.0 15200.0 1.04 179200.0 5310.0 0.4 1.0123 0.9128 3556409 BCB03_000682 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)c4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 B24 compound treatment 212440.0 38100.0 2.6 197520.0 23600.0 1.76 3.0814 0.9819 3614398 BCB03_000683 ONC(=O)/C=C/c1ccc(OCCCCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C01 compound treatment 164520.0 -9800.0 -0.67 171360.0 -2530.0 -0.19 -0.6055 -0.8721 3188790 BCB03_000684 COCC1=C([C@H](O)CCc2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C02 compound treatment 162320.0 -12000.0 -0.82 166680.0 -7210.0 -0.54 -0.9579 -0.979 3563126 BCB03_000685 COC(=O)C1=CN(Cc2ccc(OC)cc2)C(C)C=C(C)C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C03 compound treatment 181400.0 7080.0 0.48 168840.0 -5050.0 -0.38 0.0756 0.1237 3188791 BCB03_000686 CN1C(=O)[C@@H]2CC(=C([C@H](O)CCc3ccccc3)[C@H](CO)[C@@H]2C1=O)COc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C04 compound treatment 217440.0 43100.0 2.94 193960.0 20100.0 1.49 3.135 0.9507 3563127 BCB03_000687 COc1ccc(CN/2C(C)C=C(C)C\C2=N\P(=O)(Oc3ccccc3)Oc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C05 compound treatment 186600.0 12300.0 0.84 168520.0 -5370.0 -0.4 0.3094 0.3337 3071437 BCB03_000688 OB1OC(CCc2ccccc2)CC=C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C06 compound treatment 169760.0 -4560.0 -0.31 162520.0 -11400.0 -0.85 -0.8182 -0.9077 3563129 BCB03_000689 COc1ccc(CN2C(C)C3C4C(C2C=C3C)C(=O)N(C)C4=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C07 compound treatment 215400.0 41100.0 2.8 198880.0 25000.0 1.86 3.2956 0.9803 3071483 BCB03_000690 COC(=O)c1ccc(OC)c(/C=C\CC(OC(=O)c2ccncc2)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C08 compound treatment 172360.0 -1960.0 -0.13 161720.0 -12200.0 -0.91 -0.7349 -0.8029 3563130 BCB03_000691 COc1ccc(CN2CCC(=CC2C)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C09 compound treatment 166120.0 -8200.0 -0.56 163760.0 -10100.0 -0.75 -0.9284 -0.9892 3071486 BCB03_000692 CC(=O)OC(C/C=C\B1OC(C)(C)C(C)(C)O1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C10 compound treatment 174880.0 556.0 0.04 169880.0 -4010.0 -0.3 -0.184 -0.6123 3563131 BCB03_000693 COC(=O)C1=CN(Cc2ccc(OC)cc2)C(C=C)C=C(C)C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C11 mock treatment 172400.0 -1920.0 -0.13 166280.0 -7610.0 -0.57 -0.493 -0.8485 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C12 mock treatment 169960.0 -4360.0 -0.3 169040.0 -4850.0 -0.36 -0.4654 -0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C13 compound treatment 483440.0 309000.0 21.07 475040.0 301000.0 22.41 30.7511 0.9995 3188011 BCB03_000694 O=C1C=C(C(=O)c2ccc(cc12)[C@H]3Oc4ccccc4S(=O)(=O)N5CCC[C@@H]35)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C14 compound treatment 220720.0 46400.0 3.16 203680.0 29800.0 2.22 3.8047 0.9849 3563132 BCB03_000695 COc1ccc(CN/2C(C=C)C=C(C)C\C2=N\P(=O)(Oc3ccccc3)Oc4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C15 mock treatment 172800.0 -1520.0 -0.1 173640.0 -245.0 -0.02 -0.0864 -0.8188 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C16 mock treatment 166120.0 -8200.0 -0.56 170720.0 -3170.0 -0.24 -0.5621 -0.9261 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C17 compound treatment 288680.0 114000.0 7.8 258040.0 84200.0 6.26 9.9418 0.9941 3071579 BCB03_000696 O=C1C=C(C(=O)C2=C1CC(=CC2)[C@H]3Oc4ccccc4S(=O)(=O)N5CCC[C@@H]35)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C18 compound treatment 175920.0 1600.0 0.11 168400.0 -5490.0 -0.41 -0.2117 -0.5011 3563134 BCB03_000697 COc1ccc(CN2C(C=C)C3C4C(C2C=C3C)C(=O)N(C)C4=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C19 compound treatment 171440.0 -2880.0 -0.2 165800.0 -8090.0 -0.6 -0.5645 -0.8917 3070932 BCB03_000698 OCC(NC(=O)OCC1c2ccccc2-c3ccccc13)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C20 compound treatment 174960.0 636.0 0.04 165880.0 -8010.0 -0.6 -0.3906 -0.6539 3563135 BCB03_000699 COc1ccc(CN2CCC(=CC2C=C)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C21 compound treatment 168560.0 -5760.0 -0.39 167520.0 -6370.0 -0.47 -0.6129 -0.9957 3188522 BCB03_000700 COc1ccc(CN([C@H](COC(=O)OC(C)(C)C)C=C)S(=O)(=O)c2ccc(Br)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C22 compound treatment 170800.0 -3520.0 -0.24 168720.0 -5170.0 -0.38 -0.4417 -0.9744 1025568 BCB03_000701 COc1cc2CCN(C)C(C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C23 compound treatment 159160.0 -15200.0 -1.03 166160.0 -7730.0 -0.57 -1.1376 -0.9617 3070934 BCB03_000702 CC(=O)OCC(NS(=O)(=O)c1ccc(Br)cc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 C24 compound treatment 162880.0 -11400.0 -0.78 162040.0 -11800.0 -0.88 -1.1751 -0.9981 3563136 BCB03_000703 COc1cc2CCN(C)C(C=C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D01 compound treatment 199160.0 24800.0 1.69 208840.0 35000.0 2.6 3.0369 0.9784 3556407 BCB03_000704 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)c4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D02 compound treatment 226440.0 52100.0 3.55 222760.0 48900.0 3.64 5.0846 0.9999 3614403 BCB03_000705 ONC(=O)/C=C/c1ccc(OCCn2c3ccccc3c4ccccc24)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D03 compound treatment 239920.0 65600.0 4.47 251320.0 77400.0 5.76 7.2375 0.9921 3556412 BCB03_000706 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@@H](Cc3ccccc3)c4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D04 compound treatment 167880.0 -6440.0 -0.44 168640.0 -5250.0 -0.39 -0.5867 -0.9983 3614405 BCB03_000707 Cc1cccc(Cl)c1NC(=O)C2=CC=C(Cl)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D05 compound treatment 245440.0 71100.0 4.85 233040.0 59200.0 4.4 6.5416 0.9988 3614406 BCB03_000708 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)C(=O)NCc4cn(C[C@@H](Cc5ccccc5)NC(=O)c6oc(CC[C@H](CO)NC(=O)N[C@H](Cc7ccccc7)C(=O)NCc8cn(C[C@@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D06 compound treatment 171360.0 -2960.0 -0.2 167560.0 -6330.0 -0.47 -0.4758 -0.9287 3614408 BCB03_000709 COc1ccc(CN(C(=O)C2=CC=C(Cl)C2)c3c(C)cccc3Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D07 compound treatment 224600.0 50300.0 3.43 213560.0 39700.0 2.95 4.5117 0.9972 3614409 BCB03_000710 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)C(=O)NCc4cn(C[C@H](Cc5ccccc5)NC(=O)c6oc(CC[C@H](CO)NC(=O)N[C@H](Cc7ccccc7)C(=O)NCc8cn(C[C@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D08 compound treatment 214440.0 40100.0 2.73 202840.0 29000.0 2.16 3.4577 0.993 3614410 BCB03_000711 COc1ccc(CN(C(=O)C2=CC=C(C2)Nc3cc(Cl)nc(C)n3)c4c(C)cccc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D09 compound treatment 207760.0 33400.0 2.28 202720.0 28800.0 2.15 3.1294 0.9995 3614411 BCB03_000712 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)C(=O)NCc4cn(C[C@@H](Cc5ccccc5)NC(=O)c6oc(CC[C@H](CO)NC(=O)N[C@@H](Cc7ccccc7)C(=O)NCc8cn(C[C@@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D10 compound treatment 193560.0 19200.0 1.31 192920.0 19000.0 1.42 1.9291 0.9993 3614412 BCB03_000713 Cc1cccc(Cl)c1NC(=O)C2=CC=C(C2)Nc3cc(Cl)nc(C)n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D11 mock treatment 161880.0 -12400.0 -0.85 163000.0 -10900.0 -0.81 -1.1728 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D12 mock treatment 164440.0 -9880.0 -0.67 173600.0 -285.0 -0.02 -0.4915 -0.729 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D13 compound treatment 271600.0 97300.0 6.63 260120.0 86200.0 6.42 9.2279 0.9999 3614413 BCB03_000714 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)C(=O)NCc4cn(C[C@H](Cc5ccccc5)NC(=O)c6oc(CC[C@H](CO)NC(=O)N[C@@H](Cc7ccccc7)C(=O)NCc8cn(C[C@H](Cc9ccccc9)NC2=O)nn8)c(C(=O)OC)c6C(=O)OC)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D14 compound treatment 207600.0 33300.0 2.27 218160.0 44300.0 3.3 3.9343 0.9834 3614414 BCB03_000715 Cc1cccc(Cl)c1NC(=O)c2cnc(Nc3cc(nc(C)n3)N4CCN(CCO)CC4)s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D15 mock treatment 166720.0 -7600.0 -0.52 167720.0 -6170.0 -0.46 -0.691 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D16 mock treatment 164600.0 -9720.0 -0.66 167360.0 -6530.0 -0.49 -0.8122 -0.9883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D17 compound treatment 170840.0 -3480.0 -0.24 161440.0 -12400.0 -0.93 -0.8229 -0.8606 3556423 BCB03_000716 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)C(=O)NCc4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D18 compound treatment 176320.0 2000.0 0.14 167240.0 -6650.0 -0.49 -0.2535 -0.4942 3614415 BCB03_000717 COC(=O)C1(CCCC1)C2CC(=C)[C@@H](/C=C/C=C)[C@@H]2[C@@H](O)CCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D19 compound treatment 184800.0 10500.0 0.71 165360.0 -8530.0 -0.63 0.0564 0.059 3556419 BCB03_000718 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@H](Cc3ccccc3)C(=O)NCc4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D20 compound treatment 182080.0 7760.0 0.53 177080.0 3190.0 0.24 0.542 0.9349 3614418 BCB03_000719 Cn1c(=O)n2[C@H]3[C@@H]4[C@H](CCN=[N+]=[N-])OC(=O)[C@H](Cc5ccccc5)N4CC3=C[C@@H](C6CC6)n2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D21 compound treatment 238680.0 64400.0 4.39 244080.0 70200.0 5.22 6.7967 0.9962 3614420 BCB03_000720 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)C(=O)NCc4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D22 compound treatment 204560.0 30200.0 2.06 198240.0 24400.0 1.81 2.7394 0.9979 3614421 BCB03_000721 [N-]=[N+]=NCC[C@@H]1OC(=O)[C@H](Cc2ccccc2)N3CC4=CCCC=C[C@H]4[C@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D23 compound treatment 167720.0 -6600.0 -0.45 163000.0 -10900.0 -0.81 -0.8912 -0.9616 3614424 BCB03_000722 COC(=O)c1cn(CC(=O)N2CCC3(CC2)N(CNC3=O)c4ccccc4)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 D24 compound treatment 185720.0 11400.0 0.78 182840.0 8950.0 0.67 1.0206 0.9971 3614425 BCB03_000723 [N-]=[N+]=NCC[C@@H]1OC(=O)[C@H](Cc2ccccc2)N3CC4=CC(=O)[C@H](C5CC5)[C@H]4[C@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E01 mock treatment 166760.0 -7560.0 -0.52 169640.0 -4250.0 -0.32 -0.5881 -0.9724 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E02 mock treatment 170040.0 -4280.0 -0.29 167160.0 -6730.0 -0.5 -0.5605 -0.9671 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E03 compound treatment 196400.0 22100.0 1.51 193640.0 19800.0 1.47 2.1039 0.9999 3070935 BCB03_000724 O=C(CCCCCCC(=O)Nc1ccccc1)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E04 compound treatment 173080.0 -1240.0 -0.08 170400.0 -3490.0 -0.26 -0.2434 -0.8918 3563137 BCB03_000725 COc1cc2CCN(C)C(C3CC3)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E05 compound treatment 172080.0 -2240.0 -0.15 173240.0 -645.0 -0.05 -0.1421 -0.8865 3070936 BCB03_000726 C/C(=N\O)/C(=O)NCCCCCNC(=O)OCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E06 compound treatment 183840.0 9520.0 0.65 181120.0 7230.0 0.54 0.8395 0.9957 3563138 BCB03_000727 COCC#CC1N(C)CCc2cc(OC)c(OC)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E07 compound treatment 174920.0 596.0 0.04 171960.0 -1930.0 -0.14 -0.0726 -0.4874 3070944 BCB03_000728 O/N=C(\Cc1ccccc1)/C(=O)NCCCCCNC(=O)OCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E08 compound treatment 174240.0 -83.9 -0.01 171880.0 -2010.0 -0.15 -0.1096 -0.7337 3562035 BCB03_000729 COc1ccc(C[N+]2=Cc3cc(OC)c(OC)cc3CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E09 mock treatment 173360.0 -964.0 -0.07 171040.0 -2850.0 -0.21 -0.1962 -0.8849 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E10 mock treatment 173760.0 -564.0 -0.04 173080.0 -805.0 -0.06 -0.0696 -0.977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E11 compound treatment 178240.0 3920.0 0.27 177160.0 3270.0 0.24 0.3611 0.999 3188539 BCB03_000730 C[C@@H]1ON([C@@H]([C@H]1C(=O)N2[C@H](Cc3ccccc3)COC2=O)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E12 compound treatment 179160.0 4840.0 0.33 177720.0 3830.0 0.29 0.4349 0.9974 3563139 BCB03_000731 COc1ccc(CN2CCc3cc(OC)c(OC)cc3C2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E13 compound treatment 204360.0 30000.0 2.05 200360.0 26500.0 1.97 2.8413 0.9998 3188540 BCB03_000732 C[C@H]1ON([C@H]([C@@H]1C(=O)N2[C@H](COC2=O)c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E14 compound treatment 178120.0 3800.0 0.26 180520.0 6630.0 0.49 0.5322 0.9546 3563140 BCB03_000733 COc1ccc(CN2CCc3cc(OC)c(OC)cc3C2C=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E15 compound treatment 184520.0 10200.0 0.7 184760.0 10900.0 0.81 1.0638 0.9971 3188541 BCB03_000734 C[C@@H]1ON([C@@H]([C@H]1C(=O)O)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E16 compound treatment 173520.0 -804.0 -0.05 175440.0 1550.0 0.12 0.0431 0.3363 3563141 BCB03_000735 COc1ccc(CN2CCc3cc(OC)c(OC)cc3C2C4CC4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E17 mock treatment 175120.0 796.0 0.05 172520.0 -1370.0 -0.1 -0.0335 -0.2906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E18 mock treatment 174880.0 556.0 0.04 174280.0 395.0 0.03 0.0476 0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E19 compound treatment 188960.0 14600.0 1.0 185040.0 11200.0 0.83 1.2926 0.9958 3070947 BCB03_000736 C[C@@H]1ON([C@@H]([C@H]1C(=O)N2[C@H](Cc3ccccc3)COC2=O)c4ccc(O)cc4)c5ccc(cc5)C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E20 compound treatment 174200.0 -124.0 -0.01 173240.0 -645.0 -0.05 -0.0399 -0.8189 3563142 BCB03_000737 COCC#CC1N(Cc2ccc(OC)cc2)CCc3cc(OC)c(OC)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E21 compound treatment 198600.0 24300.0 1.66 198080.0 24200.0 1.8 2.4436 0.9991 3188544 BCB03_000738 C[C@H]1ON([C@H]([C@@H]1C(=O)N2[C@H](COC2=O)c3ccccc3)c4ccc(O)cc4)c5ccc(cc5)C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E22 compound treatment 182720.0 8400.0 0.57 179960.0 6070.0 0.45 0.7245 0.9932 3563143 BCB03_000739 COc1cc2CCN(C)C(C)(C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E23 compound treatment 191800.0 17500.0 1.19 183080.0 9190.0 0.68 1.3264 0.9653 3188657 BCB03_000740 C[C@@H]1ON([C@@H]([C@H]1C(=O)N2[C@H](Cc3ccccc3)COC2=O)c4ccc(Br)cc4)c5cccc(c5)C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 E24 compound treatment 176720.0 2400.0 0.16 167000.0 -6890.0 -0.51 -0.2469 -0.4589 3563144 BCB03_000741 COc1cc2CCN(C)C(C)(C=C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F01 mock treatment 165800.0 -8520.0 -0.58 163560.0 -10300.0 -0.77 -0.9543 -0.9905 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F02 mock treatment 170600.0 -3720.0 -0.25 166880.0 -7010.0 -0.52 -0.5482 -0.9453 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F03 compound treatment 180240.0 5920.0 0.4 170200.0 -3690.0 -0.27 0.0913 0.1871 3614432 BCB03_000742 COC(=O)c1cn(C[C@@H](Cc2ccccc2)NC(=O)Nc3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F04 compound treatment 172040.0 -2280.0 -0.16 169920.0 -3970.0 -0.3 -0.3188 -0.9554 3614434 BCB03_000743 COC(=O)[C@H](Cc1ccccc1)N[C@H](/C=C/C2CC2)[C@@H](O)CCN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F05 compound treatment 175120.0 796.0 0.05 174680.0 795.0 0.06 0.0802 0.9991 3614437 BCB03_000744 COC(=O)c1cn(C[C@H](Cc2ccccc2)NC(=O)c3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F06 compound treatment 184280.0 9960.0 0.68 178960.0 5070.0 0.38 0.747 0.9617 3614440 BCB03_000745 [N-]=[N+]=NCC[C@@H]1OC(=O)[C@H](Cc2ccccc2)N(CC#C)[C@@H]1/C=C/C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F07 compound treatment 243080.0 68800.0 4.69 247720.0 73800.0 5.5 7.2004 0.9969 3614442 BCB03_000746 COC(=O)c1cn(CCCNC(=S)Nc2ccc(cc2)[N+](=O)[O-])nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F08 compound treatment 203320.0 29000.0 1.98 201960.0 28100.0 2.09 2.8754 0.9996 3614443 BCB03_000747 C=C/C=C/[C@H]1[C@@H]2[C@H](CCN=[N+]=[N-])OC(=O)[C@H](Cc3ccccc3)N2CC1=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F09 mock treatment 175160.0 836.0 0.06 175560.0 1670.0 0.12 0.1284 0.9371 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F10 mock treatment 169400.0 -4920.0 -0.34 171400.0 -2490.0 -0.18 -0.3682 -0.9606 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F11 compound treatment 183360.0 9040.0 0.62 173720.0 -165.0 -0.01 0.4269 0.6928 3614446 BCB03_000748 COC(=O)c1cn(CCCNC(=O)Nc2ccccc2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F12 compound treatment 195640.0 21300.0 1.45 181920.0 8030.0 0.6 1.4505 0.923 3614447 BCB03_000749 COC(=O)[C@H](Cc1ccccc1)N2C[C@](C)(OC(C)C)O[C@@H](CCN=[N+]=[N-])[C@H]2/C=C/C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F13 compound treatment 175840.0 1520.0 0.1 177600.0 3710.0 0.28 0.2686 0.91 3614451 BCB03_000750 COC(=O)c1cn(CCNC(=O)Nc2ccccc2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F14 compound treatment 190960.0 16600.0 1.13 188200.0 14300.0 1.07 1.5553 0.9995 3614452 BCB03_000751 COC(=O)C1(CCCC1)C2CC3=C[C@@H](C4CC4)n5n([C@H]3[C@@H]2[C@@H](O)CCO)c(=O)n(C)c5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F15 compound treatment 174920.0 596.0 0.04 183200.0 9310.0 0.69 0.5189 0.7473 3614455 BCB03_000752 COC(=O)c1cn(CCCNC(=O)[C@H](Cc2ccccc2)NS(=O)(=O)c3ccc(C)cc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F16 compound treatment 172440.0 -1880.0 -0.13 175640.0 1750.0 0.13 0.0015 0.0083 3614458 BCB03_000753 OCC[C@@H]1OC(=O)C2(CCCC2)N3CC4=CC(=O)[C@H](C5CC5)[C@H]4[C@H]13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F17 mock treatment 174400.0 76.1 0.01 173160.0 -725.0 -0.05 -0.0345 -0.6362 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F18 mock treatment 175560.0 1240.0 0.08 170320.0 -3570.0 -0.27 -0.128 -0.4599 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F19 compound treatment 184080.0 9760.0 0.67 180800.0 6910.0 0.51 0.8342 0.992 3614462 BCB03_000754 COC(=O)c1cn(CCNC(=O)[C@H](Cc2ccccc2)NS(=O)(=O)c3ccc(C)cc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F20 compound treatment 174520.0 196.0 0.01 175840.0 1950.0 0.15 0.1123 0.7688 3563105 BCB03_000755 COC(=O)C1=CN(C)C(C=C)c2ccccc2C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F21 compound treatment 170280.0 -4040.0 -0.28 169160.0 -4730.0 -0.35 -0.4436 -0.9927 3614464 BCB03_000756 COC(=O)c1cn(CCNC(=O)[C@@H](NS(=O)(=O)c2ccc(C)cc2)C(C)C)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F22 compound treatment 169160.0 -5160.0 -0.35 174840.0 955.0 0.07 -0.1987 -0.5532 3563108 BCB03_000757 COC(=O)C1=CN(C)C(C2CC2)c3ccccc3C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F23 compound treatment 173440.0 -884.0 -0.06 170880.0 -3010.0 -0.22 -0.2008 -0.8667 3614467 BCB03_000758 COC(=O)c1cn(C[C@@H]2CCCN2S(=O)(=O)c3ccc(C)cc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 F24 compound treatment 165800.0 -8520.0 -0.58 170040.0 -3850.0 -0.29 -0.6133 -0.9468 3188926 BCB03_000759 CC(C)CCC[C@@H](C)[C@H]1CC[C@@]2(C)C3=C(CC[C@]12C)[C@@]4(C)CC[C@H](OC(=O)c5ccc(nc5)C(F)(F)F)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G01 compound treatment 190120.0 15800.0 1.08 180520.0 6630.0 0.49 1.1107 0.9375 3188658 BCB03_000760 C[C@@H]1ON([C@@H]([C@H]1C(=O)N2[C@H](Cc3ccccc3)COC2=O)c4ccc(Br)cc4)c5ccc(cc5)C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G02 compound treatment 179200.0 4880.0 0.33 177360.0 3470.0 0.26 0.4179 0.9923 3563145 BCB03_000761 COCC#CC1(C)N(C)CCc2cc(OC)c(OC)cc21 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G03 mock treatment 175320.0 996.0 0.07 173720.0 -165.0 -0.01 0.0393 0.5697 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G04 mock treatment 181880.0 7560.0 0.52 175120.0 1230.0 0.09 0.4292 0.8203 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G05 compound treatment 217720.0 43400.0 2.96 219240.0 45400.0 3.38 4.479 0.9978 3188659 BCB03_000762 C[C@@H]1ON([C@@H]([C@H]1C(=O)N2[C@H](Cc3ccccc3)COC2=O)c4cccc(NC(=O)OCC5c6ccccc6-c7ccccc57)c4)c8ccc(I)cc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G06 compound treatment 183920.0 9600.0 0.65 182320.0 8430.0 0.63 0.9065 0.9998 3563146 BCB03_000763 COc1ccc(C[N+]2=C(C)c3cc(OC)c(OC)cc3CC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G07 compound treatment 217760.0 43400.0 2.96 219120.0 45200.0 3.37 4.4746 0.998 3188672 BCB03_000764 C[C@@H]1ON([C@@H]([C@H]1C(=O)N2[C@H](Cc3ccccc3)COC2=O)c4ccc(OC(=O)OC(C)(C)C)cc4)c5ccc(I)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G08 compound treatment 187800.0 13500.0 0.92 186160.0 12300.0 0.91 1.2956 1.0 3563147 BCB03_000765 COc1ccc(CN2CCc3cc(OC)c(OC)cc3C2(C)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G09 compound treatment 187520.0 13200.0 0.9 188480.0 14600.0 1.09 1.4042 0.9956 3188673 BCB03_000766 COC(=O)CCCCCCC(=O)Nc1ccc(NC(=O)CCCC[P+](c2ccccc2)(c3ccccc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G10 compound treatment 184960.0 10600.0 0.73 181600.0 7710.0 0.57 0.9188 0.9933 3563148 BCB03_000767 COc1ccc(CN2CCc3cc(OC)c(OC)cc3C2(C)C=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G11 compound treatment 192600.0 18300.0 1.25 189920.0 16000.0 1.19 1.7249 0.9998 3188674 BCB03_000768 CC(C)[C@H]1COC(=O)N1C(=O)[C@@H]2[C@@H](C)ON([C@@H]2c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G12 compound treatment 191600.0 17300.0 1.18 189040.0 15200.0 1.13 1.6304 0.9998 3563149 BCB03_000769 COc1ccc(CN2CCc3cc(OC)c(OC)cc3C2(C)C4CC4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G13 compound treatment 186720.0 12400.0 0.85 179760.0 5870.0 0.44 0.9068 0.953 3188675 BCB03_000770 CC(C)[C@@H](CO)NC(=O)[C@@H]1[C@@H](C)ON([C@@H]1c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G14 compound treatment 184080.0 9760.0 0.67 176880.0 2990.0 0.22 0.6279 0.8951 3563150 BCB03_000771 COCC#CC1(C)N(Cc2ccc(OC)cc2)CCc3cc(OC)c(OC)cc31 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G15 compound treatment 195800.0 21500.0 1.46 194920.0 21000.0 1.57 2.1423 0.9994 3071001 BCB03_000772 COC(=O)[C@@H]1N[C@H]2[C@@H](COc3ccccc23)[C@@H]1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G16 compound treatment 192680.0 18400.0 1.25 190760.0 16900.0 1.26 1.773 1.0 3563151 BCB03_000773 COc1cc2CC(C)N(C)C(C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G17 compound treatment 177040.0 2720.0 0.19 175680.0 1790.0 0.13 0.2254 0.9871 3071002 BCB03_000774 OCC1CC(=NO1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G18 compound treatment 181480.0 7160.0 0.49 185080.0 11200.0 0.83 0.9341 0.9675 3563152 BCB03_000775 COc1cc2CC(C)N(C)C(C=C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G19 mock treatment 176640.0 2320.0 0.16 181920.0 8030.0 0.6 0.5345 0.8642 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G20 mock treatment 177000.0 2680.0 0.18 176920.0 3030.0 0.23 0.2887 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G21 compound treatment 170880.0 -3440.0 -0.23 172480.0 -1410.0 -0.1 -0.24 -0.9337 3071004 BCB03_000776 O[C@H](C=C)[C@H]1CC(=NO1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G22 compound treatment 172560.0 -1760.0 -0.12 175120.0 1230.0 0.09 -0.0201 -0.1325 3563153 BCB03_000777 COc1cc2CC(C)N(C)C(C3CC3)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G23 compound treatment 188040.0 13700.0 0.94 190320.0 16400.0 1.22 1.5261 0.9912 3414065 BCB03_000778 O[C@@H]([C@H]1CC(=NO1)c2ccccc2)[C@@H]3CC(=NO3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 G24 compound treatment 172680.0 -1640.0 -0.11 172120.0 -1770.0 -0.13 -0.1722 -0.9969 3563154 BCB03_000779 COCC#CC1N(C)C(C)Cc2cc(OC)c(OC)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H01 compound treatment 176600.0 2280.0 0.16 168320.0 -5570.0 -0.41 -0.1832 -0.4141 3614478 BCB03_000780 COC(=O)c1cn(CC(=O)N2CCN(C)CC2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H02 compound treatment 190680.0 16400.0 1.12 192480.0 18600.0 1.38 1.7671 0.9943 3061928 BCB03_000781 COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H03 mock treatment 172600.0 -1720.0 -0.12 173760.0 -125.0 -0.01 -0.0897 -0.7608 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H04 mock treatment 175120.0 796.0 0.05 180160.0 6270.0 0.47 0.3686 0.784 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H05 compound treatment 178480.0 4160.0 0.28 174120.0 235.0 0.02 0.2127 0.7493 3614479 BCB03_000782 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)Cn2cc(nn2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H06 compound treatment 209400.0 35100.0 2.39 208440.0 34600.0 2.57 3.5095 0.9993 3614483 BCB03_000783 COCCOc1cc2ncnc(Nc3cccc(C#C)c3)c2cc1OCCOC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H07 compound treatment 178520.0 4200.0 0.29 183520.0 9630.0 0.72 0.7093 0.9188 3614485 BCB03_000784 COC(=O)[C@@H](NC(=O)Cn1cc(nn1)C(=O)OC)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H08 mock treatment 176400.0 2080.0 0.14 179480.0 5590.0 0.42 0.3945 0.8971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H09 compound treatment 179560.0 5240.0 0.36 177640.0 3750.0 0.28 0.45 0.9927 3614488 BCB03_000785 CCOC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)Cn3cc(nn3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H10 mock treatment 173680.0 -644.0 -0.04 179000.0 5110.0 0.38 0.2381 0.6214 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H11 compound treatment 185880.0 11600.0 0.79 186280.0 12400.0 0.92 1.2094 0.9969 3614492 BCB03_000786 COC(=O)c1cn(nn1)c2cccc(N)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H12 mock treatment 183920.0 9600.0 0.65 175400.0 1510.0 0.11 0.5423 0.8169 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H13 compound treatment 180800.0 6480.0 0.44 179720.0 5830.0 0.43 0.6193 1.0 3614494 BCB03_000787 COC(=O)c1cn(CC(=O)N2CCN(CC2)c3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H14 mock treatment 180520.0 6200.0 0.42 179560.0 5670.0 0.42 0.5973 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H15 compound treatment 182320.0 8000.0 0.55 177440.0 3550.0 0.26 0.5726 0.9449 3614495 BCB03_000788 COC(=O)c1cn(CC(=O)N2CCOCC2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H16 mock treatment 177160.0 2840.0 0.19 177200.0 3310.0 0.25 0.3112 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H17 compound treatment 183920.0 9600.0 0.65 178280.0 4390.0 0.33 0.6939 0.9487 3614498 BCB03_000789 COC(=O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H18 mock treatment 182800.0 8480.0 0.58 177120.0 3230.0 0.24 0.5788 0.9247 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H19 mock treatment 176760.0 2440.0 0.17 178240.0 4350.0 0.32 0.3466 0.9518 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H20 mock treatment 179240.0 4920.0 0.34 173880.0 -5.36 0.0 0.2367 0.7063 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H21 compound treatment 174680.0 356.0 0.02 171240.0 -2650.0 -0.2 -0.1221 -0.6153 3614499 BCB03_000790 COC(=O)c1cn(CC(=O)Nc2cc(OC)ccc2OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H22 mock treatment 180120.0 5800.0 0.4 175760.0 1870.0 0.14 0.3781 0.9022 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H23 compound treatment 194240.0 19900.0 1.36 192640.0 18800.0 1.4 1.9471 0.9999 3614501 BCB03_000791 COC(=O)c1cn(CC(=O)Nc2nccs2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 H24 mock treatment 163600.0 -10700.0 -0.73 166280.0 -7610.0 -0.57 -0.9172 -0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I01 compound treatment 173720.0 -604.0 -0.04 173080.0 -805.0 -0.06 -0.0715 -0.9832 3071008 BCB03_000792 CC[C@H](C)C(=O)O[C@H]1CC[C@@]2(C)C(CCC3=C2CC[C@]4(C)[C@H](CC[C@@]34C)[C@H](C)CCCC(C)C)C1(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I02 compound treatment 177640.0 3320.0 0.23 172320.0 -1570.0 -0.12 0.0775 0.3046 3563155 BCB03_000793 COc1ccc(C[N+]2=Cc3cc(OC)c(OC)cc3CC2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I03 compound treatment 198240.0 23900.0 1.63 194960.0 21100.0 1.57 2.2621 0.9998 3188792 BCB03_000794 CC(C)CCC[C@@H](C)[C@H]1CC[C@@]2(C)C3=C(CC[C@]12C)[C@@]4(C)CC[C@H](OC(=O)CCl)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I04 compound treatment 182080.0 7760.0 0.53 180920.0 7030.0 0.52 0.7441 1.0 3563156 BCB03_000795 COc1ccc(CN2C(C)Cc3cc(OC)c(OC)cc3C2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I05 mock treatment 176680.0 2360.0 0.16 177200.0 3310.0 0.25 0.288 0.9784 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I06 mock treatment 176200.0 1880.0 0.13 176680.0 2790.0 0.21 0.2375 0.9727 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I07 compound treatment 189000.0 14700.0 1.0 186640.0 12800.0 0.95 1.3788 0.9997 3188805 BCB03_000796 CC(C)CCC[C@@H](C)[C@H]1CC[C@@]2(C)C3=C(CC[C@]12C)[C@@]4(C)CC[C@H](OC(=O)C(C)(C)C)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I08 compound treatment 187600.0 13300.0 0.91 182600.0 8710.0 0.65 1.0986 0.9866 3563157 BCB03_000797 COc1ccc(CN2C(C)Cc3cc(OC)c(OC)cc3C2C=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I09 compound treatment 200440.0 26100.0 1.78 193280.0 19400.0 1.44 2.2797 0.9946 3188806 BCB03_000798 CC(C)CCC[C@@H](C)[C@H]1CC[C@@]2(C)C3=C(CC[C@]12C)[C@@]4(C)CC[C@H](OC(=O)c5ccccc5)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I10 compound treatment 180160.0 5840.0 0.4 183880.0 9990.0 0.74 0.8073 0.957 3563158 BCB03_000799 COc1ccc(CN2C(C)Cc3cc(OC)c(OC)cc3C2C4CC4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I11 compound treatment 185680.0 11400.0 0.77 185240.0 11400.0 0.85 1.145 0.999 3188807 BCB03_000800 COc1ccc(cc1)C(=O)O[C@H]2CC[C@@]3(C)C(CCC4=C3CC[C@]5(C)[C@H](CC[C@@]45C)[C@H](C)CCCC(C)C)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I12 compound treatment 181880.0 7560.0 0.52 178880.0 4990.0 0.37 0.6271 0.9872 3563159 BCB03_000801 COCC#CC1N(Cc2ccc(OC)cc2)C(C)Cc3cc(OC)c(OC)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I13 compound treatment 180760.0 6440.0 0.44 181600.0 7710.0 0.57 0.7163 0.9912 3071124 BCB03_000802 COc1cccc(c1)C(=O)O[C@H]2CC[C@@]3(C)C(CCC4=C3CC[C@]5(C)[C@H](CC[C@@]45C)[C@H](C)CCCC(C)C)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I14 compound treatment 191720.0 17400.0 1.19 192320.0 18400.0 1.37 1.8088 0.9974 3614506 BCB03_000803 CCCCOc1ccc(/C=C/C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I15 compound treatment 172120.0 -2200.0 -0.15 178120.0 4230.0 0.32 0.1166 0.334 3188924 BCB03_000804 CC(C)CCC[C@@H](C)[C@H]1CC[C@@]2(C)C3=C(CC[C@]12C)[C@@]4(C)CC[C@H](OC(=O)c5ccc(Br)cc5)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I16 compound treatment 232320.0 58000.0 3.95 232120.0 58200.0 4.33 5.8607 0.9989 3614510 BCB03_000805 ONC(=O)/C=C/c1ccc(OC2CCCCC2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I17 compound treatment 183840.0 9520.0 0.65 180920.0 7030.0 0.52 0.829 0.9943 3188925 BCB03_000806 CC(C)CCC[C@@H](C)[C@H]1CC[C@@]2(C)C3=C(CC[C@]12C)[C@@]4(C)CC[C@H](OC(=O)c5ccc(N)cc5)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I18 compound treatment 201000.0 26700.0 1.82 199160.0 25300.0 1.88 2.6162 0.9999 3614513 BCB03_000807 COc1ccc(/C=C/C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I19 compound treatment 178880.0 4560.0 0.31 179280.0 5390.0 0.4 0.5035 0.992 3614517 BCB03_000808 COC(=O)[C@H](Cc1ccccc1)N(CC#C)O[C@@H](/C=C/[C@@H](O)Cc2ccccc2)C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I20 compound treatment 238960.0 64600.0 4.41 236760.0 62900.0 4.68 6.4249 0.9995 3614521 BCB03_000809 ONC(=O)/C=C/c1ccc(O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I21 mock treatment 174560.0 236.0 0.02 172400.0 -1490.0 -0.11 -0.0668 -0.5979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I22 mock treatment 170840.0 -3480.0 -0.24 169120.0 -4770.0 -0.35 -0.4187 -0.981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I23 compound treatment 219160.0 44800.0 3.06 209880.0 36000.0 2.68 4.0558 0.9978 3614524 BCB03_000810 COC(=O)[C@H](Cc1ccccc1)N2CC3=CCCC=C[C@H]3[C@@H]2[C@@H](O)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 I24 compound treatment 237200.0 62900.0 4.29 222240.0 48400.0 3.6 5.5759 0.9962 3614525 BCB03_000811 ONC(=O)/C=C/c1ccc(OCCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J01 compound treatment 168560.0 -5760.0 -0.39 167640.0 -6250.0 -0.46 -0.6065 -0.9965 3614528 BCB03_000812 COC(=O)c1cn(CC(=O)Nc2ccon2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J02 mock treatment 170480.0 -3840.0 -0.26 177160.0 3270.0 0.24 -0.013 -0.0362 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J03 compound treatment 181120.0 6800.0 0.46 175080.0 1190.0 0.09 0.3905 0.8277 3614530 BCB03_000813 COC(=O)c1cn(C[C@H](Cc2ccccc2)NC(=O)Nc3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J04 mock treatment 183120.0 8800.0 0.6 180400.0 6510.0 0.48 0.7669 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J05 mock treatment 179200.0 4880.0 0.33 171000.0 -2890.0 -0.21 0.0832 0.2103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J06 mock treatment 178920.0 4600.0 0.31 177360.0 3470.0 0.26 0.4044 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J07 compound treatment 199960.0 25600.0 1.75 197160.0 23300.0 1.73 2.4608 1.0 3614532 BCB03_000814 O=C(Cn1cc(nn1)C2(CCCCC2)NC(=O)Nc3ccccc3)N4CCN(CC4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J08 mock treatment 178600.0 4280.0 0.29 179400.0 5510.0 0.41 0.4964 0.986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J09 compound treatment 184200.0 9880.0 0.67 182760.0 8870.0 0.66 0.9432 1.0 3614534 BCB03_000815 NC(=N)NCc1cn(CC(=O)N2CCN(CC2)c3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J10 mock treatment 178360.0 4040.0 0.28 180080.0 6190.0 0.46 0.5206 0.9696 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J11 compound treatment 180760.0 6440.0 0.44 181800.0 7910.0 0.59 0.7268 0.9895 3614535 BCB03_000816 CC(=O)Nc1ccccc1c2cn(CC(=O)N3CCN(CC3)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J12 mock treatment 179080.0 4760.0 0.32 179000.0 5110.0 0.38 0.4985 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J13 compound treatment 177400.0 3080.0 0.21 174960.0 1070.0 0.08 0.2048 0.9127 3614536 BCB03_000817 O=C(Cn1cc(nn1)C2(CCCCC2)NC(=O)Nc3ccccc3)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J14 mock treatment 176840.0 2520.0 0.17 176760.0 2870.0 0.21 0.2726 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J15 compound treatment 178760.0 4440.0 0.3 174960.0 1070.0 0.08 0.2704 0.8644 3614537 BCB03_000818 CC(=O)Nc1ccccc1c2cn(CC(=O)N3CCOCC3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J16 mock treatment 178400.0 4080.0 0.28 173640.0 -245.0 -0.02 0.1836 0.6592 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J17 compound treatment 183440.0 9120.0 0.62 178160.0 4270.0 0.32 0.6644 0.9516 3556424 BCB03_000819 COC(=O)c1c(C(=O)OC)c2oc1CC[C@H](CO)NC(=O)N[C@@H](Cc3ccccc3)C(=O)NCc4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J18 mock treatment 177480.0 3160.0 0.22 176920.0 3030.0 0.23 0.3119 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J19 compound treatment 194480.0 20200.0 1.37 198080.0 24200.0 1.8 2.245 0.9911 3614538 BCB03_000820 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCCn3cc(nn3)c4ccccc4N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J20 mock treatment 174560.0 236.0 0.02 170440.0 -3450.0 -0.26 -0.1699 -0.6614 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J21 mock treatment 174840.0 516.0 0.04 170240.0 -3650.0 -0.27 -0.167 -0.6103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J22 mock treatment 171360.0 -2960.0 -0.2 168320.0 -5570.0 -0.41 -0.4358 -0.9455 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J23 compound treatment 207920.0 33600.0 2.29 221640.0 47800.0 3.55 4.1328 0.9774 3614540 BCB03_000821 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCn3cc(nn3)c4ccccc4N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 J24 mock treatment 165640.0 -8680.0 -0.59 164360.0 -9530.0 -0.71 -0.9199 -0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K01 compound treatment 200640.0 26300.0 1.79 186840.0 13000.0 0.96 1.9504 0.9576 3614545 BCB03_000822 COC(=O)[C@H](Cc1ccccc1)N2CC3=CC(=O)[C@H](C4CC4)[C@H]3[C@@H]2[C@@H](O)Cc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K02 compound treatment 237040.0 62700.0 4.28 231440.0 57600.0 4.28 6.0524 1.0 3614548 BCB03_000823 COc1ccc(CCCOc2ccc(/C=C/C(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K03 compound treatment 227040.0 52700.0 3.59 220720.0 46800.0 3.49 5.0062 0.9999 3614553 BCB03_000824 O=C1C=C2CN3[C@H]([C@@H]2[C@H]1C4CC4)[C@H](Cc5ccccc5)OC(=O)[C@@H]3Cc6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K04 compound treatment 202480.0 28200.0 1.92 192080.0 18200.0 1.35 2.3149 0.9854 3614558 BCB03_000825 ONC(=O)/C=C/c1ccc(OCCc2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K05 compound treatment 234920.0 60600.0 4.13 216200.0 42300.0 3.15 5.1482 0.991 3614560 BCB03_000826 COC(=O)C1(CCCC1)N2CC3=CCCC=C[C@H]3[C@@H]2[C@@H](O)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K06 compound treatment 217080.0 42800.0 2.91 209640.0 35800.0 2.66 3.9429 0.999 3614562 BCB03_000827 ONC(=O)/C=C/c1ccc(OCCNCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K07 mock treatment 181160.0 6840.0 0.47 177560.0 3670.0 0.27 0.5229 0.9677 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K08 mock treatment 181080.0 6760.0 0.46 178160.0 4270.0 0.32 0.5507 0.9837 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K09 compound treatment 197120.0 22800.0 1.55 200880.0 27000.0 2.01 2.5196 0.9919 3614565 BCB03_000828 C=C/C=C/[C@H]1[C@@H]2[C@H](Cc3ccccc3)OC(=O)C4(CCCC4)N2CC1=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K10 compound treatment 194840.0 20500.0 1.4 198040.0 24200.0 1.8 2.2603 0.9923 1065487 BCB03_000829 ONC(=O)CCCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K11 compound treatment 197480.0 23200.0 1.58 198280.0 24400.0 1.82 2.4002 0.9976 3614570 BCB03_000830 O=C1O[C@@H](Cc2ccccc2)[C@H]3[C@@H]4C=CCCC=C4CN3C51CCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K12 compound treatment 188400.0 14100.0 0.96 186320.0 12400.0 0.93 1.333 0.9998 3614573 BCB03_000831 CCCC(CCC)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K13 compound treatment 187080.0 12800.0 0.87 180080.0 6190.0 0.46 0.941 0.9559 3614575 BCB03_000832 COC(=O)C1(CCCC1)N2CC3=C[C@@H]([C@@H](O)Cc4ccccc4)n5n([C@@H]3[C@H](O2)C6CC6)c(=O)n(C)c5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K14 compound treatment 201880.0 27600.0 1.88 198040.0 24200.0 1.8 2.5996 0.9998 3614578 BCB03_000833 Oc1ccc2ncnc(NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K15 mock treatment 178880.0 4560.0 0.31 178160.0 4270.0 0.32 0.4446 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K16 mock treatment 178000.0 3680.0 0.25 176080.0 2190.0 0.16 0.2927 0.9785 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K17 compound treatment 194600.0 20300.0 1.38 189480.0 15600.0 1.16 1.7982 0.9962 3614579 BCB03_000834 COC(=O)C1(CCCC1)N2CC3=C[C@@H](C4CC4)n5n([C@H]3[C@@H]2[C@@H](O)Cc6ccccc6)c(=O)n(C)c5=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K18 compound treatment 206600.0 32300.0 2.2 206760.0 32900.0 2.45 3.2861 0.9986 3614582 BCB03_000835 CCCNc1ncnc2ccc(O)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K19 compound treatment 179400.0 5080.0 0.35 177480.0 3590.0 0.27 0.4339 0.9919 3614584 BCB03_000836 COC(=O)C1(CCCC1)N2C[C@](C)(OC)O[C@@H](Cc3ccccc3)[C@H]2/C=C/C4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K20 compound treatment 182640.0 8320.0 0.57 184200.0 10300.0 0.77 0.9437 0.9889 2065681 BCB03_000837 CC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K21 compound treatment 220560.0 46200.0 3.15 226560.0 52700.0 3.92 5.0011 0.9942 3614590 BCB03_000838 COC(=O)C1(CCCC1)N2CC(=C)[C@@H](/C=C/C=C)[C@@H]2[C@@H](O)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K22 compound treatment 197040.0 22700.0 1.55 191440.0 17600.0 1.31 2.019 0.9964 3216001 BCB03_000839 COCC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K23 mock treatment 166480.0 -7840.0 -0.53 169200.0 -4690.0 -0.35 -0.6247 -0.9785 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 K24 mock treatment 163840.0 -10500.0 -0.71 162080.0 -11800.0 -0.88 -1.1267 -0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L01 compound treatment 178520.0 4200.0 0.29 177560.0 3670.0 0.27 0.3957 0.9997 3614594 BCB03_000840 Nc1ccccc1c2cn(CC(=O)Nc3nccs3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L02 mock treatment 177560.0 3240.0 0.22 175560.0 1670.0 0.12 0.2441 0.9635 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L03 compound treatment 175640.0 1320.0 0.09 180480.0 6590.0 0.49 0.4105 0.8227 3614596 BCB03_000841 Nc1ccccc1c2cn(CC(=O)Nc3ccon3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L04 mock treatment 180080.0 5760.0 0.39 172280.0 -1610.0 -0.12 0.193 0.4705 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L05 compound treatment 202600.0 28300.0 1.93 200400.0 26500.0 1.97 2.7585 0.9999 3556414 BCB03_000842 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@H](Cc3ccccc3)c4cn(C[C@@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L06 mock treatment 181520.0 7200.0 0.49 180400.0 6510.0 0.48 0.6898 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L07 mock treatment 176920.0 2600.0 0.18 174400.0 515.0 0.04 0.1522 0.8407 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L08 mock treatment 174080.0 -244.0 -0.02 177880.0 3990.0 0.3 0.1985 0.6665 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L09 compound treatment 188080.0 13800.0 0.94 190200.0 16300.0 1.21 1.5218 0.9919 3556416 BCB03_000843 COC(=O)c1c(C(=O)OC)c2oc1CC[C@@H](CO)NC(=O)N[C@H](Cc3ccccc3)c4cn(C[C@H](Cc5ccccc5)NC2=O)nn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L10 mock treatment 182480.0 8160.0 0.56 180880.0 6990.0 0.52 0.7613 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L11 compound treatment 172680.0 -1640.0 -0.11 179680.0 5790.0 0.43 0.2257 0.5065 3614599 BCB03_000844 CN1C(=O)[C@@H]2[C@H](C1=O)[C@]34COC[C@@H](N4C(=O)[C@@]2(O3)C(=O)C)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L12 mock treatment 180960.0 6640.0 0.45 181440.0 7550.0 0.56 0.7175 0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L13 compound treatment 184800.0 10500.0 0.71 182360.0 8470.0 0.63 0.951 0.9981 3614605 BCB03_000845 Cc1ccc(cc1)S(=O)(=O)N2CCC[C@H]2Cn3cc(nn3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L14 mock treatment 178520.0 4200.0 0.29 177080.0 3190.0 0.24 0.3704 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L15 mock treatment 177240.0 2920.0 0.2 175920.0 2030.0 0.15 0.2477 0.991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L16 mock treatment 176280.0 1960.0 0.13 179480.0 5590.0 0.42 0.3887 0.8891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L17 compound treatment 178760.0 4440.0 0.3 177680.0 3790.0 0.28 0.4136 0.9994 3614607 BCB03_000846 CN1C(=O)[C@H]2[C@@H](C1=O)[C@@]34COC[C@@H](N4C(=O)[C@]2(O3)C(=O)C)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L18 mock treatment 180000.0 5680.0 0.39 174280.0 395.0 0.03 0.2944 0.7586 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L19 compound treatment 174000.0 -324.0 -0.02 173840.0 -45.4 0.0 -0.018 -0.8058 3614609 BCB03_000847 CC(=O)[C@@]1(O[C@@]23COC[C@@H](N3C1=O)c4ccccc4)[C@H]5[C@@H]2C(=O)N(C5=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L20 mock treatment 171880.0 -2440.0 -0.17 169400.0 -4490.0 -0.33 -0.3539 -0.9485 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L21 compound treatment 176440.0 2120.0 0.14 177560.0 3670.0 0.27 0.2954 0.9553 3614611 BCB03_000848 CC(=O)[C@]1(O[C@]23COC[C@@H](N3C1=O)c4ccccc4)[C@@H]5[C@H]2C(=O)N(C5=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L22 mock treatment 169080.0 -5240.0 -0.36 169440.0 -4450.0 -0.33 -0.4868 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L23 mock treatment 163080.0 -11200.0 -0.77 169840.0 -4050.0 -0.3 -0.7549 -0.9167 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 L24 mock treatment 164560.0 -9760.0 -0.67 166640.0 -7250.0 -0.54 -0.852 -0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M01 compound treatment 217160.0 42800.0 2.92 215920.0 42000.0 3.13 4.2772 0.9994 3614612 BCB03_000849 COC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](N3CC4=CC(=O)[C@H](C5CC5)[C@H]4[C@@H]3[C@@H](O)Cc6ccccc6)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M02 compound treatment 210480.0 36200.0 2.47 212440.0 38600.0 2.87 3.7721 0.9971 3215997 BCB03_000850 OB1C[C@@H]2[C@H]3[C@@H](CC(=C2[C@H](O1)c4ccccc4)COc5ccccc5)C(=O)N(Cc6ccccc6)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M03 compound treatment 230800.0 56500.0 3.85 240680.0 66800.0 4.97 6.2379 0.992 3614614 BCB03_000851 COC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](N3CC(=C)[C@@H](/C=C/C=C)[C@@H]3[C@@H](O)Cc4ccccc4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M04 compound treatment 197920.0 23600.0 1.61 190880.0 17000.0 1.26 2.0319 0.9929 3216003 BCB03_000852 CN1C(=O)[C@@H]2CC(=C3[C@H](OB(O)C[C@@H]3[C@@H]2C1=O)c4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M05 compound treatment 208360.0 34000.0 2.32 200720.0 26800.0 2.0 3.0531 0.9972 3614616 BCB03_000853 O=C1C=C2CN3[C@H]([C@@H]2[C@H]1C4CC4)[C@H](Cc5ccccc5)OC(=O)C63CCCC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M06 compound treatment 192640.0 18300.0 1.25 191040.0 17200.0 1.28 1.7858 0.9999 3215999 BCB03_000854 COCC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)N(C)C3=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M07 compound treatment 215920.0 41600.0 2.84 216840.0 43000.0 3.2 4.2659 0.9982 3614620 BCB03_000855 COC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](N[C@@H](/C=C/C3CC3)[C@H](O)Cc4ccccc4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M08 compound treatment 189800.0 15500.0 1.06 189120.0 15200.0 1.13 1.5478 0.9994 3215995 BCB03_000856 CN1C(=O)[C@@H]2CC(=C3[C@H](OB(O)C[C@@H]3[C@@H]2C1=O)c4ccccc4)COc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M09 mock treatment 179200.0 4880.0 0.33 180200.0 6310.0 0.47 0.5674 0.9856 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M10 mock treatment 177960.0 3640.0 0.25 184600.0 10700.0 0.8 0.7392 0.8851 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M11 compound treatment 208000.0 33700.0 2.3 199200.0 25300.0 1.88 2.9557 0.9952 3614624 BCB03_000857 COC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](N(CC#C)[C@@H](/C=C/C3CC3)[C@H](O)Cc4ccccc4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M12 compound treatment 201240.0 26900.0 1.84 199560.0 25700.0 1.91 2.6488 0.9998 3215892 BCB03_000858 CC1=C2[C@H](OB(O)C[C@@H]2n3n(C1)c(=O)n(c4ccccc4)c3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M13 mock treatment 182400.0 8080.0 0.55 180560.0 6670.0 0.5 0.7406 0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M14 mock treatment 179320.0 5000.0 0.34 182160.0 8270.0 0.62 0.6763 0.961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M15 compound treatment 201360.0 27000.0 1.84 195560.0 21700.0 1.61 2.4441 0.9978 3614627 BCB03_000859 O[C@@H](Cc1ccccc1)[C@H]2O[C@@H](Cc3ccccc3)[C@@H](/C=C/C4CC4)N2CC#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M16 compound treatment 198640.0 24300.0 1.66 196320.0 22400.0 1.67 2.3529 1.0 3215890 BCB03_000860 COCC1=C2[C@H](OB(O)C[C@@H]2n3n(C1)c(=O)n(c4ccccc4)c3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M17 compound treatment 183760.0 9440.0 0.64 184280.0 10400.0 0.77 1.0019 0.9958 3562141 BCB03_000861 COC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](N(CC#C)[C@H](/C=C/C3CC3)[C@@H](O)Cc4ccccc4)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M18 compound treatment 203000.0 28700.0 1.96 201840.0 28000.0 2.08 2.8536 0.9995 3215888 BCB03_000862 OB1C[C@H]2C(=C(COc3ccccc3)Cn4n2c(=O)n(c5ccccc5)c4=O)[C@H](O1)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M19 compound treatment 185960.0 11600.0 0.79 186440.0 12600.0 0.93 1.2217 0.9967 3614632 BCB03_000863 O=C1O[C@H](C2CCCCC2)[C@H](/C=C/C3CC3)N(CC#C)C1Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M20 compound treatment 204440.0 30100.0 2.05 203320.0 29400.0 2.19 3.0009 0.9995 3215943 BCB03_000864 CC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)c4ccccc4C3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M21 compound treatment 216920.0 42600.0 2.9 214320.0 40400.0 3.01 4.1815 0.9998 3614636 BCB03_000865 O=C1O[C@@H]([C@@H]2[C@H]3C=CCCC=C3CN2C1Cc4ccccc4)C5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M22 compound treatment 193080.0 18800.0 1.28 200520.0 26600.0 1.98 2.3059 0.9775 3215941 BCB03_000866 COCC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)c4ccccc4C3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M23 compound treatment 188320.0 14000.0 0.95 189000.0 15100.0 1.12 1.4702 0.9966 3614641 BCB03_000867 COC(=O)[C@@H]1N2[C@H](SC1(C)C)[C@H](N3[C@H](/C=C/C4CC4)[C@H](Cc5ccccc5)OC3=O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 M24 compound treatment 212280.0 38000.0 2.59 219680.0 45800.0 3.41 4.2399 0.9908 3215939 BCB03_000868 OB1C[C@@H]2[C@H]3[C@@H](CC(=C2[C@H](O1)c4ccccc4)COc5ccccc5)C(=O)c6ccccc6C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N01 compound treatment 181280.0 6960.0 0.47 175360.0 1470.0 0.11 0.4129 0.8483 3614646 BCB03_000869 C=CCOC(=O)[C@@]1(O[C@@]23COC[C@@H](N3C1=O)c4ccccc4)[C@H]5[C@@H]2C(=O)N(C5=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N02 mock treatment 176000.0 1680.0 0.11 176960.0 3070.0 0.23 0.2426 0.9485 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N03 compound treatment 182720.0 8400.0 0.57 187120.0 13200.0 0.99 1.1013 0.9667 3614650 BCB03_000870 C=CCOC(=O)[C@]1(O[C@]23COC[C@@H](N3C1=O)c4ccccc4)[C@@H]5[C@H]2C(=O)N(C5=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N04 mock treatment 179760.0 5440.0 0.37 176320.0 2430.0 0.18 0.3902 0.9458 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N05 compound treatment 188880.0 14600.0 0.99 194280.0 20400.0 1.52 1.775 0.9788 3614652 BCB03_000871 O=C(NCc1ccccc1)[C@@]2(O[C@@]34COC[C@@H](N4C2=O)c5ccccc5)[C@H]6[C@@H]3C(=O)N(C6=O)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N06 mock treatment 184600.0 10300.0 0.7 176040.0 2150.0 0.16 0.6088 0.8471 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N07 compound treatment 189080.0 14800.0 1.01 187040.0 13200.0 0.98 1.4037 0.9999 3614656 BCB03_000872 O=C(NCCc1c[nH]c2ccccc12)[C@@]3(O[C@@]45COC[C@@H](N5C3=O)c6ccccc6)[C@H]7[C@@H]4C(=O)N(C7=O)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N08 mock treatment 172800.0 -1520.0 -0.1 183600.0 9710.0 0.72 0.4378 0.5993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N09 mock treatment 180680.0 6360.0 0.43 183960.0 10100.0 0.75 0.8366 0.966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N10 mock treatment 181360.0 7040.0 0.48 178160.0 4270.0 0.32 0.5642 0.9801 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N11 compound treatment 192200.0 17900.0 1.22 199560.0 25700.0 1.91 2.213 0.9764 3614660 BCB03_000873 COC(=O)c1c(COC[C@@H](NC(=O)N(C)Cc2ccccc2)c3ccccc3)oc(C(=O)OCC=C)c1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N12 mock treatment 184960.0 10600.0 0.73 182400.0 8510.0 0.63 0.9609 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N13 mock treatment 180680.0 6360.0 0.43 180520.0 6630.0 0.49 0.6556 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N14 mock treatment 177960.0 3640.0 0.25 177400.0 3510.0 0.26 0.3603 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N15 compound treatment 182040.0 7720.0 0.53 184960.0 11100.0 0.82 0.9548 0.9765 3614664 BCB03_000874 COc1cc(/C=C(\C#N)/C(=O)Nc2nnc(s2)C(F)(F)F)ccc1OCc3ccc(cc3C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N16 mock treatment 182520.0 8200.0 0.56 177360.0 3470.0 0.26 0.578 0.9387 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N17 compound treatment 190120.0 15800.0 1.08 195320.0 21400.0 1.6 1.8896 0.9817 1917883 BCB03_000875 O/N=C/1\C2(CCCCC2)C(=O)N(O)C31CCCC=C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N18 mock treatment 181240.0 6920.0 0.47 177760.0 3870.0 0.29 0.5373 0.9722 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N19 compound treatment 281600.0 107000.0 7.31 257400.0 83500.0 6.22 9.5668 0.9967 3614668 BCB03_000876 C[C@@]12CCC3[C@@]4(C)CC[C@H](O)CC54C=CC3(C2CC[C@@]1(O)CN6CCC(CC6)n7c(=O)[nH]c8ccccc78)C(=C5)C(=O)c9cc%10ccccc%10s9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N20 mock treatment 177600.0 3280.0 0.22 174520.0 635.0 0.05 0.1913 0.8381 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N21 compound treatment 247480.0 73200.0 4.99 230080.0 56200.0 4.18 6.4841 0.9962 3614669 BCB03_000877 C[C@@]12CCC3[C@@]4(C)CC[C@H](O)CC54C=CC3(C2CC[C@@]1(O)CN6CCC(CC6)n7c(=O)[nH]c8ccccc78)C(=C5)C(=O)C9CCCCC9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N22 mock treatment 173280.0 -1040.0 -0.07 173600.0 -285.0 -0.02 -0.0653 -0.8798 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N23 compound treatment 190920.0 16600.0 1.13 183600.0 9710.0 0.72 1.3113 0.9766 3614671 BCB03_000878 C[C@@]12CCC3[C@@]4(C)CC[C@H](O)CC54C=CC3(C2CC[C@@]1(O)CN6CCC(CC6)C(=O)N)C(=C5)C(=O)c7ccc(F)c(F)c7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 N24 mock treatment 166200.0 -8120.0 -0.55 167840.0 -6050.0 -0.45 -0.7098 -0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O01 compound treatment 252280.0 78000.0 5.31 241400.0 67500.0 5.02 7.3113 0.9996 3614673 BCB03_000879 COC(=O)[C@H](Cc1ccccc1)N2[C@@H](/C=C/C3CC3)[C@@H](Cc4ccccc4)OC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O02 compound treatment 171680.0 -2640.0 -0.18 180680.0 6790.0 0.51 0.2301 0.4286 2065712 BCB03_000880 CC1=C([C@H](O)c2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O03 compound treatment 178520.0 4200.0 0.29 177000.0 3110.0 0.23 0.3662 0.9946 3614677 BCB03_000881 COC(=O)C1(CCCC1)N2[C@H](/C=C/C3CC3)[C@H](Cc4ccccc4)OC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O04 compound treatment 179480.0 5160.0 0.35 178680.0 4790.0 0.36 0.5009 1.0 3215981 BCB03_000882 COCC1=C([C@H](O)c2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O05 compound treatment 227360.0 53000.0 3.62 220600.0 46700.0 3.48 5.0153 0.9998 3614680 BCB03_000883 COC(=O)[C@H](Cc1ccccc1)N2[C@H](/C=C/C3CC3)[C@H](Cc4ccccc4)OC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O06 compound treatment 183960.0 9640.0 0.66 184280.0 10400.0 0.77 1.0116 0.9967 3215977 BCB03_000884 OC[C@@H]1[C@H]2[C@@H](CC(=C1[C@H](O)c3ccccc3)COc4ccccc4)C(=O)N(Cc5ccccc5)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O07 compound treatment 175280.0 956.0 0.07 180320.0 6430.0 0.48 0.3847 0.796 3563099 BCB03_000885 COC(=O)C1=CN(C)C(C)c2ccccc2C=C1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O08 compound treatment 182400.0 8080.0 0.55 174920.0 1030.0 0.08 0.4438 0.7982 2065737 BCB03_000886 CN1C(=O)[C@@H]2CC(=C([C@H](O)c3ccccc3)[C@H](CO)[C@@H]2C1=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O09 compound treatment 172720.0 -1600.0 -0.11 177920.0 4030.0 0.3 0.135 0.4225 3563100 BCB03_000887 CCOC(=O)C1=C2[C@@H](ON1)N(C)[C@H](C)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O10 compound treatment 180000.0 5680.0 0.39 183760.0 9870.0 0.73 0.7933 0.9551 3215979 BCB03_000888 COCC1=C([C@H](O)c2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O11 mock treatment 168360.0 -5960.0 -0.41 174840.0 955.0 0.07 -0.2373 -0.5748 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O12 mock treatment 177800.0 3480.0 0.24 173440.0 -445.0 -0.03 0.1441 0.6023 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O13 compound treatment 180360.0 6040.0 0.41 181600.0 7710.0 0.57 0.697 0.9867 3563102 BCB03_000889 CCOC(=O)C1=C2[C@@H](ON1)N(C)[C@@H](C)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O14 compound treatment 183080.0 8760.0 0.6 187600.0 13700.0 1.02 1.1439 0.9674 3215975 BCB03_000890 CN1C(=O)[C@@H]2CC(=C([C@H](O)c3ccccc3)[C@H](CO)[C@@H]2C1=O)COc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O15 compound treatment 206960.0 32600.0 2.23 194040.0 20200.0 1.5 2.634 0.9816 3563103 BCB03_000891 CC1N(C)/C(=N\P(=O)(Oc2ccccc2)Oc3ccccc3)/Cc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O16 compound treatment 177880.0 3560.0 0.24 175000.0 1110.0 0.08 0.2301 0.898 3215878 BCB03_000892 CC1=C([C@H](O)c2ccccc2)[C@H](CO)n3n(C1)c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O17 compound treatment 213520.0 39200.0 2.67 228840.0 55000.0 4.09 4.7817 0.9787 3563106 BCB03_000893 CN/1C(C=C)c2ccccc2C\C1=N\P(=O)(Oc3ccccc3)Oc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O18 compound treatment 172760.0 -1560.0 -0.11 174040.0 155.0 0.01 -0.0673 -0.6271 3215876 BCB03_000894 COCC1=C([C@H](O)c2ccccc2)[C@H](CO)n3n(C1)c(=O)n(c4ccccc4)c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O19 compound treatment 170720.0 -3600.0 -0.25 173000.0 -885.0 -0.07 -0.2203 -0.8661 3563109 BCB03_000895 CCOC(=O)C1=C2[C@H](ON1)N(C)[C@@H](C3CC3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O20 compound treatment 183960.0 9640.0 0.66 176720.0 2830.0 0.21 0.6137 0.8894 3215874 BCB03_000896 OC[C@H]1C(=C(COc2ccccc2)Cn3n1c(=O)n(c4ccccc4)c3=O)[C@H](O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O21 compound treatment 168400.0 -5920.0 -0.4 172360.0 -1530.0 -0.11 -0.3659 -0.8721 3563111 BCB03_000897 CCOC(=O)C1=C2[C@@H](ON1)N(C)[C@@H](C3CC3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O22 compound treatment 188560.0 14200.0 0.97 194800.0 20900.0 1.56 1.787 0.9742 3216007 BCB03_000898 C[C@]1(C[C@@H]2[C@H]([C@H]/3CO1)C(=O)N(Cc4ccccc4)C2=O)\C3=C\c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O23 compound treatment 208360.0 34000.0 2.32 196080.0 22200.0 1.65 2.8089 0.9861 3563112 BCB03_000899 CN/1C(C2CC2)c3ccccc3C\C1=N\P(=O)(Oc4ccccc4)Oc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 O24 compound treatment 185000.0 10700.0 0.73 161120.0 -12800.0 -0.95 -0.1571 -0.1313 3216011 BCB03_000900 COC[C@]1(C[C@@H]2[C@H]([C@H]/3CO1)C(=O)N(Cc4ccccc4)C2=O)\C3=C\c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P01 compound treatment 190080.0 15800.0 1.07 187400.0 13500.0 1.01 1.4708 0.9995 3614688 BCB03_000901 COc1ccc(cc1OC2CCCC2)C3=NOC(C3)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P02 mock treatment 174440.0 116.0 0.01 174960.0 1070.0 0.08 0.0622 0.7733 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P03 compound treatment 227840.0 53500.0 3.65 233160.0 59300.0 4.41 5.6994 0.9955 3614690 BCB03_000902 CC(=O)c1ccc(NC(=S)Nc2ccc(Nc3ccccc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P04 mock treatment 173080.0 -1240.0 -0.08 171440.0 -2450.0 -0.18 -0.1887 -0.9396 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P05 compound treatment 172160.0 -2160.0 -0.15 172840.0 -1050.0 -0.08 -0.1593 -0.9553 3614693 BCB03_000903 COC(=O)c1cn(CC(=O)O)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P06 mock treatment 176920.0 2600.0 0.18 172720.0 -1170.0 -0.09 0.0638 0.3238 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P07 compound treatment 174240.0 -83.9 -0.01 173360.0 -525.0 -0.04 -0.0317 -0.802 3614695 BCB03_000904 COC(=O)c1cn(CCC(=O)O)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P08 mock treatment 172800.0 -1520.0 -0.1 173480.0 -405.0 -0.03 -0.0948 -0.8762 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P09 compound treatment 214200.0 39900.0 2.72 217120.0 43200.0 3.22 4.1977 0.9965 1366116 BCB03_000905 Brc1ccc2ncnc(NCC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P10 mock treatment 171400.0 -2920.0 -0.2 173640.0 -245.0 -0.02 -0.1539 -0.7687 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P11 mock treatment 172600.0 -1720.0 -0.12 174800.0 915.0 0.07 -0.035 -0.2575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P12 mock treatment 173920.0 -404.0 -0.03 172320.0 -1570.0 -0.12 -0.1019 -0.8508 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P13 compound treatment 194520.0 20200.0 1.38 199560.0 25700.0 1.91 2.3248 0.9871 1263689 BCB03_000906 Brc1ccc2ncnc(NCc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P14 mock treatment 173240.0 -1080.0 -0.07 172880.0 -1010.0 -0.07 -0.1052 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P15 compound treatment 214360.0 40000.0 2.73 219200.0 45300.0 3.37 4.3149 0.9945 1385097 BCB03_000907 CCCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P16 mock treatment 169280.0 -5040.0 -0.34 171640.0 -2250.0 -0.17 -0.3613 -0.9451 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P17 compound treatment 176640.0 2320.0 0.16 175280.0 1390.0 0.1 0.1851 0.9793 3614697 BCB03_000908 CC(C)(C)OC(=O)NCCOCCOCCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P18 mock treatment 169840.0 -4480.0 -0.31 169680.0 -4210.0 -0.31 -0.4375 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P19 compound treatment 174720.0 396.0 0.03 175040.0 1150.0 0.09 0.0799 0.8866 3614698 BCB03_000909 CCOc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P20 mock treatment 163240.0 -11100.0 -0.76 170240.0 -3650.0 -0.27 -0.7262 -0.9045 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P21 compound treatment 180440.0 6120.0 0.42 181600.0 7710.0 0.57 0.7009 0.9877 1985613 BCB03_000910 C=CCNc1ncnc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P22 mock treatment 162920.0 -11400.0 -0.78 165280.0 -8610.0 -0.64 -1.0026 -0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P23 compound treatment 168720.0 -5600.0 -0.38 170600.0 -3290.0 -0.24 -0.4431 -0.9767 1412880 BCB03_000911 C(Nc1ncnc2ccccc12)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2283 P24 mock treatment 159280.0 -15000.0 -1.03 164800.0 -9090.0 -0.68 -1.2034 -0.9796 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A01 mock treatment 159760.0 -6320.0 -0.43 162800.0 -3690.0 -0.27 -0.4991 -0.9763 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A02 mock treatment 160920.0 -5160.0 -0.35 162280.0 -4210.0 -0.31 -0.4705 -0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A03 compound treatment 161760.0 -4320.0 -0.29 164000.0 -2490.0 -0.19 -0.3395 -0.975 3614734 CMLD4_000001 CCC#CCOCC(=S)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A04 compound treatment 169960.0 3880.0 0.26 170520.0 4030.0 0.3 0.3989 0.998 3614738 CMLD4_000002 CNC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A05 compound treatment 227480.0 61400.0 4.19 240480.0 74000.0 5.51 6.8537 0.9908 3614742 CMLD4_000003 CC[C@@]1(O)C(=O)COc2c1cc3-c4nc5cccc(C(C)C)c5c(c4Cn3c2=O)[Si](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A06 compound treatment 163440.0 -2640.0 -0.18 161240.0 -5250.0 -0.39 -0.4038 -0.9383 3614746 CMLD4_000004 COC(=O)[C@@H]1C[C@@]1(C)[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A07 compound treatment 177160.0 11100.0 0.76 200400.0 33900.0 2.52 2.3186 0.8801 3614748 CMLD4_000005 CC(C)c1cccc2nc-3c(Cn4c3cccc4=O)c(c12)[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A08 compound treatment 163560.0 -2520.0 -0.17 163520.0 -2970.0 -0.22 -0.278 -0.9923 3614750 CMLD4_000006 CN(C)C(=O)[C@H]1C[C@@H]1[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A09 compound treatment 171040.0 4960.0 0.34 168960.0 2470.0 0.18 0.3689 0.959 3614755 CMLD4_000007 CCc1cccc2c(c3CCOc3nc12)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A10 compound treatment 186160.0 20100.0 1.37 182560.0 16100.0 1.2 1.8136 0.9977 3614756 CMLD4_000008 CC(C)NC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A11 compound treatment 207520.0 41400.0 2.83 204320.0 37800.0 2.82 3.9885 1.0 3614760 CMLD4_000009 COc1ccc2nc-3c(Cn4c3cccc4=O)c(c2c1)[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A12 compound treatment 196960.0 30900.0 2.11 191800.0 25300.0 1.88 2.8205 0.9985 3614761 CMLD4_000010 CCOC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A13 compound treatment 165080.0 -1000.0 -0.07 159960.0 -6530.0 -0.49 -0.3921 -0.7988 3614762 CMLD4_000011 CCC#CCOCC(=O)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A14 compound treatment 188840.0 22800.0 1.55 190160.0 23700.0 1.76 2.3427 0.998 3614764 CMLD4_000012 COC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A15 compound treatment 164160.0 -1920.0 -0.13 163400.0 -3090.0 -0.23 -0.2554 -0.9645 3614765 CMLD4_000013 CCc1c2COCc2nc3cc(SC)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A16 compound treatment 185760.0 19700.0 1.34 186760.0 20300.0 1.51 2.0153 0.9983 3614766 CMLD4_000014 CCOC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A17 compound treatment 162120.0 -3960.0 -0.27 161840.0 -4650.0 -0.35 -0.4358 -0.9925 3614767 CMLD4_000015 Cc1ccc(/C=C/C(=O)NCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A18 compound treatment 158120.0 -7960.0 -0.54 159120.0 -7370.0 -0.55 -0.7718 -1.0 3614770 CMLD4_000016 ClC1=C(NC2CCc3ccccc23)C(=O)c4ncccc4C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A19 compound treatment 193360.0 27300.0 1.86 173240.0 6750.0 0.5 1.6702 0.867 1965263 CMLD4_000017 CCCC[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A20 compound treatment 168920.0 2840.0 0.19 162480.0 -4010.0 -0.3 -0.0743 -0.209 3614771 CMLD4_000018 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(Cl)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A21 compound treatment 194720.0 28600.0 1.95 190760.0 24300.0 1.81 2.6578 0.9992 3614772 CMLD4_000019 CC(C)NC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A22 compound treatment 159560.0 -6520.0 -0.44 160000.0 -6490.0 -0.48 -0.6561 -0.9991 3614773 CMLD4_000020 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A23 mock treatment 164680.0 -1400.0 -0.1 161960.0 -4530.0 -0.34 -0.3061 -0.8733 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 A24 mock treatment 161920.0 -4160.0 -0.28 156560.0 -9930.0 -0.74 -0.7233 -0.9136 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B01 mock treatment 154480.0 -11600.0 -0.79 156280.0 -10200.0 -0.76 -1.0967 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B02 mock treatment 156560.0 -9520.0 -0.65 158800.0 -7690.0 -0.57 -0.8638 -0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B03 compound treatment 159440.0 -6640.0 -0.45 162080.0 -4410.0 -0.33 -0.5524 -0.9875 3614775 CMLD4_000021 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B04 compound treatment 188080.0 22000.0 1.5 180760.0 14300.0 1.06 1.8114 0.9857 1693791 CMLD4_000022 CCOC(=O)C1=C(C)NC(=O)NC1c2ccc(Cl)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B05 compound treatment 165640.0 -444.0 -0.03 164080.0 -2410.0 -0.18 -0.1482 -0.8148 3614778 CMLD4_000023 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B06 compound treatment 183560.0 17500.0 1.19 175760.0 9270.0 0.69 1.3303 0.9663 3614780 CMLD4_000024 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B07 compound treatment 165520.0 -564.0 -0.04 165400.0 -1090.0 -0.08 -0.0846 -0.9417 3614783 CMLD4_000025 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B08 compound treatment 165200.0 -884.0 -0.06 165080.0 -1410.0 -0.1 -0.1168 -0.9653 1965278 CMLD4_000026 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B09 compound treatment 173360.0 7280.0 0.5 161840.0 -4650.0 -0.35 0.106 0.1753 3614786 CMLD4_000027 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc3ccccc3c2)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B10 compound treatment 162440.0 -3640.0 -0.25 164120.0 -2370.0 -0.18 -0.3004 -0.9859 3614789 CMLD4_000028 CC(Cc1ccccc1)C(=O)NCc2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B11 compound treatment 174360.0 8280.0 0.56 173800.0 7310.0 0.54 0.7837 0.9998 3614790 CMLD4_000029 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc3OCOc3c2)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B12 compound treatment 181400.0 15300.0 1.04 184880.0 18400.0 1.37 1.7062 0.9911 3614792 CMLD4_000030 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccc(cc4)S(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B13 compound treatment 174280.0 8200.0 0.56 168280.0 1790.0 0.13 0.4893 0.8518 1775499 CMLD4_000031 CCOC(=O)C1=C(C)N(C)C(=O)NC1c2cccc(c2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B14 compound treatment 163080.0 -3000.0 -0.2 160840.0 -5650.0 -0.42 -0.4422 -0.9453 3614798 CMLD4_000032 CNC(=O)[C@H](C)[C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B15 compound treatment 167080.0 996.0 0.07 170960.0 4470.0 0.33 0.2833 0.8343 3614802 CMLD4_000033 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccccc2Cl)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B16 compound treatment 167800.0 1720.0 0.12 171200.0 4710.0 0.35 0.3306 0.8946 3614804 CMLD4_000034 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4cc(C)n(C)n4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B17 compound treatment 161800.0 -4280.0 -0.29 160400.0 -6090.0 -0.45 -0.527 -0.9774 3614808 CMLD4_000035 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(Br)cc2)C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B18 compound treatment 182000.0 15900.0 1.09 177680.0 11200.0 0.83 1.3562 0.9915 3614810 CMLD4_000036 O=C(NCc1ccccc1)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B19 compound treatment 202080.0 36000.0 2.45 192000.0 25500.0 1.9 3.0778 0.992 3614814 CMLD4_000037 CCCCN1C(=C(C(NC1=O)c2ccc(OC)cc2)C(=O)OCc3ccccc3)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B20 compound treatment 163200.0 -2880.0 -0.2 159320.0 -7170.0 -0.53 -0.5164 -0.9079 3614816 CMLD4_000038 O=C(NCc1ccccn1)[C@@H]2C[C@H]2[C@@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B21 compound treatment 168080.0 2000.0 0.14 166280.0 -210.0 -0.02 0.0852 0.6217 3614818 CMLD4_000039 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cc3ccccc3c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B22 compound treatment 158720.0 -7360.0 -0.5 157640.0 -8850.0 -0.66 -0.8208 -0.991 3614821 CMLD4_000040 COCCNC(=O)[C@H](C)[C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B23 mock treatment 160520.0 -5560.0 -0.38 159080.0 -7410.0 -0.55 -0.6582 -0.9833 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 B24 mock treatment 158480.0 -7600.0 -0.52 152240.0 -14300.0 -1.06 -1.1165 -0.9458 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C01 mock treatment 166240.0 156.0 0.01 161760.0 -4730.0 -0.35 -0.2414 -0.6854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C02 mock treatment 161880.0 -4200.0 -0.29 163720.0 -2770.0 -0.21 -0.3484 -0.9869 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C03 compound treatment 200600.0 34500.0 2.35 197520.0 31000.0 2.31 3.297 1.0 3614824 CMLD4_000041 COc1cc2nc-3c(Cn4c3cccc4=O)c(c2cc1OC)[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C04 compound treatment 174880.0 8800.0 0.6 165760.0 -730.0 -0.05 0.3856 0.6404 3614825 CMLD4_000042 C[C@]1(C[C@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C05 compound treatment 214920.0 48800.0 3.33 210080.0 43600.0 3.24 4.6483 0.9999 3614827 CMLD4_000043 CC(C)c1ccc2c(c3Cn4c(cccc4=O)-c3nc2c1)[Si](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C06 compound treatment 210840.0 44800.0 3.05 203840.0 37300.0 2.78 4.1233 0.9989 3614828 CMLD4_000044 COC(=O)[C@@]1(C)C[C@@H]1[C@@H](NC(=O)[C@@]2(C)C[C@@H]2[C@@H](NC(=O)[C@@]3(C)C[C@@H]3[C@@H](NC(=O)[C@@]4(C)C[C@@H]4[C@@H](NC(=O)OCc5ccccc5)c6ccccc6)c7ccccc7)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C07 compound treatment 229240.0 63200.0 4.31 229120.0 62600.0 4.66 6.3407 0.9992 3614830 CMLD4_000045 CC(C)c1cccc2c(c3Cn4c(cccc4=O)-c3nc12)[Si](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C08 compound treatment 174200.0 8120.0 0.55 167120.0 630.0 0.05 0.4244 0.7643 3614832 CMLD4_000046 COC(=O)[C@@H]1CCCN1C(=O)[C@H]2C[C@@H]2[C@H](NC(=O)OCc3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C09 compound treatment 173720.0 7640.0 0.52 173640.0 7150.0 0.53 0.7444 0.9999 3614834 CMLD4_000047 CCc1c2CC(C)Oc2nc3ccc(OC)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C10 compound treatment 162200.0 -3880.0 -0.26 162200.0 -4290.0 -0.32 -0.413 -0.9957 4981 CMLD4_000048 CNC1=C(Br)C(=O)c2ccncc2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C11 compound treatment 187040.0 21000.0 1.43 190120.0 23600.0 1.76 2.2538 0.9947 3614836 CMLD4_000049 CCCCc1c2c3ccccc3[nH]c2nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C12 compound treatment 189080.0 23000.0 1.57 193880.0 27400.0 2.04 2.5501 0.9916 3614839 CMLD4_000050 CCOC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C13 compound treatment 169080.0 3000.0 0.2 171040.0 4550.0 0.34 0.3839 0.9707 3614841 CMLD4_000051 CCc1c2COCc2nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C14 compound treatment 186200.0 20100.0 1.37 174800.0 8310.0 0.62 1.4071 0.9353 3614843 CMLD4_000052 COC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C15 compound treatment 179240.0 13200.0 0.9 173680.0 7190.0 0.54 1.0126 0.9695 3614845 CMLD4_000053 [O-][N+](=O)c1ccc(OC(=O)N2CCC(CC2)N3CCCCC3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C16 compound treatment 179480.0 13400.0 0.91 179240.0 12700.0 0.95 1.3168 0.9998 1605644 CMLD4_000054 CCOC(=O)C1=C(C)NC(=O)NC1C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C17 compound treatment 197680.0 31600.0 2.15 188240.0 21700.0 1.62 2.6678 0.9901 3614848 CMLD4_000055 O=C(/C=C/c1ccccc1)N(CC#C)Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C18 compound treatment 185240.0 19200.0 1.31 175200.0 8710.0 0.65 1.3819 0.9478 3614852 CMLD4_000056 CC1(C)OCC(CSC2=C(SCC3COC(C)(C)O3)C(=O)c4ncccc4C2=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C19 mock treatment 188240.0 22200.0 1.51 183520.0 17000.0 1.27 1.9644 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C20 compound treatment 164720.0 -1360.0 -0.09 164440.0 -2050.0 -0.15 -0.1736 -0.9718 3614855 CMLD4_000057 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C21 compound treatment 191600.0 25500.0 1.74 185480.0 19000.0 1.41 2.2295 0.9947 3614856 CMLD4_000058 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)[C@H]2C[C@@H]2[C@H](NC(=O)OCc3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C22 compound treatment 170360.0 4280.0 0.29 157480.0 -9010.0 -0.67 -0.268 -0.3665 3614859 CMLD4_000059 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OC(=O)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C23 mock treatment 159640.0 -6440.0 -0.44 155040.0 -11500.0 -0.85 -0.9132 -0.9525 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 C24 mock treatment 163520.0 -2560.0 -0.17 159040.0 -7450.0 -0.55 -0.5157 -0.887 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D01 mock treatment 161600.0 -4480.0 -0.31 159280.0 -7210.0 -0.54 -0.5956 -0.9644 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D02 mock treatment 158680.0 -7400.0 -0.5 160880.0 -5610.0 -0.42 -0.6522 -0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D03 compound treatment 179000.0 12900.0 0.88 174240.0 7750.0 0.58 1.0305 0.979 3614862 CMLD4_000060 OC(=O)C1=CC(NC(=O)N1)c2cccc(Cl)c2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D04 compound treatment 165560.0 -524.0 -0.04 162600.0 -3890.0 -0.29 -0.23 -0.7883 3614864 CMLD4_000061 OC(=O)CCCNC(=O)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D05 compound treatment 165040.0 -1040.0 -0.07 168520.0 2030.0 0.15 0.0565 0.3384 3614866 CMLD4_000062 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D06 compound treatment 185040.0 19000.0 1.29 182880.0 16400.0 1.22 1.7764 0.9996 3614867 CMLD4_000063 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D07 compound treatment 167520.0 1440.0 0.1 164600.0 -1890.0 -0.14 -0.0302 -0.1764 3614869 CMLD4_000064 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D08 compound treatment 166680.0 596.0 0.04 164120.0 -2370.0 -0.18 -0.096 -0.5302 3614871 CMLD4_000065 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCn7cc(nc7C)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D09 compound treatment 166760.0 676.0 0.05 161720.0 -4770.0 -0.36 -0.2184 -0.6101 3614876 CMLD4_000066 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(Cl)cc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D10 compound treatment 180720.0 14600.0 1.0 178920.0 12400.0 0.93 1.3597 0.9993 3614878 CMLD4_000067 COC(=O)[C@H](C)[C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D11 compound treatment 194280.0 28200.0 1.92 195920.0 29400.0 2.19 2.9081 0.9979 3614882 CMLD4_000068 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2OS(=O)(=O)c3ccc(C)cc3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D12 compound treatment 178520.0 12400.0 0.85 176880.0 10400.0 0.77 1.1463 0.9989 3614884 CMLD4_000069 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D13 compound treatment 206440.0 40400.0 2.75 200680.0 34200.0 2.54 3.7448 0.9992 3614888 CMLD4_000070 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cc3OCOc3cc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D14 compound treatment 193280.0 27200.0 1.85 172880.0 6390.0 0.48 1.6474 0.8606 3614889 CMLD4_000071 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccc(cc4)S(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D15 compound treatment 244120.0 78000.0 5.32 252640.0 86100.0 6.41 8.2959 0.9957 3614890 CMLD4_000072 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(cc2)c3ccccc3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D16 compound treatment 166160.0 76.4 0.01 169720.0 3230.0 0.24 0.1737 0.7223 3614891 CMLD4_000073 OC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D17 compound treatment 211320.0 45200.0 3.08 208880.0 42400.0 3.15 4.4116 0.9999 3614893 CMLD4_000074 CCOC(=O)C1=C(C)N(CCCC(=O)NCCn2c(C)c(cc2c3ccccc3)C(=O)OC)C(=O)NC1c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D18 compound treatment 197960.0 31900.0 2.17 190480.0 24000.0 1.79 2.7992 0.9952 3614894 CMLD4_000075 O=C(NCCc1c[nH]c2ccccc12)[C@H]3C[C@@H]3[C@H](NP(=O)(c4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D19 compound treatment 170920.0 4840.0 0.33 162280.0 -4210.0 -0.31 0.0116 0.0254 3614896 CMLD4_000076 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2)C(=O)OCC(Br)(Br)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D20 compound treatment 180360.0 14300.0 0.97 180760.0 14300.0 1.06 1.4392 0.9991 3614897 CMLD4_000077 Cc1ccc(CNC(=O)[C@@H]2C[C@H]2[C@@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D21 compound treatment 188600.0 22500.0 1.54 192280.0 25800.0 1.92 2.4427 0.9939 3614900 CMLD4_000078 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2OC(=O)c3ccc(I)cc3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D22 compound treatment 182800.0 16700.0 1.14 181840.0 15300.0 1.14 1.6137 1.0 3614902 CMLD4_000079 COc1ccc(CNC(=O)[C@H](C)[C@H]2C[C@]2(C)[C@H](NC(=O)OCc3ccccc3)c4ccccc4)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D23 mock treatment 161280.0 -4800.0 -0.33 157920.0 -8570.0 -0.64 -0.6826 -0.952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 D24 mock treatment 160920.0 -5160.0 -0.35 158480.0 -8010.0 -0.6 -0.6705 -0.9684 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E01 mock treatment 171240.0 5160.0 0.35 169920.0 3430.0 0.26 0.4291 0.9876 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E02 mock treatment 163040.0 -3040.0 -0.21 169760.0 3270.0 0.24 0.0253 0.0793 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E03 compound treatment 235000.0 68900.0 4.7 230960.0 64500.0 4.8 6.7152 0.9999 3614906 CMLD4_000080 CN(C)c1ccc2nc-3c(Cn4c3cccc4=O)c(c2c1)[Si](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E04 compound treatment 178080.0 12000.0 0.82 174280.0 7790.0 0.58 0.9883 0.9858 3614908 CMLD4_000081 COC(=O)[C@]1(C)C[C@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E05 compound treatment 225000.0 58900.0 4.02 227440.0 60900.0 4.54 6.0479 0.9982 3614912 CMLD4_000082 CCc1cccc2nc-3c(Cn4c3cccc4=O)c(c12)[Si](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E06 compound treatment 176040.0 9960.0 0.68 173240.0 6750.0 0.5 0.8352 0.989 3614914 CMLD4_000083 CC(C)NC(=O)[C@]1(C)C[C@H]1[C@H](NC(=O)[C@]2(C)C[C@H]2[C@H](NC(=O)OCc3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E07 compound treatment 241880.0 75800.0 5.17 253560.0 87100.0 6.48 8.2363 0.9937 3614917 CMLD4_000084 CC(C)c1cccc2nc-3c(Cn4c3cccc4=O)c(c12)[Si](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E08 compound treatment 179200.0 13100.0 0.89 173520.0 7030.0 0.52 1.0023 0.9674 3614919 CMLD4_000085 CN(C)C(=O)[C@H]1C[C@@H]1[C@H](NC(=O)CNC(=O)[C@@H]2CCCN2C(=O)[C@H]3C[C@@H]3[C@H](NC(=O)OCc4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E09 compound treatment 202120.0 36000.0 2.46 199240.0 32700.0 2.44 3.4608 1.0 3614923 CMLD4_000086 COc1ccc2nc3CCCc3c(c4ccccc4)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E10 compound treatment 163200.0 -2880.0 -0.2 162640.0 -3850.0 -0.29 -0.3416 -0.9831 4982 CMLD4_000087 CNC1=C(Cl)C(=O)c2ccncc2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E11 compound treatment 203160.0 37100.0 2.53 208920.0 42400.0 3.16 4.0204 0.9939 3614925 CMLD4_000088 CCC1Cc2c(O1)nc3cccc(OC)c3c2CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E12 compound treatment 219240.0 53200.0 3.62 219640.0 53100.0 3.96 5.3597 0.999 3614926 CMLD4_000089 CCOC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E13 compound treatment 185600.0 19500.0 1.33 186920.0 20400.0 1.52 2.016 0.9978 3614928 CMLD4_000090 CC(C)c1cccc2nc-3c(Cn4c3cccc4=O)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E14 compound treatment 203960.0 37900.0 2.58 198160.0 31700.0 2.36 3.4927 0.999 3614930 CMLD4_000091 COC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E15 compound treatment 192840.0 26800.0 1.82 190160.0 23700.0 1.76 2.5356 0.9998 1071887 CMLD4_000092 O=c1cccc2-c3nc4ccccc4cc3Cn21 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E16 compound treatment 208680.0 42600.0 2.9 207880.0 41400.0 3.08 4.2317 0.9996 3614934 CMLD4_000093 CCOC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E17 compound treatment 197440.0 31400.0 2.14 199440.0 32900.0 2.45 3.2457 0.9977 3614936 CMLD4_000094 CC(C#C)N(Cc1ccccc1)C(=O)/C=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E18 compound treatment 175280.0 9200.0 0.63 173800.0 7310.0 0.54 0.828 0.9975 3614939 CMLD4_000095 ClC1=C(NCCN2CCOCC2)C(=O)c3cnncc3C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E19 compound treatment 171520.0 5440.0 0.37 172520.0 6030.0 0.45 0.5794 0.9955 3614941 CMLD4_000096 OCC[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E20 compound treatment 175160.0 9080.0 0.62 177200.0 10700.0 0.8 1.0012 0.9922 3614943 CMLD4_000097 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1C(CC)CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E21 compound treatment 216000.0 49900.0 3.4 211640.0 45100.0 3.36 4.7825 1.0 3614944 CMLD4_000098 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccc(cc4)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E22 compound treatment 171600.0 5520.0 0.38 168880.0 2390.0 0.18 0.3917 0.9415 3614946 CMLD4_000099 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OC(=O)c3cccc(I)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E23 mock treatment 168520.0 2440.0 0.17 166000.0 -490.0 -0.04 0.0916 0.5389 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 E24 mock treatment 167080.0 996.0 0.07 164800.0 -1690.0 -0.13 -0.0409 -0.2862 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F01 mock treatment 164600.0 -1480.0 -0.1 166080.0 -410.0 -0.03 -0.0931 -0.8813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F02 mock treatment 167320.0 1240.0 0.08 171760.0 5270.0 0.39 0.3369 0.8399 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F03 compound treatment 178440.0 12400.0 0.84 172000.0 5510.0 0.41 0.8856 0.9453 3614947 CMLD4_000100 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F04 compound treatment 173680.0 7600.0 0.52 172120.0 5630.0 0.42 0.6625 0.9945 3614948 CMLD4_000101 NC(=O)NCc1ccc(cc1)C(=O)OCc2ccncc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F05 compound treatment 172560.0 6480.0 0.44 169640.0 3150.0 0.23 0.478 0.9561 3614949 CMLD4_000102 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F06 compound treatment 198080.0 32000.0 2.18 199320.0 32800.0 2.44 3.2702 0.9984 3614950 CMLD4_000103 CCC/C=C(\CCC)/C(NC(=O)c1ccco1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F07 compound treatment 178240.0 12200.0 0.83 173280.0 6790.0 0.51 0.9434 0.9718 3614952 CMLD4_000104 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F08 compound treatment 207120.0 41000.0 2.8 207960.0 41500.0 3.09 4.1608 0.9988 3614953 CMLD4_000105 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)N[C@@H](CO)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F09 compound treatment 174320.0 8240.0 0.56 174400.0 7910.0 0.59 0.8133 0.9997 3614957 CMLD4_000106 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2Cl)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F10 compound treatment 182240.0 16200.0 1.1 185600.0 19100.0 1.42 1.7846 0.992 3614959 CMLD4_000107 COC(=O)[C@H](C)[C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F11 compound treatment 193560.0 27500.0 1.87 191200.0 24700.0 1.84 2.625 1.0 3614961 CMLD4_000108 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2OS(=O)(=O)c3ccccc3[N+](=O)[O-])C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F12 compound treatment 191240.0 25200.0 1.72 189320.0 22800.0 1.7 2.4142 1.0 3614963 CMLD4_000109 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccc(C)o4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F13 compound treatment 185600.0 19500.0 1.33 183120.0 16600.0 1.24 1.816 0.9993 3614967 CMLD4_000110 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccccc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F14 compound treatment 181240.0 15200.0 1.03 183440.0 16900.0 1.26 1.6227 0.9951 3614968 CMLD4_000111 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F15 compound treatment 181360.0 15300.0 1.04 183240.0 16700.0 1.25 1.6179 0.996 3614971 CMLD4_000112 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(cc2)[N+](=O)[O-])C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F16 compound treatment 179120.0 13000.0 0.89 173840.0 7350.0 0.55 1.0153 0.9728 3614973 CMLD4_000113 CNC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F17 compound treatment 226800.0 60700.0 4.14 228960.0 62500.0 4.65 6.2147 0.9983 3614976 CMLD4_000114 CCOC(=O)C1=C(C)N(CCCC(=O)NCCn2c(C)c(cc2c3ccccc3)C(=O)OC)C(=O)NC1c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F18 compound treatment 181000.0 14900.0 1.02 178600.0 12100.0 0.9 1.3564 0.9982 3614979 CMLD4_000115 O=C(NCC1CC1)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F19 compound treatment 183800.0 17700.0 1.21 192320.0 25800.0 1.92 2.2134 0.9749 3614983 CMLD4_000116 CC1=C(C(NC(=O)N1CCCC(=O)O)c2cccc3ccccc23)C(=O)OCC(Br)(Br)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F20 compound treatment 172360.0 6280.0 0.43 173280.0 6790.0 0.51 0.6599 0.9966 3614985 CMLD4_000117 C[C@H](CO)NC(=O)[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F21 compound treatment 179040.0 13000.0 0.88 178680.0 12200.0 0.91 1.2661 0.9999 3614990 CMLD4_000118 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F22 compound treatment 181200.0 15100.0 1.03 184960.0 18500.0 1.37 1.7008 0.9899 3614992 CMLD4_000119 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccc(C)c(F)c4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F23 mock treatment 167720.0 1640.0 0.11 163680.0 -2810.0 -0.21 -0.069 -0.2911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 F24 mock treatment 165640.0 -444.0 -0.03 160640.0 -5850.0 -0.44 -0.3293 -0.7544 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G01 mock treatment 168720.0 2640.0 0.18 174520.0 8030.0 0.6 0.5497 0.8808 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G02 mock treatment 174080.0 8000.0 0.55 176200.0 9710.0 0.72 0.8965 0.9903 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G03 compound treatment 247000.0 80900.0 5.52 247760.0 81300.0 6.05 8.1779 0.9989 3614996 CMLD4_000120 CC(C)(C)[Si](C)(C)c1c2Cn3c(cccc3=O)-c2nc4ccc(OCc5ccccc5)cc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G04 compound treatment 181880.0 15800.0 1.08 189240.0 22700.0 1.69 1.9588 0.9761 3614998 CMLD4_000121 COC(=O)[C@]1(C)C[C@H]1[C@H](NC(=O)c2ccc(Br)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G05 compound treatment 196240.0 30200.0 2.06 194840.0 28300.0 2.11 2.9458 0.9999 3615000 CMLD4_000122 CC[Si](CC)(CC)c1c2Cn3c(cccc3=O)-c2nc4ccc(OC)cc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G06 compound treatment 188080.0 22000.0 1.5 184800.0 18300.0 1.36 2.024 0.9989 3615001 CMLD4_000123 CNC(=O)[C@]1(C)C[C@H]1[C@H](NC(=O)[C@]2(C)C[C@H]2[C@H](NC(=O)OCc3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G07 compound treatment 210880.0 44800.0 3.05 217680.0 51200.0 3.81 4.8536 0.994 3615005 CMLD4_000124 CCc1c2Cn3c(cccc3=O)-c2nc4c(cccc14)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G08 compound treatment 187520.0 21400.0 1.46 178280.0 11800.0 0.88 1.6539 0.9702 3615006 CMLD4_000125 COC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G09 compound treatment 185320.0 19200.0 1.31 183320.0 16800.0 1.25 1.8131 0.9997 3615008 CMLD4_000126 CCCCC#Cc1ccccc1CC(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G10 compound treatment 174360.0 8280.0 0.56 170720.0 4230.0 0.31 0.6216 0.962 4983 CMLD4_000127 OCCNC1=CC(=O)c2ccncc2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G11 compound treatment 187200.0 21100.0 1.44 188360.0 21900.0 1.63 2.1689 0.9981 3615009 CMLD4_000128 CCC1Cc2c(O1)nc3ccc(OC)cc3c2CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G12 compound treatment 208200.0 42100.0 2.87 198200.0 31700.0 2.36 3.6992 0.9953 3615010 CMLD4_000129 CCOC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G13 compound treatment 195920.0 29800.0 2.03 197600.0 31100.0 2.32 3.0756 0.9979 3615011 CMLD4_000130 CC(C)c1cccc2cc3Cn4c(cccc4=O)-c3nc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G14 compound treatment 202120.0 36000.0 2.46 201400.0 34900.0 2.6 3.5745 0.9996 3615012 CMLD4_000131 COC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G15 compound treatment 97680.0 -68400.0 -4.66 111200.0 -55300.0 -4.12 -6.2074 -0.9981 3615014 CMLD4_000132 C1Oc2cc3cc4Cc5ccccc5-c4nc3cc2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G16 compound treatment 192360.0 26300.0 1.79 180600.0 14100.0 1.05 2.0093 0.9676 3615016 CMLD4_000133 CC(=O)OCC(=O)NCC(=O)c1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G17 compound treatment 187560.0 21500.0 1.46 181200.0 14700.0 1.09 1.8095 0.9897 3615017 CMLD4_000134 CC(C)OC1=C(OC(C)C)C(O)(C#CCN(C(=O)/C=C/c2ccccc2)C(C)(C)C)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G18 compound treatment 180640.0 14600.0 0.99 186400.0 19900.0 1.48 1.7495 0.981 3615021 CMLD4_000135 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G19 compound treatment 192200.0 26100.0 1.78 186520.0 20000.0 1.49 2.3131 0.9961 3615024 CMLD4_000136 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccc(Br)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G20 compound treatment 184720.0 18600.0 1.27 178320.0 11800.0 0.88 1.521 0.9839 1237977 CMLD4_000137 CCOC(=O)C1=C(C)NC(=O)NC1c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G21 compound treatment 184760.0 18700.0 1.27 183040.0 16500.0 1.23 1.7713 0.9999 3615028 CMLD4_000138 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)c2ccccc2)c3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G22 compound treatment 175640.0 9560.0 0.65 173040.0 6550.0 0.49 0.8054 0.9898 3615032 CMLD4_000139 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(Cl)cc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G23 mock treatment 171200.0 5120.0 0.35 172120.0 5630.0 0.42 0.5429 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 G24 mock treatment 166560.0 476.0 0.03 163120.0 -3370.0 -0.25 -0.1544 -0.6105 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H01 mock treatment 166920.0 836.0 0.06 168240.0 1750.0 0.13 0.1324 0.9314 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H02 mock treatment 171760.0 5680.0 0.39 171560.0 5070.0 0.38 0.5405 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H03 compound treatment 176440.0 10400.0 0.71 172000.0 5510.0 0.41 0.7892 0.9666 3615033 CMLD4_000140 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H04 compound treatment 178480.0 12400.0 0.85 179880.0 13400.0 1.0 1.3023 0.9966 3615034 CMLD4_000141 NCC#CC(CCc1ccccc1)OCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H05 compound treatment 175160.0 9080.0 0.62 175640.0 9150.0 0.68 0.9191 0.9989 3615036 CMLD4_000142 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cccc(OC)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H06 compound treatment 189720.0 23600.0 1.61 188320.0 21800.0 1.62 2.2883 1.0 1965336 CMLD4_000143 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)Cc2ccccc2)c3ccc(cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H07 compound treatment 211040.0 45000.0 3.06 208440.0 41900.0 3.12 4.375 1.0 3615038 CMLD4_000144 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H08 compound treatment 181560.0 15500.0 1.06 185280.0 18800.0 1.4 1.7349 0.9904 3615040 CMLD4_000145 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)N[C@@H](CO)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H09 compound treatment 217800.0 51700.0 3.53 209080.0 42600.0 3.17 4.7346 0.9986 3615042 CMLD4_000146 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(cc2)c3ccccc3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H10 compound treatment 176040.0 9960.0 0.68 177280.0 10800.0 0.8 1.0478 0.9965 3615006 CMLD4_000147 COC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H11 compound treatment 194000.0 27900.0 1.9 188760.0 22300.0 1.66 2.5178 0.9976 3615045 CMLD4_000148 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2OS(=O)(=O)c3ccc(cc3)[N+](=O)[O-])C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H12 compound treatment 176560.0 10500.0 0.71 180640.0 14100.0 1.05 1.2497 0.9821 3615047 CMLD4_000149 C[C@H](CO)NC(=O)[C@H](C)[C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H13 compound treatment 181400.0 15300.0 1.04 178920.0 12400.0 0.93 1.3925 0.9982 3615049 CMLD4_000150 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cccc(Cl)c2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H14 compound treatment 200280.0 34200.0 2.33 193760.0 27300.0 2.03 3.0837 0.9976 3615050 CMLD4_000151 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccc(C)o4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H15 compound treatment 193160.0 27100.0 1.85 195080.0 28600.0 2.13 2.8099 0.9975 3615051 CMLD4_000152 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2cccc(Cl)c2Cl)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H16 compound treatment 202880.0 36800.0 2.51 205560.0 39100.0 2.91 3.83 0.9973 3615052 CMLD4_000153 O=C(Nc1ccc2ccccc2c1)[C@H]3C[C@@H]3[C@H](NP(=O)(c4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H17 compound treatment 208880.0 42800.0 2.92 201520.0 35000.0 2.61 3.9067 0.9984 3615054 CMLD4_000154 COC(=O)c1cc(c2ccccc2)n(CCNC(=O)CCCCCN3C(=C(C(NC3=O)c4ccc(cc4)c5ccccc5)C(=O)OCc6ccccc6)C)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H18 compound treatment 182040.0 16000.0 1.09 177680.0 11200.0 0.83 1.3581 0.9913 3615057 CMLD4_000155 Cc1cc(CNC(=O)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)nn1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H19 compound treatment 176200.0 10100.0 0.69 182840.0 16300.0 1.22 1.3481 0.9638 3615059 CMLD4_000156 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(Br)cc2)C(=O)OCC(Br)(Br)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H20 compound treatment 188240.0 22200.0 1.51 192680.0 26200.0 1.95 2.4464 0.9921 3615061 CMLD4_000157 O=C(NCc1ccccc1)[C@@H]2C[C@H]2[C@@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H21 compound treatment 211240.0 45200.0 3.08 212720.0 46200.0 3.44 4.6099 0.9985 3615063 CMLD4_000158 CCOC(=O)C(=CNc1ccc(O)c(c1)C(=O)OC)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H22 compound treatment 196400.0 30300.0 2.07 191960.0 25500.0 1.9 2.8019 0.9991 3615065 CMLD4_000159 COc1ccc(CNC(=O)[C@H](C)[C@@H]2C[C@@]2(C)[C@@H](NC(=O)OCc3ccccc3)c4ccccc4)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H23 mock treatment 167800.0 1720.0 0.12 170640.0 4150.0 0.31 0.3011 0.9118 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 H24 mock treatment 163520.0 -2560.0 -0.17 166000.0 -490.0 -0.04 -0.1494 -0.8367 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I01 mock treatment 166760.0 676.0 0.05 170720.0 4230.0 0.31 0.2552 0.8021 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I02 mock treatment 173080.0 7000.0 0.48 170040.0 3550.0 0.26 0.5241 0.9612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I03 compound treatment 191480.0 25400.0 1.73 186880.0 20400.0 1.52 2.2974 0.9978 3615067 CMLD4_000160 CC(C)(C)[Si](C)(C)c1c2Cn3c(cccc3=O)-c2nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I04 compound treatment 187440.0 21400.0 1.46 186720.0 20200.0 1.51 2.0942 0.9999 3615069 CMLD4_000161 COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@]2(C)C[C@H]2[C@H](NC(=O)OCc3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I05 compound treatment 206160.0 40100.0 2.73 211240.0 44700.0 3.33 4.2871 0.9952 3615073 CMLD4_000162 CCc1c2Cn3c(cccc3=O)-c2nc4ccc(cc14)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I06 compound treatment 182840.0 16800.0 1.14 179160.0 12700.0 0.94 1.4746 0.9955 3615075 CMLD4_000163 CN(C)C(=C)[C@]1(C)C[C@H]1[C@H](NC(=O)CNC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I07 compound treatment 233200.0 67100.0 4.58 233200.0 66700.0 4.96 6.7464 0.9992 3615079 CMLD4_000164 CCc1c2Cn3c(cccc3=O)-c2nc4cccc(C(C)C)c14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I08 compound treatment 180000.0 13900.0 0.95 176600.0 10100.0 0.75 1.2029 0.9934 3615081 CMLD4_000165 OC[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I09 compound treatment 175280.0 9200.0 0.63 177640.0 11100.0 0.83 1.0301 0.9904 3615085 CMLD4_000166 Nc1ccccc1C#Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I10 compound treatment 209600.0 43500.0 2.97 207640.0 41100.0 3.06 4.2635 0.9999 3615087 CMLD4_000167 CCOC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I11 compound treatment 194680.0 28600.0 1.95 201200.0 34700.0 2.58 3.2053 0.9904 3615089 CMLD4_000168 COc1ccc(NC(=O)CCCCC#Cc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I12 compound treatment 240320.0 74200.0 5.06 236800.0 70300.0 5.23 7.2791 0.9999 3615091 CMLD4_000169 CCOC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I13 compound treatment 181480.0 15400.0 1.05 182920.0 16400.0 1.22 1.6069 0.9971 3615093 CMLD4_000170 O=C(CCCC#C)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I14 compound treatment 202280.0 36200.0 2.47 201240.0 34700.0 2.59 3.5738 0.9997 3615094 CMLD4_000171 COC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I15 compound treatment 218840.0 52800.0 3.6 223640.0 57100.0 4.25 5.551 0.9965 3615095 CMLD4_000172 Cc1c2Cn3c(cccc3=O)-c2nc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I16 compound treatment 208120.0 42000.0 2.87 210680.0 44200.0 3.29 4.3521 0.9976 3615096 CMLD4_000173 CCOC(=O)n1cc(c2cnc(CNC(=O)C(C)(c3ccccc3)c4ccccc4)o2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I17 compound treatment 181120.0 15000.0 1.03 180160.0 13700.0 1.02 1.4443 1.0 3615097 CMLD4_000174 COc1ccc(CN([C@@H](CO[Si](c2ccccc2)(c3ccccc3)C(C)(C)C)c4cccc(NC(=O)C)c4OC)C(=O)CO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I18 compound treatment 182560.0 16500.0 1.12 178280.0 11800.0 0.88 1.4148 0.9925 3615099 CMLD4_000175 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I19 compound treatment 206480.0 40400.0 2.75 199560.0 33100.0 2.46 3.6878 0.9984 3615100 CMLD4_000176 C[C@H](NC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I20 compound treatment 189240.0 23200.0 1.58 190920.0 24400.0 1.82 2.402 0.9975 3615102 CMLD4_000177 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccc(Cl)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I21 compound treatment 188080.0 22000.0 1.5 186880.0 20400.0 1.52 2.1335 1.0 3615104 CMLD4_000178 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NS(=O)(=O)c2ccccc2)c3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I22 compound treatment 180520.0 14400.0 0.98 174200.0 7710.0 0.57 1.1017 0.967 3615107 CMLD4_000179 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I23 mock treatment 170600.0 4520.0 0.31 172400.0 5910.0 0.44 0.5287 0.9848 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 I24 mock treatment 167760.0 1680.0 0.11 164200.0 -2290.0 -0.17 -0.0397 -0.1935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J01 mock treatment 167200.0 1120.0 0.08 170320.0 3830.0 0.29 0.2554 0.8656 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J02 mock treatment 170840.0 4760.0 0.32 170480.0 3990.0 0.3 0.4393 0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J03 compound treatment 175200.0 9120.0 0.62 177280.0 10800.0 0.8 1.0073 0.992 3615110 CMLD4_000180 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(OC)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J04 compound treatment 209680.0 43600.0 2.97 209960.0 43500.0 3.24 4.3894 0.9991 3615111 CMLD4_000181 O=C(NCC#CC(CCc1ccccc1)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J05 compound treatment 180720.0 14600.0 1.0 177680.0 11200.0 0.83 1.2945 0.996 3615114 CMLD4_000182 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(cc2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J06 compound treatment 175240.0 9160.0 0.62 179640.0 13100.0 0.98 1.1335 0.9764 1965280 CMLD4_000183 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C[C@H](O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J07 compound treatment 256480.0 90400.0 6.16 252080.0 85600.0 6.37 8.8623 0.9999 3615115 CMLD4_000184 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J08 compound treatment 193680.0 27600.0 1.88 189120.0 22600.0 1.68 2.5213 0.9985 3615117 CMLD4_000185 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4nc5ccccc5[nH]4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J09 compound treatment 178400.0 12300.0 0.84 177120.0 10600.0 0.79 1.1532 0.9996 3615122 CMLD4_000186 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(C#N)cc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J10 compound treatment 178560.0 12500.0 0.85 183160.0 16700.0 1.24 1.4788 0.983 3615124 CMLD4_000187 COC(=O)[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J11 compound treatment 183360.0 17300.0 1.18 185040.0 18500.0 1.38 1.8091 0.9969 3615125 CMLD4_000188 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccc(cc2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J12 compound treatment 197280.0 31200.0 2.13 195400.0 28900.0 2.15 3.0254 1.0 3615127 CMLD4_000189 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J13 compound treatment 179600.0 13500.0 0.92 180160.0 13700.0 1.02 1.371 0.9988 3615130 CMLD4_000190 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J14 compound treatment 174080.0 8000.0 0.55 176880.0 10400.0 0.77 0.9323 0.9854 3615131 CMLD4_000191 C[C@H](CO)NC(=O)[C@H](C)[C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J15 compound treatment 213760.0 47700.0 3.25 214720.0 48200.0 3.59 4.8366 0.9988 3615134 CMLD4_000192 CCOC(=O)C1=C(C)N(CCCC(=O)NCc2ccc3OCOc3c2)C(=O)NC1c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J16 compound treatment 191800.0 25700.0 1.75 189240.0 22700.0 1.69 2.437 0.9998 3615135 CMLD4_000193 CS(=O)(=O)c1ccc(CNC(=O)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J17 compound treatment 193120.0 27000.0 1.84 190520.0 24000.0 1.79 2.568 0.9999 3615140 CMLD4_000194 CCOC(=O)C1=C(C)N(CCCC(=O)NCCn2c(C)c(cc2c3ccccc3)C(=O)OC(C)(C)C)C(=O)NC1c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J18 compound treatment 177240.0 11200.0 0.76 175040.0 8550.0 0.64 0.9878 0.9961 3615142 CMLD4_000195 OC(=O)[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J19 compound treatment 208200.0 42100.0 2.87 202440.0 35900.0 2.68 3.9223 0.9994 3615143 CMLD4_000196 CCOC(=O)C1=C(C)N(Cc2ccccc2)C(=O)NC1c3ccccc3OS(=O)(=O)c4ccccc4[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J20 compound treatment 202440.0 36400.0 2.48 195640.0 29100.0 2.17 3.2868 0.9978 3615145 CMLD4_000197 O=C(NCCc1c[nH]c2ccccc12)[C@@H]3C[C@H]3[C@@H](NP(=O)(c4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J21 compound treatment 172080.0 6000.0 0.41 170960.0 4470.0 0.33 0.5243 0.9948 3615147 CMLD4_000198 CCOC(=O)C(=CN(CCc1ccccc1)CC(=O)OC)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J22 compound treatment 187680.0 21600.0 1.47 181960.0 15500.0 1.15 1.8553 0.9926 3615148 CMLD4_000199 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccc(C)c(F)c4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J23 mock treatment 165920.0 -164.0 -0.01 166800.0 310.0 0.02 0.0084 0.3284 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 J24 mock treatment 161480.0 -4600.0 -0.31 164920.0 -1570.0 -0.12 -0.3046 -0.9094 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K01 mock treatment 173720.0 7640.0 0.52 168400.0 1910.0 0.14 0.4686 0.8684 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K02 mock treatment 174960.0 8880.0 0.61 170960.0 4470.0 0.33 0.6631 0.9603 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K03 compound treatment 186280.0 20200.0 1.38 181840.0 15300.0 1.14 1.7815 0.9957 3615149 CMLD4_000200 CC(C)(C)[Si](C)(C)c1c2Cn3c(cccc3=O)-c2nc4cc5OCCOc5cc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K04 compound treatment 238440.0 72400.0 4.93 234280.0 67800.0 5.05 7.0558 0.9999 3615150 CMLD4_000201 CNC(=O)[C@]1(C)C[C@H]1[C@H](NC(=O)[C@]2(C)C[C@H]2[C@H](NC(=O)[C@]3(C)C[C@H]3[C@H](NC(=O)[C@]4(C)C[C@H]4[C@H](NC(=O)OCc5ccccc5)c6ccccc6)c7ccccc7)c8ccccc8)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K05 compound treatment 197160.0 31100.0 2.12 194280.0 27800.0 2.07 2.9606 0.9999 3615154 CMLD4_000202 CSc1ccc2nc-3c(Cn4c3cccc4=O)c(c2c1)[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K06 compound treatment 193880.0 27800.0 1.9 198600.0 32100.0 2.39 3.0299 0.9934 3615155 CMLD4_000203 COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@]2(C)C[C@@H]2[C@@H](NC(=O)OCc3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K07 compound treatment 222920.0 56800.0 3.87 224640.0 58100.0 4.33 5.8003 0.9985 3615156 CMLD4_000204 CC(C)c1cccc2nc-3c(Cn4c3cccc4=O)c(c12)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K08 compound treatment 236760.0 70700.0 4.82 230640.0 64100.0 4.77 6.7832 1.0 3615157 CMLD4_000205 CCCC/C(=C/[C@@H](NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K09 compound treatment 195640.0 29600.0 2.02 190400.0 23900.0 1.78 2.6832 0.9981 3615159 CMLD4_000206 Nc1ccccc1C#CCCCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K10 compound treatment 205920.0 39800.0 2.72 201040.0 34500.0 2.57 3.7387 0.9996 3615160 CMLD4_000207 COC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K11 compound treatment 185760.0 19700.0 1.34 188560.0 22100.0 1.64 2.11 0.9949 3615163 CMLD4_000208 Ic1ccccc1CC(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K12 compound treatment 190080.0 24000.0 1.64 185560.0 19100.0 1.42 2.1604 0.9975 3615164 CMLD4_000209 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K13 compound treatment 191000.0 24900.0 1.7 184760.0 18300.0 1.36 2.1627 0.9939 3615166 CMLD4_000210 S=C(CCCC#C)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K14 compound treatment 210160.0 44100.0 3.0 208160.0 41700.0 3.1 4.3178 0.9999 3615167 CMLD4_000211 CCOC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K15 compound treatment 149120.0 -17000.0 -1.16 145480.0 -21000.0 -1.56 -1.9235 -0.989 3615169 CMLD4_000212 COc1ccc2nc-3c(Cc4ccccc43)cc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K16 compound treatment 178200.0 12100.0 0.83 173320.0 6830.0 0.51 0.9435 0.9728 3615171 CMLD4_000213 NC(=N)NCCC[C@H](NC(=O)OCc1ccccc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K17 compound treatment 181200.0 15100.0 1.03 178520.0 12000.0 0.9 1.3618 0.9975 3615174 CMLD4_000214 COc1ccc(/C=C/C(=O)NCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K18 compound treatment 182240.0 16200.0 1.1 175120.0 8630.0 0.64 1.233 0.967 3615177 CMLD4_000215 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(cc2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K19 compound treatment 240040.0 74000.0 5.04 237560.0 71100.0 5.29 7.3056 0.9997 3615179 CMLD4_000216 COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]2C[C@H]2[C@@H](NC(=O)OCc3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K20 compound treatment 174800.0 8720.0 0.59 176680.0 10200.0 0.76 0.9565 0.9927 3615184 CMLD4_000217 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(Br)cc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K21 compound treatment 178280.0 12200.0 0.83 187520.0 21000.0 1.57 1.6947 0.9562 3615186 CMLD4_000218 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)Oc2ccccc2)c3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K22 compound treatment 169760.0 3680.0 0.25 170760.0 4270.0 0.32 0.4019 0.9931 3615190 CMLD4_000219 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2OC(=O)c3cccs3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K23 mock treatment 162560.0 -3520.0 -0.24 171520.0 5030.0 0.37 0.0948 0.2132 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 K24 mock treatment 163920.0 -2160.0 -0.15 164520.0 -1970.0 -0.15 -0.208 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L01 mock treatment 170280.0 4200.0 0.29 168760.0 2270.0 0.17 0.3217 0.9684 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L02 mock treatment 172520.0 6440.0 0.44 173000.0 6510.0 0.48 0.6529 0.9988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L03 compound treatment 177240.0 11200.0 0.76 176200.0 9710.0 0.72 1.0488 0.9997 3615192 CMLD4_000220 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L04 compound treatment 178680.0 12600.0 0.86 179760.0 13300.0 0.99 1.3056 0.9976 3615193 CMLD4_000221 OC(C#CCNC(=O)CCc1ccccc1)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L05 compound treatment 178320.0 12200.0 0.83 180360.0 13900.0 1.03 1.3198 0.9944 3615195 CMLD4_000222 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L06 compound treatment 177040.0 11000.0 0.75 176400.0 9910.0 0.74 1.0497 1.0 3615197 CMLD4_000223 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5[nH]c(cc35)C(=O)N6CCCC6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L07 compound treatment 181440.0 15400.0 1.05 182560.0 16100.0 1.2 1.586 0.9978 3615201 CMLD4_000224 CCOC(=O)C1=C(C)N(Cc2ccc(cc2)C(=O)O)C(=O)NC1c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L08 compound treatment 178640.0 12600.0 0.86 181280.0 14800.0 1.1 1.3837 0.9923 3615203 CMLD4_000225 O=C(N[C@H]([C@@H]1C[C@H]1C(=O)NCc2ccccc2)c3ccccc3)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L09 compound treatment 178240.0 12200.0 0.83 181600.0 15100.0 1.12 1.3812 0.9887 3615205 CMLD4_000226 COc1cccc(c1)C2NC(=O)N(CCCC(=O)O)C(=C2C(=O)OCc3ccccc3)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L10 compound treatment 179120.0 13000.0 0.89 180840.0 14300.0 1.07 1.3837 0.9958 3615207 CMLD4_000227 COCCNC(=O)[C@H](C)[C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L11 compound treatment 180840.0 14800.0 1.01 176000.0 9510.0 0.71 1.2119 0.9852 3615209 CMLD4_000228 CCOC(=O)C1=C(C)N(CCC(=O)O)C(=O)NC1c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L12 compound treatment 202040.0 36000.0 2.45 197640.0 31100.0 2.32 3.3727 0.9996 3615210 CMLD4_000229 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCCc4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L13 compound treatment 202360.0 36300.0 2.47 201600.0 35100.0 2.61 3.5966 0.9996 3615214 CMLD4_000230 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(Cl)cc2Cl)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L14 compound treatment 201240.0 35200.0 2.4 208680.0 42200.0 3.14 3.9152 0.9911 3615217 CMLD4_000231 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L15 compound treatment 251920.0 85800.0 5.85 238800.0 72300.0 5.38 7.9435 0.9991 3615218 CMLD4_000232 CCOC(=O)C1=C(C)N(CCCC(=O)N(Cc2ccc3OCOc3c2)C(C(=O)NC(C)(C)C)c4ccc5OCOc5c4)C(=O)NC1c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L16 compound treatment 177920.0 11800.0 0.81 180080.0 13600.0 1.01 1.2858 0.9937 3615220 CMLD4_000233 O=C(NCc1ccccn1)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L17 compound treatment 176880.0 10800.0 0.74 172760.0 6270.0 0.47 0.8504 0.9758 3615222 CMLD4_000234 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2cccc(c2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L18 compound treatment 179720.0 13600.0 0.93 177680.0 11200.0 0.83 1.2463 0.9985 3615224 CMLD4_000235 CNC(=O)[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L19 compound treatment 193960.0 27900.0 1.9 187320.0 20800.0 1.55 2.4401 0.9949 3615226 CMLD4_000236 CCCCN1C(=C(C(NC1=O)c2cccc(c2)[N+](=O)[O-])C(=O)OCC)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L20 compound treatment 177400.0 11300.0 0.77 172320.0 5830.0 0.43 0.8523 0.9629 3615228 CMLD4_000237 O=C(NCC1CC1)[C@@H]2C[C@H]2[C@@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L21 compound treatment 177480.0 11400.0 0.78 172400.0 5910.0 0.44 0.8604 0.9637 3615230 CMLD4_000238 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2ccccc2OC(=O)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L22 compound treatment 168240.0 2160.0 0.15 168800.0 2310.0 0.17 0.2255 0.997 3615232 CMLD4_000239 FCCNC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L23 mock treatment 165560.0 -524.0 -0.04 162000.0 -4490.0 -0.33 -0.2616 -0.7782 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 L24 mock treatment 162200.0 -3880.0 -0.26 158520.0 -7970.0 -0.59 -0.6067 -0.9339 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M01 mock treatment 165840.0 -244.0 -0.02 176120.0 9630.0 0.72 0.495 0.6905 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M02 mock treatment 175720.0 9640.0 0.66 175880.0 9390.0 0.7 0.9587 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M03 compound treatment 199720.0 33600.0 2.29 199880.0 33400.0 2.49 3.3788 0.9992 3615236 CMLD4_000240 CCCCC#Cc1ccccc1NC(=S)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M04 compound treatment 179640.0 13600.0 0.92 184120.0 17600.0 1.31 1.5813 0.9853 3615237 CMLD4_000241 C[C@]1(C[C@H]1CCO)[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M05 compound treatment 198320.0 32200.0 2.2 191120.0 24600.0 1.83 2.8503 0.9959 3615242 CMLD4_000242 Cc1ccc2nc-3c(Cn4c3cccc4=O)c(c2c1)[Si](C)(C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M06 compound treatment 190240.0 24200.0 1.65 189760.0 23300.0 1.73 2.3892 0.9997 3615244 CMLD4_000243 COC(=O)[C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M07 compound treatment 231160.0 65100.0 4.44 224800.0 58300.0 4.34 6.2059 0.9999 3615247 CMLD4_000244 CN(C)c1ccc2nc-3c(Cn4c3cccc4=O)c(c2c1)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M08 compound treatment 202200.0 36100.0 2.46 207480.0 41000.0 3.05 3.8983 0.9944 3615249 CMLD4_000245 C/C(=C\[C@@H](NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3)/CO[Si](c4ccccc4)(c5ccccc5)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M09 compound treatment 205280.0 39200.0 2.67 207520.0 41000.0 3.05 4.0489 0.9978 3615253 CMLD4_000246 S=C(Nc1ccccc1)Nc2ccccc2C#Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M10 compound treatment 214320.0 48200.0 3.29 222880.0 56400.0 4.2 5.2931 0.9927 3615255 CMLD4_000247 COC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M11 compound treatment 211320.0 45200.0 3.08 216040.0 49500.0 3.69 4.7885 0.996 3615256 CMLD4_000248 Cc1c2CCOc2nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M12 compound treatment 190200.0 24100.0 1.64 179800.0 13300.0 0.99 1.8631 0.9706 3615258 CMLD4_000249 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2cccc(Cl)c2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M13 compound treatment 229000.0 62900.0 4.29 223440.0 56900.0 4.24 6.0302 1.0 3615260 CMLD4_000250 CCc1c2COCc2nc3ccc(OC)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M14 compound treatment 187040.0 21000.0 1.43 182320.0 15800.0 1.18 1.8434 0.9954 1003776 CMLD4_000251 CCOC(=O)C1=C(C)NC(=O)NC1c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M15 compound treatment 180440.0 14400.0 0.98 183000.0 16500.0 1.23 1.561 0.9936 1037061 CMLD4_000252 OC1c2ccccc2-c3nc4ccccc4cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M16 compound treatment 176040.0 9960.0 0.68 178960.0 12500.0 0.93 1.1362 0.9882 3615263 CMLD4_000253 COC(=O)[C@@H]1C[C@]2(OC(=O)c3ccccc3)C=CC(=O)C[C@@H]2N1C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M17 compound treatment 175760.0 9680.0 0.66 180240.0 13700.0 1.02 1.1901 0.9774 3615267 CMLD4_000254 CSCC(=O)NS(=O)(=O)c1ccc(C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M18 compound treatment 181360.0 15300.0 1.04 181720.0 15200.0 1.13 1.538 0.9991 3615269 CMLD4_000255 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M19 compound treatment 218560.0 52500.0 3.58 220720.0 54200.0 4.04 5.3838 0.9982 3615271 CMLD4_000256 COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]2C[C@@H]2[C@H](NC(=O)OCc3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M20 compound treatment 176320.0 10200.0 0.7 179480.0 13000.0 0.97 1.1771 0.9872 3615274 CMLD4_000257 CC1=C(C(NC(=O)N1CCCC(=O)O)c2cccs2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M21 compound treatment 177440.0 11400.0 0.77 168840.0 2350.0 0.17 0.6711 0.8455 3615276 CMLD4_000258 CN(C)C(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M22 compound treatment 173440.0 7360.0 0.5 170760.0 4270.0 0.32 0.5793 0.9758 3615277 CMLD4_000259 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(Cl)cc2Cl)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M23 mock treatment 165400.0 -684.0 -0.05 169240.0 2750.0 0.2 0.1118 0.5324 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 M24 mock treatment 165080.0 -1000.0 -0.07 162600.0 -3890.0 -0.29 -0.2531 -0.8508 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N01 mock treatment 168080.0 2000.0 0.14 173200.0 6710.0 0.5 0.4494 0.8682 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N02 mock treatment 174400.0 8320.0 0.57 172640.0 6150.0 0.46 0.7246 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N03 compound treatment 174080.0 8000.0 0.55 176560.0 10100.0 0.75 0.9154 0.9878 3615279 CMLD4_000260 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(Cl)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N04 compound treatment 191560.0 25500.0 1.74 186960.0 20500.0 1.52 2.3054 0.9979 3615281 CMLD4_000261 O=C(NCC#CCOCc1ccccc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N05 compound treatment 183480.0 17400.0 1.19 178000.0 11500.0 0.86 1.4444 0.9872 3615282 CMLD4_000262 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(OC)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N06 compound treatment 185360.0 19300.0 1.31 181480.0 15000.0 1.12 1.7182 0.9967 1965352 CMLD4_000263 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N07 compound treatment 179920.0 13800.0 0.94 179680.0 13200.0 0.98 1.3612 0.9998 3615284 CMLD4_000264 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccccc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N08 compound treatment 182920.0 16800.0 1.15 181400.0 14900.0 1.11 1.5963 0.9999 3615287 CMLD4_000265 O=C(N[C@H]([C@@H]1C[C@H]1C(=O)NCc2ccccn2)c3ccccc3)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N09 compound treatment 179800.0 13700.0 0.94 181800.0 15300.0 1.14 1.467 0.9952 3615291 CMLD4_000266 CC1=C(C(NC(=O)N1CCCC(=O)O)c2ccc(cc2)[N+](=O)[O-])C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N10 compound treatment 183560.0 17500.0 1.19 181240.0 14700.0 1.1 1.6188 0.9992 3615293 CMLD4_000267 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N11 compound treatment 220280.0 54200.0 3.69 209040.0 42500.0 3.17 4.852 0.9971 3615296 CMLD4_000268 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc3ccccc3c2)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N12 compound treatment 181920.0 15800.0 1.08 175400.0 8910.0 0.66 1.2323 0.9726 3615298 CMLD4_000269 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCC4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N13 compound treatment 190640.0 24600.0 1.67 188400.0 21900.0 1.63 2.3369 0.9999 3615302 CMLD4_000270 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2cccc(c2)[N+](=O)[O-])C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N14 compound treatment 180640.0 14600.0 0.99 182880.0 16400.0 1.22 1.5643 0.9948 3615304 CMLD4_000271 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCCc4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N15 compound treatment 268760.0 103000.0 7.0 260480.0 94000.0 7.0 9.8963 1.0 3615305 CMLD4_000272 CCOC(=O)C1=C(C)N(CCCC(=O)N(Cc2ccc3OCOc3c2)C(C(=O)NC(C)(C)C)c4ccc5OCOc5c4)C(=O)NC1c6ccc(cc6)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N16 compound treatment 196040.0 30000.0 2.04 197920.0 31400.0 2.34 3.0982 0.9977 3615307 CMLD4_000273 Cc1ccc(CNC(=O)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N17 compound treatment 264960.0 98900.0 6.74 256000.0 89500.0 6.66 9.4774 1.0 3615310 CMLD4_000274 CCOC(=O)c1cn(Cc2ccccc2)c(C(=O)OC(C)(C)C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N18 compound treatment 203480.0 37400.0 2.55 195440.0 28900.0 2.15 3.3264 0.9965 3615311 CMLD4_000275 O=C(Nc1ccc2ccccc2c1)[C@@H]3C[C@H]3[C@@H](NP(=O)(c4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N19 compound treatment 184720.0 18600.0 1.27 174800.0 8310.0 0.62 1.3357 0.9453 3615313 CMLD4_000276 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OC(=O)c3ccc(I)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N20 compound treatment 174880.0 8800.0 0.6 180800.0 14300.0 1.07 1.1771 0.9631 3615315 CMLD4_000277 Cc1cc(CNC(=O)[C@@H]2C[C@H]2[C@@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)nn1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N21 compound treatment 183400.0 17300.0 1.18 187880.0 21400.0 1.59 1.9605 0.9892 3615317 CMLD4_000278 NCCn1c(cc(C(=O)O)c1c2ccccc2F)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N22 compound treatment 169680.0 3600.0 0.25 164360.0 -2130.0 -0.16 0.0613 0.2098 3615319 CMLD4_000279 COCCNC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N23 mock treatment 167440.0 1360.0 0.09 172880.0 6390.0 0.48 0.4017 0.8291 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 N24 mock treatment 159880.0 -6200.0 -0.42 163960.0 -2530.0 -0.19 -0.4322 -0.9336 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O01 mock treatment 171560.0 5480.0 0.37 173440.0 6950.0 0.52 0.6298 0.9872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O02 mock treatment 166080.0 -3.64 0.0 172040.0 5550.0 0.41 0.2919 0.7067 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O03 compound treatment 260600.0 94500.0 6.44 248040.0 81500.0 6.07 8.8483 0.9996 3615322 CMLD4_000280 CCc1cccc2nc-3c(Cn4c3cccc4=O)c(c12)[Si](CC)(CC)CC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O04 compound treatment 213560.0 47500.0 3.24 208360.0 41900.0 3.12 4.4923 0.9998 3615323 CMLD4_000281 CC(C)(C)[Si](OCC[C@@H]1C[C@@]1(C)[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4)(c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O05 compound treatment 235080.0 69000.0 4.7 239440.0 72900.0 5.43 7.1654 0.9974 3615327 CMLD4_000282 CC(C)(C)[Si](C)(C)c1c2Cn3c(cccc3=O)-c2nc4ccc(O)cc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O06 compound treatment 181040.0 15000.0 1.02 173920.0 7430.0 0.55 1.112 0.9587 3615329 CMLD4_000283 CC(C)NC(=O)[C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O07 compound treatment 180640.0 14600.0 0.99 177800.0 11300.0 0.84 1.2969 0.9966 3615332 CMLD4_000284 CCc1c2CC(C)Oc2nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O08 compound treatment 177600.0 11500.0 0.79 177640.0 11100.0 0.83 1.142 0.9996 3615334 CMLD4_000285 CNC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)CNC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O09 compound treatment 217880.0 51800.0 3.53 213240.0 46700.0 3.48 4.9573 1.0 3615338 CMLD4_000286 c1ccc(cc1)c2c3c4ccccc4[nH]c3nc5ccccc25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O10 compound treatment 238520.0 72400.0 4.94 229000.0 62500.0 4.65 6.7818 0.9996 3615340 CMLD4_000287 COC(=O)C1=C(COc2ccccc2)NC(=O)NC1c3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O11 compound treatment 225560.0 59500.0 4.05 229560.0 63100.0 4.69 6.1865 0.9973 3615342 CMLD4_000288 C[Si](C)(C)C#Cc1ccccc1NC(=S)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O12 compound treatment 197880.0 31800.0 2.17 199280.0 32800.0 2.44 3.2585 0.9983 3615344 CMLD4_000289 CCOC(=O)C1=C(C)N(CCCCCC(=O)O)C(=O)NC1c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O13 compound treatment 174680.0 8600.0 0.59 180040.0 13500.0 1.01 1.1275 0.9667 3615346 CMLD4_000290 CCc1c2COCc2nc3cccc(SC)c13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O14 compound treatment 194480.0 28400.0 1.94 198120.0 31600.0 2.35 3.0335 0.9953 3615347 CMLD4_000291 CCOC(=O)C1=C(CCc2ccccc2)NC(=O)NC1c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O15 compound treatment 173720.0 7640.0 0.52 178720.0 12200.0 0.91 1.0118 0.9649 1067287 CMLD4_000292 C1c2ccccc2-c3nc4ccccc4cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O16 compound treatment 197480.0 31400.0 2.14 205320.0 38800.0 2.89 3.5571 0.9891 3615350 CMLD4_000293 COC(=O)[C@@H]1C=C2CCC(=O)C[C@H]2N1C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O17 compound treatment 216640.0 50600.0 3.45 218840.0 52300.0 3.9 5.1923 0.9981 3615354 CMLD4_000294 CCCC/C=C/[C@@H](NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O18 compound treatment 170200.0 4120.0 0.28 173120.0 6630.0 0.49 0.5473 0.9642 3615358 CMLD4_000295 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2cccc(OC)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O19 compound treatment 177080.0 11000.0 0.75 177320.0 10800.0 0.81 1.1001 0.9993 3615361 CMLD4_000296 CN(C)C(=O)[C@]1(C)C[C@H]1[C@H](NC(=O)CNC(=O)[C@@H]2CCCN2C(=O)[C@]3(C)C[C@H]3[C@H](NC(=O)OCc4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O20 compound treatment 172920.0 6840.0 0.47 174840.0 8350.0 0.62 0.769 0.9899 3615364 CMLD4_000297 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2OS(=O)(=O)c3ccc(C)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O21 compound treatment 212280.0 46200.0 3.15 226240.0 59700.0 4.45 5.3715 0.9857 3615366 CMLD4_000298 CC/C(=C\C1CCCCC1)/C(NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O22 compound treatment 175080.0 9000.0 0.61 175160.0 8670.0 0.65 0.89 0.9997 3615369 CMLD4_000299 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(Cl)cc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O23 mock treatment 159040.0 -7040.0 -0.48 163720.0 -2770.0 -0.21 -0.4854 -0.9287 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 O24 mock treatment 159320.0 -6760.0 -0.46 163760.0 -2730.0 -0.2 -0.4698 -0.9322 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P01 mock treatment 170760.0 4680.0 0.32 164720.0 -1770.0 -0.13 0.1323 0.3834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P02 mock treatment 169840.0 3760.0 0.26 176000.0 9510.0 0.71 0.6816 0.9055 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P03 compound treatment 175920.0 9840.0 0.67 170280.0 3790.0 0.28 0.6736 0.9259 3615371 CMLD4_000300 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P04 compound treatment 170480.0 4400.0 0.3 171160.0 4670.0 0.35 0.4577 0.9973 3615373 CMLD4_000301 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P05 compound treatment 195560.0 29500.0 2.01 187160.0 20700.0 1.54 2.5088 0.9913 3615374 CMLD4_000302 COC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P06 compound treatment 174600.0 8520.0 0.58 171640.0 5150.0 0.38 0.6816 0.9797 3615376 CMLD4_000303 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCn7cc(nc7C)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P07 compound treatment 171640.0 5560.0 0.38 172880.0 6390.0 0.48 0.6041 0.9936 3615379 CMLD4_000304 CC1=C(C(NC(=O)N1CCCC(=O)O)c2cccc3ccccc23)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P08 compound treatment 171960.0 5880.0 0.4 174640.0 8150.0 0.61 0.7122 0.9797 3615381 CMLD4_000305 OC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P09 compound treatment 172040.0 5960.0 0.41 173680.0 7190.0 0.54 0.6655 0.9907 3615385 CMLD4_000306 COc1ccc(cc1)C2NC(=O)N(CCCC(=O)O)C(=C2C(=O)OCc3ccccc3)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P10 compound treatment 175040.0 8960.0 0.61 175440.0 8950.0 0.67 0.9028 0.9991 3615387 CMLD4_000307 CNC(=O)[C@H](C)[C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P11 compound treatment 182680.0 16600.0 1.13 179880.0 13400.0 1.0 1.5048 0.998 3615389 CMLD4_000308 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(Br)cc2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P12 compound treatment 182000.0 15900.0 1.09 178080.0 11600.0 0.86 1.3772 0.9935 3615392 CMLD4_000309 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCc4cc(C)n(C)n4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P13 compound treatment 193240.0 27200.0 1.85 187640.0 21100.0 1.57 2.4222 0.9967 3615395 CMLD4_000310 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(cc2)C(F)(F)F)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P14 compound treatment 178960.0 12900.0 0.88 180240.0 13700.0 1.02 1.3444 0.9971 3615397 CMLD4_000311 C[C@H](CO)NC(=O)[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P15 compound treatment 185400.0 19300.0 1.32 184520.0 18000.0 1.34 1.8801 1.0 3615399 CMLD4_000312 COC(=O)c1cc(c2ccccc2)n(CCN)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P16 mock treatment 166400.0 316.0 0.02 171280.0 4790.0 0.36 0.2673 0.7485 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P17 compound treatment 168640.0 2560.0 0.17 175000.0 8510.0 0.63 0.5711 0.8694 3615400 CMLD4_000313 CC1=C(C(NC(=O)N1CCCC(=O)O)c2cccc(c2)[N+](=O)[O-])C(=O)OCC(Br)(Br)Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P18 compound treatment 177400.0 11300.0 0.77 175440.0 8950.0 0.67 1.0165 0.9973 3615403 CMLD4_000314 CS(=O)(=O)c1ccc(CNC(=O)[C@@H]2C[C@H]2[C@@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P19 compound treatment 170160.0 4080.0 0.28 166320.0 -170.0 -0.01 0.1876 0.6742 3615404 CMLD4_000315 CCOC(=O)C1=C(C)N(CCCC(=O)O)C(=O)NC1c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P20 compound treatment 172360.0 6280.0 0.43 171800.0 5310.0 0.4 0.582 0.9992 3615405 CMLD4_000316 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)OCc2ccccc2)c3ccccc3)C(=O)NCCF 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P21 compound treatment 164360.0 -1720.0 -0.12 160840.0 -5650.0 -0.42 -0.3805 -0.8713 3615409 CMLD4_000317 CC(C)(C)NC(=O)C(N(CCN1CCOCC1)C(=O)CCCNC(=O)c2ccccc2)c3ccc(I)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P22 compound treatment 194440.0 28400.0 1.93 190640.0 24100.0 1.8 2.638 0.9993 3615411 CMLD4_000318 Cc1ccc(CNC(=O)[C@H]2C[C@@H]2[C@H](NP(=O)(c3ccccc3)c4ccccc4)c5ccccc5)c(F)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P23 mock treatment 160960.0 -5120.0 -0.35 160880.0 -5610.0 -0.42 -0.5423 -0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2288 P24 mock treatment 161320.0 -4760.0 -0.32 163760.0 -2730.0 -0.2 -0.3733 -0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A01 mock treatment 165880.0 -757.0 -0.05 160920.0 -2760.0 -0.21 -0.1816 -0.8582 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A02 mock treatment 165120.0 -1520.0 -0.1 160440.0 -3240.0 -0.24 -0.2435 -0.9287 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A03 compound treatment 166080.0 -557.0 -0.04 163160.0 -517.0 -0.04 -0.054 -1.0 3615415 CMLD4_000319 O=C(NCc1nc2ccccc2[nH]1)[C@H]3C[C@@H]3[C@H](NP(=O)(c4ccccc4)c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A04 compound treatment 165920.0 -717.0 -0.05 160240.0 -3440.0 -0.26 -0.2154 -0.8272 3615419 CMLD4_000320 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCN3CCOCC3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A05 compound treatment 164400.0 -2240.0 -0.15 164080.0 403.0 0.03 -0.0866 -0.5573 3615423 CMLD4_000321 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A06 compound treatment 187720.0 21100.0 1.44 174920.0 11200.0 0.84 1.6081 0.9669 3615427 CMLD4_000322 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)Nc3ccccc3)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A07 compound treatment 186480.0 19800.0 1.35 180720.0 17000.0 1.27 1.8535 0.9995 3615430 CMLD4_000323 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)c2cc(C)on2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A08 compound treatment 191720.0 25100.0 1.71 182560.0 18900.0 1.41 2.203 0.9953 3615433 CMLD4_000324 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCc3c[nH]c4ccc(OC)cc34)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A09 compound treatment 177240.0 10600.0 0.72 172720.0 9040.0 0.67 0.9871 0.9994 3615437 CMLD4_000325 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)c2cc(C)on2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A10 compound treatment 228400.0 61800.0 4.21 212680.0 49000.0 3.65 5.5564 0.9974 3615439 CMLD4_000326 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(F)cc(F)c3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A11 compound treatment 189320.0 22700.0 1.55 183000.0 19300.0 1.44 2.1104 0.9993 3615442 CMLD4_000327 COC(=O)[C@H]1C[C@@H]1[C@H](NS(=O)(=O)c2ccc(cc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A12 compound treatment 184280.0 17600.0 1.2 174840.0 11200.0 0.83 1.438 0.9837 3615445 CMLD4_000328 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(OC)c(O)c3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A13 compound treatment 172760.0 6120.0 0.42 169760.0 6080.0 0.45 0.6153 0.9992 3615448 CMLD4_000329 COC(=O)[C@H]1C[C@@H]1[C@H](NS(=O)(=O)c2ccc3ccccc3c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A14 compound treatment 161840.0 -4800.0 -0.33 161960.0 -1720.0 -0.13 -0.3216 -0.916 3615452 CMLD4_000330 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccncc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A15 compound treatment 160440.0 -6200.0 -0.42 162280.0 -1400.0 -0.1 -0.3723 -0.8556 3615456 CMLD4_000331 CC(Cc1ccccc1)C(=O)N2CCN(C)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A16 compound treatment 166560.0 -76.9 -0.01 163040.0 -637.0 -0.05 -0.0372 -0.7805 3615458 CMLD4_000332 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCF)/c3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A17 compound treatment 161280.0 -5360.0 -0.37 158560.0 -5120.0 -0.38 -0.5275 -0.9998 3615462 CMLD4_000333 CC(Cc1ccccc1)C(=O)NCc2cc(C)n(C)n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A18 compound treatment 180000.0 13400.0 0.91 178080.0 14400.0 1.07 1.4022 0.9967 3615463 CMLD4_000334 CCCCCCN(C(C(=O)NCCCC)c1cccc(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A19 compound treatment 158640.0 -8000.0 -0.55 161080.0 -2600.0 -0.19 -0.5222 -0.9027 3615465 CMLD4_000335 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCc3ccc(cc3)S(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A20 compound treatment 163080.0 -3560.0 -0.24 160160.0 -3520.0 -0.26 -0.3566 -0.9993 3615469 CMLD4_000336 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(cc2)C(C)(C)C)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A21 compound treatment 183320.0 16700.0 1.14 167520.0 3840.0 0.29 1.0065 0.8582 3615472 CMLD4_000337 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3nn(nc3C)c4ccccc4)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A22 compound treatment 161960.0 -4680.0 -0.32 159440.0 -4240.0 -0.32 -0.4484 -1.0 3615476 CMLD4_000338 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)C(C)(C)C)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A23 mock treatment 160600.0 -6040.0 -0.41 158160.0 -5520.0 -0.41 -0.5814 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 A24 mock treatment 157200.0 -9440.0 -0.64 152760.0 -10900.0 -0.81 -1.0295 -0.9933 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B01 mock treatment 155400.0 -11200.0 -0.77 154200.0 -9480.0 -0.71 -1.0405 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B02 mock treatment 159240.0 -7400.0 -0.5 156800.0 -6880.0 -0.51 -0.7185 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B03 compound treatment 180760.0 14100.0 0.96 177920.0 14200.0 1.06 1.4304 0.9988 3615478 CMLD4_000339 CCCCNC(=O)C(N(Cc1ccccc1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C)c6ccc(OCC(=O)OC)c(c6)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B04 compound treatment 167360.0 723.0 0.05 162440.0 -1240.0 -0.09 -0.0302 -0.2895 3615481 CMLD4_000340 COC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B05 compound treatment 178960.0 12300.0 0.84 174840.0 11200.0 0.83 1.1816 1.0 3615485 CMLD4_000341 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)C4CCCCC4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B06 compound treatment 163320.0 -3320.0 -0.23 154440.0 -9240.0 -0.69 -0.646 -0.8926 3615486 CMLD4_000342 CC1(C=CC2(CCCCC2)N1C(=O)c3ccccc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B07 compound treatment 161000.0 -5640.0 -0.38 162440.0 -1240.0 -0.09 -0.3368 -0.8524 3615488 CMLD4_000343 CC(C)CC1(C=CCN1C(=O)C)C(=O)NCC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B08 compound treatment 166480.0 -157.0 -0.01 165160.0 1480.0 0.11 0.0705 0.6356 3615489 CMLD4_000344 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)c3ccccc3)C(=O)NCC4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B09 compound treatment 182320.0 15700.0 1.07 178440.0 14800.0 1.1 1.533 0.9999 3615493 CMLD4_000345 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCc3cc(F)cc(c3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B10 compound treatment 180480.0 13800.0 0.94 169520.0 5840.0 0.43 0.9749 0.9381 3615495 CMLD4_000346 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)C)C(=O)NCCc3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B11 compound treatment 166280.0 -357.0 -0.02 163320.0 -357.0 -0.03 -0.036 -0.999 3615498 CMLD4_000347 CC(=O)N1CC=CC1(C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B12 compound treatment 168920.0 2280.0 0.16 164760.0 1080.0 0.08 0.1671 0.9531 3615500 CMLD4_000348 COCCNC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B13 compound treatment 185960.0 19300.0 1.32 181240.0 17600.0 1.31 1.8558 1.0 3615504 CMLD4_000349 CC(=O)N1C(C)(C=CC21CCCCC2)C(=O)NCc3cc(F)cc(c3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B14 compound treatment 159200.0 -7440.0 -0.51 155920.0 -7760.0 -0.58 -0.7667 -0.9979 3615505 CMLD4_000350 COC(=O)CNC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B15 compound treatment 174400.0 7760.0 0.53 159440.0 -4240.0 -0.32 0.1513 0.2455 3615507 CMLD4_000351 COC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B16 compound treatment 167280.0 643.0 0.04 162680.0 -997.0 -0.07 -0.0215 -0.249 3615512 CMLD4_000352 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(cc3)S(=O)(=O)C)/C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B17 compound treatment 165680.0 -957.0 -0.07 161160.0 -2520.0 -0.19 -0.1786 -0.9003 3615515 CMLD4_000353 COC(=O)CNC(=O)C1(C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B18 mock treatment 158280.0 -8360.0 -0.57 157880.0 -5800.0 -0.43 -0.7079 -0.9906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B19 compound treatment 188600.0 22000.0 1.5 185840.0 22200.0 1.65 2.2252 0.9988 3615517 CMLD4_000354 C[C@@]1(C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3)C(=O)NCc4cc(F)cc(c4)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B20 mock treatment 162840.0 -3800.0 -0.26 157400.0 -6280.0 -0.47 -0.5134 -0.9612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B21 compound treatment 180280.0 13600.0 0.93 183400.0 19700.0 1.47 1.6957 0.9758 3615521 CMLD4_000355 CC(=O)N1C(C)(C=CC21CCCCC2)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B22 mock treatment 155880.0 -10800.0 -0.73 157680.0 -6000.0 -0.45 -0.8342 -0.9717 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B23 mock treatment 156880.0 -9760.0 -0.67 153600.0 -10100.0 -0.75 -1.0007 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 B24 mock treatment 158960.0 -7680.0 -0.52 152680.0 -11000.0 -0.82 -0.9488 -0.9767 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C01 mock treatment 159560.0 -7080.0 -0.48 165880.0 2200.0 0.16 -0.2252 -0.442 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C02 mock treatment 159040.0 -7600.0 -0.52 159360.0 -4320.0 -0.32 -0.5934 -0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C03 compound treatment 165520.0 -1120.0 -0.08 162720.0 -957.0 -0.07 -0.1042 -0.9994 3615523 CMLD4_000356 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](N)c2ccccc2)C(=O)Nc3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C04 compound treatment 164960.0 -1680.0 -0.11 163800.0 123.0 0.01 -0.0744 -0.6484 3615526 CMLD4_000357 CNC(=O)[C@H](C)/C=C/C(NC(=O)OCc1ccccc1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C05 compound treatment 184120.0 17500.0 1.19 172680.0 9000.0 0.67 1.3166 0.9629 3615529 CMLD4_000358 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)c2cc(C)on2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C06 compound treatment 176560.0 9920.0 0.68 177280.0 13600.0 1.01 1.1943 0.9808 3615533 CMLD4_000359 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCC3CC3)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C07 compound treatment 185400.0 18800.0 1.28 179600.0 15900.0 1.19 1.7425 0.9993 3615535 CMLD4_000360 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)c2cnccn2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C08 compound treatment 165680.0 -957.0 -0.07 164480.0 803.0 0.06 -0.0039 -0.0437 3615539 CMLD4_000361 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCO)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C09 compound treatment 191760.0 25100.0 1.71 179960.0 16300.0 1.21 2.0681 0.9856 3615542 CMLD4_000362 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)c2cnccn2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C10 compound treatment 203160.0 36500.0 2.49 191600.0 27900.0 2.08 3.2302 0.996 3615543 CMLD4_000363 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(C)on3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C11 compound treatment 190240.0 23600.0 1.61 190360.0 26700.0 1.99 2.5421 0.9946 3615547 CMLD4_000364 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NS(=O)(=O)c2ccc(cc2)c3ccccc3)c4ccccc4)C(=O)Nc5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C12 compound treatment 188080.0 21400.0 1.46 180800.0 17100.0 1.27 1.9349 0.9977 3615552 CMLD4_000365 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCc3c[nH]c4ccccc34)/c5cccnc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C13 compound treatment 181960.0 15300.0 1.04 179000.0 15300.0 1.14 1.5451 0.999 3615555 CMLD4_000366 C[C@H]([C@H]1C[C@]1(C)[C@H](NS(=O)(=O)c2ccc3ccccc3c2)c4ccccc4)C(=O)Nc5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C14 compound treatment 195680.0 29000.0 1.98 192360.0 28700.0 2.13 2.9096 0.9993 3615559 CMLD4_000367 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccccc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C15 compound treatment 165720.0 -917.0 -0.06 157240.0 -6440.0 -0.48 -0.383 -0.7927 3615563 CMLD4_000368 CC(Cc1ccccc1)C(=O)N(C)Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C16 compound treatment 158240.0 -8400.0 -0.57 165840.0 2160.0 0.16 -0.291 -0.4893 3615565 CMLD4_000369 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N(C)Cc3cccnc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C17 compound treatment 172280.0 5640.0 0.38 168840.0 5160.0 0.38 0.5438 1.0 3615568 CMLD4_000370 CC(Cc1ccccc1)C(=O)NCc2nn(nc2C)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C18 compound treatment 185840.0 19200.0 1.31 180680.0 17000.0 1.27 1.8206 0.9999 3615570 CMLD4_000371 CCCCCCN(C(C)C(=O)NCCCC)C(=O)CCCCCN1C(=C(C(NC1=O)c2ccc(cc2)c3ccccc3)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C19 compound treatment 179080.0 12400.0 0.85 175160.0 11500.0 0.85 1.2042 1.0 3615571 CMLD4_000372 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C20 compound treatment 200960.0 34300.0 2.34 190120.0 26400.0 1.97 3.0463 0.9963 3615573 CMLD4_000373 CC1=C(C(NC(=O)N1CCCCCC(=O)O)C2CC2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C21 compound treatment 189760.0 23100.0 1.58 180960.0 17300.0 1.29 2.0243 0.9949 3615575 CMLD4_000374 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3nc4ccccc4s3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C22 compound treatment 180400.0 13800.0 0.94 180520.0 16800.0 1.25 1.5499 0.9898 3615579 CMLD4_000375 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3cccc(c3)[N+](=O)[O-])C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C23 mock treatment 157120.0 -9520.0 -0.65 155520.0 -8160.0 -0.61 -0.8881 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 C24 mock treatment 161040.0 -5600.0 -0.38 154760.0 -8920.0 -0.66 -0.7391 -0.9655 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D01 mock treatment 162160.0 -4480.0 -0.31 154120.0 -9560.0 -0.71 -0.7188 -0.9286 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D02 mock treatment 155800.0 -10800.0 -0.74 156880.0 -6800.0 -0.51 -0.8801 -0.9829 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D03 compound treatment 180120.0 13500.0 0.92 177360.0 13700.0 1.02 1.3701 0.9987 3615581 CMLD4_000376 CCCCNC(=O)C(N(CCc1ccccc1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C)c6ccc(OCC(=O)OC)c(c6)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D04 compound treatment 170880.0 4240.0 0.29 168240.0 4560.0 0.34 0.4447 0.9968 3615583 CMLD4_000377 COC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D05 compound treatment 167640.0 1000.0 0.07 160120.0 -3560.0 -0.26 -0.1388 -0.5078 3615587 CMLD4_000378 CC(C)CC1(C=CCN1C(=O)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D06 compound treatment 169040.0 2400.0 0.16 161840.0 -1840.0 -0.14 0.0192 0.0899 3615590 CMLD4_000379 CC1(C=CC2(CCCCC2)N1C(=O)c3ccccc3)C(=O)NCC4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D07 compound treatment 165520.0 -1120.0 -0.08 163200.0 -477.0 -0.04 -0.0789 -0.9396 3615591 CMLD4_000380 CNC(=O)C1(CC(C)C)C=CCN1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D08 compound treatment 196320.0 29700.0 2.02 188280.0 24600.0 1.83 2.7258 0.9988 3615593 CMLD4_000381 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)c3ccccc3)C(=O)NCCc4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D09 compound treatment 169800.0 3160.0 0.22 155800.0 -7880.0 -0.59 -0.2621 -0.4195 3615596 CMLD4_000382 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D10 compound treatment 182520.0 15900.0 1.08 176960.0 13300.0 0.99 1.4648 0.999 3615598 CMLD4_000383 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)C)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D11 compound treatment 167120.0 483.0 0.03 169160.0 5480.0 0.41 0.3119 0.7617 3615601 CMLD4_000384 COCCNC(=O)C1(C)C=CCN1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D12 compound treatment 201280.0 34600.0 2.36 188040.0 24400.0 1.81 2.9523 0.9915 3615603 CMLD4_000385 COC(=O)N1[C@H](C)C=C[C@]1(Cc2ccccc2)C(=O)NCc3ccc(cc3)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D13 compound treatment 170160.0 3520.0 0.24 167000.0 3320.0 0.25 0.3447 0.9999 3615607 CMLD4_000386 COC(=O)N1CC=CC1(C)C(=O)NCc2cc(F)cc(c2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D14 compound treatment 194960.0 28300.0 1.93 186520.0 22800.0 1.7 2.5676 0.998 3615609 CMLD4_000387 COC(=O)N1C(C)(C=CC21CCCCC2)C(=O)NCc3ccc(cc3)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D15 compound treatment 172760.0 6120.0 0.42 164400.0 723.0 0.05 0.3332 0.7917 3615611 CMLD4_000388 COC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D16 compound treatment 178240.0 11600.0 0.79 163680.0 3.11 0.0 0.5595 0.7073 3615615 CMLD4_000389 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)Nc3ccccc3)/C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D17 compound treatment 193360.0 26700.0 1.82 184640.0 21000.0 1.56 2.3915 0.997 3615617 CMLD4_000390 CN(C)c1ccc(CNC(=O)C2(C)C=CCN2C(=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D18 mock treatment 164080.0 -2560.0 -0.17 163600.0 -76.9 -0.01 -0.1273 -0.7299 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D19 compound treatment 166000.0 -637.0 -0.04 160480.0 -3200.0 -0.24 -0.1989 -0.8226 3615619 CMLD4_000391 C[C@@]1(C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D20 mock treatment 161960.0 -4680.0 -0.32 156960.0 -6720.0 -0.5 -0.579 -0.9764 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D21 compound treatment 171200.0 4560.0 0.31 166400.0 2720.0 0.2 0.3633 0.9784 3615623 CMLD4_000392 COC(=O)CNC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D22 mock treatment 166440.0 -197.0 -0.01 159960.0 -3720.0 -0.28 -0.2051 -0.7405 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D23 mock treatment 163360.0 -3280.0 -0.22 155960.0 -7720.0 -0.57 -0.5641 -0.9153 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 D24 mock treatment 157200.0 -9440.0 -0.64 155480.0 -8200.0 -0.61 -0.8863 -0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E01 mock treatment 166760.0 123.0 0.01 168080.0 4400.0 0.33 0.2377 0.725 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E02 mock treatment 165920.0 -717.0 -0.05 167840.0 4160.0 0.31 0.1845 0.5883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E03 compound treatment 176640.0 10000.0 0.68 177560.0 13900.0 1.03 1.2129 0.9797 3615628 CMLD4_000393 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E04 compound treatment 175280.0 8640.0 0.59 172200.0 8520.0 0.63 0.8652 0.9993 3615630 CMLD4_000394 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCCN3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E05 compound treatment 185800.0 19200.0 1.31 171680.0 8000.0 0.6 1.345 0.9367 3615633 CMLD4_000395 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)c2cnccn2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E06 compound treatment 214000.0 47400.0 3.23 211120.0 47400.0 3.53 4.7801 0.999 3615635 CMLD4_000396 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(OC)c(O)c3)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E07 compound treatment 182120.0 15500.0 1.06 177840.0 14200.0 1.05 1.4918 1.0 3615638 CMLD4_000397 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)c2cc(C)nn2C)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E08 compound treatment 213560.0 46900.0 3.2 199720.0 36000.0 2.68 4.159 0.9962 3615641 CMLD4_000398 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)Nc3ccc(OC)cc3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E09 compound treatment 193480.0 26800.0 1.83 182080.0 18400.0 1.37 2.2626 0.9898 3615645 CMLD4_000399 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)c2cc(C)nn2C)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E10 compound treatment 225240.0 58600.0 4.0 217960.0 54300.0 4.04 5.682 1.0 3615647 CMLD4_000400 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3nn(nc3C)c4ccccc4)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E11 compound treatment 173240.0 6600.0 0.45 175040.0 11400.0 0.85 0.9163 0.9564 3615651 CMLD4_000401 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E12 compound treatment 177040.0 10400.0 0.71 176560.0 12900.0 0.96 1.1795 0.989 3615655 CMLD4_000402 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(C)n(C)n3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E13 compound treatment 192640.0 26000.0 1.77 191400.0 27700.0 2.06 2.7126 0.9971 3615658 CMLD4_000403 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NS(=O)(=O)c2ccc3ccccc3c2)c4ccccc4)C(=O)Nc5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E14 compound treatment 216600.0 50000.0 3.41 208080.0 44400.0 3.3 4.7455 0.9999 3615660 CMLD4_000404 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(OC)c(OC)c3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E15 compound treatment 175360.0 8720.0 0.59 173840.0 10200.0 0.76 0.9554 0.9929 3615663 CMLD4_000405 CC(Cc1ccccc1)C(=O)NCCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E16 compound treatment 219520.0 52900.0 3.61 201800.0 38100.0 2.84 4.5557 0.993 3615666 CMLD4_000406 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3nc4ccccc4s3)/c5cccnc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E17 compound treatment 178280.0 11600.0 0.79 170480.0 6800.0 0.51 0.9193 0.9764 3615670 CMLD4_000407 CC(Cc1ccccc1)C(=O)NCc2nc3ccccc3s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E18 compound treatment 187240.0 20600.0 1.4 187160.0 23500.0 1.75 2.2291 0.9941 3615672 CMLD4_000408 CCCCCCN(C(C1CCCCC1)C(=O)NCCCC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E19 compound treatment 186960.0 20300.0 1.39 187360.0 23700.0 1.76 2.2261 0.9929 3615674 CMLD4_000409 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCc3cc(C)n(C)n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E20 compound treatment 173440.0 6800.0 0.46 174720.0 11000.0 0.82 0.9091 0.9633 3615678 CMLD4_000410 COC(=O)CCCCCN1C(=C(C(NC1=O)c2ccc(cc2)c3ccccc3)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E21 compound treatment 184400.0 17800.0 1.21 181320.0 17600.0 1.31 1.7848 0.9992 3615679 CMLD4_000411 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cccnc3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E22 compound treatment 194600.0 28000.0 1.91 189720.0 26000.0 1.94 2.7186 1.0 3615683 CMLD4_000412 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccccc3)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E23 mock treatment 165520.0 -1120.0 -0.08 161280.0 -2400.0 -0.18 -0.18 -0.9279 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 E24 mock treatment 165720.0 -917.0 -0.06 160720.0 -2960.0 -0.22 -0.1998 -0.8734 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F01 mock treatment 167600.0 963.0 0.07 166760.0 3080.0 0.23 0.2087 0.8744 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F02 mock treatment 167200.0 563.0 0.04 169560.0 5880.0 0.44 0.3368 0.7662 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F03 compound treatment 192800.0 26200.0 1.78 187920.0 24200.0 1.8 2.5371 1.0 3615684 CMLD4_000413 CCCCNC(=O)C(N(CCc1ccccn1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C)c6ccc(OCC(=O)OC)c(c6)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F04 compound treatment 185320.0 18700.0 1.27 180720.0 17000.0 1.27 1.7976 1.0 3615687 CMLD4_000414 COC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F05 compound treatment 171840.0 5200.0 0.35 170840.0 7160.0 0.53 0.6278 0.9804 3615690 CMLD4_000415 COCCNC(=O)C1(CC(C)C)C=CCN1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F06 compound treatment 192440.0 25800.0 1.76 181960.0 18300.0 1.36 2.2061 0.9919 3615692 CMLD4_000416 CC1(C=CC2(CCCCC2)N1C(=O)c3ccccc3)C(=O)NCCc4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F07 compound treatment 177120.0 10500.0 0.71 170000.0 6320.0 0.47 0.8381 0.9794 3615694 CMLD4_000417 CC(C)CC1(C=CCN1C(=O)C)C(=O)NCCc2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F08 compound treatment 199520.0 32900.0 2.24 190760.0 27100.0 2.02 3.0106 0.9986 3615696 CMLD4_000418 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)c3ccccc3)C(=O)NCCCNc4ncc(cc4Cl)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F09 compound treatment 172960.0 6320.0 0.43 173040.0 9360.0 0.7 0.7976 0.9733 3615700 CMLD4_000419 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F10 compound treatment 178800.0 12200.0 0.83 174120.0 10400.0 0.78 1.136 0.9995 3615701 CMLD4_000420 COC(=O)N1[C@H](C)C=C[C@]1(Cc2ccccc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F11 compound treatment 184480.0 17800.0 1.22 183840.0 20200.0 1.5 1.9213 0.9946 3615704 CMLD4_000421 CC(=O)N1CC=CC1(C)C(=O)NCc2cc(F)cc(c2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F12 compound treatment 173920.0 7280.0 0.5 173480.0 9800.0 0.73 0.867 0.9824 3615706 CMLD4_000422 COC(=O)N1[C@H](C)C=C[C@]1(Cc2ccccc2)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F13 compound treatment 177160.0 10500.0 0.72 171160.0 7480.0 0.56 0.9011 0.9922 3615709 CMLD4_000423 COC(=O)N1CC=CC1(C)C(=O)NCCN2CCOCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F14 compound treatment 170800.0 4160.0 0.28 172480.0 8800.0 0.66 0.664 0.9299 3615712 CMLD4_000424 COC(=O)N1C(C)(C=CC21CCCCC2)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F15 compound treatment 175600.0 8960.0 0.61 170520.0 6840.0 0.51 0.7922 0.9959 3615713 CMLD4_000425 COC(=O)[C@]1(Cc2ccccc2)N[C@H](C)C=C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F16 compound treatment 178440.0 11800.0 0.8 176400.0 12700.0 0.95 1.2386 0.9967 3615717 CMLD4_000426 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)O)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F17 compound treatment 175760.0 9120.0 0.62 175680.0 12000.0 0.89 1.0715 0.9843 3615721 CMLD4_000427 CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F18 mock treatment 166360.0 -277.0 -0.02 170960.0 7280.0 0.54 0.3699 0.6821 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F19 compound treatment 170880.0 4240.0 0.29 170200.0 6520.0 0.49 0.5479 0.9694 3615723 CMLD4_000428 C[C@@]1(C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3)C(=O)NCC4CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F20 mock treatment 173080.0 6440.0 0.44 170920.0 7240.0 0.54 0.6918 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F21 compound treatment 168400.0 1760.0 0.12 162600.0 -1080.0 -0.08 0.0283 0.196 3615726 CMLD4_000429 CC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCc3cc(F)cc(c3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F22 mock treatment 168080.0 1440.0 0.1 158440.0 -5240.0 -0.39 -0.206 -0.5125 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F23 mock treatment 168960.0 2320.0 0.16 162600.0 -1080.0 -0.08 0.0553 0.3116 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 F24 mock treatment 166000.0 -637.0 -0.04 159880.0 -3800.0 -0.28 -0.2305 -0.8063 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G01 mock treatment 171120.0 4480.0 0.31 169120.0 5440.0 0.41 0.5026 0.9903 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G02 mock treatment 175440.0 8800.0 0.6 174680.0 11000.0 0.82 1.0035 0.9883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G03 compound treatment 194520.0 27900.0 1.9 192680.0 29000.0 2.16 2.8706 0.998 3615730 CMLD4_000430 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)c2cc(C)on2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G04 compound treatment 222640.0 56000.0 3.82 215080.0 51400.0 3.83 5.405 1.0 3615732 CMLD4_000431 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCO)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G05 compound treatment 175400.0 8760.0 0.6 174720.0 11000.0 0.82 1.0036 0.9877 3615736 CMLD4_000432 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)c2cc(C)nn2C)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G06 compound treatment 188280.0 21600.0 1.48 182080.0 18400.0 1.37 2.0119 0.9993 3615739 CMLD4_000433 CNC(=O)[C@H](C)/C=C(\I)/C(NC(=O)OCc1ccccc1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G07 compound treatment 195040.0 28400.0 1.94 192720.0 29000.0 2.16 2.8977 0.9985 3615744 CMLD4_000434 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)c2cccnc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G08 compound treatment 230440.0 63800.0 4.35 225240.0 61600.0 4.58 6.3158 0.9997 3615747 CMLD4_000435 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N[C@@H](CO)Cc3ccccc3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G09 compound treatment 208520.0 41900.0 2.86 196280.0 32600.0 2.43 3.7349 0.9967 3615751 CMLD4_000436 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)c2cccnc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G10 compound treatment 195400.0 28800.0 1.96 186080.0 22400.0 1.67 2.5656 0.9967 3615753 CMLD4_000437 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cccnc3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G11 compound treatment 195120.0 28500.0 1.94 184800.0 21100.0 1.57 2.4848 0.9945 3615756 CMLD4_000438 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)C)c2ccccc2)C(=O)Nc3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G12 compound treatment 185320.0 18700.0 1.27 182400.0 18700.0 1.39 1.886 0.999 3615759 CMLD4_000439 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCC3CC3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G13 compound treatment 183120.0 16500.0 1.12 181280.0 17600.0 1.31 1.721 0.9971 3615762 CMLD4_000440 COC(=O)C1CC1C(NC(=O)[C@@H]2CCCN2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G14 compound treatment 192880.0 26200.0 1.79 188600.0 24900.0 1.85 2.5768 0.9998 3615765 CMLD4_000441 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(F)cc(F)c3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G15 compound treatment 190600.0 24000.0 1.63 183920.0 20200.0 1.51 2.2206 0.9992 3615769 CMLD4_000442 CC(Cc1ccccc1)C(=O)NCCc2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G16 compound treatment 186920.0 20300.0 1.38 177760.0 14100.0 1.05 1.719 0.9907 3615771 CMLD4_000443 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cccnc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G17 compound treatment 175600.0 8960.0 0.61 176920.0 13200.0 0.99 1.1291 0.9736 3615775 CMLD4_000444 CC(Cc1ccccc1)C(=O)N(C)Cc2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G18 compound treatment 220320.0 53700.0 3.66 206200.0 42500.0 3.16 4.8259 0.9974 3615777 CMLD4_000445 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccccc2c3ccccc3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G19 compound treatment 194040.0 27400.0 1.87 189560.0 25900.0 1.93 2.6832 0.9999 3615779 CMLD4_000446 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NC3CCCCC3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G20 compound treatment 189120.0 22500.0 1.53 182640.0 19000.0 1.41 2.0819 0.9992 3615783 CMLD4_000447 COC(=O)CCCCCN1C(=C(C(NC1=O)c2ccccc2)C(=O)OCc3ccccc3)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G21 compound treatment 175320.0 8680.0 0.59 167840.0 4160.0 0.31 0.6377 0.9544 3615784 CMLD4_000448 CC(Cc1ccccc1)C(=O)NCC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G22 compound treatment 191480.0 24800.0 1.69 180280.0 16600.0 1.24 2.0714 0.988 3615786 CMLD4_000449 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(Cl)cc3)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G23 mock treatment 170520.0 3880.0 0.26 167240.0 3560.0 0.27 0.3747 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 G24 mock treatment 162760.0 -3880.0 -0.26 160080.0 -3600.0 -0.27 -0.3762 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H01 mock treatment 174560.0 7920.0 0.54 168680.0 5000.0 0.37 0.6453 0.9835 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H02 mock treatment 170680.0 4040.0 0.28 169360.0 5680.0 0.42 0.494 0.9785 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H03 compound treatment 206400.0 39800.0 2.71 196320.0 32600.0 2.43 3.6348 0.9985 3615788 CMLD4_000450 CCCCNC(=O)C(N(CCc1c[nH]c2ccccc12)C(=O)CCCCCN3C(=C(C(NC3=O)c4ccc(cc4)c5ccccc5)C(=O)OCc6ccccc6)C)c7ccc(OCC(=O)OC)c(c7)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H04 compound treatment 181680.0 15000.0 1.03 168560.0 4880.0 0.36 0.9822 0.9027 3615789 CMLD4_000451 COC(=O)N1[C@H](C)C=C[C@]1(Cc2ccccc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H05 compound treatment 181800.0 15200.0 1.03 173120.0 9440.0 0.7 1.228 0.9823 3615793 CMLD4_000452 COC(=O)C1(CC(C)C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H06 compound treatment 202120.0 35500.0 2.42 197920.0 34200.0 2.55 3.5127 0.9997 3615794 CMLD4_000453 CC1(C=CC2(CCCCC2)N1C(=O)c3ccccc3)C(=O)NCCCNc4ncc(cc4Cl)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H07 compound treatment 181360.0 14700.0 1.0 182280.0 18600.0 1.38 1.6888 0.9875 3615796 CMLD4_000454 CC(C)CC1(C=CCN1C(=O)C)C(=O)NCc2ccc(C)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H08 compound treatment 180040.0 13400.0 0.91 177200.0 13500.0 1.01 1.3578 0.9988 3615798 CMLD4_000455 COCCNC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H09 compound treatment 176880.0 10200.0 0.7 174240.0 10600.0 0.79 1.0497 0.9983 3615801 CMLD4_000456 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCC3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H10 compound treatment 184080.0 17400.0 1.19 179720.0 16000.0 1.19 1.6852 1.0 3615803 CMLD4_000457 COC(=O)CNC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H11 compound treatment 179920.0 13300.0 0.91 175520.0 11800.0 0.88 1.2636 0.9999 3615807 CMLD4_000458 CC(=O)N1CC=CC1(C)C(=O)NCC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H12 compound treatment 179560.0 12900.0 0.88 177680.0 14000.0 1.04 1.36 0.9965 3615809 CMLD4_000459 CNC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H13 compound treatment 184120.0 17500.0 1.19 181000.0 17300.0 1.29 1.7545 0.9992 3615813 CMLD4_000460 COC(=O)N1CC=CC1(C)C(=O)NCC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H14 compound treatment 173880.0 7240.0 0.49 169280.0 5600.0 0.42 0.6441 0.9965 3615815 CMLD4_000461 CNC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H15 compound treatment 176760.0 10100.0 0.69 171720.0 8040.0 0.6 0.9113 0.9975 3615817 CMLD4_000462 CC1(C=CCN1C(=O)c2ccccc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H16 compound treatment 180520.0 13900.0 0.95 174400.0 10700.0 0.8 1.2336 0.9964 3615818 CMLD4_000463 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H17 compound treatment 177640.0 11000.0 0.75 172400.0 8720.0 0.65 0.9895 0.9974 3615823 CMLD4_000464 CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H18 mock treatment 176520.0 9880.0 0.67 172160.0 8480.0 0.63 0.9229 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H19 compound treatment 196320.0 29700.0 2.02 196760.0 33100.0 2.46 3.1721 0.9953 3615825 CMLD4_000465 C[C@@]1(C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3)C(=O)NCCc4c[nH]c5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H20 mock treatment 171600.0 4960.0 0.34 166080.0 2400.0 0.18 0.3657 0.9556 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H21 compound treatment 172680.0 6040.0 0.41 168800.0 5120.0 0.38 0.5609 0.9993 3615830 CMLD4_000466 CC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H22 mock treatment 170720.0 4080.0 0.28 167880.0 4200.0 0.31 0.418 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H23 mock treatment 169320.0 2680.0 0.18 165200.0 1520.0 0.11 0.2095 0.9735 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 H24 mock treatment 164000.0 -2640.0 -0.18 163120.0 -557.0 -0.04 -0.1564 -0.8479 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I01 mock treatment 170000.0 3360.0 0.23 162440.0 -1240.0 -0.09 0.097 0.3927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I02 mock treatment 173600.0 6960.0 0.47 164800.0 1120.0 0.08 0.3948 0.819 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I03 compound treatment 175840.0 9200.0 0.63 173120.0 9440.0 0.7 0.9406 0.9984 3615834 CMLD4_000467 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)c2cnccn2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I04 compound treatment 201320.0 34700.0 2.36 194880.0 31200.0 2.32 3.3142 1.0 3615836 CMLD4_000468 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)Nc3ccc(OC)cc3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I05 compound treatment 183160.0 16500.0 1.13 173800.0 10100.0 0.75 1.3293 0.9809 3615841 CMLD4_000469 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)c2cccnc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I06 compound treatment 214200.0 47600.0 3.24 213160.0 49500.0 3.68 4.8971 0.998 3615847 CMLD4_000470 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(C)o3)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I07 compound treatment 197080.0 30400.0 2.08 197840.0 34200.0 2.54 3.2655 0.9949 3615851 CMLD4_000471 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)Oc2ccc(F)cc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I08 compound treatment 261000.0 94400.0 6.43 239800.0 76100.0 5.67 8.5553 0.998 3615856 CMLD4_000472 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3nc4ccccc4s3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I09 compound treatment 199760.0 33100.0 2.26 197800.0 34100.0 2.54 3.3926 0.9983 3615862 CMLD4_000473 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)Oc2ccc(F)cc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I10 compound treatment 240000.0 73400.0 5.0 222360.0 58700.0 4.37 6.6251 0.9977 3615864 CMLD4_000474 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(cc3)c4ccccc4)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I11 compound treatment 216160.0 49500.0 3.38 194040.0 30400.0 2.26 3.9854 0.9809 3615868 CMLD4_000475 C[C@H]([C@H]1C[C@]1(C)[C@H](NS(=O)(=O)c2ccc(cc2)c3ccccc3)c4ccccc4)C(=O)Nc5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I12 compound treatment 197520.0 30900.0 2.11 186560.0 22900.0 1.7 2.6931 0.9945 3615870 CMLD4_000476 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)Nc3ccccc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I13 compound treatment 187760.0 21100.0 1.44 183200.0 19500.0 1.45 2.0458 1.0 3615875 CMLD4_000477 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)OCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I14 compound treatment 178000.0 11400.0 0.77 177160.0 13500.0 1.0 1.2574 0.9918 3615881 CMLD4_000478 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(C)on3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I15 compound treatment 179080.0 12400.0 0.85 175520.0 11800.0 0.88 1.2231 0.9998 3615886 CMLD4_000479 CC(Cc1ccccc1)C(=O)N[C@@H](CO)Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I16 compound treatment 174480.0 7840.0 0.53 173920.0 10200.0 0.76 0.9172 0.9849 3615892 CMLD4_000480 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N[C@@H](CO)Cc3ccccc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I17 compound treatment 195360.0 28700.0 1.96 193120.0 29400.0 2.19 2.9342 0.9984 3615898 CMLD4_000481 COc1ccc(CNC(=O)C(C)Cc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I18 compound treatment 198040.0 31400.0 2.14 199680.0 36000.0 2.68 3.4087 0.9938 3615902 CMLD4_000482 CCCCNC(=O)C(N(CCC1=CCCCC1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C)c6ccc(OCC(=O)OC)c(c6)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I19 compound treatment 175480.0 8840.0 0.6 173880.0 10200.0 0.76 0.9633 0.9935 3615904 CMLD4_000483 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N3CCN(C)CC3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I20 compound treatment 201240.0 34600.0 2.36 198160.0 34500.0 2.57 3.4829 0.9991 3615909 CMLD4_000484 COC(=O)CCCCCN1C(=C(C(CC2CC2)NC1=O)C(=O)OCc3ccccc3)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I21 compound treatment 172240.0 5600.0 0.38 170120.0 6440.0 0.48 0.6092 0.9937 3615913 CMLD4_000485 CC(Cc1ccccc1)C(=O)NCc2ccncc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I22 compound treatment 184080.0 17400.0 1.19 174600.0 10900.0 0.81 1.4158 0.9828 3615915 CMLD4_000486 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)[N+](=O)[O-])C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I23 mock treatment 169600.0 2960.0 0.2 167160.0 3480.0 0.26 0.3262 0.9924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 I24 mock treatment 162200.0 -4440.0 -0.3 160200.0 -3480.0 -0.26 -0.3969 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J01 mock treatment 171920.0 5280.0 0.36 167680.0 4000.0 0.3 0.4654 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J02 mock treatment 172600.0 5960.0 0.41 166800.0 3120.0 0.23 0.4518 0.9648 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J03 compound treatment 195280.0 28600.0 1.95 187280.0 23600.0 1.76 2.623 0.9986 3615919 CMLD4_000487 CCCCCCN(C(C(=O)NCCCC)c1ccc(O)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J04 compound treatment 184600.0 18000.0 1.22 173720.0 10000.0 0.75 1.3945 0.972 3615921 CMLD4_000488 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J05 compound treatment 181400.0 14800.0 1.01 176480.0 12800.0 0.95 1.3855 0.9996 3615929 CMLD4_000489 COC(=O)CNC(=O)C1(CC(C)C)C=CCN1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J06 compound treatment 210880.0 44200.0 3.02 199360.0 35700.0 2.66 4.0108 0.998 3615932 CMLD4_000490 COC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J07 compound treatment 181280.0 14600.0 1.0 176800.0 13100.0 0.98 1.3966 0.9999 3615938 CMLD4_000491 COCCNC(=O)C1(CC(C)C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J08 compound treatment 179520.0 12900.0 0.88 174640.0 11000.0 0.82 1.198 0.9993 3615940 CMLD4_000492 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)C)C(=O)NCc3cc(F)cc(c3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J09 compound treatment 179760.0 13100.0 0.89 175120.0 11400.0 0.85 1.2349 0.9997 3615946 CMLD4_000493 CNC(=O)C1(CC(C)C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J10 compound treatment 204680.0 38000.0 2.59 203800.0 40100.0 2.99 3.9456 0.9975 3615948 CMLD4_000494 COC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCc3ccc(cc3)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J11 compound treatment 198360.0 31700.0 2.16 197840.0 34200.0 2.54 3.3272 0.9968 3615953 CMLD4_000495 CC(=O)N1CC=CC1(C)C(=O)NCc2ccc(C)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J12 compound treatment 200160.0 33500.0 2.29 194320.0 30600.0 2.28 3.2288 1.0 3615957 CMLD4_000496 COC(=O)N1[C@H](C)C=C[C@]1(Cc2ccccc2)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J13 compound treatment 177600.0 11000.0 0.75 174200.0 10500.0 0.78 1.0823 0.9997 3615962 CMLD4_000497 CNC(=O)C1(C)C=CCN1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J14 compound treatment 186600.0 20000.0 1.36 186200.0 22500.0 1.68 2.1477 0.9947 3615964 CMLD4_000498 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N(C)Cc3ccccc3)/C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J15 compound treatment 183000.0 16400.0 1.12 177080.0 13400.0 1.0 1.4942 0.9984 3615969 CMLD4_000499 CC1(C=CC2(CCCCC2)N1C(=O)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J16 compound treatment 176200.0 9560.0 0.65 171600.0 7920.0 0.59 0.878 0.9987 3615973 CMLD4_000500 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)CO)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J17 compound treatment 170600.0 3960.0 0.27 174800.0 11100.0 0.83 0.7764 0.8916 3615978 CMLD4_000501 CNC(=O)C1(C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J18 mock treatment 174440.0 7800.0 0.53 171400.0 7720.0 0.57 0.7826 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J19 compound treatment 187520.0 20900.0 1.42 185040.0 21400.0 1.59 2.131 0.9985 3615981 CMLD4_000502 C[C@@]1(C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3)C(=O)NCCCNc4ncc(cc4Cl)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J20 mock treatment 172840.0 6200.0 0.42 167720.0 4040.0 0.3 0.5118 0.9861 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J21 compound treatment 176720.0 10100.0 0.69 173880.0 10200.0 0.76 1.0231 0.9988 3615989 CMLD4_000503 CC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J22 mock treatment 162400.0 -4240.0 -0.29 169720.0 6040.0 0.45 0.1138 0.2129 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J23 mock treatment 169120.0 2480.0 0.17 163040.0 -637.0 -0.05 0.0862 0.4903 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 J24 mock treatment 159200.0 -7440.0 -0.51 161520.0 -2160.0 -0.16 -0.472 -0.8876 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K01 mock treatment 173880.0 7240.0 0.49 163720.0 43.1 0.0 0.3514 0.7117 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K02 mock treatment 174960.0 8320.0 0.57 166120.0 2440.0 0.18 0.5298 0.8892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K03 compound treatment 178120.0 11500.0 0.78 171280.0 7600.0 0.57 0.9537 0.9873 3615993 CMLD4_000504 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)c2cc(C)nn2C)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K04 compound treatment 205320.0 38700.0 2.64 196720.0 33000.0 2.46 3.6038 0.9994 3615994 CMLD4_000505 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N[C@@H](CO)Cc3ccccc3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K05 compound treatment 183440.0 16800.0 1.15 181520.0 17800.0 1.33 1.7491 0.9973 3615998 CMLD4_000506 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)Oc2ccc(F)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K06 compound treatment 208120.0 41500.0 2.83 205640.0 42000.0 3.12 4.2083 0.9988 3616001 CMLD4_000507 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(C)n(C)n3)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K07 compound treatment 192880.0 26200.0 1.79 188560.0 24900.0 1.85 2.5747 0.9999 3616006 CMLD4_000508 C[C@H]([C@H]1C[C@]1(C)[C@H](NS(=O)(=O)c2ccccc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K08 compound treatment 181160.0 14500.0 0.99 176160.0 12500.0 0.93 1.3571 0.9995 3616010 CMLD4_000509 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N3CCN(C)CC3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K09 compound treatment 198440.0 31800.0 2.17 188200.0 24500.0 1.83 2.8238 0.9963 3616013 CMLD4_000510 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NS(=O)(=O)c2ccccc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K10 compound treatment 218600.0 52000.0 3.54 210280.0 46600.0 3.47 4.9577 0.9999 3616016 CMLD4_000511 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(OC)c(OC)c3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K11 compound treatment 185560.0 18900.0 1.29 181560.0 17900.0 1.33 1.8534 0.9999 3616021 CMLD4_000512 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)C)c2ccccc2)C(=O)Nc3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K12 compound treatment 181080.0 14400.0 0.98 177520.0 13800.0 1.03 1.4248 0.9997 3616024 CMLD4_000513 CNC(=O)[C@H](C)/C=C(/C(NC(=O)OCc1ccccc1)c2ccc(cc2)C(=O)OC)\c3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K13 compound treatment 186600.0 20000.0 1.36 186080.0 22400.0 1.67 2.1414 0.9949 3616029 CMLD4_000514 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)c2ccncc2Cl)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K14 compound treatment 204960.0 38300.0 2.61 205360.0 41700.0 3.1 4.0412 0.9964 3616034 CMLD4_000515 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(cc3)c4ccccc4)/c5cccnc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K15 compound treatment 210040.0 43400.0 2.96 204880.0 41200.0 3.07 4.2608 0.9998 3616042 CMLD4_000516 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K16 compound treatment 189200.0 22600.0 1.54 184480.0 20800.0 1.55 2.1826 1.0 3616048 CMLD4_000517 CCCCCCN(C(C(=O)NCCCC)c1ccccc1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K17 compound treatment 187120.0 20500.0 1.4 178400.0 14700.0 1.1 1.7623 0.9928 3616050 CMLD4_000518 COCCNC(=O)[C@H](C)/C=C/C(NC(=O)OCc1ccccc1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K18 compound treatment 237880.0 71200.0 4.86 228440.0 64800.0 4.82 6.8428 1.0 3616056 CMLD4_000519 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)O)c(c1)C(=O)O)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K19 compound treatment 186880.0 20200.0 1.38 183360.0 19700.0 1.46 2.0118 0.9996 3616058 CMLD4_000520 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N(C)Cc3cccnc3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K20 compound treatment 193160.0 26500.0 1.81 187640.0 24000.0 1.78 2.5398 1.0 3616062 CMLD4_000521 CCCCNC(=O)C(N(CCOC)C(=O)CCCCCN1C(=C(C(NC1=O)c2ccc(cc2)c3ccccc3)C(=O)OCc4ccccc4)C)c5ccc(OCC(=O)OC)c(c5)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K21 compound treatment 208800.0 42200.0 2.87 211240.0 47600.0 3.54 4.5358 0.9947 3616065 CMLD4_000522 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCc3ccc(OC)c(O)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K22 compound treatment 186080.0 19400.0 1.33 180640.0 17000.0 1.26 1.8301 0.9997 3616070 CMLD4_000523 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc4ccccc4c3)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K23 mock treatment 171160.0 4520.0 0.31 161480.0 -2200.0 -0.16 0.1024 0.2935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 K24 mock treatment 162800.0 -3840.0 -0.26 158120.0 -5560.0 -0.41 -0.4774 -0.9756 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L01 mock treatment 166120.0 -517.0 -0.04 165920.0 2240.0 0.17 0.0931 0.5458 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L02 mock treatment 172680.0 6040.0 0.41 168200.0 4520.0 0.34 0.5294 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L03 compound treatment 178400.0 11800.0 0.8 176920.0 13200.0 0.99 1.264 0.9948 3616072 CMLD4_000524 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)cc1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L04 compound treatment 190360.0 23700.0 1.62 182840.0 19200.0 1.43 2.1522 0.998 3616077 CMLD4_000525 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L05 compound treatment 175520.0 8880.0 0.61 172680.0 9000.0 0.67 0.9021 0.9987 3616082 CMLD4_000526 CC(C)CC1(C=CCN1C(=O)C)C(=O)NCc2cc(F)cc(c2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L06 compound treatment 229720.0 63100.0 4.3 224600.0 60900.0 4.53 6.2474 0.9997 3616084 CMLD4_000527 COC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L07 compound treatment 176440.0 9800.0 0.67 174800.0 11100.0 0.83 1.058 0.9944 3616089 CMLD4_000528 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L08 compound treatment 178600.0 12000.0 0.82 172640.0 8960.0 0.67 1.0484 0.995 3616091 CMLD4_000529 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)C)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L09 compound treatment 189760.0 23100.0 1.58 174440.0 10800.0 0.8 1.6812 0.9507 3616096 CMLD4_000530 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCCc3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L10 compound treatment 178440.0 11800.0 0.8 175240.0 11600.0 0.86 1.1775 0.9994 3616098 CMLD4_000531 COC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L11 compound treatment 181600.0 15000.0 1.02 173000.0 9320.0 0.69 1.212 0.9824 3616102 CMLD4_000532 COC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L12 compound treatment 187640.0 21000.0 1.43 182800.0 19100.0 1.42 2.0189 1.0 3616103 CMLD4_000533 COC(=O)N1[C@H](C)C=C[C@]1(Cc2ccccc2)C(=O)NCCCNc3ncc(cc3Cl)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L13 compound treatment 190360.0 23700.0 1.62 185080.0 21400.0 1.59 2.27 1.0 3616109 CMLD4_000534 COC(=O)N1CC=CC1(C)C(=O)NCc2ccc(C)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L14 compound treatment 189520.0 22900.0 1.56 183520.0 19800.0 1.48 2.1475 0.9996 3616111 CMLD4_000535 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCc3c[nH]c4ccccc34)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L15 compound treatment 186600.0 20000.0 1.36 183200.0 19500.0 1.45 1.9898 0.9995 3616118 CMLD4_000536 CC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L16 compound treatment 174880.0 8240.0 0.56 172320.0 8640.0 0.64 0.8523 0.9977 3616124 CMLD4_000537 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)O)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L17 compound treatment 179920.0 13300.0 0.91 172320.0 8640.0 0.64 1.0952 0.986 3616130 CMLD4_000538 CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCCc3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L18 mock treatment 174840.0 8200.0 0.56 169640.0 5960.0 0.44 0.7093 0.9934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L19 compound treatment 179680.0 13000.0 0.89 167160.0 3480.0 0.26 0.8121 0.8768 3616134 CMLD4_000539 CC(=O)N1C(C)(C=CC21CCCCC2)C(=O)NCCN3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L20 mock treatment 174840.0 8200.0 0.56 168400.0 4720.0 0.35 0.644 0.975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L21 compound treatment 179680.0 13000.0 0.89 176080.0 12400.0 0.92 1.2815 0.9998 3616137 CMLD4_000540 CNC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L22 mock treatment 166000.0 -637.0 -0.04 165160.0 1480.0 0.11 0.0473 0.3992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L23 mock treatment 163600.0 -3040.0 -0.21 160360.0 -3320.0 -0.25 -0.321 -0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 L24 mock treatment 158480.0 -8160.0 -0.56 157080.0 -6600.0 -0.49 -0.7404 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M01 mock treatment 173480.0 6840.0 0.47 168520.0 4840.0 0.36 0.5848 0.9919 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M02 mock treatment 172560.0 5920.0 0.4 171720.0 8040.0 0.6 0.7088 0.9816 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M03 compound treatment 177440.0 10800.0 0.74 173560.0 9880.0 0.74 1.0409 1.0 3616142 CMLD4_000541 COC(=O)[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccnc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M04 compound treatment 198040.0 31400.0 2.14 193640.0 30000.0 2.23 3.0908 0.9998 3616146 CMLD4_000542 CCNC(=O)[C@H](C)/C=C/C(NC(=O)OCc1ccccc1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M05 compound treatment 179760.0 13100.0 0.89 181760.0 18100.0 1.35 1.5843 0.9803 3616155 CMLD4_000543 COC(=O)[C@H]1C[C@@H]1[C@H](NS(=O)(=O)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M06 compound treatment 200960.0 34300.0 2.34 192680.0 29000.0 2.16 3.181 0.9992 3616159 CMLD4_000544 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccncc3)/I 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M07 compound treatment 185840.0 19200.0 1.31 181240.0 17600.0 1.31 1.8501 1.0 3616164 CMLD4_000545 C[C@H]([C@H]1C[C@]1(C)[C@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4)C(=O)Nc5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M08 compound treatment 216880.0 50200.0 3.43 214240.0 50600.0 3.76 5.0832 0.9989 3616170 CMLD4_000546 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NC3CCCCC3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M09 compound treatment 203680.0 37000.0 2.53 194280.0 30600.0 2.28 3.3964 0.9987 3616175 CMLD4_000547 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4)C(=O)Nc5ccc6ccccc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M10 compound treatment 178840.0 12200.0 0.83 182960.0 19300.0 1.44 1.6031 0.9664 3616177 CMLD4_000548 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)O)/c3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M11 compound treatment 197840.0 31200.0 2.13 201680.0 38000.0 2.83 3.5043 0.9901 3616183 CMLD4_000549 COC(=O)[C@H]1C[C@@H]1[C@H](NC(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M12 compound treatment 180160.0 13500.0 0.92 180240.0 16600.0 1.23 1.5236 0.9898 3616187 CMLD4_000550 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3nc4ccccc4n3C)/c5cccnc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M13 compound treatment 204840.0 38200.0 2.6 202280.0 38600.0 2.87 3.8733 0.9988 3616193 CMLD4_000551 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NS(=O)(=O)c2c(C)nn(C)c2Cl)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M14 compound treatment 181560.0 14900.0 1.02 177600.0 13900.0 1.04 1.4522 1.0 3616197 CMLD4_000552 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NC3CCCCC3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M15 compound treatment 200520.0 33900.0 2.31 194760.0 31100.0 2.31 3.2693 1.0 3616201 CMLD4_000553 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(cc3)c4ccccc4)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M16 compound treatment 199680.0 33000.0 2.25 187440.0 23800.0 1.77 2.8436 0.9928 3616205 CMLD4_000554 CCCCCCN(C(C(=O)NCCCC)c1ccc(O)cc1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M17 compound treatment 180080.0 13400.0 0.92 176480.0 12800.0 0.95 1.3219 0.9998 3616207 CMLD4_000555 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M18 compound treatment 209040.0 42400.0 2.89 211000.0 47300.0 3.52 4.5347 0.9952 3616215 CMLD4_000556 CCCCNC(=O)C(N(CCN1CCOCC1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)[N+](=O)[O-])C(=O)OCc4ccccc4)C)c5ccc(cc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M19 compound treatment 191760.0 25100.0 1.71 183680.0 20000.0 1.49 2.2639 0.9976 3616217 CMLD4_000557 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(F)cc(F)c3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M20 compound treatment 200120.0 33500.0 2.28 187600.0 23900.0 1.78 2.8732 0.9924 3616223 CMLD4_000558 CCCCCCN(C(C(=O)NCCCC)c1ccccn1)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M21 compound treatment 192760.0 26100.0 1.78 187120.0 23400.0 1.74 2.4931 0.9999 3616226 CMLD4_000559 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)NCCc3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M22 compound treatment 173840.0 7200.0 0.49 166480.0 2800.0 0.21 0.4948 0.9273 3616232 CMLD4_000560 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccccc3c4ccccc4)C(=O)OCc5ccccc5)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M23 mock treatment 168720.0 2080.0 0.14 167120.0 3440.0 0.26 0.2816 0.9612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 M24 mock treatment 165880.0 -757.0 -0.05 160320.0 -3360.0 -0.25 -0.2132 -0.8355 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N01 mock treatment 171400.0 4760.0 0.32 168320.0 4640.0 0.35 0.474 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N02 mock treatment 172960.0 6320.0 0.43 167560.0 3880.0 0.29 0.5092 0.9811 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N03 compound treatment 256240.0 89600.0 6.11 230200.0 66500.0 4.95 7.8206 0.9946 3616235 CMLD4_000561 CC1=C(C(NC(=O)N1CCCCCC(=O)O)c2ccc(cc2)C3CCCCC3)C(=O)OCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N04 compound treatment 177800.0 11200.0 0.76 175680.0 12000.0 0.89 1.1699 0.9968 3616238 CMLD4_000562 COCCNC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N05 compound treatment 178360.0 11700.0 0.8 166600.0 2920.0 0.22 0.719 0.868 3616240 CMLD4_000563 CC(C)CC1(C=CCN1C(=O)C)C(=O)NCCN2CCOCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N06 compound treatment 185600.0 19000.0 1.29 180600.0 16900.0 1.26 1.8048 0.9999 3616243 CMLD4_000564 COC(=O)CNC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N07 compound treatment 185040.0 18400.0 1.25 178040.0 14400.0 1.07 1.6431 0.9968 3616248 CMLD4_000565 COC(=O)C1(CC(C)C)C=CC[N+]1(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N08 compound treatment 182880.0 16200.0 1.11 171440.0 7760.0 0.58 1.1916 0.954 3616251 CMLD4_000566 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)C)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N09 compound treatment 217560.0 50900.0 3.47 210160.0 46500.0 3.46 4.9012 1.0 3616256 CMLD4_000567 CC(C)CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N10 compound treatment 184200.0 17600.0 1.2 175800.0 12100.0 0.9 1.4847 0.9903 3616260 CMLD4_000568 CNC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N11 compound treatment 186600.0 20000.0 1.36 177080.0 13400.0 1.0 1.6678 0.9883 3616264 CMLD4_000569 COC(=O)N1CC=CC1(C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N12 compound treatment 289840.0 123000.0 8.4 277760.0 114000.0 8.49 11.9434 1.0 3616268 CMLD4_000570 CN(C)c1ccc(CNC(=O)[C@@]2(C)C=C[C@@H](Cc3ccccc3)N2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N13 compound treatment 182320.0 15700.0 1.07 178480.0 14800.0 1.1 1.5351 0.9999 3616276 CMLD4_000571 COC(=O)C1(C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N14 compound treatment 207400.0 40800.0 2.78 190480.0 26800.0 1.99 3.3757 0.9868 3616277 CMLD4_000572 COCCNC(=O)[C@H](C)/C=C(\I)/C(NC(=O)OCc1ccccc1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N15 compound treatment 181040.0 14400.0 0.98 176320.0 12600.0 0.94 1.3597 0.9998 3616282 CMLD4_000573 C[C@@]1(C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N16 mock treatment 174680.0 8040.0 0.55 180520.0 16800.0 1.25 1.2742 0.9312 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N17 compound treatment 175640.0 9000.0 0.61 170920.0 7240.0 0.54 0.8152 0.9979 3616287 CMLD4_000574 CC1(C=CCN1C(=O)c2ccccc2)C(=O)NCCCNc3ncc(cc3Cl)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N18 mock treatment 173760.0 7120.0 0.49 172360.0 8680.0 0.65 0.8004 0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N19 compound treatment 182280.0 15600.0 1.07 181200.0 17500.0 1.3 1.6763 0.995 3616288 CMLD4_000575 CC(=O)N1C(C)(C=CC21CCCCC2)C(=O)NCc3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N20 mock treatment 173640.0 7000.0 0.48 172720.0 9040.0 0.67 0.8135 0.9859 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N21 compound treatment 176000.0 9360.0 0.64 172960.0 9280.0 0.69 0.9399 0.9992 3616289 CMLD4_000576 CC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCCc3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N22 mock treatment 165160.0 -1480.0 -0.1 160840.0 -2840.0 -0.21 -0.2205 -0.9426 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N23 mock treatment 162800.0 -3840.0 -0.26 162200.0 -1480.0 -0.11 -0.2627 -0.9258 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 N24 mock treatment 165240.0 -1400.0 -0.1 161840.0 -1840.0 -0.14 -0.164 -0.9844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O01 mock treatment 165880.0 -757.0 -0.05 168800.0 5120.0 0.38 0.2331 0.6059 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O02 mock treatment 169200.0 2560.0 0.17 167640.0 3960.0 0.29 0.3321 0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O03 compound treatment 174000.0 7360.0 0.5 171720.0 8040.0 0.6 0.7783 0.9962 3616291 CMLD4_000577 COC(=O)[C@@H]1C[C@H]1[C@@H](NS(=O)(=O)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O04 compound treatment 174760.0 8120.0 0.55 171280.0 7600.0 0.57 0.7917 0.9999 3616292 CMLD4_000578 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)N[C@H](C)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O05 compound treatment 179880.0 13200.0 0.9 173200.0 9520.0 0.71 1.1396 0.9928 3616295 CMLD4_000579 C[C@H]([C@H]1C[C@]1(C)[C@H](NC(=O)c2ccccc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O06 compound treatment 197520.0 30900.0 2.11 187080.0 23400.0 1.74 2.7205 0.9956 3616298 CMLD4_000580 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N(C)Cc3cccnc3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O07 compound treatment 204120.0 37500.0 2.56 198080.0 34400.0 2.56 3.6176 1.0 3616302 CMLD4_000581 C[C@H]([C@@H]1C[C@@]1(C)[C@@H](NC(=O)c2ccccc2)c3ccccc3)C(=O)Nc4ccc5ccccc5c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O08 compound treatment 175720.0 9080.0 0.62 167480.0 3800.0 0.28 0.638 0.9371 3616304 CMLD4_000582 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCN3CCOCC3)/F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O09 compound treatment 202560.0 35900.0 2.45 188200.0 24500.0 1.83 3.0224 0.9895 3616308 CMLD4_000583 COC(=O)[C@@H]1C[C@H]1[C@@H](NS(=O)(=O)c2ccc(cc2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O10 compound treatment 195440.0 28800.0 1.96 192280.0 28600.0 2.13 2.8939 0.9992 3616311 CMLD4_000584 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)N(C)Cc3ccccc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O11 compound treatment 179080.0 12400.0 0.85 178120.0 14400.0 1.07 1.36 0.9931 3616314 CMLD4_000585 COC(=O)[C@@H]1C[C@H]1[C@@H](NS(=O)(=O)c2ccc3ccccc3c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O12 compound treatment 179200.0 12600.0 0.86 182840.0 19200.0 1.43 1.6142 0.9702 3616316 CMLD4_000586 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(C)o3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O13 compound treatment 176280.0 9640.0 0.66 180400.0 16700.0 1.24 1.345 0.9555 1089379 CMLD4_000587 CC(Cc1ccccc1)C(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O14 compound treatment 192360.0 25700.0 1.75 188200.0 24500.0 1.83 2.5307 0.9998 3616321 CMLD4_000588 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)Nc3ccc(OC)cc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O15 compound treatment 188800.0 22200.0 1.51 188000.0 24300.0 1.81 2.3485 0.996 3616325 CMLD4_000589 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccc(OC)c(OC)c3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O16 compound treatment 198240.0 31600.0 2.15 196000.0 32300.0 2.41 3.2246 0.9985 3616328 CMLD4_000590 CCCCCCN(C(C(=O)NCCCC)c1ccc(cc1)c2ccccc2)C(=O)CCCCCN3C(=C(C(NC3=O)c4ccc(cc4)c5ccccc5)C(=O)OCc6ccccc6)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O17 compound treatment 198560.0 31900.0 2.18 192240.0 28600.0 2.13 3.0422 0.9999 3616330 CMLD4_000591 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C=C/[C@@H](C)C(=O)N(C)Cc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O18 compound treatment 175000.0 8360.0 0.57 178040.0 14400.0 1.07 1.1591 0.9567 3616333 CMLD4_000592 CC1=C(C(NC(=O)N1CCCCCC(=O)O)C2CCCCC2)C(=O)OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O19 compound treatment 179560.0 12900.0 0.88 185120.0 21400.0 1.6 1.7515 0.9608 3616334 CMLD4_000593 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3cc(C)on3)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O20 compound treatment 167640.0 1000.0 0.07 170360.0 6680.0 0.5 0.4001 0.7968 3616338 CMLD4_000594 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)c3ccc(cc3)C(F)(F)F)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O21 compound treatment 185920.0 19300.0 1.31 177840.0 14200.0 1.05 1.675 0.994 3616340 CMLD4_000595 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCCc3c[nH]c4ccc(OC)cc34)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O22 compound treatment 191400.0 24800.0 1.69 182880.0 19200.0 1.43 2.2044 0.9966 3616344 CMLD4_000596 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)C3CCCCC3)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O23 mock treatment 162920.0 -3720.0 -0.25 159960.0 -3720.0 -0.28 -0.3748 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 O24 mock treatment 162040.0 -4600.0 -0.31 163160.0 -517.0 -0.04 -0.2488 -0.788 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P01 mock treatment 170000.0 3360.0 0.23 169040.0 5360.0 0.4 0.4444 0.9654 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P02 mock treatment 173480.0 6840.0 0.47 162040.0 -1640.0 -0.12 0.2437 0.5055 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P03 compound treatment 220040.0 53400.0 3.64 211400.0 47700.0 3.55 5.086 0.9999 3616346 CMLD4_000597 CCCCCCN(C(C(=O)NCCCC)c1ccc(OCC(=O)OC)c(c1)C(=O)OC)C(=O)CCCCCN2C(=C(C(NC2=O)C3CC3)C(=O)OCc4ccccc4)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P04 compound treatment 193240.0 26600.0 1.81 175160.0 11500.0 0.85 1.8868 0.9411 3616349 CMLD4_000598 CC1(C=CC2(CCCCC2)N1C(=O)c3ccccc3)C(=O)NCc4cc(F)cc(c4)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P05 compound treatment 172440.0 5800.0 0.4 170680.0 7000.0 0.52 0.6483 0.9907 3616350 CMLD4_000599 CC(C)CC1(C=CCN1C(=O)C)C(=O)NCc2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P06 compound treatment 175120.0 8480.0 0.58 170280.0 6600.0 0.49 0.7565 0.9967 3616352 CMLD4_000600 C[C@@H]1C=C[C@@](Cc2ccccc2)(N1C(=O)c3ccccc3)C(=O)NCCN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P07 compound treatment 175680.0 9040.0 0.62 173880.0 10200.0 0.76 0.9729 0.9947 3616355 CMLD4_000601 COC(=O)CNC(=O)C1(CC(C)C)C=CCN1C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P08 compound treatment 176440.0 9800.0 0.67 169120.0 5440.0 0.41 0.7591 0.9712 3616356 CMLD4_000602 CNC(=O)[C@@]1(Cc2ccccc2)C=C[C@@H](C)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P09 compound treatment 174680.0 8040.0 0.55 171360.0 7680.0 0.57 0.7921 0.9998 3616358 CMLD4_000603 COCCNC(=O)C1(CC(C)C)C=CCN1C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P10 compound treatment 183520.0 16900.0 1.15 174400.0 10700.0 0.8 1.3782 0.984 3616360 CMLD4_000604 COC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P11 compound treatment 179040.0 12400.0 0.85 173320.0 9640.0 0.72 1.1054 0.9967 3616362 CMLD4_000605 COC(=O)CNC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P12 compound treatment 172240.0 5600.0 0.38 170280.0 6600.0 0.49 0.6176 0.9922 3616363 CMLD4_000606 CN1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCC3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P13 compound treatment 171400.0 4760.0 0.32 171880.0 8200.0 0.61 0.6613 0.9563 3616367 CMLD4_000607 COC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P14 compound treatment 186040.0 19400.0 1.32 191280.0 27600.0 2.05 2.3881 0.9773 3616369 CMLD4_000608 COC(=O)c1ccc(cc1)C(NC(=O)OCc2ccccc2)/C(=C/[C@@H](C)C(=O)NCc3ccccc3)/C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P15 compound treatment 173520.0 6880.0 0.47 168640.0 4960.0 0.37 0.593 0.993 3616372 CMLD4_000609 COC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P16 mock treatment 171280.0 4640.0 0.32 169160.0 5480.0 0.41 0.5124 0.9921 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P17 compound treatment 171200.0 4560.0 0.31 170040.0 6360.0 0.47 0.5549 0.9792 3616374 CMLD4_000610 COCCNC(=O)[C@@]1(C)C=C[C@@H](Cc2ccccc2)N1C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P18 mock treatment 168600.0 1960.0 0.13 166760.0 3080.0 0.23 0.2569 0.9671 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P19 compound treatment 171600.0 4960.0 0.34 164080.0 403.0 0.03 0.2605 0.7668 3616378 CMLD4_000611 CNC(=O)C1(C)C=CC2(CCCCC2)N1C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P20 mock treatment 165640.0 -997.0 -0.07 162080.0 -1600.0 -0.12 -0.1321 -0.9648 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P21 compound treatment 168560.0 1920.0 0.13 158360.0 -5320.0 -0.4 -0.1871 -0.4488 3616381 CMLD4_000612 CC(=O)N1[C@H](Cc2ccccc2)C=C[C@]1(C)C(=O)NCc3ccc(C)o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P22 mock treatment 163400.0 -3240.0 -0.22 159800.0 -3880.0 -0.29 -0.3601 -0.9912 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P23 mock treatment 163400.0 -3240.0 -0.22 161160.0 -2520.0 -0.19 -0.2885 -0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2289 P24 mock treatment 161440.0 -5200.0 -0.35 158960.0 -4720.0 -0.35 -0.4988 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A01 compound treatment 160520.0 -8710.0 -0.59 162520.0 -9000.0 -0.67 -0.8937 -0.9982 3622978 BCB04_000001 COC(=O)c1ccc(CNC(=N)N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A02 compound treatment 160400.0 -8830.0 -0.6 166240.0 -5280.0 -0.39 -0.7037 -0.9787 3622979 BCB04_000002 COC(=O)[C@@H](NC(=O)Cn1cc(nn1)c2ccc(OC)c(OC)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A03 compound treatment 161520.0 -7710.0 -0.53 178880.0 7360.0 0.55 0.0155 0.0204 3622981 BCB04_000003 Nc1ccccc1NC(=O)c2ccc(CNc3nccc(n3)c4cccnc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A04 compound treatment 166600.0 -2630.0 -0.18 166840.0 -4680.0 -0.35 -0.3733 -0.9524 3622982 BCB04_000004 CCOC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)Cn3cc(nn3)c4ccc(OC)c(OC)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A05 compound treatment 159680.0 -9550.0 -0.65 161520.0 -10000.0 -0.74 -0.9868 -0.9978 525 BCB04_000005 CC(=O)Nc1ccc(cc1)C(=O)Nc2ccccc2N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A06 compound treatment 166400.0 -2830.0 -0.19 162640.0 -8880.0 -0.66 -0.6039 -0.877 3622984 BCB04_000006 COC(=O)[C@@H](O)[C@H](c1ccc(OC)cc1)n2cc(nn2)c3ccc(OC)c(OC)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A07 compound treatment 161760.0 -7470.0 -0.51 162960.0 -8560.0 -0.64 -0.8108 -0.9938 3622986 BCB04_000007 CC(=O)Nc1ccc(cc1)C(=O)Nc2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A08 compound treatment 163080.0 -6150.0 -0.42 170120.0 -1400.0 -0.1 -0.3703 -0.8569 3622987 BCB04_000008 O=C1CC[C@H]2N1CCc3c2[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A09 compound treatment 187800.0 18600.0 1.27 189200.0 17700.0 1.32 1.8255 0.9998 3622988 BCB04_000009 ONC(=O)/C=C/c1cccc(c1)S(=O)(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A10 compound treatment 161800.0 -7430.0 -0.51 165800.0 -5720.0 -0.43 -0.6594 -0.9963 3622990 BCB04_000010 COc1ccc2[nH]c3[C@H]4CCC(=O)N4CCc3c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A11 compound treatment 182960.0 13700.0 0.94 187080.0 15600.0 1.16 1.4806 0.9944 3622992 BCB04_000011 CCN(CC)Cc1ccc2cc(COC(=O)Nc3ccc(cc3)C(=O)NO)ccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A12 compound treatment 165320.0 -3910.0 -0.27 167000.0 -4520.0 -0.34 -0.4265 -0.9934 3622993 BCB04_000012 Fc1ccc2[nH]c3[C@H]4CCC(=O)N4CCc3c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A13 mock treatment 162640.0 -6590.0 -0.45 161080.0 -10400.0 -0.78 -0.8673 -0.9661 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A14 mock treatment 162160.0 -7070.0 -0.48 158760.0 -12800.0 -0.95 -1.0125 -0.9506 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A15 compound treatment 169320.0 88.4 0.01 172080.0 558.0 0.04 0.0336 0.8013 3622995 BCB04_000013 ONC(=O)CCCCCC(=O)Nc1cccnc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A16 compound treatment 160000.0 -9230.0 -0.63 157280.0 -14200.0 -1.06 -1.1946 -0.969 3622996 BCB04_000014 Brc1ccc2[nH]c3[C@H]4CCC(=O)N4CCc3c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A17 compound treatment 171680.0 2450.0 0.17 169640.0 -1880.0 -0.14 0.019 0.0872 3622998 BCB04_000015 OCCN(CCc1c[nH]c2ccccc12)Cc3ccc(/C=C/C(=O)NO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A18 compound treatment 160720.0 -8510.0 -0.58 165600.0 -5920.0 -0.44 -0.722 -0.9908 3623000 BCB04_000016 Cc1cccc2c3CCN4[C@H](CCC4=O)c3[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A19 compound treatment 188440.0 19200.0 1.31 195640.0 24100.0 1.8 2.1953 0.988 3623002 BCB04_000017 Cc1[nH]c2ccccc2c1CCNCc3ccc(/C=C/C(=O)NO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A20 compound treatment 162800.0 -6430.0 -0.44 165320.0 -6200.0 -0.46 -0.6364 -0.9997 3623004 BCB04_000018 O=C1CCC[C@H]2N1CCc3c2[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A21 compound treatment 180280.0 11000.0 0.75 183280.0 11800.0 0.88 1.1514 0.9972 3623005 BCB04_000019 CN(C)Cc1c(oc2ccccc12)C(=O)NCCOc3ccc(cc3)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A22 compound treatment 160120.0 -9110.0 -0.62 161240.0 -10300.0 -0.77 -0.9804 -0.9946 3623006 BCB04_000020 C[C@@]12CCC(=O)N2CCc3c1[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A23 compound treatment 160240.0 -8990.0 -0.61 156080.0 -15400.0 -1.15 -1.2461 -0.9567 3615849 BCB04_000021 COc1cc2CCN(CC(C)O)CCCc3c(noc3-c2cc1OC)c4ccc(OCCO[Si](C(C)C)(C(C)C)C(C)C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 A24 compound treatment 153800.0 -15400.0 -1.05 158320.0 -13200.0 -0.98 -1.4387 -0.9994 3623006 BCB04_000022 C[C@@]12CCC(=O)N2CCc3c1[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B01 compound treatment 152000.0 -17200.0 -1.17 154880.0 -16600.0 -1.24 -1.7065 -0.9997 3623008 BCB04_000023 CN1C(=O)N[C@H]2[C@@H](COC(=O)c3ccccc3)[C@]1(CO)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B02 compound treatment 190240.0 21000.0 1.43 192520.0 21000.0 1.56 2.1179 0.9991 3623010 BCB04_000024 CC(C)(C)OC(=O)N[C@@H]1CN(CC2=C1CC(COC(=O)c3ccccc3)C4=C2CN(C4)S(=O)(=O)c5ccc(Br)cc5)S(=O)(=O)c6ccccc6[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B03 compound treatment 172680.0 3450.0 0.24 177680.0 6160.0 0.46 0.4903 0.9519 3623012 BCB04_000025 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO)N=C5SCc6ccccc6CN45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B04 compound treatment 175440.0 6210.0 0.42 171440.0 -81.8 -0.01 0.295 0.6969 3623014 BCB04_000026 Cn1c(=O)n2CC(=C3CN(C[C@H](NC(=O)OC(C)(C)C)[C@H]3n2c1=O)S(=O)(=O)c4ccc(Br)cc4)COC(=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B05 compound treatment 193440.0 24200.0 1.65 184840.0 13300.0 0.99 1.868 0.9702 3623016 BCB04_000027 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2COC(=O)c5ccccc5)N=C6SCc7ccccc7CN46)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B06 compound treatment 170120.0 888.0 0.06 169360.0 -2160.0 -0.16 -0.0709 -0.4126 3623018 BCB04_000028 Cn1c(=O)n2CC(=C3CN(C[C@H](NC(=O)OC(C)(C)C)[C@@H]3n2c1=O)S(=O)(=O)c4ccc(Br)cc4)COC(=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B07 compound treatment 167880.0 -1350.0 -0.09 168520.0 -3000.0 -0.22 -0.2231 -0.9233 3623019 BCB04_000029 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO[Si](C)(C)C(C)(C)C)N=C5SCCCN45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B08 compound treatment 186040.0 16800.0 1.15 185920.0 14400.0 1.07 1.5681 0.9994 3623021 BCB04_000030 Cn1c(=O)n2[C@@H]3[C@@H](COC(=O)c4ccccc4)N(CC3=C5CN(C[C@H](NC(=O)OC(C)(C)C)[C@@H]5n2c1=O)S(=O)(=O)c6ccccc6[N+](=O)[O-])S(=O)(=O)c7ccc(Br)cc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B09 compound treatment 163320.0 -5910.0 -0.4 165960.0 -5560.0 -0.41 -0.5777 -0.9999 3623023 BCB04_000031 OC[C@@]1(Oc2ccccc2[C@@H]3[C@H]1COC(=O)c4ccccc4)N=C5SCc6ccccc6CN35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B10 compound treatment 199680.0 30400.0 2.08 185720.0 14200.0 1.06 2.2151 0.9509 3623025 BCB04_000032 Cn1c(=O)n2[C@@H]3[C@@H](COC(=O)c4ccccc4)N(CC3=C5CN(C[C@@H](NC(=O)OC(C)(C)C)[C@@H]5n2c1=O)S(=O)(=O)c6ccccc6[N+](=O)[O-])S(=O)(=O)c7ccc(Br)cc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B11 compound treatment 162400.0 -6830.0 -0.47 161920.0 -9600.0 -0.71 -0.8347 -0.9785 3623026 BCB04_000033 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO)N=C5SCCCN45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B12 compound treatment 212120.0 42900.0 2.92 207120.0 35600.0 2.65 3.941 0.9988 3623028 BCB04_000034 Cn1c(=O)n2n(c1=O)C34CC(COC(=O)c5ccccc5)C62CN(CC6=C4CN(CC3NC(=O)OC(C)(C)C)S(=O)(=O)c7ccccc7[N+](=O)[O-])S(=O)(=O)c8ccc(Br)cc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B13 mock treatment 164360.0 -4870.0 -0.33 158840.0 -12700.0 -0.94 -0.9023 -0.9017 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B14 mock treatment 158120.0 -11100.0 -0.76 162320.0 -9200.0 -0.68 -1.0199 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B15 compound treatment 174400.0 5170.0 0.35 180720.0 9200.0 0.68 0.7332 0.9523 3623029 BCB04_000035 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2COC(=O)c5ccccc5)N=C6SCCCN46)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B16 compound treatment 193400.0 24200.0 1.65 187560.0 16000.0 1.19 2.0092 0.9875 3623031 BCB04_000036 CC(C)(C)OC(=O)N[C@H]1CN(CC2=C(COC(=O)c3ccccc3)C[C@@H]4[C@H]([C@@H]12)C(=O)N(C4=O)c5ccccc5)S(=O)(=O)c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B17 compound treatment 167560.0 -1670.0 -0.11 171760.0 238.0 0.02 -0.068 -0.59 3623033 BCB04_000037 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2COC(=O)c5ccccc5)N(C)C(=O)N4C(=O)CC(=O)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B18 compound treatment 190840.0 21600.0 1.47 194400.0 22900.0 1.7 2.2457 0.9974 3623035 BCB04_000038 CC(C)(C)OC(=O)N[C@H]1CN(CC2=C(COC(=O)c3ccccc3)C[C@H]4[C@@H]([C@H]12)C(=O)N(C4=O)c5ccccc5)S(=O)(=O)c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B19 compound treatment 160160.0 -9070.0 -0.62 168440.0 -3080.0 -0.23 -0.5995 -0.9089 3623036 BCB04_000039 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO)N(C)c5c6C(=O)N(C)C(=O)c6c(C(=O)C)c(=O)n45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B20 compound treatment 178240.0 9010.0 0.61 182560.0 11000.0 0.82 1.0152 0.9897 3623038 BCB04_000040 CC(C)(C)OC(=O)NCC1=C2CN([C@H](COC(=O)c3ccccc3)[C@@H]2[C@H]4[C@H](C1)C(=O)N(C4=O)c5ccccc5)S(=O)(=O)c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B21 compound treatment 156440.0 -12800.0 -0.87 158680.0 -12800.0 -0.96 -1.2925 -0.999 3623040 BCB04_000041 OC[C@@]1(Oc2ccccc2[C@@H]3[C@H]1COC(=O)c4ccccc4)N=C5SCCCN35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B22 compound treatment 179240.0 10000.0 0.68 173480.0 1960.0 0.15 0.5855 0.8392 3623042 BCB04_000042 CC(C)(C)OC(=O)NCC1=C2CN([C@H](COC(=O)c3ccccc3)[C@H]2[C@@H]4[C@@H](C1)C(=O)N(C4=O)c5ccccc5)S(=O)(=O)c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B23 compound treatment 153320.0 -15900.0 -1.08 155480.0 -16000.0 -1.19 -1.6113 -0.9989 3623043 BCB04_000043 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO[Si](C)(C)C(C)(C)C)N=C5SCC(=O)N45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 B24 compound treatment 155200.0 -14000.0 -0.96 151440.0 -20100.0 -1.49 -1.7333 -0.9768 3623045 BCB04_000044 CC(C)(C)OC(=O)N[C@H]1CN(CC2=C(COC(=O)c3ccccc3)C[C@@]4(Cl)C(Cl)(Cl)[C@@]4(Cl)[C@H]12)S(=O)(=O)c5ccc(Br)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C01 compound treatment 160960.0 -8270.0 -0.56 161880.0 -9640.0 -0.72 -0.9062 -0.9929 3623047 BCB04_000045 COc1cc2CCN(CC(C)O)CCCc3c(noc3-c2cc1OC)c4ccc(OCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C02 compound treatment 163760.0 -5470.0 -0.37 164920.0 -6600.0 -0.49 -0.6112 -0.9908 3623048 BCB04_000046 COc1ccc2[nH]c3c(CCN4C(=O)CC[C@@]43C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C03 compound treatment 165080.0 -4150.0 -0.28 166440.0 -5080.0 -0.38 -0.4676 -0.9898 3623049 BCB04_000047 COc1cc2CCN(CC=C)CCCc3c(noc3-c2cc1OC)c4ccc(OCCO)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C04 compound treatment 160040.0 -9190.0 -0.63 168400.0 -3120.0 -0.23 -0.6074 -0.9088 3623050 BCB04_000048 C[C@@]12C=CC(=O)N2CCc3c1[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C05 compound treatment 165480.0 -3750.0 -0.26 169120.0 -2400.0 -0.18 -0.3073 -0.9847 3556313 BCB04_000049 COc1cc2CCN3CC[C@H]4C(=NO[C@]43c2cc1OC)c5ccc(OCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C06 compound treatment 166920.0 -2310.0 -0.16 166560.0 -4960.0 -0.37 -0.3726 -0.9279 3623052 BCB04_000050 C[C@@]12CCCC(=O)N2CCc3c1[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C07 compound treatment 157080.0 -12200.0 -0.83 166360.0 -5160.0 -0.38 -0.8575 -0.939 3556309 BCB04_000051 COc1cc2CCN3CCC[C@H]4C(=NO[C@]43c2cc1OC)c5ccc(OCCO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C08 compound treatment 164200.0 -5030.0 -0.34 168000.0 -3520.0 -0.26 -0.4279 -0.9912 3623054 BCB04_000052 CCCC[C@@]12CCCC(=O)N2CCc3c1[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C09 compound treatment 159720.0 -9510.0 -0.65 166120.0 -5400.0 -0.4 -0.7428 -0.9736 3623056 BCB04_000053 [N-]=[N+]=NCC(=O)N1CCC2(CC1)N(CNC2=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C10 compound treatment 173240.0 4010.0 0.27 179880.0 8360.0 0.62 0.6331 0.9318 3623057 BCB04_000054 CCCCCCC1=C[C@@H]2[C@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C11 mock treatment 159120.0 -10100.0 -0.69 163320.0 -8200.0 -0.61 -0.9191 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C12 mock treatment 166320.0 -2910.0 -0.2 163880.0 -7640.0 -0.57 -0.5425 -0.9006 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C13 compound treatment 165760.0 -3470.0 -0.24 161160.0 -10400.0 -0.77 -0.7127 -0.8834 3623059 BCB04_000055 CN1CCN(CC1)C(=O)CN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C14 compound treatment 166960.0 -2270.0 -0.15 169560.0 -1960.0 -0.15 -0.2128 -0.9996 3623060 BCB04_000056 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C15 mock treatment 159520.0 -9710.0 -0.66 167280.0 -4240.0 -0.32 -0.6914 -0.9426 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C16 mock treatment 165440.0 -3790.0 -0.26 161640.0 -9880.0 -0.74 -0.7028 -0.9016 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C17 compound treatment 169200.0 -31.6 0.0 173480.0 1960.0 0.15 0.1015 0.6966 3623061 BCB04_000057 [N-]=[N+]=NCC(=O)N1CCN(CC1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C18 compound treatment 179320.0 10100.0 0.69 186880.0 15400.0 1.14 1.2946 0.9704 3623062 BCB04_000058 CCCCCCC1=C[C@H]([C@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N([C@@H](C)c3ccccc3)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C19 compound treatment 156280.0 -13000.0 -0.88 164560.0 -6960.0 -0.52 -0.9908 -0.9677 3623064 BCB04_000059 [N-]=[N+]=NCC(=O)N1CCOCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C20 compound treatment 188360.0 19100.0 1.3 184160.0 12600.0 0.94 1.5873 0.9871 3623065 BCB04_000060 CCCCCCC1=C[C@H]([C@@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N([C@@H](C)c3ccccc3)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C21 compound treatment 164400.0 -4830.0 -0.33 169120.0 -2400.0 -0.18 -0.3593 -0.9588 3623066 BCB04_000061 COc1ccc(NC(=O)CN=[N+]=[N-])cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C22 compound treatment 194160.0 24900.0 1.7 198440.0 26900.0 2.0 2.6184 0.9966 3623067 BCB04_000062 CCCCCCC1=C[C@H]([C@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C23 compound treatment 157200.0 -12000.0 -0.82 162320.0 -9200.0 -0.68 -1.0643 -0.996 3623069 BCB04_000063 COc1ccc(OC)c(NC(=O)CN=[N+]=[N-])c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 C24 compound treatment 213960.0 44700.0 3.05 218960.0 47400.0 3.53 4.6529 0.9973 3623070 BCB04_000064 CCCCCCC1=C[C@H]([C@@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D01 compound treatment 158880.0 -10400.0 -0.71 164840.0 -6680.0 -0.5 -0.8507 -0.9853 3623071 BCB04_000065 CN1C(=O)N[C@H]2[C@@H](COC(=O)c3ccc(cc3)[N+](=O)[O-])[C@]1(C)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D02 compound treatment 172120.0 2890.0 0.2 182040.0 10500.0 0.78 0.6928 0.8582 3623073 BCB04_000066 CC(C)(C)OC(=O)N[C@H]1CN(CC2=C(COC(=O)c3ccccc3)C[C@]4(Cl)C(Cl)(Cl)[C@]4(Cl)[C@@H]12)S(=O)(=O)c5ccc(Br)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D03 compound treatment 164680.0 -4550.0 -0.31 165200.0 -6320.0 -0.47 -0.5521 -0.9796 3623074 BCB04_000067 CN1C(=O)N([C@H]2[C@@H](COC(=O)c3ccc(cc3)[N+](=O)[O-])[C@]1(C)Oc4ccccc24)C(=O)CC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D04 compound treatment 213760.0 44500.0 3.04 203240.0 31700.0 2.36 3.8159 0.9923 3623076 BCB04_000068 COc1ccc(CN([C@@H](CO)[C@H]2CO2)S(=O)(=O)c3ccc(Br)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D05 compound treatment 166400.0 -2830.0 -0.19 163280.0 -8240.0 -0.61 -0.5703 -0.8868 3623078 BCB04_000069 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO)N=C5SCC(=O)N45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D06 compound treatment 176440.0 7210.0 0.49 180560.0 9040.0 0.67 0.8232 0.9881 3623080 BCB04_000070 COc1ccc(CN([C@H](CN(CCCO[Si](C(C)C)(C(C)C)C(C)C)S(=O)(=O)c2ccc(Br)cc2)[C@H]3CO3)S(=O)(=O)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D07 compound treatment 173880.0 4650.0 0.32 172360.0 838.0 0.06 0.2682 0.8304 3623082 BCB04_000071 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2COC(=O)c5ccccc5)N=C6SCC(=O)N46)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D08 compound treatment 173880.0 4650.0 0.32 184080.0 12600.0 0.93 0.885 0.8967 3623084 BCB04_000072 COc1ccc(CN([C@H](CN(CCCO[Si](C(C)C)(C(C)C)C(C)C)S(=O)(=O)c2ccc(Br)cc2)[C@@H](O)CO)S(=O)(=O)c3ccc(Br)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D09 compound treatment 159680.0 -9550.0 -0.65 166640.0 -4880.0 -0.36 -0.7174 -0.962 3623086 BCB04_000073 OC[C@@]1(Oc2ccccc2[C@@H]3[C@H]1COC(=O)c4ccccc4)N=C5SCC(=O)N35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D10 compound treatment 174720.0 5490.0 0.37 179000.0 7480.0 0.56 0.6582 0.9813 3623088 BCB04_000074 [O-][N+](=O)c1ccc(cc1)C2Sc3ccccc3C=C2C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D11 mock treatment 158960.0 -10300.0 -0.7 164040.0 -7480.0 -0.56 -0.8889 -0.9936 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D12 mock treatment 161680.0 -7550.0 -0.51 163680.0 -7840.0 -0.58 -0.7767 -0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D13 compound treatment 184080.0 14800.0 1.01 180720.0 9200.0 0.68 1.1999 0.9819 3623089 BCB04_000075 CC(C)(C)[Si](C)(C)OC[C@@H]1[C@@H]2N(C(=O)c3ccccc3)C(=S)N[C@@]1(C)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D14 compound treatment 177000.0 7770.0 0.53 170720.0 -802.0 -0.06 0.3323 0.6235 3623091 BCB04_000076 [O-][N+](=O)c1ccc(cc1)C2Oc3ccccc3C=C2C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D15 mock treatment 167760.0 -1470.0 -0.1 162400.0 -9120.0 -0.68 -0.551 -0.8029 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D16 mock treatment 161560.0 -7670.0 -0.52 167760.0 -3760.0 -0.28 -0.5678 -0.9571 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D17 compound treatment 160160.0 -9070.0 -0.62 170680.0 -842.0 -0.06 -0.4816 -0.7748 3623092 BCB04_000077 CCOC(=O)OC[C@@H]1[C@@H]2NC(=O)N(C)[C@@]1(COCc3ccc(OC)cc3)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D18 compound treatment 178520.0 9290.0 0.63 190800.0 19300.0 1.43 1.4624 0.9324 3623094 BCB04_000078 O=CC1=Cc2ccccc2OC1c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D19 compound treatment 189120.0 19900.0 1.36 186880.0 15400.0 1.14 1.7671 0.9964 3623095 BCB04_000079 COc1ccc(COC[C@]2(Oc3ccccc3[C@H]4NC(=O)N2C)[C@@H]4COC(=O)c5ccc(cc5)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D20 compound treatment 186200.0 17000.0 1.16 180480.0 8960.0 0.67 1.2895 0.9657 3623097 BCB04_000080 CCOC(=O)C1Nc2cc(OC)c(OC)cc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D21 compound treatment 171480.0 2250.0 0.15 168440.0 -3080.0 -0.23 -0.0538 -0.195 3623098 BCB04_000081 CCOC(=O)OC[C@@H]1[C@@H]2NC(=O)N(C)[C@@]1(CO)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D22 compound treatment 164040.0 -5190.0 -0.35 174400.0 2880.0 0.21 -0.0988 -0.2388 3623100 BCB04_000082 CCOC(=O)C1Oc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D23 compound treatment 166280.0 -2950.0 -0.2 171120.0 -402.0 -0.03 -0.1634 -0.8034 3623101 BCB04_000083 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2COC(=O)c5ccc(cc5)[N+](=O)[O-])N(C)C(=O)N4C(=O)CC(=O)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 D24 compound treatment 187400.0 18200.0 1.24 188160.0 16600.0 1.24 1.7515 1.0 3623103 BCB04_000084 CCOC(=O)C1Oc2ccccc2C=C1/C=N/Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E01 mock treatment 164480.0 -4750.0 -0.32 164760.0 -6760.0 -0.5 -0.5849 -0.9773 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E02 mock treatment 172920.0 3690.0 0.25 164360.0 -7160.0 -0.53 -0.1991 -0.3378 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E03 compound treatment 170000.0 768.0 0.05 174440.0 2920.0 0.22 0.1906 0.8532 3623105 BCB04_000085 [N-]=[N+]=NCC(=O)Nc1nccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E04 compound treatment 219160.0 49900.0 3.4 226720.0 55200.0 4.11 5.3119 0.9956 3623106 BCB04_000086 CCCCCCC1=C[C@H](C(O)CCCCC)n2n(C1)c(=O)n(c3ccccc3)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E05 compound treatment 168240.0 -992.0 -0.07 176840.0 5320.0 0.4 0.2321 0.578 3623108 BCB04_000087 [N-]=[N+]=NCC(=O)Nc1ccon1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E06 compound treatment 174200.0 4970.0 0.34 177520.0 6000.0 0.45 0.5552 0.9907 3623109 BCB04_000088 CCCCCC(O)C1=C[C@@H](C(C)C)n2n(C1)c(=O)n(C)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E07 compound treatment 168880.0 -352.0 -0.02 183320.0 11800.0 0.88 0.604 0.6876 3623111 BCB04_000089 [N-]=[N+]=NC[C@H](Cc1ccccc1)NC(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E08 compound treatment 171680.0 2450.0 0.17 179600.0 8080.0 0.6 0.5432 0.8705 3623113 BCB04_000090 CCCCCCC1=CCn2n([C@H]1C(O)CCCCC)c(=O)n(C)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E09 mock treatment 172120.0 2890.0 0.2 175720.0 4200.0 0.31 0.3602 0.9752 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E10 mock treatment 171400.0 2170.0 0.15 175000.0 3480.0 0.26 0.2876 0.9647 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E11 compound treatment 172160.0 2930.0 0.2 174320.0 2800.0 0.21 0.2884 0.9998 3623115 BCB04_000091 [N-]=[N+]=NC[C@@H](Cc1ccccc1)NC(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E12 compound treatment 180120.0 10900.0 0.74 185520.0 14000.0 1.04 1.2616 0.9862 3623116 BCB04_000092 CCCCCCC1=C[C@H](C(O)CCCCC)n2n(C1)c(=O)n(C)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E13 compound treatment 174120.0 4890.0 0.33 172520.0 998.0 0.07 0.2882 0.844 3189423 BCB04_000093 [N-]=[N+]=NC[C@H](Cc1ccccc1)NC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E14 compound treatment 200360.0 31100.0 2.12 200160.0 28600.0 2.13 3.0078 1.0 3623067 BCB04_000094 CCCCCCC1=C[C@H]([C@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E15 compound treatment 213040.0 43800.0 2.99 216880.0 45400.0 3.38 4.499 0.9981 3623118 BCB04_000095 CC(C)(C)OC(=O)N/C(=N/C(=O)OC(C)(C)C)/NCCN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E16 compound treatment 223800.0 54600.0 3.72 228440.0 56900.0 4.24 5.6261 0.9979 3623070 BCB04_000096 CCCCCCC1=C[C@H]([C@@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E17 mock treatment 173840.0 4610.0 0.31 172480.0 958.0 0.07 0.2726 0.8461 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E18 mock treatment 166160.0 -3070.0 -0.21 170240.0 -1280.0 -0.1 -0.2155 -0.9366 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E19 compound treatment 199880.0 30600.0 2.09 202280.0 30800.0 2.29 3.0962 0.999 3623120 BCB04_000097 CC(C)(C)OC(=O)N/C(=N/C(=O)OC(C)(C)C)/NCCCN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E20 compound treatment 183200.0 14000.0 0.95 184600.0 13100.0 0.97 1.3617 0.9999 3623122 BCB04_000098 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cc(F)cc(Br)c3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E21 compound treatment 167000.0 -2230.0 -0.15 170360.0 -1160.0 -0.09 -0.1687 -0.9641 3623124 BCB04_000099 [N-]=[N+]=NCCCNC(=O)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E22 compound treatment 164920.0 -4310.0 -0.29 169760.0 -1760.0 -0.13 -0.3006 -0.9338 3623125 BCB04_000100 CCCCCCC1=C[C@@H]2C(CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cc(nn3C)c4sc5ccc(Cl)cc5c4C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E23 compound treatment 160920.0 -8310.0 -0.57 162800.0 -8720.0 -0.65 -0.8597 -0.9977 3623127 BCB04_000101 [N-]=[N+]=NCCNC(=O)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 E24 compound treatment 161680.0 -7550.0 -0.51 164760.0 -6760.0 -0.5 -0.7199 -0.9999 3623128 BCB04_000102 CCCCCCC1=C[C@@H]2[C@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F01 mock treatment 167920.0 -1310.0 -0.09 165800.0 -5720.0 -0.43 -0.3644 -0.8373 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F02 mock treatment 167760.0 -1470.0 -0.1 166680.0 -4840.0 -0.36 -0.3258 -0.8708 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F03 compound treatment 166520.0 -2710.0 -0.18 164480.0 -7040.0 -0.52 -0.5013 -0.9021 3623130 BCB04_000103 OC[C@@H]1[C@@H]2N3C(=O)CSC3=N[C@@]1(CO)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F04 compound treatment 171600.0 2370.0 0.16 176640.0 5120.0 0.38 0.3835 0.927 3623132 BCB04_000104 CCOC(=O)C1Oc2ccc(OC)cc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F05 compound treatment 172600.0 3370.0 0.23 176360.0 4840.0 0.36 0.417 0.9764 3623133 BCB04_000105 OC[C@@H]1[C@@H]2N3Cc4ccccc4CSC3=N[C@@]1(CO)Oc5ccccc25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F06 compound treatment 173760.0 4530.0 0.31 195080.0 23600.0 1.75 1.4581 0.819 3623135 BCB04_000106 O=CC1=Cc2ccccc2NC1c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F07 compound treatment 171520.0 2290.0 0.16 181960.0 10400.0 0.78 0.6597 0.8325 3623136 BCB04_000107 OC[C@@H]1[C@@H]2N3CCCSC3=N[C@@]1(CO)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F08 compound treatment 215840.0 46600.0 3.18 211200.0 39700.0 2.95 4.3351 0.9993 3623138 BCB04_000108 [O-][N+](=O)c1ccc(cc1)C2Sc3ccccc3C=C2/C=N/Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F09 mock treatment 169480.0 248.0 0.02 173360.0 1840.0 0.14 0.1087 0.7886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F10 mock treatment 169600.0 368.0 0.03 178960.0 7440.0 0.55 0.4092 0.7384 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F11 compound treatment 190120.0 20900.0 1.42 190480.0 19000.0 1.41 2.0047 1.0 3623140 BCB04_000109 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO)N=C5Sc6ccc(cc6C(=O)N45)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F12 compound treatment 193600.0 24400.0 1.66 194400.0 22900.0 1.7 2.3788 0.9999 3623142 BCB04_000110 COc1cc2NC(C(=Cc2cc1OC)C=O)c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F13 compound treatment 180760.0 11500.0 0.79 189200.0 17700.0 1.32 1.4861 0.9697 3623143 BCB04_000111 CC(C)(C)OC(=O)NC(CN(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccc(Br)cc2)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F14 compound treatment 213280.0 44000.0 3.0 207440.0 35900.0 2.67 4.0138 0.9983 3623144 BCB04_000112 CCOC(=O)C1Oc2ccc3ccccc3c2C=C1/C=N/Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F15 compound treatment 186840.0 17600.0 1.2 192560.0 21000.0 1.57 1.9561 0.9914 3623146 BCB04_000113 CC(C)(C)OC(=O)NCC#CCN(C(COC(=O)c1ccccc1)C=C)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F16 compound treatment 194200.0 25000.0 1.7 201880.0 30400.0 2.26 2.8014 0.9903 3623147 BCB04_000114 O=CC1=Cc2ccccc2SC1c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F17 mock treatment 172520.0 3290.0 0.22 176160.0 4640.0 0.35 0.4026 0.9782 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F18 mock treatment 170600.0 1370.0 0.09 174040.0 2520.0 0.19 0.1985 0.9481 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F19 compound treatment 166360.0 -2870.0 -0.2 172240.0 718.0 0.05 -0.1006 -0.4959 3623148 BCB04_000115 CC(C)(C)OC(=O)NCC#CCO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F20 compound treatment 186920.0 17700.0 1.21 193480.0 22000.0 1.63 2.0083 0.9888 3623149 BCB04_000116 CCCCC1Nc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F21 compound treatment 166840.0 -2390.0 -0.16 169160.0 -2360.0 -0.18 -0.2396 -0.9993 3623150 BCB04_000117 CC(C)(C)OC(=O)N(CC#CCO)S(=O)(=O)c1ccccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F22 compound treatment 182160.0 12900.0 0.88 182280.0 10800.0 0.8 1.1894 0.9989 3623151 BCB04_000118 O=CC1=Cc2ccccc2OC1c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F23 compound treatment 178680.0 9450.0 0.64 180200.0 8680.0 0.65 0.9122 1.0 3623152 BCB04_000119 Brc1ccc(cc1)S(=O)(=O)NCC#CCOC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 F24 compound treatment 160520.0 -8710.0 -0.59 174720.0 3200.0 0.24 -0.2517 -0.3933 3623153 BCB04_000120 CCCCC1Sc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G01 compound treatment 181840.0 12600.0 0.86 182560.0 11000.0 0.82 1.1887 0.9997 3623154 BCB04_000121 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCCN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G02 compound treatment 181440.0 12200.0 0.83 181160.0 9640.0 0.72 1.0958 0.9973 3623156 BCB04_000122 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G03 mock treatment 174520.0 5290.0 0.36 173600.0 2080.0 0.15 0.3643 0.9286 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G04 mock treatment 176600.0 7370.0 0.5 176280.0 4760.0 0.35 0.6056 0.9854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G05 compound treatment 179520.0 10300.0 0.7 184960.0 13400.0 1.0 1.2032 0.9849 3623157 BCB04_000123 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G06 compound treatment 264600.0 95400.0 6.5 272240.0 101000.0 7.5 9.8981 0.9975 3623159 BCB04_000124 CCCCCCC1=C[C@H]([C@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C2=O)c3cc(F)ccc3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G07 compound treatment 179600.0 10400.0 0.71 180640.0 9120.0 0.68 0.9797 0.9998 3623161 BCB04_000125 CC(C)[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)NCCN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G08 compound treatment 185640.0 16400.0 1.12 189840.0 18300.0 1.36 1.7551 0.9952 3623163 BCB04_000126 CCCCCCC1=C[C@H]([C@@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C2=O)c3cc(F)ccc3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G09 compound treatment 179440.0 10200.0 0.7 181080.0 9560.0 0.71 0.9952 0.9999 3623164 BCB04_000127 Cc1ccc(cc1)S(=O)(=O)N2CCC[C@H]2CN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G10 compound treatment 197280.0 28000.0 1.91 200840.0 29300.0 2.18 2.8951 0.9978 3623166 BCB04_000128 CCCCCCC1=C[C@H]([C@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C2=O)c3cc(Cl)ccc3OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G11 compound treatment 176640.0 7410.0 0.51 184040.0 12500.0 0.93 1.016 0.9586 3623168 BCB04_000129 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)CN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G12 compound treatment 184280.0 15000.0 1.03 179280.0 7760.0 0.58 1.1338 0.963 3623116 BCB04_000130 CCCCCCC1=C[C@H](C(O)CCCCC)n2n(C1)c(=O)n(C)c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G13 compound treatment 179560.0 10300.0 0.7 181120.0 9600.0 0.71 1.0031 1.0 3623170 BCB04_000131 COC(=O)[C@@H](NC(=O)CN=[N+]=[N-])c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G14 compound treatment 439120.0 270000.0 18.4 441280.0 270000.0 20.08 27.2076 0.9991 3623172 BCB04_000132 CCCCCCC1=C[C@H]([C@H](O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(Cc3ccccc3)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G15 compound treatment 177840.0 8610.0 0.59 185280.0 13800.0 1.02 1.1391 0.9651 3623174 BCB04_000133 CCOC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN=[N+]=[N-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G16 compound treatment 203760.0 34500.0 2.35 205960.0 34400.0 2.56 3.477 0.9991 3623176 BCB04_000134 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G17 compound treatment 201280.0 32000.0 2.18 206320.0 34800.0 2.59 3.3764 0.9964 3623178 BCB04_000135 COC(=O)[C@H](O)[C@H](N=[N+]=[N-])c1ccc(OC)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G18 compound treatment 320720.0 151000.0 10.33 312200.0 141000.0 10.47 14.7066 1.0 3623180 BCB04_000136 CCCCCCC1=C[C@H](C(O)CCCCC)[C@H]2[C@@H](C1)C(=O)N(C2=O)c3ccc(F)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G19 mock treatment 174080.0 4850.0 0.33 180120.0 8600.0 0.64 0.6862 0.9528 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G20 mock treatment 174280.0 5050.0 0.34 174120.0 2600.0 0.19 0.3801 0.9628 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G21 compound treatment 168160.0 -1070.0 -0.07 173960.0 2440.0 0.18 0.0767 0.3919 3623182 BCB04_000137 COC(=O)c1cn(CC(=O)Nc2nc3ccccc3s2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G22 compound treatment 180280.0 11000.0 0.75 182920.0 11400.0 0.85 1.1325 0.9982 3623183 BCB04_000138 CCCCCCC1=C[C@@H]2C(CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cccc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G23 compound treatment 172240.0 3010.0 0.21 168800.0 -2720.0 -0.2 0.0018 0.0062 3623185 BCB04_000139 O=C1COC[C@H](N1CC#C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 G24 compound treatment 161360.0 -7870.0 -0.54 166000.0 -5520.0 -0.41 -0.6701 -0.9913 3623187 BCB04_000140 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cccc(Cl)c3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H01 compound treatment 169600.0 368.0 0.03 170680.0 -842.0 -0.06 -0.0265 -0.3932 3623189 BCB04_000141 CC(C)(C)OC(=O)N(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H02 compound treatment 164400.0 -4830.0 -0.33 181640.0 10100.0 0.75 0.2996 0.3645 3623190 BCB04_000142 CCOC(=O)C1Oc2cccc(C)c2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H03 mock treatment 173040.0 3810.0 0.26 172960.0 1440.0 0.11 0.2593 0.9232 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H04 mock treatment 172400.0 3170.0 0.22 177960.0 6440.0 0.48 0.4916 0.9352 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H05 compound treatment 180240.0 11000.0 0.75 182800.0 11300.0 0.84 1.1242 0.9984 3623191 BCB04_000143 Brc1ccc(cc1)S(=O)(=O)NC(COC(=O)c2ccccc2)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H06 compound treatment 219200.0 50000.0 3.41 225040.0 53500.0 3.98 5.2254 0.997 3623192 BCB04_000144 CCOC(=O)C1Nc2cc3OCOc3cc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H07 compound treatment 176360.0 7130.0 0.49 178400.0 6880.0 0.51 0.7056 0.9997 3623193 BCB04_000145 CC(C)(C)OC(=O)N(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H08 compound treatment 208680.0 39400.0 2.69 212120.0 40600.0 3.02 4.0383 0.9983 3623194 BCB04_000146 CCCC1Oc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H09 compound treatment 174640.0 5410.0 0.37 185760.0 14200.0 1.06 1.0101 0.9002 3623195 BCB04_000147 CC(C)(C)OC(=O)NS(=O)(=O)c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H10 compound treatment 194560.0 25300.0 1.73 209720.0 38200.0 2.84 3.2313 0.9714 3623196 BCB04_000148 CCCC1Sc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H11 compound treatment 188200.0 19000.0 1.29 188520.0 17000.0 1.27 1.809 0.9999 3623197 BCB04_000149 CC(C)(C)OC(=O)NC(CN(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccccc2[N+](=O)[O-])C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H12 compound treatment 200800.0 31600.0 2.15 210440.0 38900.0 2.9 3.57 0.9893 3623198 BCB04_000150 CCCCC1Oc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H13 compound treatment 201480.0 32200.0 2.2 200040.0 28500.0 2.12 3.0555 0.9998 3623199 BCB04_000151 CC(C)(C)OC(=O)NCC#CCN(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H14 compound treatment 219920.0 50700.0 3.46 222680.0 51200.0 3.81 5.1359 0.9988 3623200 BCB04_000152 CCOC(=O)C1Oc2cc(OC)ccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H15 compound treatment 186800.0 17600.0 1.2 185760.0 14200.0 1.06 1.5963 0.9981 3623201 BCB04_000153 CC(C)(C)OC(=O)N(CC#CCN(C(COC(=O)c1ccccc1)C=C)S(=O)(=O)c2ccc(Br)cc2)S(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H16 compound treatment 217080.0 47800.0 3.26 211000.0 39500.0 2.94 4.3843 0.9986 3623202 BCB04_000154 CCOC(=O)C1Oc2c(OC)cccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H17 compound treatment 180080.0 10800.0 0.74 179160.0 7640.0 0.57 0.925 0.9916 3623203 BCB04_000155 CC(C)(C)OC(=O)NC1CN(CC(=C1)C(=C)COC(=O)c2ccccc2)S(=O)(=O)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H18 compound treatment 189280.0 20000.0 1.37 207080.0 35600.0 2.65 2.8379 0.9527 3623204 BCB04_000156 CCOC(=O)C1Sc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H19 mock treatment 170800.0 1570.0 0.11 174440.0 2920.0 0.22 0.2292 0.9467 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H20 mock treatment 166200.0 -3030.0 -0.21 172600.0 1080.0 0.08 -0.0894 -0.4032 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H21 compound treatment 177200.0 7970.0 0.54 177160.0 5640.0 0.42 0.6809 0.9919 3623205 BCB04_000157 CC(C)(C)OC(=O)NCC#CCN(CC#CCN([C@H](COC(=O)c1ccccc1)C=C)S(=O)(=O)c2ccc(Br)cc2)S(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H22 compound treatment 170200.0 968.0 0.07 170160.0 -1360.0 -0.1 -0.025 -0.2065 3623207 BCB04_000158 O=CC1=Cc2ccccc2OC1c3ccc4ccccc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H23 compound treatment 167840.0 -1390.0 -0.09 176200.0 4680.0 0.35 0.1791 0.4963 3623208 BCB04_000159 CC(C)(C)OC(=O)N(CC#CCN(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccc(Br)cc2)S(=O)(=O)c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 H24 compound treatment 167400.0 -1830.0 -0.12 181960.0 10400.0 0.78 0.461 0.5859 3623209 BCB04_000160 [O-][N+](=O)c1ccc(cc1)C2Oc3ccccc3C=C2/C=N/Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I01 compound treatment 170280.0 1050.0 0.07 179000.0 7480.0 0.56 0.4441 0.7914 3623211 BCB04_000161 O=C(Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)N4CCC5(CC4)N(CNC5=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I02 compound treatment 168040.0 -1190.0 -0.08 173000.0 1480.0 0.11 0.0204 0.1488 3623213 BCB04_000162 CCCCCCC1=C[C@@H]2[C@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cccc(Cl)c3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I03 compound treatment 169440.0 208.0 0.01 175280.0 3760.0 0.28 0.2078 0.7421 3623214 BCB04_000163 CN1CCN(CC1)C(=O)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I04 compound treatment 354800.0 186000.0 12.65 358840.0 187000.0 13.94 18.8041 0.9988 3623216 BCB04_000164 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3ccc(Br)c(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I05 mock treatment 174200.0 4970.0 0.34 176680.0 5160.0 0.38 0.511 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I06 mock treatment 176520.0 7290.0 0.5 172520.0 998.0 0.07 0.4039 0.8039 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I07 compound treatment 177840.0 8610.0 0.59 179720.0 8200.0 0.61 0.8465 0.9998 3623218 BCB04_000165 O=C(Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)N4CCN(CC4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I08 compound treatment 181440.0 12200.0 0.83 184120.0 12600.0 0.94 1.2516 0.9982 3623220 BCB04_000166 CCCCCCC1=C[C@@H]2[C@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3ccc(Br)c(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I09 compound treatment 171200.0 1970.0 0.13 182200.0 10700.0 0.79 0.6569 0.815 3623221 BCB04_000167 O=C(Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I10 compound treatment 200440.0 31200.0 2.13 205360.0 33800.0 2.52 3.2853 0.9965 3623223 BCB04_000168 CCCCCCC1=C[C@@H]2[C@@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cccc(Cl)n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I11 compound treatment 177080.0 7850.0 0.54 179560.0 8040.0 0.6 0.8014 0.9984 3623225 BCB04_000169 COc1ccc(NC(=O)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I12 compound treatment 196360.0 27100.0 1.85 190080.0 18600.0 1.38 2.2845 0.9897 3623227 BCB04_000170 CCCCCCC1=C[C@@H]2[C@H](CCCCC)OC(=O)[C@@H]2[C@@H](C1)C(=O)Nc3cccc(Cl)n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I13 compound treatment 179160.0 9930.0 0.68 178360.0 6840.0 0.51 0.8385 0.9901 3623228 BCB04_000171 COc1ccc(OC)c(NC(=O)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I14 compound treatment 176280.0 7050.0 0.48 174720.0 3200.0 0.24 0.5081 0.9475 2108247 BCB04_000172 CCOC(=O)[C@@H]1[C@@H]2NC(=O)N[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I15 compound treatment 185600.0 16400.0 1.12 190920.0 19400.0 1.44 1.81 0.9919 3623230 BCB04_000173 O=C(Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)Nc4nccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I16 compound treatment 179080.0 9850.0 0.67 180200.0 8680.0 0.65 0.9315 0.9998 3623232 BCB04_000174 CCOC(=O)[C@@H]1[C@@H]2NC(=O)N(CC=C)[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I17 compound treatment 173560.0 4330.0 0.3 175920.0 4400.0 0.33 0.4401 0.9987 3623234 BCB04_000175 O=C(Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)Nc4ccon4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I18 compound treatment 187160.0 17900.0 1.22 185280.0 13800.0 1.02 1.5884 0.9961 3623236 BCB04_000176 CCOC(=O)[C@@H]1[C@@H]2NC(=S)N[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I19 compound treatment 171520.0 2290.0 0.16 173120.0 1600.0 0.12 0.1944 0.991 3623237 BCB04_000177 O=C(N[C@@H](Cc1ccccc1)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I20 compound treatment 170360.0 1130.0 0.08 174160.0 2640.0 0.2 0.1932 0.9163 3623239 BCB04_000178 CCOC(=O)[C@@H]1[C@@H]2NC(=S)N(CC=C)[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I21 mock treatment 167920.0 -1310.0 -0.09 167960.0 -3560.0 -0.27 -0.2507 -0.896 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I22 mock treatment 166680.0 -2550.0 -0.17 163760.0 -7760.0 -0.58 -0.5315 -0.881 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I23 compound treatment 162360.0 -6870.0 -0.47 175920.0 4400.0 0.33 -0.0998 -0.1746 3623241 BCB04_000179 O=C(N[C@H](Cc1ccccc1)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2)Nc5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 I24 compound treatment 169440.0 208.0 0.01 174320.0 2800.0 0.21 0.1573 0.7536 3623242 BCB04_000180 C[C@]1(Oc2ccccc2[C@H]3NC(=S)N1CC=C)[C@@H]3CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J01 compound treatment 178960.0 9730.0 0.66 175200.0 3680.0 0.27 0.6626 0.9234 3623244 BCB04_000181 CC(C)(C)OC(=O)NCC#CCOC(=O)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J02 compound treatment 212880.0 43600.0 2.98 218160.0 46600.0 3.47 4.5587 0.9971 3623245 BCB04_000182 N#Cc1ccc(cc1)C2Oc3ccccc3C=C2/C=N/Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J03 compound treatment 174360.0 5130.0 0.35 174520.0 3000.0 0.22 0.405 0.9765 3623247 BCB04_000183 CC(C)(C)OC(=O)NC(COC(=O)c1ccccc1)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J04 compound treatment 233400.0 64200.0 4.37 228560.0 57000.0 4.25 6.0952 0.9999 3623248 BCB04_000184 Clc1ccc(cc1)C2Nc3ccccc3C=C2C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J05 mock treatment 172840.0 3610.0 0.25 176120.0 4600.0 0.34 0.416 0.9869 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J06 mock treatment 171640.0 2410.0 0.16 176160.0 4640.0 0.35 0.3602 0.9423 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J07 compound treatment 194440.0 25200.0 1.72 197480.0 26000.0 1.93 2.5814 0.9983 3623249 BCB04_000185 CC(C)(C)OC(=O)N[C@@H](CN(CC#CCN([C@H](COC(=O)c1ccccc1)C=C)S(=O)(=O)c2ccc(Br)cc2)S(=O)(=O)c3ccccc3[N+](=O)[O-])C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J08 compound treatment 217520.0 48300.0 3.29 221320.0 49800.0 3.71 4.9487 0.9983 3623251 BCB04_000186 Clc1ccc(cc1)C2Nc3ccccc3C=C2/C=N/Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J09 compound treatment 185480.0 16200.0 1.11 190040.0 18500.0 1.38 1.7579 0.9941 3623253 BCB04_000187 CC(C)(C)OC(=O)NC(CN(CC#CCN(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccc(Br)cc2)S(=O)(=O)c3ccccc3[N+](=O)[O-])C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J10 compound treatment 200080.0 30800.0 2.1 206360.0 34800.0 2.59 3.3206 0.9946 3623254 BCB04_000188 CCOC(=O)C1Nc2cc(F)ccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J11 compound treatment 177240.0 8010.0 0.55 177800.0 6280.0 0.47 0.7165 0.997 3623255 BCB04_000189 [O-][N+](=O)c1ccccc1S(=O)(=O)NCC#CCN(CC#CCOC(=O)c2ccccc2)S(=O)(=O)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J12 compound treatment 168320.0 -912.0 -0.06 181200.0 9680.0 0.72 0.4654 0.6437 3623256 BCB04_000190 O=CC1=Cc2ccccc2SC1c3ccc(C#N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J13 compound treatment 184280.0 15000.0 1.03 188000.0 16500.0 1.23 1.5927 0.9961 3623257 BCB04_000191 CC(C)(C)OC(=O)N[C@H](CN(CC#CCN([C@H](COC(=O)c1ccccc1)C=C)S(=O)(=O)c2ccc(Br)cc2)S(=O)(=O)c3ccccc3[N+](=O)[O-])C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J14 compound treatment 188560.0 19300.0 1.32 189240.0 17700.0 1.32 1.8643 1.0 3623258 BCB04_000192 Brc1ccc(cc1)C2Oc3ccccc3C=C2C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J15 compound treatment 186520.0 17300.0 1.18 186640.0 15100.0 1.13 1.6291 0.9997 3623259 BCB04_000193 CC(C)(C)OC(=O)N[C@H](CN([C@H](COC(=O)c1ccccc1)C=C)S(=O)(=O)c2ccc(Br)cc2)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J16 compound treatment 206120.0 36900.0 2.51 203360.0 31800.0 2.37 3.4539 0.9996 3623261 BCB04_000194 CCOC(=O)C1Oc2ccc(OC)cc2C=C1/C=N/Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J17 compound treatment 214880.0 45600.0 3.11 201960.0 30400.0 2.27 3.8025 0.9878 3623263 BCB04_000195 CC(C)(C)OC(=O)N[C@@H]1CN([C@H](COC(=O)c2ccccc2)C=C1)S(=O)(=O)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J18 compound treatment 179280.0 10000.0 0.69 184320.0 12800.0 0.95 1.158 0.9869 3623265 BCB04_000196 CCOC(=O)C1Nc2cc(Cl)ccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J19 compound treatment 187120.0 17900.0 1.22 191280.0 19800.0 1.47 1.9022 0.9957 3623266 BCB04_000197 CC(C)(C)OC(=O)N[C@H]1CN(CC(=C1)C2=C[C@@H](COC(=O)c3ccccc3)N(C2)S(=O)(=O)c4ccc(Br)cc4)S(=O)(=O)c5ccccc5[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J20 compound treatment 172960.0 3730.0 0.25 185800.0 14300.0 1.06 0.9312 0.8522 3623268 BCB04_000198 CCOC(=O)C1Oc2c(F)cccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J21 mock treatment 168440.0 -792.0 -0.05 168440.0 -3080.0 -0.23 -0.2003 -0.8503 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J22 mock treatment 166040.0 -3190.0 -0.22 166840.0 -4680.0 -0.35 -0.4003 -0.9743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J23 compound treatment 167960.0 -1270.0 -0.09 167760.0 -3760.0 -0.28 -0.2593 -0.8846 3623269 BCB04_000199 CC(C)(C)OC(=O)N[C@@H]1CN(CC(=C1)C2=C[C@@H](COC(=O)c3ccccc3)N(C2)S(=O)(=O)c4ccc(Br)cc4)S(=O)(=O)c5ccccc5[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 J24 compound treatment 165840.0 -3390.0 -0.23 166600.0 -4920.0 -0.37 -0.4225 -0.9754 3623270 BCB04_000200 CCCC1Nc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K01 compound treatment 171480.0 2250.0 0.15 176400.0 4880.0 0.36 0.3651 0.9265 3623271 BCB04_000201 O=C(N[C@@H](Cc1ccccc1)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K02 compound treatment 173800.0 4570.0 0.31 179120.0 7600.0 0.57 0.6201 0.9605 3623273 BCB04_000202 CCOC(=O)[C@@H]1[C@@H]2NC(=O)N[C@@]1(COCc3ccc(OC)cc3)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K03 compound treatment 171600.0 2370.0 0.16 181520.0 10000.0 0.74 0.6404 0.841 3623275 BCB04_000203 O=C(NCCCn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K04 compound treatment 202760.0 33500.0 2.29 195760.0 24200.0 1.8 2.892 0.9931 3623277 BCB04_000204 CCOC(=O)[C@@H]1[C@@H]2NC(=S)N[C@@]1(COCc3ccc(OC)cc3)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K05 compound treatment 176400.0 7170.0 0.49 177120.0 5600.0 0.42 0.6402 0.9968 3623279 BCB04_000205 O=C(NCCn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K06 compound treatment 167560.0 -1670.0 -0.11 171040.0 -482.0 -0.04 -0.1059 -0.8867 3623281 BCB04_000206 COc1ccc(COC[C@]2(Oc3ccccc3[C@H]4NC(=O)N2CC=C)[C@@H]4CO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K07 mock treatment 173720.0 4490.0 0.31 182040.0 10500.0 0.78 0.7699 0.916 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K08 mock treatment 176080.0 6850.0 0.47 182120.0 10600.0 0.79 0.8879 0.9687 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K09 compound treatment 177120.0 7890.0 0.54 183240.0 11700.0 0.87 0.997 0.973 3623283 BCB04_000207 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCCn3cc(CN4[C@@H](COCC4=O)c5ccccc5)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K10 compound treatment 181960.0 12700.0 0.87 189080.0 17600.0 1.31 1.5377 0.9802 3623285 BCB04_000208 COc1ccc(COC[C@]2(NC(=O)N[C@H]3[C@H]2CO)Oc4ccccc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K11 compound treatment 179760.0 10500.0 0.72 185080.0 13600.0 1.01 1.2211 0.9861 3623287 BCB04_000209 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCn3cc(CN4[C@@H](COCC4=O)c5ccccc5)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K12 compound treatment 181680.0 12400.0 0.85 181360.0 9840.0 0.73 1.1179 0.9973 3623289 BCB04_000210 C[C@]1(NC(=S)N[C@H]2[C@H]1CO)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K13 compound treatment 176280.0 7050.0 0.48 177440.0 5920.0 0.44 0.6513 0.9991 3623291 BCB04_000211 CC(C)[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)NCCn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K14 compound treatment 213280.0 44000.0 3.0 198640.0 27100.0 2.02 3.5507 0.9813 3623293 BCB04_000212 CC(C)(C)[Si](C)(C)OC[C@@H]1[C@@H]2NC(=S)N[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K15 mock treatment 173840.0 4610.0 0.31 175680.0 4160.0 0.31 0.441 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K16 mock treatment 178480.0 9250.0 0.63 170760.0 -762.0 -0.06 0.4058 0.6409 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K17 compound treatment 182480.0 13200.0 0.9 177520.0 6000.0 0.45 0.9544 0.9472 3623295 BCB04_000213 Cc1ccc(cc1)S(=O)(=O)N2CCC[C@H]2Cn3cc(CN4[C@@H](COCC4=O)c5ccccc5)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K18 compound treatment 172680.0 3450.0 0.24 172120.0 598.0 0.04 0.1977 0.8263 3623297 BCB04_000214 CC(C)(C)[Si](C)(C)OC[C@@H]1[C@@H]2N3Cc4ccccc4CSC3=N[C@@]1(C)Oc5ccccc25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K19 compound treatment 167880.0 -1350.0 -0.09 173040.0 1520.0 0.11 0.0147 0.1011 3623299 BCB04_000215 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)Cn2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K20 compound treatment 187560.0 18300.0 1.25 184720.0 13200.0 0.98 1.5782 0.9929 3623301 BCB04_000216 COc1ccc(COC[C@]2(NC(=S)N[C@H]3[C@H]2CO)Oc4ccccc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K21 compound treatment 168040.0 -1190.0 -0.08 169920.0 -1600.0 -0.12 -0.1417 -0.9825 3623303 BCB04_000217 COC(=O)[C@@H](NC(=O)Cn1cc(CN2[C@@H](COCC2=O)c3ccccc3)nn1)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K22 compound treatment 165520.0 -3710.0 -0.25 172720.0 1200.0 0.09 -0.1159 -0.4319 3623305 BCB04_000218 C[C@]1(NC(=O)N[C@H]2[C@H]1CO)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K23 mock treatment 161880.0 -7350.0 -0.5 165240.0 -6280.0 -0.47 -0.685 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 K24 mock treatment 159240.0 -9990.0 -0.68 158720.0 -12800.0 -0.95 -1.1554 -0.9865 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L01 compound treatment 166160.0 -3070.0 -0.21 165320.0 -6200.0 -0.46 -0.4745 -0.9361 3616022 BCB04_000219 CC(C)(C)OC(=O)NC(CO)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L02 compound treatment 178440.0 9210.0 0.63 187960.0 16400.0 1.22 1.309 0.9519 3623307 BCB04_000220 CCOC(=O)C1Nc2ccccc2C=C1C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L03 compound treatment 184040.0 14800.0 1.01 181520.0 10000.0 0.74 1.2401 0.9887 3623308 BCB04_000221 [O-][N+](=O)c1ccccc1S(=O)(=O)NCC#CCN(C(COC(=O)c2ccccc2)C=C)S(=O)(=O)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L04 compound treatment 172840.0 3610.0 0.25 173200.0 1680.0 0.12 0.2623 0.9506 3623309 BCB04_000222 CC(CN1CCCC1)C(=O)c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L05 compound treatment 204680.0 35400.0 2.42 212400.0 40900.0 3.04 3.8602 0.9935 3623310 BCB04_000223 CC(C)(C)OC(=O)NCC(=C)C1=CC(COC(=O)c2ccccc2)N(C1)S(=O)(=O)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L06 compound treatment 173240.0 4010.0 0.27 180840.0 9320.0 0.69 0.6836 0.9171 3623311 BCB04_000224 Cc1ccccc1n2c(Cn3cnc4c(N)ncnc34)nc5cccc(C)c5c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L07 mock treatment 171280.0 2050.0 0.14 174800.0 3280.0 0.24 0.2713 0.965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L08 mock treatment 171080.0 1850.0 0.13 180600.0 9080.0 0.68 0.5669 0.8248 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L09 compound treatment 253680.0 84400.0 5.76 258400.0 86900.0 6.47 8.6433 0.9983 3623312 BCB04_000225 CC(C)(C)OC(=O)N[C@H]1CN(CC2=C(COC(=O)c3ccccc3)C[C@H]4[C@@H]([C@H]12)C(=O)c5ccccc5C4=O)S(=O)(=O)c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L10 compound treatment 175680.0 6450.0 0.44 183680.0 12200.0 0.9 0.9507 0.945 3623314 BCB04_000226 Cc1ccccc1Oc2cccc3c(=O)cc([nH]c23)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L11 compound treatment 220720.0 51500.0 3.51 224680.0 53200.0 3.96 5.2798 0.9982 3623315 BCB04_000227 CC(C)(C)OC(=O)NC1CC=C(CN(C1)S(=O)(=O)c2ccc(Br)cc2)C(=C)COC(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L12 mock treatment 178080.0 8850.0 0.6 175960.0 4440.0 0.33 0.6601 0.9598 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L13 compound treatment 189360.0 20100.0 1.37 184560.0 13000.0 0.97 1.6565 0.9856 3623316 BCB04_000228 CC(C)(C)OC(=O)NC(CC=C)CN(CC#CCOC(=O)c1ccccc1)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L14 mock treatment 172200.0 2970.0 0.2 173040.0 1520.0 0.11 0.223 0.9621 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L15 mock treatment 168800.0 -432.0 -0.03 178920.0 7400.0 0.55 0.3685 0.6684 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L16 mock treatment 176120.0 6890.0 0.47 174000.0 2480.0 0.18 0.4625 0.9167 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L17 compound treatment 194560.0 25300.0 1.73 200280.0 28800.0 2.14 2.7345 0.9943 3623317 BCB04_000229 CC(C)(C)OC(=O)N[C@H]1CN(CC2=C(COC(=O)c3ccccc3)C[C@@H]4[C@H]([C@@H]12)C(=O)c5ccccc5C4=O)S(=O)(=O)c6ccc(Br)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L18 mock treatment 170960.0 1730.0 0.12 174000.0 2480.0 0.18 0.2137 0.9766 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L19 compound treatment 191200.0 22000.0 1.5 190840.0 19300.0 1.44 2.0757 0.9998 3623318 BCB04_000230 CC(C)(C)OC(=O)NCC1=CC(COC(=O)c2ccccc2)N(CC1=C)S(=O)(=O)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L20 mock treatment 168600.0 -632.0 -0.04 170160.0 -1360.0 -0.1 -0.1021 -0.9273 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L21 compound treatment 202800.0 33600.0 2.29 199240.0 27700.0 2.06 3.077 0.9987 3623319 BCB04_000231 COc1ccc(CN(C2=CCC3(C#N)C(=O)C=CC(=O)C3(C2)C=N)S(=O)(=O)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L22 mock treatment 161200.0 -8030.0 -0.55 166240.0 -5280.0 -0.39 -0.6652 -0.9868 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L23 mock treatment 158520.0 -10700.0 -0.73 159960.0 -11600.0 -0.86 -1.1249 -0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 L24 mock treatment 156640.0 -12600.0 -0.86 154800.0 -16700.0 -1.24 -1.487 -0.9836 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M01 compound treatment 168560.0 -672.0 -0.05 170240.0 -1280.0 -0.1 -0.0998 -0.9434 3623320 BCB04_000232 CCOC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)Cn3cc(CN4[C@@H](COCC4=O)c5ccccc5)nn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M02 compound treatment 184920.0 15700.0 1.07 192600.0 21100.0 1.57 1.8656 0.9826 3623322 BCB04_000233 CC(C)(C)[Si](C)(C)OC[C@@H]1[C@@H]2NC(=O)N[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M03 compound treatment 176440.0 7210.0 0.49 183000.0 11500.0 0.85 0.9516 0.9655 3623324 BCB04_000234 COC(=O)[C@@H](O)[C@H](c1ccc(OC)cc1)n2cc(CN3[C@@H](COCC3=O)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M04 compound treatment 172640.0 3410.0 0.23 177800.0 6280.0 0.47 0.4947 0.948 3623326 BCB04_000235 CCOC(=O)[C@@H]1[C@@H]2NC(=O)N(C)[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M05 compound treatment 176720.0 7490.0 0.51 176760.0 5240.0 0.39 0.6367 0.9911 3623328 BCB04_000236 COc1ccc(C#C)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M06 compound treatment 186640.0 17400.0 1.19 183880.0 12400.0 0.92 1.4896 0.9921 3623329 BCB04_000237 C[C@@]1(Oc2ccccc2[C@@H]3[C@H]1CO)N=C4SCc5ccccc5CN34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M07 compound treatment 185440.0 16200.0 1.11 190400.0 18900.0 1.41 1.7749 0.9929 3623331 BCB04_000238 COc1ccc(cc1OC)c2cn(CC(=O)N3CCC4(CC3)N(CNC4=O)c5ccccc5)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M08 compound treatment 175840.0 6610.0 0.45 183840.0 12300.0 0.92 0.9669 0.9465 3623332 BCB04_000239 CCOC(=O)[C@@H]1[C@@H]2NC(=O)N(C)[C@@]1(COCc3ccc(OC)cc3)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M09 mock treatment 179000.0 9770.0 0.67 182680.0 11200.0 0.83 1.0582 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M10 mock treatment 179000.0 9770.0 0.67 180000.0 8480.0 0.63 0.9171 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M11 compound treatment 183040.0 13800.0 0.94 180000.0 8480.0 0.63 1.1119 0.9811 3623334 BCB04_000240 COc1ccc(cc1OC)c2cn(CC(=O)N3CCN(C)CC3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M12 compound treatment 182560.0 13300.0 0.91 189600.0 18100.0 1.35 1.594 0.9817 3623335 BCB04_000241 CC(C)(C)[Si](C)(C)OC[C@@H]1[C@@H]2N3C(=O)CSC3=N[C@@]1(C)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M13 mock treatment 176880.0 7650.0 0.52 173800.0 2280.0 0.17 0.4886 0.8911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M14 mock treatment 169880.0 648.0 0.04 180520.0 9000.0 0.67 0.5048 0.7521 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M15 compound treatment 176280.0 7050.0 0.48 188360.0 16800.0 1.25 1.226 0.9134 3623337 BCB04_000242 COc1ccc(cc1OC)c2cn(CC(=O)N3CCN(CC3)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M16 compound treatment 237000.0 67800.0 4.62 236960.0 65400.0 4.87 6.7109 0.9997 3623338 BCB04_000243 COc1ccc(COC[C@]2(NC(=O)N[C@H]3[C@H]2CO[Si](C)(C)C(C)(C)C)Oc4ccccc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M17 compound treatment 174920.0 5690.0 0.39 180200.0 8680.0 0.65 0.7309 0.9702 3623340 BCB04_000244 COc1ccc(cc1OC)c2cn(CC(=O)N3CCOCC3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M18 compound treatment 181240.0 12000.0 0.82 180880.0 9360.0 0.7 1.0714 0.9968 3623341 BCB04_000245 C[C@@]1(Oc2ccccc2[C@@H]3[C@H]1CO)N=C4SCC(=O)N34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M19 compound treatment 178520.0 9290.0 0.63 186640.0 15100.0 1.13 1.2434 0.963 3623343 BCB04_000246 COc1ccc(NC(=O)Cn2cc(nn2)c3ccc(OC)c(OC)c3)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M20 compound treatment 189040.0 19800.0 1.35 187120.0 15600.0 1.16 1.7758 0.9972 3623344 BCB04_000247 CCOC(=O)[C@@H]1[C@@H]2NC(=S)N(C)[C@@]1(COCc3ccc(OC)cc3)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M21 compound treatment 179760.0 10500.0 0.72 175560.0 4040.0 0.3 0.7201 0.9253 3623346 BCB04_000248 COc1ccc(OC)c(NC(=O)Cn2cc(nn2)c3ccc(OC)c(OC)c3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M22 compound treatment 172680.0 3450.0 0.24 172840.0 1320.0 0.1 0.2356 0.9249 3623347 BCB04_000249 CCOC(=O)[C@@H]1[C@@H]2NC(=S)N(C)[C@@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M23 compound treatment 174320.0 5090.0 0.35 173880.0 2360.0 0.18 0.3694 0.9502 3623349 BCB04_000250 COc1ccc(cc1OC)c2cn(CC(=O)Nc3nccs3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 M24 compound treatment 162360.0 -6870.0 -0.47 161720.0 -9800.0 -0.73 -0.8471 -0.9771 3623350 BCB04_000251 CN1C(=O)N[C@H]2[C@@H](CO)[C@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N01 compound treatment 202520.0 33300.0 2.27 199400.0 27900.0 2.07 3.0719 0.999 3623352 BCB04_000252 COc1ccc(CN(C2=CCC3C(C2)C(=O)c4ccccc4C3=O)S(=O)(=O)c5ccc(Br)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N02 mock treatment 171240.0 2010.0 0.14 173880.0 2360.0 0.18 0.2209 0.9925 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N03 compound treatment 173920.0 4690.0 0.32 179840.0 8320.0 0.62 0.6638 0.9527 3623353 BCB04_000253 CO[C@@](C(=O)OC[C@@H](NC(=O)OC(C)(C)C)C=C)(c1ccccc1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N04 mock treatment 172800.0 3570.0 0.24 178480.0 6960.0 0.52 0.5382 0.9407 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N05 compound treatment 175120.0 5890.0 0.4 180040.0 8520.0 0.63 0.7322 0.9757 3623355 BCB04_000254 CO[C@](C(=O)OC[C@@H](NC(=O)OC(C)(C)C)C=C)(c1ccccc1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N06 mock treatment 178560.0 9330.0 0.64 179000.0 7480.0 0.56 0.8433 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N07 compound treatment 180080.0 10800.0 0.74 183640.0 12100.0 0.9 1.1607 0.9951 3623356 BCB04_000255 CC(C)(C)OC(=O)N(CC#CCO[Si](C)(C)C(C)(C)C)S(=O)(=O)c1ccccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N08 mock treatment 176320.0 7090.0 0.48 176320.0 4800.0 0.36 0.5942 0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N09 mock treatment 179680.0 10400.0 0.71 178400.0 6880.0 0.51 0.8657 0.9869 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N10 mock treatment 179480.0 10200.0 0.7 181360.0 9840.0 0.73 1.0118 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N11 compound treatment 184240.0 15000.0 1.02 194440.0 22900.0 1.71 1.9297 0.9701 3068087 BCB04_000256 COc1cc(CN([C@@H](COC(=O)C)C=C)S(=O)(=O)c2ccc(Br)cc2)ccc1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N12 mock treatment 174120.0 4890.0 0.33 184320.0 12800.0 0.95 0.9092 0.901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N13 mock treatment 173960.0 4730.0 0.32 181800.0 10300.0 0.76 0.7689 0.9262 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N14 mock treatment 173280.0 4050.0 0.28 180920.0 9400.0 0.7 0.6898 0.9173 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N15 compound treatment 174960.0 5730.0 0.39 183840.0 12300.0 0.92 0.9244 0.9277 3068089 BCB04_000257 CC[Si](CC)(CC)OC[C@@H](C=C)N(Cc1ccc(OC(=O)C)c(OC)c1)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N16 mock treatment 173280.0 4050.0 0.28 176480.0 4960.0 0.37 0.4561 0.9898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N17 compound treatment 174880.0 5650.0 0.39 184440.0 12900.0 0.96 0.9522 0.9193 3623357 BCB04_000258 COc1ccc(CN(C(=C)C=C)S(=O)(=O)c2ccc(Br)cc2)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N18 mock treatment 170240.0 1010.0 0.07 180440.0 8920.0 0.66 0.518 0.7762 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N19 compound treatment 174360.0 5130.0 0.35 180280.0 8760.0 0.65 0.7082 0.9574 3623358 BCB04_000259 CCOC(=O)/C=C/C(CN(Cc1c(OC)cc(OC)cc1OC)S(=O)(=O)c2ccc(Br)cc2)OC(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N20 mock treatment 164600.0 -4630.0 -0.32 171800.0 278.0 0.02 -0.2086 -0.6593 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N21 compound treatment 171280.0 2050.0 0.14 174640.0 3120.0 0.23 0.2629 0.9705 3623360 BCB04_000260 COc1cc(OC)c(CN(C[C@H]2CO2)S(=O)(=O)c3ccc(Br)cc3)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N22 mock treatment 165720.0 -3510.0 -0.24 164320.0 -7200.0 -0.54 -0.5483 -0.934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N23 compound treatment 165840.0 -3390.0 -0.23 161880.0 -9640.0 -0.72 -0.6709 -0.8899 3623362 BCB04_000261 Brc1ccc(cc1)S(=O)(=O)NCC(OC(=O)c2ccccc2)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 N24 mock treatment 156720.0 -12500.0 -0.85 160760.0 -10800.0 -0.8 -1.1695 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O01 compound treatment 171800.0 2570.0 0.18 171120.0 -402.0 -0.03 0.1027 0.578 3623363 BCB04_000262 COc1ccc(cc1OC)c2cn(CC(=O)Nc3ccon3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O02 compound treatment 165240.0 -3990.0 -0.27 175120.0 3600.0 0.27 -0.0031 -0.008 3623364 BCB04_000263 CN1C(=S)N[C@H]2[C@@H](CO)[C@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O03 compound treatment 176480.0 7250.0 0.49 181640.0 10100.0 0.75 0.8819 0.9791 3623366 BCB04_000264 COc1ccc(cc1OC)c2cn(C[C@H](Cc3ccccc3)NC(=O)Nc4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O04 compound treatment 173640.0 4410.0 0.3 172920.0 1400.0 0.1 0.2861 0.8995 3623368 BCB04_000265 CN1C(=O)N[C@H]2[C@@H](CO[Si](C)(C)C(C)(C)C)[C@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O05 compound treatment 195240.0 26000.0 1.77 196640.0 25100.0 1.87 2.5757 0.9997 3623370 BCB04_000266 COc1ccc(cc1OC)c2cn(C[C@@H](Cc3ccccc3)NC(=O)Nc4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O06 compound treatment 190640.0 21400.0 1.46 192800.0 21300.0 1.58 2.1519 0.9992 3623371 BCB04_000267 CN1C(=S)N[C@H]2[C@@H](CO[Si](C)(C)C(C)(C)C)[C@]1(C)Oc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O07 compound treatment 198840.0 29600.0 2.02 195000.0 23500.0 1.75 2.663 0.9974 3623373 BCB04_000268 COc1ccc(cc1OC)c2cn(C[C@H](Cc3ccccc3)NC(=O)c4ccccc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O08 compound treatment 178400.0 9170.0 0.63 176080.0 4560.0 0.34 0.6819 0.9588 3623375 BCB04_000269 CN1C(=O)N([C@H]2[C@@H](CO[Si](C)(C)C(C)(C)C)[C@]1(C)Oc3ccccc23)C(=O)CC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O09 compound treatment 171160.0 1930.0 0.13 178280.0 6760.0 0.5 0.4486 0.8629 3623377 BCB04_000270 COc1ccc(cc1OC)c2cn(CCCNC(=O)Nc3ccccc3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O10 compound treatment 173600.0 4370.0 0.3 176640.0 5120.0 0.38 0.48 0.9926 3623378 BCB04_000271 CN1C(=O)N[C@H]2[C@@H](COC(=O)c3ccccc3)[C@]1(C)Oc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O11 mock treatment 163320.0 -5910.0 -0.4 178760.0 7240.0 0.54 0.0959 0.1426 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O12 mock treatment 167840.0 -1390.0 -0.09 181640.0 10100.0 0.75 0.4654 0.6132 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O13 compound treatment 170600.0 1370.0 0.09 178600.0 7080.0 0.53 0.4385 0.8196 3623380 BCB04_000272 COc1ccc(cc1OC)c2cn(CCNC(=O)Nc3ccccc3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O14 compound treatment 177120.0 7890.0 0.54 186360.0 14800.0 1.1 1.1612 0.9453 3623381 BCB04_000273 CN1C(=O)N([C@H]2[C@@H](COC(=O)c3ccccc3)[C@]1(C)Oc4ccccc24)C(=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O15 compound treatment 171680.0 2450.0 0.17 181520.0 10000.0 0.74 0.6442 0.8447 3623383 BCB04_000274 COc1ccc(cc1OC)c2cn(CCCNC(=O)[C@H](Cc3ccccc3)NS(=O)(=O)c4ccc(C)cc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O16 compound treatment 169160.0 -71.6 0.0 175600.0 4080.0 0.3 0.2112 0.6957 3623385 BCB04_000275 CN1C(=O)N([C@H]2[C@@H](COC(=O)c3ccccc3)[C@]1(C)Oc4ccccc24)C(=O)CC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O17 compound treatment 176440.0 7210.0 0.49 186320.0 14800.0 1.1 1.1263 0.9339 3623387 BCB04_000276 COc1ccc(cc1OC)c2cn(CCNC(=O)[C@H](Cc3ccccc3)NS(=O)(=O)c4ccc(C)cc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O18 compound treatment 214600.0 45400.0 3.09 213360.0 41800.0 3.11 4.389 1.0 3623389 BCB04_000277 COc1ccc(COC[C@]2(NC(=S)N[C@H]3[C@H]2CO[Si](C)(C)C(C)(C)C)Oc4ccccc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O19 compound treatment 169640.0 408.0 0.03 169880.0 -1640.0 -0.12 -0.0667 -0.5323 3623391 BCB04_000278 COc1ccc(cc1OC)c2cn(CCNC(=O)[C@@H](NS(=O)(=O)c3ccc(C)cc3)C(C)C)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O20 compound treatment 166520.0 -2710.0 -0.18 160360.0 -11200.0 -0.83 -0.7181 -0.8438 3623393 BCB04_000279 COc1ccc(COC[C@]2(Oc3ccccc3[C@H]4NC(=O)N2C)[C@@H]4CO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O21 compound treatment 168440.0 -792.0 -0.05 165520.0 -6000.0 -0.45 -0.354 -0.7868 3623395 BCB04_000280 COc1ccc(cc1OC)c2cn(C[C@@H]3CCCN3S(=O)(=O)c4ccc(C)cc4)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O22 compound treatment 166240.0 -2990.0 -0.2 164240.0 -7280.0 -0.54 -0.5274 -0.9108 3623397 BCB04_000281 COc1ccc(COC[C@@]2(Oc3ccccc3[C@@H]4[C@H]2CO[Si](C)(C)C(C)(C)C)N=C5SCc6ccccc6CN45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O23 compound treatment 156520.0 -12700.0 -0.87 158120.0 -13400.0 -1.0 -1.3181 -0.9975 3623399 BCB04_000282 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)Cn2cc(nn2)c3ccc(OC)c(OC)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 O24 compound treatment 158960.0 -10300.0 -0.7 158960.0 -12600.0 -0.93 -1.1563 -0.9899 3623401 BCB04_000283 COc1ccc(COC[C@]2(Oc3ccccc3[C@H]4NC(=O)N2C)[C@@H]4COC(=O)c5ccccc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P01 compound treatment 172680.0 3450.0 0.24 174600.0 3080.0 0.23 0.3282 0.9999 3616028 BCB04_000284 COc1cc(OC)c(CN(CC#CCO)S(=O)(=O)c2ccccc2[N+](=O)[O-])c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P02 mock treatment 173880.0 4650.0 0.32 170080.0 -1440.0 -0.11 0.1482 0.443 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P03 compound treatment 174640.0 5410.0 0.37 180680.0 9160.0 0.68 0.7427 0.9584 3623403 BCB04_000285 COc1cc(OC)c(CN(CC#CCN(CC(OC(=O)c2ccccc2)C=C)S(=O)(=O)c3c(OC)cc(OC)cc3OC)S(=O)(=O)c4ccccc4[N+](=O)[O-])c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P04 mock treatment 167880.0 -1350.0 -0.09 169720.0 -1800.0 -0.13 -0.16 -0.9832 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P05 compound treatment 169760.0 528.0 0.04 171880.0 358.0 0.03 0.0443 0.989 3623404 BCB04_000286 CCOC(=O)/C=C/C(CN(CC#CCN(Cc1c(OC)cc(OC)cc1OC)S(=O)(=O)c2ccccc2[N+](=O)[O-])S(=O)(=O)c3c(OC)cc(OC)cc3OC)OC(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P06 mock treatment 172520.0 3290.0 0.22 171520.0 -1.78 0.0 0.1584 0.7067 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P07 compound treatment 167920.0 -1310.0 -0.09 168320.0 -3200.0 -0.24 -0.2317 -0.9105 3623406 BCB04_000287 COc1cc(OC)c(CN(CC#CCOC(=O)c2ccccc2)S(=O)(=O)c3ccccc3[N+](=O)[O-])c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P08 mock treatment 167120.0 -2110.0 -0.14 173600.0 2080.0 0.15 0.0076 0.0359 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P09 compound treatment 181080.0 11800.0 0.81 185160.0 13600.0 1.02 1.2889 0.9936 3623407 BCB04_000288 CCOC(=O)/C=C/C(CNS(=O)(=O)c1ccc(Br)cc1)OC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P10 mock treatment 166360.0 -2870.0 -0.2 172080.0 558.0 0.04 -0.1091 -0.5449 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P11 mock treatment 166440.0 -2790.0 -0.19 171600.0 78.2 0.01 -0.1305 -0.6852 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P12 mock treatment 167000.0 -2230.0 -0.15 176640.0 5120.0 0.38 0.1618 0.3944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P13 compound treatment 177400.0 8170.0 0.56 179640.0 8120.0 0.6 0.821 0.9992 3623409 BCB04_000289 COc1cc(OC)c(CNS(=O)(=O)c2ccccc2[N+](=O)[O-])c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P14 mock treatment 169880.0 648.0 0.04 169000.0 -2520.0 -0.19 -0.1015 -0.5262 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P15 compound treatment 181560.0 12300.0 0.84 186440.0 14900.0 1.11 1.3794 0.9906 3623410 BCB04_000290 CCOC(=O)/C=C/C(O)CN(Cc1c(OC)cc(OC)cc1OC)S(=O)(=O)c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P16 mock treatment 171360.0 2130.0 0.15 169440.0 -2080.0 -0.15 -0.007 -0.0327 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P17 compound treatment 172000.0 2770.0 0.19 171200.0 -322.0 -0.02 0.1165 0.6125 3623412 BCB04_000291 COc1cc(OC)c(CN(CC(O)C=C)S(=O)(=O)c2ccc(Br)cc2)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P18 mock treatment 168960.0 -272.0 -0.02 167720.0 -3800.0 -0.28 -0.2132 -0.7518 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P19 compound treatment 193720.0 24500.0 1.67 184200.0 12700.0 0.94 1.8478 0.9635 3623413 BCB04_000292 COc1cc(OC)c(CN(CC#CCN(CC#CCOC(=O)c2ccccc2)S(=O)(=O)c3ccccc3[N+](=O)[O-])S(=O)(=O)c4ccccc4[N+](=O)[O-])c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P20 mock treatment 163120.0 -6110.0 -0.42 163040.0 -8480.0 -0.63 -0.741 -0.9797 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P21 compound treatment 194000.0 24800.0 1.69 206880.0 35400.0 2.63 3.0549 0.977 3623414 BCB04_000293 CC(C)(C)OC(=O)NCC1=C2CN(CC2=C3CN(C(COC(=O)c4ccccc4)C3C1)S(=O)(=O)c5ccc(Br)cc5)S(=O)(=O)c6ccccc6[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P22 mock treatment 160000.0 -9230.0 -0.63 160440.0 -11100.0 -0.82 -1.0282 -0.9911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P23 compound treatment 167080.0 -2150.0 -0.15 159760.0 -11800.0 -0.88 -0.7227 -0.8142 3623415 BCB04_000294 CC(C)(C)OC(=O)N[C@@H]1CN(CC2=C1C[C@H](COC(=O)c3ccccc3)C4=C2CN(C4)S(=O)(=O)c5ccc(Br)cc5)S(=O)(=O)c6ccccc6[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2319 P24 mock treatment 161040.0 -8190.0 -0.56 156240.0 -15300.0 -1.14 -1.1991 -0.9464 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A01 compound treatment 159080.0 -10300.0 -0.7 160920.0 -7270.0 -0.54 -0.8778 -0.9918 2019929 DHPC8.1_000001 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)O)c3ccsc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A02 compound treatment 168360.0 -994.0 -0.07 160800.0 -7390.0 -0.55 -0.4367 -0.7883 3557052 DHPC8.1_000002 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A03 compound treatment 160720.0 -8630.0 -0.59 161120.0 -7070.0 -0.53 -0.7882 -0.9984 3556472 DHPC8.1_000003 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)O)c3csc4ccccc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A04 compound treatment 166200.0 -3150.0 -0.22 164640.0 -3550.0 -0.26 -0.3387 -0.9948 3557032 DHPC8.1_000004 COc1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A05 compound treatment 162600.0 -6750.0 -0.46 159360.0 -8830.0 -0.66 -0.7902 -0.9849 2020334 DHPC8.1_000005 CC(C)[C@H]1C[C@@H](OCCCCO)OC(=C1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A06 compound treatment 161640.0 -7710.0 -0.53 157120.0 -11100.0 -0.82 -0.9543 -0.9765 3557033 DHPC8.1_000006 COc1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A07 compound treatment 162920.0 -6430.0 -0.44 162080.0 -6110.0 -0.45 -0.6316 -0.9998 2019875 DHPC8.1_000007 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A08 compound treatment 163160.0 -6190.0 -0.42 161480.0 -6710.0 -0.5 -0.6516 -0.9965 3556956 DHPC8.1_000008 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)Nc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A09 compound treatment 167760.0 -1590.0 -0.11 167160.0 -1030.0 -0.08 -0.1309 -0.9852 3556348 DHPC8.1_000009 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)O)c2csc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A10 compound treatment 162000.0 -7350.0 -0.5 162040.0 -6150.0 -0.46 -0.6781 -0.999 3557040 DHPC8.1_000010 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A11 compound treatment 161480.0 -7870.0 -0.54 162560.0 -5630.0 -0.42 -0.6758 -0.9925 2020415 DHPC8.1_000011 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A12 compound treatment 197760.0 28400.0 1.94 194080.0 25900.0 1.93 2.7321 1.0 2020331 DHPC8.1_000012 CC(C)[C@H]1C[C@@H](OCCCCO)OC(=C1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A13 mock treatment 161160.0 -8190.0 -0.56 157680.0 -10500.0 -0.78 -0.948 -0.9864 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A14 mock treatment 158680.0 -10700.0 -0.73 159440.0 -8750.0 -0.65 -0.9749 -0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A15 compound treatment 161400.0 -7950.0 -0.54 163200.0 -4990.0 -0.37 -0.6459 -0.9829 3556774 DHPC8.1_000013 COc1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A16 compound treatment 168680.0 -674.0 -0.05 165040.0 -3150.0 -0.23 -0.1981 -0.83 3640820 DHPC8.1_000014 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCCCC3)c4ccc-5c(Cc6ccccc65)c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A17 compound treatment 196000.0 26600.0 1.82 197800.0 29600.0 2.2 2.843 0.9954 2019902 DHPC8.1_000015 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)O)c3ccc4OCOc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A18 compound treatment 158520.0 -10800.0 -0.74 163640.0 -4550.0 -0.34 -0.7616 -0.9374 3557021 DHPC8.1_000016 CC(C)[C@@H]1C[C@H](OCCCCO)OC(=C1)C(=O)N2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A19 compound treatment 164080.0 -5270.0 -0.36 164240.0 -3950.0 -0.29 -0.462 -0.995 3556749 DHPC8.1_000017 COc1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A20 compound treatment 208040.0 38700.0 2.64 205360.0 37200.0 2.77 3.8213 0.9997 2020412 DHPC8.1_000018 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A21 compound treatment 161560.0 -7790.0 -0.53 164280.0 -3910.0 -0.29 -0.5814 -0.9598 2019389 DHPC8.1_000019 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2ccsc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A22 compound treatment 164720.0 -4630.0 -0.32 163720.0 -4470.0 -0.33 -0.4585 -0.9997 3556360 DHPC8.1_000020 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCCCC2)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A23 compound treatment 157680.0 -11700.0 -0.8 160640.0 -7550.0 -0.56 -0.96 -0.9854 2020901 DHPC8.1_000021 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 A24 compound treatment 191440.0 22100.0 1.51 196240.0 28100.0 2.09 2.5411 0.9871 2020439 DHPC8.1_000022 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B01 compound treatment 187360.0 18000.0 1.23 185600.0 17400.0 1.3 1.7844 0.9996 2019899 DHPC8.1_000023 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccc7OCOc7c6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B02 compound treatment 154000.0 -15400.0 -1.05 158040.0 -10100.0 -0.76 -1.2742 -0.9872 3556793 DHPC8.1_000024 CC(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B03 compound treatment 188360.0 19000.0 1.3 192640.0 24500.0 1.82 2.2031 0.9861 3556950 DHPC8.1_000025 COc1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B04 compound treatment 193320.0 24000.0 1.63 191760.0 23600.0 1.75 2.3959 0.9994 3557001 DHPC8.1_000026 COc1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCN(Cc5ccc6OCOc6c5)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B05 compound treatment 175400.0 6050.0 0.41 170400.0 2210.0 0.16 0.4079 0.919 3557015 DHPC8.1_000027 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)Nc3ccccc3)c4cccs4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B06 compound treatment 158480.0 -10900.0 -0.74 159280.0 -8910.0 -0.66 -0.993 -0.9984 3556910 DHPC8.1_000028 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B07 compound treatment 190680.0 21300.0 1.45 191680.0 23500.0 1.75 2.2644 0.9958 3556593 DHPC8.1_000029 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCC2)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B08 compound treatment 155840.0 -13500.0 -0.92 154840.0 -13300.0 -0.99 -1.3539 -0.9993 1952202 DHPC8.1_000030 CC(C)/C=C/C(=O)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B09 compound treatment 199480.0 30100.0 2.05 197000.0 28800.0 2.14 2.9687 0.9998 3556823 DHPC8.1_000031 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)Nc3ccccc3)c4ccc5OCOc5c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B10 compound treatment 162680.0 -6670.0 -0.46 158360.0 -9830.0 -0.73 -0.8389 -0.9739 3644571 DHPC8.1_000032 C=CCOC(=O)C(=O)/C=C/c1ccc2Cc3ccccc3-c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B11 compound treatment 204800.0 35400.0 2.42 201560.0 33400.0 2.48 3.4651 0.9999 2019332 DHPC8.1_000033 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B12 compound treatment 172240.0 2890.0 0.2 166320.0 -1870.0 -0.14 0.0408 0.1696 1952204 DHPC8.1_000034 C=CCOC(=O)C(=O)/C=C/c1ccc2OCOc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B13 mock treatment 159320.0 -10000.0 -0.68 157680.0 -10500.0 -0.78 -1.0367 -0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B14 mock treatment 157040.0 -12300.0 -0.84 154640.0 -13500.0 -1.01 -1.3066 -0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B15 compound treatment 156360.0 -13000.0 -0.89 156240.0 -11900.0 -0.89 -1.2552 -1.0 3557022 DHPC8.1_000035 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B16 compound treatment 158200.0 -11200.0 -0.76 160960.0 -7230.0 -0.54 -0.9181 -0.9856 3644223 DHPC8.1_000036 COc1ccc(/C=C/C(=O)C(=O)OCC=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B17 compound treatment 202800.0 33400.0 2.28 196160.0 28000.0 2.08 3.0845 0.999 3641348 DHPC8.1_000037 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccc-6c(Cc7ccccc76)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B18 compound treatment 160400.0 -8950.0 -0.61 160680.0 -7510.0 -0.56 -0.8268 -0.999 3644225 DHPC8.1_000038 COC(=O)c1ccc(/C=C/C(=O)C(=O)OCC=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B19 compound treatment 193960.0 24600.0 1.68 196000.0 27800.0 2.07 2.6499 0.9946 3556975 DHPC8.1_000039 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5csc6ccccc56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B20 compound treatment 163480.0 -5870.0 -0.4 160840.0 -7350.0 -0.55 -0.6699 -0.9883 3644221 DHPC8.1_000040 C=CCOC(=O)C(=O)/C=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B21 compound treatment 164640.0 -4710.0 -0.32 159800.0 -8390.0 -0.62 -0.6687 -0.9524 3641365 DHPC8.1_000041 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)NCc2ccccc2)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B22 compound treatment 156920.0 -12400.0 -0.85 155160.0 -13000.0 -0.97 -1.285 -0.9978 1952200 DHPC8.1_000042 C=CCOC(=O)C(=O)/C=C/c1ccsc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B23 compound treatment 193760.0 24400.0 1.66 191240.0 23100.0 1.72 2.3898 0.9999 2020358 DHPC8.1_000043 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 B24 compound treatment 160320.0 -9030.0 -0.62 172320.0 4130.0 0.31 -0.218 -0.3167 3644241 DHPC8.1_000044 C=CCOC(=O)C(=O)/C=C/c1csc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C01 compound treatment 159440.0 -9910.0 -0.68 161800.0 -6390.0 -0.48 -0.8141 -0.9852 2019335 DHPC8.1_000045 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C02 compound treatment 175200.0 5850.0 0.4 176000.0 7810.0 0.58 0.693 0.983 3556887 DHPC8.1_000046 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)Nc3ccccc3)c4cccs4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C03 compound treatment 164280.0 -5070.0 -0.35 170720.0 2530.0 0.19 -0.1113 -0.2826 3641369 DHPC8.1_000047 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)O)c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C04 compound treatment 204480.0 35100.0 2.39 196920.0 28700.0 2.14 3.2055 0.9984 3556899 DHPC8.1_000048 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6cccs6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C05 compound treatment 179520.0 10200.0 0.69 169360.0 1170.0 0.09 0.5518 0.7899 3221232 DHPC8.1_000049 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C06 compound treatment 201200.0 31800.0 2.17 188640.0 20500.0 1.52 2.6116 0.9849 2019386 DHPC8.1_000050 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccsc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C07 compound treatment 166760.0 -2590.0 -0.18 163360.0 -4830.0 -0.36 -0.3791 -0.9467 2019821 DHPC8.1_000051 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C08 compound treatment 206680.0 37300.0 2.54 192880.0 24700.0 1.84 3.0989 0.9872 2020898 DHPC8.1_000052 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccccc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C09 compound treatment 167160.0 -2190.0 -0.15 163600.0 -4590.0 -0.34 -0.3472 -0.9314 2019281 DHPC8.1_000053 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C10 compound treatment 174840.0 5490.0 0.37 171320.0 3130.0 0.23 0.4293 0.9741 3556999 DHPC8.1_000054 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C11 mock treatment 169880.0 526.0 0.04 162320.0 -5870.0 -0.44 -0.2834 -0.6469 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C12 mock treatment 167880.0 -1470.0 -0.1 159280.0 -8910.0 -0.66 -0.5398 -0.8051 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C13 compound treatment 165800.0 -3550.0 -0.24 158520.0 -9670.0 -0.72 -0.6801 -0.8958 3556650 DHPC8.1_000055 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)O)c3csc4ccccc34)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C14 compound treatment 168880.0 -474.0 -0.03 167760.0 -427.0 -0.03 -0.0454 -1.0 3557047 DHPC8.1_000056 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2csc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C15 mock treatment 163480.0 -5870.0 -0.4 155320.0 -12900.0 -0.96 -0.9604 -0.9252 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C16 mock treatment 160120.0 -9230.0 -0.63 154680.0 -13500.0 -1.01 -1.156 -0.9746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C17 compound treatment 164520.0 -4830.0 -0.33 162760.0 -5430.0 -0.4 -0.5187 -0.9949 2019794 DHPC8.1_000057 CC(C)[C@@H]1C[C@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C18 compound treatment 168520.0 -834.0 -0.06 158480.0 -9710.0 -0.72 -0.5511 -0.7604 3556969 DHPC8.1_000058 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2ccsc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C19 compound treatment 166680.0 -2670.0 -0.18 155920.0 -12300.0 -0.91 -0.7745 -0.8319 2020361 DHPC8.1_000059 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C20 compound treatment 174600.0 5250.0 0.36 172000.0 3810.0 0.28 0.4535 0.9934 2020983 DHPC8.1_000060 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)NCc3ccccc3)c4ccsc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C21 compound treatment 174480.0 5130.0 0.35 169960.0 1770.0 0.13 0.3404 0.9113 3556698 DHPC8.1_000061 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)O)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C22 compound treatment 167920.0 -1430.0 -0.1 164000.0 -4190.0 -0.31 -0.2895 -0.8864 3556867 DHPC8.1_000062 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)Nc3ccccc3)c4ccsc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C23 compound treatment 159640.0 -9710.0 -0.66 156440.0 -11700.0 -0.87 -1.0865 -0.9906 2020955 DHPC8.1_000063 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 C24 compound treatment 168640.0 -714.0 -0.05 166960.0 -1230.0 -0.09 -0.099 -0.9566 3188423 DHPC8.1_000064 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D01 compound treatment 166160.0 -3190.0 -0.22 166200.0 -1990.0 -0.15 -0.2586 -0.9822 3557016 DHPC8.1_000065 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4cccs4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D02 compound treatment 156200.0 -13200.0 -0.9 163640.0 -4550.0 -0.34 -0.8735 -0.9112 3644239 DHPC8.1_000066 C=CCOC(=O)C(=O)/C=C/c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D03 compound treatment 162600.0 -6750.0 -0.46 167800.0 -387.0 -0.03 -0.346 -0.7499 3639708 DHPC8.1_000067 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCC2)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D04 compound treatment 172840.0 3490.0 0.24 163520.0 -4670.0 -0.35 -0.0776 -0.1843 3644573 DHPC8.1_000068 OCc1ccc(COC=C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D05 compound treatment 172880.0 3530.0 0.24 164160.0 -4030.0 -0.3 -0.042 -0.1093 3640829 DHPC8.1_000069 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D06 compound treatment 162840.0 -6510.0 -0.44 166160.0 -2030.0 -0.15 -0.4207 -0.897 3644574 DHPC8.1_000070 OCCCCOC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D07 compound treatment 170400.0 1050.0 0.07 167360.0 -827.0 -0.06 0.0069 0.073 3556952 DHPC8.1_000071 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D08 compound treatment 163560.0 -5790.0 -0.4 156680.0 -11500.0 -0.86 -0.8849 -0.9383 1009811 DHPC8.1_000072 Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D09 compound treatment 166800.0 -2550.0 -0.17 169280.0 1090.0 0.08 -0.0656 -0.3415 3557002 DHPC8.1_000073 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D10 compound treatment 161440.0 -7910.0 -0.54 167200.0 -987.0 -0.07 -0.4335 -0.7961 1020810 DHPC8.1_000074 C1CCNCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D11 mock treatment 164240.0 -5110.0 -0.35 158520.0 -9670.0 -0.72 -0.7553 -0.9447 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D12 mock treatment 162800.0 -6550.0 -0.45 156760.0 -11400.0 -0.85 -0.9174 -0.9549 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D13 compound treatment 195840.0 26500.0 1.81 186400.0 18200.0 1.36 2.2353 0.99 2019791 DHPC8.1_000075 CC(C)[C@@H]1C[C@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D14 compound treatment 169480.0 126.0 0.01 164840.0 -3350.0 -0.25 -0.1701 -0.6824 1009903 DHPC8.1_000076 NCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D15 mock treatment 162200.0 -7150.0 -0.49 161080.0 -7110.0 -0.53 -0.7189 -0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D16 mock treatment 152600.0 -16800.0 -1.14 159560.0 -8630.0 -0.64 -1.2617 -0.9629 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D17 compound treatment 178200.0 8850.0 0.6 178760.0 10600.0 0.79 0.9829 0.9914 3638708 DHPC8.1_000077 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)NCc3ccccc3)c4ccc-5c(Cc6ccccc65)c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D18 compound treatment 166400.0 -2950.0 -0.2 160880.0 -7310.0 -0.54 -0.527 -0.9087 1237515 DHPC8.1_000078 C(N1CCNCC1)c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D19 compound treatment 171040.0 1690.0 0.11 156760.0 -11400.0 -0.85 -0.5201 -0.606 3556986 DHPC8.1_000079 CC(C)[C@@H]1C[C@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D20 mock treatment 162320.0 -7030.0 -0.48 155360.0 -12800.0 -0.95 -1.0142 -0.9493 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D21 compound treatment 197000.0 27600.0 1.88 194000.0 25800.0 1.92 2.6912 1.0 3638674 DHPC8.1_000080 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccc-7c(Cc8ccccc87)c6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D22 mock treatment 163720.0 -5630.0 -0.38 157400.0 -10800.0 -0.8 -0.8393 -0.943 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D23 compound treatment 175520.0 6170.0 0.42 171480.0 3290.0 0.25 0.4705 0.967 3557017 DHPC8.1_000081 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 D24 mock treatment 155160.0 -14200.0 -0.97 156760.0 -11400.0 -0.85 -1.2857 -0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E01 mock treatment 162720.0 -6630.0 -0.45 163880.0 -4310.0 -0.32 -0.5465 -0.9858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E02 mock treatment 165840.0 -3510.0 -0.24 169480.0 1290.0 0.1 -0.1014 -0.3927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E03 compound treatment 180440.0 11100.0 0.76 185960.0 17800.0 1.32 1.4698 0.9648 3556755 DHPC8.1_000082 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)O)c3cccs3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E04 compound treatment 204640.0 35300.0 2.41 203000.0 34800.0 2.59 3.5332 0.9993 3556452 DHPC8.1_000083 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCCCC3)c4ccc5OCOc5c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E05 compound treatment 185320.0 16000.0 1.09 182600.0 14400.0 1.07 1.5282 1.0 3638716 DHPC8.1_000084 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)O)c3ccc-4c(Cc5ccccc54)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E06 compound treatment 208120.0 38800.0 2.64 198800.0 30600.0 2.28 3.4799 0.9973 3556638 DHPC8.1_000085 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4ccc5OCOc5c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E07 compound treatment 174000.0 4650.0 0.32 171040.0 2850.0 0.21 0.3741 0.9811 3556765 DHPC8.1_000086 COc1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E08 compound treatment 173960.0 4610.0 0.31 175520.0 7330.0 0.55 0.6079 0.9655 3641363 DHPC8.1_000087 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)Nc2ccccc2)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E09 mock treatment 169440.0 85.7 0.01 170480.0 2290.0 0.17 0.1248 0.7309 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E10 mock treatment 169600.0 246.0 0.02 165480.0 -2710.0 -0.2 -0.1306 -0.6461 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E11 compound treatment 186080.0 16700.0 1.14 183160.0 15000.0 1.11 1.5943 0.9999 3556778 DHPC8.1_000088 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)O)c3cccs3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E12 compound treatment 212760.0 43400.0 2.96 208280.0 40100.0 2.98 4.2025 1.0 2020416 DHPC8.1_000089 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)NCc2ccccc2)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E13 compound treatment 183800.0 14400.0 0.98 168160.0 -27.3 0.0 0.695 0.7056 3640846 DHPC8.1_000090 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)O)c3ccc-4c(Cc5ccccc54)c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E14 compound treatment 180440.0 11100.0 0.76 174640.0 6450.0 0.48 0.874 0.976 3557004 DHPC8.1_000091 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)Nc3ccccc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E15 compound treatment 175080.0 5730.0 0.39 173320.0 5130.0 0.38 0.5461 0.9999 2020469 DHPC8.1_000092 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)O)c2ccsc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E16 compound treatment 186400.0 17000.0 1.16 178960.0 10800.0 0.8 1.3887 0.9836 2019363 DHPC8.1_000093 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E17 mock treatment 168320.0 -1030.0 -0.07 171840.0 3650.0 0.27 0.1424 0.5069 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E18 mock treatment 173920.0 4570.0 0.31 169360.0 1170.0 0.09 0.2818 0.8718 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E19 compound treatment 173920.0 4570.0 0.31 171320.0 3130.0 0.23 0.385 0.9899 3639760 DHPC8.1_000094 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E20 compound treatment 170440.0 1090.0 0.07 168880.0 693.0 0.05 0.0888 0.9844 3556954 DHPC8.1_000095 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E21 compound treatment 203600.0 34200.0 2.33 202040.0 33900.0 2.52 3.4325 0.9993 2020982 DHPC8.1_000096 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)O)c3ccc4OCOc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E22 compound treatment 176120.0 6770.0 0.46 180480.0 12300.0 0.91 0.9731 0.9497 2020389 DHPC8.1_000097 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E23 compound treatment 171840.0 2490.0 0.17 169880.0 1690.0 0.13 0.2089 0.9893 3556782 DHPC8.1_000098 COc1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 E24 compound treatment 173400.0 4050.0 0.28 170920.0 2730.0 0.2 0.3389 0.9888 3556973 DHPC8.1_000099 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2csc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F01 mock treatment 160120.0 -9230.0 -0.63 162640.0 -5550.0 -0.41 -0.7371 -0.9791 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F02 mock treatment 169560.0 206.0 0.01 171640.0 3450.0 0.26 0.1916 0.7446 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F03 compound treatment 181320.0 12000.0 0.82 181200.0 13000.0 0.97 1.2617 0.9964 3557044 DHPC8.1_000100 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCC2)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F04 mock treatment 166720.0 -2630.0 -0.18 169040.0 853.0 0.06 -0.0821 -0.4311 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F05 compound treatment 167480.0 -1870.0 -0.13 172000.0 3810.0 0.28 0.1103 0.3544 3556797 DHPC8.1_000101 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F06 mock treatment 168240.0 -1110.0 -0.08 168120.0 -67.3 -0.01 -0.0573 -0.7521 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F07 compound treatment 176200.0 6850.0 0.47 182320.0 14100.0 1.05 1.0738 0.9331 3556966 DHPC8.1_000102 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)Nc2ccccc2)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F08 mock treatment 168680.0 -674.0 -0.05 166800.0 -1390.0 -0.1 -0.1055 -0.9336 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F09 mock treatment 169440.0 85.7 0.01 167680.0 -507.0 -0.04 -0.0226 -0.5906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F10 mock treatment 169320.0 -34.3 0.0 168520.0 333.0 0.02 0.0159 0.6375 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F11 compound treatment 179320.0 9970.0 0.68 173320.0 5130.0 0.38 0.7506 0.9629 2019255 DHPC8.1_000103 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F12 mock treatment 173920.0 4570.0 0.31 174240.0 6050.0 0.45 0.5386 0.9837 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F13 compound treatment 202000.0 32600.0 2.23 201920.0 33700.0 2.51 3.3491 0.9982 2020871 DHPC8.1_000104 CC(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F14 mock treatment 168960.0 -394.0 -0.03 170080.0 1890.0 0.14 0.0806 0.562 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F15 compound treatment 182440.0 13100.0 0.89 181920.0 13700.0 1.02 1.3536 0.9977 3556490 DHPC8.1_000105 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCCCC3)c4csc5ccccc45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F16 mock treatment 171760.0 2410.0 0.16 168240.0 52.7 0.0 0.1187 0.7238 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F17 mock treatment 165440.0 -3910.0 -0.27 165560.0 -2630.0 -0.2 -0.327 -0.9883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F18 mock treatment 170640.0 1290.0 0.09 170320.0 2130.0 0.16 0.1742 0.9608 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F19 compound treatment 211480.0 42100.0 2.87 212520.0 44300.0 3.3 4.3639 0.9976 3557014 DHPC8.1_000106 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6csc7ccccc67)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F20 mock treatment 167440.0 -1910.0 -0.13 163360.0 -4830.0 -0.36 -0.3463 -0.906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F21 compound treatment 182560.0 13200.0 0.9 179200.0 11000.0 0.82 1.2162 0.9989 3556602 DHPC8.1_000107 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F22 mock treatment 169160.0 -194.0 -0.01 164000.0 -4190.0 -0.31 -0.2297 -0.7365 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F23 compound treatment 178840.0 9490.0 0.65 176400.0 8210.0 0.61 0.8895 0.9996 3556662 DHPC8.1_000108 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4csc5ccccc45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 F24 mock treatment 163600.0 -5750.0 -0.39 160480.0 -7710.0 -0.57 -0.683 -0.9828 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G01 compound treatment 176280.0 6930.0 0.47 171360.0 3170.0 0.24 0.5008 0.9487 2021009 DHPC8.1_000109 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)O)c3ccsc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G02 compound treatment 215800.0 46400.0 3.17 220400.0 52200.0 3.89 4.9869 0.9948 3557048 DHPC8.1_000110 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5csc6ccccc56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G03 mock treatment 175400.0 6050.0 0.41 175080.0 6890.0 0.51 0.6542 0.9941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G04 mock treatment 175120.0 5770.0 0.39 173280.0 5090.0 0.38 0.546 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G05 compound treatment 180240.0 10900.0 0.74 174600.0 6410.0 0.48 0.8623 0.9772 3556597 DHPC8.1_000111 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2csc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G06 compound treatment 187200.0 17800.0 1.22 189720.0 21500.0 1.6 1.9935 0.9908 3556981 DHPC8.1_000112 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G07 compound treatment 207960.0 38600.0 2.63 208760.0 40600.0 3.02 3.9964 0.9977 2019362 DHPC8.1_000113 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)O)c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G08 compound treatment 208000.0 38600.0 2.63 202200.0 34000.0 2.53 3.6531 0.9998 3556934 DHPC8.1_000114 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G09 compound treatment 179440.0 10100.0 0.69 178400.0 10200.0 0.76 1.0237 0.9987 2020874 DHPC8.1_000115 CC(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G10 compound treatment 183040.0 13700.0 0.93 180240.0 12100.0 0.9 1.2941 0.9998 3556586 DHPC8.1_000116 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCC2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G11 compound treatment 187920.0 18600.0 1.27 185480.0 17300.0 1.29 1.8051 1.0 2019928 DHPC8.1_000117 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)OCC=C)c3ccsc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G12 compound treatment 184920.0 15600.0 1.06 182080.0 13900.0 1.03 1.4815 0.9999 2019309 DHPC8.1_000118 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G13 compound treatment 176680.0 7330.0 0.5 175160.0 6970.0 0.52 0.7201 0.9998 2019820 DHPC8.1_000119 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)OCC=C)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G14 compound treatment 182600.0 13200.0 0.9 179400.0 11200.0 0.83 1.2287 0.9992 3557020 DHPC8.1_000120 CC(C)[C@@H]1C[C@H](OCCCCO)OC(=C1)C(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G15 compound treatment 183360.0 14000.0 0.95 178800.0 10600.0 0.79 1.2337 0.9956 3556710 DHPC8.1_000121 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)OCC=C)c3cccs3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G16 compound treatment 177280.0 7930.0 0.54 179320.0 11100.0 0.83 0.968 0.9785 2019228 DHPC8.1_000122 CC(C)[C@@H]1C[C@H](OCCCCO)OC(=C1)C(=O)NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G17 compound treatment 205920.0 36600.0 2.49 214160.0 46000.0 3.42 4.1822 0.9879 2019901 DHPC8.1_000123 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)OCC=C)c3ccc4OCOc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G18 compound treatment 183040.0 13700.0 0.93 176880.0 8690.0 0.65 1.1172 0.984 3556839 DHPC8.1_000124 COc1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G19 mock treatment 174560.0 5210.0 0.35 175280.0 7090.0 0.53 0.6242 0.9813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G20 mock treatment 170480.0 1130.0 0.08 174520.0 6330.0 0.47 0.3875 0.8116 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G21 compound treatment 206480.0 37100.0 2.53 198400.0 30200.0 2.25 3.3798 0.9983 2019361 DHPC8.1_000125 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)OCC=C)c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G22 compound treatment 179320.0 9970.0 0.68 180880.0 12700.0 0.94 1.1484 0.9869 3556997 DHPC8.1_000126 COc1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G23 compound treatment 173080.0 3730.0 0.25 171160.0 2970.0 0.22 0.3361 0.9976 3556739 DHPC8.1_000127 COc1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 G24 compound treatment 171360.0 2010.0 0.14 178600.0 10400.0 0.77 0.6447 0.8192 3556979 DHPC8.1_000128 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCCCC2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H01 compound treatment 186600.0 17200.0 1.18 180520.0 12300.0 0.92 1.4804 0.9925 3557049 DHPC8.1_000129 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H02 mock treatment 167080.0 -2270.0 -0.16 169000.0 813.0 0.06 -0.0669 -0.4018 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H03 mock treatment 174160.0 4810.0 0.33 173080.0 4890.0 0.36 0.4892 0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H04 mock treatment 169120.0 -234.0 -0.02 174240.0 6050.0 0.45 0.3072 0.6816 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H05 compound treatment 175160.0 5810.0 0.4 176200.0 8010.0 0.6 0.7016 0.9802 3556944 DHPC8.1_000130 COc1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H06 mock treatment 174200.0 4850.0 0.33 171040.0 2850.0 0.21 0.3837 0.9771 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H07 compound treatment 172400.0 3050.0 0.21 175960.0 7770.0 0.58 0.5559 0.9044 2020308 DHPC8.1_000131 CC(C)[C@H]1C[C@@H](OCCCCO)OC(=C1)C(=O)NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H08 mock treatment 175200.0 5850.0 0.4 171560.0 3370.0 0.25 0.4593 0.9752 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H09 compound treatment 212120.0 42800.0 2.92 210760.0 42600.0 3.17 4.3022 0.9991 3556994 DHPC8.1_000132 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H10 mock treatment 176520.0 7170.0 0.49 175120.0 6930.0 0.52 0.7103 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H11 compound treatment 179920.0 10600.0 0.72 178440.0 10300.0 0.76 1.0489 0.9996 3556903 DHPC8.1_000133 CC(C)[C@H]1C[C@@H](OCCCCO)OC(=C1)C(=O)Nc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H12 mock treatment 170560.0 1210.0 0.08 169360.0 1170.0 0.09 0.1198 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H13 compound treatment 181800.0 12400.0 0.85 176840.0 8650.0 0.64 1.0554 0.9907 3556855 DHPC8.1_000134 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H14 mock treatment 172720.0 3370.0 0.23 176680.0 8490.0 0.63 0.6092 0.906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H15 compound treatment 211040.0 41700.0 2.84 219400.0 51200.0 3.81 4.7048 0.9895 3557036 DHPC8.1_000135 COc1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H16 mock treatment 176440.0 7090.0 0.48 173400.0 5210.0 0.39 0.6159 0.9941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H17 compound treatment 193960.0 24600.0 1.68 185520.0 17300.0 1.29 2.0984 0.9916 3556893 DHPC8.1_000136 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H18 mock treatment 170560.0 1210.0 0.08 171000.0 2810.0 0.21 0.2062 0.9166 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H19 mock treatment 170440.0 1090.0 0.07 171040.0 2850.0 0.21 0.2025 0.9005 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H20 mock treatment 171040.0 1690.0 0.11 170360.0 2170.0 0.16 0.1956 0.986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H21 compound treatment 173520.0 4170.0 0.28 173160.0 4970.0 0.37 0.4625 0.9914 3556789 DHPC8.1_000137 CC(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H22 mock treatment 170640.0 1290.0 0.09 167000.0 -1190.0 -0.09 -5.0E-4 -0.004 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H23 compound treatment 174480.0 5130.0 0.35 176880.0 8690.0 0.65 0.7046 0.9582 2019849 DHPC8.1_000138 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 H24 mock treatment 163080.0 -6270.0 -0.43 164480.0 -3710.0 -0.28 -0.4976 -0.9775 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I01 compound treatment 185480.0 16100.0 1.1 184280.0 16100.0 1.2 1.6243 0.9991 2020954 DHPC8.1_000139 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I02 compound treatment 199800.0 30400.0 2.08 194160.0 26000.0 1.93 2.8346 0.9994 2019818 DHPC8.1_000140 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccccc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I03 compound treatment 170440.0 1090.0 0.07 171920.0 3730.0 0.28 0.2488 0.8653 2020414 DHPC8.1_000141 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I04 compound treatment 177680.0 8330.0 0.57 171200.0 3010.0 0.22 0.5599 0.9174 3556987 DHPC8.1_000142 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I05 mock treatment 174720.0 5370.0 0.37 171200.0 3010.0 0.22 0.4172 0.9724 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I06 mock treatment 176640.0 7290.0 0.5 170680.0 2490.0 0.19 0.4824 0.9098 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I07 compound treatment 207000.0 37600.0 2.57 204080.0 35900.0 2.67 3.7038 0.9998 2020441 DHPC8.1_000143 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)OCC=C)c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I08 compound treatment 176640.0 7290.0 0.5 174080.0 5890.0 0.44 0.6614 0.9981 3557003 DHPC8.1_000144 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I09 compound treatment 174280.0 4930.0 0.34 173160.0 4970.0 0.37 0.4992 0.9988 2019253 DHPC8.1_000145 CC(C)[C@@H]1C[C@H](OCCCCO)OC(=C1)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I10 compound treatment 210760.0 41400.0 2.82 208520.0 40300.0 3.0 4.1187 0.9995 3556993 DHPC8.1_000146 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)Nc3ccccc3)c4ccc5OCOc5c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I11 compound treatment 176960.0 7610.0 0.52 177000.0 8810.0 0.66 0.8305 0.9932 3556703 DHPC8.1_000147 COc1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I12 compound treatment 216000.0 46600.0 3.18 214400.0 46200.0 3.44 4.6808 0.9992 2019872 DHPC8.1_000148 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCN(Cc5ccc6OCOc6c5)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I13 compound treatment 176600.0 7250.0 0.49 174880.0 6690.0 0.5 0.7015 1.0 2020873 DHPC8.1_000149 CC(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I14 compound treatment 187480.0 18100.0 1.24 186360.0 18200.0 1.35 1.8302 0.999 3556847 DHPC8.1_000150 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I15 compound treatment 183440.0 14100.0 0.96 180720.0 12500.0 0.93 1.3386 0.9999 3556735 DHPC8.1_000151 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)OCC=C)c3cccs3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I16 compound treatment 219080.0 49700.0 3.39 206480.0 38300.0 2.85 4.4125 0.9963 3557019 DHPC8.1_000152 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6cccs6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I17 compound treatment 175880.0 6530.0 0.44 171840.0 3650.0 0.27 0.5068 0.9721 3556716 DHPC8.1_000153 COc1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I18 compound treatment 206920.0 37600.0 2.56 198680.0 30500.0 2.27 3.4157 0.9982 3557029 DHPC8.1_000154 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccc3OCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I19 compound treatment 203000.0 33600.0 2.29 204560.0 36400.0 2.71 3.5362 0.9966 2020981 DHPC8.1_000155 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)OCC=C)c3ccc4OCOc4c3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I20 compound treatment 181960.0 12600.0 0.86 178760.0 10600.0 0.79 1.1641 0.999 3639748 DHPC8.1_000156 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I21 mock treatment 169440.0 85.7 0.01 165640.0 -2550.0 -0.19 -0.1299 -0.685 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I22 mock treatment 167560.0 -1790.0 -0.12 165880.0 -2310.0 -0.17 -0.2079 -0.9862 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I23 compound treatment 165960.0 -3390.0 -0.23 170040.0 1850.0 0.14 -0.0661 -0.2455 2019388 DHPC8.1_000157 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)OCC=C)c2ccsc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 I24 compound treatment 170040.0 686.0 0.05 168520.0 333.0 0.02 0.0506 0.9558 3556942 DHPC8.1_000158 COc1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J01 compound treatment 174720.0 5370.0 0.37 172240.0 4050.0 0.3 0.472 0.9954 3556857 DHPC8.1_000159 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)Nc3ccccc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J02 mock treatment 170560.0 1210.0 0.08 170320.0 2130.0 0.16 0.1704 0.9531 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J03 compound treatment 215760.0 46400.0 3.16 210600.0 42400.0 3.16 4.4692 1.0 3556332 DHPC8.1_000160 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCCCC2)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J04 mock treatment 171200.0 1850.0 0.13 173240.0 5050.0 0.38 0.3549 0.8949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J05 mock treatment 170960.0 1610.0 0.11 169680.0 1490.0 0.11 0.156 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J06 mock treatment 178560.0 9210.0 0.63 171560.0 3370.0 0.25 0.6213 0.9191 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J07 compound treatment 234800.0 65400.0 4.46 230720.0 62500.0 4.65 6.446 0.9998 3639718 DHPC8.1_000161 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccc-6c(Cc7ccccc76)c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J08 mock treatment 172080.0 2730.0 0.19 174280.0 6090.0 0.45 0.452 0.9224 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J09 compound treatment 184640.0 15300.0 1.04 179880.0 11700.0 0.87 1.3523 0.996 3556660 DHPC8.1_000162 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)NCc3ccccc3)c4csc5ccccc45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J10 mock treatment 174120.0 4770.0 0.32 173800.0 5610.0 0.42 0.5251 0.9923 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J11 compound treatment 189320.0 20000.0 1.36 179720.0 11500.0 0.86 1.5695 0.9753 3556488 DHPC8.1_000163 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)NCc3ccccc3)c4csc5ccccc45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J12 mock treatment 178880.0 9530.0 0.65 174200.0 6010.0 0.45 0.7757 0.9835 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J13 compound treatment 181520.0 12200.0 0.83 179720.0 11500.0 0.86 1.1934 0.9999 2020335 DHPC8.1_000164 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)NCc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J14 mock treatment 171280.0 1930.0 0.13 173000.0 4810.0 0.36 0.3461 0.9073 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J15 compound treatment 209880.0 40500.0 2.76 210520.0 42300.0 3.15 4.1816 0.9979 3556851 DHPC8.1_000165 COc1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCN(Cc5ccc6OCOc6c5)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J16 mock treatment 171120.0 1770.0 0.12 172120.0 3930.0 0.29 0.2921 0.9229 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J17 compound treatment 177040.0 7690.0 0.52 172920.0 4730.0 0.35 0.6196 0.9813 3556946 DHPC8.1_000166 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2ccc(OC)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J18 mock treatment 172680.0 3330.0 0.23 171280.0 3090.0 0.23 0.3231 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J19 compound treatment 179120.0 9770.0 0.67 178200.0 10000.0 0.75 0.9977 0.9984 3556621 DHPC8.1_000167 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J20 mock treatment 167000.0 -2350.0 -0.16 164360.0 -3830.0 -0.28 -0.3149 -0.9632 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J21 mock treatment 165240.0 -4110.0 -0.28 161960.0 -6230.0 -0.46 -0.5261 -0.9711 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J22 mock treatment 165200.0 -4150.0 -0.28 166680.0 -1510.0 -0.11 -0.2796 -0.9178 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J23 compound treatment 199760.0 30400.0 2.07 205920.0 37700.0 2.81 3.4516 0.9888 2019336 DHPC8.1_000168 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 J24 mock treatment 158240.0 -11100.0 -0.76 156920.0 -11300.0 -0.84 -1.1288 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K01 compound treatment 175360.0 6010.0 0.41 165480.0 -2710.0 -0.2 0.147 0.3222 2019874 DHPC8.1_000169 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K02 compound treatment 193600.0 24200.0 1.65 188680.0 20500.0 1.53 2.2473 0.9992 3556977 DHPC8.1_000170 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)Nc2ccccc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K03 compound treatment 179200.0 9850.0 0.67 178520.0 10300.0 0.77 1.0184 0.9977 3641368 DHPC8.1_000171 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)OCC=C)c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K04 compound treatment 181760.0 12400.0 0.85 176360.0 8170.0 0.61 1.0282 0.9869 3557011 DHPC8.1_000172 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K05 compound treatment 182800.0 13400.0 0.92 176280.0 8090.0 0.6 1.0741 0.9792 2020468 DHPC8.1_000173 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)OCC=C)c2ccsc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K06 compound treatment 187720.0 18400.0 1.25 183320.0 15100.0 1.13 1.6818 0.9986 3556880 DHPC8.1_000174 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K07 mock treatment 172920.0 3570.0 0.24 172080.0 3890.0 0.29 0.3768 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K08 mock treatment 170000.0 646.0 0.04 171600.0 3410.0 0.25 0.2107 0.8175 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K09 compound treatment 175560.0 6210.0 0.42 173880.0 5690.0 0.42 0.5988 1.0 3556729 DHPC8.1_000175 COc1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K10 compound treatment 177880.0 8530.0 0.58 171400.0 3210.0 0.24 0.5801 0.9229 3556843 DHPC8.1_000176 COc1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K11 compound treatment 173800.0 4450.0 0.3 172960.0 4770.0 0.36 0.4655 0.9969 2019793 DHPC8.1_000177 CC(C)[C@@H]1C[C@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K12 compound treatment 200160.0 30800.0 2.1 196480.0 28300.0 2.11 2.9741 1.0 3556896 DHPC8.1_000178 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)NCc3ccccc3)c4cccs4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K13 compound treatment 178840.0 9490.0 0.65 174120.0 5930.0 0.44 0.7695 0.9827 2020900 DHPC8.1_000179 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)OCC=C)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K14 compound treatment 192040.0 22700.0 1.55 187560.0 19400.0 1.44 2.1132 0.9994 3638682 DHPC8.1_000180 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K15 mock treatment 176200.0 6850.0 0.47 166720.0 -1470.0 -0.11 0.2528 0.5274 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K16 mock treatment 173120.0 3770.0 0.26 167080.0 -1110.0 -0.08 0.1233 0.4571 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K17 compound treatment 174440.0 5090.0 0.35 172560.0 4370.0 0.33 0.4753 0.9995 2020360 DHPC8.1_000181 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)OCC=C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K18 compound treatment 184440.0 15100.0 1.03 182480.0 14300.0 1.06 1.4795 0.9999 3556872 DHPC8.1_000182 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K19 compound treatment 175760.0 6410.0 0.44 172480.0 4290.0 0.32 0.5347 0.9882 3639758 DHPC8.1_000183 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)OCC=C)c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K20 compound treatment 211320.0 42000.0 2.86 205920.0 37700.0 2.81 4.0089 1.0 2020979 DHPC8.1_000184 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccc7OCOc7c6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K21 compound treatment 183040.0 13700.0 0.93 174200.0 6010.0 0.45 0.9762 0.9434 3556742 DHPC8.1_000185 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)OCC=C)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K22 compound treatment 173040.0 3690.0 0.25 171320.0 3130.0 0.23 0.3425 0.9993 3556630 DHPC8.1_000186 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K23 mock treatment 164480.0 -4870.0 -0.33 164880.0 -3310.0 -0.25 -0.409 -0.9891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 K24 mock treatment 161320.0 -8030.0 -0.55 160880.0 -7310.0 -0.54 -0.7719 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L01 compound treatment 211000.0 41600.0 2.84 208120.0 39900.0 2.97 4.1092 0.9997 3557053 DHPC8.1_000187 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5cccs5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L02 mock treatment 167320.0 -2030.0 -0.14 167800.0 -387.0 -0.03 -0.1185 -0.8362 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L03 compound treatment 177480.0 8130.0 0.55 169400.0 1210.0 0.09 0.4555 0.8116 3556907 DHPC8.1_000188 CC(C)[C@H]1C[C@@H](OCCCCO)OC(=C1)C(=O)N2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L04 mock treatment 171360.0 2010.0 0.14 168360.0 173.0 0.01 0.1058 0.7702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L05 compound treatment 183000.0 13600.0 0.93 186440.0 18300.0 1.36 1.6184 0.9829 3641352 DHPC8.1_000189 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L06 mock treatment 174440.0 5090.0 0.35 168400.0 213.0 0.02 0.2564 0.7386 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L07 mock treatment 169280.0 -74.3 -0.01 167680.0 -507.0 -0.04 -0.0303 -0.7948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L08 mock treatment 169640.0 286.0 0.02 171520.0 3330.0 0.25 0.1892 0.7603 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L09 compound treatment 184360.0 15000.0 1.02 181200.0 13000.0 0.97 1.4082 0.9996 2020443 DHPC8.1_000190 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)NCc2ccccc2)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L10 mock treatment 177480.0 8130.0 0.55 170160.0 1970.0 0.15 0.4955 0.8647 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L11 compound treatment 184040.0 14700.0 1.0 182000.0 13800.0 1.03 1.4349 0.9999 3638704 DHPC8.1_000191 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)Nc3ccccc3)c4ccc-5c(Cc6ccccc65)c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L12 mock treatment 174200.0 4850.0 0.33 174600.0 6410.0 0.48 0.5711 0.9839 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L13 compound treatment 180800.0 11400.0 0.78 178080.0 9890.0 0.74 1.0724 0.9996 3556998 DHPC8.1_000192 COc1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L14 mock treatment 174120.0 4770.0 0.32 171400.0 3210.0 0.24 0.3988 0.9886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L15 mock treatment 172360.0 3010.0 0.2 169160.0 973.0 0.07 0.1961 0.9023 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L16 mock treatment 172000.0 2650.0 0.18 172920.0 4730.0 0.35 0.3766 0.9517 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L17 compound treatment 180360.0 11000.0 0.75 177760.0 9570.0 0.71 1.0344 0.9997 3639752 DHPC8.1_000193 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)NCc2ccccc2)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L18 mock treatment 177640.0 8290.0 0.56 165760.0 -2430.0 -0.18 0.2717 0.4581 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L19 compound treatment 176040.0 6690.0 0.46 177240.0 9050.0 0.67 0.7987 0.9819 2019903 DHPC8.1_000194 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)NCc3ccccc3)c4ccsc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L20 mock treatment 166640.0 -2710.0 -0.19 168800.0 613.0 0.05 -0.0986 -0.5174 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L21 compound treatment 178120.0 8770.0 0.6 176680.0 8490.0 0.63 0.8695 0.9996 3557046 DHPC8.1_000195 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L22 mock treatment 164840.0 -4510.0 -0.31 164320.0 -3870.0 -0.29 -0.4212 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L23 mock treatment 162960.0 -6390.0 -0.44 158520.0 -9670.0 -0.72 -0.817 -0.9712 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 L24 mock treatment 154680.0 -14700.0 -1.0 164000.0 -4190.0 -0.31 -0.9278 -0.8854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M01 compound treatment 165680.0 -3670.0 -0.25 169160.0 973.0 0.07 -0.1259 -0.483 2020333 DHPC8.1_000196 CC(C)[C@H]1C[C@@H](OCCCCO)OC(=C1)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M02 compound treatment 193480.0 24100.0 1.64 190360.0 22200.0 1.65 2.33 1.0 3640842 DHPC8.1_000197 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)NCc3ccccc3)c4ccc-5c(Cc6ccccc65)c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M03 compound treatment 175720.0 6370.0 0.43 174080.0 5890.0 0.44 0.617 1.0 2019280 DHPC8.1_000198 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)OCC=C)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M04 compound treatment 223120.0 53800.0 3.67 219360.0 51200.0 3.81 5.2851 0.9998 3556983 DHPC8.1_000199 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5cccs5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M05 compound treatment 182480.0 13100.0 0.89 176440.0 8250.0 0.61 1.0671 0.9831 3556596 DHPC8.1_000200 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)OCC=C)c2csc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M06 compound treatment 227240.0 57900.0 3.95 215000.0 46800.0 3.48 5.2542 0.9981 2020466 DHPC8.1_000201 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccsc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M07 compound treatment 182040.0 12700.0 0.86 174920.0 6730.0 0.5 0.9659 0.9663 2019334 DHPC8.1_000202 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M08 compound treatment 181720.0 12400.0 0.84 180600.0 12400.0 0.92 1.2494 0.999 3557045 DHPC8.1_000203 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccsc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M09 mock treatment 173400.0 4050.0 0.28 174800.0 6610.0 0.49 0.543 0.9625 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M10 mock treatment 176000.0 6650.0 0.45 172960.0 4770.0 0.36 0.5716 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M11 compound treatment 189680.0 20300.0 1.39 186840.0 18700.0 1.39 1.9615 1.0 3556721 DHPC8.1_000204 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)OCC=C)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M12 compound treatment 228400.0 59000.0 4.03 224800.0 56600.0 4.21 5.8259 0.9997 2019926 DHPC8.1_000205 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccsc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M13 mock treatment 177360.0 8010.0 0.55 173080.0 4890.0 0.36 0.6434 0.9806 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M14 mock treatment 175440.0 6090.0 0.41 176440.0 8250.0 0.61 0.7277 0.9818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M15 compound treatment 181640.0 12300.0 0.84 181160.0 13000.0 0.97 1.275 0.9975 3556344 DHPC8.1_000206 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)OCC=C)c2csc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M16 compound treatment 207800.0 38400.0 2.62 204200.0 36000.0 2.68 3.7487 0.9999 2019278 DHPC8.1_000207 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M17 compound treatment 185320.0 16000.0 1.09 180520.0 12300.0 0.92 1.4187 0.9964 3556849 DHPC8.1_000208 COc1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M18 compound treatment 187040.0 17700.0 1.21 189640.0 21500.0 1.6 1.9816 0.9904 3556358 DHPC8.1_000209 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)NCc2ccccc2)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M19 compound treatment 172920.0 3570.0 0.24 179400.0 11200.0 0.83 0.762 0.8767 2019768 DHPC8.1_000210 CC(C)[C@@H]1C[C@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M20 compound treatment 190040.0 20700.0 1.41 183640.0 15500.0 1.15 1.8105 0.9949 3557035 DHPC8.1_000211 COc1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M21 compound treatment 176640.0 7290.0 0.5 180440.0 12300.0 0.91 0.9961 0.9592 3640840 DHPC8.1_000212 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)Nc3ccccc3)c4ccc-5c(Cc6ccccc65)c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M22 compound treatment 180600.0 11200.0 0.77 176640.0 8450.0 0.63 0.987 0.9952 3557039 DHPC8.1_000213 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M23 compound treatment 204240.0 34900.0 2.38 201840.0 33700.0 2.5 3.4528 0.9997 2020956 DHPC8.1_000214 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)NCc3ccccc3)c4ccc5OCOc5c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 M24 compound treatment 170640.0 1290.0 0.09 170200.0 2010.0 0.15 0.1679 0.9674 3557034 DHPC8.1_000215 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccc(OC)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N01 compound treatment 175280.0 5930.0 0.4 173400.0 5210.0 0.39 0.56 0.9998 3557012 DHPC8.1_000216 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)Nc3ccccc3)c4csc5ccccc45)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N02 mock treatment 167000.0 -2350.0 -0.16 169640.0 1450.0 0.11 -0.037 -0.1914 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N03 compound treatment 172440.0 3090.0 0.21 172200.0 4010.0 0.3 0.3599 0.9853 2020848 DHPC8.1_000217 CC(C)[C@H]1C[C@@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N04 mock treatment 173240.0 3890.0 0.26 174080.0 5890.0 0.44 0.4974 0.9709 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N05 compound treatment 171160.0 1810.0 0.12 175520.0 7330.0 0.55 0.473 0.8454 3556985 DHPC8.1_000218 CC(C)[C@@H]1C[C@H](OCc2ccc(CO)cc2)OC(=C1)C(=O)Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N06 mock treatment 175320.0 5970.0 0.41 173360.0 5170.0 0.38 0.5598 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N07 compound treatment 209680.0 40300.0 2.75 218320.0 50100.0 3.73 4.5824 0.9887 3556931 DHPC8.1_000219 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)Nc2ccccc2)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N08 mock treatment 175880.0 6530.0 0.44 178400.0 10200.0 0.76 0.8521 0.9675 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N09 mock treatment 175560.0 6210.0 0.42 174480.0 6290.0 0.47 0.6303 0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N10 mock treatment 181000.0 11600.0 0.79 182680.0 14500.0 1.08 1.3241 0.9886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N11 compound treatment 207520.0 38200.0 2.6 205600.0 37400.0 2.78 3.8089 0.9994 3557018 DHPC8.1_000220 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)NCc3ccccc3)c4cccs4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N12 mock treatment 178120.0 8770.0 0.6 174800.0 6610.0 0.49 0.7706 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N13 mock treatment 180160.0 10800.0 0.74 173720.0 5530.0 0.41 0.8121 0.9622 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N14 mock treatment 173480.0 4130.0 0.28 173680.0 5490.0 0.41 0.488 0.9833 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N15 compound treatment 180440.0 11100.0 0.76 180840.0 12700.0 0.94 1.2003 0.9941 3557010 DHPC8.1_000221 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4ccsc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N16 mock treatment 177640.0 8290.0 0.56 169120.0 933.0 0.07 0.4485 0.7881 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N17 compound treatment 185480.0 16100.0 1.1 185320.0 17100.0 1.28 1.679 0.9973 3557051 DHPC8.1_000222 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N18 mock treatment 175080.0 5730.0 0.39 179320.0 11100.0 0.83 0.8619 0.941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N19 compound treatment 178480.0 9130.0 0.62 179720.0 11500.0 0.86 1.0469 0.9875 3638664 DHPC8.1_000223 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)N3CCCCC3)c4ccc-5c(Cc6ccccc65)c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N20 mock treatment 167520.0 -1830.0 -0.13 171840.0 3650.0 0.27 0.1038 0.3469 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N21 compound treatment 219680.0 50300.0 3.43 212480.0 44300.0 3.3 4.7571 0.9998 2020952 DHPC8.1_000224 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCN(Cc5ccc6OCOc6c5)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N22 mock treatment 173240.0 3890.0 0.26 169280.0 1090.0 0.08 0.2448 0.8835 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N23 compound treatment 202840.0 33500.0 2.28 202360.0 34200.0 2.54 3.4127 0.9985 3556827 DHPC8.1_000225 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 N24 mock treatment 158040.0 -11300.0 -0.77 163960.0 -4230.0 -0.31 -0.7679 -0.9218 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O01 compound treatment 171560.0 2210.0 0.15 171600.0 3410.0 0.25 0.2859 0.9687 3557000 DHPC8.1_000226 COc1ccc(cc1)[C@@H]2C[C@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O02 compound treatment 202880.0 33500.0 2.29 211760.0 43600.0 3.24 3.9094 0.9853 3557028 DHPC8.1_000227 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)Nc2ccccc2)c3ccc4OCOc4c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O03 compound treatment 180360.0 11000.0 0.75 195120.0 26900.0 2.0 1.948 0.9101 3556890 DHPC8.1_000228 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCCCC3)c4cccs4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O04 compound treatment 168280.0 -1070.0 -0.07 174160.0 5970.0 0.44 0.2625 0.5827 3557013 DHPC8.1_000229 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O05 compound treatment 176200.0 6850.0 0.47 171400.0 3210.0 0.24 0.4991 0.9517 3556591 DHPC8.1_000230 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O06 compound treatment 218880.0 49500.0 3.38 223600.0 55400.0 4.12 5.3038 0.9951 2019359 DHPC8.1_000231 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2)c5ccc6OCOc6c5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O07 compound treatment 186640.0 17300.0 1.18 180200.0 12000.0 0.89 1.4655 0.9907 3557037 DHPC8.1_000232 COC(=O)c1ccc(cc1)[C@@H]2C[C@H](OCCCCO)OC(=C2)C(=O)Nc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O08 compound treatment 187120.0 17800.0 1.21 179640.0 11500.0 0.85 1.4592 0.9852 3556948 DHPC8.1_000233 COc1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O09 compound treatment 212840.0 43500.0 2.96 206800.0 38600.0 2.87 4.1285 0.9999 2019876 DHPC8.1_000234 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)NCc3ccccc3)c4ccc5OCOc5c4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O10 compound treatment 172160.0 2810.0 0.19 171160.0 2970.0 0.22 0.2917 0.9974 3556311 DHPC8.1_000235 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCCCC2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O11 mock treatment 170600.0 1250.0 0.08 166320.0 -1870.0 -0.14 -0.0382 -0.2346 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O12 mock treatment 172280.0 2930.0 0.2 166280.0 -1910.0 -0.14 0.0407 0.1661 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O13 compound treatment 221120.0 51800.0 3.53 207520.0 39300.0 2.93 4.5655 0.9957 3640825 DHPC8.1_000236 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccc-7c(Cc8ccccc87)c6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O14 compound treatment 171080.0 1730.0 0.12 179640.0 11500.0 0.85 0.6859 0.7971 3556326 DHPC8.1_000237 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCCCCO)OC(=C2)C(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O15 compound treatment 203840.0 34500.0 2.35 201680.0 33500.0 2.49 3.4251 0.9996 2019251 DHPC8.1_000238 CC(C)[C@@H]1C[C@H](OCCCCO)OC(=C1)C(=O)N2CCN(Cc3ccc4OCOc4c3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O16 compound treatment 173040.0 3690.0 0.25 173680.0 5490.0 0.41 0.4668 0.9727 3556958 DHPC8.1_000239 CNC(=O)C1=C[C@H](C[C@@H](OCCCCO)O1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O17 compound treatment 177520.0 8170.0 0.56 183040.0 14900.0 1.11 1.1753 0.9496 2019795 DHPC8.1_000240 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)NCc3ccccc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O18 compound treatment 203320.0 34000.0 2.32 208360.0 40200.0 2.99 3.7516 0.992 3556884 DHPC8.1_000241 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6csc7ccccc67)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O19 compound treatment 185560.0 16200.0 1.1 185960.0 17800.0 1.32 1.7166 0.996 3557009 DHPC8.1_000242 OCc1ccc(CO[C@H]2C[C@H](C=C(O2)C(=O)Nc3ccccc3)c4ccsc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O20 compound treatment 177920.0 8570.0 0.58 177800.0 9610.0 0.72 0.9188 0.9949 3556869 DHPC8.1_000243 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCCCC3)c4ccsc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O21 compound treatment 176800.0 7450.0 0.51 171680.0 3490.0 0.26 0.5428 0.9517 2020929 DHPC8.1_000244 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)NCc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O22 compound treatment 169600.0 246.0 0.02 165000.0 -3190.0 -0.24 -0.1559 -0.6555 3556441 DHPC8.1_000245 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)N4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O23 compound treatment 164680.0 -4670.0 -0.32 161800.0 -6390.0 -0.48 -0.5615 -0.9811 3557050 DHPC8.1_000246 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCC2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 O24 compound treatment 156440.0 -12900.0 -0.88 158080.0 -10100.0 -0.75 -1.1545 -0.9969 3557038 DHPC8.1_000247 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccc(cc2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P01 compound treatment 175960.0 6610.0 0.45 171960.0 3770.0 0.28 0.517 0.9741 2020875 DHPC8.1_000248 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)NCc3ccccc3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P02 mock treatment 167880.0 -1470.0 -0.1 167600.0 -587.0 -0.04 -0.102 -0.9304 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P03 compound treatment 170360.0 1010.0 0.07 174520.0 6330.0 0.47 0.3818 0.8015 3557005 DHPC8.1_000249 CNC(=O)C1=C[C@@H](C[C@H](OCc2ccc(CO)cc2)O1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P04 mock treatment 162640.0 -6710.0 -0.46 170520.0 2330.0 0.17 -0.2009 -0.4104 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P05 compound treatment 172960.0 3610.0 0.25 174800.0 6610.0 0.49 0.5218 0.9486 3556853 DHPC8.1_000250 COC(=O)c1ccc(cc1)[C@H]2C[C@@H](OCc3ccc(CO)cc3)OC(=C2)C(=O)Nc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P06 mock treatment 163920.0 -5430.0 -0.37 169680.0 1490.0 0.11 -0.1834 -0.4742 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P07 compound treatment 181480.0 12100.0 0.83 180280.0 12100.0 0.9 1.221 0.9991 3556603 DHPC8.1_000251 OCCCCO[C@H]1C[C@H](C=C(O1)C(=O)N2CCCCC2)c3csc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P08 mock treatment 171360.0 2010.0 0.14 162360.0 -5830.0 -0.43 -0.21 -0.4618 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P09 compound treatment 179160.0 9810.0 0.67 173440.0 5250.0 0.39 0.7492 0.9673 3556967 DHPC8.1_000252 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCCCC2)c3ccsc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P10 mock treatment 171120.0 1770.0 0.12 170960.0 2770.0 0.21 0.231 0.9671 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P11 mock treatment 165400.0 -3950.0 -0.27 169000.0 813.0 0.06 -0.1479 -0.5352 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P12 mock treatment 178840.0 9490.0 0.65 175640.0 7450.0 0.55 0.8495 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P13 compound treatment 184520.0 15200.0 1.03 181880.0 13700.0 1.02 1.4517 1.0 2023656 DHPC8.1_000253 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)NCc2ccccc2)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P14 mock treatment 168280.0 -1070.0 -0.07 168480.0 293.0 0.02 -0.0364 -0.4762 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P15 compound treatment 174680.0 5330.0 0.36 174920.0 6730.0 0.5 0.6111 0.9875 3641343 DHPC8.1_000254 OCCCCO[C@@H]1C[C@@H](C=C(O1)C(=O)N2CCCCC2)c3ccc-4c(Cc5ccccc54)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P16 mock treatment 167320.0 -2030.0 -0.14 165720.0 -2470.0 -0.18 -0.2279 -0.9904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P17 compound treatment 210760.0 41400.0 2.82 204400.0 36200.0 2.7 3.9019 0.9997 2021006 DHPC8.1_000255 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3)c6ccsc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P18 mock treatment 170520.0 1170.0 0.08 166400.0 -1790.0 -0.13 -0.0379 -0.2444 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P19 compound treatment 168560.0 -794.0 -0.05 171200.0 3010.0 0.22 0.1203 0.5213 3556431 DHPC8.1_000256 OCc1ccc(CO[C@@H]2C[C@@H](C=C(O2)C(=O)N3CCCCC3)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P20 mock treatment 162800.0 -6550.0 -0.45 165040.0 -3150.0 -0.23 -0.4816 -0.9546 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P21 compound treatment 163000.0 -6350.0 -0.43 161680.0 -6510.0 -0.48 -0.6488 -0.9985 3556859 DHPC8.1_000257 CNC(=O)C1=C[C@H](C[C@@H](OCc2ccc(CO)cc2)O1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P22 mock treatment 162920.0 -6430.0 -0.44 164080.0 -4110.0 -0.31 -0.5263 -0.9844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P23 compound treatment 163360.0 -5990.0 -0.41 160600.0 -7590.0 -0.56 -0.6883 -0.9874 3639726 DHPC8.1_000258 CNC(=O)C1=C[C@@H](C[C@H](OCCCCO)O1)c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2402 P24 mock treatment 156040.0 -13300.0 -0.91 161200.0 -6990.0 -0.52 -1.0096 -0.9651 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A01 compound treatment 164560.0 3490.0 0.24 167040.0 7790.0 0.58 0.5784 0.9226 3213058 CHDI2_000001 NNC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A02 compound treatment 185320.0 24300.0 1.65 174560.0 15300.0 1.14 1.9749 0.9835 3213102 CHDI2_000002 ONC(=O)CCCCCCC(=O)N/N=C/c1c(O)ccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A03 compound treatment 174520.0 13500.0 0.92 156440.0 -2810.0 -0.21 0.5007 0.5323 3213060 CHDI2_000003 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A04 compound treatment 196480.0 35400.0 2.41 189200.0 30000.0 2.23 3.2834 0.9992 3213106 CHDI2_000004 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A05 compound treatment 165800.0 4730.0 0.32 159400.0 152.0 0.01 0.2361 0.7314 3213064 CHDI2_000005 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A06 compound treatment 171000.0 9930.0 0.68 166960.0 7710.0 0.57 0.8846 0.9966 3213110 CHDI2_000006 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc([N+](=O)[O-])c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A07 compound treatment 160560.0 -509.0 -0.03 162280.0 3030.0 0.23 0.135 0.5915 3213068 CHDI2_000007 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A08 compound treatment 185440.0 24400.0 1.66 181320.0 22100.0 1.64 2.3365 1.0 3213114 CHDI2_000008 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(O)ccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A09 compound treatment 165840.0 4770.0 0.33 165360.0 6110.0 0.45 0.5517 0.9865 3213072 CHDI2_000009 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc2OCCOc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A10 compound treatment 161640.0 571.0 0.04 162960.0 3710.0 0.28 0.2229 0.7989 3213118 CHDI2_000010 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)n2ccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A11 compound treatment 169400.0 8330.0 0.57 172440.0 13200.0 0.98 1.0959 0.9662 3213076 CHDI2_000011 ONC(=O)CCCCCCC(=O)N/N=C/COCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A12 compound treatment 167400.0 6330.0 0.43 168360.0 9110.0 0.68 0.7848 0.9762 3213122 CHDI2_000012 ONC(=O)CCCCCCC(=O)N/N=C/c1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A13 compound treatment 196520.0 35500.0 2.42 195480.0 36200.0 2.7 3.6158 0.9985 3214258 CHDI2_000013 ONC(=O)CCCCCC(=O)N/N=C/c1c(O)ccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A14 compound treatment 175120.0 14100.0 0.96 175200.0 16000.0 1.19 1.5169 0.9943 3214354 CHDI2_000014 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A15 compound treatment 208920.0 47900.0 3.26 207120.0 47900.0 3.56 4.8262 0.999 3213080 CHDI2_000015 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A16 compound treatment 186640.0 25600.0 1.74 186880.0 27600.0 2.06 2.6869 0.9966 3213126 CHDI2_000016 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(I)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A17 compound treatment 170160.0 9090.0 0.62 165360.0 6110.0 0.45 0.7599 0.9884 3213084 CHDI2_000017 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A18 compound treatment 166520.0 5450.0 0.37 160760.0 1510.0 0.11 0.3424 0.8817 3213130 CHDI2_000018 C/C=C(/C)\C=N\NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A19 compound treatment 175640.0 14600.0 0.99 168480.0 9230.0 0.69 1.1883 0.9838 3213088 CHDI2_000019 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A20 compound treatment 178400.0 17300.0 1.18 175320.0 16100.0 1.2 1.6813 1.0 3213206 CHDI2_000020 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(s1)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A21 compound treatment 181040.0 20000.0 1.36 175240.0 16000.0 1.19 1.8044 0.9978 3213092 CHDI2_000021 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A22 compound treatment 166840.0 5770.0 0.39 161560.0 2310.0 0.17 0.3999 0.9312 3213138 CHDI2_000022 Cc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A23 mock treatment 161160.0 91.3 0.01 152800.0 -6450.0 -0.48 -0.335 -0.6979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 A24 mock treatment 156680.0 -4390.0 -0.3 152160.0 -7090.0 -0.53 -0.5846 -0.9639 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B01 compound treatment 162440.0 1370.0 0.09 154960.0 -4290.0 -0.32 -0.1596 -0.4798 3213059 CHDI2_000023 NNC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B02 compound treatment 191440.0 30400.0 2.07 210720.0 51500.0 3.83 4.173 0.9583 3213100 CHDI2_000024 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2c(O)ccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B03 compound treatment 169040.0 7970.0 0.54 315200.0 156000.0 11.61 8.5917 0.7394 3213062 CHDI2_000025 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B04 compound treatment 187760.0 26700.0 1.82 190680.0 31400.0 2.34 2.9409 0.9923 3213104 CHDI2_000026 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(O)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B05 compound treatment 159200.0 -1870.0 -0.13 159960.0 712.0 0.05 -0.0526 -0.3814 3213066 CHDI2_000027 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B06 compound treatment 178280.0 17200.0 1.17 183920.0 24700.0 1.84 2.1281 0.9766 3213108 CHDI2_000028 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc([N+](=O)[O-])c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B07 compound treatment 163240.0 2170.0 0.15 164560.0 5310.0 0.4 0.3842 0.9102 3213070 CHDI2_000029 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B08 compound treatment 205720.0 44700.0 3.04 206640.0 47400.0 3.53 4.6467 0.9973 3213112 CHDI2_000030 Oc1ccc([N+](=O)[O-])c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B09 compound treatment 174360.0 13300.0 0.91 169080.0 9830.0 0.73 1.1582 0.9944 3213074 CHDI2_000031 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc3OCCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B10 compound treatment 161880.0 811.0 0.06 160200.0 952.0 0.07 0.0892 0.9925 3213116 CHDI2_000032 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)n3ccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B11 compound treatment 174920.0 13900.0 0.94 173960.0 14700.0 1.09 1.442 0.9973 3213078 CHDI2_000033 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/COCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B12 compound treatment 170960.0 9890.0 0.67 167800.0 8550.0 0.64 0.9269 0.9996 3213120 CHDI2_000034 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B13 compound treatment 366080.0 205000.0 13.98 365720.0 206000.0 15.37 20.7494 0.9989 3214500 CHDI2_000035 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B14 mock treatment 157120.0 -3950.0 -0.27 155640.0 -3610.0 -0.27 -0.3803 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B15 compound treatment 162280.0 1210.0 0.08 158120.0 -1130.0 -0.08 -0.001 -0.0083 3213082 CHDI2_000036 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B16 compound treatment 156360.0 -4710.0 -0.32 157960.0 -1290.0 -0.1 -0.2948 -0.8799 3213124 CHDI2_000037 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(I)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B17 compound treatment 175040.0 14000.0 0.95 168720.0 9470.0 0.7 1.172 0.989 3213086 CHDI2_000038 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B18 compound treatment 166440.0 5370.0 0.37 159880.0 632.0 0.05 0.2922 0.7914 3213128 CHDI2_000039 C/C=C(/C)\C=N\NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B19 compound treatment 167200.0 6130.0 0.42 165720.0 6470.0 0.48 0.6362 0.9975 3213090 CHDI2_000040 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B20 compound treatment 179000.0 17900.0 1.22 176560.0 17300.0 1.29 1.7755 0.9997 3213204 CHDI2_000041 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B21 compound treatment 156880.0 -4190.0 -0.29 152240.0 -7010.0 -0.52 -0.5708 -0.9598 3213094 CHDI2_000042 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B22 compound treatment 164360.0 3290.0 0.22 159000.0 -248.0 -0.02 0.1456 0.6467 3213136 CHDI2_000043 Cc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B23 mock treatment 149560.0 -11500.0 -0.78 151640.0 -7610.0 -0.57 -0.9552 -0.9872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 B24 mock treatment 147920.0 -13100.0 -0.9 147600.0 -11600.0 -0.87 -1.2469 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C01 compound treatment 165920.0 4850.0 0.33 158680.0 -568.0 -0.04 0.204 0.6117 3213144 CHDI2_000044 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(Br)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C02 compound treatment 168600.0 7530.0 0.51 161920.0 2670.0 0.2 0.5037 0.9148 3213186 CHDI2_000045 Cc1ccsc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C03 compound treatment 175080.0 14000.0 0.96 178320.0 19100.0 1.42 1.6792 0.9814 3213148 CHDI2_000046 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C04 compound treatment 173120.0 12100.0 0.82 173600.0 14400.0 1.07 1.3363 0.9916 3213190 CHDI2_000047 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C05 compound treatment 176640.0 15600.0 1.06 172560.0 13300.0 0.99 1.4512 0.9994 3213152 CHDI2_000048 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(O)ccc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C06 compound treatment 171120.0 10100.0 0.69 173720.0 14500.0 1.08 1.2462 0.9762 3213194 CHDI2_000049 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C07 compound treatment 207600.0 46500.0 3.17 212200.0 53000.0 3.94 5.0299 0.9942 3213156 CHDI2_000050 COc1cc(Br)cc(/C=N/NC(=O)CCCCCCC(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C08 compound treatment 190440.0 29400.0 2.0 186200.0 27000.0 2.01 2.8344 1.0 3213202 CHDI2_000051 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc2ccccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C09 compound treatment 169400.0 8330.0 0.57 172320.0 13100.0 0.97 1.0896 0.9672 3213160 CHDI2_000052 COc1ccc(Br)c(/C=N/NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C10 compound treatment 180080.0 19000.0 1.3 178680.0 19400.0 1.45 1.9392 0.9985 3213134 CHDI2_000053 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C11 compound treatment 189880.0 28800.0 1.96 189760.0 30500.0 2.27 2.9947 0.9974 3214262 CHDI2_000054 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C12 compound treatment 174640.0 13600.0 0.93 167160.0 7910.0 0.59 1.0706 0.9762 3214366 CHDI2_000055 ONC(=O)CCCCCC(=O)N/N=C/c1c(F)c(F)c(F)c(F)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C13 compound treatment 168160.0 7090.0 0.48 163880.0 4630.0 0.34 0.5856 0.9863 3213164 CHDI2_000056 COc1ccc(Br)cc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C14 compound treatment 175400.0 14300.0 0.98 176240.0 17000.0 1.26 1.5851 0.9919 3213198 CHDI2_000057 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C15 compound treatment 174960.0 13900.0 0.95 169400.0 10200.0 0.76 1.2039 0.9937 3214266 CHDI2_000058 ONC(=O)CCCCCC(=O)N/N=C/c1ccc([N+](=O)[O-])c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C16 compound treatment 166680.0 5610.0 0.38 162640.0 3390.0 0.25 0.449 0.9796 3214370 CHDI2_000059 ONC(=O)CCCCCC(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C17 compound treatment 165920.0 4850.0 0.33 167880.0 8630.0 0.64 0.6881 0.9523 3213168 CHDI2_000060 ONC(=O)CCCCCCC(=O)N/N=C/c1cc2OCOc2cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C18 compound treatment 171000.0 9930.0 0.68 168840.0 9590.0 0.71 0.9836 0.9997 3213210 CHDI2_000061 ONC(=O)CCCCCCC(=O)N/N=C/c1c(F)c(F)c(F)c(F)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C19 compound treatment 162760.0 1690.0 0.12 160840.0 1590.0 0.12 0.1653 0.9999 3213172 CHDI2_000062 ONC(=O)CCCCCCC(=O)N/N=C/c1cccnc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C20 compound treatment 157480.0 -3590.0 -0.24 156000.0 -3250.0 -0.24 -0.344 -1.0 3213214 CHDI2_000063 ONC(=O)CCCCCCC(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C21 compound treatment 166760.0 5690.0 0.39 173720.0 14500.0 1.08 1.036 0.9049 3213176 CHDI2_000064 ONC(=O)CCCCCCC(=O)N/N=C/c1ccncc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C22 compound treatment 160840.0 -229.0 -0.02 166760.0 7510.0 0.56 0.3843 0.6871 3213218 CHDI2_000065 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C23 mock treatment 151960.0 -9110.0 -0.62 153360.0 -5890.0 -0.44 -0.749 -0.9854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 C24 mock treatment 154360.0 -6710.0 -0.46 150920.0 -8330.0 -0.62 -0.7617 -0.9888 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D01 compound treatment 180680.0 19600.0 1.34 180080.0 20800.0 1.55 2.0418 0.9973 3213146 CHDI2_000066 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(Br)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D02 compound treatment 164560.0 3490.0 0.24 167240.0 7990.0 0.59 0.5889 0.9192 3213184 CHDI2_000067 Cc1ccsc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D03 compound treatment 183040.0 22000.0 1.5 232240.0 73000.0 5.43 4.9006 0.8696 3213150 CHDI2_000068 Oc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D04 compound treatment 161080.0 11.3 0.0 275320.0 116000.0 8.64 6.1091 0.7072 3213188 CHDI2_000069 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)CCCCCCC(=O)Nc3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D05 compound treatment 188120.0 27100.0 1.84 184360.0 25100.0 1.87 2.6257 1.0 3213154 CHDI2_000070 Oc1ccc(Br)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D06 compound treatment 178240.0 17200.0 1.17 181160.0 21900.0 1.63 1.981 0.9868 3213192 CHDI2_000071 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D07 compound treatment 198600.0 37500.0 2.56 201160.0 41900.0 3.12 4.015 0.9952 3213158 CHDI2_000072 COc1cc(Br)cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D08 compound treatment 165280.0 4210.0 0.29 165800.0 6550.0 0.49 0.5478 0.9681 3213200 CHDI2_000073 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D09 compound treatment 181080.0 20000.0 1.36 180000.0 20800.0 1.54 2.0568 0.9981 3213162 CHDI2_000074 COc1ccc(Br)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D10 compound treatment 209880.0 48800.0 3.33 201560.0 42300.0 3.15 4.5799 0.9996 3213132 CHDI2_000075 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D11 compound treatment 262120.0 101000.0 6.89 254000.0 94800.0 7.05 9.8581 0.9999 3214504 CHDI2_000076 ONC(=O)CCCCCC(=O)N/N=C/c1c(O)cc(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D12 mock treatment 161680.0 611.0 0.04 161600.0 2350.0 0.18 0.1532 0.8517 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D13 compound treatment 177960.0 16900.0 1.15 177320.0 18100.0 1.35 1.7654 0.997 3213166 CHDI2_000077 COc1ccc(Br)cc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D14 compound treatment 194600.0 33500.0 2.29 190280.0 31000.0 2.31 3.2496 1.0 3213196 CHDI2_000078 COc1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D15 compound treatment 166000.0 4930.0 0.34 166760.0 7510.0 0.56 0.6331 0.9704 3214508 CHDI2_000079 COc1cc(OC)c(/C=N/NC(=O)CCCCCC(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D16 compound treatment 169480.0 8410.0 0.57 167000.0 7750.0 0.58 0.8135 1.0 3214630 CHDI2_000080 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D17 compound treatment 179160.0 18100.0 1.23 166920.0 7670.0 0.57 1.2759 0.9387 3213170 CHDI2_000081 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc3OCOc3cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D18 compound treatment 176600.0 15500.0 1.06 166080.0 6830.0 0.51 1.1083 0.9435 3213208 CHDI2_000082 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2c(F)c(F)c(F)c(F)c2F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D19 compound treatment 172720.0 11700.0 0.79 168280.0 9030.0 0.67 1.037 0.9965 3213174 CHDI2_000083 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccnc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D20 compound treatment 169160.0 8090.0 0.55 163760.0 4510.0 0.34 0.6275 0.9717 3213212 CHDI2_000084 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D21 compound treatment 166400.0 5330.0 0.36 161200.0 1950.0 0.15 0.3597 0.919 3213178 CHDI2_000085 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccncc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D22 compound treatment 158360.0 -2710.0 -0.18 158840.0 -408.0 -0.03 -0.1521 -0.8125 3213216 CHDI2_000086 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D23 mock treatment 153120.0 -7950.0 -0.54 154680.0 -4570.0 -0.34 -0.6236 -0.9748 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 D24 mock treatment 157800.0 -3270.0 -0.22 151840.0 -7410.0 -0.55 -0.5475 -0.9206 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E01 compound treatment 196480.0 35400.0 2.41 192280.0 33000.0 2.46 3.4455 1.0 3214270 CHDI2_000087 ONC(=O)CCCCCC(=O)N/N=C/c1cc(O)ccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E02 compound treatment 180720.0 19700.0 1.34 176040.0 16800.0 1.25 1.8311 0.9994 3214374 CHDI2_000088 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E03 compound treatment 185240.0 24200.0 1.65 177600.0 18400.0 1.37 2.1311 0.9956 3213224 CHDI2_000089 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(Br)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E04 compound treatment 332520.0 171000.0 11.69 337200.0 178000.0 13.24 17.6306 0.9981 3213262 CHDI2_000090 ONC(=O)CCCCCCC(=O)N/N=C/c1cn(c2ccccc12)S(=O)(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E05 compound treatment 209280.0 48200.0 3.29 207600.0 48400.0 3.6 4.8688 0.999 3213228 CHDI2_000091 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E06 compound treatment 183520.0 22500.0 1.53 173280.0 14000.0 1.04 1.8208 0.9826 3213266 CHDI2_000092 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E07 compound treatment 215800.0 54700.0 3.73 222320.0 63100.0 4.69 5.9578 0.9935 3213232 CHDI2_000093 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E08 compound treatment 175520.0 14500.0 0.99 170320.0 11100.0 0.82 1.2794 0.9961 3213270 CHDI2_000094 ONC(=O)CCCCCCC(=O)N/N=C/c1cccnc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E09 compound treatment 178760.0 17700.0 1.21 177440.0 18200.0 1.35 1.8103 0.9983 3214274 CHDI2_000095 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)n2ccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E10 compound treatment 184840.0 23800.0 1.62 179440.0 20200.0 1.5 2.2086 0.9993 3214378 CHDI2_000096 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(Oc2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E11 compound treatment 180800.0 19700.0 1.35 174000.0 14800.0 1.1 1.7276 0.9949 3213236 CHDI2_000097 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E12 compound treatment 187640.0 26600.0 1.81 184080.0 24800.0 1.85 2.5878 0.9999 3213274 CHDI2_000098 Cc1ncc(CO)c(/C=N/NC(=O)CCCCCCC(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E13 compound treatment 178840.0 17800.0 1.21 172280.0 13000.0 0.97 1.5426 0.9939 3213240 CHDI2_000099 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E14 compound treatment 178120.0 17100.0 1.16 177000.0 17800.0 1.32 1.7563 0.998 3213278 CHDI2_000100 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E15 compound treatment 222440.0 61400.0 4.18 224200.0 65000.0 4.83 6.3769 0.9974 3213244 CHDI2_000101 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E16 compound treatment 184240.0 23200.0 1.58 179360.0 20100.0 1.5 2.1755 0.9996 3213282 CHDI2_000102 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)N2CCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E17 compound treatment 182000.0 20900.0 1.43 181360.0 22100.0 1.65 2.1728 0.9975 3214278 CHDI2_000103 ONC(=O)CCCCCC(=O)N/N=C/c1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E18 compound treatment 269360.0 108000.0 7.38 256480.0 97200.0 7.24 10.3376 0.9999 3214418 CHDI2_000104 ONC(=O)CCCCCC(=O)N/N=C/c1cn(c2ccccc12)S(=O)(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E19 compound treatment 170240.0 9170.0 0.63 172480.0 13200.0 0.98 1.1385 0.976 3213248 CHDI2_000105 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(c1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E20 compound treatment 181400.0 20300.0 1.39 177160.0 17900.0 1.33 1.9228 0.9998 3213286 CHDI2_000106 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E21 compound treatment 179080.0 18000.0 1.23 166280.0 7030.0 0.52 1.2384 0.9277 3213252 CHDI2_000107 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E22 compound treatment 178960.0 17900.0 1.22 176680.0 17400.0 1.3 1.7799 0.9995 3213290 CHDI2_000108 CCCCCCC/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E23 mock treatment 161920.0 851.0 0.06 159480.0 232.0 0.02 0.0532 0.8793 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 E24 mock treatment 160040.0 -1030.0 -0.07 154520.0 -4730.0 -0.35 -0.2984 -0.8317 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F01 compound treatment 167600.0 6530.0 0.45 164680.0 5430.0 0.4 0.6007 0.9988 3214512 CHDI2_000109 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F02 compound treatment 171840.0 10800.0 0.73 169360.0 10100.0 0.75 1.0514 0.9999 3214634 CHDI2_000110 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F03 compound treatment 184920.0 23900.0 1.63 190880.0 31600.0 2.35 2.8145 0.9837 3213226 CHDI2_000111 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(Br)s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F04 compound treatment 216480.0 55400.0 3.78 201640.0 42400.0 3.16 4.9023 0.996 3213260 CHDI2_000112 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cn(c3ccccc23)S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F05 compound treatment 193800.0 32700.0 2.23 194560.0 35300.0 2.63 3.4363 0.9967 3213230 CHDI2_000113 COc1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F06 compound treatment 184800.0 23700.0 1.62 177640.0 18400.0 1.37 2.112 0.9965 3213264 CHDI2_000114 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F07 compound treatment 199000.0 37900.0 2.59 197240.0 38000.0 2.83 3.828 0.999 3213234 CHDI2_000115 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCc3ccccc3)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F08 compound treatment 180320.0 19300.0 1.31 178240.0 19000.0 1.41 1.9276 0.9993 3213268 CHDI2_000116 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F09 compound treatment 179360.0 18300.0 1.25 177080.0 17800.0 1.33 1.8202 0.9995 3214516 CHDI2_000117 CC(C)(C)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F10 compound treatment 175360.0 14300.0 0.97 180440.0 21200.0 1.58 1.8042 0.9732 3214638 CHDI2_000118 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F11 compound treatment 175360.0 14300.0 0.97 179920.0 20700.0 1.54 1.7769 0.9757 3213238 CHDI2_000119 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F12 compound treatment 186760.0 25700.0 1.75 185760.0 26500.0 1.97 2.6338 0.9982 3213272 CHDI2_000120 Cc1ncc(CO)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F13 compound treatment 180960.0 19900.0 1.36 174800.0 15600.0 1.16 1.7774 0.9969 3213242 CHDI2_000121 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F14 compound treatment 178200.0 17100.0 1.17 177320.0 18100.0 1.35 1.7769 0.9975 3213276 CHDI2_000122 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F15 compound treatment 213040.0 52000.0 3.54 208440.0 49200.0 3.66 5.0943 0.9999 3213246 CHDI2_000123 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F16 compound treatment 183680.0 22600.0 1.54 183080.0 23800.0 1.77 2.3443 0.9976 3213280 CHDI2_000124 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)N3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F17 compound treatment 188760.0 27700.0 1.89 183080.0 23800.0 1.77 2.5892 0.9995 3214520 CHDI2_000125 CC1=C(C/C=N/NC(=O)CCCCCC(=O)NO)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F18 compound treatment 175080.0 14000.0 0.96 172080.0 12800.0 0.96 1.3508 1.0 3214641 CHDI2_000126 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F19 compound treatment 170280.0 9210.0 0.63 173600.0 14400.0 1.07 1.1994 0.9679 3213250 CHDI2_000127 OC(=O)c1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F20 compound treatment 191880.0 30800.0 2.1 202400.0 43200.0 3.21 3.7563 0.9788 3213284 CHDI2_000128 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F21 compound treatment 174200.0 13100.0 0.9 167120.0 7870.0 0.59 1.0473 0.9789 3213254 CHDI2_000129 OC(=O)c1ccccc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F22 compound treatment 168080.0 7010.0 0.48 168160.0 8910.0 0.66 0.807 0.9871 3213288 CHDI2_000130 CCCCCCC/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F23 mock treatment 159200.0 -1870.0 -0.13 159400.0 152.0 0.01 -0.0821 -0.6419 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 F24 mock treatment 155560.0 -5510.0 -0.38 154800.0 -4450.0 -0.33 -0.4997 -0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G01 compound treatment 174040.0 13000.0 0.88 175360.0 16100.0 1.2 1.4733 0.9888 3213296 CHDI2_000131 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G02 compound treatment 180320.0 19300.0 1.31 177920.0 18700.0 1.39 1.9107 0.9996 3213336 CHDI2_000132 ONC(=O)CCCCCCC(=O)N/N=C/c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G03 compound treatment 188400.0 27300.0 1.86 188440.0 29200.0 2.17 2.8539 0.9971 3214282 CHDI2_000133 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(I)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G04 compound treatment 182240.0 21200.0 1.44 176960.0 17700.0 1.32 1.9528 0.999 3214422 CHDI2_000134 ONC(=O)CCCCCC(=O)N/N=C/c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G05 compound treatment 176080.0 15000.0 1.02 181760.0 22500.0 1.68 1.9084 0.972 3213300 CHDI2_000135 ONC(=O)CCCCCCC(=O)N/N=C/c1cccnc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G06 compound treatment 188160.0 27100.0 1.85 181880.0 22600.0 1.68 2.4971 0.9989 3213340 CHDI2_000136 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G07 compound treatment 187240.0 26200.0 1.78 184000.0 24800.0 1.84 2.5643 0.9999 3213304 CHDI2_000137 ONC(=O)CCCCCCC(=O)N/N=C/C=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G08 compound treatment 398720.0 238000.0 16.2 375280.0 216000.0 16.08 22.826 1.0 3213344 CHDI2_000138 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G09 compound treatment 195200.0 34100.0 2.33 196440.0 37200.0 2.77 3.6027 0.9963 3213308 CHDI2_000139 C[C@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G10 compound treatment 251600.0 90500.0 6.17 251000.0 91800.0 6.83 9.1931 0.9987 3213348 CHDI2_000140 ONC(=O)CCCCCCC(=O)N/N=C/c1c(O)cc(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G11 compound treatment 190360.0 29300.0 2.0 189520.0 30300.0 2.25 3.0052 0.9982 3213312 CHDI2_000141 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G12 compound treatment 181600.0 20500.0 1.4 178200.0 19000.0 1.41 1.9872 1.0 3213352 CHDI2_000142 COc1cc(OC)c(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G13 compound treatment 185520.0 24500.0 1.67 185520.0 26300.0 1.96 2.5614 0.9968 3213314 CHDI2_000143 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G14 compound treatment 178880.0 17800.0 1.21 180800.0 21600.0 1.6 1.9929 0.9906 3213356 CHDI2_000144 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G15 compound treatment 181920.0 20900.0 1.42 181240.0 22000.0 1.64 2.1626 0.9975 3213318 CHDI2_000145 ONC(=O)CCCCCCC(=O)N/N=C/C1CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G16 compound treatment 176320.0 15300.0 1.04 179160.0 19900.0 1.48 1.7832 0.985 3213360 CHDI2_000146 CC(C)(C)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G17 compound treatment 188760.0 27700.0 1.89 181640.0 22400.0 1.67 2.5134 0.9981 3213322 CHDI2_000147 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G18 compound treatment 185920.0 24900.0 1.69 187360.0 28100.0 2.09 2.6775 0.9945 3213364 CHDI2_000148 CC1=C(C/C=N/NC(=O)CCCCCCC(=O)NO)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G19 compound treatment 182640.0 21600.0 1.47 175160.0 15900.0 1.18 1.8773 0.9942 3214286 CHDI2_000149 C/C=C(/C)\C=N\NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G20 compound treatment 185240.0 24200.0 1.65 179760.0 20500.0 1.53 2.2447 0.9993 3214426 CHDI2_000150 ONC(=O)CCCCCC(=O)N/N=C/c1cccnc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G21 compound treatment 241760.0 80700.0 5.5 234000.0 74800.0 5.56 7.824 1.0 3213326 CHDI2_000151 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(Br)cc(Br)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G22 compound treatment 166680.0 5610.0 0.38 174160.0 14900.0 1.11 1.0553 0.8989 3213368 CHDI2_000152 NC(=O)COc1ccccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G23 mock treatment 164840.0 3770.0 0.26 167160.0 7910.0 0.59 0.5982 0.931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 G24 mock treatment 158920.0 -2150.0 -0.15 164040.0 4790.0 0.36 0.1486 0.3854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H01 compound treatment 179720.0 18700.0 1.27 177200.0 18000.0 1.34 1.8439 0.9997 3213298 CHDI2_000153 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H02 compound treatment 173640.0 12600.0 0.86 168240.0 8990.0 0.67 1.0793 0.9925 3213334 CHDI2_000154 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H03 compound treatment 191320.0 30300.0 2.06 175880.0 16600.0 1.24 2.3337 0.9702 3214524 CHDI2_000155 NC(=O)COc1ccccc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H04 compound treatment 184120.0 23100.0 1.57 177280.0 18000.0 1.34 2.0602 0.9969 3214643 CHDI2_000156 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H05 compound treatment 187000.0 25900.0 1.77 185480.0 26200.0 1.95 2.6306 0.9988 3213302 CHDI2_000157 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccnc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H06 compound treatment 179320.0 18300.0 1.24 319760.0 161000.0 11.95 9.3272 0.7766 3213338 CHDI2_000158 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H07 compound treatment 211960.0 50900.0 3.47 260000.0 101000.0 7.5 7.7557 0.9387 3213306 CHDI2_000159 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/C=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H08 compound treatment 370320.0 209000.0 14.27 373880.0 215000.0 15.97 21.3832 0.9984 3213342 CHDI2_000160 Oc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H09 compound treatment 206000.0 44900.0 3.06 199680.0 40400.0 3.01 4.2939 1.0 3213310 CHDI2_000161 C[C@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H10 compound treatment 249760.0 88700.0 6.05 241800.0 82600.0 6.14 8.6202 1.0 3213346 CHDI2_000162 Oc1cc(O)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H11 compound treatment 193360.0 32300.0 2.2 197800.0 38600.0 2.87 3.5856 0.9914 3213313 CHDI2_000163 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H12 compound treatment 189760.0 28700.0 1.96 189080.0 29800.0 2.22 2.9531 0.998 3213350 CHDI2_000164 COc1cc(OC)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H13 compound treatment 191560.0 30500.0 2.08 185120.0 25900.0 1.93 2.8315 0.9993 3213316 CHDI2_000165 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H14 compound treatment 178200.0 17100.0 1.17 182400.0 23200.0 1.72 2.0443 0.9821 3213354 CHDI2_000166 COc1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H15 compound treatment 179480.0 18400.0 1.26 183160.0 23900.0 1.78 2.146 0.9854 3213320 CHDI2_000167 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/C2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H16 compound treatment 179920.0 18900.0 1.29 180040.0 20800.0 1.55 2.003 0.9957 3213358 CHDI2_000168 CC(C)(C)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H17 compound treatment 181600.0 20500.0 1.4 178480.0 19200.0 1.43 2.0019 0.9999 3213324 CHDI2_000169 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H18 compound treatment 194760.0 33700.0 2.3 192880.0 33600.0 2.5 3.3942 0.9991 3213362 CHDI2_000170 CC1=C(C/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H19 compound treatment 179200.0 18100.0 1.24 179440.0 20200.0 1.5 1.9367 0.9953 3214528 CHDI2_000171 NC(=O)COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H20 compound treatment 176440.0 15400.0 1.05 175080.0 15800.0 1.18 1.5742 0.9983 3214646 CHDI2_000172 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H21 compound treatment 218760.0 57700.0 3.93 212120.0 52900.0 3.94 5.5637 1.0 3213328 CHDI2_000173 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(Br)cc(Br)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H22 compound treatment 180720.0 19700.0 1.34 190240.0 31000.0 2.31 2.5784 0.9666 3213366 CHDI2_000174 NC(=O)COc1ccccc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H23 mock treatment 162840.0 1770.0 0.12 163360.0 4110.0 0.31 0.3018 0.9173 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 H24 mock treatment 162560.0 1490.0 0.1 161160.0 1910.0 0.14 0.1725 0.9864 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I01 compound treatment 181960.0 20900.0 1.42 177720.0 18500.0 1.37 1.9793 0.9998 3213374 CHDI2_000175 COc1cc(Cl)c(/C=N/NC(=O)CCCCCCC(=O)NO)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I02 compound treatment 178240.0 17200.0 1.17 169960.0 10700.0 0.8 1.3915 0.9825 3213415 CHDI2_000176 ONC(=O)CCCCCCC(=O)NN=C1CCCCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I03 compound treatment 223640.0 62600.0 4.27 215280.0 56000.0 4.17 5.9653 0.9999 3213378 CHDI2_000177 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(Cl)cc(Cl)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I04 compound treatment 181120.0 20100.0 1.37 173120.0 13900.0 1.03 1.6967 0.9904 3213417 CHDI2_000178 ONC(=O)CCCCCCC(=O)NN=C1CCCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I05 compound treatment 190680.0 29600.0 2.02 187800.0 28600.0 2.13 2.9301 0.9997 3214362 CHDI2_000179 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(s1)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I06 compound treatment 187160.0 26100.0 1.78 184280.0 25000.0 1.86 2.5752 0.9997 3214430 CHDI2_000180 Cc1ncc(CO)c(/C=N/NC(=O)CCCCCC(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I07 compound treatment 217120.0 56100.0 3.82 216640.0 57400.0 4.27 5.7225 0.9985 3213382 CHDI2_000181 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(Br)cc([N+](=O)[O-])c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I08 compound treatment 178920.0 17900.0 1.22 178560.0 19300.0 1.44 1.8769 0.9966 3213419 CHDI2_000182 ONC(=O)CCCCCCC(=O)NN=C1CCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I09 compound treatment 202800.0 41700.0 2.85 200560.0 41300.0 3.07 4.1859 0.9992 3213386 CHDI2_000183 CCN(CC)c1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I10 mock treatment 176320.0 15300.0 1.04 167280.0 8030.0 0.6 1.1579 0.9654 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I11 compound treatment 189520.0 28500.0 1.94 182960.0 23700.0 1.76 2.6195 0.9989 3213390 CHDI2_000184 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc2OCCc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I12 compound treatment 191160.0 30100.0 2.05 181640.0 22400.0 1.67 2.6291 0.9947 3213422 CHDI2_000185 COc1cc(Br)c(/C=N/NC(=O)CCCCCCC(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I13 compound treatment 339920.0 179000.0 12.19 353440.0 194000.0 14.45 18.842 0.9964 3213394 CHDI2_000186 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I14 compound treatment 190160.0 29100.0 1.98 190840.0 31600.0 2.35 3.065 0.9964 3213426 CHDI2_000187 ONC(=O)CCCCCCC(=O)N/N=C/CCC1CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I15 compound treatment 210080.0 49000.0 3.34 211600.0 52400.0 3.9 5.1179 0.9971 3213398 CHDI2_000188 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I16 compound treatment 255640.0 94600.0 6.45 234840.0 75600.0 5.63 8.5374 0.9977 3213430 CHDI2_000189 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I17 compound treatment 394000.0 233000.0 15.88 394360.0 235000.0 17.5 23.6026 0.9988 3213402 CHDI2_000190 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I18 compound treatment 188920.0 27900.0 1.9 189800.0 30600.0 2.27 2.9505 0.996 3213434 CHDI2_000191 ONC(=O)CCCCCCC(=O)N/N=C/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I19 compound treatment 258720.0 97700.0 6.66 257080.0 97800.0 7.28 9.8563 0.999 3213406 CHDI2_000192 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I20 mock treatment 176680.0 15600.0 1.06 173040.0 13800.0 1.03 1.4784 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I21 compound treatment 183840.0 22800.0 1.55 177120.0 17900.0 1.33 2.0383 0.997 3214294 CHDI2_000193 Cc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I22 compound treatment 166080.0 5010.0 0.34 168600.0 9350.0 0.7 0.7337 0.9463 3214434 CHDI2_000194 ONC(=O)CCCCCC(=O)N/N=C/c1ccc[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I23 mock treatment 162480.0 1410.0 0.1 159840.0 592.0 0.04 0.0992 0.9373 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 I24 mock treatment 160160.0 -909.0 -0.06 156040.0 -3210.0 -0.24 -0.2126 -0.862 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J01 compound treatment 210360.0 49300.0 3.36 197200.0 38000.0 2.82 4.3736 0.9963 3213376 CHDI2_000195 COc1cc(Cl)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J02 compound treatment 178040.0 17000.0 1.16 176200.0 17000.0 1.26 1.7103 0.9991 3213414 CHDI2_000196 Oc1ccccc1NC(=O)CCCCCCC(=O)NN=C2CCCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J03 compound treatment 213080.0 52000.0 3.55 207720.0 48500.0 3.61 5.0583 1.0 3213380 CHDI2_000197 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J04 compound treatment 185320.0 24300.0 1.65 181400.0 22200.0 1.65 2.3349 1.0 3213416 CHDI2_000198 Oc1ccccc1NC(=O)CCCCCCC(=O)NN=C2CCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J05 compound treatment 181760.0 20700.0 1.41 237680.0 78400.0 5.84 5.1252 0.8534 3214571 CHDI2_000199 ONC(=O)CCCCCC(=O)NN=C1CCCCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J06 compound treatment 186040.0 25000.0 1.7 365840.0 207000.0 15.38 12.0763 0.7806 3214650 CHDI2_000200 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(Oc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J07 compound treatment 202520.0 41500.0 2.83 201840.0 42600.0 3.17 4.2398 0.9984 3213384 CHDI2_000201 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(Br)cc([N+](=O)[O-])c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J08 compound treatment 182120.0 21100.0 1.44 196760.0 37500.0 2.79 2.989 0.9522 3213418 CHDI2_000202 Oc1ccccc1NC(=O)CCCCCCC(=O)NN=C2CCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J09 compound treatment 214520.0 53500.0 3.64 214240.0 55000.0 4.09 5.4709 0.9983 3213388 CHDI2_000203 CCN(CC)c1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J10 mock treatment 169120.0 8050.0 0.55 175720.0 16500.0 1.23 1.255 0.9343 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J11 compound treatment 186960.0 25900.0 1.77 181120.0 21900.0 1.63 2.3992 0.9992 3213392 CHDI2_000204 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc3OCCc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J12 compound treatment 188800.0 27700.0 1.89 188440.0 29200.0 2.17 2.8732 0.9976 3213420 CHDI2_000205 COc1cc(Br)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J13 compound treatment 251720.0 90700.0 6.18 239520.0 80300.0 5.97 8.5947 0.9999 3213396 CHDI2_000206 Oc1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J14 compound treatment 185640.0 24600.0 1.68 183960.0 24700.0 1.84 2.4851 0.9989 3213424 CHDI2_000207 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/CCC2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J15 compound treatment 205400.0 44300.0 3.02 199400.0 40200.0 2.99 4.2502 1.0 3213400 CHDI2_000208 Oc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J16 compound treatment 180560.0 19500.0 1.33 176640.0 17400.0 1.29 1.8549 0.9999 3213428 CHDI2_000209 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J17 compound treatment 355080.0 194000.0 13.23 349080.0 190000.0 14.13 19.3434 0.9995 3213404 CHDI2_000210 Oc1ccc(O)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J18 compound treatment 190600.0 29500.0 2.01 186920.0 27700.0 2.06 2.88 0.9999 3213432 CHDI2_000211 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J19 compound treatment 267120.0 106000.0 7.23 264080.0 105000.0 7.8 10.6296 0.9993 3213408 CHDI2_000212 Oc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J20 mock treatment 171960.0 10900.0 0.74 171320.0 12100.0 0.9 1.1604 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J21 compound treatment 172240.0 11200.0 0.76 169360.0 10100.0 0.75 1.0707 1.0 3214573 CHDI2_000213 ONC(=O)CCCCCC(=O)NN=C1CCCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J22 compound treatment 165880.0 4810.0 0.33 163480.0 4230.0 0.31 0.4547 0.9998 3214654 CHDI2_000214 ONC(=O)CCCCCC(=O)N/N=C/c1cc[n+]([O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J23 mock treatment 159960.0 -1110.0 -0.08 160600.0 1350.0 0.1 0.0177 0.1406 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 J24 mock treatment 159120.0 -1950.0 -0.13 155520.0 -3730.0 -0.28 -0.2902 -0.9431 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K01 compound treatment 172680.0 11600.0 0.79 172960.0 13700.0 1.02 1.2814 0.9921 3213436 CHDI2_000215 COc1cccc(OC)c1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K02 compound treatment 175920.0 14900.0 1.01 168400.0 9150.0 0.68 1.1976 0.9814 3213474 CHDI2_000216 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K03 compound treatment 175720.0 14700.0 1.0 178040.0 18800.0 1.4 1.6953 0.9864 3213440 CHDI2_000217 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K04 compound treatment 177280.0 16200.0 1.11 169920.0 10700.0 0.79 1.3432 0.9869 3213478 CHDI2_000218 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K05 compound treatment 178400.0 17300.0 1.18 172240.0 13000.0 0.97 1.5192 0.995 3213444 CHDI2_000219 COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K06 compound treatment 175120.0 14100.0 0.96 181680.0 22400.0 1.67 1.8579 0.9652 3213482 CHDI2_000220 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K07 compound treatment 183880.0 22800.0 1.56 183800.0 24600.0 1.83 2.3918 0.9968 3214298 CHDI2_000221 Cc1[nH]cnc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K08 compound treatment 187760.0 26700.0 1.82 189600.0 30400.0 2.26 2.8841 0.9943 3214438 CHDI2_000222 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)N2CCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K09 compound treatment 182280.0 21200.0 1.45 180240.0 21000.0 1.56 2.1273 0.9993 3213448 CHDI2_000223 CC1(C)COC(CCC/C=N/NC(=O)CCCCCCC(=O)NO)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K10 compound treatment 179840.0 18800.0 1.28 179280.0 20000.0 1.49 1.9592 0.9971 3213485 CHDI2_000224 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K11 compound treatment 192880.0 31800.0 2.17 192040.0 32800.0 2.44 3.2593 0.9983 3213452 CHDI2_000225 Cc1nnc(Sc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K12 compound treatment 178600.0 17500.0 1.2 178080.0 18800.0 1.4 1.8362 0.9969 3213487 CHDI2_000226 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K13 compound treatment 188720.0 27700.0 1.89 188640.0 29400.0 2.19 2.8798 0.9973 3213456 CHDI2_000227 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(Br)cs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K14 compound treatment 178000.0 16900.0 1.15 175360.0 16100.0 1.2 1.6642 0.9998 3213490 CHDI2_000228 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K15 compound treatment 185760.0 24700.0 1.68 181200.0 22000.0 1.63 2.3456 0.9999 3214342 CHDI2_000229 Cc1ccsc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K16 compound treatment 189000.0 27900.0 1.9 183120.0 23900.0 1.78 2.6028 0.9994 3214442 CHDI2_000230 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K17 compound treatment 181840.0 20800.0 1.42 184320.0 25100.0 1.87 2.3208 0.9907 3213460 CHDI2_000231 CC(C)(C)OC(=O)NC/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K18 compound treatment 221120.0 60100.0 4.09 219520.0 60300.0 4.49 6.0669 0.999 3213494 CHDI2_000232 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(Oc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K19 compound treatment 254080.0 93000.0 6.34 248360.0 89100.0 6.63 9.1737 0.9997 3213464 CHDI2_000233 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc-2c(Cc3ccccc32)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K20 compound treatment 184480.0 23400.0 1.6 168400.0 9150.0 0.68 1.6103 0.9279 3213498 CHDI2_000234 ONC(=O)CCCCCCC(=O)N/N=C/c1cc[n+]([O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K21 compound treatment 176280.0 15200.0 1.04 173160.0 13900.0 1.04 1.4655 1.0 3213468 CHDI2_000235 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K22 compound treatment 177680.0 16600.0 1.13 175760.0 16500.0 1.23 1.6698 0.9992 3213502 CHDI2_000236 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc2ccccc2n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K23 mock treatment 165920.0 4850.0 0.33 156280.0 -2970.0 -0.22 0.0777 0.1953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 K24 mock treatment 157760.0 -3310.0 -0.23 154360.0 -4890.0 -0.36 -0.4168 -0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L01 compound treatment 179480.0 18400.0 1.26 175320.0 16100.0 1.2 1.7334 0.9997 3213438 CHDI2_000237 COc1cccc(OC)c1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L02 compound treatment 172120.0 11100.0 0.75 167560.0 8310.0 0.62 0.9702 0.9952 3213472 CHDI2_000238 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L03 compound treatment 181000.0 19900.0 1.36 181160.0 21900.0 1.63 2.114 0.9959 3213442 CHDI2_000239 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L04 compound treatment 176160.0 15100.0 1.03 192160.0 32900.0 2.45 2.4596 0.9258 3213476 CHDI2_000240 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L05 compound treatment 205480.0 44400.0 3.03 378040.0 219000.0 16.28 13.6555 0.8245 3213446 CHDI2_000241 COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L06 compound treatment 179480.0 18400.0 1.26 199920.0 40700.0 3.03 3.028 0.924 3213480 CHDI2_000242 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L07 compound treatment 183120.0 22100.0 1.5 185040.0 25800.0 1.92 2.4204 0.9927 3214575 CHDI2_000243 ONC(=O)CCCCCC(=O)NN=C1CCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L08 compound treatment 185760.0 24700.0 1.68 179680.0 20400.0 1.52 2.2656 0.9987 3214658 CHDI2_000244 ONC(=O)CCCCCC(=O)N/N=C/c1ccc2ccccc2n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L09 compound treatment 177800.0 16700.0 1.14 180200.0 21000.0 1.56 1.9092 0.9882 3213450 CHDI2_000245 CC1(C)COC(CCC/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L10 compound treatment 175760.0 14700.0 1.0 179080.0 19800.0 1.48 1.7519 0.9822 3213484 CHDI2_000246 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L11 compound treatment 191720.0 30700.0 2.09 192160.0 32900.0 2.45 3.2097 0.9969 3213454 CHDI2_000247 Cc1nnc(Sc2ccc(/C=N/NC(=O)CCCCCCC(=O)Nc3ccccc3O)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L12 compound treatment 183120.0 22100.0 1.5 179320.0 20100.0 1.49 2.1194 1.0 3213486 CHDI2_000248 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L13 compound treatment 183280.0 22200.0 1.51 180600.0 21400.0 1.59 2.1945 0.9997 3213458 CHDI2_000249 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(Br)cs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L14 compound treatment 175320.0 14300.0 0.97 173960.0 14700.0 1.09 1.4613 0.9982 3213488 CHDI2_000250 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L15 mock treatment 169680.0 8610.0 0.59 166400.0 7150.0 0.53 0.7915 0.9988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L16 compound treatment 179640.0 18600.0 1.27 173520.0 14300.0 1.06 1.6464 0.9962 3214702 CHDI2_000251 Cc1ccccc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L17 compound treatment 183160.0 22100.0 1.51 179920.0 20700.0 1.54 2.1529 0.9999 3213462 CHDI2_000252 CC(C)(C)OC(=O)NC/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L18 compound treatment 178680.0 17600.0 1.2 176120.0 16900.0 1.26 1.7369 0.9997 3213492 CHDI2_000253 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(Oc3ccccc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L19 compound treatment 175480.0 14400.0 0.98 169560.0 10300.0 0.77 1.2374 0.9925 3213466 CHDI2_000254 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L20 compound treatment 176320.0 15300.0 1.04 172640.0 13400.0 1.0 1.44 0.9998 3213496 CHDI2_000255 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc[n+]([O-])cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L21 compound treatment 171040.0 9970.0 0.68 166880.0 7630.0 0.57 0.8823 0.996 3213470 CHDI2_000256 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(F)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L22 compound treatment 200520.0 39500.0 2.69 184840.0 25600.0 1.9 3.2487 0.9857 3213500 CHDI2_000257 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L23 mock treatment 163640.0 2570.0 0.18 159320.0 71.8 0.01 0.1277 0.7283 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 L24 mock treatment 159560.0 -1510.0 -0.1 159320.0 71.8 0.01 -0.069 -0.6695 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M01 compound treatment 188480.0 27400.0 1.87 185880.0 26600.0 1.98 2.723 0.9996 3213504 CHDI2_000258 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M02 compound treatment 180800.0 19700.0 1.35 181320.0 22100.0 1.64 2.1128 0.9951 3213546 CHDI2_000259 Cc1ccccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M03 compound treatment 200720.0 39700.0 2.7 201200.0 42000.0 3.12 4.1194 0.9974 3213508 CHDI2_000260 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(F)c(Oc2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M04 compound treatment 215320.0 54300.0 3.7 211760.0 52500.0 3.91 5.3789 0.9996 3213550 CHDI2_000261 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M05 compound treatment 203000.0 41900.0 2.86 195640.0 36400.0 2.71 3.9367 0.9996 3213512 CHDI2_000262 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(F)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M06 compound treatment 187360.0 26300.0 1.79 187760.0 28500.0 2.12 2.768 0.9965 3213554 CHDI2_000263 ONC(=O)CCCCCCC(=O)N/N=C/[C@H](O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M07 compound treatment 222160.0 61100.0 4.17 226960.0 67700.0 5.04 6.5086 0.9955 3213516 CHDI2_000264 ONC(=O)CCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M08 compound treatment 186280.0 25200.0 1.72 182600.0 23400.0 1.74 2.4443 1.0 3213557 CHDI2_000265 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M09 compound treatment 187040.0 26000.0 1.77 187800.0 28600.0 2.13 2.7546 0.9959 3214350 CHDI2_000266 ONC(=O)CCCCCC(=O)N/N=C/c1cccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M10 compound treatment 180480.0 19400.0 1.32 181080.0 21800.0 1.62 2.0847 0.9948 3214450 CHDI2_000267 ONC(=O)CCCCCC(=O)N/N=C/c1nccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M11 compound treatment 187920.0 26900.0 1.83 184040.0 24800.0 1.85 2.5992 1.0 3213520 CHDI2_000268 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M12 compound treatment 192280.0 31200.0 2.13 184720.0 25500.0 1.9 2.8452 0.9983 3213560 CHDI2_000269 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M13 compound treatment 190520.0 29500.0 2.01 188040.0 28800.0 2.14 2.935 0.9995 3214358 CHDI2_000270 ONC(=O)CCCCCC(=O)N/N=C/c1ccc2ccccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M14 compound treatment 183400.0 22300.0 1.52 186760.0 27500.0 2.05 2.5244 0.9894 3214492 CHDI2_000271 ONC(=O)CCCCCC(=O)N/N=C/c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M15 compound treatment 184600.0 23500.0 1.6 183840.0 24600.0 1.83 2.4286 0.9978 3213524 CHDI2_000272 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(c1)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M16 compound treatment 184920.0 23900.0 1.63 183640.0 24400.0 1.82 2.4335 0.9985 3213564 CHDI2_000273 CCOc1cccc(/C=N/NC(=O)CCCCCCC(=O)NO)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M17 compound treatment 192200.0 31100.0 2.12 191480.0 32200.0 2.4 3.1971 0.9981 3213528 CHDI2_000274 ONC(=O)CCCCCCC(=O)N/N=C/c1ccco1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M18 compound treatment 243520.0 82500.0 5.62 246480.0 87200.0 6.49 8.5657 0.9974 3213568 CHDI2_000275 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(I)cc(I)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M19 compound treatment 170960.0 9890.0 0.67 172360.0 13100.0 0.98 1.1669 0.9837 3213532 CHDI2_000276 ONC(=O)CCCCCCC(=O)N/N=C/c1ccoc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M20 compound treatment 173000.0 11900.0 0.81 171520.0 12300.0 0.91 1.221 0.9983 3213572 CHDI2_000277 CN(C)c1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M21 compound treatment 182520.0 21500.0 1.46 178600.0 19400.0 1.44 2.0526 1.0 3213536 CHDI2_000278 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M22 compound treatment 244840.0 83800.0 5.71 242120.0 82900.0 6.17 8.3998 0.9993 3213576 CHDI2_000279 CCn1c2ccccc2c3cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M23 mock treatment 168360.0 7290.0 0.5 172320.0 13100.0 0.97 1.0394 0.9514 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 M24 mock treatment 160000.0 -1070.0 -0.07 160760.0 1510.0 0.11 0.028 0.2092 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N01 compound treatment 192360.0 31300.0 2.13 195320.0 36100.0 2.68 3.4069 0.9935 3213506 CHDI2_000280 Oc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N02 compound treatment 180520.0 19500.0 1.33 179800.0 20600.0 1.53 2.0193 0.9975 3213544 CHDI2_000281 Cc1ccccc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N03 compound treatment 176480.0 15400.0 1.05 176760.0 17500.0 1.3 1.6646 0.9943 3213510 CHDI2_000282 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(F)c(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N04 compound treatment 199560.0 38500.0 2.62 193520.0 34300.0 2.55 3.6592 0.9999 3213548 CHDI2_000283 COc1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N05 compound treatment 201480.0 40400.0 2.76 200560.0 41300.0 3.07 4.1223 0.9985 3213514 CHDI2_000284 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(F)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N06 compound treatment 186800.0 25700.0 1.75 315280.0 156000.0 11.61 9.4521 0.8048 3213552 CHDI2_000285 O[C@@H](/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N07 compound treatment 207920.0 46900.0 3.19 352280.0 193000.0 14.37 12.4175 0.8437 3213518 CHDI2_000286 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N08 compound treatment 184520.0 23500.0 1.6 184680.0 25400.0 1.89 2.469 0.9965 3213556 CHDI2_000287 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N09 compound treatment 194760.0 33700.0 2.3 189480.0 30200.0 2.25 3.2152 0.9999 3214582 CHDI2_000288 ONC(=O)CCCCCC(=O)N/N=C/CCC1CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N10 compound treatment 186240.0 25200.0 1.72 187160.0 27900.0 2.08 2.6824 0.9955 3214710 CHDI2_000289 ONC(=O)CCCCCC(=O)N/N=C/[C@H](O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N11 compound treatment 198320.0 37300.0 2.54 199240.0 40000.0 2.98 3.9005 0.9969 3213522 CHDI2_000290 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N12 compound treatment 197400.0 36300.0 2.48 196480.0 37200.0 2.77 3.7109 0.9984 3213558 CHDI2_000291 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N13 compound treatment 257040.0 96000.0 6.54 249320.0 90100.0 6.7 9.3669 0.9999 3214586 CHDI2_000292 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N14 compound treatment 184000.0 22900.0 1.56 177400.0 18200.0 1.35 2.0608 0.9974 3214713 CHDI2_000293 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N15 compound treatment 186920.0 25900.0 1.76 182280.0 23000.0 1.71 2.4584 0.9999 3213526 CHDI2_000294 OB(O)c1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N16 compound treatment 176000.0 14900.0 1.02 178400.0 19200.0 1.43 1.7277 0.9864 3213562 CHDI2_000295 CCOc1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N17 compound treatment 182800.0 21700.0 1.48 182000.0 22800.0 1.69 2.245 0.9978 3213530 CHDI2_000296 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N18 compound treatment 211640.0 50600.0 3.45 210440.0 51200.0 3.81 5.1321 0.9988 3213566 CHDI2_000297 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(I)cc(I)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N19 compound treatment 179960.0 18900.0 1.29 184600.0 25400.0 1.89 2.2449 0.9827 3213534 CHDI2_000298 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccoc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N20 compound treatment 179640.0 18600.0 1.27 170320.0 11100.0 0.82 1.478 0.9784 3213570 CHDI2_000299 CN(C)c1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N21 compound treatment 194880.0 33800.0 2.31 179280.0 20000.0 1.49 2.6842 0.9778 3213538 CHDI2_000300 Oc1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N22 compound treatment 173520.0 12500.0 0.85 172480.0 13200.0 0.98 1.2966 0.9973 3213574 CHDI2_000301 CCn1c2ccccc2c3cc(/C=N/NC(=O)CCCCCCC(=O)Nc4ccccc4O)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N23 mock treatment 163480.0 2410.0 0.16 163360.0 4110.0 0.31 0.3326 0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 N24 mock treatment 161280.0 211.0 0.01 159240.0 -8.21 0.0 0.0098 0.6765 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O01 compound treatment 171360.0 10300.0 0.7 170160.0 10900.0 0.81 1.0704 0.9973 3213582 CHDI2_000302 OCCOc1ccccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O02 compound treatment 167440.0 6370.0 0.43 172200.0 13000.0 0.96 0.9888 0.9352 3213628 CHDI2_000303 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(o1)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O03 compound treatment 172920.0 11900.0 0.81 170480.0 11200.0 0.84 1.1624 0.9999 3213586 CHDI2_000304 OCCOc1cccc(/C=N/NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O04 compound treatment 178600.0 17500.0 1.2 177400.0 18200.0 1.35 1.8004 0.9981 3213632 CHDI2_000305 Cn1cc(/C=N/NC(=O)CCCCCCC(=O)NO)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O05 compound treatment 184160.0 23100.0 1.57 172720.0 13500.0 1.0 1.8222 0.9763 3213590 CHDI2_000306 OCCOc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O06 compound treatment 200480.0 39400.0 2.69 206920.0 47700.0 3.55 4.4088 0.9906 3213636 CHDI2_000307 ONC(=O)CCCCCCC(=O)N/N=C/c1cn(Cc2ccccc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O07 compound treatment 200880.0 39800.0 2.71 199960.0 40700.0 3.03 4.0618 0.9985 3213594 CHDI2_000308 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O08 compound treatment 178080.0 17000.0 1.16 178360.0 19100.0 1.42 1.8259 0.9949 3213640 CHDI2_000309 ONC(=O)CCCCCCC(=O)N/N=C/C1=CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O09 compound treatment 195680.0 34600.0 2.36 197560.0 38300.0 2.85 3.6848 0.9956 3213598 CHDI2_000310 COc1ccc(O)c(/C=N/NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O10 compound treatment 171440.0 10400.0 0.71 177400.0 18200.0 1.35 1.4553 0.9544 3213643 CHDI2_000311 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O11 compound treatment 195200.0 34100.0 2.33 194920.0 35700.0 2.65 3.5227 0.9978 3214290 CHDI2_000312 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O12 compound treatment 185480.0 24400.0 1.66 180600.0 21400.0 1.59 2.3005 0.9997 3214496 CHDI2_000313 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O13 compound treatment 203800.0 42700.0 2.91 199480.0 40200.0 2.99 4.1773 0.9999 3213602 CHDI2_000314 COc1cc(/C=C/C=N/NC(=O)CCCCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O14 compound treatment 174760.0 13700.0 0.93 175240.0 16000.0 1.19 1.5016 0.9928 3213646 CHDI2_000315 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O15 compound treatment 185560.0 24500.0 1.67 189720.0 30500.0 2.27 2.7843 0.9887 3213606 CHDI2_000316 Cc1ccc(O)c(/C=N/NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O16 compound treatment 169240.0 8170.0 0.56 173080.0 13800.0 1.03 1.1219 0.9584 3213650 CHDI2_000317 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)NO)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O17 compound treatment 174880.0 13800.0 0.94 178240.0 19000.0 1.41 1.6653 0.9805 3213610 CHDI2_000318 OCc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O18 compound treatment 176040.0 15000.0 1.02 176520.0 17300.0 1.29 1.6307 0.9935 3213654 CHDI2_000319 C/C(=N\NC(=O)CCCCCCC(=O)NO)/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O19 compound treatment 239520.0 78500.0 5.35 230440.0 71200.0 5.3 7.5287 1.0 3213614 CHDI2_000320 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc2ccccc2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O20 compound treatment 173440.0 12400.0 0.84 163440.0 4190.0 0.31 0.817 0.9085 3213658 CHDI2_000321 CN(C)CCCOc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O21 compound treatment 230920.0 69900.0 4.76 225560.0 66300.0 4.94 6.8573 0.9998 3213618 CHDI2_000322 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(o1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O22 compound treatment 194280.0 33200.0 2.26 190080.0 30800.0 2.29 3.2237 1.0 3213662 CHDI2_000323 CCOc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O23 mock treatment 163800.0 2730.0 0.19 157120.0 -2130.0 -0.16 0.0197 0.0805 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 O24 mock treatment 155720.0 -5350.0 -0.36 156760.0 -2490.0 -0.19 -0.3888 -0.9506 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P01 compound treatment 184320.0 23300.0 1.59 173520.0 14300.0 1.06 1.872 0.981 3213584 CHDI2_000324 OCCOc1ccccc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P02 compound treatment 179120.0 18100.0 1.23 175280.0 16000.0 1.19 1.7139 0.9999 3213626 CHDI2_000325 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(o2)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P03 compound treatment 178000.0 16900.0 1.15 179080.0 19800.0 1.48 1.8599 0.9926 3213588 CHDI2_000326 OCCOc1cccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P04 compound treatment 182160.0 21100.0 1.44 189200.0 30000.0 2.23 2.5931 0.9775 3213630 CHDI2_000327 Cn1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P05 compound treatment 175640.0 14600.0 0.99 185480.0 26200.0 1.95 2.083 0.9509 3213592 CHDI2_000328 OCCOc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P06 compound treatment 193760.0 32700.0 2.23 233760.0 74500.0 5.55 5.4974 0.9198 3213634 CHDI2_000329 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cn(Cc3ccccc3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P07 compound treatment 202440.0 41400.0 2.82 385840.0 227000.0 16.86 13.9195 0.8141 3213596 CHDI2_000330 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P08 compound treatment 174160.0 13100.0 0.89 246240.0 87000.0 6.47 5.2093 0.797 3213638 CHDI2_000331 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/C2=CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P09 compound treatment 196280.0 35200.0 2.4 196720.0 37500.0 2.79 3.6695 0.9972 3213600 CHDI2_000332 COc1ccc(O)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P10 compound treatment 173760.0 12700.0 0.87 183960.0 24700.0 1.84 1.9124 0.9408 3213642 CHDI2_000333 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P11 compound treatment 178040.0 17000.0 1.16 180760.0 21500.0 1.6 1.9503 0.9873 3214590 CHDI2_000334 ONC(=O)CCCCCC(=O)N/N=C/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P12 compound treatment 189600.0 28500.0 1.95 191920.0 32700.0 2.43 3.0949 0.9939 3214716 CHDI2_000335 COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P13 compound treatment 199240.0 38200.0 2.6 202280.0 43000.0 3.2 4.1048 0.9947 3213604 CHDI2_000336 COc1cc(/C=C/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P14 compound treatment 172680.0 11600.0 0.79 174480.0 15200.0 1.13 1.3614 0.9846 3213644 CHDI2_000337 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P15 compound treatment 199520.0 38500.0 2.62 200840.0 41600.0 3.1 4.0426 0.9966 3213608 CHDI2_000338 Cc1ccc(O)c(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P16 compound treatment 174800.0 13700.0 0.94 170720.0 11500.0 0.85 1.2657 0.9989 3213648 CHDI2_000339 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P17 compound treatment 189360.0 28300.0 1.93 187640.0 28400.0 2.11 2.8581 0.999 3213612 CHDI2_000340 OCc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P18 compound treatment 176600.0 15500.0 1.06 175360.0 16100.0 1.2 1.5967 0.9981 3213652 CHDI2_000341 C/C(=N\NC(=O)CCCCCCC(=O)Nc1ccccc1O)/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P19 compound treatment 218360.0 57300.0 3.91 215360.0 56100.0 4.18 5.715 0.9994 3213616 CHDI2_000342 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc3ccccc3c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P20 compound treatment 173440.0 12400.0 0.84 168280.0 9030.0 0.67 1.0717 0.9937 3213656 CHDI2_000343 CN(C)CCCOc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P21 compound treatment 177280.0 16200.0 1.11 194040.0 34800.0 2.59 2.6125 0.9279 3213620 CHDI2_000344 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(o2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P22 compound treatment 197440.0 36400.0 2.48 199840.0 40600.0 3.02 3.8897 0.9952 3213660 CHDI2_000345 CCOc1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P23 mock treatment 154400.0 -6670.0 -0.45 155160.0 -4090.0 -0.3 -0.5366 -0.9809 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2403 P24 mock treatment 165040.0 3970.0 0.27 154760.0 -4490.0 -0.33 -0.0448 -0.1041 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A01 compound treatment 165880.0 9500.0 0.65 163600.0 9010.0 0.67 0.932 0.9999 3214214 CHDI2_000346 NNC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A02 compound treatment 160880.0 4500.0 0.31 162360.0 7770.0 0.58 0.6257 0.9561 3214215 CHDI2_000347 NNC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A03 compound treatment 171080.0 14700.0 1.0 166280.0 11700.0 0.87 1.3237 0.9975 3214216 CHDI2_000348 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A04 compound treatment 179800.0 23400.0 1.6 168600.0 14000.0 1.04 1.8662 0.9786 3214218 CHDI2_000349 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A05 compound treatment 167720.0 11300.0 0.77 164560.0 9970.0 0.74 1.0712 0.9998 3214220 CHDI2_000350 COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A06 compound treatment 164120.0 7740.0 0.53 164040.0 9450.0 0.7 0.8703 0.99 3214222 CHDI2_000351 COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A07 compound treatment 159800.0 3420.0 0.23 162800.0 8210.0 0.61 0.5967 0.9129 3214224 CHDI2_000352 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A08 compound treatment 160120.0 3740.0 0.26 163600.0 9010.0 0.67 0.6543 0.9124 3214226 CHDI2_000353 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A09 compound treatment 163440.0 7060.0 0.48 165760.0 11200.0 0.83 0.928 0.9663 3214228 CHDI2_000354 ONC(=O)CCCCCC(=O)N/N=C/c1ccc2OCCOc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A10 compound treatment 172080.0 15700.0 1.07 173040.0 18400.0 1.37 1.7277 0.9924 3214230 CHDI2_000355 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc3OCCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A11 compound treatment 169840.0 13500.0 0.92 173080.0 18500.0 1.38 1.6218 0.9806 3214232 CHDI2_000356 ONC(=O)CCCCCC(=O)N/N=C/COCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A12 compound treatment 180560.0 24200.0 1.65 174600.0 20000.0 1.49 2.2186 0.9987 3214234 CHDI2_000357 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/COCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A13 compound treatment 167880.0 11500.0 0.78 163160.0 8570.0 0.64 1.0052 0.9947 3214720 CHDI2_000358 CCOc1cccc(/C=N/NC(=O)CCCCCC(=O)NO)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A14 compound treatment 262840.0 106000.0 7.26 249080.0 94500.0 7.03 10.1049 0.9999 3553354 CHDI2_000359 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2c(O)ccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A15 compound treatment 195080.0 38700.0 2.64 198440.0 43800.0 3.26 4.1732 0.9944 3214236 CHDI2_000360 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A16 compound treatment 200000.0 43600.0 2.97 179200.0 24600.0 1.83 3.3978 0.9729 3214238 CHDI2_000361 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A17 compound treatment 162720.0 6340.0 0.43 162040.0 7450.0 0.55 0.6975 0.9925 3214240 CHDI2_000362 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A18 compound treatment 169040.0 12700.0 0.86 173200.0 18600.0 1.38 1.5895 0.9741 3214242 CHDI2_000363 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A19 compound treatment 163120.0 6740.0 0.46 163440.0 8850.0 0.66 0.7905 0.9846 3214244 CHDI2_000364 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A20 compound treatment 167920.0 11500.0 0.79 162880.0 8290.0 0.62 0.9924 0.9927 3214246 CHDI2_000365 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A21 compound treatment 167040.0 10700.0 0.73 159240.0 4650.0 0.35 0.7584 0.9423 3214248 CHDI2_000366 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A22 compound treatment 166760.0 10400.0 0.71 164600.0 10000.0 0.74 1.027 0.9997 3214250 CHDI2_000367 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A23 mock treatment 152680.0 -3700.0 -0.25 149200.0 -5400.0 -0.4 -0.4622 -0.9749 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 A24 mock treatment 153000.0 -3380.0 -0.23 148120.0 -6480.0 -0.48 -0.5036 -0.9429 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B01 compound treatment 185920.0 29500.0 2.01 188320.0 33700.0 2.51 3.199 0.994 3214256 CHDI2_000368 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2c(O)ccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B02 compound treatment 151800.0 -4580.0 -0.31 160920.0 6330.0 0.47 0.1121 0.1985 3214824 CHDI2_000369 NNC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B03 compound treatment 180640.0 24300.0 1.65 183000.0 28400.0 2.11 2.6645 0.9926 3214260 CHDI2_000370 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(O)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B04 compound treatment 170000.0 13600.0 0.93 167520.0 12900.0 0.96 1.3369 0.9998 3214826 CHDI2_000371 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B05 compound treatment 181840.0 25500.0 1.74 179840.0 25200.0 1.88 2.556 0.9992 3214264 CHDI2_000372 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc([N+](=O)[O-])c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B06 compound treatment 161560.0 5180.0 0.35 162720.0 8130.0 0.6 0.6774 0.9672 3214830 CHDI2_000373 COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B07 compound treatment 186360.0 30000.0 2.04 180480.0 25900.0 1.93 2.8076 0.9996 3214268 CHDI2_000374 Oc1ccc([N+](=O)[O-])c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B08 compound treatment 161720.0 5340.0 0.36 161680.0 7090.0 0.53 0.6304 0.9837 3214834 CHDI2_000375 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B09 compound treatment 168160.0 11800.0 0.8 171440.0 16800.0 1.25 1.4545 0.9768 3214272 CHDI2_000376 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)n3ccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B10 compound treatment 164080.0 7700.0 0.53 168760.0 14200.0 1.05 1.1167 0.9482 3214838 CHDI2_000377 ONC(=O)CCCCC(=O)N/N=C/c1ccc2OCCOc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B11 compound treatment 165800.0 9420.0 0.64 167680.0 13100.0 0.97 1.1428 0.9796 3214276 CHDI2_000378 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B12 compound treatment 183200.0 26800.0 1.83 172600.0 18000.0 1.34 2.2406 0.9883 3214842 CHDI2_000379 ONC(=O)CCCCC(=O)N/N=C/COCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B13 compound treatment 221240.0 64900.0 4.42 207080.0 52500.0 3.91 5.889 0.9981 3553415 CHDI2_000380 COc1cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B14 compound treatment 412680.0 256000.0 17.47 407160.0 253000.0 18.8 25.6478 0.9993 3553478 CHDI2_000381 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)c(O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B15 compound treatment 177120.0 20700.0 1.41 177120.0 22500.0 1.68 2.1853 0.9964 3214280 CHDI2_000382 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(I)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B16 compound treatment 183600.0 27200.0 1.86 184120.0 29500.0 2.2 2.8661 0.9965 3214846 CHDI2_000383 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B17 compound treatment 160520.0 4140.0 0.28 162880.0 8290.0 0.62 0.6357 0.9373 3214284 CHDI2_000384 C/C=C(/C)\C=N\NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B18 compound treatment 158160.0 1780.0 0.12 168040.0 13400.0 1.0 0.7935 0.7871 3214850 CHDI2_000385 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B19 compound treatment 175240.0 18900.0 1.29 176920.0 22300.0 1.66 2.0842 0.992 3214360 CHDI2_000386 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B20 compound treatment 168880.0 12500.0 0.85 167240.0 12600.0 0.94 1.2681 0.9988 3214854 CHDI2_000387 ONC(=O)CCCCC(=O)N/N=C/c1cccc(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B21 compound treatment 161240.0 4860.0 0.33 159360.0 4770.0 0.35 0.4851 0.9994 3214292 CHDI2_000388 Cc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B22 compound treatment 160040.0 3660.0 0.25 158960.0 4370.0 0.32 0.4062 0.9915 3214858 CHDI2_000389 ONC(=O)CCCCC(=O)N/N=C/c1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B23 mock treatment 152720.0 -3660.0 -0.25 149640.0 -4960.0 -0.37 -0.4372 -0.9819 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 B24 mock treatment 144320.0 -12100.0 -0.82 147040.0 -7560.0 -0.56 -0.9789 -0.9828 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C01 compound treatment 173240.0 16900.0 1.15 166440.0 11800.0 0.88 1.4362 0.9914 3214300 CHDI2_000390 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(Br)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C02 compound treatment 179600.0 23200.0 1.58 176560.0 22000.0 1.63 2.2754 0.9999 3214302 CHDI2_000391 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(Br)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C03 compound treatment 179640.0 23300.0 1.59 176720.0 22100.0 1.65 2.2858 0.9998 3214304 CHDI2_000392 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C04 compound treatment 177600.0 21200.0 1.45 178080.0 23500.0 1.75 2.259 0.9956 3214306 CHDI2_000393 Oc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C05 compound treatment 176680.0 20300.0 1.38 172720.0 18100.0 1.35 1.9326 0.9999 3214308 CHDI2_000394 ONC(=O)CCCCCC(=O)N/N=C/c1cc(O)ccc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C06 compound treatment 181160.0 24800.0 1.69 172720.0 18100.0 1.35 2.1485 0.9938 3214310 CHDI2_000395 Oc1ccc(Br)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C07 compound treatment 210000.0 53600.0 3.66 205000.0 50400.0 3.75 5.2377 0.9999 3214312 CHDI2_000396 COc1cc(Br)cc(/C=N/NC(=O)CCCCCC(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C08 compound treatment 213160.0 56800.0 3.87 202680.0 48100.0 3.58 5.2679 0.9992 3214314 CHDI2_000397 COc1cc(Br)cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C09 compound treatment 173520.0 17100.0 1.17 169160.0 14600.0 1.08 1.5929 0.9993 3214316 CHDI2_000398 COc1ccc(Br)c(/C=N/NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C10 compound treatment 172360.0 16000.0 1.09 179720.0 25100.0 1.87 2.0927 0.9669 3214318 CHDI2_000399 COc1ccc(Br)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C11 compound treatment 228000.0 71600.0 4.88 222720.0 68100.0 5.07 7.038 0.9998 3214724 CHDI2_000400 ONC(=O)CCCCCC(=O)N/N=C/c1cc(I)cc(I)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C12 compound treatment 234360.0 78000.0 5.32 222720.0 68100.0 5.07 7.3446 0.9997 3553358 CHDI2_000401 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C13 compound treatment 182920.0 26500.0 1.81 173080.0 18500.0 1.38 2.2523 0.9909 3214320 CHDI2_000402 COc1ccc(Br)cc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C14 compound treatment 180840.0 24500.0 1.67 177120.0 22500.0 1.68 2.3647 1.0 3214322 CHDI2_000403 COc1ccc(Br)cc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C15 compound treatment 168720.0 12300.0 0.84 162000.0 7410.0 0.55 0.9847 0.979 3214728 CHDI2_000404 CN(C)c1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C16 compound treatment 184400.0 28000.0 1.91 180480.0 25900.0 1.93 2.7131 1.0 3553362 CHDI2_000405 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc([N+](=O)[O-])c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C17 compound treatment 176040.0 19700.0 1.34 172760.0 18200.0 1.35 1.9038 1.0 3214324 CHDI2_000406 ONC(=O)CCCCCC(=O)N/N=C/c1cc2OCOc2cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C18 compound treatment 176560.0 20200.0 1.38 178000.0 23400.0 1.74 2.2047 0.9932 3214326 CHDI2_000407 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc3OCOc3cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C19 compound treatment 163560.0 7180.0 0.49 170200.0 15600.0 1.16 1.1675 0.9262 3214328 CHDI2_000408 ONC(=O)CCCCCC(=O)N/N=C/c1cccnc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C20 compound treatment 177160.0 20800.0 1.42 167760.0 13200.0 0.98 1.6947 0.9838 3214330 CHDI2_000409 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccnc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C21 compound treatment 174880.0 18500.0 1.26 167600.0 13000.0 0.97 1.5763 0.9914 3214332 CHDI2_000410 ONC(=O)CCCCCC(=O)N/N=C/c1ccncc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C22 compound treatment 171200.0 14800.0 1.01 177120.0 22500.0 1.68 1.8999 0.9706 3214334 CHDI2_000411 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccncc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C23 mock treatment 150920.0 -5460.0 -0.37 148600.0 -6000.0 -0.45 -0.5787 -0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 C24 mock treatment 153960.0 -2420.0 -0.16 145040.0 -9560.0 -0.71 -0.6195 -0.8486 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D01 compound treatment 164280.0 7900.0 0.54 161960.0 7370.0 0.55 0.7685 1.0 3214340 CHDI2_000412 Cc1ccsc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D02 compound treatment 172400.0 16000.0 1.09 165240.0 10600.0 0.79 1.3326 0.9876 3214910 CHDI2_000413 ONC(=O)CCCCC(=O)N/N=C/c1ccc(Br)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D03 compound treatment 171520.0 15100.0 1.03 170800.0 16200.0 1.21 1.5828 0.997 3214344 CHDI2_000414 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)CCCCCC(=O)Nc3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D04 compound treatment 177480.0 21100.0 1.44 168080.0 13500.0 1.0 1.7269 0.9845 3214914 CHDI2_000415 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D05 compound treatment 184680.0 28300.0 1.93 172960.0 18400.0 1.37 2.3309 0.9857 3214348 CHDI2_000416 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D06 compound treatment 176560.0 20200.0 1.38 173320.0 18700.0 1.39 1.9584 1.0 3214918 CHDI2_000417 ONC(=O)CCCCC(=O)N/N=C/c1cc(O)ccc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D07 compound treatment 176640.0 20300.0 1.38 179360.0 24800.0 1.84 2.2801 0.9899 3214356 CHDI2_000418 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D08 compound treatment 205160.0 48800.0 3.33 203160.0 48600.0 3.61 4.9075 0.9991 3214922 CHDI2_000419 COc1cc(Br)cc(/C=N/NC(=O)CCCCC(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D09 compound treatment 175520.0 19100.0 1.3 177160.0 22600.0 1.68 2.1103 0.9922 3214288 CHDI2_000420 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D10 compound treatment 172720.0 16300.0 1.11 172640.0 18000.0 1.34 1.7375 0.9957 3214926 CHDI2_000421 COc1ccc(Br)c(/C=N/NC(=O)CCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D11 compound treatment 196640.0 40300.0 2.74 195920.0 41300.0 3.08 4.1158 0.9984 3553419 CHDI2_000422 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2c(F)c(F)c(F)c(F)c2F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D12 compound treatment 421440.0 265000.0 18.07 407480.0 253000.0 18.82 26.0869 0.9998 3553482 CHDI2_000423 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2c(O)cc(O)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D13 compound treatment 184640.0 28300.0 1.93 169800.0 15200.0 1.13 2.1626 0.9678 3214352 CHDI2_000424 COc1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D14 compound treatment 172600.0 16200.0 1.11 172480.0 17900.0 1.33 1.7232 0.9958 3214930 CHDI2_000425 COc1ccc(Br)cc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D15 compound treatment 175040.0 18700.0 1.27 178200.0 23600.0 1.76 2.1419 0.9874 3553423 CHDI2_000426 ONC(=O)c1cccc(c1)C(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D16 compound treatment 170680.0 14300.0 0.98 174040.0 19400.0 1.45 1.7128 0.9815 3553485 CHDI2_000427 COc1cc(OC)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D17 compound treatment 166480.0 10100.0 0.69 170000.0 15400.0 1.15 1.2977 0.9703 3214364 CHDI2_000428 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2c(F)c(F)c(F)c(F)c2F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D18 compound treatment 173480.0 17100.0 1.17 172160.0 17600.0 1.31 1.7488 0.9984 3214934 CHDI2_000429 ONC(=O)CCCCC(=O)N/N=C/c1cc2OCOc2cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D19 compound treatment 160000.0 3620.0 0.25 165160.0 10600.0 0.79 0.7306 0.8865 3214368 CHDI2_000430 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D20 compound treatment 162640.0 6260.0 0.43 162240.0 7650.0 0.57 0.7042 0.99 3214938 CHDI2_000431 ONC(=O)CCCCC(=O)N/N=C/c1cccnc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D21 compound treatment 170960.0 14600.0 0.99 171800.0 17200.0 1.28 1.6084 0.9922 3214372 CHDI2_000432 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D22 compound treatment 168360.0 12000.0 0.82 159640.0 5050.0 0.38 0.8431 0.9378 3214942 CHDI2_000433 ONC(=O)CCCCC(=O)N/N=C/c1ccncc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D23 mock treatment 149440.0 -6940.0 -0.47 145040.0 -9560.0 -0.71 -0.8374 -0.9804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 D24 mock treatment 146920.0 -9460.0 -0.64 142440.0 -12200.0 -0.9 -1.0957 -0.9862 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E01 compound treatment 201120.0 44700.0 3.05 207080.0 52500.0 3.91 4.9191 0.9925 3214732 CHDI2_000434 CCn1c2ccccc2c3cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E02 compound treatment 238960.0 82600.0 5.63 239360.0 84800.0 6.31 8.4421 0.9984 3553366 CHDI2_000435 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(O)ccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E03 compound treatment 176080.0 19700.0 1.34 179280.0 24700.0 1.84 2.2489 0.9881 3214380 CHDI2_000436 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(Br)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E04 compound treatment 186720.0 30300.0 2.07 179040.0 24400.0 1.82 2.7492 0.998 3214382 CHDI2_000437 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(Br)s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E05 compound treatment 205400.0 49000.0 3.34 209120.0 54500.0 4.06 5.2328 0.9954 3214384 CHDI2_000438 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E06 compound treatment 190080.0 33700.0 2.3 197360.0 42800.0 3.18 3.8753 0.9872 3214386 CHDI2_000439 COc1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E07 compound treatment 211120.0 54700.0 3.73 213160.0 58600.0 4.36 5.7211 0.997 3214388 CHDI2_000440 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E08 compound treatment 197920.0 41500.0 2.83 209360.0 54800.0 4.08 4.8848 0.9842 3214390 CHDI2_000441 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCc3ccccc3)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E09 compound treatment 182160.0 25800.0 1.76 184640.0 30000.0 2.24 2.8241 0.9929 3214736 CHDI2_000442 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(c(F)c1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E10 compound treatment 200520.0 44100.0 3.01 189680.0 35100.0 2.61 3.9744 0.9975 3553369 CHDI2_000443 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)n3ccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E11 compound treatment 179800.0 23400.0 1.6 173160.0 18600.0 1.38 2.1061 0.9974 3214392 CHDI2_000444 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E12 compound treatment 178760.0 22400.0 1.53 179600.0 25000.0 1.86 2.3949 0.9951 3214394 CHDI2_000445 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E13 compound treatment 182160.0 25800.0 1.76 180440.0 25800.0 1.92 2.603 0.999 3214396 CHDI2_000446 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E14 compound treatment 179440.0 23100.0 1.57 183200.0 28600.0 2.13 2.6172 0.9889 3214398 CHDI2_000447 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E15 compound treatment 180480.0 24100.0 1.64 185000.0 30400.0 2.26 2.762 0.9876 3214400 CHDI2_000448 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E16 compound treatment 185200.0 28800.0 1.96 183560.0 29000.0 2.16 2.9138 0.9989 3214402 CHDI2_000449 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E17 compound treatment 171160.0 14800.0 1.01 177720.0 23100.0 1.72 1.9296 0.9675 3214784 CHDI2_000450 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(o1)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E18 compound treatment 183320.0 26900.0 1.84 182520.0 27900.0 2.08 2.7684 0.9981 3553372 CHDI2_000451 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E19 compound treatment 172120.0 15700.0 1.07 170800.0 16200.0 1.21 1.6117 0.9983 3214404 CHDI2_000452 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(c1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E20 compound treatment 170800.0 14400.0 0.98 169280.0 14700.0 1.09 1.4681 0.9986 3214406 CHDI2_000453 OC(=O)c1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E21 compound treatment 169600.0 13200.0 0.9 165960.0 11400.0 0.85 1.2355 0.9995 3214408 CHDI2_000454 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E22 compound treatment 170400.0 14000.0 0.96 170000.0 15400.0 1.15 1.4867 0.9959 3214410 CHDI2_000455 OC(=O)c1ccccc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E23 mock treatment 158960.0 2580.0 0.18 152320.0 -2280.0 -0.17 0.0047 0.0193 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 E24 mock treatment 155400.0 -979.0 -0.07 150440.0 -4160.0 -0.31 -0.2659 -0.8403 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F01 compound treatment 198040.0 41700.0 2.84 204120.0 49500.0 3.69 4.6148 0.9917 3553427 CHDI2_000456 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F02 compound treatment 182320.0 25900.0 1.77 177800.0 23200.0 1.73 2.4718 0.9999 3553487 CHDI2_000457 COc1cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F03 compound treatment 185840.0 29500.0 2.01 186280.0 31700.0 2.36 3.0878 0.9968 3214416 CHDI2_000458 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cn(c3ccccc23)S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F04 compound treatment 172680.0 16300.0 1.11 174360.0 19800.0 1.47 1.826 0.9904 3214990 CHDI2_000459 ONC(=O)CCCCC(=O)N/N=C/c1ccc(Br)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F05 compound treatment 180720.0 24300.0 1.66 180040.0 25400.0 1.89 2.5126 0.9978 3214420 CHDI2_000460 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F06 compound treatment 189200.0 32800.0 2.24 196600.0 42000.0 3.13 3.7929 0.9866 3214994 CHDI2_000461 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F07 compound treatment 177880.0 21500.0 1.47 183640.0 29000.0 2.16 2.5651 0.9821 3214424 CHDI2_000462 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F08 compound treatment 195720.0 39300.0 2.68 201680.0 47100.0 3.5 4.3746 0.9913 3214998 CHDI2_000463 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F09 compound treatment 236280.0 79900.0 5.45 230000.0 75400.0 5.61 7.8203 0.9999 3553430 CHDI2_000464 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F10 compound treatment 179520.0 23100.0 1.58 180400.0 25800.0 1.92 2.4737 0.9952 3553491 CHDI2_000465 CC(C)(C)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F11 compound treatment 180920.0 24500.0 1.67 183720.0 29100.0 2.17 2.7159 0.9918 3214428 CHDI2_000466 Cc1ncc(CO)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F12 compound treatment 175560.0 19200.0 1.31 188720.0 34100.0 2.54 2.7206 0.9524 3215002 CHDI2_000467 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F13 compound treatment 178840.0 22500.0 1.53 181760.0 27200.0 2.02 2.5125 0.9906 3214432 CHDI2_000468 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F14 compound treatment 175880.0 19500.0 1.33 183000.0 28400.0 2.11 2.435 0.975 3215006 CHDI2_000469 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F15 compound treatment 194000.0 37600.0 2.56 199440.0 44800.0 3.34 4.1738 0.9915 3214436 CHDI2_000470 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)N3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F16 compound treatment 183440.0 27100.0 1.84 188240.0 33600.0 2.5 3.0752 0.9887 3215010 CHDI2_000471 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)CCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F17 compound treatment 272200.0 116000.0 7.9 292840.0 138000.0 10.29 12.8591 0.9915 3553434 CHDI2_000472 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cn(c3ccccc23)S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F18 compound treatment 201760.0 45400.0 3.09 214040.0 59400.0 4.42 5.3162 0.9847 3553494 CHDI2_000473 CC1=C(C/C=N/NC(=O)c2cccc(c2)C(=O)NO)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F19 compound treatment 189240.0 32900.0 2.24 181520.0 26900.0 2.0 3.0012 0.9985 3214440 CHDI2_000474 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F20 compound treatment 170560.0 14200.0 0.97 171400.0 16800.0 1.25 1.5681 0.9919 3215014 CHDI2_000475 ONC(=O)CCCCC(=O)N/N=C/c1cccc(c1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F21 compound treatment 173480.0 17100.0 1.17 174840.0 20200.0 1.51 1.8899 0.992 3214444 CHDI2_000476 CCCCCCC/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F22 compound treatment 169160.0 12800.0 0.87 170160.0 15600.0 1.16 1.4353 0.9901 3215018 CHDI2_000477 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F23 mock treatment 163680.0 7300.0 0.5 159080.0 4490.0 0.33 0.588 0.9811 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 F24 mock treatment 157800.0 1420.0 0.1 153480.0 -1120.0 -0.08 0.0098 0.0771 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G01 compound treatment 175120.0 18700.0 1.28 173720.0 19100.0 1.42 1.91 0.9985 3214452 CHDI2_000478 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G02 compound treatment 188040.0 31700.0 2.16 180480.0 25900.0 1.93 2.8886 0.9984 3214454 CHDI2_000479 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G03 compound treatment 181560.0 25200.0 1.72 180480.0 25900.0 1.93 2.5762 0.9983 3214788 CHDI2_000480 Cn1cc(/C=N/NC(=O)CCCCCC(=O)NO)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G04 compound treatment 204840.0 48500.0 3.3 205120.0 50500.0 3.76 4.9953 0.9979 3553376 CHDI2_000481 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(I)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G05 compound treatment 176800.0 20400.0 1.39 183320.0 28700.0 2.14 2.4962 0.9784 3214456 CHDI2_000482 ONC(=O)CCCCCC(=O)N/N=C/c1cccnc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G06 compound treatment 179000.0 22600.0 1.54 185240.0 30600.0 2.28 2.7033 0.9818 3214458 CHDI2_000483 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccnc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G07 compound treatment 184640.0 28300.0 1.93 187360.0 32800.0 2.44 3.0868 0.9932 3214460 CHDI2_000484 ONC(=O)CCCCCC(=O)N/N=C/C=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G08 compound treatment 210360.0 54000.0 3.68 192040.0 37400.0 2.79 4.573 0.9906 3214462 CHDI2_000485 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/C=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G09 compound treatment 186760.0 30400.0 2.07 187920.0 33300.0 2.48 3.2184 0.996 3214464 CHDI2_000486 C[C@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G10 compound treatment 190680.0 34300.0 2.34 190080.0 35500.0 2.64 3.5211 0.9982 3214466 CHDI2_000487 C[C@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G11 compound treatment 187000.0 30600.0 2.09 181880.0 27300.0 2.03 2.9121 0.9999 3214468 CHDI2_000488 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G12 compound treatment 185760.0 29400.0 2.0 181760.0 27200.0 2.02 2.8461 1.0 3214469 CHDI2_000489 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G13 compound treatment 183240.0 26900.0 1.83 178400.0 23800.0 1.77 2.5477 0.9999 3214470 CHDI2_000490 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G14 compound treatment 187680.0 31300.0 2.13 164840.0 10200.0 0.76 2.0482 0.9038 3214472 CHDI2_000491 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G15 compound treatment 185360.0 29000.0 1.98 182760.0 28200.0 2.1 2.8794 0.9996 3214474 CHDI2_000492 ONC(=O)CCCCCC(=O)N/N=C/C1CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G16 compound treatment 185760.0 29400.0 2.0 182600.0 28000.0 2.08 2.8903 0.9998 3214476 CHDI2_000493 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/C2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G17 compound treatment 187440.0 31100.0 2.12 184400.0 29800.0 2.22 3.066 0.9997 3214478 CHDI2_000494 COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G18 compound treatment 188200.0 31800.0 2.17 187720.0 33100.0 2.47 3.2773 0.998 3214480 CHDI2_000495 COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G19 compound treatment 195960.0 39600.0 2.7 192200.0 37600.0 2.8 3.8872 0.9998 3214792 CHDI2_000496 ONC(=O)CCCCCC(=O)N/N=C/c1cn(Cc2ccccc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G20 compound treatment 185480.0 29100.0 1.98 184160.0 29600.0 2.2 2.9589 0.9987 3553380 CHDI2_000497 C/C=C(/C)\C=N\NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G21 compound treatment 199840.0 43500.0 2.96 218240.0 63600.0 4.74 5.4447 0.9745 3214482 CHDI2_000498 ONC(=O)CCCCCC(=O)N/N=C/c1cc(Br)cc(Br)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G22 compound treatment 200360.0 44000.0 3.0 203920.0 49300.0 3.67 4.7161 0.995 3214484 CHDI2_000499 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(Br)cc(Br)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G23 mock treatment 161160.0 4780.0 0.33 160160.0 5570.0 0.41 0.5234 0.993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 G24 mock treatment 159840.0 3460.0 0.24 162720.0 8130.0 0.6 0.5945 0.9158 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H01 compound treatment 175200.0 18800.0 1.28 170600.0 16000.0 1.19 1.7496 0.9993 3214490 CHDI2_000500 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H02 compound treatment 171800.0 15400.0 1.05 174520.0 19900.0 1.48 1.792 0.9858 3215062 CHDI2_000501 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H03 compound treatment 189160.0 32800.0 2.23 185640.0 31000.0 2.31 3.2142 0.9999 3553438 CHDI2_000502 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H04 compound treatment 206120.0 49700.0 3.39 201360.0 46800.0 3.48 4.8591 0.9999 3553498 CHDI2_000503 NC(=O)COc1ccccc1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H05 compound treatment 184720.0 28300.0 1.93 184880.0 30300.0 2.25 2.9601 0.9971 3214494 CHDI2_000504 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H06 compound treatment 184480.0 28100.0 1.92 182720.0 28100.0 2.09 2.8349 0.999 3215066 CHDI2_000505 ONC(=O)CCCCC(=O)N/N=C/c1cccnc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H07 compound treatment 426520.0 270000.0 18.42 425560.0 271000.0 20.17 27.2833 0.999 3214498 CHDI2_000506 Oc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H08 compound treatment 198440.0 42100.0 2.87 193040.0 38400.0 2.86 4.051 1.0 3215070 CHDI2_000507 ONC(=O)CCCCC(=O)N/N=C/C=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H09 compound treatment 259520.0 103000.0 7.03 256120.0 102000.0 7.56 10.3153 0.9994 3214502 CHDI2_000508 Oc1cc(O)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H10 compound treatment 185720.0 29300.0 2.0 188000.0 33400.0 2.49 3.1725 0.9942 3215074 CHDI2_000509 C[C@H](CCC=C(C)C)C/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H11 compound treatment 184920.0 28500.0 1.95 180760.0 26200.0 1.95 2.7529 1.0 3214506 CHDI2_000510 COc1cc(OC)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H12 compound treatment 184280.0 27900.0 1.9 182520.0 27900.0 2.08 2.8147 0.999 3215078 CHDI2_000511 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H13 compound treatment 189480.0 33100.0 2.26 186040.0 31400.0 2.34 3.2506 0.9998 3214510 CHDI2_000512 COc1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H14 compound treatment 178000.0 21600.0 1.47 180000.0 25400.0 1.89 2.3793 0.9924 3215080 CHDI2_000513 ONC(=O)CCCCC(=O)N/N=C/c1ccc(C#N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H15 compound treatment 177240.0 20900.0 1.42 178880.0 24300.0 1.81 2.2838 0.993 3214514 CHDI2_000514 CC(C)(C)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H16 compound treatment 175960.0 19600.0 1.33 179680.0 25100.0 1.87 2.2641 0.9865 3215084 CHDI2_000515 ONC(=O)CCCCC(=O)N/N=C/C1CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H17 compound treatment 191160.0 34800.0 2.37 190280.0 35700.0 2.66 3.5548 0.9984 3214518 CHDI2_000516 CC1=C(C/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H18 compound treatment 181360.0 25000.0 1.7 183080.0 28500.0 2.12 2.7034 0.9941 3215088 CHDI2_000517 COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H19 compound treatment 181560.0 25200.0 1.72 185480.0 30900.0 2.3 2.8394 0.9897 3553442 CHDI2_000518 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H20 compound treatment 177120.0 20700.0 1.41 178520.0 23900.0 1.78 2.259 0.9935 3553502 CHDI2_000519 NC(=O)COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H21 compound treatment 181480.0 25100.0 1.71 180760.0 26200.0 1.95 2.5871 0.9979 3214522 CHDI2_000520 NC(=O)COc1ccccc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H22 compound treatment 205880.0 49500.0 3.37 202720.0 48100.0 3.58 4.9191 0.9996 3215092 CHDI2_000521 ONC(=O)CCCCC(=O)N/N=C/c1cc(Br)cc(Br)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H23 mock treatment 161360.0 4980.0 0.34 164040.0 9450.0 0.7 0.7372 0.9443 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 H24 mock treatment 151400.0 -4980.0 -0.34 157960.0 3370.0 0.25 -0.0629 -0.1492 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I01 compound treatment 178800.0 22400.0 1.53 177560.0 23000.0 1.71 2.2895 0.9984 3214530 CHDI2_000522 COc1cc(Cl)c(/C=N/NC(=O)CCCCCC(=O)NO)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I02 compound treatment 169720.0 13300.0 0.91 168640.0 14000.0 1.05 1.3823 0.9976 3214532 CHDI2_000523 COc1cc(Cl)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I03 compound treatment 212240.0 55900.0 3.81 211040.0 56400.0 4.2 5.6636 0.9988 3214534 CHDI2_000524 ONC(=O)CCCCCC(=O)N/N=C/c1cc(Cl)cc(Cl)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I04 compound treatment 212200.0 55800.0 3.81 204960.0 50400.0 3.75 5.3416 1.0 3214536 CHDI2_000525 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I05 compound treatment 177040.0 20700.0 1.41 178320.0 23700.0 1.77 2.2446 0.9937 3214796 CHDI2_000526 ONC(=O)CCCCCC(=O)N/N=C/C1=CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I06 compound treatment 212200.0 55800.0 3.81 207640.0 53000.0 3.95 5.4827 0.9998 3553384 CHDI2_000527 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I07 compound treatment 200840.0 44500.0 3.03 199680.0 45100.0 3.36 4.5161 0.9987 3214538 CHDI2_000528 ONC(=O)CCCCCC(=O)N/N=C/c1cc(Br)cc([N+](=O)[O-])c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I08 compound treatment 208120.0 51700.0 3.53 202400.0 47800.0 3.56 5.0102 1.0 3214540 CHDI2_000529 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(Br)cc([N+](=O)[O-])c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I09 compound treatment 205440.0 49100.0 3.34 198880.0 44300.0 3.3 4.6958 1.0 3214542 CHDI2_000530 CCN(CC)c1ccc(/C=N/NC(=O)CCCCCC(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I10 compound treatment 208160.0 51800.0 3.53 215840.0 61200.0 4.56 5.7195 0.992 3214544 CHDI2_000531 CCN(CC)c1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I11 compound treatment 184400.0 28000.0 1.91 186160.0 31600.0 2.35 3.0121 0.9947 3214546 CHDI2_000532 ONC(=O)CCCCCC(=O)N/N=C/c1ccc2OCCc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I12 compound treatment 185440.0 29100.0 1.98 190800.0 36200.0 2.69 3.3064 0.9886 3214548 CHDI2_000533 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc3OCCc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I13 compound treatment 347720.0 191000.0 13.05 331920.0 177000.0 13.2 18.5565 1.0 3214550 CHDI2_000534 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I14 compound treatment 265000.0 109000.0 7.41 274760.0 120000.0 8.94 11.5605 0.9956 3214552 CHDI2_000535 Oc1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I15 compound treatment 192560.0 36200.0 2.47 192360.0 37800.0 2.81 3.7317 0.9979 3214554 CHDI2_000536 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I16 compound treatment 196280.0 39900.0 2.72 202080.0 47500.0 3.53 4.4226 0.9916 3214556 CHDI2_000537 Oc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I17 compound treatment 383400.0 227000.0 15.48 375040.0 220000.0 16.41 22.5458 0.9996 3214558 CHDI2_000538 ONC(=O)CCCCCC(=O)N/N=C/c1cc(O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I18 compound treatment 310920.0 155000.0 10.54 325760.0 171000.0 12.74 16.4582 0.9956 3214560 CHDI2_000539 Oc1ccc(O)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I19 compound treatment 240680.0 84300.0 5.75 245600.0 91000.0 6.77 8.8534 0.9967 3214562 CHDI2_000540 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I20 compound treatment 256400.0 100000.0 6.82 256840.0 102000.0 7.61 10.2028 0.9985 3214564 CHDI2_000541 Oc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I21 compound treatment 169920.0 13500.0 0.92 169800.0 15200.0 1.13 1.453 0.9949 3214799 CHDI2_000542 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I22 compound treatment 187560.0 31200.0 2.13 189400.0 34800.0 2.59 3.3349 0.9952 3553388 CHDI2_000543 Cc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I23 mock treatment 158280.0 1900.0 0.13 160200.0 5610.0 0.42 0.3866 0.8851 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 I24 mock treatment 155440.0 -939.0 -0.06 157080.0 2490.0 0.18 0.0855 0.437 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J01 compound treatment 172640.0 16300.0 1.11 170760.0 16200.0 1.2 1.6347 0.9992 3214570 CHDI2_000544 Oc1ccccc1NC(=O)CCCCCC(=O)NN=C2CCCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J02 compound treatment 174680.0 18300.0 1.25 179920.0 25300.0 1.88 2.2151 0.9799 3215140 CHDI2_000545 COc1cc(Cl)c(/C=N/NC(=O)CCCCC(=O)NO)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J03 compound treatment 172280.0 15900.0 1.08 175120.0 20500.0 1.53 1.8468 0.9859 3214572 CHDI2_000546 Oc1ccccc1NC(=O)CCCCCC(=O)NN=C2CCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J04 compound treatment 205200.0 48800.0 3.33 207520.0 52900.0 3.94 5.1389 0.9965 3215144 CHDI2_000547 ONC(=O)CCCCC(=O)N/N=C/c1cc(Cl)cc(Cl)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J05 compound treatment 217760.0 61400.0 4.18 219200.0 64600.0 4.81 6.3591 0.9976 3553446 CHDI2_000548 Cc1ncc(CO)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J06 compound treatment 182040.0 25700.0 1.75 182480.0 27900.0 2.08 2.7046 0.9964 3554234 CHDI2_000549 ONC(=O)c1cccc(c1)C(=O)NN=C2CCCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J07 compound treatment 180760.0 24400.0 1.66 181880.0 27300.0 2.03 2.6113 0.9951 3214574 CHDI2_000550 Oc1ccccc1NC(=O)CCCCCC(=O)NN=C2CCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J08 compound treatment 194200.0 37800.0 2.58 201880.0 47300.0 3.52 4.3118 0.9883 3215148 CHDI2_000551 ONC(=O)CCCCC(=O)N/N=C/c1cc(Br)cc([N+](=O)[O-])c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J09 compound treatment 183680.0 27300.0 1.86 180360.0 25800.0 1.92 2.6721 0.9999 3214215 CHDI2_000552 NNC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J10 compound treatment 199200.0 42800.0 2.92 212040.0 57400.0 4.28 5.0875 0.9827 3215152 CHDI2_000553 CCN(CC)c1ccc(/C=N/NC(=O)CCCCC(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J11 compound treatment 185720.0 29300.0 2.0 190280.0 35700.0 2.66 3.2925 0.9902 3214576 CHDI2_000554 COc1cc(Br)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J12 compound treatment 186800.0 30400.0 2.07 191040.0 36400.0 2.71 3.3846 0.9912 3215156 CHDI2_000555 ONC(=O)CCCCC(=O)N/N=C/c1ccc2OCCc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J13 compound treatment 198560.0 42200.0 2.88 199000.0 44400.0 3.3 4.3704 0.9976 3214580 CHDI2_000556 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/CCC2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J14 compound treatment 324720.0 168000.0 11.48 341960.0 187000.0 13.95 17.9761 0.9953 3215160 CHDI2_000557 ONC(=O)CCCCC(=O)N/N=C/c1cccc(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J15 compound treatment 196920.0 40500.0 2.76 203160.0 48600.0 3.61 4.5103 0.9912 3214584 CHDI2_000558 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J16 compound treatment 212960.0 56600.0 3.86 216520.0 61900.0 4.61 5.9867 0.9961 3215164 CHDI2_000559 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J17 compound treatment 190960.0 34600.0 2.36 190320.0 35700.0 2.66 3.5472 0.9982 3214588 CHDI2_000560 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J18 compound treatment 373120.0 217000.0 14.78 390640.0 236000.0 17.57 22.8713 0.9963 3215168 CHDI2_000561 ONC(=O)CCCCC(=O)N/N=C/c1cc(O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J19 compound treatment 194600.0 38200.0 2.61 186840.0 32200.0 2.4 3.5396 0.9992 3214215 CHDI2_000562 NNC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J20 compound treatment 265680.0 109000.0 7.45 267840.0 113000.0 8.43 11.2291 0.9981 3215172 CHDI2_000563 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J21 compound treatment 193320.0 36900.0 2.52 197600.0 43000.0 3.2 4.0441 0.993 3553450 CHDI2_000564 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J22 compound treatment 167840.0 11500.0 0.78 167880.0 13300.0 0.99 1.2517 0.9932 3554232 CHDI2_000565 ONC(=O)c1cccc(c1)C(=O)NN=C2CCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J23 mock treatment 160040.0 3660.0 0.25 157680.0 3090.0 0.23 0.3389 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 J24 mock treatment 153160.0 -3220.0 -0.22 152080.0 -2520.0 -0.19 -0.2875 -0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K01 compound treatment 172480.0 16100.0 1.1 167280.0 12700.0 0.94 1.4438 0.9972 3214592 CHDI2_000566 COc1cccc(OC)c1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K02 compound treatment 177880.0 21500.0 1.47 174680.0 20100.0 1.49 2.0936 1.0 3214594 CHDI2_000567 COc1cccc(OC)c1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K03 compound treatment 177720.0 21300.0 1.45 179960.0 25400.0 1.89 2.3637 0.9917 3214596 CHDI2_000568 COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K04 compound treatment 184200.0 27800.0 1.9 182440.0 27800.0 2.07 2.8066 0.999 3214598 CHDI2_000569 COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K05 compound treatment 189680.0 33300.0 2.27 186240.0 31600.0 2.36 3.2708 0.9998 3214600 CHDI2_000570 COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K06 compound treatment 200320.0 43900.0 3.0 199960.0 45400.0 3.38 4.5058 0.9982 3214602 CHDI2_000571 COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K07 compound treatment 180000.0 23600.0 1.61 176000.0 21400.0 1.59 2.2652 1.0 3214802 CHDI2_000572 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K08 compound treatment 188760.0 32400.0 2.21 186040.0 31400.0 2.34 3.2159 0.9996 3553391 CHDI2_000573 Cc1[nH]cnc1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K09 compound treatment 178080.0 21700.0 1.48 180920.0 26300.0 1.96 2.4316 0.9904 3214604 CHDI2_000574 CC1(C)COC(CCC/C=N/NC(=O)CCCCCC(=O)NO)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K10 compound treatment 180160.0 23800.0 1.62 180320.0 25700.0 1.91 2.5003 0.9966 3214606 CHDI2_000575 CC1(C)COC(CCC/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K11 compound treatment 182880.0 26500.0 1.81 186600.0 32000.0 2.38 2.9619 0.9907 3214608 CHDI2_000576 Cc1nnc(Sc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K12 compound treatment 190120.0 33700.0 2.3 187800.0 33200.0 2.47 3.3741 0.9994 3214610 CHDI2_000577 Cc1nnc(Sc2ccc(/C=N/NC(=O)CCCCCC(=O)Nc3ccccc3O)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K13 compound treatment 189880.0 33500.0 2.28 186400.0 31800.0 2.37 3.2889 0.9998 3214612 CHDI2_000578 ONC(=O)CCCCCC(=O)N/N=C/c1cc(Br)cs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K14 compound treatment 189960.0 33600.0 2.29 184680.0 30100.0 2.24 3.2022 0.9999 3214614 CHDI2_000579 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(Br)cs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K15 compound treatment 178200.0 21800.0 1.49 177400.0 22800.0 1.7 2.2521 0.9978 3214806 CHDI2_000580 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)NO)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K16 compound treatment 181560.0 25200.0 1.72 179880.0 25300.0 1.88 2.5446 0.9989 3553395 CHDI2_000581 Cc1ccsc1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K17 compound treatment 175840.0 19500.0 1.33 177200.0 22600.0 1.68 2.1278 0.9931 3214616 CHDI2_000582 CC(C)(C)OC(=O)NC/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K18 compound treatment 177200.0 20800.0 1.42 179080.0 24500.0 1.82 2.2923 0.9924 3214618 CHDI2_000583 CC(C)(C)OC(=O)NC/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K19 compound treatment 208480.0 52100.0 3.55 204600.0 50000.0 3.72 5.1434 0.9997 3214620 CHDI2_000584 ONC(=O)CCCCCC(=O)N/N=C/c1ccc-2c(Cc3ccccc32)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K20 compound treatment 174080.0 17700.0 1.21 184640.0 30000.0 2.24 2.4345 0.9581 3214622 CHDI2_000585 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K21 compound treatment 176160.0 19800.0 1.35 171160.0 16600.0 1.23 1.8254 0.999 3214624 CHDI2_000586 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K22 compound treatment 171400.0 15000.0 1.02 171360.0 16800.0 1.25 1.6065 0.9952 3214626 CHDI2_000587 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(F)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K23 mock treatment 157400.0 1020.0 0.07 158600.0 4010.0 0.3 0.26 0.8494 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 K24 mock treatment 158600.0 2220.0 0.15 154160.0 -435.0 -0.03 0.0842 0.5437 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L01 compound treatment 164280.0 7900.0 0.54 168160.0 13600.0 1.01 1.0948 0.9567 3214628 CHDI2_000588 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L02 compound treatment 175080.0 18700.0 1.27 169320.0 14700.0 1.1 1.6765 0.9972 3215202 CHDI2_000589 COc1cccc(OC)c1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L03 compound treatment 172560.0 16200.0 1.1 173600.0 19000.0 1.41 1.7803 0.9924 3214632 CHDI2_000590 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L04 compound treatment 179520.0 23100.0 1.58 177040.0 22400.0 1.67 2.2968 0.9996 3215206 CHDI2_000591 COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L05 compound treatment 173200.0 16800.0 1.15 174800.0 20200.0 1.5 1.8743 0.9911 3214636 CHDI2_000592 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L06 compound treatment 186480.0 30100.0 2.05 190840.0 36200.0 2.7 3.3586 0.9909 3215210 CHDI2_000593 COc1cc(O)cc(OC)c1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L07 compound treatment 241120.0 84700.0 5.78 233200.0 78600.0 5.85 8.222 1.0 3553454 CHDI2_000594 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)N3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L08 compound treatment 202960.0 46600.0 3.18 197960.0 43400.0 3.23 4.5278 1.0 3553643 CHDI2_000595 ONC(=O)c1cccc(c1)C(=O)N/N=C/Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L09 compound treatment 175760.0 19400.0 1.32 172040.0 17400.0 1.3 1.8524 1.0 3214640 CHDI2_000596 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L10 compound treatment 176520.0 20100.0 1.37 177840.0 23200.0 1.73 2.1943 0.9935 3215214 CHDI2_000597 CC1(C)COC(CCC/C=N/NC(=O)CCCCC(=O)NO)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L11 compound treatment 179680.0 23300.0 1.59 183280.0 28700.0 2.13 2.6329 0.9894 3214642 CHDI2_000598 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L12 compound treatment 183840.0 27500.0 1.87 179200.0 24600.0 1.83 2.6188 0.9999 3215218 CHDI2_000599 Cc1nnc(Sc2ccc(/C=N/NC(=O)CCCCC(=O)NO)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L13 compound treatment 177000.0 20600.0 1.41 182080.0 27500.0 2.05 2.4406 0.9833 3214644 CHDI2_000600 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L14 compound treatment 179520.0 23100.0 1.58 186800.0 32200.0 2.4 2.8105 0.9794 3215222 CHDI2_000601 ONC(=O)CCCCC(=O)N/N=C/c1cc(Br)cs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L15 compound treatment 189640.0 33300.0 2.27 194720.0 40100.0 2.99 3.7152 0.9908 3553458 CHDI2_000602 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L16 compound treatment 174360.0 18000.0 1.23 177120.0 22500.0 1.68 2.0523 0.9882 3553647 CHDI2_000603 COC(=O)c1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L17 compound treatment 190560.0 34200.0 2.33 201400.0 46800.0 3.48 4.1111 0.9809 3214648 CHDI2_000604 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(Oc3ccccc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L18 compound treatment 177640.0 21300.0 1.45 177000.0 22400.0 1.67 2.2041 0.9976 3215226 CHDI2_000605 CC(C)(C)OC(=O)NC/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L19 compound treatment 173400.0 17000.0 1.16 169760.0 15200.0 1.13 1.6187 0.9999 3214652 CHDI2_000606 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc[n+]([O-])cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L20 compound treatment 228000.0 71600.0 4.88 243960.0 89400.0 6.65 8.1558 0.9885 3215230 CHDI2_000607 ONC(=O)CCCCC(=O)N/N=C/c1ccc-2c(Cc3ccccc32)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L21 compound treatment 179200.0 22800.0 1.56 182280.0 27700.0 2.06 2.5572 0.9904 3214656 CHDI2_000608 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L22 compound treatment 173920.0 17500.0 1.2 171560.0 17000.0 1.26 1.7385 0.9996 3215234 CHDI2_000609 ONC(=O)CCCCC(=O)N/N=C/c1ccc(F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L23 mock treatment 157920.0 1540.0 0.11 156360.0 1770.0 0.13 0.1672 0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 L24 mock treatment 155680.0 -699.0 -0.05 155720.0 1130.0 0.08 0.0255 0.2649 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M01 compound treatment 181800.0 25400.0 1.73 181720.0 27100.0 2.02 2.653 0.9971 3214660 CHDI2_000610 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M02 compound treatment 191120.0 34700.0 2.37 192960.0 38400.0 2.86 3.6939 0.9957 3214662 CHDI2_000611 Oc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M03 compound treatment 191040.0 34700.0 2.36 190800.0 36200.0 2.69 3.5763 0.9979 3214664 CHDI2_000612 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(F)c(Oc2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M04 compound treatment 205880.0 49500.0 3.37 198480.0 43900.0 3.27 4.6959 0.9999 3214666 CHDI2_000613 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(F)c(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M05 compound treatment 191560.0 35200.0 2.4 193920.0 39300.0 2.93 3.7656 0.9951 3214668 CHDI2_000614 ONC(=O)CCCCCC(=O)N/N=C/c1cc(F)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M06 compound treatment 193360.0 37000.0 2.52 192760.0 38200.0 2.84 3.7913 0.9982 3214670 CHDI2_000615 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(F)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M07 compound treatment 219480.0 63100.0 4.3 221800.0 67200.0 5.0 6.5789 0.9972 3214672 CHDI2_000616 ONC(=O)CCCCCC(=O)N/N=C/c1coc2ccccc2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M08 compound treatment 209400.0 53000.0 3.61 211240.0 56600.0 4.22 5.5372 0.9971 3214674 CHDI2_000617 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M09 compound treatment 181160.0 24800.0 1.69 180720.0 26100.0 1.94 2.5696 0.9975 3214814 CHDI2_000618 CN(C)CCCOc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M10 compound treatment 216160.0 59800.0 4.08 214760.0 60200.0 4.48 6.0483 0.9989 3553403 CHDI2_000619 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M11 compound treatment 190800.0 34400.0 2.35 183040.0 28400.0 2.12 3.1564 0.9987 3214676 CHDI2_000620 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M12 compound treatment 191680.0 35300.0 2.41 190760.0 36200.0 2.69 3.6051 0.9984 3214678 CHDI2_000621 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M13 compound treatment 206720.0 50300.0 3.43 209840.0 55200.0 4.11 5.3343 0.996 3214818 CHDI2_000622 CCOc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M14 compound treatment 228080.0 71700.0 4.89 229280.0 74700.0 5.56 7.3871 0.9979 3553407 CHDI2_000623 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M15 compound treatment 186160.0 29800.0 2.03 188320.0 33700.0 2.51 3.2106 0.9945 3214680 CHDI2_000624 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(c1)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M16 compound treatment 180920.0 24500.0 1.67 183600.0 29000.0 2.16 2.7096 0.9921 3214682 CHDI2_000625 OB(O)c1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M17 compound treatment 191560.0 35200.0 2.4 189720.0 35100.0 2.61 3.5446 0.9991 3214684 CHDI2_000626 ONC(=O)CCCCCC(=O)N/N=C/c1ccco1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M18 compound treatment 182440.0 26100.0 1.78 186040.0 31400.0 2.34 2.9112 0.9908 3214686 CHDI2_000627 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M19 compound treatment 181680.0 25300.0 1.72 182960.0 28400.0 2.11 2.7125 0.995 3214688 CHDI2_000628 ONC(=O)CCCCCC(=O)N/N=C/c1ccoc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M20 compound treatment 177360.0 21000.0 1.43 182440.0 27800.0 2.07 2.4769 0.9836 3214690 CHDI2_000629 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccoc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M21 compound treatment 180880.0 24500.0 1.67 177320.0 22700.0 1.69 2.3771 1.0 3214692 CHDI2_000630 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M22 compound treatment 177800.0 21400.0 1.46 175520.0 20900.0 1.56 2.1339 0.9995 3214694 CHDI2_000631 Oc1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M23 mock treatment 164680.0 8300.0 0.57 167320.0 12700.0 0.95 1.0699 0.9697 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 M24 mock treatment 162240.0 5860.0 0.4 158680.0 4090.0 0.3 0.4975 0.9909 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N01 compound treatment 177360.0 21000.0 1.43 176760.0 22200.0 1.65 2.178 0.9975 3214700 CHDI2_000632 Cc1ccccc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N02 compound treatment 180560.0 24200.0 1.65 181600.0 27000.0 2.01 2.587 0.9952 3215270 CHDI2_000633 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N03 compound treatment 188480.0 32100.0 2.19 195400.0 40800.0 3.04 3.695 0.9871 3214704 CHDI2_000634 COc1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N04 compound treatment 186080.0 29700.0 2.02 182760.0 28200.0 2.1 2.9141 0.9999 3215274 CHDI2_000635 ONC(=O)CCCCC(=O)N/N=C/c1ccc(F)c(Oc2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N05 compound treatment 179720.0 23300.0 1.59 182040.0 27400.0 2.04 2.5696 0.9924 3214708 CHDI2_000636 O[C@@H](/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N06 compound treatment 192920.0 36500.0 2.49 194680.0 40100.0 2.98 3.8712 0.996 3215278 CHDI2_000637 ONC(=O)CCCCC(=O)N/N=C/c1cc(F)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N07 compound treatment 180520.0 24100.0 1.65 181720.0 27100.0 2.02 2.5913 0.9949 3214712 CHDI2_000638 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N08 compound treatment 209320.0 52900.0 3.61 210600.0 56000.0 4.17 5.4996 0.9974 3215282 CHDI2_000639 ONC(=O)CCCCC(=O)N/N=C/c1coc2ccccc2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N09 compound treatment 189440.0 33100.0 2.25 189440.0 34800.0 2.59 3.4276 0.9976 3553466 CHDI2_000640 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2nccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N10 compound treatment 316120.0 160000.0 10.89 315600.0 161000.0 11.98 16.1742 0.9989 3553651 CHDI2_000641 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc3ccccc3n2S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N11 compound treatment 188880.0 32500.0 2.22 192360.0 37800.0 2.81 3.5543 0.9931 3214714 CHDI2_000642 COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N12 compound treatment 187640.0 31300.0 2.13 188760.0 34200.0 2.54 3.3051 0.9961 3215286 CHDI2_000643 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N13 compound treatment 188240.0 31900.0 2.17 187200.0 32600.0 2.43 3.2519 0.9985 3553471 CHDI2_000644 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N14 compound treatment 289520.0 133000.0 9.08 298320.0 144000.0 10.7 13.9824 0.9967 3553510 CHDI2_000645 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N15 compound treatment 182920.0 26500.0 1.81 185520.0 30900.0 2.3 2.907 0.9929 3214718 CHDI2_000646 CCOc1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N16 compound treatment 180560.0 24200.0 1.65 185040.0 30400.0 2.27 2.768 0.9878 3215290 CHDI2_000647 ONC(=O)CCCCC(=O)N/N=C/c1cccc(c1)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N17 compound treatment 205760.0 49400.0 3.37 208640.0 54000.0 4.02 5.2249 0.9961 3214722 CHDI2_000648 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(I)cc(I)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N18 compound treatment 180360.0 24000.0 1.63 177200.0 22600.0 1.68 2.3457 0.9999 3215294 CHDI2_000649 ONC(=O)CCCCC(=O)N/N=C/c1ccco1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N19 compound treatment 180640.0 24300.0 1.65 183920.0 29300.0 2.18 2.7129 0.9906 3214726 CHDI2_000650 CN(C)c1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N20 compound treatment 180840.0 24500.0 1.67 177040.0 22400.0 1.67 2.3605 1.0 3215298 CHDI2_000651 ONC(=O)CCCCC(=O)N/N=C/c1ccoc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N21 compound treatment 175760.0 19400.0 1.32 181880.0 27300.0 2.03 2.3703 0.9783 3214730 CHDI2_000652 CCn1c2ccccc2c3cc(/C=N/NC(=O)CCCCCC(=O)Nc4ccccc4O)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N22 compound treatment 168440.0 12100.0 0.82 173320.0 18700.0 1.39 1.5669 0.9683 3215302 CHDI2_000653 ONC(=O)CCCCC(=O)N/N=C/c1cccc(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N23 mock treatment 159360.0 2980.0 0.2 159960.0 5370.0 0.4 0.4261 0.9509 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 N24 mock treatment 157320.0 941.0 0.06 156200.0 1610.0 0.12 0.1298 0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O01 compound treatment 172440.0 16100.0 1.1 165760.0 11200.0 0.83 1.3619 0.9907 3214738 CHDI2_000654 OCCOc1ccccc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O02 compound treatment 169080.0 12700.0 0.87 172280.0 17700.0 1.32 1.543 0.9794 3214740 CHDI2_000655 OCCOc1ccccc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O03 compound treatment 170400.0 14000.0 0.96 168160.0 13600.0 1.01 1.3898 0.9996 3214742 CHDI2_000656 OCCOc1cccc(/C=N/NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O04 compound treatment 171360.0 15000.0 1.02 170360.0 15800.0 1.17 1.5519 0.9976 3214744 CHDI2_000657 OCCOc1cccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O05 compound treatment 176960.0 20600.0 1.4 173400.0 18800.0 1.4 1.9819 1.0 3214746 CHDI2_000658 OCCOc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O06 compound treatment 173120.0 16700.0 1.14 179160.0 24600.0 1.83 2.0999 0.9743 3214748 CHDI2_000659 OCCOc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O07 compound treatment 190080.0 33700.0 2.3 186400.0 31800.0 2.37 3.2985 0.9999 3214750 CHDI2_000660 COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O08 compound treatment 191360.0 35000.0 2.38 191200.0 36600.0 2.72 3.6128 0.9978 3214752 CHDI2_000661 COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O09 compound treatment 192040.0 35700.0 2.43 188960.0 34400.0 2.56 3.5277 0.9997 3214754 CHDI2_000662 COc1ccc(O)c(/C=N/NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O10 compound treatment 187160.0 30800.0 2.1 187600.0 33000.0 2.46 3.2209 0.9969 3214756 CHDI2_000663 COc1ccc(O)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O11 compound treatment 166640.0 10300.0 0.7 166880.0 12300.0 0.91 1.1412 0.9913 3214822 CHDI2_000664 CN(CCO)c1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O12 compound treatment 189440.0 33100.0 2.25 186440.0 31800.0 2.37 3.2698 0.9997 3553411 CHDI2_000665 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O13 compound treatment 213640.0 57300.0 3.9 219760.0 65200.0 4.85 6.19 0.9942 3214758 CHDI2_000666 COc1cc(/C=C/C=N/NC(=O)CCCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O14 compound treatment 192520.0 36100.0 2.46 203640.0 49000.0 3.65 4.3234 0.9817 3214760 CHDI2_000667 COc1cc(/C=C/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O15 compound treatment 185920.0 29500.0 2.01 185160.0 30600.0 2.27 3.0327 0.9982 3214762 CHDI2_000668 Cc1ccc(O)c(/C=N/NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O16 compound treatment 189440.0 33100.0 2.25 188160.0 33600.0 2.5 3.3603 0.9987 3214764 CHDI2_000669 Cc1ccc(O)c(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O17 compound treatment 182160.0 25800.0 1.76 182400.0 27800.0 2.07 2.7062 0.9967 3214766 CHDI2_000670 OCc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O18 compound treatment 184120.0 27700.0 1.89 184320.0 29700.0 2.21 2.9017 0.997 3214768 CHDI2_000671 OCc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O19 compound treatment 228080.0 71700.0 4.89 226360.0 71800.0 5.34 7.2334 0.999 3214770 CHDI2_000672 ONC(=O)CCCCCC(=O)N/N=C/c1ccc2ccccc2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O20 compound treatment 199760.0 43400.0 2.96 204360.0 49800.0 3.7 4.7104 0.9938 3214772 CHDI2_000673 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc3ccccc3c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O21 compound treatment 205040.0 48700.0 3.32 207040.0 52400.0 3.9 5.1059 0.9967 3214774 CHDI2_000674 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(o1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O22 compound treatment 177640.0 21300.0 1.45 183440.0 28800.0 2.15 2.543 0.9817 3214776 CHDI2_000675 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(o2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O23 mock treatment 158080.0 1700.0 0.12 158320.0 3730.0 0.28 0.2781 0.9252 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 O24 mock treatment 157120.0 741.0 0.05 154040.0 -555.0 -0.04 0.0065 0.1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P01 compound treatment 171480.0 15100.0 1.03 171320.0 16700.0 1.24 1.6082 0.9956 3214782 CHDI2_000676 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(o2)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P02 compound treatment 169880.0 13500.0 0.92 167960.0 13400.0 0.99 1.3542 0.9992 3215348 CHDI2_000677 OCCOc1ccccc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P03 compound treatment 177080.0 20700.0 1.41 179960.0 25400.0 1.89 2.3329 0.9897 3214786 CHDI2_000678 Cn1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P04 compound treatment 171360.0 15000.0 1.02 171520.0 16900.0 1.26 1.6129 0.9946 3215352 CHDI2_000679 OCCOc1cccc(/C=N/NC(=O)CCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P05 compound treatment 201440.0 45100.0 3.07 205040.0 50400.0 3.75 4.8271 0.995 3214790 CHDI2_000680 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cn(Cc3ccccc3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P06 compound treatment 174160.0 17800.0 1.21 171200.0 16600.0 1.24 1.7311 1.0 3215356 CHDI2_000681 OCCOc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P07 compound treatment 174960.0 18600.0 1.27 180760.0 26200.0 1.95 2.2728 0.9783 3214794 CHDI2_000682 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/C2=CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P08 compound treatment 189680.0 33300.0 2.27 188840.0 34200.0 2.55 3.4076 0.9983 3215360 CHDI2_000683 COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P09 compound treatment 172600.0 16200.0 1.11 176400.0 21800.0 1.62 1.9295 0.9825 3214798 CHDI2_000684 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P10 compound treatment 200040.0 43700.0 2.98 200760.0 46200.0 3.44 4.5344 0.9974 3215364 CHDI2_000685 COc1ccc(O)c(/C=N/NC(=O)CCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P11 compound treatment 178760.0 22400.0 1.53 177560.0 23000.0 1.71 2.2876 0.9984 3553474 CHDI2_000686 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P12 compound treatment 204880.0 48500.0 3.31 205520.0 50900.0 3.79 5.0182 0.9977 3553514 CHDI2_000687 ONC(=O)c1cccc(c1)C(=O)N/N=C/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P13 compound treatment 176120.0 19700.0 1.35 179800.0 25200.0 1.88 2.2782 0.9867 3214800 CHDI2_000688 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P14 compound treatment 207440.0 51100.0 3.48 214360.0 59800.0 4.45 5.6069 0.9926 3215368 CHDI2_000689 COc1cc(/C=C/C=N/NC(=O)CCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P15 compound treatment 170640.0 14300.0 0.97 178440.0 23800.0 1.77 1.9424 0.9599 3214804 CHDI2_000690 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P16 compound treatment 179920.0 23500.0 1.6 183440.0 28800.0 2.15 2.6529 0.9897 3215372 CHDI2_000691 Cc1ccc(O)c(/C=N/NC(=O)CCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P17 compound treatment 171360.0 15000.0 1.02 174280.0 19700.0 1.47 1.7582 0.9844 3214808 CHDI2_000692 C/C(=N\NC(=O)CCCCCC(=O)Nc1ccccc1O)/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P18 compound treatment 171960.0 15600.0 1.06 178320.0 23700.0 1.77 1.9997 0.9704 3215376 CHDI2_000693 OCc1ccc(/C=N/NC(=O)CCCCC(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P19 compound treatment 168560.0 12200.0 0.83 174000.0 19400.0 1.44 1.6085 0.9655 3214812 CHDI2_000694 CN(C)CCCOc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P20 compound treatment 204880.0 48500.0 3.31 209680.0 55100.0 4.1 5.2372 0.9943 3215380 CHDI2_000695 ONC(=O)CCCCC(=O)N/N=C/c1ccc2ccccc2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P21 compound treatment 185880.0 29500.0 2.01 193000.0 38400.0 2.86 3.4434 0.9852 3214816 CHDI2_000696 CCOc1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P22 compound treatment 190000.0 33600.0 2.29 192440.0 37800.0 2.82 3.6125 0.9948 3215384 CHDI2_000697 ONC(=O)CCCCC(=O)N/N=C/c1ccc(o1)c2cccc(Cl)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P23 mock treatment 157360.0 981.0 0.07 152440.0 -2160.0 -0.16 -0.0661 -0.3804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2404 P24 mock treatment 157880.0 1500.0 0.1 152880.0 -1720.0 -0.13 -0.0179 -0.1093 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A01 compound treatment 183320.0 27700.0 1.89 185120.0 30100.0 2.24 2.9171 0.9963 3214868 CHDI2_000698 ONC(=O)CCCCC(=O)N/N=C/c1c(O)ccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A02 compound treatment 170520.0 14900.0 1.01 169040.0 14000.0 1.04 1.4538 0.9999 3551921 CHDI2_000699 NNC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A03 compound treatment 192320.0 36700.0 2.5 181400.0 26400.0 1.96 3.1552 0.9929 3214872 CHDI2_000700 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A04 compound treatment 182680.0 27000.0 1.84 180560.0 25500.0 1.9 2.6463 0.9999 3552997 CHDI2_000701 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A05 compound treatment 172960.0 17300.0 1.18 175720.0 20700.0 1.54 1.923 0.9913 3214876 CHDI2_000702 ONC(=O)CCCCC(=O)N/N=C/c1ccc([N+](=O)[O-])c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A06 compound treatment 166640.0 11000.0 0.75 165480.0 10500.0 0.78 1.0794 0.9998 3553001 CHDI2_000703 COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A07 compound treatment 180200.0 24500.0 1.67 184200.0 29200.0 2.17 2.7183 0.9917 3214880 CHDI2_000704 ONC(=O)CCCCC(=O)N/N=C/c1cc(O)ccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A08 compound treatment 171360.0 15700.0 1.07 164240.0 9220.0 0.69 1.2417 0.9769 3553005 CHDI2_000705 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A09 compound treatment 178080.0 22400.0 1.53 168400.0 13400.0 1.0 1.7846 0.9785 3214884 CHDI2_000706 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)n2ccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A10 compound treatment 168600.0 12900.0 0.88 166800.0 11800.0 0.88 1.2433 1.0 3553009 CHDI2_000707 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc3OCCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A11 compound treatment 166200.0 10500.0 0.72 167720.0 12700.0 0.95 1.1761 0.9908 3214888 CHDI2_000708 ONC(=O)CCCCC(=O)N/N=C/c1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A12 compound treatment 180920.0 25300.0 1.72 181080.0 26100.0 1.94 2.5888 0.9982 3553013 CHDI2_000709 ONC(=O)c1cccc(c1)C(=O)N/N=C/COCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A13 compound treatment 176560.0 20900.0 1.42 174760.0 19700.0 1.47 2.046 0.9999 3553655 CHDI2_000710 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A14 compound treatment 173840.0 18200.0 1.24 177880.0 22900.0 1.7 2.0791 0.9879 3553589 CHDI2_000711 CCOc1cccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A15 compound treatment 170800.0 15100.0 1.03 167360.0 12300.0 0.92 1.3789 0.9983 3214892 CHDI2_000712 ONC(=O)CCCCC(=O)N/N=C/c1ccc(I)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A16 compound treatment 195160.0 39500.0 2.69 188080.0 33100.0 2.46 3.6437 0.999 3553017 CHDI2_000713 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A17 compound treatment 159840.0 4170.0 0.28 163200.0 8180.0 0.61 0.6316 0.94 3214896 CHDI2_000714 C/C=C(/C)\C=N\NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A18 compound treatment 171360.0 15700.0 1.07 175800.0 20800.0 1.55 1.85 0.9838 3553021 CHDI2_000715 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A19 compound treatment 170840.0 15200.0 1.03 169360.0 14300.0 1.07 1.4861 0.9999 3214972 CHDI2_000716 ONC(=O)CCCCC(=O)N/N=C/c1ccc(s1)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A20 compound treatment 163880.0 8210.0 0.56 163800.0 8780.0 0.65 0.8579 0.9971 3553025 CHDI2_000717 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A21 compound treatment 164960.0 9290.0 0.63 163560.0 8540.0 0.64 0.8973 1.0 3214904 CHDI2_000718 Cc1ccc(/C=N/NC(=O)CCCCC(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A22 compound treatment 171160.0 15500.0 1.06 170520.0 15500.0 1.15 1.5625 0.999 3553029 CHDI2_000719 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A23 mock treatment 150280.0 -5390.0 -0.37 150160.0 -4860.0 -0.36 -0.5156 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 A24 mock treatment 146840.0 -8830.0 -0.6 149960.0 -5060.0 -0.38 -0.6919 -0.9746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B01 compound treatment 167320.0 11700.0 0.79 165680.0 10700.0 0.79 1.1227 1.0 3551923 CHDI2_000720 NNC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B02 compound treatment 277760.0 122000.0 8.32 281600.0 127000.0 9.42 12.5474 0.9981 3553956 CHDI2_000721 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2c(O)ccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B03 compound treatment 174480.0 18800.0 1.28 180560.0 25500.0 1.9 2.251 0.9817 3553662 CHDI2_000722 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B04 compound treatment 201440.0 45800.0 3.12 196960.0 41900.0 3.12 4.4138 1.0 3553960 CHDI2_000723 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B05 compound treatment 172160.0 16500.0 1.12 165440.0 10400.0 0.78 1.3434 0.9835 3553666 CHDI2_000724 COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B06 compound treatment 180960.0 25300.0 1.72 182880.0 27900.0 2.07 2.6854 0.9958 3553964 CHDI2_000725 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc([N+](=O)[O-])c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B07 compound treatment 167480.0 11800.0 0.81 166080.0 11100.0 0.82 1.1515 0.9999 3553670 CHDI2_000726 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B08 compound treatment 195280.0 39600.0 2.7 200000.0 45000.0 3.35 4.2768 0.9943 3553968 CHDI2_000727 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(O)ccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B09 compound treatment 182600.0 26900.0 1.84 181720.0 26700.0 1.99 2.7035 0.9992 3553675 CHDI2_000728 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc3OCCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B10 compound treatment 213920.0 58300.0 3.97 199320.0 44300.0 3.3 5.1396 0.9957 3553971 CHDI2_000729 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)n3ccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B11 compound treatment 179280.0 23600.0 1.61 180920.0 25900.0 1.93 2.5013 0.996 3553679 CHDI2_000730 ONC(=O)c1ccc(cc1)C(=O)N/N=C/COCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B12 compound treatment 180400.0 24700.0 1.69 173760.0 18700.0 1.39 2.1785 0.9955 3553975 CHDI2_000731 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B13 compound treatment 241800.0 86100.0 5.87 244760.0 89700.0 6.68 8.875 0.9979 3552713 CHDI2_000732 Oc1ccc2ccccc2c1/C=N/NC(=O)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B14 compound treatment 177600.0 21900.0 1.5 175840.0 20800.0 1.55 2.153 0.9998 3552763 CHDI2_000733 COc1cc(/C=N/NC(=O)c2ccccn2)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B15 compound treatment 198560.0 42900.0 2.92 190760.0 35700.0 2.66 3.9486 0.9989 3553682 CHDI2_000734 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B16 compound treatment 175760.0 20100.0 1.37 172480.0 17500.0 1.3 1.8874 0.9997 3553978 CHDI2_000735 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(I)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B17 compound treatment 173600.0 17900.0 1.22 171560.0 16500.0 1.23 1.7349 1.0 3553686 CHDI2_000736 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B18 compound treatment 169560.0 13900.0 0.95 166640.0 11600.0 0.86 1.2812 0.999 3553981 CHDI2_000737 C/C=C(/C)\C=N\NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B19 compound treatment 169440.0 13800.0 0.94 171720.0 16700.0 1.24 1.5428 0.9905 3553690 CHDI2_000738 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B20 compound treatment 203280.0 47600.0 3.25 212600.0 57600.0 4.29 5.3256 0.9906 3553985 CHDI2_000739 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B21 compound treatment 174960.0 19300.0 1.32 173280.0 18300.0 1.36 1.891 0.9999 3553695 CHDI2_000740 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B22 compound treatment 203640.0 48000.0 3.27 210880.0 55900.0 4.16 5.2524 0.993 3553989 CHDI2_000741 Cc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B23 mock treatment 149960.0 -5710.0 -0.39 153000.0 -2020.0 -0.15 -0.3815 -0.9146 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 B24 mock treatment 147720.0 -7950.0 -0.54 149880.0 -5140.0 -0.38 -0.6537 -0.9855 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C01 compound treatment 167640.0 12000.0 0.82 162640.0 7620.0 0.57 0.9781 0.9841 3214952 CHDI2_000742 Cc1ccsc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C02 compound treatment 188600.0 32900.0 2.25 194560.0 39500.0 2.94 3.6685 0.9911 3553037 CHDI2_000743 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(Br)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C03 compound treatment 173320.0 17700.0 1.2 172040.0 17000.0 1.27 1.7467 0.9997 3214956 CHDI2_000744 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C04 compound treatment 185000.0 29300.0 2.0 180880.0 25900.0 1.92 2.775 0.9998 3553041 CHDI2_000745 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C05 compound treatment 180440.0 24800.0 1.69 178440.0 23400.0 1.74 2.4267 0.9999 3214960 CHDI2_000746 ONC(=O)CCCCC(=O)N/N=C/c1cccc2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C06 compound treatment 182520.0 26900.0 1.83 179960.0 24900.0 1.86 2.607 1.0 3553045 CHDI2_000747 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(O)ccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C07 compound treatment 175120.0 19500.0 1.33 178960.0 23900.0 1.78 2.1976 0.9894 3214968 CHDI2_000748 ONC(=O)CCCCC(=O)N/N=C/c1ccc2ccccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C08 compound treatment 296440.0 141000.0 9.6 283840.0 129000.0 9.59 13.5658 1.0 3553049 CHDI2_000749 COc1cc(Br)cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C09 compound treatment 182120.0 26500.0 1.8 184600.0 29600.0 2.2 2.8319 0.9951 3214900 CHDI2_000750 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C10 compound treatment 188800.0 33100.0 2.26 187200.0 32200.0 2.39 3.2908 0.9996 3553053 CHDI2_000751 COc1ccc(Br)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C11 compound treatment 173160.0 17500.0 1.19 182280.0 27300.0 2.03 2.2778 0.9679 3553658 CHDI2_000752 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C12 compound treatment 260360.0 105000.0 7.14 277600.0 123000.0 9.12 11.4981 0.9926 3553593 CHDI2_000753 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(I)cc(I)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C13 compound treatment 180400.0 24700.0 1.69 181040.0 26000.0 1.94 2.5616 0.9976 3214964 CHDI2_000754 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C14 compound treatment 189040.0 33400.0 2.28 188760.0 33700.0 2.51 3.3844 0.9988 3553057 CHDI2_000755 COc1ccc(Br)cc1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C15 compound treatment 179920.0 24300.0 1.65 167480.0 12500.0 0.93 1.8248 0.9626 3553517 CHDI2_000756 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C16 compound treatment 179120.0 23500.0 1.6 177720.0 22700.0 1.69 2.3252 0.9996 3553597 CHDI2_000757 CN(C)c1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C17 compound treatment 174480.0 18800.0 1.28 171080.0 16100.0 1.2 1.752 0.9994 3214976 CHDI2_000758 ONC(=O)CCCCC(=O)N/N=C/c1c(F)c(F)c(F)c(F)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C18 compound treatment 172320.0 16700.0 1.14 165200.0 10200.0 0.76 1.3385 0.9806 3553061 CHDI2_000759 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc3OCOc3cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C19 compound treatment 171880.0 16200.0 1.11 164440.0 9420.0 0.7 1.2773 0.9758 3214980 CHDI2_000760 ONC(=O)CCCCC(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C20 compound treatment 167200.0 11500.0 0.79 172880.0 17900.0 1.33 1.4958 0.9686 3553065 CHDI2_000761 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccnc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C21 compound treatment 179680.0 24000.0 1.64 166760.0 11700.0 0.87 1.7754 0.9567 3214984 CHDI2_000762 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C22 compound treatment 172320.0 16700.0 1.14 171080.0 16100.0 1.2 1.6479 0.9997 3553069 CHDI2_000763 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccncc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C23 mock treatment 149120.0 -6550.0 -0.45 153960.0 -1060.0 -0.08 -0.3715 -0.8196 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 C24 mock treatment 148600.0 -7070.0 -0.48 152520.0 -2500.0 -0.19 -0.4724 -0.9145 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D01 compound treatment 212760.0 57100.0 3.89 206880.0 51900.0 3.86 5.4815 1.0 3553703 CHDI2_000764 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(Br)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D02 compound treatment 174240.0 18600.0 1.27 176840.0 21800.0 1.62 2.0436 0.9924 3553995 CHDI2_000765 Cc1ccsc1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D03 compound treatment 178520.0 22900.0 1.56 182760.0 27700.0 2.06 2.5615 0.9904 3553706 CHDI2_000766 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D04 compound treatment 181320.0 25700.0 1.75 182640.0 27600.0 2.06 2.6902 0.9968 3553998 CHDI2_000767 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)c3ccc(cc3)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D05 compound treatment 183560.0 27900.0 1.9 180440.0 25400.0 1.89 2.6824 1.0 3553710 CHDI2_000768 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(O)ccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D06 compound treatment 218000.0 62300.0 4.25 206640.0 51600.0 3.84 5.7215 0.9987 3554002 CHDI2_000769 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D07 compound treatment 247400.0 91700.0 6.25 273960.0 119000.0 8.85 10.6817 0.9855 3553714 CHDI2_000770 COc1cc(Br)cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D08 compound treatment 211680.0 56000.0 3.82 213720.0 58700.0 4.37 5.7894 0.9978 3554006 CHDI2_000771 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D09 compound treatment 186640.0 31000.0 2.11 189880.0 34900.0 2.59 3.3277 0.9948 3553718 CHDI2_000772 COc1ccc(Br)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D10 compound treatment 190760.0 35100.0 2.39 188600.0 33600.0 2.5 3.4589 0.9998 3554009 CHDI2_000773 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D11 compound treatment 189080.0 33400.0 2.28 181160.0 26100.0 1.95 2.9864 0.9969 3552716 CHDI2_000774 Oc1ccc(/C=N/NC(=O)c2ccccn2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D12 compound treatment 176040.0 20400.0 1.39 176160.0 21100.0 1.57 2.0946 0.9981 3552765 CHDI2_000775 Fc1c(F)c(F)c(/C=N/NC(=O)c2ccccn2)c(F)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D13 compound treatment 188920.0 33300.0 2.27 189320.0 34300.0 2.55 3.4081 0.9982 3553722 CHDI2_000776 COc1ccc(Br)cc1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D14 compound treatment 197880.0 42200.0 2.88 199440.0 44400.0 3.31 4.3726 0.9976 3554013 CHDI2_000777 COc1cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D15 compound treatment 167840.0 12200.0 0.83 167120.0 12100.0 0.9 1.2235 0.9992 3552720 CHDI2_000778 Oc1cc(/C=N/NC(=O)c2ccccn2)ccc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D16 compound treatment 170120.0 14500.0 0.99 173640.0 18600.0 1.39 1.6766 0.9861 3552767 CHDI2_000779 C=CCC/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D17 compound treatment 200600.0 44900.0 3.06 187760.0 32700.0 2.44 3.8891 0.9936 3553726 CHDI2_000780 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc3OCOc3cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D18 compound treatment 191280.0 35600.0 2.43 179920.0 24900.0 1.85 3.0272 0.9911 3554017 CHDI2_000781 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2c(F)c(F)c(F)c(F)c2F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D19 compound treatment 179800.0 24100.0 1.65 165760.0 10700.0 0.8 1.7285 0.945 3553730 CHDI2_000782 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccnc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D20 compound treatment 168600.0 12900.0 0.88 171120.0 16100.0 1.2 1.4707 0.9886 3554021 CHDI2_000783 ONC(=O)c1ccc(cc1)C(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D21 compound treatment 181160.0 25500.0 1.74 181160.0 26100.0 1.95 2.6046 0.9984 3553734 CHDI2_000784 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccncc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D22 compound treatment 189440.0 33800.0 2.3 189720.0 34700.0 2.58 3.4542 0.9984 3554025 CHDI2_000785 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D23 mock treatment 152880.0 -2790.0 -0.19 152520.0 -2500.0 -0.19 -0.266 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 D24 mock treatment 148280.0 -7390.0 -0.5 145000.0 -10000.0 -0.75 -0.8835 -0.9817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E01 compound treatment 177400.0 21700.0 1.48 173760.0 18700.0 1.39 2.0339 0.9995 3553522 CHDI2_000786 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E02 compound treatment 258400.0 103000.0 7.0 262320.0 107000.0 7.99 10.5995 0.9979 3553601 CHDI2_000787 CCn1c2ccccc2c3cc(/C=N/NC(=O)c4cccc(c4)C(=O)NO)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E03 compound treatment 241120.0 85500.0 5.83 249240.0 94200.0 7.01 9.078 0.9958 3215028 CHDI2_000788 ONC(=O)CCCCC(=O)N/N=C/c1cn(c2ccccc12)S(=O)(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E04 compound treatment 196080.0 40400.0 2.76 192080.0 37100.0 2.76 3.8985 1.0 3553077 CHDI2_000789 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(Br)s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E05 compound treatment 179880.0 24200.0 1.65 178840.0 23800.0 1.77 2.4208 0.9994 3215032 CHDI2_000790 ONC(=O)CCCCC(=O)N/N=C/c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E06 compound treatment 200040.0 44400.0 3.03 190440.0 35400.0 2.64 4.0031 0.9976 3553081 CHDI2_000791 COc1cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E07 compound treatment 176440.0 20800.0 1.42 186840.0 31800.0 2.37 2.676 0.9698 3215036 CHDI2_000792 ONC(=O)CCCCC(=O)N/N=C/c1cccnc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E08 compound treatment 275720.0 120000.0 8.18 281280.0 126000.0 9.4 12.4322 0.9976 3553084 CHDI2_000793 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCc3ccccc3)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E09 compound treatment 179200.0 23500.0 1.6 174360.0 19300.0 1.44 2.1522 0.9985 3553525 CHDI2_000794 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E10 compound treatment 245480.0 89800.0 6.12 224240.0 69200.0 5.15 7.9725 0.9963 3553605 CHDI2_000795 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(c(F)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E11 compound treatment 182920.0 27300.0 1.86 181160.0 26100.0 1.95 2.6894 0.9997 3215040 CHDI2_000796 Cc1ncc(CO)c(/C=N/NC(=O)CCCCC(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E12 compound treatment 181920.0 26300.0 1.79 177840.0 22800.0 1.7 2.4665 0.9997 3553088 CHDI2_000797 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E13 compound treatment 182120.0 26500.0 1.8 179440.0 24400.0 1.82 2.5603 1.0 3215044 CHDI2_000798 ONC(=O)CCCCC(=O)N/N=C/c1ccc[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E14 compound treatment 185160.0 29500.0 2.01 180520.0 25500.0 1.9 2.7637 0.9996 3553092 CHDI2_000799 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E15 compound treatment 188160.0 32500.0 2.22 186720.0 31700.0 2.36 3.2346 0.9995 3215048 CHDI2_000800 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)N2CCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E16 compound treatment 203240.0 47600.0 3.24 196680.0 41700.0 3.1 4.4858 0.9997 3553096 CHDI2_000801 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E17 compound treatment 178240.0 22600.0 1.54 175080.0 20100.0 1.49 2.1438 0.9999 3553530 CHDI2_000802 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E18 compound treatment 181760.0 26100.0 1.78 178920.0 23900.0 1.78 2.5156 1.0 3553608 CHDI2_000803 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(o2)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E19 compound treatment 182200.0 26500.0 1.81 179760.0 24700.0 1.84 2.581 1.0 3215052 CHDI2_000804 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E20 compound treatment 181400.0 25700.0 1.75 167760.0 12700.0 0.95 1.9109 0.9582 3553100 CHDI2_000805 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(c2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E21 compound treatment 178800.0 23100.0 1.58 172520.0 17500.0 1.3 2.0361 0.9955 3215056 CHDI2_000806 CCCCCCC/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E22 compound treatment 164520.0 8850.0 0.6 164880.0 9860.0 0.73 0.9456 0.9953 3553104 CHDI2_000807 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E23 mock treatment 162360.0 6690.0 0.46 156000.0 978.0 0.07 0.3741 0.8096 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 E24 mock treatment 158160.0 2490.0 0.17 155960.0 938.0 0.07 0.1696 0.9226 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F01 compound treatment 208080.0 52400.0 3.57 200560.0 45500.0 3.39 4.9233 0.9997 1936929 CHDI2_000808 Oc1ccc([N+](=O)[O-])c(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F02 compound treatment 109840.0 -45800.0 -3.12 108600.0 -46400.0 -3.46 -4.6523 -0.9987 3552769 CHDI2_000809 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F03 compound treatment 202800.0 47100.0 3.21 204720.0 49700.0 3.7 4.8877 0.9975 3553741 CHDI2_000810 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(Br)s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F04 compound treatment 302280.0 147000.0 10.0 304360.0 149000.0 11.11 14.9273 0.9986 3554032 CHDI2_000811 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cn(c3ccccc23)S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F05 compound treatment 194720.0 39100.0 2.66 197400.0 42400.0 3.15 4.1129 0.9964 3553745 CHDI2_000812 COc1cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F06 compound treatment 185160.0 29500.0 2.01 185720.0 30700.0 2.28 3.0374 0.998 3554034 CHDI2_000813 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F07 compound treatment 268560.0 113000.0 7.7 256960.0 102000.0 7.59 10.8072 1.0 3553748 CHDI2_000814 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCc3ccccc3)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F08 compound treatment 185760.0 30100.0 2.05 180880.0 25900.0 1.92 2.8116 0.9995 3554036 CHDI2_000815 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F09 compound treatment 169840.0 14200.0 0.97 167320.0 12300.0 0.92 1.3305 0.9996 3552725 CHDI2_000816 O=C(N/N=C/c1ccc(cc1)n2ccnc2)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F10 compound treatment 167200.0 11500.0 0.79 166520.0 11500.0 0.86 1.1611 0.9991 3552771 CHDI2_000817 O=C(N/N=C/c1cccc(Oc2ccccc2)c1)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F11 compound treatment 177240.0 21600.0 1.47 176240.0 21200.0 1.58 2.1567 0.9994 3553752 CHDI2_000818 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F12 compound treatment 190800.0 35100.0 2.4 186960.0 31900.0 2.38 3.3745 1.0 3554038 CHDI2_000819 Cc1ncc(CO)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F13 compound treatment 180800.0 25100.0 1.71 179680.0 24700.0 1.84 2.5093 0.9994 3553756 CHDI2_000820 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F14 compound treatment 184720.0 29100.0 1.98 181400.0 26400.0 1.96 2.7888 1.0 3554040 CHDI2_000821 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F15 compound treatment 269600.0 114000.0 7.77 248760.0 93700.0 6.98 10.4258 0.9986 3553759 CHDI2_000822 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F16 compound treatment 197800.0 42100.0 2.87 192880.0 37900.0 2.82 4.0236 1.0 3554042 CHDI2_000823 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F17 compound treatment 174160.0 18500.0 1.26 166960.0 11900.0 0.89 1.5198 0.9853 3552730 CHDI2_000824 O=C(N/N=C/c1c[nH]c2ccccc12)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F18 compound treatment 175280.0 19600.0 1.34 174680.0 19700.0 1.46 1.9801 0.999 3552773 CHDI2_000825 O=C(N/N=C/c1cn(c2ccccc12)S(=O)(=O)c3ccccc3)c4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F19 compound treatment 181760.0 26100.0 1.78 172640.0 17600.0 1.31 2.1851 0.9887 3553763 CHDI2_000826 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(c2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F20 compound treatment 193040.0 37400.0 2.55 183080.0 28100.0 2.09 3.2783 0.9951 3554044 CHDI2_000827 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F21 compound treatment 181680.0 26000.0 1.77 171000.0 16000.0 1.19 2.0949 0.9811 3553767 CHDI2_000828 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F22 compound treatment 180040.0 24400.0 1.66 176160.0 21100.0 1.57 2.2874 0.9996 3554046 CHDI2_000829 CCCCCCC/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F23 mock treatment 160560.0 4890.0 0.33 155120.0 97.5 0.01 0.2411 0.7223 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 F24 mock treatment 151560.0 -4110.0 -0.28 151720.0 -3300.0 -0.25 -0.3718 -0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G01 compound treatment 176600.0 20900.0 1.43 176160.0 21100.0 1.57 2.1216 0.9988 3215102 CHDI2_000830 ONC(=O)CCCCC(=O)N/N=C/c1cccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G02 compound treatment 184200.0 28500.0 1.95 184080.0 29100.0 2.16 2.9048 0.9986 3553111 CHDI2_000831 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G03 compound treatment 184640.0 29000.0 1.98 190080.0 35100.0 2.61 3.2418 0.9906 3553531 CHDI2_000832 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G04 compound treatment 204840.0 49200.0 3.35 203000.0 48000.0 3.57 4.8955 0.9995 3553612 CHDI2_000833 Cn1cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G05 compound treatment 185000.0 29300.0 2.0 190240.0 35200.0 2.62 3.2675 0.9911 3215106 CHDI2_000834 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G06 compound treatment 188440.0 32800.0 2.23 194240.0 39200.0 2.92 3.6439 0.9913 3553115 CHDI2_000835 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccnc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G07 compound treatment 402800.0 247000.0 16.85 417400.0 262000.0 19.53 25.7222 0.9973 3215110 CHDI2_000836 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G08 compound treatment 204720.0 49100.0 3.34 206360.0 51300.0 3.82 5.0666 0.9978 3553118 CHDI2_000837 ONC(=O)c1cccc(c1)C(=O)N/N=C/C=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G09 compound treatment 292280.0 137000.0 9.31 297640.0 143000.0 10.61 14.0916 0.9979 3215114 CHDI2_000838 ONC(=O)CCCCC(=O)N/N=C/c1c(O)cc(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G10 compound treatment 199280.0 43600.0 2.97 208160.0 53100.0 3.95 4.8991 0.9901 3553123 CHDI2_000839 C[C@H](CCC=C(C)C)C/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G11 compound treatment 188320.0 32700.0 2.23 190360.0 35300.0 2.63 3.4339 0.9966 3215118 CHDI2_000840 COc1cc(OC)c(/C=N/NC(=O)CCCCC(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G12 compound treatment 194560.0 38900.0 2.65 191480.0 36500.0 2.71 3.7937 0.9999 3553127 CHDI2_000841 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G13 compound treatment 186600.0 30900.0 2.11 181680.0 26700.0 1.98 2.8942 0.9995 3215122 CHDI2_000842 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G14 compound treatment 195480.0 39800.0 2.71 182320.0 27300.0 2.03 3.356 0.9898 3553128 CHDI2_000843 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G15 compound treatment 186400.0 30700.0 2.1 182920.0 27900.0 2.08 2.9498 1.0 3215126 CHDI2_000844 CC(C)(C)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G16 compound treatment 186120.0 30500.0 2.08 183240.0 28200.0 2.1 2.9531 1.0 3553133 CHDI2_000845 ONC(=O)c1cccc(c1)C(=O)N/N=C/C2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G17 compound treatment 183920.0 28300.0 1.93 182120.0 27100.0 2.02 2.7881 0.9997 3215130 CHDI2_000846 CC1=C(C/C=N/NC(=O)CCCCC(=O)NO)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G18 compound treatment 199760.0 44100.0 3.01 198760.0 43700.0 3.26 4.4275 0.9992 3553137 CHDI2_000847 COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G19 compound treatment 182440.0 26800.0 1.83 179200.0 24200.0 1.8 2.5631 1.0 3553533 CHDI2_000848 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G20 compound treatment 214840.0 59200.0 4.03 213720.0 58700.0 4.37 5.9418 0.9992 3553614 CHDI2_000849 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cn(Cc3ccccc3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G21 compound treatment 179160.0 23500.0 1.6 178480.0 23500.0 1.75 2.3671 0.9991 3215134 CHDI2_000850 NC(=O)COc1ccccc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G22 compound treatment 260880.0 105000.0 7.17 254080.0 99100.0 7.37 10.2854 0.9999 3553141 CHDI2_000851 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(Br)cc(Br)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G23 mock treatment 167440.0 11800.0 0.8 162640.0 7620.0 0.57 0.9685 0.9855 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 G24 mock treatment 154280.0 -1390.0 -0.09 153640.0 -1380.0 -0.1 -0.1396 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H01 compound treatment 179800.0 24100.0 1.65 179040.0 24000.0 1.79 2.4274 0.9991 3553774 CHDI2_000852 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H02 compound treatment 181720.0 26100.0 1.78 182440.0 27400.0 2.04 2.6989 0.9976 3554050 CHDI2_000853 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H03 compound treatment 162320.0 6650.0 0.45 168760.0 13700.0 1.02 1.0437 0.9331 3552734 CHDI2_000854 Ic1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H04 compound treatment 170840.0 15200.0 1.03 170680.0 15700.0 1.17 1.5555 0.9982 3552775 CHDI2_000855 O=C(N/N=C/c1ccccn1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H05 compound treatment 191480.0 35800.0 2.44 184600.0 29600.0 2.2 3.2831 0.9987 3553778 CHDI2_000856 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccnc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H06 compound treatment 190120.0 34500.0 2.35 190240.0 35200.0 2.62 3.5144 0.9985 3554054 CHDI2_000857 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H07 compound treatment 215600.0 59900.0 4.09 211280.0 56300.0 4.19 5.85 0.9999 3553782 CHDI2_000858 ONC(=O)c1ccc(cc1)C(=O)N/N=C/C=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H08 compound treatment 437600.0 282000.0 19.22 420720.0 266000.0 19.78 27.5746 0.9999 3554058 CHDI2_000859 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)c(O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H09 compound treatment 210320.0 54700.0 3.73 211600.0 56600.0 4.21 5.6123 0.9981 3553785 CHDI2_000860 C[C@H](CCC=C(C)C)C/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H10 compound treatment 449120.0 293000.0 20.01 451160.0 296000.0 22.04 29.732 0.9988 3554062 CHDI2_000861 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2c(O)cc(O)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H11 compound treatment 205320.0 49700.0 3.39 201720.0 46700.0 3.48 4.8513 0.9999 3553788 CHDI2_000862 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H12 compound treatment 190760.0 35100.0 2.39 190640.0 35600.0 2.65 3.5663 0.9987 3554066 CHDI2_000863 COc1cc(OC)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H13 compound treatment 189000.0 33300.0 2.27 189960.0 34900.0 2.6 3.4456 0.9977 3553791 CHDI2_000864 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H14 compound treatment 189560.0 33900.0 2.31 186880.0 31900.0 2.37 3.3106 0.9999 3554070 CHDI2_000865 COc1cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H15 compound treatment 186160.0 30500.0 2.08 184320.0 29300.0 2.18 3.0119 0.9997 3553793 CHDI2_000866 ONC(=O)c1ccc(cc1)C(=O)N/N=C/C2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H16 compound treatment 186440.0 30800.0 2.1 183160.0 28100.0 2.09 2.9644 1.0 3554074 CHDI2_000867 CC(C)(C)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H17 compound treatment 219360.0 63700.0 4.34 214040.0 59000.0 4.39 6.1765 1.0 3553797 CHDI2_000868 COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H18 compound treatment 210040.0 54400.0 3.71 208880.0 53900.0 4.01 5.4557 0.9992 3554078 CHDI2_000869 CC1=C(C/C=N/NC(=O)c2ccc(cc2)C(=O)NO)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H19 compound treatment 179160.0 23500.0 1.6 184480.0 29500.0 2.19 2.6829 0.9881 3552737 CHDI2_000870 C/C=C(/C)\C=N\NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H20 compound treatment 164920.0 9250.0 0.63 165680.0 10700.0 0.79 1.007 0.9936 3552777 CHDI2_000871 O=C(N/N=C/c1cccnc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H21 compound treatment 314120.0 158000.0 10.8 282680.0 128000.0 9.5 14.3571 0.998 3553801 CHDI2_000872 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(Br)cc(Br)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H22 compound treatment 195600.0 39900.0 2.72 190480.0 35500.0 2.64 3.7912 0.9999 3554082 CHDI2_000873 NC(=O)COc1ccccc1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H23 mock treatment 158640.0 2970.0 0.2 161200.0 6180.0 0.46 0.4685 0.9323 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 H24 mock treatment 156720.0 1050.0 0.07 155520.0 498.0 0.04 0.077 0.9525 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I01 compound treatment 173920.0 18300.0 1.24 174600.0 19600.0 1.46 1.9103 0.9969 3215181 CHDI2_000874 ONC(=O)CCCCC(=O)NN=C1CCCCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I02 compound treatment 188600.0 32900.0 2.25 191000.0 36000.0 2.68 3.4811 0.9962 3553148 CHDI2_000875 COc1cc(Cl)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I03 compound treatment 180200.0 24500.0 1.67 181720.0 26700.0 1.99 2.5878 0.9963 3215183 CHDI2_000876 ONC(=O)CCCCC(=O)NN=C1CCCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I04 compound treatment 248320.0 92700.0 6.32 265640.0 111000.0 8.23 10.2882 0.9914 3553152 CHDI2_000877 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I05 compound treatment 262360.0 107000.0 7.27 252520.0 97500.0 7.26 10.2746 1.0 3553537 CHDI2_000878 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(Oc3ccccc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I06 compound treatment 191880.0 36200.0 2.47 186080.0 31100.0 2.31 3.3803 0.9995 3553618 CHDI2_000879 ONC(=O)c1cccc(c1)C(=O)N/N=C/C2=CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I07 compound treatment 188160.0 32500.0 2.22 180000.0 25000.0 1.86 2.881 0.9962 3215185 CHDI2_000880 ONC(=O)CCCCC(=O)NN=C1CCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I08 compound treatment 271360.0 116000.0 7.89 250240.0 95200.0 7.09 10.5885 0.9986 3553156 CHDI2_000881 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(Br)cc([N+](=O)[O-])c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I09 compound treatment 193760.0 38100.0 2.6 187080.0 32100.0 2.39 3.5236 0.9991 3214824 CHDI2_000882 NNC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I10 compound treatment 277440.0 122000.0 8.3 270520.0 115000.0 8.6 11.9489 0.9998 3553212 CHDI2_000883 CCN(CC)c1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I11 compound treatment 185360.0 29700.0 2.02 184640.0 29600.0 2.2 2.9902 0.9991 3215188 CHDI2_000884 COc1cc(Br)c(/C=N/NC(=O)CCCCC(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I12 compound treatment 185640.0 30000.0 2.04 182480.0 27500.0 2.04 2.89 1.0 3553216 CHDI2_000885 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc3OCCc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I13 compound treatment 201000.0 45300.0 3.09 195640.0 40600.0 3.02 4.3231 0.9999 3215192 CHDI2_000886 ONC(=O)CCCCC(=O)N/N=C/CCC1CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I14 compound treatment 419040.0 263000.0 17.96 405400.0 250000.0 18.63 25.8736 0.9998 3553220 CHDI2_000887 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I15 compound treatment 260760.0 105000.0 7.16 262320.0 107000.0 7.99 10.7132 0.9985 3215196 CHDI2_000888 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I16 compound treatment 322800.0 167000.0 11.39 312840.0 158000.0 11.75 16.3628 0.9999 3553224 CHDI2_000889 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I17 compound treatment 193800.0 38100.0 2.6 192400.0 37400.0 2.78 3.8055 0.9994 3215200 CHDI2_000890 ONC(=O)CCCCC(=O)N/N=C/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I18 compound treatment 443720.0 288000.0 19.64 446600.0 292000.0 21.7 29.2317 0.9988 3553228 CHDI2_000891 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(O)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I19 compound treatment 189520.0 33900.0 2.31 184440.0 29400.0 2.19 3.1802 0.9997 3214824 CHDI2_000892 NNC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I20 compound treatment 275120.0 119000.0 8.14 282760.0 128000.0 9.51 12.4812 0.997 3553231 CHDI2_000893 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I21 compound treatment 180240.0 24600.0 1.68 174880.0 19900.0 1.48 2.2297 0.998 3553541 CHDI2_000894 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc[n+]([O-])cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I22 compound treatment 169120.0 13500.0 0.92 168200.0 13200.0 0.98 1.3421 0.9994 3553622 CHDI2_000895 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I23 mock treatment 161200.0 5530.0 0.38 157880.0 2860.0 0.21 0.4172 0.9632 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 I24 mock treatment 155640.0 -26.3 0.0 153440.0 -1580.0 -0.12 -0.0845 -0.7178 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J01 compound treatment 196720.0 41100.0 2.8 193040.0 38000.0 2.83 3.9799 1.0 3553809 CHDI2_000896 COc1cc(Cl)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J02 compound treatment 181960.0 26300.0 1.79 183680.0 28700.0 2.13 2.7758 0.9963 3554238 CHDI2_000897 ONC(=O)c1ccc(cc1)C(=O)NN=C2CCCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J03 compound treatment 288600.0 133000.0 9.06 284840.0 130000.0 9.66 13.2405 0.9995 3553812 CHDI2_000898 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J04 compound treatment 183440.0 27800.0 1.89 187520.0 32500.0 2.42 3.0492 0.9927 3554236 CHDI2_000899 ONC(=O)c1ccc(cc1)C(=O)NN=C2CCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J05 compound treatment 191080.0 35400.0 2.41 181920.0 26900.0 2.0 3.1228 0.9957 3552741 CHDI2_000900 [O-][N+](=O)c1ccc(/C=N/NC(=O)c2ccccn2)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J06 compound treatment 187360.0 31700.0 2.16 185960.0 30900.0 2.3 3.1561 0.9995 3552779 CHDI2_000901 Cc1ncc(CO)c(/C=N/NC(=O)c2ccccn2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J07 compound treatment 246040.0 90400.0 6.16 241080.0 86100.0 6.4 8.8858 0.9998 3553816 CHDI2_000902 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(Br)cc([N+](=O)[O-])c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J08 compound treatment 202880.0 47200.0 3.22 205760.0 50700.0 3.78 4.9463 0.9968 3554206 CHDI2_000903 ONC(=O)c1ccc(cc1)C(=O)N/N=C/Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J09 compound treatment 297960.0 142000.0 9.7 279200.0 124000.0 9.24 13.3949 0.9997 3553820 CHDI2_000904 CCN(CC)c1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J10 compound treatment 183840.0 28200.0 1.92 180680.0 25700.0 1.91 2.7085 1.0 3554209 CHDI2_000905 COC(=O)c1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J11 compound treatment 191480.0 35800.0 2.44 188040.0 33000.0 2.46 3.4642 1.0 3553823 CHDI2_000906 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc3OCCc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J12 compound treatment 217720.0 62100.0 4.23 214880.0 59900.0 4.46 6.1417 0.9997 3554090 CHDI2_000907 COc1cc(Br)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J13 compound treatment 435320.0 280000.0 19.07 434200.0 279000.0 20.78 28.1741 0.9991 3553827 CHDI2_000908 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J14 compound treatment 285800.0 130000.0 8.87 275240.0 120000.0 8.95 12.6003 1.0 3554213 CHDI2_000909 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc3ccccc3n2S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J15 compound treatment 305920.0 150000.0 10.24 322600.0 168000.0 12.47 16.0627 0.9952 3553831 CHDI2_000910 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J16 compound treatment 334720.0 179000.0 12.21 314320.0 159000.0 11.86 17.0154 0.9999 3554094 CHDI2_000911 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J17 compound treatment 385120.0 229000.0 15.64 404040.0 249000.0 18.53 24.1668 0.9964 3553835 CHDI2_000912 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(O)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J18 compound treatment 210280.0 54600.0 3.72 208400.0 53400.0 3.97 5.442 0.9995 3554098 CHDI2_000913 ONC(=O)c1ccc(cc1)C(=O)N/N=C/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J19 compound treatment 275760.0 120000.0 8.19 274360.0 119000.0 8.88 12.07 0.9992 3553839 CHDI2_000914 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J20 compound treatment 189640.0 34000.0 2.32 191480.0 36500.0 2.71 3.5565 0.9969 3554217 CHDI2_000915 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J21 compound treatment 173640.0 18000.0 1.23 171760.0 16700.0 1.25 1.7473 1.0 3552745 CHDI2_000916 Cc1ccc(/C=N/NC(=O)c2ccccn2)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J22 compound treatment 167680.0 12000.0 0.82 171480.0 16500.0 1.22 1.4453 0.9809 1936582 CHDI2_000917 O=C(N/N=C/c1ccc[nH]1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J23 mock treatment 162480.0 6810.0 0.46 159600.0 4580.0 0.34 0.5694 0.9884 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 J24 mock treatment 154160.0 -1510.0 -0.1 154400.0 -623.0 -0.05 -0.1054 -0.9353 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K01 compound treatment 172800.0 17100.0 1.17 169560.0 14500.0 1.08 1.5911 0.9993 3215240 CHDI2_000918 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K02 compound treatment 178800.0 23100.0 1.58 176360.0 21300.0 1.59 2.2382 1.0 3553239 CHDI2_000919 COc1cccc(OC)c1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K03 compound treatment 179480.0 23800.0 1.62 180920.0 25900.0 1.93 2.5109 0.9964 3215244 CHDI2_000920 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K04 compound treatment 184120.0 28500.0 1.94 186840.0 31800.0 2.37 3.0462 0.9951 3553243 CHDI2_000921 COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K05 compound treatment 185280.0 29600.0 2.02 175160.0 20100.0 1.5 2.4874 0.9892 3215248 CHDI2_000922 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K06 compound treatment 204560.0 48900.0 3.33 203120.0 48100.0 3.58 4.8884 0.9994 3553247 CHDI2_000923 COc1cc(O)cc(OC)c1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K07 compound treatment 208720.0 53100.0 3.62 202160.0 47100.0 3.51 5.0384 0.9999 3553544 CHDI2_000924 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K08 compound treatment 180360.0 24700.0 1.68 185640.0 30600.0 2.28 2.8018 0.9889 3553623 CHDI2_000925 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K09 compound treatment 182840.0 27200.0 1.85 176520.0 21500.0 1.6 2.4414 0.9973 3215251 CHDI2_000926 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K10 compound treatment 184160.0 28500.0 1.94 180560.0 25500.0 1.9 2.7176 0.9999 3553250 CHDI2_000927 CC1(C)COC(CCC/C=N/NC(=O)c2cccc(c2)C(=O)NO)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K11 compound treatment 180760.0 25100.0 1.71 185760.0 30700.0 2.29 2.8274 0.9898 3215253 CHDI2_000928 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K12 compound treatment 226000.0 70300.0 4.8 216960.0 61900.0 4.61 6.6503 0.9998 3553254 CHDI2_000929 Cc1nnc(Sc2ccc(/C=N/NC(=O)c3cccc(c3)C(=O)NO)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K13 compound treatment 183480.0 27800.0 1.9 179920.0 24900.0 1.85 2.6512 0.9999 3215256 CHDI2_000930 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K14 compound treatment 201240.0 45600.0 3.11 195440.0 40400.0 3.01 4.3241 0.9999 3553258 CHDI2_000931 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(Br)cs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K15 compound treatment 185320.0 29700.0 2.02 184800.0 29800.0 2.22 2.9967 0.9989 3553549 CHDI2_000932 Cc1ccccc1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K16 compound treatment 188040.0 32400.0 2.21 179920.0 24900.0 1.85 2.871 0.9962 3553627 CHDI2_000933 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2cccc(c2)C(=O)NO)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K17 compound treatment 189200.0 33500.0 2.29 185040.0 30000.0 2.23 3.1964 0.9999 3215260 CHDI2_000934 ONC(=O)CCCCC(=O)N/N=C/c1ccc(Oc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K18 compound treatment 187360.0 31700.0 2.16 181880.0 26900.0 2.0 2.9414 0.9992 3553262 CHDI2_000935 CC(C)(C)OC(=O)NC/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K19 compound treatment 171280.0 15600.0 1.06 173040.0 18000.0 1.34 1.7009 0.9935 3215264 CHDI2_000936 ONC(=O)CCCCC(=O)N/N=C/c1cc[n+]([O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K20 compound treatment 296680.0 141000.0 9.61 296440.0 141000.0 10.53 14.2405 0.999 3553266 CHDI2_000937 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K21 compound treatment 178600.0 22900.0 1.56 180680.0 25700.0 1.91 2.4559 0.9951 3215268 CHDI2_000938 ONC(=O)CCCCC(=O)N/N=C/c1ccc2ccccc2n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K22 compound treatment 173760.0 18100.0 1.23 173720.0 18700.0 1.39 1.8563 0.9982 3553269 CHDI2_000939 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(F)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K23 mock treatment 160120.0 4450.0 0.3 160760.0 5740.0 0.43 0.5167 0.986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 K24 mock treatment 156200.0 534.0 0.04 152440.0 -2580.0 -0.19 -0.1102 -0.5632 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L01 compound treatment 175960.0 20300.0 1.38 172680.0 17700.0 1.31 1.9076 0.9997 3553847 CHDI2_000940 COc1cccc(OC)c1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L02 compound treatment 175960.0 20300.0 1.38 177840.0 22800.0 1.7 2.1792 0.9948 3554102 CHDI2_000941 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L03 compound treatment 181840.0 26200.0 1.78 186840.0 31800.0 2.37 2.9363 0.9903 3553851 CHDI2_000942 COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L04 compound treatment 182560.0 26900.0 1.83 179840.0 24800.0 1.85 2.6026 1.0 3554105 CHDI2_000943 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L05 compound treatment 196080.0 40400.0 2.76 198400.0 43400.0 3.23 4.2311 0.9969 3553855 CHDI2_000944 COc1cc(O)cc(OC)c1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L06 compound treatment 181760.0 26100.0 1.78 174680.0 19700.0 1.46 2.2925 0.9953 3554109 CHDI2_000945 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L07 compound treatment 161560.0 5890.0 0.4 156560.0 1540.0 0.11 0.365 0.8737 3552749 CHDI2_000946 Cc1[nH]cnc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L08 compound treatment 163800.0 8130.0 0.55 173720.0 18700.0 1.39 1.3761 0.9186 3552781 CHDI2_000947 O=C(N/N=C/c1ccc(cc1)N2CCCC2)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L09 compound treatment 185200.0 29500.0 2.01 183040.0 28000.0 2.09 2.8983 0.9998 3553858 CHDI2_000948 CC1(C)COC(CCC/C=N/NC(=O)c2ccc(cc2)C(=O)NO)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L10 compound treatment 179840.0 24200.0 1.65 185200.0 30200.0 2.25 2.7536 0.9884 3554113 CHDI2_000949 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L11 compound treatment 228040.0 72400.0 4.93 227520.0 72500.0 5.4 7.3044 0.999 3553862 CHDI2_000950 Cc1nnc(Sc2ccc(/C=N/NC(=O)c3ccc(cc3)C(=O)NO)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L12 compound treatment 184200.0 28500.0 1.95 175680.0 20700.0 1.54 2.4627 0.9932 3554115 CHDI2_000951 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L13 compound treatment 215520.0 59900.0 4.08 211080.0 56100.0 4.17 5.8356 0.9999 3553866 CHDI2_000952 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(Br)cs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L14 compound treatment 180520.0 24900.0 1.69 179560.0 24500.0 1.83 2.4895 0.9993 3554117 CHDI2_000953 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L15 compound treatment 148400.0 -7270.0 -0.5 152000.0 -3020.0 -0.22 -0.5094 -0.9362 3552753 CHDI2_000954 Cc1ccsc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L16 compound treatment 183400.0 27700.0 1.89 187960.0 32900.0 2.45 3.0704 0.9918 3552783 CHDI2_000955 Oc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L17 compound treatment 188920.0 33300.0 2.27 184160.0 29100.0 2.17 3.1365 0.9998 3553870 CHDI2_000956 CC(C)(C)OC(=O)NC/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L18 compound treatment 255960.0 100000.0 6.84 254440.0 99400.0 7.4 10.0671 0.9992 3554121 CHDI2_000957 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(Oc3ccccc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L19 compound treatment 288040.0 132000.0 9.02 284400.0 129000.0 9.63 13.1904 0.9995 3553873 CHDI2_000958 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L20 compound treatment 181840.0 26200.0 1.78 178560.0 23500.0 1.75 2.5005 1.0 3554125 CHDI2_000959 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc[n+]([O-])cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L21 compound treatment 176680.0 21000.0 1.43 178440.0 23400.0 1.74 2.2454 0.9953 3553877 CHDI2_000960 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(F)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L22 compound treatment 190160.0 34500.0 2.35 186840.0 31800.0 2.37 3.3374 1.0 3554129 CHDI2_000961 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L23 mock treatment 156880.0 1210.0 0.08 156600.0 1580.0 0.12 0.1415 0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 L24 mock treatment 156320.0 654.0 0.04 154400.0 -623.0 -0.05 -0.0012 -0.0194 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M01 compound treatment 174040.0 18400.0 1.25 178440.0 23400.0 1.74 2.1182 0.9869 3215312 CHDI2_000962 Cc1ccccc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M02 compound treatment 185800.0 30100.0 2.05 191480.0 36500.0 2.71 3.3714 0.9906 3553273 CHDI2_000963 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M03 compound treatment 221760.0 66100.0 4.51 230120.0 75100.0 5.59 7.1385 0.9943 3215316 CHDI2_000964 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M04 compound treatment 238640.0 83000.0 5.66 242080.0 87100.0 6.48 8.5817 0.9977 3553277 CHDI2_000965 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(F)c(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M05 compound treatment 187000.0 31300.0 2.14 192600.0 37600.0 2.8 3.4882 0.9912 3215320 CHDI2_000966 ONC(=O)CCCCC(=O)N/N=C/[C@H](O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M06 compound treatment 220400.0 64700.0 4.41 214120.0 59100.0 4.4 6.2309 1.0 3553281 CHDI2_000967 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(F)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M07 compound treatment 186160.0 30500.0 2.08 191400.0 36400.0 2.71 3.3845 0.9915 3215323 CHDI2_000968 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M08 compound treatment 193760.0 38100.0 2.6 200400.0 45400.0 3.38 4.2246 0.9916 3553285 CHDI2_000969 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M09 compound treatment 204920.0 49300.0 3.36 209160.0 54100.0 4.03 5.2236 0.9959 3553579 CHDI2_000970 ONC(=O)c1cccc(c1)C(=O)N/N=C/[C@H](O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M10 compound treatment 188960.0 33300.0 2.27 192400.0 37400.0 2.78 3.5721 0.9949 3553631 CHDI2_000971 CN(C)CCCOc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M11 compound treatment 187800.0 32100.0 2.19 186320.0 31300.0 2.33 3.1962 0.9995 3215326 CHDI2_000972 COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M12 compound treatment 202480.0 46800.0 3.19 199960.0 44900.0 3.34 4.6218 0.9997 3553289 CHDI2_000973 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M13 compound treatment 193200.0 37500.0 2.56 186680.0 31700.0 2.36 3.4755 0.9992 3553584 CHDI2_000974 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M14 compound treatment 202960.0 47300.0 3.22 200520.0 45500.0 3.39 4.6744 0.9997 3553635 CHDI2_000975 CCOc1cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M15 compound treatment 184720.0 29100.0 1.98 185920.0 30900.0 2.3 3.0267 0.9972 3215330 CHDI2_000976 CCOc1cccc(/C=N/NC(=O)CCCCC(=O)NO)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M16 compound treatment 186960.0 31300.0 2.13 187240.0 32200.0 2.4 3.2042 0.9983 3553293 CHDI2_000977 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(c2)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M17 compound treatment 224440.0 68800.0 4.69 227120.0 72100.0 5.37 7.1098 0.9977 3215334 CHDI2_000978 ONC(=O)CCCCC(=O)N/N=C/c1cc(I)cc(I)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M18 compound treatment 196480.0 40800.0 2.78 193560.0 38500.0 2.87 3.9957 0.9999 3553297 CHDI2_000979 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M19 compound treatment 180600.0 24900.0 1.7 183320.0 28300.0 2.11 2.6912 0.9944 3215338 CHDI2_000980 CN(C)c1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M20 compound treatment 194240.0 38600.0 2.63 192960.0 37900.0 2.82 3.8561 0.9994 3553301 CHDI2_000981 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccoc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M21 compound treatment 200080.0 44400.0 3.03 191320.0 36300.0 2.7 4.0514 0.9984 3215342 CHDI2_000982 CCn1c2ccccc2c3cc(/C=N/NC(=O)CCCCC(=O)NO)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M22 compound treatment 172560.0 16900.0 1.15 177280.0 22300.0 1.66 1.9858 0.9842 3553305 CHDI2_000983 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M23 mock treatment 159680.0 4010.0 0.27 161760.0 6740.0 0.5 0.5481 0.9594 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 M24 mock treatment 161120.0 5450.0 0.37 157080.0 2060.0 0.15 0.3712 0.9231 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N01 compound treatment 185120.0 29500.0 2.01 183440.0 28400.0 2.12 2.9155 0.9997 3553880 CHDI2_000984 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)c(F)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N02 compound treatment 182120.0 26500.0 1.8 191760.0 36700.0 2.73 3.2087 0.9796 3554133 CHDI2_000985 Cc1ccccc1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N03 compound treatment 234040.0 78400.0 5.34 248280.0 93300.0 6.94 8.6862 0.9916 3553882 CHDI2_000986 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(F)c(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N04 compound treatment 194200.0 38500.0 2.63 201240.0 46200.0 3.44 4.29 0.9911 3554137 CHDI2_000987 COc1cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N05 compound treatment 226440.0 70800.0 4.83 233160.0 78100.0 5.82 7.5241 0.9957 3553886 CHDI2_000988 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(F)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N06 compound treatment 192440.0 36800.0 2.51 189880.0 34900.0 2.59 3.6073 0.9999 3554141 CHDI2_000989 ONC(=O)c1ccc(cc1)C(=O)N/N=C/[C@H](O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N07 compound treatment 198320.0 42700.0 2.91 192880.0 37900.0 2.82 4.0486 0.9999 3553889 CHDI2_000990 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N08 compound treatment 188920.0 33300.0 2.27 185200.0 30200.0 2.25 3.1913 1.0 3554145 CHDI2_000991 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N09 compound treatment 181640.0 26000.0 1.77 178080.0 23100.0 1.72 2.4656 0.9999 3552757 CHDI2_000992 O=C(N/N=C/c1cccc2ccccc12)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N10 compound treatment 168240.0 12600.0 0.86 166280.0 11300.0 0.84 1.1986 0.9999 3552787 CHDI2_000993 O=C(N/N=C/c1nccs1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N11 compound treatment 205000.0 49300.0 3.36 205400.0 50400.0 3.75 5.0296 0.9985 3553894 CHDI2_000994 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N12 compound treatment 189040.0 33400.0 2.28 189160.0 34100.0 2.54 3.4055 0.9985 3554147 CHDI2_000995 COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N13 compound treatment 167000.0 11300.0 0.77 168640.0 13600.0 1.01 1.263 0.991 3552759 CHDI2_000996 O=C(N/N=C/c1ccc2ccccc2c1)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N14 compound treatment 147120.0 -8550.0 -0.58 152600.0 -2420.0 -0.18 -0.5395 -0.8845 3552789 CHDI2_000997 O=C(N/N=C/c1cccs1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N15 compound treatment 190240.0 34600.0 2.36 187760.0 32700.0 2.44 3.3896 0.9999 3553898 CHDI2_000998 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(c2)B(O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N16 compound treatment 195280.0 39600.0 2.7 190760.0 35700.0 2.66 3.7905 1.0 3554152 CHDI2_000999 CCOc1cccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N17 compound treatment 220440.0 64800.0 4.42 220720.0 65700.0 4.89 6.5801 0.9987 3553901 CHDI2_001000 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N18 compound treatment 269840.0 114000.0 7.78 273360.0 118000.0 8.81 11.732 0.9981 3554155 CHDI2_001001 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(I)cc(I)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N19 compound treatment 209720.0 54100.0 3.69 202720.0 47700.0 3.55 5.1161 0.9998 3553905 CHDI2_001002 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccoc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N20 compound treatment 185360.0 29700.0 2.02 182240.0 27200.0 2.03 2.8639 1.0 3554159 CHDI2_001003 CN(C)c1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N21 compound treatment 182360.0 26700.0 1.82 179160.0 24100.0 1.8 2.5572 1.0 3553909 CHDI2_001004 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N22 compound treatment 278640.0 123000.0 8.38 294920.0 140000.0 10.41 13.2909 0.9942 3554162 CHDI2_001005 CCn1c2ccccc2c3cc(/C=N/NC(=O)c4ccc(cc4)C(=O)NO)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N23 mock treatment 164360.0 8690.0 0.59 160880.0 5860.0 0.44 0.7274 0.9886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 N24 mock treatment 153520.0 -2150.0 -0.15 156800.0 1780.0 0.13 -0.0099 -0.0503 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O01 compound treatment 168280.0 12600.0 0.86 175000.0 20000.0 1.49 1.6595 0.9661 3215394 CHDI2_001006 ONC(=O)CCCCC(=O)N/N=C/c1ccc(o1)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O02 compound treatment 173480.0 17800.0 1.21 177480.0 22500.0 1.67 2.0407 0.9877 3553313 CHDI2_001007 OCCOc1ccccc1/C=N/NC(=O)c2cccc(c2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O03 compound treatment 175120.0 19500.0 1.33 172960.0 17900.0 1.34 1.8818 1.0 3215398 CHDI2_001008 Cn1cc(/C=N/NC(=O)CCCCC(=O)NO)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O04 compound treatment 169120.0 13500.0 0.92 171320.0 16300.0 1.21 1.5063 0.9905 3553317 CHDI2_001009 OCCOc1cccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O05 compound treatment 192880.0 37200.0 2.54 193160.0 38100.0 2.84 3.8011 0.9984 3215402 CHDI2_001010 ONC(=O)CCCCC(=O)N/N=C/c1cn(Cc2ccccc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O06 compound treatment 178960.0 23300.0 1.59 179840.0 24800.0 1.85 2.429 0.9972 3553320 CHDI2_001011 OCCOc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O07 compound treatment 183520.0 27900.0 1.9 185160.0 30100.0 2.24 2.9289 0.9966 3215406 CHDI2_001012 ONC(=O)CCCCC(=O)N/N=C/C1=CCCCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O08 compound treatment 227600.0 71900.0 4.9 220840.0 65800.0 4.9 6.9316 1.0 3553323 CHDI2_001013 COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O09 compound treatment 176640.0 21000.0 1.43 177040.0 22000.0 1.64 2.1698 0.9977 3215409 CHDI2_001014 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O10 compound treatment 206360.0 50700.0 3.46 206080.0 51100.0 3.8 5.1309 0.9989 3553327 CHDI2_001015 COc1ccc(O)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O11 compound treatment 185640.0 30000.0 2.04 192560.0 37500.0 2.79 3.4205 0.9882 3553585 CHDI2_001016 COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O12 compound treatment 190440.0 34800.0 2.37 186280.0 31300.0 2.33 3.3214 1.0 3553639 CHDI2_001017 CN(CCO)c1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O13 compound treatment 184600.0 28900.0 1.97 174480.0 19500.0 1.45 2.4189 0.9885 3215412 CHDI2_001018 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O14 compound treatment 209960.0 54300.0 3.7 212480.0 57500.0 4.28 5.6413 0.9974 3553331 CHDI2_001019 COc1cc(/C=C/C=N/NC(=O)c2cccc(c2)C(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O15 compound treatment 170560.0 14900.0 1.02 175520.0 20500.0 1.53 1.7967 0.9804 3215416 CHDI2_001020 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)CCCCC(=O)NO)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O16 compound treatment 212240.0 56600.0 3.86 218600.0 63600.0 4.73 6.0733 0.9949 3553334 CHDI2_001021 Cc1ccc(O)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O17 compound treatment 172800.0 17100.0 1.17 182000.0 27000.0 2.01 2.2458 0.9668 3215420 CHDI2_001022 C/C(=N\NC(=O)CCCCC(=O)NO)/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O18 compound treatment 183440.0 27800.0 1.89 185600.0 30600.0 2.28 2.9482 0.9958 3553338 CHDI2_001023 OCc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O19 compound treatment 177040.0 21400.0 1.46 173080.0 18100.0 1.34 1.9807 0.9992 3215424 CHDI2_001024 CN(C)CCCOc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O20 compound treatment 252480.0 96800.0 6.6 243960.0 88900.0 6.62 9.3478 1.0 3553342 CHDI2_001025 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc3ccccc3c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O21 compound treatment 199640.0 44000.0 3.0 198920.0 43900.0 3.27 4.4301 0.9991 3215428 CHDI2_001026 CCOc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O22 compound treatment 241840.0 86200.0 5.88 240680.0 85700.0 6.38 8.6623 0.9992 3553346 CHDI2_001027 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(o2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O23 mock treatment 157520.0 1850.0 0.13 155800.0 778.0 0.06 0.1303 0.9373 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 O24 mock treatment 151160.0 -4510.0 -0.31 151200.0 -3820.0 -0.28 -0.4184 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P01 compound treatment 174920.0 19300.0 1.31 176880.0 21900.0 1.63 2.0785 0.9943 3553917 CHDI2_001028 OCCOc1ccccc1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P02 compound treatment 201400.0 45700.0 3.12 192120.0 37100.0 2.76 4.1571 0.9982 3554170 CHDI2_001029 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(o2)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P03 compound treatment 172560.0 16900.0 1.15 176640.0 21600.0 1.61 1.9521 0.9866 3553921 CHDI2_001030 OCCOc1cccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P04 compound treatment 191360.0 35700.0 2.43 189920.0 34900.0 2.6 3.5573 0.9995 3554174 CHDI2_001031 Cn1cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P05 compound treatment 176040.0 20400.0 1.39 176760.0 21700.0 1.62 2.1262 0.9971 3553924 CHDI2_001032 OCCOc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P06 compound treatment 298080.0 142000.0 9.71 272480.0 117000.0 8.74 13.0471 0.9986 3554177 CHDI2_001033 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cn(Cc3ccccc3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P07 compound treatment 225480.0 69800.0 4.76 227920.0 72900.0 5.43 7.202 0.9979 3553927 CHDI2_001034 COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P08 compound treatment 184600.0 28900.0 1.97 184800.0 29800.0 2.22 2.962 0.9983 3554181 CHDI2_001035 ONC(=O)c1ccc(cc1)C(=O)N/N=C/C2=CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P09 compound treatment 242080.0 86400.0 5.89 232080.0 77100.0 5.74 8.2212 0.9999 3553931 CHDI2_001036 COc1ccc(O)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P10 compound treatment 174360.0 18700.0 1.27 181160.0 26100.0 1.95 2.2768 0.979 3554185 CHDI2_001037 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P11 compound treatment 181720.0 26100.0 1.78 182440.0 27400.0 2.04 2.6989 0.9976 3552761 CHDI2_001038 [O-][N+](=O)c1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P12 compound treatment 160320.0 4650.0 0.32 184880.0 29900.0 2.22 1.7957 0.8 3552791 CHDI2_001039 FC(F)(F)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P13 compound treatment 220040.0 64400.0 4.39 211520.0 56500.0 4.2 6.0767 0.9998 3553935 CHDI2_001040 COc1cc(/C=C/C=N/NC(=O)c2ccc(cc2)C(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P14 compound treatment 176760.0 21100.0 1.44 174560.0 19500.0 1.45 2.0451 1.0 3554187 CHDI2_001041 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P15 compound treatment 207880.0 52200.0 3.56 210920.0 55900.0 4.16 5.4589 0.997 3553938 CHDI2_001042 Cc1ccc(O)c(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P16 compound treatment 169240.0 13600.0 0.93 170960.0 15900.0 1.19 1.4931 0.9925 3554191 CHDI2_001043 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2ccc(cc2)C(=O)NO)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P17 compound treatment 191600.0 35900.0 2.45 195800.0 40800.0 3.03 3.8783 0.9944 3553942 CHDI2_001044 OCc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P18 compound treatment 182160.0 26500.0 1.81 184760.0 29700.0 2.21 2.8422 0.9949 3554251 CHDI2_001045 C/C(=N\NC(=O)c1ccc(cc1)C(=O)NO)/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P19 compound treatment 292280.0 137000.0 9.31 283560.0 129000.0 9.57 13.3506 0.9999 3553946 CHDI2_001046 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc3ccccc3c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P20 compound treatment 173120.0 17500.0 1.19 175480.0 20500.0 1.52 1.918 0.9926 3554194 CHDI2_001047 CN(C)CCCOc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P21 compound treatment 270320.0 115000.0 7.82 259520.0 104000.0 7.78 11.0267 1.0 3553950 CHDI2_001048 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(o2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P22 compound treatment 188800.0 33100.0 2.26 188520.0 33500.0 2.49 3.3602 0.9988 3554198 CHDI2_001049 CCOc1cc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P23 mock treatment 151840.0 -3830.0 -0.26 156360.0 1340.0 0.1 -0.1141 -0.4085 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2405 P24 mock treatment 155720.0 53.8 0.0 152520.0 -2500.0 -0.19 -0.1291 -0.6931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A01 compound treatment 175160.0 18400.0 1.26 176200.0 21100.0 1.57 1.9976 0.994 1006361 CHDI2_001050 NNC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A02 compound treatment 194040.0 37300.0 2.54 187880.0 32700.0 2.44 3.5225 0.9998 3552205 CHDI2_001051 Oc1ccc2ccccc2c1/C=N/NC(=O)c3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A03 compound treatment 176320.0 19600.0 1.34 175000.0 19900.0 1.48 1.9904 0.9987 3551925 CHDI2_001052 Oc1ccccc1C(=O)N/N=C/c2ccccc2OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A04 compound treatment 181760.0 25000.0 1.71 180440.0 25300.0 1.88 2.5389 0.9988 3552209 CHDI2_001053 Oc1ccccc1C(=O)N/N=C/c2ccc(O)c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A05 compound treatment 174680.0 18000.0 1.22 173800.0 18700.0 1.39 1.8482 0.998 1913714 CHDI2_001054 COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A06 compound treatment 172920.0 16200.0 1.1 170400.0 15300.0 1.14 1.5844 0.9999 3552211 CHDI2_001055 Oc1ccccc1C(=O)N/N=C/c2ccc([N+](=O)[O-])c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A07 compound treatment 172520.0 15800.0 1.08 171800.0 16700.0 1.24 1.6388 0.9975 3551931 CHDI2_001056 Oc1ccccc1C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A08 compound treatment 177840.0 21100.0 1.44 181640.0 26500.0 1.97 2.4131 0.988 3552215 CHDI2_001057 Oc1ccc([N+](=O)[O-])c(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A09 compound treatment 159000.0 2280.0 0.16 160560.0 5420.0 0.4 0.3955 0.914 3551934 CHDI2_001058 Oc1ccccc1C(=O)N/N=C/c2ccc3OCCOc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A10 compound treatment 178920.0 22200.0 1.51 179920.0 24800.0 1.84 2.3746 0.9952 3552219 CHDI2_001059 Oc1ccccc1C(=O)N/N=C/c2ccc(cc2)n3ccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A11 compound treatment 182800.0 26100.0 1.78 180840.0 25700.0 1.91 2.6101 0.9993 3551938 CHDI2_001060 Oc1ccccc1C(=O)N/N=C/COCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A12 compound treatment 174560.0 17800.0 1.22 176160.0 21000.0 1.56 1.9666 0.9922 3552223 CHDI2_001061 Oc1ccccc1C(=O)N/N=C/c2c[nH]c3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A13 compound treatment 414080.0 257000.0 17.55 419920.0 265000.0 19.71 26.342 0.9983 3552793 CHDI2_001062 Oc1ccc(/C=N/NC(=O)c2ccccn2)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A14 compound treatment 158440.0 1720.0 0.12 160760.0 5620.0 0.42 0.379 0.8717 3552989 CHDI2_001063 OB(O)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A15 compound treatment 175360.0 18600.0 1.27 174960.0 19800.0 1.48 1.942 0.9972 3551942 CHDI2_001064 Oc1ccccc1C(=O)N/N=C/c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A16 compound treatment 164960.0 8240.0 0.56 169640.0 14500.0 1.08 1.1606 0.9537 1922439 CHDI2_001065 Oc1ccccc1C(=O)N/N=C/c2ccc(I)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A17 compound treatment 164680.0 7960.0 0.54 168840.0 13700.0 1.02 1.105 0.9564 3551946 CHDI2_001066 Oc1ccccc1C(=O)N/N=C/c2ccccc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A18 compound treatment 172120.0 15400.0 1.05 174560.0 19400.0 1.45 1.7647 0.9877 3552228 CHDI2_001067 C/C=C(/C)\C=N\NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A19 compound treatment 173360.0 16600.0 1.13 173640.0 18500.0 1.38 1.7761 0.9954 3551950 CHDI2_001068 Oc1ccccc1C(=O)N/N=C/c2cccc(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A20 compound treatment 174400.0 17700.0 1.21 166880.0 11700.0 0.87 1.4705 0.9875 3552232 CHDI2_001069 Oc1ccccc1C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A21 compound treatment 169240.0 12500.0 0.85 165040.0 9900.0 0.74 1.1249 0.9973 3551953 CHDI2_001070 Oc1ccccc1C(=O)N/N=C/c2ccc(Br)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A22 compound treatment 169880.0 13200.0 0.9 169480.0 14300.0 1.07 1.3894 0.9963 1912639 CHDI2_001071 Cc1ccc(/C=N/NC(=O)c2ccccc2O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A23 mock treatment 153080.0 -3640.0 -0.25 152520.0 -2620.0 -0.19 -0.3131 -0.9928 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 A24 mock treatment 151560.0 -5160.0 -0.35 150480.0 -4660.0 -0.35 -0.4937 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B01 compound treatment 165160.0 8440.0 0.58 165880.0 10700.0 0.8 0.9724 0.987 1047348 CHDI2_001072 NNC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B02 compound treatment 159440.0 2720.0 0.19 168000.0 12900.0 0.96 0.8082 0.8287 3213096 CHDI2_001073 ONC(=O)CCCCCCC(=O)N/N=C/C(=C/c1ccccc1)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B03 compound treatment 164080.0 7360.0 0.5 165320.0 10200.0 0.76 0.8909 0.98 3552424 CHDI2_001074 C=CCOc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B04 compound treatment 158280.0 1560.0 0.11 159240.0 4100.0 0.31 0.2913 0.9004 3213142 CHDI2_001075 Cc1[nH]cnc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B05 compound treatment 115200.0 -41500.0 -2.83 113920.0 -41200.0 -3.07 -4.1706 -0.9992 3552426 CHDI2_001076 COc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B06 compound treatment 170600.0 13900.0 0.95 177120.0 22000.0 1.64 1.8262 0.9661 3213098 CHDI2_001077 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/C(=C/c2ccccc2)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B07 compound treatment 162000.0 5280.0 0.36 158880.0 3740.0 0.28 0.4517 0.992 3552428 CHDI2_001078 O=C(N/N=C/c1ccccc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B08 compound treatment 163200.0 6480.0 0.44 163560.0 8420.0 0.63 0.7558 0.9853 3213140 CHDI2_001079 Cc1[nH]cnc1/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B09 compound treatment 58400.0 -98300.0 -6.7 55440.0 -99700.0 -7.42 -9.9865 -0.9987 3552430 CHDI2_001080 O=C(N/N=C/c1ccc2OCCOc2c1)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B10 compound treatment 156360.0 -359.0 -0.02 172760.0 17600.0 1.31 0.9103 0.6938 3214252 CHDI2_001081 ONC(=O)CCCCCC(=O)N/N=C/C(=C/c1ccccc1)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B11 compound treatment 181200.0 24500.0 1.67 183720.0 28600.0 2.13 2.6845 0.9928 3552432 CHDI2_001082 O=C(N/N=C/COCc1ccccc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B12 compound treatment 184280.0 27600.0 1.88 186880.0 31700.0 2.36 2.9993 0.9936 3214254 CHDI2_001083 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/C(=C/c2ccccc2)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B13 compound treatment 167320.0 10600.0 0.72 167120.0 12000.0 0.89 1.1418 0.9946 3552919 CHDI2_001084 CCOc1cccc(/C=N/NC(=O)c2ccccn2)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B14 compound treatment 163160.0 6440.0 0.44 161760.0 6620.0 0.49 0.6592 0.9983 3214296 CHDI2_001085 Cc1[nH]cnc1/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B15 compound treatment 144720.0 -12000.0 -0.82 136840.0 -18300.0 -1.36 -1.5413 -0.9703 3552436 CHDI2_001086 O=C(N/N=C/c1ccc(cc1)c2ccccc2)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B16 compound treatment 159160.0 2440.0 0.17 163360.0 8220.0 0.61 0.5505 0.8679 3214862 CHDI2_001087 ONC(=O)CCCCC(=O)N/N=C/C(=C/c1ccccc1)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B17 compound treatment 156840.0 121.0 0.01 151400.0 -3740.0 -0.28 -0.1907 -0.6858 3552440 CHDI2_001088 Brc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B18 compound treatment 161480.0 4760.0 0.32 162080.0 6940.0 0.52 0.595 0.9749 3214908 CHDI2_001089 Cc1[nH]cnc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B19 compound treatment 171120.0 14400.0 0.98 168720.0 13600.0 1.01 1.4092 0.9999 3552445 CHDI2_001090 Brc1cccc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B20 compound treatment 209880.0 53200.0 3.62 195200.0 40100.0 2.98 4.6713 0.9953 3553033 CHDI2_001091 ONC(=O)c1cccc(c1)C(=O)N/N=C/C(=C/c2ccccc2)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B21 compound treatment 147200.0 -9520.0 -0.65 146440.0 -8700.0 -0.65 -0.9165 -1.0 3552449 CHDI2_001092 Brc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B22 compound treatment 178160.0 21400.0 1.46 179720.0 24600.0 1.83 2.3275 0.9938 3553699 CHDI2_001093 ONC(=O)c1ccc(cc1)C(=O)N/N=C/C(=C/c2ccccc2)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B23 mock treatment 149360.0 -7360.0 -0.5 150800.0 -4340.0 -0.32 -0.5829 -0.9772 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 B24 mock treatment 149720.0 -7000.0 -0.48 145480.0 -9660.0 -0.72 -0.8455 -0.9802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C01 compound treatment 172680.0 16000.0 1.09 179400.0 24300.0 1.81 2.0465 0.9706 3551960 CHDI2_001094 Oc1ccccc1C(=O)N/N=C/c2ccc(Br)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C02 compound treatment 158000.0 1280.0 0.09 164320.0 9180.0 0.68 0.5451 0.791 3552241 CHDI2_001095 Cc1ccsc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C03 compound treatment 169920.0 13200.0 0.9 176560.0 21400.0 1.59 1.7639 0.9634 3551964 CHDI2_001096 Oc1ccc(/C=N/NC(=O)c2ccccc2O)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C04 compound treatment 171680.0 15000.0 1.02 179400.0 24300.0 1.81 1.9983 0.9634 3552245 CHDI2_001097 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)c3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C05 compound treatment 174880.0 18200.0 1.24 174840.0 19700.0 1.47 1.9125 0.9965 3551968 CHDI2_001098 Oc1ccc(Br)c(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C06 compound treatment 176280.0 19600.0 1.33 172560.0 17400.0 1.3 1.86 0.9999 3552249 CHDI2_001099 Oc1ccccc1C(=O)N/N=C/c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C07 compound treatment 186800.0 30100.0 2.05 190960.0 35800.0 2.67 3.3355 0.9916 3551973 CHDI2_001100 COc1cc(Br)cc(/C=N/NC(=O)c2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C08 compound treatment 178200.0 21500.0 1.46 171640.0 16500.0 1.23 1.9042 0.9962 3552253 CHDI2_001101 Oc1ccccc1C(=O)N/N=C/c2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C09 compound treatment 177400.0 20700.0 1.41 178320.0 23200.0 1.73 2.2172 0.995 3551976 CHDI2_001102 COc1ccc(Br)c(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C10 compound treatment 161960.0 5240.0 0.36 161000.0 5860.0 0.44 0.5613 0.9951 1918554 CHDI2_001103 Oc1ccccc1C(=O)N/N=C/c2ccccc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C11 compound treatment 398080.0 241000.0 16.46 398040.0 243000.0 18.08 24.4192 0.9989 3552795 CHDI2_001104 Oc1cc(O)c(/C=N/NC(=O)c2ccccn2)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C12 compound treatment 113480.0 -43200.0 -2.95 107680.0 -47500.0 -3.53 -4.5819 -0.996 3552993 CHDI2_001105 O=C(N/N=C/c1ccc(OCC#C)cc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C13 compound treatment 170920.0 14200.0 0.97 174840.0 19700.0 1.47 1.7216 0.9797 3551980 CHDI2_001106 COc1ccc(Br)cc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C14 compound treatment 174680.0 18000.0 1.22 171360.0 16200.0 1.21 1.7197 1.0 1919338 CHDI2_001107 COc1cc(/C=N/NC(=O)c2ccccc2O)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C15 compound treatment 172280.0 15600.0 1.06 164000.0 8860.0 0.66 1.2167 0.9739 3552797 CHDI2_001108 COc1cc(OC)c(/C=N/NC(=O)c2ccccn2)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C16 compound treatment 169680.0 13000.0 0.88 169240.0 14100.0 1.05 1.3671 0.9963 3552870 CHDI2_001109 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C17 compound treatment 172760.0 16000.0 1.09 166840.0 11700.0 0.87 1.3893 0.9936 1922614 CHDI2_001110 Oc1ccccc1C(=O)N/N=C/c2cc3OCOc3cc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C18 compound treatment 173080.0 16400.0 1.12 171680.0 16500.0 1.23 1.6595 0.9988 3552261 CHDI2_001111 Oc1ccccc1C(=O)N/N=C/c2c(F)c(F)c(F)c(F)c2F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C19 compound treatment 162120.0 5400.0 0.37 164080.0 8940.0 0.67 0.7311 0.961 3551985 CHDI2_001112 Oc1ccccc1C(=O)N/N=C/c2cccnc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C20 compound treatment 171080.0 14400.0 0.98 166080.0 10900.0 0.81 1.2683 0.9958 3552264 CHDI2_001113 Oc1ccccc1C(=O)N/N=C/CCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C21 compound treatment 169760.0 13000.0 0.89 171200.0 16100.0 1.2 1.4741 0.9894 3551989 CHDI2_001114 Oc1ccccc1C(=O)N/N=C/c2ccncc2Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C22 compound treatment 167720.0 11000.0 0.75 167840.0 12700.0 0.95 1.199 0.9934 3552269 CHDI2_001115 CC(=C)[C@H]1CCC(=CC1)/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C23 mock treatment 152840.0 -3880.0 -0.26 148520.0 -6620.0 -0.49 -0.5351 -0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 C24 mock treatment 150600.0 -6120.0 -0.42 143000.0 -12100.0 -0.9 -0.9336 -0.9384 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D01 compound treatment 161440.0 4720.0 0.32 163440.0 8300.0 0.62 0.6647 0.9538 3552455 CHDI2_001116 Brc1ccc(/C=N/NC(=O)c2ccccn2)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D02 compound treatment 178040.0 21300.0 1.45 182320.0 27200.0 2.02 2.4585 0.9868 3213180 CHDI2_001117 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(Br)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D03 compound treatment 157560.0 841.0 0.06 157600.0 2460.0 0.18 0.1703 0.8859 3552459 CHDI2_001118 Oc1ccc(/C=N/NC(=O)c2ccccn2)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D04 compound treatment 172440.0 15700.0 1.07 175160.0 20000.0 1.49 1.8117 0.9869 3213222 CHDI2_001119 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(Oc2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D05 compound treatment 157040.0 321.0 0.02 157400.0 2260.0 0.17 0.1347 0.7923 3552463 CHDI2_001120 Oc1ccc(Br)c(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D06 compound treatment 195080.0 38400.0 2.62 193760.0 38600.0 2.87 3.8821 0.9989 3213182 CHDI2_001121 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(Br)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D07 compound treatment 234040.0 77300.0 5.27 233720.0 78600.0 5.85 7.8633 0.9987 3552467 CHDI2_001122 COc1cc(Br)cc(/C=N/NC(=O)c2ccccn2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D08 compound treatment 165480.0 8760.0 0.6 164840.0 9700.0 0.72 0.9331 0.9955 3213220 CHDI2_001123 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D09 compound treatment 148880.0 -7840.0 -0.53 147480.0 -7660.0 -0.57 -0.7808 -0.9995 3552471 CHDI2_001124 COc1ccc(Br)c(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D10 compound treatment 184360.0 27600.0 1.88 188040.0 32900.0 2.45 3.0642 0.9916 3214336 CHDI2_001125 ONC(=O)CCCCCC(=O)N/N=C/c1cc(Br)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D11 compound treatment 185120.0 28400.0 1.94 187440.0 32300.0 2.4 3.0693 0.9942 3552923 CHDI2_001126 Oc1c(I)cc(I)cc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D12 compound treatment 198040.0 41300.0 2.82 191800.0 36700.0 2.73 3.9216 0.9999 3214338 CHDI2_001127 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(Br)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D13 compound treatment 171360.0 14600.0 1.0 170720.0 15600.0 1.16 1.526 0.9972 3552475 CHDI2_001128 COc1ccc(Br)cc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D14 compound treatment 189040.0 32300.0 2.2 185840.0 30700.0 2.29 3.1741 0.9998 3214376 CHDI2_001129 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D15 compound treatment 101760.0 -55000.0 -3.75 105520.0 -49600.0 -3.69 -5.2606 -1.0 3552927 CHDI2_001130 CN(C)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D16 compound treatment 185200.0 28500.0 1.94 183720.0 28600.0 2.13 2.8774 0.999 3214946 CHDI2_001131 ONC(=O)CCCCC(=O)N/N=C/c1cc(Br)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D17 compound treatment 167880.0 11200.0 0.76 163680.0 8540.0 0.64 0.9878 0.996 3552479 CHDI2_001132 Brc1cc2OCOc2cc1/C=N/NC(=O)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D18 compound treatment 165040.0 8320.0 0.57 166680.0 11500.0 0.86 1.0087 0.9797 3214988 CHDI2_001133 ONC(=O)CCCCC(=O)N/N=C/c1cccc(Oc2ccccc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D19 compound treatment 145920.0 -10800.0 -0.74 147200.0 -7940.0 -0.59 -0.9382 -0.994 3552483 CHDI2_001134 Brc1ncccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D20 compound treatment 241880.0 85200.0 5.81 234440.0 79300.0 5.9 8.2791 1.0 3553073 CHDI2_001135 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(Br)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D21 compound treatment 146680.0 -10000.0 -0.68 138480.0 -16700.0 -1.24 -1.3605 -0.9608 3552486 CHDI2_001136 Brc1cnccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D22 compound treatment 181280.0 24600.0 1.67 183520.0 28400.0 2.11 2.6779 0.9934 3553737 CHDI2_001137 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(Br)ccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D23 mock treatment 149520.0 -7200.0 -0.49 147360.0 -7780.0 -0.58 -0.7562 -0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 D24 mock treatment 151240.0 -5480.0 -0.37 144440.0 -10700.0 -0.8 -0.827 -0.9405 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E01 compound treatment 171480.0 14800.0 1.01 166760.0 11600.0 0.87 1.3234 0.9972 3552839 CHDI2_001138 COc1cc(/C=N/NC(=O)c2ccccn2)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E02 compound treatment 159240.0 2520.0 0.17 159680.0 4540.0 0.34 0.3607 0.9507 3552874 CHDI2_001139 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E03 compound treatment 191720.0 35000.0 2.39 188760.0 33600.0 2.5 3.4569 0.9997 3551996 CHDI2_001140 Oc1ccccc1C(=O)N/N=C/c2ccc(Br)s2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E04 compound treatment 187400.0 30700.0 2.09 192600.0 37500.0 2.79 3.4508 0.99 3552276 CHDI2_001141 Oc1ccccc1C(=O)N/N=C/c2cn(c3ccccc23)S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E05 compound treatment 181120.0 24400.0 1.66 189600.0 34500.0 2.57 2.9901 0.978 3552001 CHDI2_001142 COc1cc(/C=N/NC(=O)c2ccccc2O)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E06 compound treatment 179800.0 23100.0 1.57 180360.0 25200.0 1.88 2.4402 0.9961 3552280 CHDI2_001143 Oc1ccccc1C(=O)N/N=C/c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E07 compound treatment 201800.0 45100.0 3.07 209400.0 54300.0 4.04 5.0291 0.9909 3552005 CHDI2_001144 Oc1ccccc1C(=O)N/N=C/c2ccc(OCc3ccccc3)cc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E08 compound treatment 174800.0 18100.0 1.23 173680.0 18500.0 1.38 1.8476 0.9984 1912699 CHDI2_001145 Oc1ccccc1C(=O)N/N=C/c2cccnc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E09 compound treatment 181000.0 24300.0 1.66 182920.0 27800.0 2.07 2.6328 0.9939 3552842 CHDI2_001146 CC(C)(C)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E10 compound treatment 176960.0 20200.0 1.38 179560.0 24400.0 1.82 2.2612 0.9908 3552878 CHDI2_001147 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E11 compound treatment 179240.0 22500.0 1.54 180720.0 25600.0 1.9 2.4322 0.9943 3552009 CHDI2_001148 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E12 compound treatment 188760.0 32000.0 2.18 186360.0 31200.0 2.32 3.1879 0.9995 3552285 CHDI2_001149 Cc1ncc(CO)c(/C=N/NC(=O)c2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E13 compound treatment 182840.0 26100.0 1.78 183960.0 28800.0 2.15 2.7762 0.9957 3552013 CHDI2_001150 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E14 compound treatment 181640.0 24900.0 1.7 180880.0 25700.0 1.92 2.5563 0.9982 1917465 CHDI2_001151 Oc1ccccc1C(=O)N/N=C/c2ccc[nH]2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E15 compound treatment 213240.0 56500.0 3.85 212920.0 57800.0 4.3 5.7659 0.9985 3552017 CHDI2_001152 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E16 compound treatment 181520.0 24800.0 1.69 179280.0 24100.0 1.8 2.4663 0.9995 3552291 CHDI2_001153 Oc1ccccc1C(=O)N/N=C/c2ccc(cc2)N3CCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E17 compound treatment 181480.0 24800.0 1.69 180760.0 25600.0 1.91 2.5423 0.9981 3552846 CHDI2_001154 CC1=C(C/C=N/NC(=O)c2ccccn2)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E18 compound treatment 174880.0 18200.0 1.24 177640.0 22500.0 1.67 2.0599 0.9889 3552881 CHDI2_001155 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E19 compound treatment 166960.0 10200.0 0.7 164080.0 8940.0 0.67 0.9644 0.9997 3552021 CHDI2_001156 OC(=O)c1cccc(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E20 compound treatment 196640.0 39900.0 2.72 192280.0 37100.0 2.76 3.8794 1.0 2119509 CHDI2_001157 Oc1ccccc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E21 compound treatment 167080.0 10400.0 0.71 164520.0 9380.0 0.7 0.9934 1.0 3552026 CHDI2_001158 OC(=O)c1ccccc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E22 compound treatment 180120.0 23400.0 1.6 176560.0 21400.0 1.59 2.2557 1.0 3552296 CHDI2_001159 CCCCCCC/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E23 mock treatment 158320.0 1600.0 0.11 158520.0 3380.0 0.25 0.2553 0.93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 E24 mock treatment 157280.0 561.0 0.04 153200.0 -1940.0 -0.14 -0.0748 -0.5019 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F01 compound treatment 187080.0 30400.0 2.07 182120.0 27000.0 2.01 2.8838 0.9999 3552931 CHDI2_001160 CCn1c2ccccc2c3cc(/C=N/NC(=O)c4ccccn4)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F02 compound treatment 166320.0 9600.0 0.65 166680.0 11500.0 0.86 1.0704 0.991 3213256 CHDI2_001161 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F03 compound treatment 169560.0 12800.0 0.88 169640.0 14500.0 1.08 1.3824 0.9946 3552494 CHDI2_001162 Brc1ccc(/C=N/NC(=O)c2ccccn2)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F04 compound treatment 172000.0 15300.0 1.04 175120.0 20000.0 1.49 1.7884 0.9848 3213294 CHDI2_001163 ONC(=O)CCCCCCC(=O)N/N=C/c1nccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F05 compound treatment 184440.0 27700.0 1.89 185560.0 30400.0 2.26 2.9376 0.996 3552498 CHDI2_001164 COc1cc(/C=N/NC(=O)c2ccccn2)c(Br)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F06 compound treatment 176360.0 19600.0 1.34 178520.0 23400.0 1.74 2.1776 0.9916 3213258 CHDI2_001165 OC(=O)c1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F07 compound treatment 211760.0 55000.0 3.75 218560.0 63400.0 4.72 5.9913 0.9935 3552502 CHDI2_001166 Oc1cc(OCc2ccccc2)ccc1/C=N/NC(=O)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F08 compound treatment 192520.0 35800.0 2.44 187920.0 32800.0 2.44 3.4513 1.0 3213292 CHDI2_001167 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2nccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F09 compound treatment 171320.0 14600.0 1.0 176720.0 21600.0 1.61 1.8399 0.9735 3552936 CHDI2_001168 Fc1cc(/C=N/NC(=O)c2ccccn2)ccc1c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F10 compound treatment 181800.0 25100.0 1.71 179600.0 24500.0 1.82 2.4966 0.9995 3214412 CHDI2_001169 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F11 compound treatment 173680.0 17000.0 1.16 178600.0 23500.0 1.75 2.0526 0.98 3552506 CHDI2_001170 CC(C)(C)OC(=O)NC1(CCCC1)/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F12 compound treatment 177680.0 21000.0 1.43 174040.0 18900.0 1.41 2.0054 1.0 3214414 CHDI2_001171 OC(=O)c1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F13 compound treatment 179160.0 22400.0 1.53 180880.0 25700.0 1.92 2.4367 0.9938 3552509 CHDI2_001172 CC(C)(C)OC(=O)N1CCC[C@H]1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F14 compound treatment 182920.0 26200.0 1.79 187160.0 32000.0 2.38 2.9485 0.9899 3214448 CHDI2_001173 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2nccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F15 compound treatment 185640.0 28900.0 1.97 187440.0 32300.0 2.4 3.0944 0.9951 3552513 CHDI2_001174 CC(C)(C)OC(=O)Nc1cccc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F16 compound treatment 171240.0 14500.0 0.99 168240.0 13100.0 0.98 1.3897 1.0 3215022 CHDI2_001175 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F17 compound treatment 168680.0 12000.0 0.82 168560.0 13400.0 1.0 1.2831 0.9949 3552940 CHDI2_001176 OS(=O)(=O)c1ccc(/C=N/NC(=O)c2ccccn2)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F18 compound treatment 180040.0 23300.0 1.59 175800.0 20700.0 1.54 2.2118 0.9999 3215060 CHDI2_001177 ONC(=O)CCCCC(=O)N/N=C/c1nccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F19 compound treatment 167000.0 10300.0 0.7 168120.0 13000.0 0.97 1.179 0.9876 3552517 CHDI2_001178 OC(=O)c1cccc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F20 compound treatment 173880.0 17200.0 1.17 173880.0 18700.0 1.4 1.8138 0.9962 3553108 CHDI2_001179 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F21 compound treatment 137880.0 -18800.0 -1.28 124720.0 -30400.0 -2.26 -2.5089 -0.964 3552521 CHDI2_001180 OC(=O)c1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F22 compound treatment 168880.0 12200.0 0.83 169200.0 14100.0 1.05 1.3265 0.9933 3553771 CHDI2_001181 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F23 mock treatment 160880.0 4160.0 0.28 155400.0 265.0 0.02 0.2145 0.7544 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 F24 mock treatment 154520.0 -2200.0 -0.15 150480.0 -4660.0 -0.35 -0.351 -0.9298 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G01 compound treatment 186080.0 29400.0 2.0 186880.0 31700.0 2.36 3.0861 0.9966 3552033 CHDI2_001182 Oc1ccccc1C(=O)N/N=C/c2ccccc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G02 compound treatment 177560.0 20800.0 1.42 180920.0 25800.0 1.92 2.3617 0.9891 1918398 CHDI2_001183 Oc1ccccc1C(=O)N/N=C/c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G03 compound treatment 181360.0 24600.0 1.68 186320.0 31200.0 2.32 2.8291 0.9874 3552850 CHDI2_001184 NC(=O)COc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G04 compound treatment 184200.0 27500.0 1.87 181320.0 26200.0 1.95 2.7029 0.9998 3552884 CHDI2_001185 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G05 compound treatment 183680.0 27000.0 1.84 177400.0 22300.0 1.66 2.4715 0.9987 3552037 CHDI2_001186 Oc1ccccc1C(=O)N/N=C/c2cccnc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G06 compound treatment 189360.0 32600.0 2.23 190840.0 35700.0 2.66 3.4526 0.9961 3552305 CHDI2_001187 Oc1ccccc1C(=O)N/N=C/c2ccc(cc2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G07 compound treatment 217920.0 61200.0 4.17 210480.0 55300.0 4.12 5.8631 1.0 3552041 CHDI2_001188 Oc1ccccc1C(=O)N/N=C/C=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G08 compound treatment 408280.0 252000.0 17.15 405240.0 250000.0 18.61 25.2898 0.9992 3552309 CHDI2_001189 Oc1ccc(/C=N/NC(=O)c2ccccc2O)c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G09 compound treatment 199480.0 42800.0 2.92 204480.0 49300.0 3.67 4.6583 0.9935 3552044 CHDI2_001190 C[C@H](CCC=C(C)C)C/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G10 compound treatment 239120.0 82400.0 5.62 245640.0 90500.0 6.74 8.7355 0.9959 3552313 CHDI2_001191 Oc1cc(O)c(/C=N/NC(=O)c2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G11 compound treatment 207800.0 51100.0 3.48 204040.0 48900.0 3.64 5.0363 0.9998 3552048 CHDI2_001192 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G12 compound treatment 191880.0 35200.0 2.4 184480.0 29300.0 2.18 3.2394 0.9989 3552317 CHDI2_001193 COc1cc(OC)c(/C=N/NC(=O)c2ccccc2O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G13 compound treatment 181680.0 25000.0 1.7 177400.0 22300.0 1.66 2.3751 0.9999 3552051 CHDI2_001194 Oc1ccccc1C(=O)N/N=C/c2ccc(C#N)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G14 compound treatment 182920.0 26200.0 1.79 187800.0 32700.0 2.43 2.9822 0.9885 3552321 CHDI2_001195 COc1cc(/C=N/NC(=O)c2ccccc2O)cc(OC)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G15 compound treatment 190840.0 34100.0 2.33 193480.0 38300.0 2.85 3.6629 0.9949 3552054 CHDI2_001196 Oc1ccccc1C(=O)N/N=C/C2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G16 compound treatment 185000.0 28300.0 1.93 186080.0 30900.0 2.3 2.9919 0.9961 3552325 CHDI2_001197 CC(C)(C)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G17 compound treatment 182480.0 25800.0 1.76 184400.0 29300.0 2.18 2.782 0.9943 3552058 CHDI2_001198 COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G18 compound treatment 195680.0 39000.0 2.66 198440.0 43300.0 3.22 4.1573 0.9954 3552329 CHDI2_001199 CC1=C(C/C=N/NC(=O)c2ccccc2O)C(C)(C)CCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G19 compound treatment 174440.0 17700.0 1.21 166520.0 11400.0 0.85 1.4535 0.9849 3552855 CHDI2_001200 NC(=O)COc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G20 compound treatment 179920.0 23200.0 1.58 172720.0 17600.0 1.31 2.0439 0.9956 3552885 CHDI2_001201 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G21 compound treatment 191600.0 34900.0 2.38 186800.0 31700.0 2.36 3.348 1.0 3552062 CHDI2_001202 Oc1ccccc1C(=O)N/N=C/c2cc(Br)cc(Br)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G22 compound treatment 179960.0 23200.0 1.58 179480.0 24300.0 1.81 2.4016 0.9978 3552333 CHDI2_001203 NC(=O)COc1ccccc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G23 mock treatment 167320.0 10600.0 0.72 161480.0 6340.0 0.47 0.845 0.9787 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 G24 mock treatment 160400.0 3680.0 0.25 151040.0 -4100.0 -0.3 -0.0381 -0.0964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H01 compound treatment 172080.0 15400.0 1.05 177880.0 22700.0 1.69 1.9375 0.9734 1936274 CHDI2_001204 Clc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H02 compound treatment 250880.0 94200.0 6.42 252200.0 97100.0 7.22 9.6477 0.9983 3213330 CHDI2_001205 CCCCN(CCCC)c1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H03 compound treatment 177840.0 21100.0 1.44 178480.0 23300.0 1.74 2.2468 0.9956 3552944 CHDI2_001206 Cn1cc(/C=N/NC(=O)c2ccccn2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H04 compound treatment 175200.0 18500.0 1.26 175000.0 19900.0 1.48 1.9364 0.9968 3213372 CHDI2_001207 NC(=O)COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H05 compound treatment 164280.0 7560.0 0.52 164040.0 8900.0 0.66 0.8331 0.9923 3552530 CHDI2_001208 Clc1ncccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H06 compound treatment 180840.0 24100.0 1.64 177600.0 22500.0 1.67 2.3451 1.0 3213332 CHDI2_001209 CCCCN(CCCC)c1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H07 compound treatment 194840.0 38100.0 2.6 191480.0 36300.0 2.71 3.7505 0.9998 3552534 CHDI2_001210 O=C(N/N=C/C=C/c1ccccc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H08 compound treatment 216560.0 59800.0 4.08 197720.0 42600.0 3.17 5.126 0.9922 3213370 CHDI2_001211 NC(=O)COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H09 compound treatment 190680.0 34000.0 2.32 190680.0 35500.0 2.65 3.5079 0.9978 3552538 CHDI2_001212 C[C@H](CCC=C(C)C)C/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H10 compound treatment 225240.0 68500.0 4.67 225960.0 70800.0 5.27 7.0306 0.9982 3214486 CHDI2_001213 CCCCN(CCCC)c1ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H11 compound treatment 187480.0 30800.0 2.1 183600.0 28500.0 2.12 2.981 1.0 3552543 CHDI2_001214 C[C@@H](CCC=C(C)C)C/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H12 compound treatment 212320.0 55600.0 3.79 213600.0 58500.0 4.35 5.7573 0.9976 3214488 CHDI2_001215 CCCCN(CCCC)c1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H13 compound treatment 166000.0 9280.0 0.63 165520.0 10400.0 0.77 0.994 0.9951 3552545 CHDI2_001216 O=C(N/N=C/c1ccc(C#N)cc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H14 compound treatment 176640.0 19900.0 1.36 182360.0 27200.0 2.03 2.3931 0.9811 3214526 CHDI2_001217 NC(=O)COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H15 compound treatment 184760.0 28000.0 1.91 188680.0 33500.0 2.5 3.1172 0.9913 3552548 CHDI2_001218 O=C(N/N=C/C1CCCCC1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H16 compound treatment 198840.0 42100.0 2.87 195640.0 40500.0 3.01 4.1623 0.9997 3215096 CHDI2_001219 CCCCN(CCCC)c1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H17 compound treatment 181440.0 24700.0 1.69 177960.0 22800.0 1.7 2.393 1.0 3552552 CHDI2_001220 COc1ccc(/C=N/NC(=O)c2ccccn2)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H18 compound treatment 178600.0 21900.0 1.49 181280.0 26100.0 1.95 2.4308 0.9914 3215138 CHDI2_001221 NC(=O)COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H19 compound treatment 186240.0 29500.0 2.01 191160.0 36000.0 2.68 3.3191 0.99 3552948 CHDI2_001222 O=C(N/N=C/c1cn(Cc2ccccc2)c3ccccc13)c4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H20 compound treatment 278240.0 122000.0 8.28 276240.0 121000.0 9.01 12.2318 0.9991 3553145 CHDI2_001223 CCCCN(CCCC)c1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H21 compound treatment 183360.0 26600.0 1.82 187000.0 31900.0 2.37 2.9613 0.9913 3552556 CHDI2_001224 Oc1c(Br)cc(Br)cc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H22 compound treatment 291840.0 135000.0 9.21 285880.0 131000.0 9.73 13.3948 0.9996 3553805 CHDI2_001225 CCCCN(CCCC)c1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H23 mock treatment 160840.0 4120.0 0.28 162400.0 7260.0 0.54 0.581 0.9535 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 H24 mock treatment 155360.0 -1360.0 -0.09 159160.0 4020.0 0.3 0.1463 0.4666 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I01 compound treatment 193120.0 36400.0 2.48 197800.0 42700.0 3.18 4.0002 0.9926 3552070 CHDI2_001226 COc1cc(Cl)c(/C=N/NC(=O)c2ccccc2O)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I02 compound treatment 181560.0 24800.0 1.69 178360.0 23200.0 1.73 2.4198 0.9999 1918345 CHDI2_001227 Oc1ccccc1C(=O)NN=C2CCCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I03 compound treatment 200880.0 44200.0 3.01 209200.0 54100.0 4.02 4.9742 0.9898 2082285 CHDI2_001228 Oc1ccccc1C(=O)N/N=C/c2cc(Cl)cc(Cl)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I04 compound treatment 187680.0 31000.0 2.11 183160.0 28000.0 2.09 2.9675 1.0 3554225 CHDI2_001229 Oc1ccccc1C(=O)NN=C2CCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I05 compound treatment 184280.0 27600.0 1.88 185040.0 29900.0 2.23 2.9025 0.9965 3554230 CHDI2_001230 O=C(NN=C1CCCCCCC1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I06 compound treatment 159880.0 3160.0 0.22 159760.0 4620.0 0.34 0.3958 0.9746 3552890 CHDI2_001231 O=C(N/N=C/c1ccc(Oc2ccccc2)cc1)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I07 compound treatment 208480.0 51800.0 3.53 206440.0 51300.0 3.82 5.1954 0.9992 3552075 CHDI2_001232 Oc1ccccc1C(=O)N/N=C/c2cc(Br)cc([N+](=O)[O-])c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I08 compound treatment 191840.0 35100.0 2.39 188520.0 33400.0 2.48 3.4501 0.9998 3552414 CHDI2_001233 Oc1ccccc1C(=O)N/N=C/Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I09 compound treatment 224440.0 67700.0 4.62 222200.0 67100.0 4.99 6.7942 0.9992 3552079 CHDI2_001234 CCN(CC)c1ccc(/C=N/NC(=O)c2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I10 compound treatment 194600.0 37900.0 2.58 188440.0 33300.0 2.48 3.5789 0.9998 3552416 CHDI2_001235 COC(=O)c1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I11 compound treatment 180400.0 23700.0 1.61 182080.0 26900.0 2.01 2.5597 0.9942 3552083 CHDI2_001236 Oc1ccccc1C(=O)N/N=C/c2ccc3OCCc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I12 compound treatment 192960.0 36200.0 2.47 192480.0 37300.0 2.78 3.7125 0.9983 3552341 CHDI2_001237 COc1cc(Br)c(/C=N/NC(=O)c2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I13 compound treatment 311320.0 155000.0 10.54 309840.0 155000.0 11.51 15.5948 0.999 3552087 CHDI2_001238 Oc1cccc(/C=N/NC(=O)c2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I14 compound treatment 200360.0 43600.0 2.98 189960.0 34800.0 2.59 3.9366 0.9976 3552418 CHDI2_001239 Oc1ccccc1C(=O)N/N=C/c2cc3ccccc3n2S(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I15 compound treatment 287080.0 130000.0 8.89 286160.0 131000.0 9.75 13.18 0.9989 3552091 CHDI2_001240 Oc1ccc(/C=N/NC(=O)c2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I16 compound treatment 189080.0 32400.0 2.21 188440.0 33300.0 2.48 3.3128 0.9983 3552345 CHDI2_001241 Oc1ccccc1C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I17 compound treatment 318640.0 162000.0 11.04 323760.0 169000.0 12.55 16.6803 0.998 3552095 CHDI2_001242 Oc1ccc(O)c(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I18 compound treatment 208720.0 52000.0 3.55 204040.0 48900.0 3.64 5.0806 0.9999 3552349 CHDI2_001243 Oc1ccccc1C(=O)N/N=C/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I19 compound treatment 209360.0 52600.0 3.59 207640.0 52500.0 3.91 5.3009 0.9991 3552098 CHDI2_001244 Oc1ccc(/C=N/NC(=O)c2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I20 compound treatment 187560.0 30800.0 2.1 184000.0 28900.0 2.15 3.0059 0.9999 3552420 CHDI2_001245 OB(O)c1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I21 compound treatment 174800.0 18100.0 1.23 174200.0 19100.0 1.42 1.875 0.9975 3554228 CHDI2_001246 O=C(NN=C1CCCCCC1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I22 compound treatment 167200.0 10500.0 0.71 165680.0 10500.0 0.78 1.0602 0.9989 3552894 CHDI2_001247 [O-][n+]1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I23 mock treatment 159320.0 2600.0 0.18 158960.0 3820.0 0.28 0.3267 0.9741 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 I24 mock treatment 154080.0 -2640.0 -0.18 155520.0 385.0 0.03 -0.107 -0.5872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J01 compound treatment 168400.0 11700.0 0.8 169480.0 14300.0 1.07 1.3181 0.9896 3552565 CHDI2_001248 COc1cc(Cl)c(/C=N/NC(=O)c2ccccn2)c(Cl)c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J02 compound treatment 179600.0 22900.0 1.56 171160.0 16000.0 1.19 1.9464 0.9912 3213410 CHDI2_001249 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J03 compound treatment 212920.0 56200.0 3.83 220200.0 65100.0 4.84 6.1336 0.9933 3552569 CHDI2_001250 Oc1c(Cl)cc(Cl)cc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J04 mock treatment 172640.0 15900.0 1.09 166240.0 11100.0 0.83 1.3519 0.991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J05 compound treatment 175320.0 18600.0 1.27 173160.0 18000.0 1.34 1.8453 0.9996 3552951 CHDI2_001251 O=C(N/N=C/C1=CCCCC1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J06 compound treatment 182520.0 25800.0 1.76 187680.0 32500.0 2.42 2.9566 0.9877 3213412 CHDI2_001252 COc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J07 compound treatment 217400.0 60700.0 4.14 215040.0 59900.0 4.46 6.078 0.9993 3552573 CHDI2_001253 Oc1c(/C=N/NC(=O)c2ccccn2)cc(Br)cc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J08 mock treatment 176440.0 19700.0 1.34 169360.0 14200.0 1.06 1.6993 0.993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J09 compound treatment 332880.0 176000.0 12.01 332680.0 178000.0 13.21 17.8362 0.9989 3552578 CHDI2_001254 CCN(CC)c1ccc(/C=N/NC(=O)c2ccccn2)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J10 compound treatment 188240.0 31500.0 2.15 187120.0 32000.0 2.38 3.2029 0.9987 3214566 CHDI2_001255 COc1ccc(/C=N/NC(=O)CCCCCC(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J11 compound treatment 180960.0 24200.0 1.65 170960.0 15800.0 1.18 2.0014 0.9862 3552582 CHDI2_001256 O=C(N/N=C/c1ccc2OCCc2c1)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J12 compound treatment 187320.0 30600.0 2.09 188160.0 33000.0 2.46 3.2132 0.9967 3214568 CHDI2_001257 COc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J13 compound treatment 167160.0 10400.0 0.71 169080.0 13900.0 1.04 1.2372 0.9831 3552586 CHDI2_001258 Oc1cccc(/C=N/NC(=O)c2ccccn2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J14 compound treatment 185800.0 29100.0 1.98 185600.0 30500.0 2.27 3.0052 0.9978 3214215 CHDI2_001259 NNC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J15 compound treatment 248440.0 91700.0 6.25 235880.0 80700.0 6.01 8.6711 0.9998 3552590 CHDI2_001260 Oc1ccc(/C=N/NC(=O)c2ccccn2)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J16 compound treatment 178600.0 21900.0 1.49 182160.0 27000.0 2.01 2.4771 0.9892 3215176 CHDI2_001261 COc1ccc(/C=N/NC(=O)CCCCC(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J17 compound treatment 209800.0 53100.0 3.62 271360.0 116000.0 8.65 8.6756 0.9252 3552594 CHDI2_001262 Oc1ccc(O)c(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J18 compound treatment 179120.0 22400.0 1.53 181960.0 26800.0 2.0 2.4916 0.9912 3214824 CHDI2_001263 NNC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J19 compound treatment 179720.0 23000.0 1.57 178920.0 23800.0 1.77 2.3606 0.9982 1936679 CHDI2_001264 Oc1ccc(/C=N/NC(=O)c2ccccn2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J20 compound treatment 180480.0 23800.0 1.62 178680.0 23500.0 1.75 2.3846 0.9992 3553235 CHDI2_001265 COc1ccc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J21 compound treatment 168200.0 11500.0 0.78 168280.0 13100.0 0.98 1.2453 0.9939 3552955 CHDI2_001266 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J22 compound treatment 180880.0 24200.0 1.65 175160.0 20000.0 1.49 2.2186 0.9988 3553843 CHDI2_001267 COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J23 mock treatment 161760.0 5040.0 0.34 154880.0 -255.0 -0.02 0.2296 0.667 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 J24 mock treatment 153880.0 -2840.0 -0.19 149760.0 -5380.0 -0.4 -0.4197 -0.9445 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K01 compound treatment 183080.0 26400.0 1.8 187280.0 32100.0 2.39 2.9625 0.9901 3552103 CHDI2_001268 COc1cccc(OC)c1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K02 compound treatment 185120.0 28400.0 1.94 184720.0 29600.0 2.2 2.9262 0.9979 3552353 CHDI2_001269 OC[C@@H](O)[C@@H](O)[C@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K03 compound treatment 181920.0 25200.0 1.72 185800.0 30700.0 2.28 2.8287 0.9902 1913656 CHDI2_001270 COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K04 compound treatment 192400.0 35700.0 2.43 192480.0 37300.0 2.78 3.6855 0.9978 3552357 CHDI2_001271 C[C@@H](O)[C@@H](O)[C@@H](O)C/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K05 compound treatment 199800.0 43100.0 2.94 201280.0 46100.0 3.43 4.5054 0.997 3552108 CHDI2_001272 COc1cc(O)cc(OC)c1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K06 compound treatment 186640.0 29900.0 2.04 186360.0 31200.0 2.32 3.0857 0.9979 3552361 CHDI2_001273 OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K07 compound treatment 180120.0 23400.0 1.6 180320.0 25200.0 1.87 2.4535 0.9968 3552977 CHDI2_001274 O=C(N/N=C/Cc1ccccc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K08 compound treatment 185080.0 28400.0 1.93 188680.0 33500.0 2.5 3.1326 0.992 3552898 CHDI2_001275 O=C(N/N=C/c1ccc2ccccc2n1)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K09 compound treatment 192760.0 36000.0 2.46 194640.0 39500.0 2.94 3.8165 0.996 3552111 CHDI2_001276 CC1(C)COC(CCC/C=N/NC(=O)c2ccccc2O)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K10 compound treatment 188000.0 31300.0 2.13 190080.0 34900.0 2.6 3.3471 0.9951 3552365 CHDI2_001277 OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K11 compound treatment 190080.0 33400.0 2.27 194320.0 39200.0 2.92 3.6705 0.9924 3552115 CHDI2_001278 Cc1nnc(Sc2ccc(/C=N/NC(=O)c3ccccc3O)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K12 compound treatment 184920.0 28200.0 1.92 189600.0 34500.0 2.57 3.1733 0.9899 3552366 CHDI2_001279 OC[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K13 compound treatment 191360.0 34600.0 2.36 197440.0 42300.0 3.15 3.8964 0.99 3552118 CHDI2_001280 Oc1ccccc1C(=O)N/N=C/c2cc(Br)cs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K14 compound treatment 184800.0 28100.0 1.91 188240.0 33100.0 2.46 3.096 0.9922 3552369 CHDI2_001281 C[C@H](O)[C@H](O)[C@@H](O)[C@@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K15 compound treatment 162960.0 6240.0 0.43 162200.0 7060.0 0.53 0.6727 0.9945 3552981 CHDI2_001282 COC(=O)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K16 compound treatment 159680.0 2960.0 0.2 163920.0 8780.0 0.65 0.6051 0.8843 3552902 CHDI2_001283 Cc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K17 compound treatment 185000.0 28300.0 1.93 180240.0 25100.0 1.87 2.6846 0.9999 3552121 CHDI2_001284 CC(C)(C)OC(=O)NC/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K18 compound treatment 200360.0 43600.0 2.98 200840.0 45700.0 3.4 4.5092 0.9978 3552373 CHDI2_001285 Oc1ccccc1C(=O)N/N=C/c2ccc(Oc3ccccc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K19 compound treatment 186720.0 30000.0 2.05 184160.0 29000.0 2.16 2.9738 0.9996 3552125 CHDI2_001286 Oc1ccccc1C(=O)N/N=C/c2ccc-3c(Cc4ccccc43)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K20 compound treatment 180920.0 24200.0 1.65 180240.0 25100.0 1.87 2.4879 0.9981 3552377 CHDI2_001287 Oc1ccccc1C(=O)N/N=C/c2cc[n+]([O-])cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K21 compound treatment 177080.0 20400.0 1.39 177240.0 22100.0 1.65 2.1449 0.9964 1922658 CHDI2_001288 Oc1ccccc1C(=O)N/N=C/c2ccc(F)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K22 compound treatment 185880.0 29200.0 1.99 186600.0 31500.0 2.34 3.0617 0.9967 3552381 CHDI2_001289 Oc1ccccc1C(=O)N/N=C/c2ccc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K23 mock treatment 156080.0 -639.0 -0.04 157600.0 2460.0 0.18 0.0989 0.5246 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 K24 mock treatment 158640.0 1920.0 0.13 155760.0 625.0 0.05 0.1255 0.9029 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L01 compound treatment 176160.0 19400.0 1.33 175920.0 20800.0 1.55 2.0311 0.997 3552603 CHDI2_001290 COc1cccc(OC)c1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L02 compound treatment 175400.0 18700.0 1.27 179960.0 24800.0 1.85 2.2071 0.9835 3214346 CHDI2_001291 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L03 compound treatment 175480.0 18800.0 1.28 174840.0 19700.0 1.47 1.9415 0.9977 3552607 CHDI2_001292 COc1ccc(/C=N/NC(=O)c2ccccn2)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L04 compound treatment 182560.0 25800.0 1.76 182520.0 27400.0 2.04 2.687 0.9974 3214446 CHDI2_001293 CCCCCCC/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L05 compound treatment 195600.0 38900.0 2.65 198520.0 43400.0 3.23 4.1576 0.9952 3552611 CHDI2_001294 COc1cc(O)cc(OC)c1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L06 compound treatment 179360.0 22600.0 1.54 185800.0 30700.0 2.28 2.7053 0.9819 3214578 CHDI2_001295 COc1cc(Br)c(/C=N/NC(=O)CCCCCC(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L07 compound treatment 169560.0 12800.0 0.88 171920.0 16800.0 1.25 1.5024 0.9849 3552957 CHDI2_001296 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L08 compound treatment 206880.0 50200.0 3.42 207080.0 51900.0 3.87 5.1519 0.9981 3214706 CHDI2_001297 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L09 compound treatment 189920.0 33200.0 2.26 186600.0 31500.0 2.34 3.2565 0.9999 3552614 CHDI2_001298 CC1(C)COC(CCC/C=N/NC(=O)c2ccccn2)OC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L10 compound treatment 178080.0 21400.0 1.46 180640.0 25500.0 1.9 2.372 0.9914 3214810 CHDI2_001299 C/C(=N\NC(=O)CCCCCC(=O)NO)/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L11 compound treatment 184440.0 27700.0 1.89 183920.0 28800.0 2.14 2.8513 0.998 3552618 CHDI2_001300 Cc1nnc(Sc2ccc(/C=N/NC(=O)c3ccccn3)o2)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L12 compound treatment 197680.0 41000.0 2.79 196360.0 41200.0 3.07 4.1442 0.9989 3553399 CHDI2_001301 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)c3cccc(c3)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L13 compound treatment 164880.0 8160.0 0.56 162880.0 7740.0 0.58 0.801 0.9998 3552622 CHDI2_001302 Brc1csc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L14 compound treatment 185880.0 29200.0 1.99 188000.0 32900.0 2.45 3.1354 0.9947 3553462 CHDI2_001303 CCCCCCC/C=N/NC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L15 compound treatment 180760.0 24000.0 1.64 176520.0 21400.0 1.59 2.2844 0.9999 3552961 CHDI2_001304 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2ccccn2)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L16 compound treatment 197320.0 40600.0 2.77 194160.0 39000.0 2.9 4.0111 0.9997 3553506 CHDI2_001305 COc1cc(Br)c(/C=N/NC(=O)c2cccc(c2)C(=O)NO)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L17 compound treatment 180120.0 23400.0 1.6 174080.0 18900.0 1.41 2.1251 0.9981 3552626 CHDI2_001306 CC(C)(C)OC(=O)NC/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L18 compound treatment 188760.0 32000.0 2.18 189080.0 33900.0 2.53 3.3311 0.9974 3553553 CHDI2_001307 COc1cc(/C=N/NC(=O)c2cccc(c2)C(=O)NO)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L19 compound treatment 171520.0 14800.0 1.01 175960.0 20800.0 1.55 1.8095 0.9784 3552630 CHDI2_001308 O=C(N/N=C/c1ccc-2c(Cc3ccccc32)c1)c4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L20 compound treatment 179000.0 22300.0 1.52 179280.0 24100.0 1.8 2.3448 0.9965 3554247 CHDI2_001309 C/C(=N\NC(=O)c1cccc(c1)C(=O)NO)/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L21 compound treatment 170440.0 13700.0 0.94 160840.0 5700.0 0.42 0.9617 0.9361 3552634 CHDI2_001310 Fc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L22 compound treatment 167320.0 10600.0 0.72 168160.0 13000.0 0.97 1.1965 0.9895 3552755 CHDI2_001311 CC1(C)[C@@H]2C[C@H]1C(=CC2)/C=N/NC(=O)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L23 mock treatment 154760.0 -1960.0 -0.13 156000.0 865.0 0.06 -0.0489 -0.33 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 L24 mock treatment 153640.0 -3080.0 -0.21 155760.0 625.0 0.05 -0.1155 -0.5375 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M01 compound treatment 184160.0 27400.0 1.87 187160.0 32000.0 2.38 3.0083 0.9928 3552129 CHDI2_001312 Oc1ccc(/C=N/NC(=O)c2ccccc2O)cc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M02 compound treatment 186280.0 29600.0 2.02 186440.0 31300.0 2.33 3.0726 0.9974 3552383 CHDI2_001313 Cc1ccccc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M03 compound treatment 213560.0 56800.0 3.88 212800.0 57700.0 4.29 5.775 0.9987 3552133 CHDI2_001314 Oc1ccccc1C(=O)N/N=C/c2ccc(F)c(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M04 compound treatment 189680.0 33000.0 2.25 193680.0 38500.0 2.87 3.6175 0.9927 3552385 CHDI2_001315 COc1cc(/C=N/NC(=O)c2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M05 compound treatment 212120.0 55400.0 3.78 209560.0 54400.0 4.05 5.535 0.9994 3552138 CHDI2_001316 Oc1ccc(F)cc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M06 compound treatment 195080.0 38400.0 2.62 199280.0 44100.0 3.29 4.1726 0.9936 3552386 CHDI2_001317 O[C@@H](/C=N/NC(=O)c1ccccc1O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M07 compound treatment 240600.0 83900.0 5.72 244520.0 89400.0 6.65 8.7479 0.9972 3552142 CHDI2_001318 Oc1ccccc1C(=O)N/N=C/c2coc3ccccc3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M08 compound treatment 192120.0 35400.0 2.41 198000.0 42900.0 3.19 3.9625 0.9905 3552388 CHDI2_001319 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M09 compound treatment 194680.0 38000.0 2.59 191120.0 36000.0 2.68 3.7238 0.9999 3552985 CHDI2_001320 O=C(N/N=C/c1cc2ccccc2n1S(=O)(=O)c3ccccc3)c4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M10 compound treatment 189280.0 32600.0 2.22 184480.0 29300.0 2.18 3.1141 1.0 3552910 CHDI2_001321 O[C@@H](/C=N/NC(=O)c1ccccn1)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M11 compound treatment 196120.0 39400.0 2.69 194040.0 38900.0 2.9 3.9469 0.9993 3552146 CHDI2_001322 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M12 compound treatment 189440.0 32700.0 2.23 193040.0 37900.0 2.82 3.5723 0.9932 1919426 CHDI2_001323 COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M13 compound treatment 191880.0 35200.0 2.4 194120.0 39000.0 2.9 3.7467 0.9955 3552862 CHDI2_001324 O=C(N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3)c4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M14 compound treatment 184480.0 27800.0 1.89 178000.0 22900.0 1.7 2.5416 0.9986 3552913 CHDI2_001325 OC[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M15 compound treatment 186920.0 30200.0 2.06 185920.0 30800.0 2.29 3.0761 0.9986 3552150 CHDI2_001326 OB(O)c1cccc(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M16 compound treatment 195480.0 38800.0 2.64 190240.0 35100.0 2.61 3.7161 1.0 3552389 CHDI2_001327 CCOc1cccc(/C=N/NC(=O)c2ccccc2O)c1OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M17 compound treatment 182120.0 25400.0 1.73 180400.0 25300.0 1.88 2.5542 0.9992 1913661 CHDI2_001328 Oc1ccccc1C(=O)N/N=C/c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M18 compound treatment 198760.0 42000.0 2.87 199880.0 44700.0 3.33 4.3815 0.9972 3552391 CHDI2_001329 Oc1ccccc1C(=O)N/N=C/c2cc(I)cc(I)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M19 compound treatment 184120.0 27400.0 1.87 189320.0 34200.0 2.54 3.12 0.9885 3552154 CHDI2_001330 Oc1ccccc1C(=O)N/N=C/c2ccoc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M20 compound treatment 183240.0 26500.0 1.81 175440.0 20300.0 1.51 2.3471 0.996 1912672 CHDI2_001331 CN(C)c1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M21 compound treatment 172120.0 15400.0 1.05 173480.0 18300.0 1.37 1.7079 0.9916 3552158 CHDI2_001332 Oc1cccc(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M22 compound treatment 192080.0 35400.0 2.41 192840.0 37700.0 2.81 3.689 0.9971 1919995 CHDI2_001333 CCn1c2ccccc2c3cc(/C=N/NC(=O)c4ccccc4O)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M23 mock treatment 163200.0 6480.0 0.44 160080.0 4940.0 0.37 0.5727 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 M24 mock treatment 157560.0 841.0 0.06 158760.0 3620.0 0.27 0.2313 0.8387 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N01 compound treatment 156880.0 161.0 0.01 159720.0 4580.0 0.34 0.2491 0.7295 3552638 CHDI2_001334 Oc1ccc(/C=N/NC(=O)c2ccccn2)cc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N02 compound treatment 175840.0 19100.0 1.3 177840.0 22700.0 1.69 2.1167 0.9918 3213540 CHDI2_001335 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N03 compound treatment 185040.0 28300.0 1.93 182480.0 27300.0 2.04 2.8044 0.9997 3552642 CHDI2_001336 Fc1ccc(/C=N/NC(=O)c2ccccn2)cc1Oc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N04 compound treatment 226200.0 69500.0 4.74 209360.0 54200.0 4.04 6.2033 0.9968 3213580 CHDI2_001337 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(c(F)c1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N05 compound treatment 234600.0 77900.0 5.31 231240.0 76100.0 5.66 7.7597 0.9995 3552646 CHDI2_001338 Oc1ccc(F)cc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N06 compound treatment 189640.0 32900.0 2.24 188200.0 33100.0 2.46 3.3272 0.9989 3213542 CHDI2_001339 Oc1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N07 compound treatment 195520.0 38800.0 2.65 199760.0 44600.0 3.32 4.219 0.9936 3552650 CHDI2_001340 O=C(N/N=C/c1coc2ccccc2c1=O)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N08 compound treatment 174280.0 17600.0 1.2 179640.0 24500.0 1.82 2.1362 0.9792 3213578 CHDI2_001341 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(c(F)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N09 compound treatment 187120.0 30400.0 2.07 190880.0 35700.0 2.66 3.3468 0.9924 3552965 CHDI2_001342 CN(C)CCCOc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N10 compound treatment 188080.0 31400.0 2.14 185760.0 30600.0 2.28 3.1236 0.9995 3214696 CHDI2_001343 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N11 compound treatment 195560.0 38800.0 2.65 188640.0 33500.0 2.49 3.6357 0.9995 3552654 CHDI2_001344 CC(C)(C)OC(=O)Nc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N12 compound treatment 199520.0 42800.0 2.92 192520.0 37400.0 2.78 4.0308 0.9997 3214698 CHDI2_001345 Oc1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N13 compound treatment 200560.0 43800.0 2.99 196960.0 41800.0 3.11 4.3147 0.9998 3552969 CHDI2_001346 CCOc1cc(/C=N/NC(=O)c2ccccn2)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N14 compound treatment 231960.0 75200.0 5.13 234600.0 79500.0 5.91 7.8093 0.9975 3214734 CHDI2_001347 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(c(F)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N15 compound treatment 179640.0 22900.0 1.56 177320.0 22200.0 1.65 2.2725 0.9996 3552658 CHDI2_001348 OB(O)c1cccc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N16 compound treatment 179640.0 22900.0 1.56 179440.0 24300.0 1.81 2.3841 0.9973 3215306 CHDI2_001349 ONC(=O)CCCCC(=O)N/N=C/c1ccc(O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N17 compound treatment 178920.0 22200.0 1.51 177480.0 22300.0 1.66 2.2462 0.9989 1937927 CHDI2_001350 O=C(N/N=C/c1ccco1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N18 compound treatment 188560.0 31800.0 2.17 189160.0 34000.0 2.53 3.3257 0.9971 3215346 CHDI2_001351 ONC(=O)CCCCC(=O)N/N=C/c1ccc(c(F)c1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N19 compound treatment 172400.0 15700.0 1.07 175640.0 20500.0 1.53 1.8351 0.9848 3552663 CHDI2_001352 O=C(N/N=C/c1ccoc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N20 compound treatment 176040.0 19300.0 1.32 177560.0 22400.0 1.67 2.1116 0.9931 3553309 CHDI2_001353 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N21 compound treatment 124040.0 -32700.0 -2.23 122920.0 -32200.0 -2.4 -3.2708 -0.9993 3552665 CHDI2_001354 Oc1cccc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N22 compound treatment 176080.0 19400.0 1.32 175360.0 20200.0 1.51 1.9978 0.9979 3553913 CHDI2_001355 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N23 mock treatment 158080.0 1360.0 0.09 160560.0 5420.0 0.4 0.3511 0.8475 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 N24 mock treatment 152640.0 -4080.0 -0.28 155560.0 425.0 0.03 -0.1743 -0.6227 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O01 compound treatment 173680.0 17000.0 1.16 181640.0 26500.0 1.97 2.2126 0.9676 3552163 CHDI2_001356 OCCOc1ccccc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O02 compound treatment 183240.0 26500.0 1.81 188200.0 33100.0 2.46 3.0187 0.9885 3552395 CHDI2_001357 Oc1ccccc1C(=O)N/N=C/c2ccc(o2)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O03 compound treatment 166840.0 10100.0 0.69 171200.0 16100.0 1.2 1.3334 0.9659 3552167 CHDI2_001358 OCCOc1cccc(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O04 compound treatment 188400.0 31700.0 2.16 183600.0 28500.0 2.12 3.0253 1.0 3552397 CHDI2_001359 Cn1cc(/C=N/NC(=O)c2ccccc2O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O05 compound treatment 180000.0 23300.0 1.59 183440.0 28300.0 2.11 2.612 0.9903 3552171 CHDI2_001360 OCCOc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O06 compound treatment 195880.0 39200.0 2.67 198800.0 43700.0 3.25 4.1859 0.9952 3552399 CHDI2_001361 Oc1ccccc1C(=O)N/N=C/c2cn(Cc3ccccc3)c4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O07 compound treatment 231320.0 74600.0 5.09 226080.0 70900.0 5.28 7.3301 0.9998 3552175 CHDI2_001362 COc1ccc(/C=N/NC(=O)c2ccccc2O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O08 compound treatment 190200.0 33500.0 2.28 180760.0 25600.0 1.91 2.9626 0.996 3552401 CHDI2_001363 Oc1ccccc1C(=O)N/N=C/C2=CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O09 compound treatment 223160.0 66400.0 4.53 221040.0 65900.0 4.91 6.6714 0.9992 3552179 CHDI2_001364 COc1ccc(O)c(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O10 compound treatment 184920.0 28200.0 1.92 184440.0 29300.0 2.18 2.9018 0.998 3552403 CHDI2_001365 OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)/C=N/NC(=O)c1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O11 compound treatment 192000.0 35300.0 2.41 187640.0 32500.0 2.42 3.4115 1.0 3552866 CHDI2_001366 O=C(N/N=C/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3)c4ccccn4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O12 compound treatment 128920.0 -27800.0 -1.9 126840.0 -28300.0 -2.11 -2.8293 -0.9986 3552915 CHDI2_001367 COc1ccc(/C=N/NC(=O)c2ccccn2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O13 compound treatment 195320.0 38600.0 2.63 195600.0 40500.0 3.01 3.9905 0.9977 3552184 CHDI2_001368 COc1cc(/C=C/C=N/NC(=O)c2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O14 compound treatment 170760.0 14000.0 0.96 191080.0 35900.0 2.68 2.5686 0.904 3552404 CHDI2_001369 OC[C@@H](O)[C@@H](O[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@H]1O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O15 compound treatment 199360.0 42600.0 2.91 199200.0 44100.0 3.28 4.3747 0.9982 3552188 CHDI2_001370 Cc1ccc(O)c(/C=N/NC(=O)c2ccccc2O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O16 compound treatment 185720.0 29000.0 1.98 184320.0 29200.0 2.17 2.934 0.9989 3552406 CHDI2_001371 OC[C@H]1O[C@H](OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)/C=N/NC(=O)c2ccccc2O)[C@H](O)[C@@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O17 compound treatment 187160.0 30400.0 2.08 186240.0 31100.0 2.32 3.1045 0.9985 3552191 CHDI2_001372 OCc1ccc(/C=N/NC(=O)c2ccccc2O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O18 compound treatment 186200.0 29500.0 2.01 186400.0 31300.0 2.33 3.0666 0.9973 3554239 CHDI2_001373 C/C(=N\NC(=O)c1ccccc1O)/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O19 compound treatment 196040.0 39300.0 2.68 205360.0 50200.0 3.74 4.5388 0.9867 3552195 CHDI2_001374 Oc1ccccc1C(=O)N/N=C/c2ccc3ccccc3c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O20 compound treatment 180600.0 23900.0 1.63 186080.0 30900.0 2.3 2.7798 0.9856 3552408 CHDI2_001375 CN(C)CCCOc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O21 compound treatment 182800.0 26100.0 1.78 186240.0 31100.0 2.32 2.8943 0.9915 3552199 CHDI2_001376 Oc1ccccc1C(=O)N/N=C/c2ccc(o2)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O22 compound treatment 173360.0 16600.0 1.13 174320.0 19200.0 1.43 1.8119 0.9935 3552410 CHDI2_001377 CCOc1cc(/C=N/NC(=O)c2ccccc2O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O23 mock treatment 155520.0 -1200.0 -0.08 165840.0 10700.0 0.8 0.5056 0.6313 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 O24 mock treatment 151640.0 -5080.0 -0.35 151680.0 -3460.0 -0.26 -0.4267 -0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P01 compound treatment 172840.0 16100.0 1.1 171600.0 16500.0 1.23 1.6437 0.9985 3552673 CHDI2_001378 OCCOc1ccccc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P02 compound treatment 180000.0 23300.0 1.59 181720.0 26600.0 1.98 2.5214 0.994 3213622 CHDI2_001379 ONC(=O)CCCCCCC(=O)N/N=C/c1cc(Br)c(O)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P03 compound treatment 78720.0 -78000.0 -5.32 77320.0 -77800.0 -5.79 -7.8554 -0.9991 3552677 CHDI2_001380 OCCOc1cccc(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P04 compound treatment 161080.0 4360.0 0.3 163160.0 8020.0 0.6 0.6326 0.9481 3213666 CHDI2_001381 CN(CCO)c1ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P05 compound treatment 124040.0 -32700.0 -2.23 123160.0 -32000.0 -2.38 -3.2582 -0.9995 3552680 CHDI2_001382 OCCOc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P06 compound treatment 190640.0 33900.0 2.31 190080.0 34900.0 2.6 3.4743 0.9983 3213624 CHDI2_001383 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cc(Br)c(O)c(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P07 compound treatment 119600.0 -37100.0 -2.53 109520.0 -45600.0 -3.4 -4.1901 -0.9895 3552684 CHDI2_001384 COc1ccc(/C=N/NC(=O)c2ccccn2)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P08 compound treatment 182280.0 25600.0 1.74 177800.0 22700.0 1.69 2.4251 0.9999 3213664 CHDI2_001385 CN(CCO)c1ccc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P09 compound treatment 240920.0 84200.0 5.74 239520.0 84400.0 6.28 8.5002 0.999 3552688 CHDI2_001386 COc1ccc(O)c(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P10 compound treatment 199520.0 42800.0 2.92 204120.0 49000.0 3.65 4.6413 0.9939 3214778 CHDI2_001387 ONC(=O)CCCCCC(=O)N/N=C/c1cc(Br)c(O)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P11 compound treatment 110440.0 -46300.0 -3.16 121000.0 -34100.0 -2.54 -4.0275 -0.9942 3552973 CHDI2_001388 CN(CCO)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P12 compound treatment 184520.0 27800.0 1.9 187120.0 32000.0 2.38 3.0235 0.9936 3214780 CHDI2_001389 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cc(Br)c(O)c(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P13 compound treatment 195520.0 38800.0 2.65 199680.0 44500.0 3.32 4.2148 0.9937 3552692 CHDI2_001390 COc1cc(/C=C/C=N/NC(=O)c2ccccn2)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P14 compound treatment 173280.0 16600.0 1.13 176000.0 20900.0 1.55 1.8964 0.9877 3214820 CHDI2_001391 CN(CCO)c1ccc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P15 compound treatment 243200.0 86500.0 5.9 258040.0 103000.0 7.66 9.5848 0.9916 3552696 CHDI2_001392 Cc1ccc(O)c(/C=N/NC(=O)c2ccccn2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P16 compound treatment 197080.0 40400.0 2.75 197120.0 42000.0 3.12 4.1553 0.998 3215388 CHDI2_001393 ONC(=O)CCCCC(=O)N/N=C/c1cc(Br)c(O)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P17 compound treatment 171520.0 14800.0 1.01 169600.0 14500.0 1.08 1.4748 0.9995 3552700 CHDI2_001394 OCc1ccc(/C=N/NC(=O)c2ccccn2)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P18 compound treatment 164840.0 8120.0 0.55 163520.0 8380.0 0.62 0.8328 0.9982 3215432 CHDI2_001395 CN(CCO)c1ccc(/C=N/NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P19 compound treatment 193120.0 36400.0 2.48 196080.0 40900.0 3.05 3.9097 0.9948 3552703 CHDI2_001396 Oc1c(/C=N/NC(=O)c2ccccn2)ccc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P20 compound treatment 183400.0 26700.0 1.82 188800.0 33700.0 2.51 3.058 0.9876 3553350 CHDI2_001397 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cc(Br)c(O)c(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P21 compound treatment 192000.0 35300.0 2.41 197080.0 41900.0 3.12 3.9083 0.9917 3552707 CHDI2_001398 Clc1cccc(c1)c2ccc(/C=N/NC(=O)c3ccccn3)o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P22 compound treatment 179720.0 23000.0 1.57 183840.0 28700.0 2.14 2.6195 0.9884 3553954 CHDI2_001399 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cc(Br)c(O)c(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P23 mock treatment 151600.0 -5120.0 -0.35 158280.0 3140.0 0.23 -0.0813 -0.1934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2406 P24 mock treatment 154120.0 -2600.0 -0.18 149720.0 -5420.0 -0.4 -0.4103 -0.9319 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A01 compound treatment 175520.0 18300.0 1.25 159280.0 6590.0 0.49 1.2282 0.9168 3553992 CHDI2_001400 Cc1[nH]cnc1/C=N/NC(=O)c2ccc(cc2)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A02 compound treatment 174880.0 17600.0 1.2 167440.0 14700.0 1.1 1.6268 0.999 3634596 CHDI2_001401 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A03 compound treatment 178240.0 21000.0 1.43 180280.0 27600.0 2.05 2.4645 0.9845 3551957 CHDI2_001402 Oc1ccccc1C(=O)N/N=C/C(=C/c2ccccc2)/Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A04 compound treatment 159560.0 2330.0 0.16 161360.0 8670.0 0.65 0.5683 0.8555 3634598 CHDI2_001403 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A05 compound treatment 175880.0 18600.0 1.27 174080.0 21400.0 1.59 2.0245 0.9938 3552237 CHDI2_001404 Cc1[nH]cnc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A06 compound treatment 160680.0 3450.0 0.23 162720.0 10000.0 0.75 0.6939 0.8868 3634600 CHDI2_001405 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OC/C=C/COc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A07 compound treatment 158560.0 1330.0 0.09 156560.0 3870.0 0.29 0.2675 0.8865 3552453 CHDI2_001406 Br/C(=C\c1ccccc1)/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A08 compound treatment 208480.0 51200.0 3.49 209560.0 56900.0 4.23 5.4633 0.9955 3634602 CHDI2_001407 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A09 compound treatment 190200.0 33000.0 2.25 184880.0 32200.0 2.4 3.2832 0.9995 3634604 CHDI2_001408 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CN3CCCCCCC3)CC(O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A10 compound treatment 162200.0 4970.0 0.34 165960.0 13300.0 0.99 0.9377 0.8982 3634605 CHDI2_001409 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A11 compound treatment 180280.0 23000.0 1.57 173800.0 21100.0 1.57 2.2219 1.0 3562114 CHDI2_001410 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CSc3nc(c(o3)c4ccccc4)c5ccccc5)CC(O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A12 compound treatment 223560.0 66300.0 4.52 213880.0 61200.0 4.55 6.4176 1.0 3634607 CHDI2_001411 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A13 compound treatment 214840.0 57600.0 3.93 188360.0 35700.0 2.65 4.6542 0.9818 3561878 CHDI2_001412 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2CC(CSc3nc(c(o3)c4ccccc4)c5ccccc5)OC(O2)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A14 compound treatment 201360.0 44100.0 3.01 186080.0 33400.0 2.48 3.8844 0.9955 3634609 CHDI2_001413 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A15 compound treatment 154840.0 -2390.0 -0.16 151760.0 -933.0 -0.07 -0.1645 -0.9274 3614528 CHDI2_001414 COC(=O)c1cn(CC(=O)Nc2ccon2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A16 compound treatment 172360.0 15100.0 1.03 173680.0 21000.0 1.56 1.8337 0.9797 3634611 CHDI2_001415 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A17 compound treatment 153880.0 -3350.0 -0.23 156240.0 3550.0 0.26 0.025 0.0716 3614462 CHDI2_001416 COC(=O)c1cn(CCNC(=O)[C@H](Cc2ccccc2)NS(=O)(=O)c3ccc(C)cc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A18 compound treatment 172760.0 15500.0 1.06 175160.0 22500.0 1.67 1.9309 0.9757 3634613 CHDI2_001417 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A19 compound treatment 198040.0 40800.0 2.78 193440.0 40700.0 3.03 4.1117 0.9991 3614540 CHDI2_001418 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCn3cc(nn3)c4ccccc4N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A20 compound treatment 175560.0 18300.0 1.25 164480.0 11800.0 0.88 1.5038 0.985 3634615 CHDI2_001419 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A21 compound treatment 237920.0 80700.0 5.5 271560.0 119000.0 8.85 10.1455 0.9739 3614392 CHDI2_001420 ONC(=O)/C=C/c1ccc(OCc2ccc(Cl)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A22 compound treatment 162600.0 5370.0 0.37 158280.0 5590.0 0.42 0.5528 0.998 3634617 CHDI2_001421 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A23 mock treatment 154400.0 -2830.0 -0.19 146440.0 -6250.0 -0.47 -0.4657 -0.9242 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 A24 mock treatment 149320.0 -7910.0 -0.54 149600.0 -3090.0 -0.23 -0.5443 -0.9279 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B01 compound treatment 160080.0 2850.0 0.19 155040.0 2350.0 0.17 0.2608 0.9986 3634619 CHDI2_001422 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B02 compound treatment 171560.0 14300.0 0.98 167080.0 14400.0 1.07 1.4478 0.9989 3634621 CHDI2_001423 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B03 compound treatment 165080.0 7850.0 0.53 167480.0 14800.0 1.1 1.1565 0.9451 3634623 CHDI2_001424 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B04 compound treatment 160480.0 3250.0 0.22 157480.0 4790.0 0.36 0.4085 0.9738 3634625 CHDI2_001425 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B05 compound treatment 163680.0 6450.0 0.44 162560.0 9870.0 0.73 0.8301 0.9699 3634627 CHDI2_001426 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OC/C=C/COc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B06 compound treatment 159520.0 2290.0 0.16 163000.0 10300.0 0.77 0.6527 0.8337 3634629 CHDI2_001427 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OC/C=C/COc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B07 compound treatment 190840.0 33600.0 2.29 184800.0 32100.0 2.39 3.3098 0.9998 3634631 CHDI2_001428 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B08 compound treatment 160080.0 2850.0 0.19 158040.0 5350.0 0.4 0.4186 0.9455 3634633 CHDI2_001429 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B09 compound treatment 165160.0 7930.0 0.54 164880.0 12200.0 0.91 1.0235 0.9694 3634635 CHDI2_001430 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B10 compound treatment 161200.0 3970.0 0.27 156160.0 3470.0 0.26 0.3737 0.9997 3634637 CHDI2_001431 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B11 compound treatment 196520.0 39300.0 2.68 193400.0 40700.0 3.03 4.0363 0.9981 3634639 CHDI2_001432 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B12 compound treatment 166680.0 9450.0 0.64 158400.0 5710.0 0.42 0.7558 0.9796 3634641 CHDI2_001433 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B13 compound treatment 170440.0 13200.0 0.9 166400.0 13700.0 1.02 1.358 0.9981 3634643 CHDI2_001434 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B14 compound treatment 165040.0 7810.0 0.53 159680.0 6990.0 0.52 0.7441 0.9999 3634645 CHDI2_001435 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B15 compound treatment 166400.0 9170.0 0.62 163600.0 10900.0 0.81 1.0159 0.9916 3634647 CHDI2_001436 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B16 compound treatment 160240.0 3010.0 0.2 152720.0 27.5 0.0 0.1464 0.7141 3634649 CHDI2_001437 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B17 compound treatment 164800.0 7570.0 0.52 159480.0 6790.0 0.51 0.722 0.9999 3634651 CHDI2_001438 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B18 compound treatment 155760.0 -1470.0 -0.1 163280.0 10600.0 0.79 0.4861 0.612 3634653 CHDI2_001439 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B19 compound treatment 164920.0 7690.0 0.52 166960.0 14300.0 1.06 1.1214 0.947 3634655 CHDI2_001440 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B20 compound treatment 159240.0 2010.0 0.14 158560.0 5870.0 0.44 0.4055 0.8861 3634657 CHDI2_001441 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B21 compound treatment 159040.0 1810.0 0.12 157400.0 4710.0 0.35 0.3348 0.9016 3634659 CHDI2_001442 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B22 compound treatment 152520.0 -4710.0 -0.32 152520.0 -173.0 -0.01 -0.2363 -0.7348 3634661 CHDI2_001443 ONC(=O)CCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B23 mock treatment 152840.0 -4390.0 -0.3 152280.0 -413.0 -0.03 -0.2335 -0.7755 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 B24 mock treatment 148960.0 -8270.0 -0.56 145480.0 -7210.0 -0.54 -0.7784 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C01 compound treatment 220200.0 63000.0 4.29 203360.0 50700.0 3.77 5.702 0.9979 3554029 CHDI2_001444 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C02 compound treatment 174440.0 17200.0 1.17 182360.0 29700.0 2.21 2.3908 0.9562 3634663 CHDI2_001445 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C03 compound treatment 187360.0 30100.0 2.05 186720.0 34000.0 2.53 3.2431 0.9946 3551993 CHDI2_001446 Oc1ccc(Br)cc1/C=N/NC(=O)c2ccccc2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C04 compound treatment 175240.0 18000.0 1.23 171200.0 18500.0 1.38 1.8421 0.9983 3634665 CHDI2_001447 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C05 compound treatment 188480.0 31200.0 2.13 184160.0 31500.0 2.34 3.1624 0.9989 3552272 CHDI2_001448 Oc1ccccc1C(=O)N/N=C/c2cccc(Oc3ccccc3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C06 compound treatment 179880.0 22600.0 1.54 181560.0 28900.0 2.15 2.611 0.9869 3634667 CHDI2_001449 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OC/C=C/COc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C07 compound treatment 234760.0 77500.0 5.29 243480.0 90800.0 6.76 8.5154 0.9926 3552490 CHDI2_001450 Oc1ccc(Br)cc1/C=N/NC(=O)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C08 compound treatment 210760.0 53500.0 3.65 214560.0 61900.0 4.6 5.8364 0.9934 3634669 CHDI2_001451 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C09 compound treatment 165320.0 8090.0 0.55 163920.0 11200.0 0.84 0.9807 0.9796 3634671 CHDI2_001452 CN(CC=C)CC1CC(OC(O1)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C10 compound treatment 170920.0 13700.0 0.93 167120.0 14400.0 1.07 1.4191 0.9976 3634672 CHDI2_001453 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C11 compound treatment 187960.0 30700.0 2.09 183560.0 30900.0 2.3 3.1057 0.9989 3634674 CHDI2_001454 OCc1ccc(cc1)[C@@H]2C[C@H](CSc3nc(c(o3)c4ccccc4)c5ccccc5)OC(O2)c6ccc(NC(=O)CCCCCCC(=O)O)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C12 compound treatment 188720.0 31500.0 2.15 188480.0 35800.0 2.66 3.4013 0.9943 3634675 CHDI2_001455 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C13 compound treatment 159600.0 2370.0 0.16 159640.0 6950.0 0.52 0.4797 0.8856 3614424 CHDI2_001456 COC(=O)c1cn(CC(=O)N2CCC3(CC2)N(CNC3=O)c4ccccc4)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C14 compound treatment 169360.0 12100.0 0.83 166520.0 13800.0 1.03 1.3123 0.9941 3634677 CHDI2_001457 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C15 compound treatment 162360.0 5130.0 0.35 164360.0 11700.0 0.87 0.8612 0.92 3614530 CHDI2_001458 COC(=O)c1cn(C[C@H](Cc2ccccc2)NC(=O)Nc3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C16 compound treatment 171880.0 14600.0 1.0 175000.0 22300.0 1.66 1.8801 0.9704 3634679 CHDI2_001459 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C17 compound treatment 157200.0 -33.8 0.0 151320.0 -1370.0 -0.1 -0.0739 -0.7229 3614464 CHDI2_001460 COC(=O)c1cn(CCNC(=O)[C@@H](NS(=O)(=O)c2ccc(C)cc2)C(C)C)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C18 compound treatment 166200.0 8970.0 0.61 163200.0 10500.0 0.78 0.9852 0.9926 3634681 CHDI2_001461 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C19 compound treatment 159280.0 2050.0 0.14 156960.0 4270.0 0.32 0.3232 0.9318 3614594 CHDI2_001462 Nc1ccccc1c2cn(CC(=O)Nc3nccs3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C20 compound treatment 165360.0 8130.0 0.55 160480.0 7790.0 0.58 0.8016 0.9997 3634683 CHDI2_001463 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C21 compound treatment 224520.0 67300.0 4.59 220160.0 67500.0 5.02 6.7944 0.999 3614389 CHDI2_001464 ONC(=O)/C=C/c1ccc(OCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C22 compound treatment 172480.0 15200.0 1.04 161840.0 9150.0 0.68 1.2164 0.979 3634685 CHDI2_001465 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(OCCCCCCCCCCCCOc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C23 mock treatment 154840.0 -2390.0 -0.16 150480.0 -2210.0 -0.16 -0.2318 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 C24 mock treatment 154840.0 -2390.0 -0.16 148800.0 -3890.0 -0.29 -0.3203 -0.9631 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D01 compound treatment 193160.0 35900.0 2.45 188560.0 35900.0 2.67 3.6196 0.9991 3634687 CHDI2_001466 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D02 compound treatment 176000.0 18800.0 1.28 177440.0 24700.0 1.84 2.2071 0.9841 3634689 CHDI2_001467 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D03 compound treatment 166160.0 8930.0 0.61 164880.0 12200.0 0.91 1.0717 0.9812 3634691 CHDI2_001468 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D04 compound treatment 179080.0 21800.0 1.49 180040.0 27300.0 2.04 2.4924 0.9882 3634693 CHDI2_001469 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D05 compound treatment 180280.0 23000.0 1.57 167040.0 14300.0 1.07 1.8661 0.9823 3634695 CHDI2_001470 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OC/C=C/COc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D06 compound treatment 172000.0 14800.0 1.01 165840.0 13100.0 0.98 1.4038 0.9999 3634697 CHDI2_001471 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OC/C=C/COc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D07 compound treatment 175920.0 18700.0 1.27 179720.0 27000.0 2.01 2.3232 0.9757 3634699 CHDI2_001472 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D08 compound treatment 181240.0 24000.0 1.64 179800.0 27100.0 2.02 2.5839 0.9946 3634701 CHDI2_001473 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D09 compound treatment 168200.0 11000.0 0.75 163280.0 10600.0 0.79 1.0859 0.9997 3634703 CHDI2_001474 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D10 compound treatment 174040.0 16800.0 1.15 171960.0 19300.0 1.43 1.8242 0.9938 3634705 CHDI2_001475 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D11 compound treatment 169920.0 12700.0 0.86 168320.0 15600.0 1.16 1.434 0.9894 3634707 CHDI2_001476 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D12 compound treatment 175320.0 18100.0 1.23 171360.0 18700.0 1.39 1.8543 0.9982 3634709 CHDI2_001477 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D13 compound treatment 164480.0 7250.0 0.49 169120.0 16400.0 1.22 1.2139 0.9205 3634711 CHDI2_001478 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D14 compound treatment 172000.0 14800.0 1.01 166200.0 13500.0 1.01 1.4227 1.0 3634713 CHDI2_001479 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D15 compound treatment 169000.0 11800.0 0.8 169800.0 17100.0 1.27 1.4676 0.9752 3634715 CHDI2_001480 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D16 compound treatment 167040.0 9810.0 0.67 162280.0 9590.0 0.71 0.9773 0.9995 3634717 CHDI2_001481 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D17 compound treatment 165880.0 8650.0 0.59 160560.0 7870.0 0.59 0.8309 1.0 3634719 CHDI2_001482 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D18 compound treatment 169680.0 12400.0 0.85 165920.0 13200.0 0.98 1.2961 0.9973 3634721 CHDI2_001483 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D19 compound treatment 175360.0 18100.0 1.24 172520.0 19800.0 1.48 1.9173 0.9961 3634723 CHDI2_001484 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D20 compound treatment 164640.0 7410.0 0.5 161720.0 9030.0 0.67 0.8321 0.9901 3634725 CHDI2_001485 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D21 compound treatment 163040.0 5810.0 0.4 161240.0 8550.0 0.64 0.7297 0.9739 3634727 CHDI2_001486 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D22 compound treatment 155080.0 -2150.0 -0.15 154160.0 1470.0 0.11 -0.0266 -0.1453 3634729 CHDI2_001487 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D23 mock treatment 152200.0 -5030.0 -0.34 149120.0 -3570.0 -0.27 -0.4307 -0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 D24 mock treatment 152840.0 -4390.0 -0.3 150240.0 -2450.0 -0.18 -0.3409 -0.9718 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E01 compound treatment 178800.0 21600.0 1.47 178520.0 25800.0 1.92 2.3989 0.9912 3554048 CHDI2_001488 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2nccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E02 compound treatment 208320.0 51100.0 3.48 194880.0 42200.0 3.14 4.683 0.9987 3634731 CHDI2_001489 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E03 compound treatment 177880.0 20600.0 1.41 175800.0 23100.0 1.72 2.2114 0.9951 3552029 CHDI2_001490 OC(=O)c1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E04 compound treatment 176760.0 19500.0 1.33 172200.0 19500.0 1.45 1.968 0.9991 3634733 CHDI2_001491 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E05 compound treatment 186840.0 29600.0 2.02 180600.0 27900.0 2.08 2.896 0.9999 3552300 CHDI2_001492 Oc1ccccc1C(=O)N/N=C/c2nccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E06 compound treatment 183040.0 25800.0 1.76 177040.0 24300.0 1.81 2.5254 0.9999 3634735 CHDI2_001493 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OC/C=C/COc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E07 compound treatment 169800.0 12600.0 0.86 169800.0 17100.0 1.27 1.5061 0.9814 3552525 CHDI2_001494 OC(=O)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E08 compound treatment 211640.0 54400.0 3.71 199680.0 47000.0 3.5 5.0957 0.9996 3634737 CHDI2_001495 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E09 compound treatment 194280.0 37000.0 2.53 189200.0 36500.0 2.72 3.7072 0.9993 3634739 CHDI2_001496 CN(CC1CC(OC(O1)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c3ccccc3)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E10 compound treatment 179560.0 22300.0 1.52 179360.0 26700.0 1.98 2.4798 0.9914 3634740 CHDI2_001497 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E11 compound treatment 189360.0 32100.0 2.19 188960.0 36300.0 2.7 3.4574 0.9946 3634742 CHDI2_001498 CN(C[C@H]1C[C@H](OC(O1)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c3ccc(CO)cc3)Cc4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E12 compound treatment 183920.0 26700.0 1.82 181920.0 29200.0 2.18 2.8247 0.9961 3634743 CHDI2_001499 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E13 compound treatment 166360.0 9130.0 0.62 165680.0 13000.0 0.97 1.1235 0.9773 3614478 CHDI2_001500 COC(=O)c1cn(CC(=O)N2CCN(C)CC2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E14 compound treatment 176800.0 19600.0 1.33 173360.0 20700.0 1.54 2.0309 0.9975 3634745 CHDI2_001501 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E15 compound treatment 166200.0 8970.0 0.61 166640.0 13900.0 1.04 1.1663 0.9681 3614432 CHDI2_001502 COC(=O)c1cn(C[C@@H](Cc2ccccc2)NC(=O)Nc3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E16 compound treatment 178920.0 21700.0 1.48 175760.0 23100.0 1.72 2.2594 0.9972 3634747 CHDI2_001503 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E17 compound treatment 166560.0 9330.0 0.64 159520.0 6830.0 0.51 0.8089 0.9938 3614467 CHDI2_001504 COC(=O)c1cn(C[C@@H]2CCCN2S(=O)(=O)c3ccc(C)cc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E18 compound treatment 178480.0 21200.0 1.45 177520.0 24800.0 1.85 2.3309 0.9927 3634749 CHDI2_001505 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E19 compound treatment 165480.0 8250.0 0.56 164720.0 12000.0 0.9 1.0305 0.9749 3614596 CHDI2_001506 Nc1ccccc1c2cn(CC(=O)Nc3ccon3)nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E20 compound treatment 181840.0 24600.0 1.68 178360.0 25700.0 1.91 2.537 0.9979 3634751 CHDI2_001507 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E21 compound treatment 238320.0 81100.0 5.53 218360.0 65700.0 4.89 7.365 0.9981 3614386 CHDI2_001508 ONC(=O)/C=C/c1ccc(OCc2ccc-3c(Cc4ccccc43)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E22 compound treatment 185720.0 28500.0 1.94 177880.0 25200.0 1.87 2.6988 0.9998 3634753 CHDI2_001509 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E23 mock treatment 158440.0 1210.0 0.08 152600.0 -92.5 -0.01 0.0533 0.6457 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 E24 mock treatment 163240.0 6010.0 0.41 157160.0 4470.0 0.33 0.5247 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F01 compound treatment 169600.0 12400.0 0.84 171000.0 18300.0 1.36 1.5596 0.9734 3634755 CHDI2_001510 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F02 compound treatment 172280.0 15000.0 1.03 173880.0 21200.0 1.58 1.8404 0.9783 3634757 CHDI2_001511 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1OC\C=C\COc2ccc(/C=N/NC(=O)CCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F03 compound treatment 172360.0 15100.0 1.03 172280.0 19600.0 1.46 1.7601 0.9856 3634759 CHDI2_001512 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F04 compound treatment 184520.0 27300.0 1.86 180640.0 27900.0 2.08 2.7862 0.9984 3634761 CHDI2_001513 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1OCCCCCOc2ccc(/C=N/NC(=O)CCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F05 compound treatment 179600.0 22400.0 1.52 171680.0 19000.0 1.41 2.0775 0.9993 3634763 CHDI2_001514 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OC/C=C/COc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F06 compound treatment 172760.0 15500.0 1.06 173440.0 20700.0 1.54 1.8404 0.983 3634765 CHDI2_001515 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1OCCCCCCOc2ccc(/C=N/NC(=O)CCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F07 compound treatment 177240.0 20000.0 1.36 179960.0 27300.0 2.03 2.3995 0.9813 3634767 CHDI2_001516 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F08 compound treatment 183760.0 26500.0 1.81 176920.0 24200.0 1.8 2.5538 1.0 3634769 CHDI2_001517 CCOc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1OC\C=C\COc2ccc(/C=N/NC(=O)CCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F09 compound treatment 179320.0 22100.0 1.51 169960.0 17300.0 1.29 1.9735 0.9969 3634771 CHDI2_001518 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F10 compound treatment 168800.0 11600.0 0.79 169480.0 16800.0 1.25 1.4411 0.9754 3634773 CHDI2_001519 CCOc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1OCCCCCOc2ccc(/C=N/NC(=O)CCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F11 compound treatment 172640.0 15400.0 1.05 170400.0 17700.0 1.32 1.6746 0.9937 3634775 CHDI2_001520 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F12 compound treatment 173040.0 15800.0 1.08 176920.0 24200.0 1.8 2.037 0.9697 3634777 CHDI2_001521 CCOc1cc(/C=N/NC(=O)CCCCC(=O)NO)ccc1OCCCCCCOc2ccc(/C=N/NC(=O)CCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F13 compound treatment 184440.0 27200.0 1.85 182600.0 29900.0 2.23 2.8855 0.9959 3634779 CHDI2_001522 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F14 compound treatment 174240.0 17000.0 1.16 164800.0 12100.0 0.9 1.457 0.9922 3634781 CHDI2_001523 COc1cc(OC/C=C/COc2cc(OC)c(\C=N\NC(=O)CCCCC(=O)NO)c(OC)c2)cc(OC)c1\C=N\NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F15 compound treatment 187280.0 30000.0 2.05 185600.0 32900.0 2.45 3.1803 0.9961 3634783 CHDI2_001524 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F16 compound treatment 169360.0 12100.0 0.83 169280.0 16600.0 1.23 1.4575 0.981 3634785 CHDI2_001525 COc1cc(OCCCCCOc2cc(OC)c(/C=N/NC(=O)CCCCC(=O)NO)c(OC)c2)cc(OC)c1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F17 compound treatment 186040.0 28800.0 1.96 182640.0 29900.0 2.23 2.9648 0.998 3634787 CHDI2_001526 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F18 compound treatment 169840.0 12600.0 0.86 167840.0 15100.0 1.13 1.4049 0.991 3634789 CHDI2_001527 COc1cc(OCCCCCCOc2cc(OC)c(/C=N/NC(=O)CCCCC(=O)NO)c(OC)c2)cc(OC)c1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F19 compound treatment 180080.0 22800.0 1.56 171720.0 19000.0 1.42 2.1028 0.9989 3634791 CHDI2_001528 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F20 compound treatment 170480.0 13200.0 0.9 167880.0 15200.0 1.13 1.4379 0.9938 3634793 CHDI2_001529 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)cc(OC)c1OC\C=C\COc2c(OC)cc(/C=N/NC(=O)CCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F21 compound treatment 177920.0 20700.0 1.41 176200.0 23500.0 1.75 2.2344 0.9943 3634795 CHDI2_001530 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(OCCCCCCCCCCCCOc3cccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F22 compound treatment 164000.0 6770.0 0.46 159800.0 7110.0 0.53 0.7002 0.9977 3634797 CHDI2_001531 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)cc(OC)c1OCCCCCOc2c(OC)cc(/C=N/NC(=O)CCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F23 mock treatment 158000.0 766.0 0.05 156200.0 3510.0 0.26 0.2215 0.8321 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 F24 mock treatment 157080.0 -154.0 -0.01 149480.0 -3210.0 -0.24 -0.1765 -0.7374 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G01 compound treatment 179200.0 22000.0 1.5 176400.0 23700.0 1.76 2.3066 0.9967 3554086 CHDI2_001532 NC(=O)COc1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G02 compound treatment 197640.0 40400.0 2.75 185440.0 32700.0 2.44 3.6713 0.9981 3634799 CHDI2_001533 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G03 compound treatment 184960.0 27700.0 1.89 181320.0 28600.0 2.13 2.8432 0.9982 3552065 CHDI2_001534 CCCCN(CCCC)c1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G04 compound treatment 185640.0 28400.0 1.94 180640.0 27900.0 2.08 2.8402 0.9994 3634801 CHDI2_001535 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G05 compound treatment 187920.0 30700.0 2.09 185520.0 32800.0 2.44 3.207 0.997 3552337 CHDI2_001536 NC(=O)COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G06 compound treatment 191440.0 34200.0 2.33 184160.0 31500.0 2.34 3.3051 1.0 3634803 CHDI2_001537 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OC/C=C/COc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G07 compound treatment 232640.0 75400.0 5.14 222600.0 69900.0 5.2 7.3143 1.0 3552561 CHDI2_001538 CCCCN(CCCC)c1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G08 compound treatment 197240.0 40000.0 2.73 190680.0 38000.0 2.83 3.9278 0.9998 3634805 CHDI2_001539 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G09 compound treatment 250640.0 93400.0 6.37 237840.0 85100.0 6.34 8.9841 1.0 3634807 CHDI2_001540 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2CC(OC(O2)c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G10 compound treatment 178280.0 21000.0 1.43 183840.0 31100.0 2.32 2.6538 0.9734 3634808 CHDI2_001541 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G11 compound treatment 201080.0 43800.0 2.99 187400.0 34700.0 2.58 3.9403 0.9974 3634810 CHDI2_001542 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C(=O)c2ccc(NC(=O)CCCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G12 compound treatment 186440.0 29200.0 1.99 180640.0 27900.0 2.08 2.8788 0.9998 3634811 CHDI2_001543 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G13 compound treatment 171360.0 14100.0 0.96 171080.0 18400.0 1.37 1.6487 0.9852 3614494 CHDI2_001544 COC(=O)c1cn(CC(=O)N2CCN(CC2)c3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G14 compound treatment 181800.0 24600.0 1.67 181240.0 28500.0 2.12 2.6867 0.9931 3634813 CHDI2_001545 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G15 compound treatment 173720.0 16500.0 1.12 172920.0 20200.0 1.51 1.8593 0.9896 3614437 CHDI2_001546 COC(=O)c1cn(C[C@H](Cc2ccccc2)NC(=O)c3ccccc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G16 compound treatment 187160.0 29900.0 2.04 184320.0 31600.0 2.35 3.1072 0.9975 3634815 CHDI2_001547 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G17 compound treatment 169240.0 12000.0 0.82 169080.0 16400.0 1.22 1.4412 0.9812 3614479 CHDI2_001548 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)Cn2cc(nn2)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G18 compound treatment 179880.0 22600.0 1.54 183400.0 30700.0 2.29 2.7078 0.9818 3634817 CHDI2_001549 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G19 compound treatment 174400.0 17200.0 1.17 168440.0 15700.0 1.17 1.6563 1.0 3614693 CHDI2_001550 COC(=O)c1cn(CC(=O)O)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G20 compound treatment 192200.0 35000.0 2.38 181760.0 29100.0 2.16 3.2154 0.9988 3634819 CHDI2_001551 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G21 compound treatment 249600.0 92400.0 6.3 229920.0 77200.0 5.75 8.5171 0.999 3614403 CHDI2_001552 ONC(=O)/C=C/c1ccc(OCCn2c3ccccc3c4ccccc24)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G22 compound treatment 178920.0 21700.0 1.48 174400.0 21700.0 1.62 2.1879 0.999 3634821 CHDI2_001553 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCCCCCCCCCCCCOc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G23 mock treatment 165280.0 8050.0 0.55 156360.0 3670.0 0.27 0.5809 0.9481 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 G24 mock treatment 157360.0 126.0 0.01 156560.0 3870.0 0.29 0.2096 0.7279 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H01 compound treatment 171640.0 14400.0 0.98 175720.0 23000.0 1.71 1.9064 0.9651 3634823 CHDI2_001554 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H02 compound treatment 173880.0 16600.0 1.13 173280.0 20600.0 1.53 1.886 0.9891 3634825 CHDI2_001555 COc1cc(OC/C=C/COc2ccc(\C=N\NC(=O)CCCCC(=O)NO)c(OC)c2)ccc1\C=N\NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H03 compound treatment 190440.0 33200.0 2.26 191960.0 39300.0 2.92 3.6674 0.992 3634827 CHDI2_001556 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H04 compound treatment 175200.0 18000.0 1.22 180280.0 27600.0 2.05 2.318 0.9695 3634829 CHDI2_001557 COc1cc(OCCCCCOc2ccc(/C=N/NC(=O)CCCCC(=O)NO)c(OC)c2)ccc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H05 compound treatment 185040.0 27800.0 1.9 185280.0 32600.0 2.43 3.0555 0.9926 3634831 CHDI2_001558 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OC/C=C/COc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H06 compound treatment 180040.0 22800.0 1.55 188560.0 35900.0 2.67 2.9871 0.9669 3634833 CHDI2_001559 COc1cc(OCCCCCCOc2ccc(/C=N/NC(=O)CCCCC(=O)NO)c(OC)c2)ccc1/C=N/NC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H07 compound treatment 189880.0 32600.0 2.23 186360.0 33700.0 2.51 3.3457 0.9983 3634835 CHDI2_001560 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H08 compound treatment 185960.0 28700.0 1.96 186160.0 33500.0 2.49 3.1462 0.9929 3634837 CHDI2_001561 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCc2ccc(COc3ccc(\C=N\NC(=O)CCCCC(=O)NO)cc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H09 compound treatment 254360.0 97100.0 6.62 236600.0 83900.0 6.24 9.0982 0.9996 3634839 CHDI2_001562 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H10 compound treatment 176720.0 19500.0 1.33 172440.0 19700.0 1.47 1.9787 0.9987 3634841 CHDI2_001563 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCc2cccc(COc3ccc(\C=N\NC(=O)CCCCC(=O)NO)cc3)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H11 compound treatment 214920.0 57700.0 3.93 209960.0 57300.0 4.26 5.7948 0.9992 3634843 CHDI2_001564 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H12 compound treatment 172600.0 15400.0 1.05 179880.0 27200.0 2.02 2.1716 0.953 3634845 CHDI2_001565 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCc2ccccc2COc3ccc(\C=N\NC(=O)CCCCC(=O)NO)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H13 compound treatment 248720.0 91500.0 6.24 235120.0 82400.0 6.13 8.7484 1.0 3634847 CHDI2_001566 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H14 compound treatment 170600.0 13400.0 0.91 173360.0 20700.0 1.54 1.732 0.9688 3634849 CHDI2_001567 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCc2ccccc2c3ccccc3COc4ccc(\C=N\NC(=O)CCCCC(=O)NO)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H15 compound treatment 172360.0 15100.0 1.03 174480.0 21800.0 1.62 1.8758 0.9761 3634851 CHDI2_001568 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H16 compound treatment 177320.0 20100.0 1.37 174200.0 21500.0 1.6 2.1002 0.997 3634853 CHDI2_001569 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H17 compound treatment 166280.0 9050.0 0.62 171960.0 19300.0 1.43 1.4501 0.9289 3634855 CHDI2_001570 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H18 compound treatment 189280.0 32000.0 2.18 184400.0 31700.0 2.36 3.2136 0.9993 3634857 CHDI2_001571 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H19 compound treatment 264800.0 108000.0 7.33 267440.0 115000.0 8.54 11.2245 0.9971 3634859 CHDI2_001572 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H20 compound treatment 177000.0 19800.0 1.35 168480.0 15800.0 1.18 1.7838 0.9977 3634861 CHDI2_001573 Cc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)c(O)c(/C=N/NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H21 compound treatment 327440.0 170000.0 11.6 264600.0 112000.0 8.33 14.0948 0.9868 3634863 CHDI2_001574 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H22 compound treatment 179880.0 22600.0 1.54 171520.0 18800.0 1.4 2.0826 0.9988 3634865 CHDI2_001575 Cc1cc(/C=N/NC(=O)CCCCCC(=O)NO)c(O)c(/C=N/NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H23 mock treatment 164280.0 7050.0 0.48 154480.0 1790.0 0.13 0.4338 0.8702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 H24 mock treatment 155600.0 -1630.0 -0.11 153120.0 428.0 0.03 -0.0563 -0.4857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I01 compound treatment 206760.0 49500.0 3.38 202800.0 50100.0 3.73 5.0246 0.9988 3554221 CHDI2_001576 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I02 compound treatment 201240.0 44000.0 3.0 197040.0 44300.0 3.3 4.4554 0.9989 3634867 CHDI2_001577 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I03 compound treatment 184120.0 26900.0 1.83 186200.0 33500.0 2.49 3.0596 0.9885 1922557 CHDI2_001578 COc1ccc(/C=N/NC(=O)c2ccccc2O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I04 compound treatment 193240.0 36000.0 2.45 195120.0 42400.0 3.16 3.9687 0.9922 3634869 CHDI2_001579 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I05 compound treatment 203480.0 46200.0 3.15 206480.0 53800.0 4.0 5.0602 0.993 3552422 CHDI2_001580 Oc1ccccc1C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I06 compound treatment 209320.0 52100.0 3.55 203720.0 51000.0 3.8 5.1965 0.9994 3634871 CHDI2_001581 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OC/C=C/COc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I07 compound treatment 181400.0 24200.0 1.65 176160.0 23500.0 1.75 2.4001 0.9996 3552599 CHDI2_001582 COc1ccc(/C=N/NC(=O)c2ccccn2)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I08 compound treatment 260280.0 103000.0 7.03 238640.0 85900.0 6.4 9.4909 0.9989 3634873 CHDI2_001583 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I09 compound treatment 179960.0 22700.0 1.55 173880.0 21200.0 1.58 2.2106 1.0 3634875 CHDI2_001584 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C(=O)NCCOCCOCCNC(=O)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I10 compound treatment 205080.0 47800.0 3.26 195520.0 42800.0 3.19 4.5605 0.9999 3634876 CHDI2_001585 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I11 compound treatment 178240.0 21000.0 1.43 178280.0 25600.0 1.9 2.3593 0.9901 468 CHDI2_001586 ONC(=O)CCCCCCC(=O)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I12 compound treatment 248680.0 91400.0 6.23 241200.0 88500.0 6.59 9.0664 0.9996 3634878 CHDI2_001587 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I13 compound treatment 176760.0 19500.0 1.33 171200.0 18500.0 1.38 1.9153 0.9999 3614495 CHDI2_001588 COC(=O)c1cn(CC(=O)N2CCOCC2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I14 compound treatment 196760.0 39500.0 2.69 191880.0 39200.0 2.92 3.9678 0.9992 3634880 CHDI2_001589 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I15 compound treatment 211080.0 53800.0 3.67 208000.0 55300.0 4.12 5.5065 0.9984 3614442 CHDI2_001590 COC(=O)c1cn(CCCNC(=S)Nc2ccc(cc2)[N+](=O)[O-])nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I16 compound treatment 219200.0 62000.0 4.22 211840.0 59100.0 4.4 6.1001 0.9998 3634882 CHDI2_001591 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I17 compound treatment 175640.0 18400.0 1.25 166200.0 13500.0 1.01 1.5982 0.994 3614485 CHDI2_001592 COC(=O)[C@@H](NC(=O)Cn1cc(nn1)C(=O)OC)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I18 compound treatment 186640.0 29400.0 2.0 182880.0 30200.0 2.25 3.0063 0.9984 3634884 CHDI2_001593 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I19 compound treatment 181280.0 24000.0 1.64 173640.0 20900.0 1.56 2.2616 0.9997 3614695 CHDI2_001594 COC(=O)c1cn(CCC(=O)O)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I20 compound treatment 189360.0 32100.0 2.19 181600.0 28900.0 2.15 3.0701 1.0 3634886 CHDI2_001595 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I21 compound treatment 240840.0 83600.0 5.7 240440.0 87700.0 6.53 8.6485 0.9977 3614398 CHDI2_001596 ONC(=O)/C=C/c1ccc(OCCCCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I22 compound treatment 174720.0 17500.0 1.19 168080.0 15400.0 1.15 1.6528 0.9998 3634888 CHDI2_001597 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(OCCCCCCCCCCCCOc3cccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I23 mock treatment 162520.0 5290.0 0.36 156080.0 3390.0 0.25 0.4331 0.9847 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 I24 mock treatment 157640.0 406.0 0.03 150680.0 -2010.0 -0.15 -0.0863 -0.5667 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J01 compound treatment 165160.0 7930.0 0.54 163680.0 11000.0 0.82 0.9604 0.9798 3634890 CHDI2_001598 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J02 compound treatment 172200.0 15000.0 1.02 173480.0 20800.0 1.55 1.8155 0.9796 3634892 CHDI2_001599 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1OC\C=C\COc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J03 compound treatment 170560.0 13300.0 0.91 170240.0 17500.0 1.31 1.5659 0.9843 3634894 CHDI2_001600 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J04 compound treatment 176480.0 19200.0 1.31 177440.0 24700.0 1.84 2.2302 0.9862 3634896 CHDI2_001601 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1OCCCCCOc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J05 compound treatment 187920.0 30700.0 2.09 183600.0 30900.0 2.3 3.1059 0.9989 3634898 CHDI2_001602 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OC/C=C/COc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J06 compound treatment 183160.0 25900.0 1.77 182240.0 29500.0 2.2 2.8049 0.9941 3634900 CHDI2_001603 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1OCCCCCCOc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J07 compound treatment 183080.0 25800.0 1.76 180200.0 27500.0 2.05 2.6937 0.9972 3634902 CHDI2_001604 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J08 compound treatment 186640.0 29400.0 2.0 180960.0 28300.0 2.1 2.9053 0.9997 3634904 CHDI2_001605 CCOc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1OC\C=C\COc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J09 compound treatment 211880.0 54600.0 3.73 208400.0 55700.0 4.15 5.5662 0.9986 3634906 CHDI2_001606 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J10 compound treatment 192680.0 35400.0 2.42 195600.0 42900.0 3.19 3.9669 0.9905 3634908 CHDI2_001607 CCOc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1OCCCCCOc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J11 compound treatment 191160.0 33900.0 2.31 188920.0 36200.0 2.7 3.5421 0.9971 3634910 CHDI2_001608 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J12 compound treatment 185400.0 28200.0 1.92 179400.0 26700.0 1.99 2.7634 0.9999 3634912 CHDI2_001609 CCOc1cc(/C=N/NC(=O)CCCCCC(=O)NO)ccc1OCCCCCCOc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J13 compound treatment 194960.0 37700.0 2.57 193440.0 40700.0 3.03 3.9632 0.9966 3634914 CHDI2_001610 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J14 compound treatment 183200.0 26000.0 1.77 181880.0 29200.0 2.17 2.7879 0.9948 3634916 CHDI2_001611 COc1cc(OC/C=C/COc2cc(OC)c(\C=N\NC(=O)CCCCCC(=O)NO)c(OC)c2)cc(OC)c1\C=N\NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J15 compound treatment 204960.0 47700.0 3.25 198320.0 45600.0 3.4 4.7021 0.9998 3634918 CHDI2_001612 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J16 compound treatment 180520.0 23300.0 1.59 175280.0 22600.0 1.68 2.3113 0.9996 3634920 CHDI2_001613 COc1cc(OCCCCCOc2cc(OC)c(/C=N/NC(=O)CCCCCC(=O)NO)c(OC)c2)cc(OC)c1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J17 compound treatment 211240.0 54000.0 3.68 207520.0 54800.0 4.08 5.489 0.9987 3634922 CHDI2_001614 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J18 compound treatment 178040.0 20800.0 1.42 176160.0 23500.0 1.75 2.2381 0.9947 3634924 CHDI2_001615 COc1cc(OCCCCCCOc2cc(OC)c(/C=N/NC(=O)CCCCCC(=O)NO)c(OC)c2)cc(OC)c1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J19 compound treatment 178600.0 21400.0 1.46 172360.0 19700.0 1.46 2.0651 1.0 3634926 CHDI2_001616 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J20 compound treatment 176400.0 19200.0 1.31 174080.0 21400.0 1.59 2.0495 0.9952 3634928 CHDI2_001617 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)cc(OC)c1OC\C=C\COc2c(OC)cc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J21 compound treatment 191160.0 33900.0 2.31 190720.0 38000.0 2.83 3.6368 0.995 3634930 CHDI2_001618 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J22 compound treatment 172600.0 15400.0 1.05 166680.0 14000.0 1.04 1.4769 1.0 3634932 CHDI2_001619 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)cc(OC)c1OCCCCCOc2c(OC)cc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J23 mock treatment 161720.0 4490.0 0.31 152720.0 27.5 0.0 0.2177 0.7118 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 J24 mock treatment 162400.0 5170.0 0.35 147240.0 -5450.0 -0.41 -0.0379 -0.0705 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K01 compound treatment 175080.0 17800.0 1.22 176000.0 23300.0 1.73 2.087 0.9849 3552785 CHDI2_001620 CCCCCCC/C=N/NC(=O)c1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K02 compound treatment 192880.0 35600.0 2.43 192960.0 40300.0 3.0 3.8376 0.9946 3634934 CHDI2_001621 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K03 compound treatment 181880.0 24600.0 1.68 180720.0 28000.0 2.09 2.6632 0.9942 3552859 CHDI2_001622 COc1cc(Br)c(/C=N/NC(=O)c2ccccn2)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K04 compound treatment 200800.0 43600.0 2.97 201720.0 49000.0 3.65 4.6805 0.9948 3634936 CHDI2_001623 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K05 compound treatment 186160.0 28900.0 1.97 188240.0 35500.0 2.65 3.2653 0.9895 3552906 CHDI2_001624 COc1cc(/C=N/NC(=O)c2ccccn2)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K06 compound treatment 199400.0 42200.0 2.87 193320.0 40600.0 3.02 4.1709 0.9997 3634938 CHDI2_001625 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OC/C=C/COc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K07 compound treatment 181640.0 24400.0 1.66 184320.0 31600.0 2.35 2.8411 0.9856 3554243 CHDI2_001626 C/C(=N\NC(=O)c1ccccn1)/C[P+](c2ccccc2)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K08 compound treatment 212640.0 55400.0 3.78 213160.0 60500.0 4.5 5.8533 0.9962 3634940 CHDI2_001627 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K09 compound treatment 185720.0 28500.0 1.94 185880.0 33200.0 2.47 3.1199 0.9929 3634942 CHDI2_001628 ONC(=O)CCCCCCC(=O)Nc1cccc(c1)C(=O)NCCOCCOCCNC(=O)c2cccc(NC(=O)CCCCCCC(=O)NO)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K10 compound treatment 192040.0 34800.0 2.37 196520.0 43800.0 3.26 3.9845 0.9878 3634943 CHDI2_001629 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K11 compound treatment 272680.0 115000.0 7.87 256440.0 104000.0 7.72 11.0255 1.0 3634945 CHDI2_001630 ONC(=O)/C=C/c1ccc(CN(CCC2=C[N]c3ccccc23)C(=O)CCCCC(=O)N(CCC4=C[N]c5ccccc45)Cc6ccc(\C=C\C(=O)NO)cc6)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K12 compound treatment 197480.0 40200.0 2.74 201360.0 48700.0 3.62 4.5015 0.9906 3634947 CHDI2_001631 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K13 compound treatment 175280.0 18000.0 1.23 174240.0 21500.0 1.6 2.004 0.9914 3614498 CHDI2_001632 COC(=O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K14 compound treatment 193200.0 36000.0 2.45 190320.0 37600.0 2.8 3.7141 0.9978 3634949 CHDI2_001633 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K15 compound treatment 170240.0 13000.0 0.89 171560.0 18900.0 1.4 1.62 0.9754 3614446 CHDI2_001634 COC(=O)c1cn(CCCNC(=O)Nc2ccccc2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K16 compound treatment 186200.0 29000.0 1.97 185560.0 32900.0 2.45 3.1262 0.9944 3634951 CHDI2_001635 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K17 compound treatment 174200.0 17000.0 1.16 171840.0 19100.0 1.43 1.8256 0.9946 3614488 CHDI2_001636 CCOC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)Cn3cc(nn3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K18 compound treatment 191520.0 34300.0 2.34 175200.0 22500.0 1.68 2.8374 0.9866 3634953 CHDI2_001637 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K19 compound treatment 214440.0 57200.0 3.9 211080.0 58400.0 4.35 5.8306 0.9985 3614383 CHDI2_001638 ONC(=O)/C=C/c1ccc(OCCc2cccs2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K20 compound treatment 181160.0 23900.0 1.63 176320.0 23600.0 1.76 2.3969 0.9993 3634955 CHDI2_001639 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K21 compound treatment 178200.0 21000.0 1.43 174600.0 21900.0 1.63 2.1637 0.9978 1917883 CHDI2_001640 O/N=C/1\C2(CCCCC2)C(=O)N(O)C31CCCC=C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K22 compound treatment 180520.0 23300.0 1.59 171960.0 19300.0 1.43 2.1366 0.9987 3634957 CHDI2_001641 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(OCCCCCCCCCCCCOc3cccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)c3)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K23 mock treatment 160240.0 3010.0 0.2 153600.0 908.0 0.07 0.1927 0.8929 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 K24 mock treatment 160960.0 3730.0 0.25 147640.0 -5050.0 -0.38 -0.0863 -0.1901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L01 compound treatment 180160.0 22900.0 1.56 172600.0 19900.0 1.48 2.1529 0.9996 3634959 CHDI2_001642 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L02 compound treatment 167480.0 10200.0 0.7 171880.0 19200.0 1.43 1.5038 0.9459 3634961 CHDI2_001643 COc1cc(OC/C=C/COc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)c(OC)c2)ccc1\C=N\NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L03 compound treatment 227640.0 70400.0 4.8 224320.0 71600.0 5.33 7.1638 0.9986 3634963 CHDI2_001644 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L04 compound treatment 183800.0 26600.0 1.81 179800.0 27100.0 2.02 2.7073 0.9986 3634965 CHDI2_001645 COc1cc(OCCCCCOc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)c(OC)c2)ccc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L05 compound treatment 197160.0 39900.0 2.72 201000.0 48300.0 3.6 4.4671 0.9906 3634967 CHDI2_001646 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OC/C=C/COc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L06 compound treatment 180720.0 23500.0 1.6 174760.0 22100.0 1.64 2.2936 0.9999 3634969 CHDI2_001647 COc1cc(OCCCCCCOc2ccc(/C=N/NC(=O)CCCCCC(=O)NO)c(OC)c2)ccc1/C=N/NC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L07 compound treatment 186000.0 28800.0 1.96 184680.0 32000.0 2.38 3.0702 0.9954 3634971 CHDI2_001648 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L08 compound treatment 177640.0 20400.0 1.39 175280.0 22600.0 1.68 2.1725 0.9956 3634973 CHDI2_001649 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCc2ccc(COc3ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L09 compound treatment 205080.0 47800.0 3.26 200080.0 47400.0 3.53 4.8005 0.9992 3634975 CHDI2_001650 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L10 compound treatment 198040.0 40800.0 2.78 194680.0 42000.0 3.13 4.1769 0.9983 3634977 CHDI2_001651 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCc2cccc(COc3ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc3)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L11 compound treatment 248040.0 90800.0 6.19 242000.0 89300.0 6.65 9.0777 0.9994 3634979 CHDI2_001652 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L12 compound treatment 184120.0 26900.0 1.83 179880.0 27200.0 2.02 2.727 0.9988 3634981 CHDI2_001653 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCc2ccccc2COc3ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L13 compound treatment 267040.0 110000.0 7.49 264040.0 111000.0 8.29 11.1535 0.9987 3634983 CHDI2_001654 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L14 compound treatment 170040.0 12800.0 0.87 168880.0 16200.0 1.2 1.4693 0.9875 3634985 CHDI2_001655 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCc2ccccc2c3ccccc3COc4ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L15 compound treatment 216000.0 58800.0 4.01 226280.0 73600.0 5.48 6.7058 0.9882 3634987 CHDI2_001656 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L16 compound treatment 177680.0 20400.0 1.39 172000.0 19300.0 1.44 2.0018 0.9999 3634989 CHDI2_001657 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(O)c(\C=N\NC(=O)CCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L17 compound treatment 309640.0 152000.0 10.39 296720.0 144000.0 10.72 14.9271 0.9999 3634991 CHDI2_001658 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L18 compound treatment 223080.0 65800.0 4.49 219920.0 67200.0 5.0 6.7124 0.9985 3634993 CHDI2_001659 Cc1cc(/C=N/NC(=O)CCCCC(=O)NO)c(O)c(/C=N/NC(=O)CCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L19 compound treatment 168880.0 11600.0 0.79 174720.0 22000.0 1.64 1.7207 0.9446 3634995 CHDI2_001660 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L20 compound treatment 196320.0 39100.0 2.66 187760.0 35100.0 2.61 3.7298 0.9999 3634997 CHDI2_001661 ONC(=O)CCCCC(=O)N/N=C/c1ccc(\C=N\NC(=O)CCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L21 compound treatment 177800.0 20600.0 1.4 173680.0 21000.0 1.56 2.096 0.9985 3634999 CHDI2_001662 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCCCCCCCCCCCCOc3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L22 compound treatment 168040.0 10800.0 0.74 164560.0 11900.0 0.88 1.1455 0.9959 3635001 CHDI2_001663 COc1cc(/C=N/NC(=O)CCCCC(=O)NO)cc(OC)c1OCCCCCCOc2c(OC)cc(/C=N/NC(=O)CCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L23 mock treatment 161160.0 3930.0 0.27 152960.0 268.0 0.02 0.2034 0.7576 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 L24 mock treatment 157400.0 166.0 0.01 150320.0 -2370.0 -0.18 -0.1168 -0.6604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M01 compound treatment 223040.0 65800.0 4.49 215600.0 62900.0 4.68 6.4831 0.9998 3554166 CHDI2_001664 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(c(F)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M02 compound treatment 186880.0 29600.0 2.02 191160.0 38500.0 2.86 3.4537 0.9855 3635003 CHDI2_001665 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M03 compound treatment 184760.0 27500.0 1.88 185120.0 32400.0 2.41 3.0336 0.9923 1922299 CHDI2_001666 Oc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M04 compound treatment 197520.0 40300.0 2.75 194000.0 41300.0 3.07 4.1161 0.9984 3635005 CHDI2_001667 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M05 compound treatment 188240.0 31000.0 2.11 187000.0 34300.0 2.55 3.3003 0.9956 3552393 CHDI2_001668 Oc1ccccc1C(=O)N/N=C/c2ccc(c(F)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M06 compound treatment 194720.0 37500.0 2.56 190120.0 37400.0 2.79 3.7769 0.9991 3635007 CHDI2_001669 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OC/C=C/COc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M07 compound treatment 172160.0 14900.0 1.02 165720.0 13000.0 0.97 1.4052 0.9997 3552669 CHDI2_001670 Oc1ccc(/C=N/NC(=O)c2ccccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M08 compound treatment 200600.0 43400.0 2.96 196160.0 43500.0 3.24 4.3782 0.999 3635009 CHDI2_001671 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M09 compound treatment 207240.0 50000.0 3.41 204240.0 51500.0 3.84 5.1235 0.9983 3635011 CHDI2_001672 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M10 compound treatment 198280.0 41000.0 2.8 196240.0 43500.0 3.24 4.2706 0.9973 3635012 CHDI2_001673 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M11 compound treatment 204360.0 47100.0 3.21 199840.0 47100.0 3.51 4.7531 0.999 3635014 CHDI2_001674 ONC(=O)/C=C/c1ccc(CNCCC2=C[N]c3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M12 compound treatment 205320.0 48100.0 3.28 198880.0 46200.0 3.44 4.7489 0.9997 3635016 CHDI2_001675 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M13 compound treatment 175480.0 18200.0 1.24 179600.0 26900.0 2.0 2.2957 0.9738 3614499 CHDI2_001676 COC(=O)c1cn(CC(=O)Nc2cc(OC)ccc2OC)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M14 compound treatment 193240.0 36000.0 2.45 195160.0 42500.0 3.16 3.9708 0.9922 3635018 CHDI2_001677 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M15 compound treatment 176640.0 19400.0 1.32 172800.0 20100.0 1.5 1.9938 0.9981 3614451 CHDI2_001678 COC(=O)c1cn(CCNC(=O)Nc2ccccc2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M16 compound treatment 193800.0 36600.0 2.49 197480.0 44800.0 3.33 4.1199 0.9898 3635020 CHDI2_001679 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M17 compound treatment 182440.0 25200.0 1.72 175840.0 23100.0 1.72 2.4334 1.0 3614488 CHDI2_001680 CCOC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)Cn3cc(nn3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M18 compound treatment 205440.0 48200.0 3.29 196080.0 43400.0 3.23 4.6073 1.0 3635022 CHDI2_001681 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M19 compound treatment 238640.0 81400.0 5.55 241600.0 88900.0 6.62 8.6035 0.9962 3614396 CHDI2_001682 ONC(=O)/C=C/c1ccc(OCCCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M20 compound treatment 198200.0 41000.0 2.79 201000.0 48300.0 3.6 4.5172 0.9922 3635024 CHDI2_001683 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M21 compound treatment 183440.0 26200.0 1.79 182440.0 29700.0 2.21 2.8289 0.9943 3614688 CHDI2_001684 COc1ccc(cc1OC2CCCC2)C3=NOC(C3)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M22 compound treatment 186320.0 29100.0 1.98 180760.0 28100.0 2.09 2.8793 0.9997 3635026 CHDI2_001685 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCCCCCCCCCCCCOc3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M23 mock treatment 165600.0 8370.0 0.57 159480.0 6790.0 0.51 0.7605 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 M24 mock treatment 159840.0 2610.0 0.18 154280.0 1590.0 0.12 0.2092 0.9803 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N01 compound treatment 168000.0 10800.0 0.73 170920.0 18200.0 1.36 1.4783 0.9584 3635028 CHDI2_001686 Cc1cc(/C=N/NC(=O)CCCCC(=O)Nc2ccccc2O)c(O)c(/C=N/NC(=O)CCCCC(=O)Nc3ccccc3O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N02 compound treatment 194600.0 37400.0 2.55 195480.0 42800.0 3.18 4.0532 0.9939 3635030 CHDI2_001687 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OC\C=C\COc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N03 compound treatment 178160.0 20900.0 1.43 176360.0 23700.0 1.76 2.2544 0.9945 3635032 CHDI2_001688 Cc1cc(/C=N/NC(=O)CCCCCC(=O)Nc2ccccc2O)c(O)c(/C=N/NC(=O)CCCCCC(=O)Nc3ccccc3O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N04 compound treatment 212600.0 55400.0 3.77 200800.0 48100.0 3.58 5.2009 0.9997 3635034 CHDI2_001689 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OCCCCCOc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N05 compound treatment 177720.0 20500.0 1.4 178280.0 25600.0 1.9 2.3342 0.9884 3635036 CHDI2_001690 Cc1cc(/C=N/NC(=O)CCCCCCC(=O)Nc2ccccc2O)c(O)c(/C=N/NC(=O)CCCCCCC(=O)Nc3ccccc3O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N06 compound treatment 206400.0 49200.0 3.35 200840.0 48100.0 3.58 4.9041 0.9994 3635038 CHDI2_001691 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OCCCCCCOc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N07 compound treatment 181680.0 24400.0 1.67 175080.0 22400.0 1.67 2.3567 1.0 3635040 CHDI2_001692 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(\C=N\NC(=O)CCCCC(=O)Nc3ccccc3O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N08 compound treatment 193880.0 36600.0 2.5 186240.0 33500.0 2.5 3.5322 1.0 3635042 CHDI2_001693 CCOc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OC\C=C\COc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N09 compound treatment 188480.0 31200.0 2.13 182040.0 29300.0 2.18 3.0508 0.9999 3635044 CHDI2_001694 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(\C=N\NC(=O)CCCCCC(=O)Nc3ccccc3O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N10 compound treatment 187080.0 29800.0 2.03 185440.0 32700.0 2.44 3.1623 0.996 3635046 CHDI2_001695 CCOc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OCCCCCOc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N11 compound treatment 186920.0 29700.0 2.02 180400.0 27700.0 2.06 2.8893 1.0 3635048 CHDI2_001696 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(\C=N\NC(=O)CCCCCCC(=O)Nc3ccccc3O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N12 compound treatment 189280.0 32000.0 2.18 177520.0 24800.0 1.85 2.8515 0.9965 3635050 CHDI2_001697 CCOc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OCCCCCCOc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N13 compound treatment 210440.0 53200.0 3.63 205720.0 53000.0 3.95 5.3557 0.9991 3635052 CHDI2_001698 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(O)c(\C=N\NC(=O)CCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N14 compound treatment 230640.0 73400.0 5.0 226240.0 73500.0 5.47 7.4094 0.999 3635054 CHDI2_001699 COc1cc(OC/C=C/COc2cc(OC)c(\C=N\NC(=O)CCCCCCC(=O)NO)c(OC)c2)cc(OC)c1\C=N\NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N15 compound treatment 222040.0 64800.0 4.42 230400.0 77700.0 5.78 7.2138 0.9912 3635056 CHDI2_001700 COc1cc(/C=N/NC(=O)CCCCCC(=O)NO)cc(OC)c1OCCCCCCOc2c(OC)cc(/C=N/NC(=O)CCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N16 compound treatment 182400.0 25200.0 1.72 180040.0 27300.0 2.04 2.6525 0.9964 3635058 CHDI2_001701 COc1cc(OCCCCCOc2cc(OC)c(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c2)cc(OC)c1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N17 compound treatment 215000.0 57800.0 3.94 206880.0 54200.0 4.03 5.6366 0.9999 3635060 CHDI2_001702 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc(OC)c1OCCCCCCOc2c(OC)cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N18 compound treatment 187840.0 30600.0 2.09 186040.0 33300.0 2.48 3.2305 0.9963 3635062 CHDI2_001703 COc1cc(OCCCCCCOc2cc(OC)c(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c2)cc(OC)c1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N19 compound treatment 186360.0 29100.0 1.99 188120.0 35400.0 2.64 3.2686 0.9902 3635064 CHDI2_001704 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CSc3nc4ccccc4o3)CC(O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N20 compound treatment 233360.0 76100.0 5.19 221240.0 68500.0 5.1 7.2774 1.0 3635065 CHDI2_001705 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc(OC)c1OC\C=C\COc2c(OC)cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N21 compound treatment 184440.0 27200.0 1.85 182920.0 30200.0 2.25 2.9024 0.9954 3215593 CHDI2_001706 OCCSCC1CC(OC(O1)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N22 compound treatment 172560.0 15300.0 1.04 172720.0 20000.0 1.49 1.7929 0.9849 3635067 CHDI2_001707 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc(OC)c1OCCCCCOc2c(OC)cc(/C=N/NC(=O)CCCCCCC(=O)NO)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N23 mock treatment 157000.0 -234.0 -0.02 163000.0 10300.0 0.77 0.5312 0.6923 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 N24 mock treatment 156320.0 -914.0 -0.06 155360.0 2670.0 0.2 0.0963 0.463 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O01 compound treatment 176840.0 19600.0 1.34 175160.0 22500.0 1.67 2.1276 0.9938 3554202 CHDI2_001708 CN(CCO)c1ccc(/C=N/NC(=O)c2ccc(cc2)C(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O02 compound treatment 181920.0 24700.0 1.68 185920.0 33200.0 2.47 2.9388 0.9824 3635069 CHDI2_001709 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O03 compound treatment 183480.0 26200.0 1.79 183960.0 31300.0 2.33 2.9108 0.9916 3552203 CHDI2_001710 Oc1ccccc1C(=O)N/N=C/c2cc(Br)c(O)c(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O04 compound treatment 196880.0 39600.0 2.7 188520.0 35800.0 2.67 3.7968 1.0 3635071 CHDI2_001711 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O05 compound treatment 180960.0 23700.0 1.62 182600.0 29900.0 2.23 2.7178 0.9877 3552412 CHDI2_001712 CN(CCO)c1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O06 compound treatment 204200.0 47000.0 3.2 197640.0 44900.0 3.35 4.6297 0.9998 3635073 CHDI2_001713 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OC/C=C/COc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O07 compound treatment 190320.0 33100.0 2.26 181400.0 28700.0 2.14 3.1058 0.9996 3552710 CHDI2_001714 Oc1c(Br)cc(/C=N/NC(=O)c2ccccn2)cc1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O08 compound treatment 187160.0 29900.0 2.04 189520.0 36800.0 2.74 3.3808 0.9894 3635075 CHDI2_001715 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O09 compound treatment 235720.0 78500.0 5.35 235240.0 82500.0 6.14 8.128 0.9976 3635077 CHDI2_001716 OCc1ccc(cc1)[C@@H]2C[C@H](CSc3nc(c(o3)c4ccccc4)c5ccccc5)OC(O2)c6ccc(NC(=O)CCCCCCC(=O)NO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O10 compound treatment 198080.0 40800.0 2.78 189040.0 36300.0 2.71 3.882 0.9999 3635078 CHDI2_001717 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O11 compound treatment 244000.0 86800.0 5.92 244240.0 91500.0 6.81 9.0008 0.9975 3635080 CHDI2_001718 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2CC(CSc3nc(c(o3)c4ccccc4)c5ccccc5)OC(O2)c6ccc(NC(=O)CCCCCCC(=O)NO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O12 compound treatment 195360.0 38100.0 2.6 186280.0 33600.0 2.5 3.6056 0.9998 3635081 CHDI2_001719 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O13 compound treatment 194160.0 36900.0 2.52 180200.0 27500.0 2.05 3.2278 0.9947 3614501 CHDI2_001720 COC(=O)c1cn(CC(=O)Nc2nccs2)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O14 compound treatment 193800.0 36600.0 2.49 189360.0 36700.0 2.73 3.6925 0.999 3635083 CHDI2_001721 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O15 compound treatment 167800.0 10600.0 0.72 169440.0 16700.0 1.25 1.3908 0.966 3614455 CHDI2_001722 COC(=O)c1cn(CCCNC(=O)[C@H](Cc2ccccc2)NS(=O)(=O)c3ccc(C)cc3)nn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O16 compound treatment 186520.0 29300.0 2.0 186280.0 33600.0 2.5 3.1795 0.9938 3635085 CHDI2_001723 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O17 compound treatment 192360.0 35100.0 2.39 189880.0 37200.0 2.77 3.6505 0.9974 3614538 CHDI2_001724 Cc1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccccc2)C(=O)NCCCn3cc(nn3)c4ccccc4N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O18 compound treatment 191360.0 34100.0 2.33 192240.0 39500.0 2.94 3.7265 0.9932 3635087 CHDI2_001725 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O19 compound treatment 214720.0 57500.0 3.92 212320.0 59600.0 4.44 5.9094 0.9981 3614394 CHDI2_001726 Nc1cccc(COc2ccc(/C=C/C(=O)NO)cc2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O20 compound treatment 183920.0 26700.0 1.82 176280.0 23600.0 1.76 2.5279 0.9998 3635089 CHDI2_001727 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O21 compound treatment 193160.0 35900.0 2.45 196000.0 43300.0 3.22 4.0111 0.9908 3614525 CHDI2_001728 ONC(=O)/C=C/c1ccc(OCCc2ccccc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O22 compound treatment 169280.0 12000.0 0.82 171800.0 19100.0 1.42 1.5863 0.966 3635091 CHDI2_001729 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCCCCCCCCCCCCOc3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O23 mock treatment 153360.0 -3870.0 -0.26 159280.0 6590.0 0.49 0.1599 0.2872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 O24 mock treatment 151440.0 -5790.0 -0.39 151240.0 -1450.0 -0.11 -0.3557 -0.8687 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P01 compound treatment 167200.0 9970.0 0.68 164640.0 11900.0 0.89 1.1092 0.9912 3635093 CHDI2_001730 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CSc3ccccc3)CC(O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P02 compound treatment 219560.0 62300.0 4.25 209960.0 57300.0 4.26 6.0185 1.0 3635094 CHDI2_001731 COc1cc(OC/C=C/COc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)c(OC)c2)ccc1\C=N\NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P03 compound treatment 193600.0 36400.0 2.48 189360.0 36700.0 2.73 3.6829 0.9989 3215583 CHDI2_001732 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CSc3ccccn3)CC(O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P04 compound treatment 210600.0 53400.0 3.64 203920.0 51200.0 3.81 5.2687 0.9997 3635096 CHDI2_001733 COc1cc(OCCCCCOc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c2)ccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P05 compound treatment 176600.0 19400.0 1.32 175600.0 22900.0 1.7 2.1392 0.992 3635098 CHDI2_001734 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CSc3nc4ccccc4s3)CC(O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P06 compound treatment 219960.0 62700.0 4.28 221360.0 68700.0 5.11 6.6377 0.9961 3635099 CHDI2_001735 COc1cc(OCCCCCCOc2ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c2)ccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P07 compound treatment 176640.0 19400.0 1.32 177600.0 24900.0 1.85 2.2464 0.9863 3635101 CHDI2_001736 CC(C)OCC1CC(OC(O1)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P08 compound treatment 180920.0 23700.0 1.61 185440.0 32700.0 2.44 2.8653 0.98 3635102 CHDI2_001737 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCc2ccc(COc3ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P09 compound treatment 190920.0 33700.0 2.3 196440.0 43700.0 3.26 3.9263 0.9854 3215599 CHDI2_001738 COCC1CC(OC(O1)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P10 compound treatment 180000.0 22800.0 1.55 181080.0 28400.0 2.11 2.5915 0.9885 3635104 CHDI2_001739 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCc2cccc(COc3ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc3)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P11 compound treatment 244400.0 87200.0 5.94 235360.0 82700.0 6.15 8.5527 0.9998 3635106 CHDI2_001740 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(COc3ccccc3)CC(O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P12 compound treatment 255280.0 98000.0 6.68 240040.0 87300.0 6.5 9.3236 0.9999 3635107 CHDI2_001741 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCc2ccccc2COc3ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P13 compound treatment 244080.0 86800.0 5.92 238280.0 85600.0 6.37 8.691 0.9993 3635109 CHDI2_001742 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)[C@@H]2O[C@H](CSc3ccncc3)C[C@@H](O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P14 compound treatment 227480.0 70200.0 4.79 224120.0 71400.0 5.32 7.1455 0.9986 3635110 CHDI2_001743 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCc2ccccc2c3ccccc3COc4ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P15 compound treatment 179360.0 22100.0 1.51 178160.0 25500.0 1.9 2.407 0.9936 3635112 CHDI2_001744 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)[C@H]2O[C@@H](CSc3ccncc3)C[C@H](O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P16 compound treatment 211640.0 54400.0 3.71 212040.0 59300.0 4.42 5.7462 0.9962 3635113 CHDI2_001745 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OCc2ccc(COc3ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc3OC)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P17 compound treatment 192600.0 35400.0 2.41 187720.0 35000.0 2.61 3.5484 0.9992 3635115 CHDI2_001746 COCC1CC(OC(O1)c2ccc(cc2)C3OC(COC)CC(O3)c4ccc(NC(=O)CCCCCCC(=O)NO)cc4)c5ccc(NC(=O)CCCCCCC(=O)NO)cc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P18 compound treatment 201280.0 44000.0 3.0 206760.0 54100.0 4.02 4.9688 0.9896 3635116 CHDI2_001747 COc1cc(/C=N/NC(=O)CCCCCCC(=O)NO)ccc1OCc2cccc(COc3ccc(/C=N/NC(=O)CCCCCCC(=O)NO)cc3OC)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P19 compound treatment 181000.0 23800.0 1.62 178360.0 25700.0 1.91 2.4966 0.9966 3215595 CHDI2_001748 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CSc3ccncc3)CC(O2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P20 compound treatment 208640.0 51400.0 3.5 207120.0 54400.0 4.05 5.3426 0.9974 3635118 CHDI2_001749 COc1cc(OCc2ccc(COc3ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c3)cc2)ccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P21 compound treatment 234560.0 77300.0 5.27 223920.0 71200.0 5.3 7.4763 1.0 3635120 CHDI2_001750 ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C2OC(CN(Cc3ccccc3)Cc4ccccc4)CC(O2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P22 compound treatment 189600.0 32400.0 2.21 190000.0 37300.0 2.78 3.5237 0.9935 3635121 CHDI2_001751 COc1cc(OCc2cccc(COc3ccc(/C=N/NC(=O)CCCCCCC(=O)NO)c(OC)c3)c2)ccc1/C=N/NC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P23 mock treatment 151920.0 -5310.0 -0.36 150840.0 -1850.0 -0.14 -0.3537 -0.9124 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2407 P24 mock treatment 152440.0 -4790.0 -0.33 153040.0 348.0 0.03 -0.2128 -0.6491 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A01 compound treatment 159560.0 -5080.0 -0.35 160440.0 -5920.0 -0.44 -0.5567 -0.9929 3622456 Ald3.1-H_000001 ONC(=O)CCCCC(=O)N/N=C/c1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A02 compound treatment 233440.0 68800.0 4.69 221160.0 54800.0 4.08 6.2005 0.9976 3622458 Ald3.1-H_000002 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A03 compound treatment 152960.0 -11700.0 -0.8 168160.0 1800.0 0.13 -0.4686 -0.5801 3622460 Ald3.1-H_000003 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A04 compound treatment 256840.0 92200.0 6.29 239960.0 73600.0 5.48 8.318 0.9976 3622462 Ald3.1-H_000004 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A05 compound treatment 173520.0 8880.0 0.61 173520.0 7160.0 0.53 0.8047 0.998 3622464 Ald3.1-H_000005 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A06 compound treatment 214520.0 49900.0 3.4 154680.0 -11700.0 -0.87 1.7897 0.5099 3622466 Ald3.1-H_000006 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A07 compound treatment 227600.0 63000.0 4.29 238000.0 71600.0 5.33 6.8052 0.9942 3622468 Ald3.1-H_000007 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A08 compound treatment 184480.0 19800.0 1.35 178920.0 12600.0 0.93 1.6172 0.9837 3622470 Ald3.1-H_000008 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A09 compound treatment 247760.0 83100.0 5.67 227920.0 61600.0 4.58 7.2466 0.9944 3622472 Ald3.1-H_000009 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A10 compound treatment 188560.0 23900.0 1.63 187960.0 21600.0 1.61 2.2897 1.0 3622474 Ald3.1-H_000010 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A11 compound treatment 242880.0 78200.0 5.33 211320.0 45000.0 3.35 6.1377 0.9748 3622476 Ald3.1-H_000011 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A12 compound treatment 197960.0 33300.0 2.27 192920.0 26600.0 1.98 3.0038 0.9976 3622478 Ald3.1-H_000012 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A13 mock treatment 154120.0 -10500.0 -0.72 153200.0 -13200.0 -0.98 -1.2 -0.9883 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A14 mock treatment 153920.0 -10700.0 -0.73 151840.0 -14500.0 -1.08 -1.2812 -0.9819 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A15 compound treatment 222320.0 57700.0 3.93 155880.0 -10500.0 -0.78 2.2289 0.556 3622480 Ald3.1-H_000013 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A16 compound treatment 160400.0 -4240.0 -0.29 158800.0 -7560.0 -0.56 -0.6025 -0.9522 3622482 Ald3.1-H_000014 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A17 compound treatment 232480.0 67800.0 4.62 222200.0 55800.0 4.16 6.2089 0.9986 3622484 Ald3.1-H_000015 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A18 compound treatment 157640.0 -7000.0 -0.48 161080.0 -5280.0 -0.39 -0.6156 -0.9953 3622486 Ald3.1-H_000016 CC(=O)N/N=C/c1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A19 compound treatment 224520.0 59900.0 4.08 222600.0 56200.0 4.19 5.8463 0.9999 3622488 Ald3.1-H_000017 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A20 compound treatment 152680.0 -12000.0 -0.82 154960.0 -11400.0 -0.85 -1.1768 -0.9998 3622490 Ald3.1-H_000018 O=Cc1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A21 compound treatment 220680.0 56000.0 3.82 242520.0 76200.0 5.67 6.7095 0.9816 3622492 Ald3.1-H_000019 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A22 compound treatment 148080.0 -16600.0 -1.13 156240.0 -10100.0 -0.75 -1.3312 -0.9806 3622494 Ald3.1-H_000020 OC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A23 compound treatment 185920.0 21300.0 1.45 186840.0 20500.0 1.52 2.1034 0.9997 3622496 Ald3.1-H_000021 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 A24 compound treatment 185120.0 20500.0 1.4 182920.0 16600.0 1.23 1.8586 0.9981 3622498 Ald3.1-H_000022 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B01 compound treatment 161840.0 -2800.0 -0.19 166120.0 -241.0 -0.02 -0.1479 -0.7701 3622500 Ald3.1-H_000023 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCC(=O)NO)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B02 compound treatment 235080.0 70400.0 4.8 237560.0 71200.0 5.3 7.1426 0.9988 3622502 Ald3.1-H_000024 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3ccc(OCCCCCCC(=O)NO)cc3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B03 compound treatment 164320.0 -324.0 -0.02 166760.0 399.0 0.03 0.0054 0.1453 3622504 Ald3.1-H_000025 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCCC(=O)NO)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B04 compound treatment 224960.0 60300.0 4.11 230240.0 63900.0 4.75 6.2695 0.9974 3622506 Ald3.1-H_000026 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3ccc(OCCCCCCC(=O)NO)c(OC)c3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B05 compound treatment 177280.0 12600.0 0.86 180280.0 13900.0 1.04 1.3417 0.9958 3622508 Ald3.1-H_000027 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCCCC(=O)NO)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B06 compound treatment 223480.0 58800.0 4.01 219280.0 52900.0 3.94 5.6214 1.0 3622510 Ald3.1-H_000028 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3ccc(OCCCCCCC(=O)NO)c4ccccc34)c2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B07 compound treatment 222600.0 58000.0 3.95 227720.0 61400.0 4.57 6.0231 0.9974 3622512 Ald3.1-H_000029 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3cccc(c3)C(=O)NO)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B08 compound treatment 179720.0 15100.0 1.03 180000.0 13600.0 1.02 1.4446 1.0 3622514 Ald3.1-H_000030 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCC(=O)Nc3ccccc3O)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B09 compound treatment 236000.0 71400.0 4.86 229280.0 62900.0 4.68 6.7512 0.9998 3622516 Ald3.1-H_000031 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3ccc(cc3)C(=O)NO)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B10 compound treatment 189000.0 24400.0 1.66 186000.0 19600.0 1.46 2.2077 0.998 3622518 Ald3.1-H_000032 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCCC(=O)Nc3ccccc3O)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B11 compound treatment 215000.0 50400.0 3.43 213360.0 47000.0 3.5 4.901 1.0 3622520 Ald3.1-H_000033 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3cccc(OCC(=O)NO)c3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B12 compound treatment 201480.0 36800.0 2.51 195520.0 29200.0 2.17 3.3104 0.9974 3622522 Ald3.1-H_000034 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCCCC(=O)Nc3ccccc3O)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B13 mock treatment 160120.0 -4520.0 -0.31 156800.0 -9560.0 -0.71 -0.7213 -0.93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B14 mock treatment 148560.0 -16100.0 -1.1 156440.0 -9920.0 -0.74 -1.2975 -0.9815 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B15 compound treatment 219440.0 54800.0 3.74 225360.0 59000.0 4.39 5.7466 0.9968 3622524 Ald3.1-H_000035 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3cccc(OCCCCCC(=O)NO)c3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B16 compound treatment 154280.0 -10400.0 -0.71 158120.0 -8240.0 -0.61 -0.9333 -0.9975 3622526 Ald3.1-H_000036 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCCCC(=O)O)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B17 compound treatment 239400.0 74800.0 5.1 238960.0 72600.0 5.4 7.4246 0.9996 3622528 Ald3.1-H_000037 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3ccc(OCCCCCC(=O)NO)cc3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B18 compound treatment 155640.0 -9000.0 -0.61 160600.0 -5760.0 -0.43 -0.7373 -0.9846 3622530 Ald3.1-H_000038 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)C)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B19 compound treatment 234960.0 70300.0 4.79 234040.0 67700.0 5.04 6.9516 0.9997 3622532 Ald3.1-H_000039 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3cccc(OCCCCCCC(=O)NO)c3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B20 compound treatment 154000.0 -10600.0 -0.73 158400.0 -7960.0 -0.59 -0.9321 -0.9949 3622534 Ald3.1-H_000040 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(C=O)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B21 compound treatment 202840.0 38200.0 2.6 182120.0 15800.0 1.17 2.6707 0.9351 3622536 Ald3.1-H_000041 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)c3ccc(OCC(=O)NO)cc3)c2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B22 compound treatment 151720.0 -12900.0 -0.88 153760.0 -12600.0 -0.94 -1.2862 -0.9995 3622538 Ald3.1-H_000042 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2cccc(\C=N\NC(=O)CCCCCC(=O)O)c2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B23 compound treatment 170760.0 6120.0 0.42 165800.0 -561.0 -0.04 0.2653 0.6331 3622540 Ald3.1-H_000043 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 B24 compound treatment 165360.0 716.0 0.05 166840.0 479.0 0.04 0.0597 0.988 3622542 Ald3.1-H_000044 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C01 compound treatment 166080.0 1440.0 0.1 164840.0 -1520.0 -0.11 -0.0108 -0.0723 3622544 Ald3.1-H_000045 ONC(=O)CCCCC(=O)N/N=C/c1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C02 compound treatment 155720.0 -8920.0 -0.61 226360.0 60000.0 4.47 2.7274 0.6052 3622546 Ald3.1-H_000046 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C03 compound treatment 172520.0 7880.0 0.54 173720.0 7360.0 0.55 0.767 1.0 3622548 Ald3.1-H_000047 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C04 compound treatment 209480.0 44800.0 3.06 219240.0 52900.0 3.94 4.9444 0.9922 3622550 Ald3.1-H_000048 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C05 compound treatment 171280.0 6640.0 0.45 175640.0 9280.0 0.69 0.8082 0.979 3622552 Ald3.1-H_000049 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C06 compound treatment 215960.0 51300.0 3.5 212280.0 45900.0 3.42 4.8905 0.9999 3622554 Ald3.1-H_000050 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C07 compound treatment 234320.0 69700.0 4.75 225920.0 59600.0 4.43 6.4934 0.9994 3622556 Ald3.1-H_000051 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C08 compound treatment 185920.0 21300.0 1.45 181120.0 14800.0 1.1 1.8024 0.9906 3622558 Ald3.1-H_000052 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C09 compound treatment 214320.0 49700.0 3.39 217880.0 51500.0 3.83 5.1061 0.9981 3622560 Ald3.1-H_000053 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C10 compound treatment 180120.0 15500.0 1.06 177760.0 11400.0 0.85 1.346 0.9942 3622562 Ald3.1-H_000054 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C11 mock treatment 159920.0 -4720.0 -0.32 162280.0 -4080.0 -0.3 -0.4425 -0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C12 mock treatment 163720.0 -924.0 -0.06 165280.0 -1080.0 -0.08 -0.1014 -0.9926 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C13 compound treatment 201520.0 36900.0 2.51 194200.0 27800.0 2.07 3.2428 0.9954 3622564 Ald3.1-H_000055 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C14 compound treatment 154600.0 -10000.0 -0.68 165400.0 -961.0 -0.07 -0.5348 -0.7768 3622566 Ald3.1-H_000056 OC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C15 mock treatment 158240.0 -6400.0 -0.44 157400.0 -8960.0 -0.67 -0.7803 -0.9789 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C16 mock treatment 151560.0 -13100.0 -0.89 158040.0 -8320.0 -0.62 -1.0687 -0.9841 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C17 compound treatment 233360.0 68700.0 4.68 253160.0 86800.0 6.46 7.8807 0.9875 3622568 Ald3.1-H_000057 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C18 compound treatment 160680.0 -3960.0 -0.27 162680.0 -3680.0 -0.27 -0.3848 -1.0 3622570 Ald3.1-H_000058 CC(=O)N/N=C/c1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C19 compound treatment 233320.0 68700.0 4.68 241520.0 75200.0 5.59 7.2662 0.9961 3622572 Ald3.1-H_000059 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C20 compound treatment 156440.0 -8200.0 -0.56 156280.0 -10100.0 -0.75 -0.926 -0.9895 3622574 Ald3.1-H_000060 O=Cc1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C21 compound treatment 218600.0 54000.0 3.68 221720.0 55400.0 4.12 5.5145 0.9984 3622576 Ald3.1-H_000061 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H](COC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C22 compound treatment 157000.0 -7640.0 -0.52 156280.0 -10100.0 -0.75 -0.8991 -0.9841 3622578 Ald3.1-H_000062 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2[C@H](COC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C23 compound treatment 146120.0 -18500.0 -1.26 155120.0 -11200.0 -0.84 -1.4846 -0.98 3622580 Ald3.1-H_000063 ONC(=O)CCCCC(=O)N/N=C/c1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 C24 compound treatment 206880.0 42200.0 2.88 231680.0 65300.0 4.86 5.4737 0.9688 3622581 Ald3.1-H_000064 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D01 compound treatment 154680.0 -9960.0 -0.68 162840.0 -3520.0 -0.26 -0.6657 -0.9142 3622582 Ald3.1-H_000065 ONC(=O)CCCCC(=O)N/N=C/c1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D02 compound treatment 212440.0 47800.0 3.26 211080.0 44700.0 3.33 4.6576 0.9999 3622584 Ald3.1-H_000066 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D03 compound treatment 168600.0 3960.0 0.27 170440.0 4080.0 0.3 0.4054 0.9983 3622586 Ald3.1-H_000067 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D04 compound treatment 213560.0 48900.0 3.33 212400.0 46000.0 3.43 4.7811 0.9999 3622588 Ald3.1-H_000068 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D05 compound treatment 166520.0 1880.0 0.13 173160.0 6800.0 0.51 0.4483 0.8588 3622590 Ald3.1-H_000069 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D06 compound treatment 232280.0 67600.0 4.61 246400.0 80000.0 5.96 7.4729 0.992 3622592 Ald3.1-H_000070 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D07 compound treatment 179600.0 15000.0 1.02 194560.0 28200.0 2.1 2.205 0.945 3622594 Ald3.1-H_000071 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D08 compound treatment 168560.0 3920.0 0.27 177600.0 11200.0 0.84 0.7803 0.8886 3622596 Ald3.1-H_000072 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D09 compound treatment 195360.0 30700.0 2.09 197440.0 31100.0 2.31 3.1164 0.9988 3622598 Ald3.1-H_000073 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D10 compound treatment 181080.0 16400.0 1.12 180640.0 14300.0 1.06 1.5438 0.9996 3622600 Ald3.1-H_000074 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D11 mock treatment 160680.0 -3960.0 -0.27 156760.0 -9600.0 -0.71 -0.6964 -0.9115 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D12 mock treatment 157280.0 -7360.0 -0.5 154040.0 -12300.0 -0.92 -1.0034 -0.9598 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D13 compound treatment 178160.0 13500.0 0.92 183360.0 17000.0 1.27 1.5462 0.9879 3622602 Ald3.1-H_000075 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D14 compound treatment 157560.0 -7080.0 -0.48 164560.0 -1800.0 -0.13 -0.4363 -0.8705 3622604 Ald3.1-H_000076 OC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D15 mock treatment 151520.0 -13100.0 -0.89 159560.0 -6800.0 -0.51 -0.9906 -0.9636 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D16 mock treatment 152720.0 -11900.0 -0.81 160040.0 -6320.0 -0.47 -0.9075 -0.9662 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D17 compound treatment 218760.0 54100.0 3.69 225960.0 59600.0 4.44 5.7454 0.9958 3622606 Ald3.1-H_000077 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D18 compound treatment 159920.0 -4720.0 -0.32 164680.0 -1680.0 -0.13 -0.3162 -0.9152 3622608 Ald3.1-H_000078 CC(=O)N/N=C/c1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D19 compound treatment 231880.0 67200.0 4.58 242120.0 75800.0 5.64 7.2284 0.9947 3622610 Ald3.1-H_000079 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D20 compound treatment 157880.0 -6760.0 -0.46 165400.0 -961.0 -0.07 -0.3767 -0.8072 3622612 Ald3.1-H_000080 O=Cc1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D21 compound treatment 190680.0 26000.0 1.78 202920.0 36600.0 2.72 3.1792 0.9786 3622614 Ald3.1-H_000081 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D22 compound treatment 156960.0 -7680.0 -0.52 154920.0 -11400.0 -0.85 -0.9726 -0.9728 3622616 Ald3.1-H_000082 OC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D23 compound treatment 164840.0 196.0 0.01 171960.0 5600.0 0.42 0.3041 0.7294 3622618 Ald3.1-H_000083 ONC(=O)CCCCC(=O)N/N=C/c1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 D24 compound treatment 196080.0 31400.0 2.14 220840.0 54500.0 4.05 4.3826 0.9556 3622620 Ald3.1-H_000084 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E01 mock treatment 160720.0 -3920.0 -0.27 160920.0 -5440.0 -0.4 -0.4755 -0.9797 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E02 mock treatment 160680.0 -3960.0 -0.27 160280.0 -6080.0 -0.45 -0.5111 -0.9696 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E03 compound treatment 184120.0 19500.0 1.33 180880.0 14500.0 1.08 1.703 0.9948 3622622 Ald3.1-H_000085 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E04 compound treatment 245960.0 81300.0 5.54 239600.0 73200.0 5.45 7.7745 1.0 3622623 Ald3.1-H_000086 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E05 compound treatment 189360.0 24700.0 1.69 191200.0 24800.0 1.85 2.4987 0.9989 3622624 Ald3.1-H_000087 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E06 compound treatment 227920.0 63300.0 4.31 229200.0 62800.0 4.68 6.3575 0.9992 3622625 Ald3.1-H_000088 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E07 compound treatment 231040.0 66400.0 4.53 223920.0 57600.0 4.28 6.23 0.9996 3622626 Ald3.1-H_000089 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E08 compound treatment 184360.0 19700.0 1.34 185680.0 19300.0 1.44 1.9672 0.9994 3622627 Ald3.1-H_000090 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E09 mock treatment 173000.0 8360.0 0.57 169880.0 3520.0 0.26 0.588 0.9378 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E10 mock treatment 163800.0 -844.0 -0.06 169040.0 2680.0 0.2 0.1003 0.4834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E11 compound treatment 223400.0 58800.0 4.01 217400.0 51000.0 3.8 5.5186 0.9996 3622628 Ald3.1-H_000091 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E12 compound treatment 198160.0 33500.0 2.29 196360.0 30000.0 2.23 3.1945 0.9999 3622629 Ald3.1-H_000092 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E13 compound treatment 236640.0 72000.0 4.91 163240.0 -3120.0 -0.23 3.3065 0.6729 3622630 Ald3.1-H_000093 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E14 compound treatment 169440.0 4800.0 0.33 169680.0 3320.0 0.25 0.4059 0.9904 3622631 Ald3.1-H_000094 OC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E15 compound treatment 230560.0 65900.0 4.49 237080.0 70700.0 5.26 6.8995 0.9969 3622632 Ald3.1-H_000095 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E16 compound treatment 175600.0 11000.0 0.75 169680.0 3320.0 0.25 0.7028 0.8934 3622633 Ald3.1-H_000096 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E17 mock treatment 166880.0 2240.0 0.15 169520.0 3160.0 0.24 0.274 0.978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E18 mock treatment 166800.0 2160.0 0.15 165920.0 -441.0 -0.03 0.0807 0.5359 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E19 compound treatment 231080.0 66400.0 4.53 234480.0 68100.0 5.07 6.7877 0.9984 3622634 Ald3.1-H_000097 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E20 compound treatment 164560.0 -83.8 -0.01 168840.0 2480.0 0.18 0.1264 0.6849 3622635 Ald3.1-H_000098 O=Cc1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E21 compound treatment 273560.0 109000.0 7.43 268240.0 102000.0 7.58 10.6123 0.9999 3622636 Ald3.1-H_000099 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E22 compound treatment 194080.0 29400.0 2.01 201200.0 34800.0 2.59 3.2526 0.992 3622637 Ald3.1-H_000100 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E23 compound treatment 235360.0 70700.0 4.82 246200.0 79800.0 5.94 7.6108 0.9946 3622638 Ald3.1-H_000101 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 E24 compound treatment 154440.0 -10200.0 -0.7 160200.0 -6160.0 -0.46 -0.8162 -0.9795 3622639 Ald3.1-H_000102 CC(=O)N/N=C/c1ccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F01 mock treatment 158920.0 -5720.0 -0.39 158760.0 -7600.0 -0.57 -0.676 -0.9836 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F02 mock treatment 167080.0 2440.0 0.17 165880.0 -481.0 -0.04 0.0921 0.5421 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F03 compound treatment 177560.0 12900.0 0.88 179480.0 13100.0 0.98 1.3131 0.9987 3622640 Ald3.1-H_000103 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F04 compound treatment 229080.0 64400.0 4.39 228520.0 62200.0 4.63 6.3776 0.9997 3622642 Ald3.1-H_000104 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F05 compound treatment 189520.0 24900.0 1.7 183440.0 17100.0 1.27 2.0981 0.9899 3622644 Ald3.1-H_000105 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F06 compound treatment 250440.0 85800.0 5.85 254440.0 88100.0 6.56 8.7715 0.9984 3622646 Ald3.1-H_000106 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F07 compound treatment 208840.0 44200.0 3.01 201680.0 35300.0 2.63 3.9894 0.9977 3622648 Ald3.1-H_000107 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F08 compound treatment 179840.0 15200.0 1.04 183640.0 17300.0 1.29 1.6419 0.9943 3622650 Ald3.1-H_000108 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F09 mock treatment 164280.0 -364.0 -0.02 168680.0 2320.0 0.17 0.1045 0.5993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F10 mock treatment 164920.0 276.0 0.02 165800.0 -561.0 -0.04 -0.0162 -0.3541 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F11 compound treatment 195880.0 31200.0 2.13 192640.0 26300.0 1.96 2.8888 0.9991 3622652 Ald3.1-H_000109 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F12 compound treatment 195280.0 30600.0 2.09 190720.0 24400.0 1.81 2.7589 0.9975 3622654 Ald3.1-H_000110 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F13 compound treatment 195640.0 31000.0 2.11 204520.0 38200.0 2.84 3.5025 0.9894 3622656 Ald3.1-H_000111 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F14 compound treatment 168520.0 3880.0 0.26 171160.0 4800.0 0.36 0.4394 0.989 3622658 Ald3.1-H_000112 OC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F15 compound treatment 226280.0 61600.0 4.2 228400.0 62000.0 4.62 6.2363 0.9989 3622660 Ald3.1-H_000113 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F16 compound treatment 170840.0 6200.0 0.42 168320.0 1960.0 0.15 0.4018 0.8991 3622662 Ald3.1-H_000114 OC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F17 mock treatment 165640.0 996.0 0.07 164440.0 -1920.0 -0.14 -0.0531 -0.3354 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F18 mock treatment 161800.0 -2840.0 -0.19 170520.0 4160.0 0.31 0.0818 0.2239 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F19 compound treatment 248120.0 83500.0 5.69 249480.0 83100.0 6.19 8.3986 0.9991 3622664 Ald3.1-H_000115 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F20 compound treatment 162480.0 -2160.0 -0.15 166600.0 239.0 0.02 -0.0917 -0.6175 3622666 Ald3.1-H_000116 O=Cc1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F21 compound treatment 207480.0 42800.0 2.92 208600.0 42200.0 3.14 4.288 0.9993 3622668 Ald3.1-H_000117 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F22 compound treatment 194480.0 29800.0 2.03 188880.0 22500.0 1.68 2.6235 0.9954 3622670 Ald3.1-H_000118 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F23 compound treatment 232880.0 68200.0 4.65 245920.0 79600.0 5.92 7.4766 0.9929 3622672 Ald3.1-H_000119 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 F24 compound treatment 152600.0 -12000.0 -0.82 162080.0 -4280.0 -0.32 -0.8059 -0.915 3622674 Ald3.1-H_000120 CC(=O)N/N=C/c1cccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G01 compound treatment 177640.0 13000.0 0.89 177040.0 10700.0 0.79 1.1885 0.9985 3622676 Ald3.1-H_000121 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G02 compound treatment 242080.0 77400.0 5.28 234960.0 68600.0 5.11 7.3433 0.9999 3622678 Ald3.1-H_000122 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3ccc(OCCCCCCC(=O)NO)cc3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G03 mock treatment 171560.0 6920.0 0.47 172520.0 6160.0 0.46 0.6575 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G04 mock treatment 175120.0 10500.0 0.71 173080.0 6720.0 0.5 0.8586 0.9848 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G05 compound treatment 199080.0 34400.0 2.35 194400.0 28000.0 2.09 3.1357 0.9983 3622680 Ald3.1-H_000123 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G06 compound treatment 257720.0 93100.0 6.35 265280.0 98900.0 7.36 9.6929 0.9973 3622682 Ald3.1-H_000124 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3ccc(OCCCCCCC(=O)NO)c4ccccc34)cc2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G07 compound treatment 243680.0 79000.0 5.39 242920.0 76600.0 5.7 7.8393 0.9996 3622684 Ald3.1-H_000125 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3cccc(c3)C(=O)NO)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G08 compound treatment 210240.0 45600.0 3.11 202360.0 36000.0 2.68 4.0926 0.9973 3622686 Ald3.1-H_000126 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCC(=O)Nc3ccccc3O)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G09 compound treatment 247920.0 83300.0 5.68 257000.0 90600.0 6.75 8.7847 0.9963 3622688 Ald3.1-H_000127 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3ccc(cc3)C(=O)NO)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G10 compound treatment 197240.0 32600.0 2.22 212640.0 46300.0 3.44 4.007 0.9775 3622690 Ald3.1-H_000128 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCCC(=O)Nc3ccccc3O)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G11 compound treatment 244560.0 79900.0 5.45 241400.0 75000.0 5.58 7.8017 0.9999 3622692 Ald3.1-H_000129 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3cccc(OCC(=O)NO)c3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G12 compound treatment 190920.0 26300.0 1.79 200120.0 33800.0 2.51 3.0434 0.9863 3622694 Ald3.1-H_000130 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCCCC(=O)Nc3ccccc3O)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G13 compound treatment 241520.0 76900.0 5.24 243520.0 77200.0 5.74 7.7668 0.999 3622696 Ald3.1-H_000131 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3ccc(OCC(=O)NO)cc3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G14 compound treatment 174960.0 10300.0 0.7 179680.0 13300.0 0.99 1.1983 0.9859 3622698 Ald3.1-H_000132 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCCC(=O)O)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G15 compound treatment 220520.0 55900.0 3.81 225360.0 59000.0 4.39 5.7987 0.9975 3622700 Ald3.1-H_000133 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3cccc(OCCCCCC(=O)NO)c3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G16 compound treatment 181160.0 16500.0 1.13 179200.0 12800.0 0.96 1.4719 0.9967 3622702 Ald3.1-H_000134 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCCCC(=O)O)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G17 compound treatment 273680.0 109000.0 7.43 270920.0 105000.0 7.78 10.7591 0.9997 3622704 Ald3.1-H_000135 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3ccc(OCCCCCC(=O)NO)cc3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G18 compound treatment 171080.0 6440.0 0.44 176840.0 10500.0 0.78 0.8618 0.963 3622706 Ald3.1-H_000136 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)C)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G19 mock treatment 168040.0 3400.0 0.23 170880.0 4520.0 0.34 0.4015 0.9834 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G20 mock treatment 164360.0 -284.0 -0.02 166760.0 399.0 0.03 0.0073 0.2061 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G21 compound treatment 180440.0 15800.0 1.08 187280.0 20900.0 1.56 1.8624 0.9838 3622708 Ald3.1-H_000137 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G22 compound treatment 253760.0 89100.0 6.08 251040.0 84700.0 6.3 8.7526 0.9998 3622710 Ald3.1-H_000138 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3ccc(OCCCCCCC(=O)NO)c(OC)c3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G23 compound treatment 224200.0 59600.0 4.06 234440.0 68100.0 5.07 6.4539 0.994 3622712 Ald3.1-H_000139 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(\C=N\NC(=O)c3cccc(OCCCCCCC(=O)NO)c3)cc2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 G24 compound treatment 161680.0 -2960.0 -0.2 166920.0 559.0 0.04 -0.1135 -0.5501 3622714 Ald3.1-H_000140 COC[C@H]1[C@@H](OC(=O)CC/C=C/CCC(=O)N1Cc2ccc(C=O)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H01 compound treatment 173920.0 9280.0 0.63 174840.0 8480.0 0.63 0.8934 1.0 3214834 Ald3.1-H_000141 ONC(=O)CCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H02 compound treatment 197360.0 32700.0 2.23 195240.0 28900.0 2.15 3.097 0.9998 3622716 Ald3.1-H_000142 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H03 mock treatment 168840.0 4200.0 0.29 167480.0 1120.0 0.08 0.2612 0.8765 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H04 mock treatment 167720.0 3080.0 0.21 165360.0 -1000.0 -0.07 0.0956 0.4295 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H05 compound treatment 175760.0 11100.0 0.76 178000.0 11600.0 0.87 1.1484 0.9978 3213068 Ald3.1-H_000143 ONC(=O)CCCCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H06 compound treatment 240280.0 75600.0 5.16 239160.0 72800.0 5.42 7.4775 0.9997 3622718 Ald3.1-H_000144 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccccc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H07 compound treatment 180720.0 16100.0 1.1 182520.0 16200.0 1.2 1.6254 0.9989 3553005 Ald3.1-H_000145 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H08 compound treatment 179840.0 15200.0 1.04 181600.0 15200.0 1.13 1.5346 0.999 3622720 Ald3.1-H_000146 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H09 compound treatment 176600.0 12000.0 0.82 184800.0 18400.0 1.37 1.5468 0.9691 3553670 Ald3.1-H_000147 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H10 compound treatment 180480.0 15800.0 1.08 186320.0 20000.0 1.49 1.8138 0.9877 3214226 Ald3.1-H_000148 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H11 compound treatment 180840.0 16200.0 1.1 183560.0 17200.0 1.28 1.6859 0.9973 3622722 Ald3.1-H_000149 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H12 compound treatment 176640.0 12000.0 0.82 184880.0 18500.0 1.38 1.5529 0.9689 3213070 Ald3.1-H_000150 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H13 compound treatment 189840.0 25200.0 1.72 184960.0 18600.0 1.38 2.1935 0.9943 3622724 Ald3.1-H_000151 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H14 compound treatment 175320.0 10700.0 0.73 177560.0 11200.0 0.83 1.104 0.9977 3213680 Ald3.1-H_000152 OC(=O)CCCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H15 compound treatment 188880.0 24200.0 1.65 199120.0 32800.0 2.44 2.8924 0.982 3622726 Ald3.1-H_000153 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H16 compound treatment 170960.0 6320.0 0.43 170960.0 4600.0 0.34 0.5465 0.9935 3213678 Ald3.1-H_000154 OC(=O)CCCCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H17 compound treatment 195720.0 31100.0 2.12 200960.0 34600.0 2.58 3.319 0.9953 3622728 Ald3.1-H_000155 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H18 compound treatment 167440.0 2800.0 0.19 174760.0 8400.0 0.63 0.5768 0.8826 3622730 Ald3.1-H_000156 CC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H19 mock treatment 162000.0 -2640.0 -0.18 171720.0 5360.0 0.4 0.1546 0.3532 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H20 mock treatment 164240.0 -404.0 -0.03 166840.0 479.0 0.04 0.0057 0.1272 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H21 compound treatment 171200.0 6560.0 0.45 173720.0 7360.0 0.55 0.7033 0.9949 3214224 Ald3.1-H_000157 ONC(=O)CCCCCC(=O)N/N=C/c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H22 compound treatment 180960.0 16300.0 1.11 185720.0 19400.0 1.44 1.8054 0.9918 3622731 Ald3.1-H_000158 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H23 compound treatment 185040.0 20400.0 1.39 193520.0 27200.0 2.02 2.4126 0.9833 3622733 Ald3.1-H_000159 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 H24 compound treatment 155200.0 -9440.0 -0.64 156360.0 -10000.0 -0.74 -0.9816 -0.9974 1009816 Ald3.1-H_000160 O=Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I01 compound treatment 174600.0 9960.0 0.68 174640.0 8280.0 0.62 0.9157 0.9988 3622735 Ald3.1-H_000161 ONC(=O)CCCCC(=O)N/N=C/c1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I02 compound treatment 246480.0 81800.0 5.58 242040.0 75700.0 5.63 7.928 1.0 3622737 Ald3.1-H_000162 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I03 compound treatment 180000.0 15400.0 1.05 179040.0 12700.0 0.94 1.4075 0.9987 3622739 Ald3.1-H_000163 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I04 compound treatment 235320.0 70700.0 4.82 223800.0 57400.0 4.27 6.4301 0.9982 3622741 Ald3.1-H_000164 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I05 mock treatment 166640.0 2000.0 0.14 170720.0 4360.0 0.32 0.3256 0.9256 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I06 mock treatment 169040.0 4400.0 0.3 173160.0 6800.0 0.51 0.5697 0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I07 compound treatment 200480.0 35800.0 2.44 210680.0 44300.0 3.3 4.06 0.9891 3622743 Ald3.1-H_000165 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I08 compound treatment 180440.0 15800.0 1.08 180240.0 13900.0 1.03 1.4919 0.9998 3622745 Ald3.1-H_000166 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I09 compound treatment 210440.0 45800.0 3.12 211200.0 44800.0 3.34 4.5675 0.9994 3622747 Ald3.1-H_000167 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I10 compound treatment 188320.0 23700.0 1.61 197080.0 30700.0 2.29 2.758 0.9855 3622749 Ald3.1-H_000168 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I11 compound treatment 188080.0 23400.0 1.6 191000.0 24600.0 1.83 2.4265 0.9976 3622751 Ald3.1-H_000169 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I12 compound treatment 202080.0 37400.0 2.55 205280.0 38900.0 2.9 3.8529 0.998 3622753 Ald3.1-H_000170 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I13 compound treatment 203440.0 38800.0 2.65 203720.0 37400.0 2.78 3.8364 0.9997 3622755 Ald3.1-H_000171 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I14 compound treatment 173440.0 8800.0 0.6 175440.0 9080.0 0.68 0.9018 0.9982 3622757 Ald3.1-H_000172 OC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I15 compound treatment 223000.0 58400.0 3.98 219400.0 53000.0 3.95 5.6046 1.0 3622759 Ald3.1-H_000173 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I16 compound treatment 171000.0 6360.0 0.43 176000.0 9640.0 0.72 0.8137 0.9709 3622761 Ald3.1-H_000174 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I17 compound treatment 256200.0 91600.0 6.24 255720.0 89400.0 6.65 9.1165 0.9995 3622763 Ald3.1-H_000175 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I18 compound treatment 170880.0 6240.0 0.43 165960.0 -401.0 -0.03 0.2795 0.6558 3622765 Ald3.1-H_000176 CC(=O)N/N=C/c1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I19 compound treatment 247640.0 83000.0 5.66 259800.0 93400.0 6.95 8.9186 0.9948 3622767 Ald3.1-H_000177 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I20 compound treatment 168960.0 4320.0 0.29 169920.0 3560.0 0.26 0.3954 0.9986 3622769 Ald3.1-H_000178 O=Cc1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I21 mock treatment 156240.0 -8400.0 -0.57 157680.0 -8680.0 -0.65 -0.862 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I22 mock treatment 161640.0 -3000.0 -0.2 161720.0 -4640.0 -0.35 -0.3891 -0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I23 compound treatment 170560.0 5920.0 0.4 173680.0 7320.0 0.54 0.6704 0.9891 3622771 Ald3.1-H_000179 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2[C@@H]3CCCC[C@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 I24 compound treatment 209520.0 44900.0 3.06 218800.0 52400.0 3.9 4.9231 0.9927 3622773 Ald3.1-H_000180 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(CN3[C@@H]4CCCC[C@H]4OC(=O)CC/C=C/CCC3=O)cc2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J01 compound treatment 223680.0 59000.0 4.02 228160.0 61800.0 4.6 6.0984 0.9978 3215196 Ald3.1-H_000181 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J02 compound treatment 232840.0 68200.0 4.65 235120.0 68800.0 5.12 6.9062 0.9989 3622775 Ald3.1-H_000182 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J03 compound treatment 238320.0 73700.0 5.02 230840.0 64500.0 4.8 6.9452 0.9997 3214586 Ald3.1-H_000183 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J04 compound treatment 210400.0 45800.0 3.12 214880.0 48500.0 3.61 4.7593 0.9973 3622777 Ald3.1-H_000184 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J05 mock treatment 181760.0 17100.0 1.17 176720.0 10400.0 0.77 1.3703 0.9798 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J06 mock treatment 185800.0 21200.0 1.44 191360.0 25000.0 1.86 2.3355 0.9921 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J07 compound treatment 286320.0 122000.0 8.3 316320.0 150000.0 11.16 13.7578 0.9893 3553510 Ald3.1-H_000185 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J08 compound treatment 200120.0 35500.0 2.42 210680.0 44300.0 3.3 4.0426 0.9884 3622779 Ald3.1-H_000186 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J09 compound treatment 295240.0 131000.0 8.9 286880.0 121000.0 8.97 12.6385 1.0 3554094 Ald3.1-H_000187 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J10 compound treatment 197320.0 32700.0 2.23 197760.0 31400.0 2.34 3.2277 0.9997 3214584 Ald3.1-H_000188 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J11 compound treatment 254760.0 90100.0 6.14 247440.0 81100.0 6.03 8.6113 1.0 3622781 Ald3.1-H_000189 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J12 compound treatment 204520.0 39900.0 2.72 204760.0 38400.0 2.86 3.9432 0.9997 3213428 Ald3.1-H_000190 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J13 compound treatment 290360.0 126000.0 8.57 275320.0 109000.0 8.11 11.7948 0.9996 3622783 Ald3.1-H_000191 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J14 compound treatment 192280.0 27600.0 1.88 194760.0 28400.0 2.11 2.8269 0.9984 3214038 Ald3.1-H_000192 OC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J15 compound treatment 235760.0 71100.0 4.85 228520.0 62200.0 4.63 6.6997 0.9997 3622785 Ald3.1-H_000193 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J16 compound treatment 210680.0 46000.0 3.14 210520.0 44200.0 3.29 4.5433 0.9997 3214040 Ald3.1-H_000194 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J17 compound treatment 268320.0 104000.0 7.07 268800.0 102000.0 7.62 10.3892 0.9993 3622787 Ald3.1-H_000195 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J18 compound treatment 193240.0 28600.0 1.95 191280.0 24900.0 1.85 2.69 0.9997 3622789 Ald3.1-H_000196 CC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J19 compound treatment 231560.0 66900.0 4.56 216000.0 49600.0 3.69 5.8383 0.9945 3622791 Ald3.1-H_000197 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J20 compound treatment 168160.0 3520.0 0.24 165760.0 -601.0 -0.04 0.1379 0.5653 1073512 Ald3.1-H_000198 O=Cc1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J21 mock treatment 156240.0 -8400.0 -0.57 162000.0 -4360.0 -0.32 -0.6347 -0.9638 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J22 mock treatment 157640.0 -7000.0 -0.48 161920.0 -4440.0 -0.33 -0.5714 -0.9839 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J23 compound treatment 219600.0 55000.0 3.75 218720.0 52400.0 3.9 5.4049 0.9998 3213430 Ald3.1-H_000199 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)N(c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 J24 compound treatment 172680.0 8040.0 0.55 176280.0 9920.0 0.74 0.9094 0.9892 3622793 Ald3.1-H_000200 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(cc2)N(c3ccccc3)c4ccccc4)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K01 compound treatment 166960.0 2320.0 0.16 161560.0 -4800.0 -0.36 -0.141 -0.361 3622795 Ald3.1-H_000201 ONC(=O)CCCCC(=O)N/N=C/c1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K02 compound treatment 261240.0 96600.0 6.59 258920.0 92600.0 6.89 9.5279 0.9997 3622797 Ald3.1-H_000202 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K03 compound treatment 133280.0 -31400.0 -2.14 137840.0 -28500.0 -2.12 -3.013 -1.0 3622799 Ald3.1-H_000203 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K04 compound treatment 246120.0 81500.0 5.55 244520.0 78200.0 5.82 8.0412 0.9997 3622801 Ald3.1-H_000204 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K05 compound treatment 183360.0 18700.0 1.28 180120.0 13800.0 1.02 1.6264 0.9941 3622803 Ald3.1-H_000205 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K06 compound treatment 270080.0 105000.0 7.19 260520.0 94200.0 7.01 10.0383 0.9999 3622805 Ald3.1-H_000206 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K07 mock treatment 169120.0 4480.0 0.31 175960.0 9600.0 0.71 0.7209 0.928 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K08 mock treatment 166280.0 1640.0 0.11 171760.0 5400.0 0.4 0.363 0.8705 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K09 compound treatment 203520.0 38900.0 2.65 203720.0 37400.0 2.78 3.8403 0.9997 3622807 Ald3.1-H_000207 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K10 compound treatment 196000.0 31400.0 2.14 210880.0 44500.0 3.31 3.8546 0.9775 3622809 Ald3.1-H_000208 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K11 compound treatment 192680.0 28000.0 1.91 199040.0 32700.0 2.43 3.0714 0.9929 3622811 Ald3.1-H_000209 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K12 compound treatment 195480.0 30800.0 2.1 196760.0 30400.0 2.26 3.0864 0.9993 3622813 Ald3.1-H_000210 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K13 compound treatment 198120.0 33500.0 2.28 198600.0 32200.0 2.4 3.3105 0.9997 3622815 Ald3.1-H_000211 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K14 compound treatment 175360.0 10700.0 0.73 170760.0 4400.0 0.33 0.7481 0.9344 3622817 Ald3.1-H_000212 OC(=O)CCCCCC(=O)N/N=C/c1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K15 mock treatment 167160.0 2520.0 0.17 171400.0 5040.0 0.38 0.3865 0.9372 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K16 mock treatment 165520.0 876.0 0.06 168960.0 2600.0 0.19 0.179 0.8843 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K17 compound treatment 249600.0 85000.0 5.79 257040.0 90700.0 6.75 8.8678 0.9971 3622819 Ald3.1-H_000213 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K18 compound treatment 170560.0 5920.0 0.4 170960.0 4600.0 0.34 0.5272 0.9967 3622821 Ald3.1-H_000214 CC(=O)N/N=C/c1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K19 compound treatment 245640.0 81000.0 5.52 246480.0 80100.0 5.96 8.1212 0.9993 3622823 Ald3.1-H_000215 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K20 compound treatment 161200.0 -3440.0 -0.23 169720.0 3360.0 0.25 0.0107 0.0313 3622825 Ald3.1-H_000216 O=Cc1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K21 compound treatment 192320.0 27700.0 1.89 197440.0 31100.0 2.31 2.9698 0.9949 3622827 Ald3.1-H_000217 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K22 compound treatment 174160.0 9520.0 0.65 172840.0 6480.0 0.48 0.7997 0.9893 3622829 Ald3.1-H_000218 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K23 mock treatment 157360.0 -7280.0 -0.5 160200.0 -6160.0 -0.46 -0.6754 -0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 K24 mock treatment 155480.0 -9160.0 -0.62 153480.0 -12900.0 -0.96 -1.1197 -0.9785 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L01 compound treatment 174160.0 9520.0 0.65 174240.0 7880.0 0.59 0.8734 0.9987 3622831 Ald3.1-H_000219 ONC(=O)CCCCC(=O)N/N=C/c1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L02 compound treatment 230440.0 65800.0 4.49 233840.0 67500.0 5.02 6.7232 0.9984 3622833 Ald3.1-H_000220 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L03 compound treatment 178640.0 14000.0 0.95 179000.0 12600.0 0.94 1.3399 1.0 3622835 Ald3.1-H_000221 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L04 compound treatment 236720.0 72100.0 4.91 236720.0 70400.0 5.24 7.1775 0.9995 3622837 Ald3.1-H_000222 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L05 compound treatment 185600.0 21000.0 1.43 183320.0 17000.0 1.26 1.9028 0.9981 3622839 Ald3.1-H_000223 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L06 compound treatment 252560.0 87900.0 5.99 254280.0 87900.0 6.54 8.8653 0.999 3622841 Ald3.1-H_000224 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(OCC#C)cc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L07 mock treatment 171920.0 7280.0 0.5 175120.0 8760.0 0.65 0.8117 0.9909 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L08 mock treatment 174680.0 10000.0 0.68 173800.0 7440.0 0.55 0.8753 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L09 compound treatment 214600.0 50000.0 3.41 229320.0 63000.0 4.69 5.7217 0.9877 3554221 Ald3.1-H_000225 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L10 compound treatment 192560.0 27900.0 1.9 191760.0 25400.0 1.89 2.6825 1.0 3622843 Ald3.1-H_000226 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L11 compound treatment 181560.0 16900.0 1.15 187560.0 21200.0 1.58 1.9311 0.9881 3622845 Ald3.1-H_000227 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L12 compound treatment 193280.0 28600.0 1.95 194240.0 27900.0 2.07 2.8477 0.9995 3622847 Ald3.1-H_000228 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L13 compound treatment 182800.0 18200.0 1.24 183200.0 16800.0 1.25 1.7615 1.0 3622849 Ald3.1-H_000229 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L14 compound treatment 171000.0 6360.0 0.43 173200.0 6840.0 0.51 0.6663 0.9968 3622851 Ald3.1-H_000230 OC(=O)CCCCCC(=O)N/N=C/c1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L15 mock treatment 168000.0 3360.0 0.23 170800.0 4440.0 0.33 0.3954 0.9839 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L16 mock treatment 167000.0 2360.0 0.16 170440.0 4080.0 0.3 0.3282 0.9557 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L17 compound treatment 205320.0 40700.0 2.77 224200.0 57800.0 4.3 5.0049 0.9774 3622853 Ald3.1-H_000231 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L18 compound treatment 167560.0 2920.0 0.2 169800.0 3440.0 0.26 0.3216 0.9922 3622855 Ald3.1-H_000232 CC(=O)N/N=C/c1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L19 compound treatment 223040.0 58400.0 3.98 220200.0 53800.0 4.01 5.6486 1.0 3622857 Ald3.1-H_000233 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L20 compound treatment 159880.0 -4760.0 -0.32 164480.0 -1880.0 -0.14 -0.3287 -0.9293 3622859 Ald3.1-H_000234 O=Cc1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L21 compound treatment 179080.0 14400.0 0.98 175400.0 9040.0 0.67 1.1716 0.9828 3553658 Ald3.1-H_000235 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L22 compound treatment 172280.0 7640.0 0.52 170560.0 4200.0 0.31 0.5891 0.9702 3622860 Ald3.1-H_000236 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L23 mock treatment 156920.0 -7720.0 -0.53 157720.0 -8640.0 -0.64 -0.8271 -0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 L24 mock treatment 203840.0 39200.0 2.67 155840.0 -10500.0 -0.78 1.3359 0.4797 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M01 compound treatment 183840.0 19200.0 1.31 177560.0 11200.0 0.83 1.5148 0.9763 3622862 Ald3.1-H_000237 ONC(=O)CCCCC(=O)N/N=C/c1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M02 compound treatment 260840.0 96200.0 6.56 265560.0 99200.0 7.38 9.8581 0.9983 3622864 Ald3.1-H_000238 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M03 compound treatment 194920.0 30300.0 2.06 197320.0 31000.0 2.3 3.0889 0.9985 3622866 Ald3.1-H_000239 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M04 compound treatment 274040.0 109000.0 7.46 267680.0 101000.0 7.54 10.606 1.0 3622868 Ald3.1-H_000240 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M05 compound treatment 200880.0 36200.0 2.47 192200.0 25800.0 1.92 3.1067 0.9923 3622870 Ald3.1-H_000241 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M06 compound treatment 267720.0 103000.0 7.03 255880.0 89500.0 6.66 9.6803 0.9996 3622872 Ald3.1-H_000242 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M07 compound treatment 274160.0 110000.0 7.47 259240.0 92900.0 6.91 10.1676 0.9993 3622874 Ald3.1-H_000243 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M08 compound treatment 198400.0 33800.0 2.3 212120.0 45800.0 3.41 4.0355 0.9818 3622876 Ald3.1-H_000244 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M09 mock treatment 176440.0 11800.0 0.8 176120.0 9760.0 0.73 1.0823 0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M10 mock treatment 176880.0 12200.0 0.83 176560.0 10200.0 0.76 1.1266 0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M11 compound treatment 232360.0 67700.0 4.62 235400.0 69000.0 5.14 6.8978 0.9986 3622878 Ald3.1-H_000245 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M12 compound treatment 209240.0 44600.0 3.04 206960.0 40600.0 3.02 4.2865 1.0 3622880 Ald3.1-H_000246 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M13 mock treatment 170320.0 5680.0 0.39 173920.0 7560.0 0.56 0.6714 0.9833 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M14 mock treatment 166960.0 2320.0 0.16 172520.0 6160.0 0.46 0.4358 0.8989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M15 compound treatment 243800.0 79200.0 5.4 241040.0 74700.0 5.56 7.7462 0.9999 3622882 Ald3.1-H_000247 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M16 compound treatment 169320.0 4680.0 0.32 175560.0 9200.0 0.68 0.7095 0.9395 3622884 Ald3.1-H_000248 OC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M17 compound treatment 282200.0 118000.0 8.01 276400.0 110000.0 8.19 11.4583 0.9999 3622886 Ald3.1-H_000249 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M18 compound treatment 166880.0 2240.0 0.15 177280.0 10900.0 0.81 0.6824 0.8254 3622888 Ald3.1-H_000250 CC(=O)N/N=C/c1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M19 compound treatment 223440.0 58800.0 4.01 208240.0 41900.0 3.12 5.0385 0.9923 3622890 Ald3.1-H_000251 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M20 compound treatment 165200.0 556.0 0.04 167640.0 1280.0 0.1 0.0941 0.9186 3622892 Ald3.1-H_000252 O=Cc1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M21 compound treatment 207960.0 43300.0 2.95 207520.0 41200.0 3.06 4.2543 0.9998 3622894 Ald3.1-H_000253 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(CN3[C@H]4CCC[C@@H]4OC(=O)CC/C=C/CCC3=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M22 compound treatment 165400.0 756.0 0.05 168240.0 1880.0 0.14 0.1353 0.9081 3622896 Ald3.1-H_000254 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(CN2[C@H]3CCC[C@@H]3OC(=O)CC/C=C/CCC2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M23 compound treatment 264760.0 100000.0 6.83 272560.0 106000.0 7.9 10.4154 0.9973 3622898 Ald3.1-H_000255 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 M24 compound treatment 201560.0 36900.0 2.52 189080.0 22700.0 1.69 2.9753 0.9813 3622900 Ald3.1-H_000256 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N01 compound treatment 189280.0 24600.0 1.68 191360.0 25000.0 1.86 2.5033 0.9987 3622902 Ald3.1-H_000257 ONC(=O)CCCCC(=O)N/N=C/c1ccc(cc1)c2ccc(\C=N\NC(=O)CCCCC(=O)NO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N02 compound treatment 194880.0 30200.0 2.06 200320.0 34000.0 2.53 3.2448 0.9949 3622904 Ald3.1-H_000258 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4ccc(OCCCCCCC(=O)NO)cc4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N03 compound treatment 196000.0 31400.0 2.14 194720.0 28400.0 2.11 3.0041 1.0 3622906 Ald3.1-H_000259 ONC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)c2ccc(\C=N\NC(=O)CCCCCC(=O)NO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N04 compound treatment 186960.0 22300.0 1.52 188720.0 22400.0 1.66 2.2525 0.999 3622908 Ald3.1-H_000260 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4ccc(OCCCCCCC(=O)NO)c(OC)c4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N05 compound treatment 182520.0 17900.0 1.22 187760.0 21400.0 1.59 1.9879 0.9913 3622910 Ald3.1-H_000261 ONC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)c2ccc(\C=N\NC(=O)CCCCCCC(=O)NO)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N06 compound treatment 201480.0 36800.0 2.51 200760.0 34400.0 2.56 3.5861 1.0 3622912 Ald3.1-H_000262 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4ccc(OCCCCCCC(=O)NO)c5ccccc45)cc3)c6ccccc16 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N07 compound treatment 200600.0 36000.0 2.45 198920.0 32600.0 2.42 3.4469 1.0 3622914 Ald3.1-H_000263 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4cccc(c4)C(=O)NO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N08 compound treatment 195520.0 30900.0 2.11 200120.0 33800.0 2.51 3.2651 0.9961 3622916 Ald3.1-H_000264 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)CCCCC(=O)Nc4ccccc4O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N09 mock treatment 177120.0 12500.0 0.85 178040.0 11700.0 0.87 1.2161 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N10 mock treatment 174920.0 10300.0 0.7 176320.0 9960.0 0.74 1.0195 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N11 compound treatment 256160.0 91500.0 6.24 261320.0 95000.0 7.07 9.4093 0.9981 3622918 Ald3.1-H_000265 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4cccc(OCC(=O)NO)c4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N12 compound treatment 182200.0 17600.0 1.2 187600.0 21200.0 1.58 1.9641 0.9906 3622920 Ald3.1-H_000266 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)CCCCCCC(=O)Nc4ccccc4O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N13 mock treatment 206920.0 42300.0 2.88 211800.0 45400.0 3.38 4.4294 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N14 mock treatment 171000.0 6360.0 0.43 174480.0 8120.0 0.6 0.7337 0.9867 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N15 compound treatment 263800.0 99200.0 6.76 296040.0 130000.0 9.65 11.6049 0.9848 3622922 Ald3.1-H_000267 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4cccc(OCCCCCC(=O)NO)c4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N16 compound treatment 178520.0 13900.0 0.95 175400.0 9040.0 0.67 1.1446 0.986 3622924 Ald3.1-H_000268 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(cc1)c2ccc(\C=N\NC(=O)CCCCCCC(=O)O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N17 compound treatment 187160.0 22500.0 1.54 188000.0 21600.0 1.61 2.2243 0.9997 3622926 Ald3.1-H_000269 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4ccc(OCCCCCC(=O)NO)cc4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N18 compound treatment 170360.0 5720.0 0.39 175400.0 9040.0 0.67 0.7513 0.9663 3622928 Ald3.1-H_000270 CC(=O)N/N=C/c1ccc(cc1)c2ccc(\C=N\NC(=O)C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N19 compound treatment 183080.0 18400.0 1.26 178880.0 12500.0 0.93 1.5476 0.9891 3622930 Ald3.1-H_000271 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4cccc(OCCCCCCC(=O)NO)c4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N20 compound treatment 163400.0 -1240.0 -0.08 163680.0 -2680.0 -0.2 -0.2011 -0.9273 3622932 Ald3.1-H_000272 O=Cc1ccc(cc1)c2ccc(C=O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N21 compound treatment 197360.0 32700.0 2.23 188000.0 21600.0 1.61 2.716 0.9872 3622933 Ald3.1-H_000273 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2ccc(OCC#C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N22 compound treatment 159960.0 -4680.0 -0.32 160880.0 -5480.0 -0.41 -0.5143 -0.9927 3622935 Ald3.1-H_000274 OC(=O)CCCCCCC(=O)N/N=C/c1ccc(OCC#C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N23 compound treatment 209200.0 44600.0 3.04 206960.0 40600.0 3.02 4.2846 1.0 3622937 Ald3.1-H_000275 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4ccc(cc4)C(=O)NO)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 N24 compound treatment 163720.0 -924.0 -0.06 165920.0 -441.0 -0.03 -0.0678 -0.9539 3622939 Ald3.1-H_000276 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)CCCCCC(=O)Nc4ccccc4O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O01 compound treatment 183000.0 18400.0 1.25 180040.0 13700.0 1.02 1.6048 0.9948 3622941 Ald3.1-H_000277 ONC(=O)CCCCC(=O)N/N=C/c1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O02 compound treatment 228360.0 63700.0 4.34 245000.0 78600.0 5.85 7.2102 0.9892 3622942 Ald3.1-H_000278 ONC(=O)CCCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O03 compound treatment 183320.0 18700.0 1.27 181480.0 15100.0 1.13 1.696 0.9981 3622943 Ald3.1-H_000279 ONC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O04 compound treatment 243760.0 79100.0 5.39 249080.0 82700.0 6.16 8.1674 0.9978 3622944 Ald3.1-H_000280 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O05 compound treatment 191600.0 27000.0 1.84 191480.0 25100.0 1.87 2.6215 1.0 3622945 Ald3.1-H_000281 ONC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O06 compound treatment 250120.0 85500.0 5.83 234280.0 67900.0 5.05 7.6951 0.9975 3622946 Ald3.1-H_000282 ONC(=O)CCCCCCOc1ccc(C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2)c5ccccc15 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O07 compound treatment 254760.0 90100.0 6.14 244200.0 77800.0 5.79 8.4408 0.9996 3622947 Ald3.1-H_000283 ONC(=O)c1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O08 compound treatment 193440.0 28800.0 1.96 195880.0 29500.0 2.2 2.9417 0.9984 3622948 Ald3.1-H_000284 Oc1ccccc1NC(=O)CCCCC(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O09 compound treatment 260480.0 95800.0 6.53 251640.0 85300.0 6.35 9.1081 0.9999 3622949 Ald3.1-H_000285 ONC(=O)c1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O10 compound treatment 205920.0 41300.0 2.81 203480.0 37100.0 2.76 3.9433 1.0 3622950 Ald3.1-H_000286 Oc1ccccc1NC(=O)CCCCCC(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O11 mock treatment 170560.0 5920.0 0.4 176480.0 10100.0 0.75 0.8177 0.9572 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O12 mock treatment 164760.0 116.0 0.01 172720.0 6360.0 0.47 0.3402 0.7188 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O13 compound treatment 246640.0 82000.0 5.59 231280.0 64900.0 4.83 7.3694 0.9974 3622951 Ald3.1-H_000287 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O14 compound treatment 167600.0 2960.0 0.2 171680.0 5320.0 0.4 0.4224 0.951 3622953 Ald3.1-H_000288 OC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O15 compound treatment 198960.0 34300.0 2.34 231440.0 65100.0 4.84 5.0793 0.9443 3622955 Ald3.1-H_000289 ONC(=O)CCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O16 compound treatment 166440.0 1800.0 0.12 184560.0 18200.0 1.35 1.0444 0.7679 3622956 Ald3.1-H_000290 OC(=O)CCCCCCC(=O)N/N=C/c1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O17 compound treatment 271960.0 107000.0 7.32 270200.0 104000.0 7.73 10.6383 0.9996 3622957 Ald3.1-H_000291 ONC(=O)CCCCCOc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O18 compound treatment 170360.0 5720.0 0.39 172280.0 5920.0 0.44 0.5871 0.9981 3622958 Ald3.1-H_000292 CC(=O)N/N=C/c1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O19 compound treatment 240760.0 76100.0 5.19 246800.0 80400.0 5.99 7.9027 0.9975 3622959 Ald3.1-H_000293 ONC(=O)CCCCCCOc1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O20 compound treatment 161800.0 -2840.0 -0.19 166840.0 479.0 0.04 -0.1119 -0.5677 3622960 Ald3.1-H_000294 O=Cc1cccc(CN2C[C@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O21 compound treatment 243160.0 78500.0 5.35 233880.0 67500.0 5.03 7.3385 0.9995 3622961 Ald3.1-H_000295 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2cccc(CN3C[C@@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O22 compound treatment 158080.0 -6560.0 -0.45 158560.0 -7800.0 -0.58 -0.727 -0.9917 3622962 Ald3.1-H_000296 OC(=O)CCCCCC(=O)N/N=C/c1cccc(CN2C[C@@H](OC(=O)CC/C=C/CCC2=O)c3ccccc3)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O23 compound treatment 223000.0 58400.0 3.98 207400.0 41000.0 3.05 4.973 0.9915 3622963 Ald3.1-H_000297 ONC(=O)COc1cccc(c1)C(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 O24 compound treatment 181080.0 16400.0 1.12 173480.0 7120.0 0.53 1.167 0.9415 3622964 Ald3.1-H_000298 Oc1ccccc1NC(=O)CCCCCCC(=O)N/N=C/c2cccc(CN3C[C@H](OC(=O)CC/C=C/CCC3=O)c4ccccc4)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P01 compound treatment 167520.0 2880.0 0.2 172200.0 5840.0 0.43 0.4459 0.9354 3214824 Ald3.1-H_000299 NNC(=O)CCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P02 compound treatment 184640.0 20000.0 1.36 186000.0 19600.0 1.46 1.9975 0.9994 3622965 Ald3.1-H_000300 NNC(=O)c1ccc(OCCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P03 compound treatment 173120.0 8480.0 0.58 172000.0 5640.0 0.42 0.7054 0.9877 3214214 Ald3.1-H_000301 NNC(=O)CCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P04 compound treatment 179640.0 15000.0 1.02 181600.0 15200.0 1.13 1.5249 0.9987 3622966 Ald3.1-H_000302 COc1cc(ccc1OCCCCCCC(=O)NO)C(=O)NN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P05 compound treatment 171560.0 6920.0 0.47 176080.0 9720.0 0.72 0.8449 0.9785 3213058 Ald3.1-H_000303 NNC(=O)CCCCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P06 compound treatment 195480.0 30800.0 2.1 194400.0 28000.0 2.09 2.9622 1.0 3622967 Ald3.1-H_000304 NNC(=O)c1ccc(OCCCCCCC(=O)NO)c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P07 compound treatment 176880.0 12200.0 0.83 181160.0 14800.0 1.1 1.3687 0.9906 3551921 Ald3.1-H_000305 NNC(=O)c1cccc(c1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P08 compound treatment 175120.0 10500.0 0.71 178160.0 11800.0 0.88 1.126 0.9947 3622968 Ald3.1-H_000306 NNC(=O)CCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P09 compound treatment 181000.0 16400.0 1.12 181840.0 15500.0 1.15 1.6031 0.9999 3551923 Ald3.1-H_000307 NNC(=O)c1ccc(cc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P10 compound treatment 174040.0 9400.0 0.64 181920.0 15600.0 1.16 1.2718 0.961 3214215 Ald3.1-H_000308 NNC(=O)CCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P11 mock treatment 159920.0 -4720.0 -0.32 172000.0 5640.0 0.42 0.069 0.1305 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P12 mock treatment 167600.0 2960.0 0.2 166560.0 199.0 0.01 0.153 0.757 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P13 compound treatment 176960.0 12300.0 0.84 184240.0 17900.0 1.33 1.5347 0.9754 3622969 Ald3.1-H_000309 NNC(=O)c1ccc(OCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P14 compound treatment 164160.0 -484.0 -0.03 171960.0 5600.0 0.42 0.2713 0.6491 3213669 Ald3.1-H_000310 NNC(=O)CCCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P15 compound treatment 187520.0 22900.0 1.56 189800.0 23400.0 1.74 2.3364 0.9984 3622970 Ald3.1-H_000311 NNC(=O)c1cccc(OCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P16 compound treatment 160560.0 -4080.0 -0.28 164920.0 -1440.0 -0.11 -0.2727 -0.914 3213668 Ald3.1-H_000312 NNC(=O)CCCCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P17 compound treatment 183440.0 18800.0 1.28 181440.0 15100.0 1.12 1.6997 0.9978 3622971 Ald3.1-H_000313 NNC(=O)c1ccc(OCCCCCC(=O)NO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P18 compound treatment 232240.0 67600.0 4.61 163120.0 -3240.0 -0.24 3.0881 0.6692 1003260 Ald3.1-H_000314 CC(=O)NN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P19 compound treatment 175480.0 10800.0 0.74 181400.0 15000.0 1.12 1.3138 0.9797 3622972 Ald3.1-H_000315 NNC(=O)c1cccc(OCCCCCCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P20 mock treatment 152880.0 -11800.0 -0.8 159680.0 -6680.0 -0.5 -0.9187 -0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P21 compound treatment 168640.0 4000.0 0.27 165880.0 -481.0 -0.04 0.1673 0.6089 3622973 Ald3.1-H_000316 ONC(=O)COc1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)c3ccc(\C=N\NC(=O)c4ccc(OCC(=O)NO)cc4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P22 compound treatment 158800.0 -5840.0 -0.4 158920.0 -7440.0 -0.55 -0.6733 -0.9869 3622975 Ald3.1-H_000317 OC(=O)CCCCCC(=O)N/N=C/c1ccc(cc1)c2ccc(\C=N\NC(=O)CCCCCC(=O)O)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P23 compound treatment 165840.0 1200.0 0.08 163840.0 -2520.0 -0.19 -0.075 -0.3667 3622977 Ald3.1-H_000318 NNC(=O)c1cccc(OCC(=O)NO)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2410 P24 compound treatment 161920.0 -2720.0 -0.19 158960.0 -7400.0 -0.55 -0.5208 -0.8959 3213059 Ald3.1-H_000319 NNC(=O)CCCCCCC(=O)Nc1ccccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A01 compound treatment 156520.0 -3360.0 -0.23 155320.0 -3900.0 -0.29 -0.367 -0.9932 DHPC8.2_000001 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A02 compound treatment 156520.0 -3360.0 -0.23 152920.0 -6300.0 -0.47 -0.4934 -0.9458 DHPC8.2_000002 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A03 compound treatment 150280.0 -9600.0 -0.65 150440.0 -8780.0 -0.65 -0.9247 -1.0 DHPC8.2_000003 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A04 compound treatment 159640.0 -239.0 -0.02 159320.0 103.0 0.01 -0.0061 -0.3402 DHPC8.2_000004 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A05 compound treatment 157360.0 -2520.0 -0.17 155400.0 -3820.0 -0.28 -0.3223 -0.9709 DHPC8.2_000005 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A06 compound treatment 153480.0 -6400.0 -0.44 150520.0 -8700.0 -0.65 -0.7662 -0.9816 DHPC8.2_000006 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A07 compound treatment 155080.0 -4800.0 -0.33 150640.0 -8580.0 -0.64 -0.6828 -0.9518 DHPC8.2_000007 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A08 compound treatment 151560.0 -8320.0 -0.57 150400.0 -8820.0 -0.66 -0.8651 -0.9974 DHPC8.2_000008 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A09 compound treatment 151000.0 -8880.0 -0.61 149640.0 -9580.0 -0.71 -0.9321 -0.9967 DHPC8.2_000009 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A10 compound treatment 151600.0 -8280.0 -0.56 150600.0 -8620.0 -0.64 -0.8526 -0.998 DHPC8.2_000010 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A11 compound treatment 154960.0 -4920.0 -0.34 152880.0 -6340.0 -0.47 -0.5707 -0.986 DHPC8.2_000011 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A12 compound treatment 151560.0 -8320.0 -0.57 150120.0 -9100.0 -0.68 -0.8798 -0.9961 DHPC8.2_000012 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A13 mock treatment 155160.0 -4720.0 -0.32 147760.0 -11500.0 -0.85 -0.8305 -0.9112 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A14 mock treatment 152600.0 -7280.0 -0.5 147880.0 -11300.0 -0.84 -0.9476 -0.968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A15 compound treatment 151680.0 -8200.0 -0.56 150200.0 -9020.0 -0.67 -0.8698 -0.9959 DHPC8.2_000013 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A16 compound treatment 149760.0 -10100.0 -0.69 148600.0 -10600.0 -0.79 -1.0466 -0.9977 DHPC8.2_000014 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A17 compound treatment 148800.0 -11100.0 -0.76 147240.0 -12000.0 -0.89 -1.1644 -0.9966 DHPC8.2_000015 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A18 compound treatment 144480.0 -15400.0 -1.05 149080.0 -10100.0 -0.75 -1.2759 -0.9869 DHPC8.2_000016 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A19 compound treatment 147920.0 -12000.0 -0.82 149960.0 -9260.0 -0.69 -1.0637 -0.9965 DHPC8.2_000017 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A20 compound treatment 168640.0 8760.0 0.6 169840.0 10600.0 0.79 0.9814 0.9904 DHPC8.2_000018 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A21 compound treatment 148640.0 -11200.0 -0.77 146680.0 -12500.0 -0.93 -1.2016 -0.9952 DHPC8.2_000019 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A22 compound treatment 176520.0 16600.0 1.13 174160.0 14900.0 1.11 1.5886 1.0 DHPC8.2_000020 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A23 compound treatment 151400.0 -8480.0 -0.58 144360.0 -14900.0 -1.11 -1.1907 -0.9542 DHPC8.2_000021 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 A24 compound treatment 155920.0 -3960.0 -0.27 149240.0 -9980.0 -0.74 -0.7159 -0.9061 DHPC8.2_000022 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B01 mock treatment 148400.0 -11500.0 -0.78 147160.0 -12100.0 -0.9 -1.1879 -0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B02 mock treatment 147320.0 -12600.0 -0.86 147000.0 -12200.0 -0.91 -1.2484 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B03 mock treatment 147320.0 -12600.0 -0.86 149280.0 -9940.0 -0.74 -1.1284 -0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B04 mock treatment 151200.0 -8680.0 -0.59 147360.0 -11900.0 -0.88 -1.0424 -0.9811 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B05 mock treatment 155840.0 -4040.0 -0.28 148800.0 -10400.0 -0.78 -0.743 -0.903 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B06 mock treatment 265760.0 106000.0 7.22 146440.0 -12800.0 -0.95 4.4319 0.6087 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B07 mock treatment 145960.0 -13900.0 -0.95 149240.0 -9980.0 -0.74 -1.1961 -0.9926 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B08 mock treatment 149520.0 -10400.0 -0.71 144480.0 -14700.0 -1.1 -1.275 -0.9773 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B09 mock treatment 149320.0 -10600.0 -0.72 145840.0 -13400.0 -1.0 -1.2131 -0.9873 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B10 mock treatment 151640.0 -8240.0 -0.56 147160.0 -12100.0 -0.9 -1.0317 -0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B11 mock treatment 151800.0 -8080.0 -0.55 147120.0 -12100.0 -0.9 -1.0261 -0.9722 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B12 mock treatment 151800.0 -8080.0 -0.55 148720.0 -10500.0 -0.78 -0.9419 -0.9854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B13 mock treatment 152240.0 -7640.0 -0.52 148920.0 -10300.0 -0.77 -0.9102 -0.9823 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B14 mock treatment 149040.0 -10800.0 -0.74 148920.0 -10300.0 -0.77 -1.0645 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B15 mock treatment 149160.0 -10700.0 -0.73 144840.0 -14400.0 -1.07 -1.2734 -0.9827 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B16 mock treatment 147720.0 -12200.0 -0.83 143720.0 -15500.0 -1.15 -1.4018 -0.9869 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B17 mock treatment 148200.0 -11700.0 -0.8 144760.0 -14500.0 -1.08 -1.3239 -0.989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B18 mock treatment 148800.0 -11100.0 -0.76 149920.0 -9300.0 -0.69 -1.0234 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B19 mock treatment 151760.0 -8120.0 -0.55 153360.0 -5860.0 -0.44 -0.6997 -0.993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B20 mock treatment 153800.0 -6080.0 -0.41 148520.0 -10700.0 -0.8 -0.856 -0.9537 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B21 mock treatment 151240.0 -8640.0 -0.59 145840.0 -13400.0 -1.0 -1.1205 -0.9686 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B22 mock treatment 151280.0 -8600.0 -0.59 147000.0 -12200.0 -0.91 -1.0575 -0.9775 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B23 mock treatment 147280.0 -12600.0 -0.86 151080.0 -8140.0 -0.61 -1.0356 -0.9854 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 B24 mock treatment 146440.0 -13400.0 -0.92 142520.0 -16700.0 -1.24 -1.5266 -0.9888 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C01 compound treatment 161560.0 1680.0 0.11 157840.0 -1380.0 -0.1 0.0085 0.0556 DHPC8.2_000023 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C02 compound treatment 154400.0 -5480.0 -0.37 159560.0 343.0 0.03 -0.2461 -0.6573 DHPC8.2_000024 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C03 compound treatment 150600.0 -9280.0 -0.63 158080.0 -1140.0 -0.08 -0.5072 -0.7946 DHPC8.2_000025 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C04 compound treatment 157520.0 -2360.0 -0.16 156400.0 -2820.0 -0.21 -0.262 -0.9914 DHPC8.2_000026 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C05 compound treatment 157840.0 -2040.0 -0.14 159400.0 183.0 0.01 -0.0887 -0.6349 DHPC8.2_000027 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C06 compound treatment 156440.0 -3440.0 -0.23 161800.0 2580.0 0.19 -0.0299 -0.0985 DHPC8.2_000028 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C07 compound treatment 152000.0 -7880.0 -0.54 156120.0 -3100.0 -0.23 -0.5428 -0.9287 DHPC8.2_000029 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C08 compound treatment 170040.0 10200.0 0.69 167280.0 8060.0 0.6 0.9142 0.9974 DHPC8.2_000030 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C09 compound treatment 158200.0 -1680.0 -0.11 162200.0 2980.0 0.22 0.076 0.3044 DHPC8.2_000031 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C10 compound treatment 156520.0 -3360.0 -0.23 152800.0 -6420.0 -0.48 -0.4997 -0.9433 DHPC8.2_000032 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C11 mock treatment 154560.0 -5320.0 -0.36 151320.0 -7900.0 -0.59 -0.672 -0.9731 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C12 mock treatment 154960.0 -4920.0 -0.34 158160.0 -1060.0 -0.08 -0.2928 -0.8499 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C13 compound treatment 177960.0 18100.0 1.23 175800.0 16600.0 1.23 1.7444 1.0 DHPC8.2_000033 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C14 compound treatment 154440.0 -5440.0 -0.37 151280.0 -7940.0 -0.59 -0.6799 -0.9748 DHPC8.2_000034 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C15 mock treatment 150360.0 -9520.0 -0.65 155360.0 -3860.0 -0.29 -0.6619 -0.9327 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C16 mock treatment 153520.0 -6360.0 -0.43 155840.0 -3380.0 -0.25 -0.4843 -0.9664 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C17 compound treatment 153040.0 -6840.0 -0.47 154960.0 -4260.0 -0.32 -0.5538 -0.9823 DHPC8.2_000035 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C18 compound treatment 155880.0 -4000.0 -0.27 151600.0 -7620.0 -0.57 -0.5937 -0.9437 DHPC8.2_000036 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C19 compound treatment 179640.0 19800.0 1.35 177480.0 18300.0 1.36 1.9138 1.0 DHPC8.2_000037 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C20 compound treatment 155520.0 -4360.0 -0.3 151320.0 -7900.0 -0.59 -0.6258 -0.9501 DHPC8.2_000038 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C21 compound treatment 160600.0 721.0 0.05 159240.0 22.6 0.0 0.0359 0.7309 DHPC8.2_000039 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C22 compound treatment 146080.0 -13800.0 -0.94 152320.0 -6900.0 -0.51 -1.0282 -0.9594 DHPC8.2_000040 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C23 compound treatment 149080.0 -10800.0 -0.74 146840.0 -12400.0 -0.92 -1.172 -0.9938 DHPC8.2_000041 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 C24 compound treatment 170840.0 11000.0 0.75 164800.0 5580.0 0.42 0.8222 0.9616 DHPC8.2_000042 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D01 mock treatment 150040.0 -9840.0 -0.67 147520.0 -11700.0 -0.87 -1.0899 -0.9917 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D02 mock treatment 149360.0 -10500.0 -0.72 149560.0 -9660.0 -0.72 -1.0154 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D03 mock treatment 153960.0 -5920.0 -0.4 155920.0 -3300.0 -0.25 -0.4589 -0.9716 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D04 mock treatment 156880.0 -3000.0 -0.2 150120.0 -9100.0 -0.68 -0.6234 -0.8813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D05 mock treatment 156360.0 -3520.0 -0.24 156640.0 -2580.0 -0.19 -0.3053 -0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D06 mock treatment 152120.0 -7760.0 -0.53 156280.0 -2940.0 -0.22 -0.5286 -0.9236 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D07 mock treatment 145480.0 -14400.0 -0.98 153120.0 -6100.0 -0.45 -1.015 -0.9386 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D08 mock treatment 155720.0 -4160.0 -0.28 151920.0 -7300.0 -0.54 -0.5845 -0.9541 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D09 mock treatment 155200.0 -4680.0 -0.32 146240.0 -13000.0 -0.97 -0.9085 -0.8932 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D10 mock treatment 156080.0 -3800.0 -0.26 154440.0 -4780.0 -0.36 -0.4346 -0.9879 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D11 mock treatment 154400.0 -5480.0 -0.37 154240.0 -4980.0 -0.37 -0.5261 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D12 mock treatment 154160.0 -5720.0 -0.39 157000.0 -2220.0 -0.17 -0.3924 -0.9268 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D13 mock treatment 158840.0 -1040.0 -0.07 154240.0 -4980.0 -0.37 -0.312 -0.8273 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D14 mock treatment 155560.0 -4320.0 -0.29 151640.0 -7580.0 -0.56 -0.607 -0.9541 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D15 mock treatment 155400.0 -4480.0 -0.31 149800.0 -9420.0 -0.7 -0.7115 -0.9307 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D16 mock treatment 155040.0 -4840.0 -0.33 149960.0 -9260.0 -0.69 -0.7205 -0.9431 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D17 mock treatment 148320.0 -11600.0 -0.79 145520.0 -13700.0 -1.02 -1.2781 -0.9919 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D18 mock treatment 158720.0 -1160.0 -0.08 154720.0 -4500.0 -0.33 -0.2926 -0.8507 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D19 mock treatment 150960.0 -8920.0 -0.61 154520.0 -4700.0 -0.35 -0.6772 -0.9655 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D20 mock treatment 153680.0 -6200.0 -0.42 152920.0 -6300.0 -0.47 -0.6303 -0.9987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D21 mock treatment 149600.0 -10300.0 -0.7 148320.0 -10900.0 -0.81 -1.069 -0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D22 mock treatment 152480.0 -7400.0 -0.5 150520.0 -8700.0 -0.65 -0.8144 -0.9924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D23 mock treatment 146360.0 -13500.0 -0.92 145880.0 -13300.0 -0.99 -1.3536 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 D24 mock treatment 148520.0 -11400.0 -0.77 145880.0 -13300.0 -0.99 -1.2495 -0.9925 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E01 mock treatment 154600.0 -5280.0 -0.36 158640.0 -577.0 -0.04 -0.2849 -0.7859 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E02 mock treatment 156240.0 -3640.0 -0.25 156360.0 -2860.0 -0.21 -0.3258 -0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E03 compound treatment 162320.0 2440.0 0.17 163160.0 3940.0 0.29 0.3252 0.9639 DHPC8.2_000043 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E04 compound treatment 179680.0 19800.0 1.35 160720.0 1500.0 0.11 1.0336 0.7631 DHPC8.2_000044 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E05 compound treatment 167200.0 7320.0 0.5 162920.0 3700.0 0.28 0.5478 0.9608 DHPC8.2_000045 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E06 compound treatment 172360.0 12500.0 0.85 168880.0 9660.0 0.72 1.1102 0.9965 DHPC8.2_000046 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E07 compound treatment 163560.0 3680.0 0.25 154120.0 -5100.0 -0.38 -0.0908 -0.1996 DHPC8.2_000047 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E08 compound treatment 165000.0 5120.0 0.35 163280.0 4060.0 0.3 0.4607 0.9974 DHPC8.2_000048 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E09 mock treatment 162520.0 2640.0 0.18 158120.0 -1100.0 -0.08 0.0696 0.3518 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E10 mock treatment 163520.0 3640.0 0.25 160680.0 1460.0 0.11 0.2525 0.9316 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E11 compound treatment 171000.0 11100.0 0.76 170520.0 11300.0 0.84 1.131 0.9987 DHPC8.2_000049 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E12 compound treatment 189160.0 29300.0 2.0 186480.0 27300.0 2.03 2.8464 1.0 DHPC8.2_000050 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E13 compound treatment 167120.0 7240.0 0.49 163960.0 4740.0 0.35 0.5987 0.9865 DHPC8.2_000051 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E14 compound treatment 201920.0 42000.0 2.87 194440.0 35200.0 2.62 3.8804 0.999 DHPC8.2_000052 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E15 compound treatment 162240.0 2360.0 0.16 161080.0 1860.0 0.14 0.2118 0.9972 DHPC8.2_000053 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E16 compound treatment 182680.0 22800.0 1.55 178880.0 19700.0 1.46 2.134 0.9995 DHPC8.2_000054 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E17 mock treatment 158000.0 -1880.0 -0.13 154760.0 -4460.0 -0.33 -0.3252 -0.9144 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E18 mock treatment 159720.0 -159.0 -0.01 160800.0 1580.0 0.12 0.0756 0.6393 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E19 compound treatment 156520.0 -3360.0 -0.23 157840.0 -1380.0 -0.1 -0.2344 -0.9343 DHPC8.2_000055 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E20 compound treatment 156480.0 -3400.0 -0.23 156760.0 -2460.0 -0.18 -0.2932 -0.9931 DHPC8.2_000056 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E21 compound treatment 166720.0 6840.0 0.47 162080.0 2860.0 0.21 0.4804 0.937 DHPC8.2_000057 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E22 compound treatment 187080.0 27200.0 1.85 183320.0 24100.0 1.79 2.5798 0.9999 DHPC8.2_000058 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E23 compound treatment 167200.0 7320.0 0.5 163120.0 3900.0 0.29 0.5583 0.9668 DHPC8.2_000059 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 E24 compound treatment 156560.0 -3320.0 -0.23 149960.0 -9260.0 -0.69 -0.6472 -0.8924 DHPC8.2_000060 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F01 mock treatment 159760.0 -119.0 -0.01 154240.0 -4980.0 -0.37 -0.2677 -0.7224 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F02 mock treatment 158000.0 -1880.0 -0.13 158960.0 -257.0 -0.02 -0.1041 -0.8039 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F03 mock treatment 158000.0 -1880.0 -0.13 158400.0 -817.0 -0.06 -0.1336 -0.9421 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F04 mock treatment 156600.0 -3280.0 -0.22 155880.0 -3340.0 -0.25 -0.3337 -0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F05 mock treatment 159640.0 -239.0 -0.02 162800.0 3580.0 0.27 0.177 0.6626 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F06 mock treatment 164680.0 4800.0 0.33 157920.0 -1300.0 -0.1 0.1632 0.4781 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F07 mock treatment 164120.0 4240.0 0.29 162480.0 3260.0 0.24 0.3762 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F08 mock treatment 161560.0 1680.0 0.11 157640.0 -1580.0 -0.12 -0.002 -0.0121 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F09 mock treatment 160080.0 201.0 0.01 161160.0 1940.0 0.14 0.1119 0.7706 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F10 mock treatment 159280.0 -599.0 -0.04 161560.0 2340.0 0.17 0.0944 0.5272 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F11 mock treatment 161400.0 1520.0 0.1 162120.0 2900.0 0.22 0.2261 0.9435 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F12 mock treatment 159040.0 -839.0 -0.06 164480.0 5260.0 0.39 0.2365 0.5975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F13 mock treatment 157360.0 -2520.0 -0.17 156920.0 -2300.0 -0.17 -0.2423 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F14 mock treatment 158080.0 -1800.0 -0.12 159520.0 303.0 0.02 -0.0708 -0.5678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F15 mock treatment 157280.0 -2600.0 -0.18 158720.0 -497.0 -0.04 -0.1515 -0.8368 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F16 mock treatment 162600.0 2720.0 0.19 160080.0 863.0 0.06 0.1766 0.8995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F17 mock treatment 160400.0 521.0 0.04 159640.0 423.0 0.03 0.0474 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F18 mock treatment 161160.0 1280.0 0.09 159240.0 22.6 0.0 0.0629 0.7206 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F19 mock treatment 157520.0 -2360.0 -0.16 156760.0 -2460.0 -0.18 -0.2431 -0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F20 mock treatment 155600.0 -4280.0 -0.29 161680.0 2460.0 0.18 -0.0767 -0.2226 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F21 mock treatment 155560.0 -4320.0 -0.29 157640.0 -1580.0 -0.12 -0.2912 -0.9187 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F22 mock treatment 155760.0 -4120.0 -0.28 163920.0 4700.0 0.35 0.0489 0.109 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F23 mock treatment 156760.0 -3120.0 -0.21 159080.0 -137.0 -0.01 -0.1576 -0.7402 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 F24 mock treatment 154720.0 -5160.0 -0.35 147880.0 -11300.0 -0.84 -0.8454 -0.9247 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G01 compound treatment 176040.0 16200.0 1.1 172080.0 12900.0 0.96 1.456 0.9975 DHPC8.2_000061 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G02 compound treatment 194400.0 34500.0 2.35 185840.0 26600.0 1.98 3.0653 0.9963 DHPC8.2_000062 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G03 mock treatment 164840.0 4960.0 0.34 162560.0 3340.0 0.25 0.4151 0.9886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G04 mock treatment 167440.0 7560.0 0.52 165680.0 6460.0 0.48 0.7046 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G05 compound treatment 190240.0 30400.0 2.07 180920.0 21700.0 1.62 2.6058 0.9925 DHPC8.2_000063 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G06 compound treatment 185200.0 25300.0 1.73 184760.0 25500.0 1.9 2.5649 0.9988 DHPC8.2_000064 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G07 compound treatment 169840.0 9960.0 0.68 170120.0 10900.0 0.81 1.054 0.9961 DHPC8.2_000065 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G08 compound treatment 168600.0 8720.0 0.59 166200.0 6980.0 0.52 0.7879 0.9978 DHPC8.2_000066 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G09 compound treatment 168880.0 9000.0 0.61 166000.0 6780.0 0.5 0.7909 0.9953 DHPC8.2_000067 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G10 compound treatment 164880.0 5000.0 0.34 162480.0 3260.0 0.24 0.4128 0.9862 DHPC8.2_000068 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G11 compound treatment 167600.0 7720.0 0.53 169240.0 10000.0 0.75 0.8997 0.9854 DHPC8.2_000069 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G12 compound treatment 168480.0 8600.0 0.59 167240.0 8020.0 0.6 0.8368 1.0 DHPC8.2_000070 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G13 compound treatment 174640.0 14800.0 1.01 174880.0 15700.0 1.17 1.5359 0.9973 DHPC8.2_000071 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G14 compound treatment 167440.0 7560.0 0.52 168960.0 9740.0 0.73 0.8772 0.986 DHPC8.2_000072 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G15 compound treatment 172880.0 13000.0 0.89 169640.0 10400.0 0.78 1.1753 0.9978 DHPC8.2_000073 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G16 compound treatment 175040.0 15200.0 1.03 173200.0 14000.0 1.04 1.4668 1.0 DHPC8.2_000074 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G17 compound treatment 166160.0 6280.0 0.43 168160.0 8940.0 0.67 0.7734 0.9773 DHPC8.2_000075 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G18 compound treatment 164560.0 4680.0 0.32 165560.0 6340.0 0.47 0.5595 0.9818 DHPC8.2_000076 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G19 mock treatment 168160.0 8280.0 0.56 165120.0 5900.0 0.44 0.7099 0.9923 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G20 mock treatment 161200.0 1320.0 0.09 162920.0 3700.0 0.28 0.2585 0.8918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G21 compound treatment 166000.0 6120.0 0.42 162600.0 3380.0 0.25 0.4731 0.9707 DHPC8.2_000077 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G22 compound treatment 158640.0 -1240.0 -0.08 161360.0 2140.0 0.16 0.053 0.2938 DHPC8.2_000078 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G23 compound treatment 171480.0 11600.0 0.79 169320.0 10100.0 0.75 1.0909 0.9997 DHPC8.2_000079 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 G24 mock treatment 160240.0 361.0 0.02 153280.0 -5940.0 -0.44 -0.2951 -0.6667 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H01 mock treatment 163120.0 3240.0 0.22 160360.0 1140.0 0.09 0.2164 0.9139 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H02 mock treatment 163560.0 3680.0 0.25 160360.0 1140.0 0.09 0.2376 0.8966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H03 mock treatment 164280.0 4400.0 0.3 164120.0 4900.0 0.36 0.4702 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H04 mock treatment 166360.0 6480.0 0.44 162680.0 3460.0 0.26 0.4947 0.9671 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H05 mock treatment 160760.0 881.0 0.06 163520.0 4300.0 0.32 0.2689 0.8253 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H06 mock treatment 163760.0 3880.0 0.26 165840.0 6620.0 0.49 0.5356 0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H07 mock treatment 165320.0 5440.0 0.37 167440.0 8220.0 0.61 0.695 0.9712 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H08 mock treatment 168960.0 9080.0 0.62 164760.0 5540.0 0.41 0.7295 0.9805 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H09 mock treatment 167560.0 7680.0 0.52 162920.0 3700.0 0.28 0.5651 0.955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H10 mock treatment 163440.0 3560.0 0.24 164560.0 5340.0 0.4 0.4528 0.972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H11 mock treatment 165080.0 5200.0 0.35 164320.0 5100.0 0.38 0.5193 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H12 mock treatment 164040.0 4160.0 0.28 163160.0 3940.0 0.29 0.4081 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H13 mock treatment 166560.0 6680.0 0.46 167920.0 8700.0 0.65 0.7801 0.9852 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H14 mock treatment 163360.0 3480.0 0.24 163160.0 3940.0 0.29 0.3753 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H15 mock treatment 164440.0 4560.0 0.31 161920.0 2700.0 0.2 0.3621 0.9778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H16 mock treatment 162880.0 3000.0 0.2 164600.0 5380.0 0.4 0.4279 0.9513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H17 mock treatment 164160.0 4280.0 0.29 161160.0 1940.0 0.14 0.3086 0.9475 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H18 mock treatment 164040.0 4160.0 0.28 162840.0 3620.0 0.27 0.3912 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H19 mock treatment 162640.0 2760.0 0.19 159800.0 583.0 0.04 0.1638 0.8478 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H20 mock treatment 159960.0 80.9 0.01 160880.0 1660.0 0.12 0.0914 0.7379 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H21 mock treatment 158880.0 -999.0 -0.07 156200.0 -3020.0 -0.22 -0.207 -0.8819 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H22 mock treatment 159640.0 -239.0 -0.02 157520.0 -1700.0 -0.13 -0.1009 -0.7918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H23 mock treatment 153560.0 -6320.0 -0.43 157000.0 -2220.0 -0.17 -0.4213 -0.9133 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 H24 mock treatment 153440.0 -6440.0 -0.44 148560.0 -10700.0 -0.79 -0.8713 -0.9611 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I01 compound treatment 163440.0 3560.0 0.24 159800.0 583.0 0.04 0.2023 0.8204 DHPC8.2_000080 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I02 mock treatment 162240.0 2360.0 0.16 163720.0 4500.0 0.34 0.3508 0.9435 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I03 compound treatment 161160.0 1280.0 0.09 161000.0 1780.0 0.13 0.1556 0.9794 DHPC8.2_000081 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I04 mock treatment 163880.0 4000.0 0.27 163520.0 4300.0 0.32 0.4193 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I05 mock treatment 168840.0 8960.0 0.61 163480.0 4260.0 0.32 0.6563 0.9534 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I06 mock treatment 164840.0 4960.0 0.34 163040.0 3820.0 0.28 0.4403 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I07 compound treatment 166160.0 6280.0 0.43 166680.0 7460.0 0.56 0.6955 0.9917 DHPC8.2_000082 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I08 mock treatment 166120.0 6240.0 0.43 163800.0 4580.0 0.34 0.542 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I09 compound treatment 172360.0 12500.0 0.85 164960.0 5740.0 0.43 0.9039 0.9493 DHPC8.2_000083 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I10 mock treatment 167920.0 8040.0 0.55 160200.0 983.0 0.07 0.4394 0.7944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I11 compound treatment 170040.0 10200.0 0.69 165600.0 6380.0 0.48 0.8257 0.9831 DHPC8.2_000084 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I12 mock treatment 180240.0 20400.0 1.39 165000.0 5780.0 0.43 1.2859 0.8848 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I13 compound treatment 197760.0 37900.0 2.58 197160.0 37900.0 2.82 3.823 0.999 DHPC8.2_000085 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I14 mock treatment 166600.0 6720.0 0.46 165960.0 6740.0 0.5 0.6789 0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I15 compound treatment 195280.0 35400.0 2.41 185560.0 26300.0 1.96 3.093 0.9947 DHPC8.2_000086 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I16 mock treatment 166720.0 6840.0 0.47 163240.0 4020.0 0.3 0.5415 0.977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I17 compound treatment 164760.0 4880.0 0.33 167400.0 8180.0 0.61 0.6659 0.9596 DHPC8.2_000087 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I18 mock treatment 159520.0 -359.0 -0.02 163240.0 4020.0 0.3 0.1944 0.6471 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I19 compound treatment 166600.0 6720.0 0.46 164920.0 5700.0 0.42 0.6241 0.9993 DHPC8.2_000088 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I20 mock treatment 158840.0 -1040.0 -0.07 159160.0 -57.4 0.0 -0.0531 -0.7484 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I21 mock treatment 160600.0 721.0 0.05 159840.0 623.0 0.05 0.0675 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I22 mock treatment 158200.0 -1680.0 -0.11 159400.0 183.0 0.01 -0.0713 -0.6188 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I23 compound treatment 150560.0 -9320.0 -0.64 156880.0 -2340.0 -0.17 -0.5723 -0.8687 DHPC8.2_000089 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 I24 mock treatment 148520.0 -11400.0 -0.77 152280.0 -6940.0 -0.52 -0.9127 -0.9806 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J01 mock treatment 158040.0 -1840.0 -0.13 157920.0 -1300.0 -0.1 -0.1569 -0.9917 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J02 mock treatment 156800.0 -3080.0 -0.21 160840.0 1620.0 0.12 -0.063 -0.2603 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J03 mock treatment 161040.0 1160.0 0.08 160200.0 983.0 0.07 0.1077 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J04 mock treatment 165200.0 5320.0 0.36 166760.0 7540.0 0.56 0.6535 0.9777 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J05 mock treatment 161640.0 1760.0 0.12 163320.0 4100.0 0.31 0.3008 0.9168 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J06 mock treatment 166080.0 6200.0 0.42 165640.0 6420.0 0.48 0.6369 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J07 mock treatment 165800.0 5920.0 0.4 160960.0 1740.0 0.13 0.3771 0.8895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J08 mock treatment 164920.0 5040.0 0.34 163480.0 4260.0 0.32 0.4673 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J09 mock treatment 164480.0 4600.0 0.31 161160.0 1940.0 0.14 0.324 0.9382 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J10 mock treatment 165720.0 5840.0 0.4 164920.0 5700.0 0.42 0.5817 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J11 mock treatment 162800.0 2920.0 0.2 162960.0 3740.0 0.28 0.3378 0.9865 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J12 mock treatment 165080.0 5200.0 0.35 161520.0 2300.0 0.17 0.3719 0.9444 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J13 mock treatment 166920.0 7040.0 0.48 162560.0 3340.0 0.25 0.5153 0.9532 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J14 mock treatment 162680.0 2800.0 0.19 168000.0 8780.0 0.65 0.5972 0.877 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J15 mock treatment 164760.0 4880.0 0.33 164120.0 4900.0 0.36 0.4933 0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J16 mock treatment 159720.0 -159.0 -0.01 160040.0 823.0 0.06 0.0356 0.5729 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J17 mock treatment 159280.0 -599.0 -0.04 168040.0 8820.0 0.66 0.4354 0.6618 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J18 mock treatment 164680.0 4800.0 0.33 165760.0 6540.0 0.49 0.5758 0.9813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J19 mock treatment 160080.0 201.0 0.01 166840.0 7620.0 0.57 0.4108 0.724 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J20 mock treatment 159640.0 -239.0 -0.02 160040.0 823.0 0.06 0.0318 0.5014 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J21 mock treatment 157120.0 -2760.0 -0.19 158240.0 -977.0 -0.07 -0.1844 -0.9145 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J22 mock treatment 152560.0 -7320.0 -0.5 152920.0 -6300.0 -0.47 -0.6843 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J23 mock treatment 154440.0 -5440.0 -0.37 153400.0 -5820.0 -0.43 -0.5684 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 J24 mock treatment 147560.0 -12300.0 -0.84 147400.0 -11800.0 -0.88 -1.2158 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K01 compound treatment 164920.0 5040.0 0.34 159160.0 -57.4 0.0 0.24 0.6983 DHPC8.2_000090 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K02 mock treatment 165000.0 5120.0 0.35 157440.0 -1780.0 -0.13 0.1533 0.4107 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K03 compound treatment 162120.0 2240.0 0.15 159760.0 543.0 0.04 0.1366 0.8643 DHPC8.2_000091 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K04 mock treatment 167600.0 7720.0 0.53 161360.0 2140.0 0.16 0.485 0.8818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K05 compound treatment 163600.0 3720.0 0.25 164640.0 5420.0 0.4 0.4648 0.975 DHPC8.2_000092 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K06 mock treatment 164280.0 4400.0 0.3 161240.0 2020.0 0.15 0.3186 0.9491 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K07 mock treatment 165080.0 5200.0 0.35 164520.0 5300.0 0.39 0.5298 0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K08 mock treatment 163880.0 4000.0 0.27 157960.0 -1260.0 -0.09 0.1267 0.4394 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K09 compound treatment 170320.0 10400.0 0.71 167760.0 8540.0 0.64 0.9529 0.9984 DHPC8.2_000093 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K10 mock treatment 166600.0 6720.0 0.46 164040.0 4820.0 0.36 0.5778 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K11 compound treatment 175200.0 15300.0 1.04 171320.0 12100.0 0.9 1.3755 0.9973 DHPC8.2_000094 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K12 mock treatment 163520.0 3640.0 0.25 166760.0 7540.0 0.56 0.5725 0.9327 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K13 compound treatment 178800.0 18900.0 1.29 175120.0 15900.0 1.18 1.7491 0.9991 DHPC8.2_000095 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K14 mock treatment 168360.0 8480.0 0.58 167000.0 7780.0 0.58 0.8184 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K15 mock treatment 165320.0 5440.0 0.37 166480.0 7260.0 0.54 0.6445 0.9831 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K16 mock treatment 163160.0 3280.0 0.22 164960.0 5740.0 0.43 0.4604 0.9544 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K17 compound treatment 173720.0 13800.0 0.94 172160.0 12900.0 0.96 1.3484 0.9999 DHPC8.2_000096 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K18 mock treatment 161840.0 1960.0 0.13 159480.0 263.0 0.02 0.1084 0.802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K19 compound treatment 167400.0 7520.0 0.51 171240.0 12000.0 0.89 0.9953 0.9651 DHPC8.2_000097 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K20 mock treatment 160080.0 201.0 0.01 163680.0 4460.0 0.33 0.2445 0.7356 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K21 compound treatment 161400.0 1520.0 0.1 156240.0 -2980.0 -0.22 -0.0834 -0.3408 DHPC8.2_000098 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K22 mock treatment 158320.0 -1560.0 -0.11 158920.0 -297.0 -0.02 -0.0908 -0.8364 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K23 mock treatment 155160.0 -4720.0 -0.32 153520.0 -5700.0 -0.42 -0.5273 -0.9907 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 K24 mock treatment 148840.0 -11000.0 -0.75 153280.0 -5940.0 -0.44 -0.8446 -0.9678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L01 mock treatment 160800.0 921.0 0.06 157440.0 -1780.0 -0.13 -0.0491 -0.3356 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L02 mock treatment 162560.0 2680.0 0.18 160360.0 1140.0 0.09 0.1894 0.9394 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L03 mock treatment 161320.0 1440.0 0.1 161080.0 1860.0 0.14 0.1675 0.9858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L04 mock treatment 164760.0 4880.0 0.33 162680.0 3460.0 0.26 0.4175 0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L05 mock treatment 162480.0 2600.0 0.18 167520.0 8300.0 0.62 0.5623 0.8747 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L06 mock treatment 162520.0 2640.0 0.18 166960.0 7740.0 0.58 0.5348 0.8858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L07 mock treatment 165120.0 5240.0 0.36 162160.0 2940.0 0.22 0.4075 0.9724 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L08 mock treatment 165320.0 5440.0 0.37 162520.0 3300.0 0.25 0.4361 0.98 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L09 mock treatment 166160.0 6280.0 0.43 162040.0 2820.0 0.21 0.4513 0.9463 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L10 mock treatment 166440.0 6560.0 0.45 164080.0 4860.0 0.36 0.5722 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L11 mock treatment 167160.0 7280.0 0.5 161000.0 1780.0 0.13 0.4448 0.8657 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L12 mock treatment 167240.0 7360.0 0.5 163400.0 4180.0 0.31 0.575 0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L13 mock treatment 162880.0 3000.0 0.2 162720.0 3500.0 0.26 0.329 0.9928 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L14 mock treatment 162200.0 2320.0 0.16 164200.0 4980.0 0.37 0.3741 0.9279 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L15 mock treatment 166760.0 6880.0 0.47 164600.0 5380.0 0.4 0.615 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L16 mock treatment 160960.0 1080.0 0.07 164560.0 5340.0 0.4 0.3333 0.8241 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L17 mock treatment 159800.0 -79.1 -0.01 166920.0 7700.0 0.57 0.4016 0.7004 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L18 mock treatment 163840.0 3960.0 0.27 159400.0 183.0 0.01 0.2006 0.7418 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L19 mock treatment 157880.0 -2000.0 -0.14 162840.0 3620.0 0.27 0.0943 0.3121 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L20 mock treatment 159920.0 40.9 0.0 154200.0 -5020.0 -0.37 -0.2621 -0.7018 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L21 mock treatment 152760.0 -7120.0 -0.49 158280.0 -937.0 -0.07 -0.3925 -0.8005 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L22 mock treatment 149760.0 -10100.0 -0.69 154840.0 -4380.0 -0.33 -0.7182 -0.9413 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L23 mock treatment 152080.0 -7800.0 -0.53 155280.0 -3940.0 -0.29 -0.5832 -0.9606 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 L24 mock treatment 148480.0 -11400.0 -0.78 146120.0 -13100.0 -0.97 -1.2388 -0.9937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M01 compound treatment 160960.0 1080.0 0.07 162360.0 3140.0 0.23 0.2175 0.8869 DHPC8.2_000099 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M02 mock treatment 162560.0 2680.0 0.18 164880.0 5660.0 0.42 0.4273 0.9301 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M03 compound treatment 165880.0 6000.0 0.41 160800.0 1580.0 0.12 0.3726 0.8751 DHPC8.2_000100 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M04 mock treatment 167160.0 7280.0 0.5 167280.0 8060.0 0.6 0.7753 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M05 compound treatment 171120.0 11200.0 0.77 176600.0 17400.0 1.29 1.4567 0.9688 DHPC8.2_000101 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M06 mock treatment 175320.0 15400.0 1.05 170640.0 11400.0 0.85 1.3455 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M07 compound treatment 204640.0 44800.0 3.05 199400.0 40200.0 2.99 4.2726 0.9999 DHPC8.2_000102 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M08 mock treatment 171720.0 11800.0 0.81 169320.0 10100.0 0.75 1.1025 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M09 mock treatment 171960.0 12100.0 0.82 169720.0 10500.0 0.78 1.1351 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M10 mock treatment 171520.0 11600.0 0.79 169680.0 10500.0 0.78 1.1118 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M11 compound treatment 179720.0 19800.0 1.35 172680.0 13500.0 1.0 1.665 0.9891 DHPC8.2_000103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M12 mock treatment 169400.0 9520.0 0.65 168200.0 8980.0 0.67 0.9317 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M13 mock treatment 169320.0 9440.0 0.64 169800.0 10600.0 0.79 1.0121 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M14 mock treatment 164960.0 5080.0 0.35 165360.0 6140.0 0.46 0.5682 0.9906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M15 compound treatment 168520.0 8640.0 0.59 166000.0 6780.0 0.5 0.7735 0.997 DHPC8.2_000104 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M16 mock treatment 163520.0 3640.0 0.25 167360.0 8140.0 0.61 0.6041 0.9224 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M17 compound treatment 172520.0 12600.0 0.86 170880.0 11700.0 0.87 1.2232 1.0 DHPC8.2_000105 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M18 mock treatment 165680.0 5800.0 0.4 165760.0 6540.0 0.49 0.624 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M19 compound treatment 171280.0 11400.0 0.78 173160.0 13900.0 1.04 1.2834 0.9899 DHPC8.2_000106 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M20 mock treatment 163120.0 3240.0 0.22 164040.0 4820.0 0.36 0.41 0.9728 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M21 compound treatment 199560.0 39700.0 2.71 194400.0 35200.0 2.62 3.7645 0.9999 DHPC8.2_000107 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M22 mock treatment 163120.0 3240.0 0.22 158400.0 -817.0 -0.06 0.1132 0.494 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M23 compound treatment 163400.0 3520.0 0.24 167840.0 8620.0 0.64 0.6235 0.91 DHPC8.2_000108 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 M24 mock treatment 155720.0 -4160.0 -0.28 153520.0 -5700.0 -0.42 -0.5003 -0.9809 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N01 mock treatment 160560.0 681.0 0.05 161440.0 2220.0 0.17 0.1498 0.8719 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N02 mock treatment 160920.0 1040.0 0.07 163560.0 4340.0 0.32 0.2787 0.8423 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N03 mock treatment 158440.0 -1440.0 -0.1 160160.0 943.0 0.07 -0.0198 -0.1639 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N04 mock treatment 162960.0 3080.0 0.21 160520.0 1300.0 0.1 0.2171 0.9384 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N05 mock treatment 166240.0 6360.0 0.43 161760.0 2540.0 0.19 0.4405 0.9309 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N06 mock treatment 165640.0 5760.0 0.39 167640.0 8420.0 0.63 0.721 0.9746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N07 mock treatment 165080.0 5200.0 0.35 170040.0 10800.0 0.81 0.8203 0.9321 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N08 mock treatment 164880.0 5000.0 0.34 167400.0 8180.0 0.61 0.6717 0.9624 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N09 mock treatment 170160.0 10300.0 0.7 173400.0 14200.0 1.06 1.242 0.9802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N10 mock treatment 175400.0 15500.0 1.06 175680.0 16500.0 1.23 1.6146 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N11 mock treatment 172400.0 12500.0 0.85 170560.0 11300.0 0.84 1.2006 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N12 mock treatment 163880.0 4000.0 0.27 168560.0 9340.0 0.7 0.6846 0.9165 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N13 mock treatment 165960.0 6080.0 0.41 171640.0 12400.0 0.92 0.9469 0.9345 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N14 mock treatment 168400.0 8520.0 0.58 164240.0 5020.0 0.37 0.6751 0.9773 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N15 mock treatment 164920.0 5040.0 0.34 167400.0 8180.0 0.61 0.6736 0.9633 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N16 mock treatment 162760.0 2880.0 0.2 164800.0 5580.0 0.42 0.4327 0.9415 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N17 mock treatment 166040.0 6160.0 0.42 166720.0 7500.0 0.56 0.6919 0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N18 mock treatment 159680.0 -199.0 -0.01 162800.0 3580.0 0.27 0.1789 0.6702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N19 mock treatment 161560.0 1680.0 0.11 163720.0 4500.0 0.34 0.318 0.8979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N20 mock treatment 162760.0 2880.0 0.2 161880.0 2660.0 0.2 0.279 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N21 mock treatment 160280.0 401.0 0.03 162920.0 3700.0 0.28 0.2142 0.7734 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N22 mock treatment 156040.0 -3840.0 -0.26 161240.0 2020.0 0.15 -0.0786 -0.2604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N23 mock treatment 158000.0 -1880.0 -0.13 154640.0 -4580.0 -0.34 -0.3315 -0.9107 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 N24 mock treatment 154840.0 -5040.0 -0.34 152600.0 -6620.0 -0.49 -0.5912 -0.9845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O01 compound treatment 197680.0 37800.0 2.58 161200.0 1980.0 0.15 1.9267 0.7464 DHPC8.2_000109 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O02 mock treatment 157880.0 -2000.0 -0.14 163720.0 4500.0 0.34 0.1406 0.3886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O03 compound treatment 155280.0 -4600.0 -0.31 165360.0 6140.0 0.46 0.1016 0.1832 DHPC8.2_000110 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O04 mock treatment 154480.0 -5400.0 -0.37 163560.0 4340.0 0.32 -0.0317 -0.0648 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O05 compound treatment 162560.0 2680.0 0.18 163920.0 4700.0 0.35 0.3767 0.9541 DHPC8.2_000111 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O06 mock treatment 166320.0 6440.0 0.44 166200.0 6980.0 0.52 0.678 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O07 compound treatment 167120.0 7240.0 0.49 167200.0 7980.0 0.59 0.7692 0.9958 DHPC8.2_000112 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O08 mock treatment 162400.0 2520.0 0.17 168960.0 9740.0 0.73 0.6343 0.8511 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O09 compound treatment 200120.0 40200.0 2.74 202600.0 43400.0 3.23 4.2231 0.9967 DHPC8.2_000113 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O10 mock treatment 165760.0 5880.0 0.4 166160.0 6940.0 0.52 0.6489 0.9921 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O11 mock treatment 164720.0 4840.0 0.33 167000.0 7780.0 0.58 0.643 0.9644 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O12 mock treatment 163240.0 3360.0 0.23 165600.0 6380.0 0.48 0.4979 0.9441 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O13 compound treatment 173880.0 14000.0 0.95 170800.0 11600.0 0.86 1.2845 0.9987 DHPC8.2_000114 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O14 mock treatment 164640.0 4760.0 0.32 161440.0 2220.0 0.17 0.3465 0.9511 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O15 compound treatment 187080.0 27200.0 1.85 193080.0 33900.0 2.52 3.0934 0.9886 DHPC8.2_000115 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O16 mock treatment 166680.0 6800.0 0.46 163640.0 4420.0 0.33 0.5606 0.9859 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O17 compound treatment 190880.0 31000.0 2.11 187240.0 28000.0 2.09 2.9693 1.0 DHPC8.2_000116 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O18 mock treatment 164160.0 4280.0 0.29 162440.0 3220.0 0.24 0.376 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O19 compound treatment 163160.0 3280.0 0.22 166640.0 7420.0 0.55 0.5488 0.9208 DHPC8.2_000117 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O20 mock treatment 161600.0 1720.0 0.12 162160.0 2940.0 0.22 0.2378 0.9572 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O21 compound treatment 183320.0 23400.0 1.6 183200.0 24000.0 1.78 2.3922 0.9985 DHPC8.2_000118 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O22 mock treatment 155480.0 -4400.0 -0.3 152440.0 -6780.0 -0.5 -0.5688 -0.9692 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O23 compound treatment 189640.0 29800.0 2.03 178840.0 19600.0 1.46 2.4674 0.987 DHPC8.2_000119 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 O24 mock treatment 153720.0 -6160.0 -0.42 150600.0 -8620.0 -0.64 -0.7504 -0.9789 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P01 mock treatment 161000.0 1120.0 0.08 160280.0 1060.0 0.08 0.11 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P02 mock treatment 159160.0 -719.0 -0.05 161680.0 2460.0 0.18 0.0949 0.5004 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P03 mock treatment 157680.0 -2200.0 -0.15 160880.0 1660.0 0.12 -0.0185 -0.0952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P04 mock treatment 157840.0 -2040.0 -0.14 160640.0 1420.0 0.11 -0.0234 -0.1341 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P05 mock treatment 158920.0 -959.0 -0.07 156680.0 -2540.0 -0.19 -0.1798 -0.8995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P06 mock treatment 164360.0 4480.0 0.31 164640.0 5420.0 0.4 0.5014 0.9906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P07 mock treatment 161360.0 1480.0 0.1 161800.0 2580.0 0.19 0.2073 0.9548 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P08 mock treatment 164440.0 4560.0 0.31 163120.0 3900.0 0.29 0.4253 0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P09 mock treatment 162880.0 3000.0 0.2 165520.0 6300.0 0.47 0.4764 0.9308 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P10 mock treatment 162040.0 2160.0 0.15 157040.0 -2180.0 -0.16 -0.0104 -0.0476 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P11 mock treatment 160600.0 721.0 0.05 163640.0 4420.0 0.33 0.2675 0.8038 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P12 mock treatment 161480.0 1600.0 0.11 161800.0 2580.0 0.19 0.2131 0.964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P13 mock treatment 159880.0 0.909 0.0 161160.0 1940.0 0.14 0.1023 0.7074 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P14 mock treatment 159920.0 40.9 0.0 161000.0 1780.0 0.13 0.0958 0.7218 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P15 mock treatment 162760.0 2880.0 0.2 161120.0 1900.0 0.14 0.239 0.9871 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P16 mock treatment 164200.0 4320.0 0.29 156680.0 -2540.0 -0.19 0.0748 0.2137 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P17 mock treatment 163320.0 3440.0 0.23 163880.0 4660.0 0.35 0.4113 0.9818 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P18 mock treatment 158680.0 -1200.0 -0.08 161320.0 2100.0 0.16 0.0529 0.2993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P19 mock treatment 156560.0 -3320.0 -0.23 156040.0 -3180.0 -0.24 -0.3272 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P20 mock treatment 156120.0 -3760.0 -0.26 153000.0 -6220.0 -0.46 -0.5084 -0.9612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P21 mock treatment 155720.0 -4160.0 -0.28 152520.0 -6700.0 -0.5 -0.553 -0.9643 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P22 mock treatment 157720.0 -2160.0 -0.15 151080.0 -8140.0 -0.61 -0.5323 -0.8541 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P23 mock treatment 156320.0 -3560.0 -0.24 151400.0 -7820.0 -0.58 -0.583 -0.9248 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2412 P24 mock treatment 152080.0 -7800.0 -0.53 149240.0 -9980.0 -0.74 -0.9011 -0.9866 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A01 compound treatment 166240.0 19300.0 1.32 162880.0 17300.0 1.29 1.8428 0.9999 1913656 CBChromo1_000001 COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A02 compound treatment 154080.0 7180.0 0.49 150040.0 4460.0 0.33 0.5808 0.9822 1920364 CBChromo1_000002 C1CCc2c(C1)sc3ncnc(N/N=C\c4ccc(cc4)c5ccccc5)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A03 compound treatment 147400.0 498.0 0.03 144680.0 -899.0 -0.07 -0.0233 -0.3109 1912983 CBChromo1_000003 O=C(Cc1ccccc1)NNc2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A04 compound treatment 152480.0 5580.0 0.38 150640.0 5060.0 0.38 0.5352 1.0 538 CBChromo1_000004 CC(CCc1ccccc1)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A05 compound treatment 170360.0 23500.0 1.6 163160.0 17600.0 1.31 2.0561 0.995 1912573 CBChromo1_000005 NC(=N)SCc1ccccc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A06 compound treatment 140440.0 -6460.0 -0.44 140000.0 -5580.0 -0.42 -0.6051 -0.9996 1244471 CBChromo1_000006 CCN(CC)CC(O)COc1ccc(cc1)C2(CC3CC4CC(C3)C2)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A07 compound treatment 162440.0 15500.0 1.06 157000.0 11400.0 0.85 1.3501 0.994 1913686 CBChromo1_000007 OC(=O)/C=C/C(=O)Nc1cccc2c(NC(=O)\C=C\C(=O)O)cccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A08 compound treatment 168200.0 21300.0 1.45 168560.0 23000.0 1.71 2.2362 0.9967 1699574 CBChromo1_000008 CN1C(N(C)c2ccccc12)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A09 compound treatment 197680.0 50800.0 3.46 185520.0 39900.0 2.97 4.5499 0.9971 1918598 CBChromo1_000009 COc1cccc(/C=N\Nc2ccccn2)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A10 compound treatment 148960.0 2060.0 0.14 149920.0 4340.0 0.32 0.3277 0.9302 1917942 CBChromo1_000010 CCOC(=O)c1c(C)c(C)sc1NC(=O)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A11 compound treatment 149720.0 2820.0 0.19 149720.0 4140.0 0.31 0.3538 0.9741 1913101 CBChromo1_000011 N=c1ccn(CC(=O)c2ccc(cc2)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A12 compound treatment 352200.0 205000.0 14.0 354600.0 209000.0 15.56 20.8974 0.9986 1002707 CBChromo1_000012 Oc1cc(cc2cc(NC(=O)Nc3ccc4c(O)cc(cc4c3)S(=O)(=O)O)ccc12)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A13 compound treatment 200680.0 53800.0 3.67 194200.0 48600.0 3.62 5.1514 1.0 1917324 CBChromo1_000013 Cc1cc(Br)cc(C)c1OCC(=O)N/N=C/c2cc(Br)c(O)c(Br)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A14 compound treatment 167840.0 20900.0 1.43 165920.0 20300.0 1.51 2.0799 0.9996 1392413 CBChromo1_000014 CN(C)c1cccc(c1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A15 compound treatment 235800.0 88900.0 6.06 219480.0 73900.0 5.5 8.1749 0.9988 1914233 CBChromo1_000015 Oc1c(Br)cc(cc1Br)S(=O)(=O)c2cc(Br)c(OCC=C)c(Br)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A16 compound treatment 151000.0 4100.0 0.28 151120.0 5540.0 0.41 0.4892 0.982 1924027 CBChromo1_000016 COc1ccc(OC)c(/C=C/C(=O)c2c(c3ccccc3)c4cc(Br)ccc4[nH]c2=O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A17 compound treatment 202520.0 55600.0 3.79 206640.0 61100.0 4.54 5.8947 0.9959 1031871 CBChromo1_000017 Oc1ccc(Cl)cc1Cc2cc(Cl)cc(Cc3cc(Cl)ccc3O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A18 compound treatment 149440.0 2540.0 0.17 141360.0 -4220.0 -0.31 -0.0997 -0.2781 1933148 CBChromo1_000018 Cc1ccc(cc1NS(=O)(=O)c2ccccc2)c3nc4cc(Cl)ccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A19 compound treatment 153680.0 6780.0 0.46 150760.0 5180.0 0.39 0.5994 0.996 1916017 CBChromo1_000019 Nc1ccc(cc1)c2cnc(nc2)c3ccc(N)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A20 compound treatment 146040.0 -863.0 -0.06 146040.0 461.0 0.03 -0.0173 -0.2542 1308836 CBChromo1_000020 Cc1cc(C)c(NC(=O)COc2cccc(Br)c2)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A21 compound treatment 156360.0 9460.0 0.64 151160.0 5580.0 0.42 0.7497 0.9774 1918845 CBChromo1_000021 Oc1ccccc1C(=O)N/N=C/c2cc3OCOc3cc2[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A22 compound treatment 143160.0 -3740.0 -0.26 143560.0 -2020.0 -0.15 -0.2867 -0.9681 1428952 CBChromo1_000022 COc1ccc(Cl)cc1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A23 mock treatment 142080.0 -4820.0 -0.33 142160.0 -3420.0 -0.25 -0.4124 -0.992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 A24 mock treatment 141240.0 -5660.0 -0.39 139000.0 -6580.0 -0.49 -0.6192 -0.9931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B01 compound treatment 139760.0 -7140.0 -0.49 138680.0 -6900.0 -0.51 -0.7074 -0.9996 1913438 CBChromo1_000023 [O-][N+](=O)c1ccc(/C=N/NC(=O)c2ccncc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B02 compound treatment 145040.0 -1860.0 -0.13 139720.0 -5860.0 -0.44 -0.3981 -0.8766 1192620 CBChromo1_000024 Clc1ccc(OCC(=O)N2CC(CC2=O)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B03 compound treatment 147440.0 538.0 0.04 138000.0 -7580.0 -0.56 -0.3729 -0.6598 1920508 CBChromo1_000025 Cc1ccc(cc1)S(=O)(=O)NC2=C(C(=O)c3ccccc3C2=O)[n+]4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B04 compound treatment 145120.0 -1780.0 -0.12 141040.0 -4540.0 -0.34 -0.3248 -0.9047 1923167 CBChromo1_000026 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(I)cc4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B05 compound treatment 153360.0 6460.0 0.44 156000.0 10400.0 0.78 0.8598 0.964 1041351 CBChromo1_000027 CN(C)Cc1c[nH]c2cc(ccc12)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B06 compound treatment 156000.0 9100.0 0.62 161200.0 15600.0 1.16 1.2607 0.9567 1921966 CBChromo1_000028 Brc1ccccc1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B07 compound treatment 149440.0 2540.0 0.17 148720.0 3140.0 0.23 0.2876 0.989 1913597 CBChromo1_000029 COc1ccccc1C2CC(=NN2c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B08 compound treatment 145440.0 -1460.0 -0.1 146080.0 501.0 0.04 -0.0441 -0.4145 1128878 CBChromo1_000030 COc1ccc(cc1OC)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B09 compound treatment 147360.0 458.0 0.03 144000.0 -1580.0 -0.12 -0.061 -0.502 1918866 CBChromo1_000031 [O-][N+](=O)c1ccc(OC(=O)CN2C(=O)c3ccccc3C2=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B10 compound treatment 144840.0 -2060.0 -0.14 144000.0 -1580.0 -0.12 -0.1825 -0.996 1496608 CBChromo1_000032 CCOc1ccc(cc1OC)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B11 compound treatment 144440.0 -2460.0 -0.17 144040.0 -1540.0 -0.11 -0.1997 -0.9826 1086418 CBChromo1_000033 ClCC(=O)Nc1ccc(Br)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B12 compound treatment 148920.0 2020.0 0.14 147120.0 1540.0 0.11 0.1784 0.9959 1207865 CBChromo1_000034 Cc1ccc(o1)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B13 compound treatment 152440.0 5540.0 0.38 153360.0 7780.0 0.58 0.6765 0.9785 1626895 CBChromo1_000035 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(OCc5ccc(F)cc5)cc4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B14 compound treatment 145880.0 -1020.0 -0.07 145840.0 261.0 0.02 -0.0355 -0.4911 1931161 CBChromo1_000036 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4c(O)ccc5ccccc45)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B15 compound treatment 144560.0 -2340.0 -0.16 141040.0 -4540.0 -0.34 -0.3518 -0.9415 1140129 CBChromo1_000037 Cc1ccc(C)c(OCC(=O)Nc2c(C)cc(C)cc2C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B16 compound treatment 147120.0 218.0 0.01 145600.0 21.3 0.0 0.0116 0.7781 1918161 CBChromo1_000038 CCCCCC(=O)N/N=C/c1ccc2cc(OC)ccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B17 compound treatment 146080.0 -823.0 -0.06 142720.0 -2860.0 -0.21 -0.1901 -0.864 3624409 CBChromo1_000039 Cc1cccc(COc2ccc(cc2)C3C4=C(CC(C)(C)CC4=O)OC5=C3C(=O)CC(C)(C)C5)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B18 compound treatment 148880.0 1980.0 0.13 138880.0 -6700.0 -0.5 -0.2572 -0.498 1152708 CBChromo1_000040 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nc4ccccc4[nH]c3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B19 compound treatment 144840.0 -2060.0 -0.14 143320.0 -2260.0 -0.17 -0.2183 -0.9961 3624410 CBChromo1_000041 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B20 compound treatment 165200.0 18300.0 1.25 163480.0 17900.0 1.33 1.8242 0.9995 1589883 CBChromo1_000042 Cc1cccc(c1)c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B21 compound treatment 142880.0 -4020.0 -0.27 143680.0 -1900.0 -0.14 -0.2938 -0.9525 3624411 CBChromo1_000043 COc1ccc(NC(CC(=O)c2ccc(Br)cc2)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B22 compound treatment 140640.0 -6260.0 -0.43 140360.0 -5220.0 -0.39 -0.5766 -0.9989 3624412 CBChromo1_000044 C[C@@H](O)[C@@H]1OC1/C=C/[C@@H]2O[C@H]2[C@H](O)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B23 mock treatment 141320.0 -5580.0 -0.38 136360.0 -9220.0 -0.69 -0.7543 -0.9613 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 B24 mock treatment 140240.0 -6660.0 -0.45 137800.0 -7780.0 -0.58 -0.7306 -0.9928 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C01 compound treatment 175320.0 28400.0 1.94 171160.0 25600.0 1.9 2.7162 1.0 1921774 CBChromo1_000045 CC/C(=C/c1sc2ccc3ccccc3c2[n+]1C)/SC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C02 compound treatment 169960.0 23100.0 1.57 161000.0 15400.0 1.15 1.9231 0.9881 1920309 CBChromo1_000046 Oc1ccc(/C=N/Nc2ncnc3sc4CCCCc4c23)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C03 compound treatment 151560.0 4660.0 0.32 149080.0 3500.0 0.26 0.4088 0.9952 1010154 CBChromo1_000047 CC(NC(=O)CCl)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C04 compound treatment 151720.0 4820.0 0.33 151400.0 5820.0 0.43 0.5386 0.9907 1121247 CBChromo1_000048 Cc1cc(C)c(NC(=O)CCc2ccccc2)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C05 compound treatment 247200.0 100000.0 6.84 207880.0 62300.0 4.64 8.114 0.9821 1003597 CBChromo1_000049 Oc1cc2oc3cc(=O)c(O)cc3c(c4ccccc4)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C06 compound treatment 162200.0 15300.0 1.04 166240.0 20700.0 1.54 1.8248 0.9821 536 CBChromo1_000050 ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C07 compound treatment 180000.0 33100.0 2.26 190480.0 44900.0 3.34 3.9586 0.9817 1913709 CBChromo1_000051 COc1ccc(/C=N/NC(=O)c2cc3ccccc3cc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C08 compound treatment 175680.0 28800.0 1.96 178400.0 32800.0 2.44 3.1146 0.9941 1918023 CBChromo1_000052 CC[n+]1c(/C=C/N(C)c2ccccc2)n(c3ccccc3)c4ccc(cc14)c5nc6ccccc6s5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C09 compound treatment 150120.0 3220.0 0.22 147480.0 1900.0 0.14 0.2552 0.9775 1919799 CBChromo1_000053 CCOc1c(OCC)c2oc(C(=O)N3CCOCC3)c(C)c2cc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C10 compound treatment 159520.0 12600.0 0.86 157920.0 12300.0 0.92 1.2578 0.9995 1919796 CBChromo1_000054 C/C(=N\NC(=O)c1ccccc1O)/Cn2nnc(n2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C11 compound treatment 145120.0 -1780.0 -0.12 143320.0 -2260.0 -0.17 -0.2048 -0.9873 1727701 CBChromo1_000055 Clc1ccc(cc1)C(=O)NCc2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C12 compound treatment 157240.0 10300.0 0.7 159480.0 13900.0 1.03 1.2299 0.9825 1921358 CBChromo1_000056 Oc1nc(cc(n1)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C13 compound treatment 183280.0 36400.0 2.48 180640.0 35100.0 2.61 3.5989 0.9997 1035314 CBChromo1_000057 Nc1ccc(NC(=O)c2ccc(cc2)C(=O)Nc3ccc(N)cc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C14 compound treatment 158160.0 11300.0 0.77 160240.0 14700.0 1.09 1.3143 0.9852 1350276 CBChromo1_000058 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C15 compound treatment 164320.0 17400.0 1.19 160640.0 15100.0 1.12 1.6323 0.9996 535 CBChromo1_000059 ONC(=O)CCCN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C16 compound treatment 169720.0 22800.0 1.56 169240.0 23700.0 1.76 2.3452 0.9981 1593689 CBChromo1_000060 Ic1ccc(cc1)c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C17 compound treatment 227080.0 80200.0 5.47 190800.0 45200.0 3.37 6.2451 0.9729 1915616 CBChromo1_000061 [O-][N+](=O)c1cc(ccc1Cl)S(=O)(=O)Nc2ccc(Br)cc2C(=O)Nc3cc(Cl)ccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C18 compound treatment 148320.0 1420.0 0.1 145360.0 -219.0 -0.02 0.0568 0.5798 1931455 CBChromo1_000062 Fc1ccc(C(=O)n2nnc3ccccc23)c(F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C19 compound treatment 151720.0 4820.0 0.33 150720.0 5140.0 0.38 0.5028 0.9971 1133700 CBChromo1_000063 CC(Oc1cccc(Cl)c1)C(=O)NN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C20 compound treatment 148200.0 1300.0 0.09 147320.0 1740.0 0.13 0.1542 0.9827 1129917 CBChromo1_000064 CCOC(=O)C(C)Oc1ccc2c(C)c(C)c(=O)oc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C21 compound treatment 155040.0 8140.0 0.55 156720.0 11100.0 0.83 0.9786 0.9809 1920217 CBChromo1_000065 Cc1ccc(/C=N/NC(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C22 compound treatment 140480.0 -6420.0 -0.44 139600.0 -5980.0 -0.44 -0.6243 -1.0 1291152 CBChromo1_000066 COc1ccc(cc1)N(CC(=O)N2CCOCC2)S(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C23 mock treatment 143040.0 -3860.0 -0.26 138560.0 -7020.0 -0.52 -0.5556 -0.9497 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 C24 mock treatment 142000.0 -4900.0 -0.33 143680.0 -1900.0 -0.14 -0.3363 -0.9267 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D01 compound treatment 227840.0 80900.0 5.52 254160.0 109000.0 8.08 9.6163 0.9827 1523100 CBChromo1_000067 Nc1cc2cccnc2c3ncccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D02 compound treatment 155520.0 8620.0 0.59 154120.0 8540.0 0.64 0.8649 0.9992 3017585 CBChromo1_000068 CN1CCc2c1nc3CCCc3c2N.OC(=O)c1cncc(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D03 compound treatment 182280.0 35400.0 2.41 181760.0 36200.0 2.69 3.6096 0.9985 1157157 CBChromo1_000069 Cc1ccc(C)n1c2cccc(c2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D04 compound treatment 157840.0 10900.0 0.75 151520.0 5940.0 0.44 0.84 0.9689 1716722 CBChromo1_000070 Cc1ccc2[nH]c3C(CCCc3c2c1)NCC4(CC5CC6CC(C5)C4)C6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D05 compound treatment 173320.0 26400.0 1.8 168880.0 23300.0 1.73 2.4998 0.9998 1913502 CBChromo1_000071 CN(C)c1ccc(/C=N/NC(=N)N[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D06 compound treatment 153080.0 6180.0 0.42 152800.0 7220.0 0.54 0.6778 0.9927 1920938 CBChromo1_000072 Brc1ccc(cc1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D07 compound treatment 211720.0 64800.0 4.42 210000.0 64400.0 4.79 6.5151 0.9992 1010375 CBChromo1_000073 Oc1cc(cc2ccc(Nc3ccccc3)cc12)S(=O)(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D08 compound treatment 152040.0 5140.0 0.35 151240.0 5660.0 0.42 0.5456 0.9958 1218659 CBChromo1_000074 O=C(c1ccc(cc1)c2ccccc2)n3nnc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D09 compound treatment 156480.0 9580.0 0.65 147320.0 1740.0 0.13 0.5534 0.8312 1026485 CBChromo1_000075 Cc1ccc(cc1)S(=O)(=O)NCCCCCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D10 compound treatment 149520.0 2620.0 0.18 152840.0 7260.0 0.54 0.5083 0.8932 1524778 CBChromo1_000076 CCOc1ccc(cc1)C(CC(=O)c2ccccc2)Nc3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D11 compound treatment 165760.0 18900.0 1.29 162240.0 16700.0 1.24 1.7859 0.9998 1914356 CBChromo1_000077 CCc1nnc(NS(=O)(=O)c2ccc(NC(=S)NC(=O)/C=C/c3ccco3)cc2)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D12 compound treatment 149880.0 2980.0 0.2 146720.0 1140.0 0.08 0.2036 0.9252 1630350 CBChromo1_000078 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(o4)c5ccc(Cl)cc5)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D13 compound treatment 152120.0 5220.0 0.36 154960.0 9380.0 0.7 0.7452 0.951 1215060 CBChromo1_000079 Brc1cccc(c1)c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D14 compound treatment 222440.0 75500.0 5.15 210880.0 65300.0 4.86 7.0782 0.9996 1917473 CBChromo1_000080 Cc1ccc(o1)c2cc3C(=O)c4ccccc4-c3nn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D15 compound treatment 152520.0 5620.0 0.38 156440.0 10900.0 0.81 0.8424 0.9418 1337439 CBChromo1_000081 CCc1ccc(OCC(=O)Nc2c(C)cc(C)cc2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D16 compound treatment 153120.0 6220.0 0.42 159440.0 13900.0 1.03 1.0292 0.9228 1918640 CBChromo1_000082 Nc1cc(c2ccccc2c1)S(=O)(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D17 compound treatment 161800.0 14900.0 1.02 155400.0 9820.0 0.73 1.2351 0.987 3624413 CBChromo1_000083 Clc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D18 compound treatment 166400.0 19500.0 1.33 163200.0 17600.0 1.31 1.8673 1.0 1374975 CBChromo1_000084 Oc1ccc(NS(=O)(=O)c2ccccc2)cc1c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D19 compound treatment 146480.0 -423.0 -0.03 146840.0 1260.0 0.09 0.046 0.4686 3624414 CBChromo1_000085 O=C(Nc1cccc(c1)C(=O)n2nnc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D20 compound treatment 148080.0 1180.0 0.08 149920.0 4340.0 0.32 0.2852 0.8567 1241852 CBChromo1_000086 O=S(=O)(Nc1ccc2oc(nc2c1)c3cccnc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D21 compound treatment 149080.0 2180.0 0.15 148920.0 3340.0 0.25 0.2808 0.9696 3624415 CBChromo1_000087 Cc1ccc(NC(=O)COc2ccc(C)c(C)c2)c(N)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D22 compound treatment 139120.0 -7780.0 -0.53 142640.0 -2940.0 -0.22 -0.5298 -0.9232 471 CBChromo1_000088 CCCC(CCC)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D23 mock treatment 141960.0 -4940.0 -0.34 145640.0 61.3 0.0 -0.235 -0.6975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 D24 mock treatment 140240.0 -6660.0 -0.45 136800.0 -8780.0 -0.65 -0.7832 -0.9842 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E01 compound treatment 148960.0 2060.0 0.14 159120.0 13500.0 1.01 0.8118 0.7978 1427482 CBChromo1_000089 Cc1c(oc2c3OCCOc3ccc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E02 compound treatment 166760.0 19900.0 1.35 169480.0 23900.0 1.78 2.2152 0.9909 1921826 CBChromo1_000090 Oc1ccc(Br)cc1/C=N/c2cccc(Nc3nc(nc(n3)N4CCOCC4)N(c5ccccc5)c6ccccc6)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E03 compound treatment 158000.0 11100.0 0.76 161040.0 15500.0 1.15 1.3487 0.9793 1913491 CBChromo1_000091 Ic1ccccc1C(=O)OCC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E04 compound treatment 225600.0 78700.0 5.37 239640.0 94100.0 7.0 8.7441 0.9914 1919107 CBChromo1_000092 Cc1cc(NCCCN2CCOCC2)nc(n1)c3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E05 compound treatment 160960.0 14100.0 0.96 153160.0 7580.0 0.56 1.0767 0.9681 1118121 CBChromo1_000093 CC1(C)CC(=C(CC2C(=O)CC(C)(C)CC2=O)C(=O)C1)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E06 compound treatment 158960.0 12100.0 0.82 155440.0 9860.0 0.73 1.1002 0.9984 1921947 CBChromo1_000094 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccccc4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E07 compound treatment 176160.0 29300.0 1.99 172400.0 26800.0 2.0 2.822 1.0 1913769 CBChromo1_000095 Oc1cc2ccccc2cc1C(=O)N/N=C/c3ccccc3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E08 compound treatment 187320.0 40400.0 2.76 191480.0 45900.0 3.42 4.3641 0.9943 1919356 CBChromo1_000096 COc1ccc(cc1)c2n(C)c3ccccc3[n+]2C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E09 compound treatment 184600.0 37700.0 2.57 182240.0 36700.0 2.73 3.7467 0.9996 1912827 CBChromo1_000097 CCN(CC)c1ccc(/C=N\NC(=O)c2cccc(Br)c2)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E10 compound treatment 157760.0 10900.0 0.74 159440.0 13900.0 1.03 1.2529 0.9867 1918577 CBChromo1_000098 O=S(=O)(c1ccccc1)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E11 compound treatment 169280.0 22400.0 1.53 163760.0 18200.0 1.35 2.0356 0.9982 1003076 CBChromo1_000099 OC(=O)c1ccccc1c2c3cc(Br)c(O)c(Br)c3oc4c(Br)c(=O)c(Br)cc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E12 compound treatment 181760.0 34900.0 2.38 179120.0 33500.0 2.5 3.4456 0.9997 1917753 CBChromo1_000100 COc1ccc2C(=O)N(C)C(=O)c3cccc1c32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E13 compound treatment 169360.0 22500.0 1.53 171320.0 25700.0 1.92 2.4373 0.9938 1470918 CBChromo1_000101 Cc1cc(C)cc(NCC(=O)Nc2c(C)cccc2C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E14 compound treatment 165960.0 19100.0 1.3 171440.0 25900.0 1.92 2.2798 0.9817 1941017 CBChromo1_000102 Cc1cc(Cl)ccc1OCCCC(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E15 compound treatment 193840.0 46900.0 3.2 189000.0 43400.0 3.23 4.5479 1.0 1914841 CBChromo1_000103 [O-][N+](=O)c1ccccc1NC(=S)NC(NC(=O)Cc2cccc3ccccc23)C(Cl)(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E16 compound treatment 158960.0 12100.0 0.82 157240.0 11700.0 0.87 1.195 0.9996 1275344 CBChromo1_000104 CCc1ccc2oc(nc2c1)c3ccc(C)c(NS(=O)(=O)c4ccccc4)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E17 compound treatment 264520.0 118000.0 8.02 226120.0 80500.0 5.99 9.9088 0.9897 1915720 CBChromo1_000105 [O-][N+](=O)c1cc(ccc1Cl)S(=O)(=O)Nc2ccc(Cl)cc2C(=O)Nc3cc(Cl)ccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E18 compound treatment 159920.0 13000.0 0.89 156880.0 11300.0 0.84 1.2223 0.9996 1931570 CBChromo1_000106 [O-][N+](=O)c1ccc(F)c(c1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E19 compound treatment 164280.0 17400.0 1.18 164880.0 19300.0 1.44 1.8535 0.9954 1920218 CBChromo1_000107 Clc1c(Cl)c(Cl)c(C(=O)OCC#C)c(C(=O)OCC#C)c1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E20 compound treatment 156520.0 9620.0 0.66 156360.0 10800.0 0.8 1.031 0.995 1291287 CBChromo1_000108 Cc1cc(C)c(NC(=O)COc2cccc(Cl)c2)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E21 compound treatment 161880.0 15000.0 1.02 170200.0 24600.0 1.83 2.0178 0.9619 1919426 CBChromo1_000109 COc1ccc(/C=N/NC(=O)c2ccccc2O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E22 compound treatment 159120.0 12200.0 0.83 158240.0 12700.0 0.94 1.2553 0.9981 1166615 CBChromo1_000110 COc1ccc(N(CC(=O)Nc2ccccc2Br)S(=O)(=O)c3ccc(C)cc3)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E23 mock treatment 152320.0 5420.0 0.37 150520.0 4940.0 0.37 0.5212 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 E24 mock treatment 152080.0 5180.0 0.35 145600.0 21.3 0.0 0.2507 0.7103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F01 compound treatment 154240.0 7340.0 0.5 150960.0 5380.0 0.4 0.6369 0.9939 1913508 CBChromo1_000111 Nc1scc[n+]1CC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F02 compound treatment 155520.0 8620.0 0.59 157240.0 11700.0 0.87 1.0291 0.9819 1915702 CBChromo1_000112 Oc1c(I)cc(I)cc1C(=O)Nc2cc(ccc2Cl)S(=O)(=O)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F03 compound treatment 155600.0 8700.0 0.59 158080.0 12500.0 0.93 1.0772 0.9763 1774290 CBChromo1_000113 [O-][N+](=O)c1ccc(cc1)C(=O)Nc2sc3CCCCc3c2C(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F04 compound treatment 162480.0 15600.0 1.06 161560.0 16000.0 1.19 1.592 0.9984 1251647 CBChromo1_000114 Fc1ccccc1CN2CCN(CC2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F05 compound treatment 158120.0 11200.0 0.76 159440.0 13900.0 1.03 1.2703 0.9891 1628747 CBChromo1_000115 COc1ccc(cc1OC)C(=O)Nc2ccccc2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F06 compound treatment 175600.0 28700.0 1.96 167800.0 22200.0 1.65 2.5529 0.9965 1921581 CBChromo1_000116 CCN(C(=O)c1ccc(cc1)c2ccccc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F07 compound treatment 157720.0 10800.0 0.74 158440.0 12900.0 0.96 1.1984 0.9917 1049687 CBChromo1_000117 Cc1ccc(cc1)S(=O)(=O)Nc2cccc3cccnc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F08 compound treatment 165440.0 18500.0 1.26 164960.0 19400.0 1.44 1.9137 0.9978 541 CBChromo1_000118 Cc1c(C)c(CONC(=O)c2ccccc2)c(C)c(C)c1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F09 compound treatment 174280.0 27400.0 1.87 163880.0 18300.0 1.36 2.283 0.988 1565273 CBChromo1_000119 Oc1ccc(Oc2ccc(Oc3ccc(O)cc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F10 compound treatment 158960.0 12100.0 0.82 156680.0 11100.0 0.83 1.1655 1.0 1176912 CBChromo1_000120 Cc1cc(C)c(NC(=O)COc2ccc(Cl)cc2)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F11 compound treatment 256720.0 110000.0 7.49 217000.0 71400.0 5.32 9.0529 0.9859 1914302 CBChromo1_000121 O=C(NC(=S)Nc1ccc(cc1)S(=O)(=O)Nc2nccs2)/C=C/c3ccco3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F12 compound treatment 156920.0 10000.0 0.68 155840.0 10300.0 0.76 1.023 0.9984 1613055 CBChromo1_000122 Cc1ccccc1C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F13 compound treatment 172200.0 25300.0 1.72 174320.0 28700.0 2.14 2.7321 0.9943 1359699 CBChromo1_000123 Brc1ccccc1c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F14 compound treatment 198400.0 51500.0 3.51 191120.0 45500.0 3.39 4.8793 0.9998 1918058 CBChromo1_000124 Oc1ccccc1C(=O)NNC(=S)NC(=O)c2ccc(cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F15 compound treatment 164440.0 17500.0 1.2 162360.0 16800.0 1.25 1.7286 0.9998 1175946 CBChromo1_000125 Cc1cc(C)c(NC(=O)COc2ccc(C)c(C)c2)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F16 compound treatment 156960.0 10100.0 0.69 155760.0 10200.0 0.76 1.0207 0.9988 1708885 CBChromo1_000126 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F17 compound treatment 180400.0 33500.0 2.28 173440.0 27900.0 2.07 3.0811 0.9988 3624416 CBChromo1_000127 Clc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F18 compound treatment 202000.0 55100.0 3.76 198000.0 52400.0 3.9 5.415 0.9998 1525986 CBChromo1_000128 Cc1ccc2oc(nc2c1)c3cccc(NS(=O)(=O)c4ccccc4)c3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F19 compound treatment 164520.0 17600.0 1.2 161560.0 16000.0 1.19 1.6904 1.0 1451943 CBChromo1_000129 Cc1ccc(NC(=O)c2ccc(OCC(=O)Nc3ccccc3)cc2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F20 compound treatment 170280.0 23400.0 1.59 170320.0 24700.0 1.84 2.4291 0.9974 1577769 CBChromo1_000130 CCc1ccc2oc(nc2c1)c3ccc(NS(=O)(=O)c4ccccc4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F21 compound treatment 152920.0 6020.0 0.41 160680.0 15100.0 1.12 1.0848 0.9067 3624417 CBChromo1_000131 Cc1ccc(C(=O)n2nnc3ccccc23)c(F)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F22 compound treatment 144880.0 -2020.0 -0.14 153800.0 8220.0 0.61 0.3352 0.5344 3069074 CBChromo1_000132 N[C@@H]1C[C@H]1c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F23 mock treatment 155120.0 8220.0 0.56 150320.0 4740.0 0.35 0.6457 0.9752 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 F24 mock treatment 145680.0 -1220.0 -0.08 140720.0 -4860.0 -0.36 -0.3146 -0.8479 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G01 compound treatment 237480.0 90600.0 6.18 232960.0 87400.0 6.5 8.9653 0.9997 1912757 CBChromo1_000133 Cc1cc2/C(=C/c3ccco3)/OC(=O)c2c(=O)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G02 compound treatment 249680.0 103000.0 7.01 239240.0 93700.0 6.97 9.8839 1.0 1915749 CBChromo1_000134 Oc1ccc(/N=C/c2ccc(o2)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G03 compound treatment 214160.0 67300.0 4.59 207640.0 62100.0 4.62 6.5085 1.0 1913613 CBChromo1_000135 CCc1c(cn2CCn3c(C)ccc3-c12)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G04 compound treatment 206440.0 59500.0 4.06 203320.0 57700.0 4.3 5.909 0.9996 1367680 CBChromo1_000136 Cc1ccc(cc1)c2cc(nc(n2)N3CCOCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G05 compound treatment 187600.0 40700.0 2.77 178480.0 32900.0 2.45 3.6935 0.9981 1913753 CBChromo1_000137 C/C(=N\NC(=O)c1ccccc1O)/c2ccc3ccccc3c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G06 compound treatment 183560.0 36700.0 2.5 174880.0 29300.0 2.18 3.3093 0.9977 540 CBChromo1_000138 CC1(CC2CC3(C)C1)CC(C2)(C3)C(=O)NO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G07 compound treatment 96040.0 -50900.0 -3.47 93840.0 -51700.0 -3.85 -5.1749 -0.9986 1913831 CBChromo1_000139 CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2CC)/C=Cc4cc(C)ccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G08 compound treatment 160320.0 13400.0 0.91 155720.0 10100.0 0.75 1.1805 0.9954 1919068 CBChromo1_000140 Clc1ccc(nn1)N2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G09 compound treatment 173920.0 27000.0 1.84 169480.0 23900.0 1.78 2.5603 0.9998 1919035 CBChromo1_000141 [O-][N+](=O)c1ccc(cc1)C(=O)Oc2c(Cl)cc(Cl)c(Cl)c2CNC(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G10 compound treatment 169280.0 22400.0 1.53 168280.0 22700.0 1.69 2.2735 0.9987 1918768 CBChromo1_000142 Clc1ccc(C(=O)n2nnc3ccccc23)c(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G11 compound treatment 122080.0 -24800.0 -1.69 121360.0 -24200.0 -1.8 -2.4712 -0.9995 1001846 CBChromo1_000143 CCNc1cc2oc3cc(=NCC)c(C)cc3c(c4ccccc4C(=O)OCC)c2cc1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G12 compound treatment 165160.0 18300.0 1.24 161920.0 16300.0 1.22 1.7402 0.9999 1294988 CBChromo1_000144 Fc1ccccc1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G13 compound treatment 161840.0 14900.0 1.02 160160.0 14600.0 1.09 1.4875 0.9995 1499150 CBChromo1_000145 Cc1ccccc1NCC(=O)Nc2c(C)cccc2C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G14 compound treatment 159720.0 12800.0 0.87 163960.0 18400.0 1.37 1.5853 0.9766 1256375 CBChromo1_000146 COc1ccc(cc1)C(=O)CC(Nc2ccc(Cl)cc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G15 compound treatment 164640.0 17700.0 1.21 165120.0 19500.0 1.45 1.8835 0.9958 1352496 CBChromo1_000147 Nc1ccc(C(=O)Nc2ccc(cc2)C(=O)O)c(c1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G16 compound treatment 186400.0 39500.0 2.69 186560.0 41000.0 3.05 4.0609 0.9981 1707305 CBChromo1_000148 O=S(=O)(Nc1ccc(cc1)c2nc3ccccc3o2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G17 compound treatment 233600.0 86700.0 5.91 243640.0 98100.0 7.3 9.3403 0.9945 1916635 CBChromo1_000149 Nc1ccc(cc1)c2nc3ccc(cc3[nH]2)c4nc5ccc(N)cc5[nH]4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G18 compound treatment 159200.0 12300.0 0.84 159680.0 14100.0 1.05 1.335 0.9938 1931472 CBChromo1_000150 Cc1cc(F)c(F)cc1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G19 compound treatment 160080.0 13200.0 0.9 159760.0 14200.0 1.06 1.3816 0.9968 3624419 CBChromo1_000151 Clc1ccc(cc1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G20 compound treatment 155880.0 8980.0 0.61 160360.0 14800.0 1.1 1.2107 0.9617 1924714 CBChromo1_000152 COc1ccc(cc1Br)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G21 compound treatment 165480.0 18600.0 1.27 168040.0 22500.0 1.67 2.0777 0.9906 1919298 CBChromo1_000153 Cc1cc(C)c(/C=N/NC(=O)c2ccccc2[N+](=O)[O-])c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G22 compound treatment 162600.0 15700.0 1.07 161000.0 15400.0 1.15 1.5683 0.9994 1924575 CBChromo1_000154 COC(=O)c1ccc(cc1)C2C(=C(C)NC(=C2C(=O)OCC=C)C)C(=O)OCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G23 mock treatment 150640.0 3740.0 0.25 153480.0 7900.0 0.59 0.596 0.93 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 G24 mock treatment 149520.0 2620.0 0.18 151520.0 5940.0 0.44 0.4389 0.9204 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H01 compound treatment 153680.0 6780.0 0.46 154600.0 9020.0 0.67 0.8015 0.9834 1913510 CBChromo1_000155 NC1=[N+](Cc2ccccc12)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H02 compound treatment 197040.0 50100.0 3.42 192400.0 46800.0 3.48 4.8811 1.0 1410511 CBChromo1_000156 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(Cc3ccc(NS(=O)(=O)c4ccc(C)cc4)c(c3)C(=O)O)cc2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H03 compound treatment 158240.0 11300.0 0.77 163320.0 17700.0 1.32 1.4802 0.9675 1913412 CBChromo1_000157 OCCSc1nnnn1c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H04 compound treatment 161480.0 14600.0 0.99 161880.0 16300.0 1.21 1.5607 0.9951 1156418 CBChromo1_000158 Cc1ccc(CN2CCN(CC2)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H05 compound treatment 160800.0 13900.0 0.95 157240.0 11700.0 0.87 1.2837 0.999 1380267 CBChromo1_000159 COc1ccc(cc1OC)C(=O)OCCN2CCOCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H06 compound treatment 158240.0 11300.0 0.77 154600.0 9020.0 0.67 1.0213 0.9975 1920603 CBChromo1_000160 CC1CCN(CC1)C(=O)Nc2ccccc2C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H07 compound treatment 255120.0 108000.0 7.38 262040.0 116000.0 8.67 11.3461 0.9968 1917951 CBChromo1_000161 Oc1ccc2ccccc2c1/C=N/NC(=O)c3ccn[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H08 compound treatment 157200.0 10300.0 0.7 156920.0 11300.0 0.84 1.0933 0.9958 3624420 CBChromo1_000162 CC1(C)CC(=O)C2=C(C1)OC3=C(C2)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H09 compound treatment 187560.0 40700.0 2.77 179320.0 33700.0 2.51 3.7358 0.9988 1913459 CBChromo1_000163 COc1ccc(NC(=S)NC(NC(=O)/C=C/c2ccccc2)C(Cl)(Cl)Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H10 compound treatment 162680.0 15800.0 1.08 156920.0 11300.0 0.84 1.3575 0.9928 3624421 CBChromo1_000164 [O-][N+](=O)c1ccc(C(=O)n2nnc3ccccc23)c(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H11 compound treatment 170520.0 23600.0 1.61 169680.0 24100.0 1.79 2.407 0.9985 3624422 CBChromo1_000165 Brc1cc(Br)c(OC(=O)CCCC(=O)OCC#C)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H12 compound treatment 172240.0 25300.0 1.73 168880.0 23300.0 1.73 2.4478 1.0 1720239 CBChromo1_000166 CCOc1ccc(cc1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H13 compound treatment 199200.0 52300.0 3.57 192080.0 46500.0 3.46 4.9684 0.9999 1604810 CBChromo1_000167 COc1ccc(cc1Br)c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H14 compound treatment 159520.0 12600.0 0.86 162840.0 17300.0 1.28 1.5167 0.981 1029030 CBChromo1_000168 OC(Cc1cccnc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H15 compound treatment 162200.0 15300.0 1.04 158040.0 12500.0 0.93 1.3933 0.9983 3624423 CBChromo1_000169 Fc1cccc(c1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H16 compound treatment 158400.0 11500.0 0.78 159040.0 13500.0 1.0 1.2627 0.9926 1777712 CBChromo1_000170 CCc1ccc(cc1)c2nc3cc(NC(=O)c4cccc(c4)[N+](=O)[O-])ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H17 compound treatment 157880.0 11000.0 0.75 160000.0 14400.0 1.07 1.2882 0.9845 3624424 CBChromo1_000171 Cc1cc(F)c(F)c(C(=O)n2nnc3ccccc23)c1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H18 compound treatment 194840.0 47900.0 3.27 191160.0 45600.0 3.39 4.7098 0.9998 1369668 CBChromo1_000172 Fc1ccccc1c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H19 compound treatment 156360.0 9460.0 0.64 154320.0 8740.0 0.65 0.916 1.0 3624425 CBChromo1_000173 COc1ccc(cc1Br)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H20 compound treatment 169560.0 22700.0 1.54 174440.0 28900.0 2.15 2.6112 0.9869 1494517 CBChromo1_000174 Clc1ccc(cc1)c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H21 compound treatment 174200.0 27300.0 1.86 168960.0 23400.0 1.74 2.5465 0.9994 3624426 CBChromo1_000175 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3nc4cc(C)ccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H22 compound treatment 154080.0 7180.0 0.49 148520.0 2940.0 0.22 0.5008 0.9342 3273 CBChromo1_000176 NNCCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H23 mock treatment 148280.0 1380.0 0.09 149720.0 4140.0 0.31 0.2844 0.8825 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 H24 mock treatment 147080.0 178.0 0.01 142240.0 -3340.0 -0.25 -0.1672 -0.6719 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I01 compound treatment 203880.0 57000.0 3.88 196400.0 50800.0 3.78 5.4214 0.9999 1912759 CBChromo1_000177 Cc1ccc(/C=C/2\OC(=O)c3c2cc(C)[nH]c3=O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I02 compound treatment 159120.0 12200.0 0.83 158600.0 13000.0 0.97 1.2743 0.9972 1004614 CBChromo1_000178 OC(=O)CNS(=O)(=O)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I03 compound treatment 164680.0 17800.0 1.21 162680.0 17100.0 1.27 1.757 0.9997 1913667 CBChromo1_000179 CCOC(=O)C/C(=N/c1cnn(c1)c2ccccc2)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I04 compound treatment 157840.0 10900.0 0.75 159800.0 14200.0 1.06 1.2757 0.9853 878 CBChromo1_000180 CC(=O)NS(=O)(=O)c1ccc(N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I05 compound treatment 163440.0 16500.0 1.13 162920.0 17300.0 1.29 1.7099 0.9977 1921399 CBChromo1_000181 [O-][N+](=O)c1ccc(Nc2ccccc2Cl)c(c1)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I06 compound treatment 169960.0 23100.0 1.57 168200.0 22600.0 1.68 2.3021 0.9994 1283442 CBChromo1_000182 O=C(Nc1ccc2OCOc2c1)C3(CC4CC5CC(C4)C3)C5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I07 compound treatment 170080.0 23200.0 1.58 164960.0 19400.0 1.44 2.1373 0.999 1921209 CBChromo1_000183 CC[n+]1c(/C=C/N(C)c2ccccc2)oc3ccc(cc13)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I08 compound treatment 161640.0 14700.0 1.0 162960.0 17400.0 1.29 1.6252 0.9922 1918103 CBChromo1_000184 CCN(CC)CCn1c2ccccc2c3nc4ccc(cc4cc13)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I09 compound treatment 170360.0 23500.0 1.6 167240.0 21700.0 1.61 2.2708 1.0 1913121 CBChromo1_000185 CCCN1C/C(=C\c2cccc(c2)[N+](=O)[O-])/C(=O)\C(=C\c3cccc(c3)[N+](=O)[O-])\C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I10 compound treatment 175920.0 29000.0 1.98 176320.0 30700.0 2.29 3.0167 0.9974 1920019 CBChromo1_000186 Cc1cc(O)c(C(=O)O)c(/C=C/c2cccc(Br)c2)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I11 compound treatment 162240.0 15300.0 1.05 161280.0 15700.0 1.17 1.5657 0.9985 1913249 CBChromo1_000187 CN(C)c1ccc(/C=C\2/C(=O)N(N=C2c3ccccc3)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I12 compound treatment 185360.0 38500.0 2.62 179560.0 34000.0 2.53 3.6423 0.9998 1921765 CBChromo1_000188 [O-][N+](=O)c1cccc(/C=C/C(=O)Nc2cccc(Cl)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I13 compound treatment 158920.0 12000.0 0.82 162800.0 17200.0 1.28 1.4857 0.9766 1558952 CBChromo1_000189 Cc1cccc(C)c1NC(=O)CNc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I14 compound treatment 158720.0 11800.0 0.81 160840.0 15300.0 1.14 1.3729 0.9858 1661743 CBChromo1_000190 COc1ccc(cc1)C(=O)CC(Nc2ccc(Br)cc2)c3ccc(F)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I15 compound treatment 156280.0 9380.0 0.64 162560.0 17000.0 1.26 1.3458 0.9502 1786058 CBChromo1_000191 [O-][N+](=O)c1ccc(cc1)C(=O)Oc2ccc(C(=O)c3ccccc3)c(OC(=O)c4ccc(cc4)[N+](=O)[O-])c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I16 compound treatment 161560.0 14700.0 1.0 167520.0 21900.0 1.63 1.8613 0.9722 1642758 CBChromo1_000192 Cc1cc(C)c2oc(nc2c1)c3ccc(NS(=O)(=O)c4ccccc4)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I17 compound treatment 198080.0 51200.0 3.49 200480.0 54900.0 4.09 5.3565 0.9969 1580129 CBChromo1_000193 Nc1ccccc1C(=O)Nc2ccc(cc2C(=O)O)c3ccc(NC(=O)c4ccccc4N)c(c3)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I18 compound treatment 160000.0 13100.0 0.89 165080.0 19500.0 1.45 1.6577 0.9728 3624427 CBChromo1_000194 Fc1ccc(cc1F)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I19 compound treatment 158560.0 11700.0 0.79 162360.0 16800.0 1.25 1.4451 0.9762 1919066 CBChromo1_000195 Brc1cccc(c1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I20 compound treatment 162880.0 16000.0 1.09 165880.0 20300.0 1.51 1.8387 0.9871 1378967 CBChromo1_000196 CCc1ccccc1N2C(=O)CC(Sc3nc(C)cc(C)n3)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I21 compound treatment 164840.0 17900.0 1.22 169600.0 24000.0 1.79 2.1289 0.9828 1919338 CBChromo1_000197 COc1cc(/C=N/NC(=O)c2ccccc2O)c(cc1OC)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I22 compound treatment 172040.0 25100.0 1.71 170360.0 24800.0 1.84 2.516 0.9993 3624428 CBChromo1_000198 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I23 mock treatment 149360.0 2460.0 0.17 144480.0 -1100.0 -0.08 0.0606 0.3253 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 I24 mock treatment 144680.0 -2220.0 -0.15 146040.0 461.0 0.03 -0.0829 -0.5334 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J01 compound treatment 169680.0 22800.0 1.55 171120.0 25500.0 1.9 2.4422 0.995 1002045 CBChromo1_000199 Oc1c(ccc2cccnc12)C(Nc3ccc(cc3)[N+](=O)[O-])c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J02 compound treatment 197120.0 50200.0 3.42 189960.0 44400.0 3.3 4.7566 0.9998 1043460 CBChromo1_000200 COC(=O)c1ccccc1NC(c2ccccc2)c3ccc4cccnc4c3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J03 compound treatment 151840.0 4940.0 0.34 151920.0 6340.0 0.47 0.5718 0.9863 1920592 CBChromo1_000201 O=c1c(=NNc2nnn[nH]2)c(=O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J04 compound treatment 159800.0 12900.0 0.88 159280.0 13700.0 1.02 1.3428 0.9973 1681672 CBChromo1_000202 CCOc1ccc(cc1)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J05 compound treatment 278320.0 131000.0 8.96 273800.0 128000.0 9.54 13.0834 0.9995 1916346 CBChromo1_000203 CCOC(=O)C1=C(C)C2C3C(C(=O)N(C3=O)c4ccc(cc4)C(=O)O)C1(C)C5C2C(=O)N(C5=O)c6ccc(cc6)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J06 compound treatment 231920.0 85000.0 5.8 270920.0 125000.0 9.33 10.695 0.9738 1382399 CBChromo1_000204 C(Cc1ccccc1)NC2CCCc3c2[nH]c4ccc(cc34)C5CCCCC5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J07 compound treatment 167040.0 20100.0 1.37 163080.0 17500.0 1.3 1.8918 0.9997 1353277 CBChromo1_000205 CCOC(=O)c1[nH]c2CCC(=C(Sc3ccccc3)c2c1C)C=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J08 compound treatment 162840.0 15900.0 1.09 160800.0 15200.0 1.13 1.5694 0.9998 1094556 CBChromo1_000206 CC1C2=C(CC(C)(C)CC2=O)OC3=C1C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J09 compound treatment 173240.0 26300.0 1.8 166440.0 20900.0 1.55 2.3676 0.9974 1913469 CBChromo1_000207 ClC(Cl)(Cl)C(NC(=O)/C=C/c1ccccc1)NC(=S)Nc2ccc(N=Nc3ccccc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J10 compound treatment 165040.0 18100.0 1.24 162200.0 16600.0 1.24 1.7491 1.0 1676891 CBChromo1_000208 COc1cccc(OC)c1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J11 compound treatment 163520.0 16600.0 1.13 160080.0 14500.0 1.08 1.5643 0.9997 1918471 CBChromo1_000209 Brc1cc(Br)c(OC(=O)c2ccccc2C(=O)OCC#C)c(Br)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J12 compound treatment 184000.0 37100.0 2.53 182960.0 37400.0 2.78 3.7557 0.9989 1262121 CBChromo1_000210 COc1cc(cc(OC)c1O)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J13 compound treatment 176840.0 29900.0 2.04 174240.0 28700.0 2.13 2.9516 0.9998 3624429 CBChromo1_000211 O=S(=O)(Nc1cccc(c1)c2nc3ccccc3o2)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J14 compound treatment 156800.0 9900.0 0.67 156440.0 10900.0 0.81 1.0487 0.996 1918243 CBChromo1_000212 CC(=O)N(CCCn1c2ccccc2c3nc4ccc(cc4cc13)[N+](=O)[O-])C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J15 compound treatment 158640.0 11700.0 0.8 162120.0 16500.0 1.23 1.4364 0.9782 3624430 CBChromo1_000213 COc1ccc(Cl)cc1C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J16 compound treatment 192720.0 45800.0 3.12 193520.0 47900.0 3.57 4.7318 0.9978 1921580 CBChromo1_000214 Oc1ccc(/N=C/C=C/c2ccccc2[N+](=O)[O-])cc1c3nc4ccccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J17 compound treatment 156920.0 10000.0 0.68 158440.0 12900.0 0.96 1.1598 0.9863 3624431 CBChromo1_000215 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(cc4)C(=O)O)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J18 compound treatment 157920.0 11000.0 0.75 156960.0 11400.0 0.85 1.1301 0.9982 3624432 CBChromo1_000216 Fc1cccc(C(=O)n2nnc3ccccc23)c1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J19 compound treatment 160640.0 13700.0 0.94 162800.0 17200.0 1.28 1.5686 0.9881 1860866 CBChromo1_000217 Cc1ccc(cc1I)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J20 compound treatment 152360.0 5460.0 0.37 153720.0 8140.0 0.61 0.6916 0.9726 199 CBChromo1_000218 C[C@H](/C=C(\C)/C=C/C(=O)NO)C(=O)c1ccc(cc1)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J21 compound treatment 162600.0 15700.0 1.07 170160.0 24600.0 1.83 2.0504 0.9674 3624433 CBChromo1_000219 Cc1ccc(cc1NS(=O)(=O)c2ccc(Cl)cc2)c3nc4ccccc4[nH]3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J22 compound treatment 145280.0 -1620.0 -0.11 148400.0 2820.0 0.21 0.0703 0.296 865102 CBChromo1_000220 O=C(CCNNC(=O)c1ccncc1)NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J23 mock treatment 150600.0 3700.0 0.25 147320.0 1740.0 0.13 0.2699 0.9522 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 J24 mock treatment 142320.0 -4580.0 -0.31 146080.0 501.0 0.04 -0.1945 -0.6183 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K01 compound treatment 164840.0 17900.0 1.22 167520.0 21900.0 1.63 2.0195 0.9898 1912767 CBChromo1_000221 COc1ccc(/C=C/2\OC(=O)c3c2cc(C)[nH]c3=O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K02 compound treatment 169960.0 23100.0 1.57 171120.0 25500.0 1.9 2.4557 0.9955 1913149 CBChromo1_000222 CC(C)(C)c1cc(Br)cc(/C=N/NC(=O)c2ccccc2O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K03 compound treatment 158840.0 11900.0 0.81 158360.0 12800.0 0.95 1.2481 0.997 1914261 CBChromo1_000223 CC/C(=N\N=C(/CC)\c1ccccc1)/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K04 compound treatment 185760.0 38900.0 2.65 182520.0 36900.0 2.75 3.8174 0.9998 1917298 CBChromo1_000224 C/C(=N\NC(=O)c1ccc(cc1)c2ccccc2)/c3cccc(N)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K05 compound treatment 207800.0 60900.0 4.15 191880.0 46300.0 3.45 5.3725 0.9957 1912543 CBChromo1_000225 O=C(Oc1ccc(/C=N/Nc2ccccc2)cc1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K06 compound treatment 222560.0 75700.0 5.16 216320.0 70700.0 5.27 7.3703 0.9999 1661768 CBChromo1_000226 Cc1ccc(cc1)C(=O)c2coc3ccc(O)c(Cl)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K07 compound treatment 197120.0 50200.0 3.42 186600.0 41000.0 3.05 4.5798 0.9984 1913935 CBChromo1_000227 Oc1ccccc1C(=O)N/N=C\c2ccc(Cl)cc2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K08 compound treatment 176160.0 29300.0 1.99 173640.0 28100.0 2.09 2.8873 0.9997 1917883 CBChromo1_000228 O/N=C/1\C2(CCCCC2)C(=O)N(O)C31CCCC=C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K09 compound treatment 168600.0 21700.0 1.48 157760.0 12200.0 0.91 1.6871 0.9724 1498599 CBChromo1_000229 CCOC(=O)C1(CCCC1=O)C2(O)C(=O)c3ccccc3C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K10 compound treatment 179280.0 32400.0 2.21 176080.0 30500.0 2.27 3.1661 0.9999 1919798 CBChromo1_000230 Oc1ccc(cc1/C=N/c2cccc3ccccc23)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K11 compound treatment 193800.0 46900.0 3.2 182800.0 37200.0 2.77 4.2197 0.9974 1920545 CBChromo1_000231 O=c1cc([nH]c(=S)[nH]1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K12 compound treatment 164640.0 17700.0 1.21 154640.0 9060.0 0.67 1.332 0.962 1975241 CBChromo1_000232 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(Cl)cc4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K13 compound treatment 188320.0 41400.0 2.82 184600.0 39000.0 2.9 4.0503 0.9999 1918634 CBChromo1_000233 [O-][n+]1ccc(N/N=C/c2ccc(F)cc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K14 compound treatment 164000.0 17100.0 1.17 160360.0 14800.0 1.1 1.6021 0.9996 1188672 CBChromo1_000234 COc1ccc(cc1)C(=O)CC(Nc2ccc(Cl)cc2)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K15 compound treatment 158520.0 11600.0 0.79 164600.0 19000.0 1.42 1.5611 0.9623 1425867 CBChromo1_000235 Oc1ccccc1C(CC(=O)N2CCCCC2)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K16 compound treatment 187640.0 40700.0 2.78 181720.0 36100.0 2.69 3.8659 0.9999 1393634 CBChromo1_000236 CCc1ccc(cc1)c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K17 compound treatment 166560.0 19700.0 1.34 168040.0 22500.0 1.67 2.1297 0.994 1709481 CBChromo1_000237 Cc1ccc(cc1)S(=O)(=O)Nc2cc(C(=O)O)c(NS(=O)(=O)c3ccc(C)cc3)cc2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K18 compound treatment 160560.0 13700.0 0.93 167760.0 22200.0 1.65 1.8258 0.9633 1931583 CBChromo1_000238 Fc1cc(Cl)c(cc1F)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K19 compound treatment 154200.0 7300.0 0.5 164080.0 18500.0 1.38 1.3255 0.9053 1473494 CBChromo1_000239 Cc1ccc(C)c(NCC(=O)Nc2c(C)cccc2C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K20 compound treatment 176960.0 30100.0 2.05 177560.0 32000.0 2.38 3.1321 0.9972 1229469 CBChromo1_000240 CCCOc1ccc(cc1OCC)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K21 compound treatment 160560.0 13700.0 0.93 169360.0 23800.0 1.77 1.91 0.955 1920306 CBChromo1_000241 CCn1c2ccccc2c3cc(/C=N/NC(=O)COc4ccccc4)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K22 compound treatment 159560.0 12700.0 0.86 160000.0 14400.0 1.07 1.3692 0.9941 1564910 CBChromo1_000242 Cc1cc(C)c(OCC(=O)Nc2c(C)cccc2C)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K23 mock treatment 148240.0 1340.0 0.09 152960.0 7380.0 0.55 0.4529 0.8133 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 K24 mock treatment 146760.0 -143.0 -0.01 145600.0 21.3 0.0 -0.0058 -0.5843 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L01 compound treatment 153920.0 7020.0 0.48 156000.0 10400.0 0.78 0.8867 0.973 1913570 CBChromo1_000243 CCC(=O)OCC1OC(C(Br)C1OC(=O)CC)n2cc(F)c(=O)[nH]c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L02 compound treatment 164720.0 17800.0 1.21 166080.0 20500.0 1.53 1.9379 0.9936 1917264 CBChromo1_000244 [O-][N+](=O)c1ccccc1NC(=O)c2cc(ccc2Cl)S(=O)(=O)N3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L03 compound treatment 168320.0 21400.0 1.46 164400.0 18800.0 1.4 2.023 0.9998 1913436 CBChromo1_000245 O=C(N/N=C\c1ccco1)c2ccncc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L04 compound treatment 177080.0 30200.0 2.06 175680.0 30100.0 2.24 3.039 0.9991 1706491 CBChromo1_000246 Fc1ccc(cc1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L05 compound treatment 399400.0 252000.0 17.21 384440.0 239000.0 17.78 24.7432 0.9999 1027977 CBChromo1_000247 O=C1C=CC(=O)N1c2cccc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L06 compound treatment 182480.0 35600.0 2.43 178760.0 33200.0 2.47 3.4614 1.0 1921008 CBChromo1_000248 Clc1ccccc1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L07 compound treatment 217680.0 70800.0 4.83 211120.0 65500.0 4.88 6.8614 1.0 1914929 CBChromo1_000249 CC1(C)C(N(O)C(=O)Nc2cccc3ccccc23)N(C(=O)N1CC(=O)N/N=C/c4cc(Br)ccc4O)c5cccc6ccccc56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L08 compound treatment 160000.0 13100.0 0.89 156280.0 10700.0 0.8 1.1946 0.9984 1970309 CBChromo1_000250 CC1(C)CC(=O)C2=C(C1)OC3=C(C(=O)CC(C)(C)C3)C2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L09 compound treatment 169440.0 22500.0 1.54 165520.0 19900.0 1.48 2.136 0.9998 1913581 CBChromo1_000251 COc1ccc(cc1)C(=O)NC(NC(=S)Nc2ccc(N=Nc3ccccc3)cc2)C(Cl)(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L10 compound treatment 169600.0 22700.0 1.55 165840.0 20300.0 1.51 2.1605 0.9999 1375710 CBChromo1_000252 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(o4)c5cccc(Cl)c5)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L11 compound treatment 165000.0 18100.0 1.23 158800.0 13200.0 0.98 1.5683 0.9937 1914613 CBChromo1_000253 O=C(COc1ccccc1)NN=C2CCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L12 compound treatment 168480.0 21600.0 1.47 165160.0 19600.0 1.46 2.0707 1.0 1413142 CBChromo1_000254 Clc1ccc(cc1)C(=O)c2ccccc2C(=O)n3nnc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L13 compound treatment 161560.0 14700.0 1.0 164160.0 18600.0 1.38 1.6845 0.9873 3624434 CBChromo1_000255 Cc1ccc(cc1Br)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L14 compound treatment 177040.0 30100.0 2.05 181600.0 36000.0 2.68 3.3486 0.9914 1919882 CBChromo1_000256 CN1C(=O)N(C(=O)/C(=C/c2ccc3OCOc3c2)/C1=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L15 compound treatment 164080.0 17200.0 1.17 166040.0 20500.0 1.52 1.9049 0.9916 1147680 CBChromo1_000257 CCc1cccc(C)c1NC(=O)COc2cc(C)cc(C)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L16 compound treatment 174880.0 28000.0 1.91 177840.0 32300.0 2.4 3.0466 0.9935 1921275 CBChromo1_000258 Cc1[nH]c2ccccc2c1C(=O)/C=C/c3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L17 compound treatment 159520.0 12600.0 0.86 157280.0 11700.0 0.87 1.2241 1.0 1136335 CBChromo1_000259 COc1ccc(cc1)C(CC(=O)c2ccccc2)Nc3ccc(F)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L18 compound treatment 157320.0 10400.0 0.71 160160.0 14600.0 1.09 1.2696 0.9789 3624435 CBChromo1_000260 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nc4ccccc4s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L19 compound treatment 158400.0 11500.0 0.78 161360.0 15800.0 1.17 1.3848 0.9807 1860865 CBChromo1_000261 COc1ccc(cc1I)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L20 compound treatment 154120.0 7220.0 0.49 157280.0 11700.0 0.87 0.9638 0.9635 541 CBChromo1_000262 Cc1c(C)c(CONC(=O)c2ccccc2)c(C)c(C)c1Br 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L21 compound treatment 165560.0 18700.0 1.27 165800.0 20200.0 1.51 1.9636 0.9965 3624436 CBChromo1_000263 O=C(Nc1ccc2OCOc2c1)c3ccccc3NS(=O)(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L22 compound treatment 149560.0 2660.0 0.18 149480.0 3900.0 0.29 0.3334 0.9742 2027357 CBChromo1_000264 OCc1ccc(cc1)[C@@H]2C[C@H](CSc3nc(c(o3)c4ccccc4)c5ccccc5)O[C@@H](O2)c6ccc(NC(=O)CCCCCCC(=O)NO)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L23 mock treatment 148800.0 1900.0 0.13 149280.0 3700.0 0.28 0.2863 0.9406 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 L24 mock treatment 149600.0 2700.0 0.18 143280.0 -2300.0 -0.17 0.0091 0.0361 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M01 compound treatment 164240.0 17300.0 1.18 162440.0 16900.0 1.25 1.7232 0.9996 1432230 CBChromo1_000265 Cc1sc2ncnc(Nc3ccc(C)c(C)c3)c2c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M02 compound treatment 181880.0 35000.0 2.38 175400.0 29800.0 2.22 3.2556 0.9994 1921141 CBChromo1_000266 CCN1/C(=C/C=C/C=C/c2sc3ccccc3[n+]2CC(=O)O)/Sc4ccccc14 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M03 compound treatment 195440.0 48500.0 3.31 195680.0 50100.0 3.73 4.9766 0.9982 1914421 CBChromo1_000267 C/C(=N\Nc1ccccc1)/c2cc3ccccc3oc2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M04 compound treatment 206560.0 59700.0 4.07 201360.0 55800.0 4.15 5.8116 0.9999 1915319 CBChromo1_000268 Nc1ccc2oc3ccc(N)cc3c(=O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M05 compound treatment 196640.0 49700.0 3.39 188760.0 43200.0 3.21 4.6703 0.9996 1913842 CBChromo1_000269 Oc1cc2ccccc2cc1C(=O)N/N=C/c3ccccc3[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M06 compound treatment 176600.0 29700.0 2.02 170560.0 25000.0 1.86 2.7464 0.9991 1917785 CBChromo1_000270 O=C(Nc1ccc(/C=C/C(=O)c2ccccc2)cc1)C(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M07 compound treatment 166720.0 19800.0 1.35 166280.0 20700.0 1.54 2.0448 0.9979 1445757 CBChromo1_000271 COc1ccc(OC)c(c1)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M08 compound treatment 174680.0 27800.0 1.89 167240.0 21700.0 1.61 2.4791 0.9968 1919359 CBChromo1_000272 COc1cc(/C=N/c2ccc(NC(=O)C)cc2)cc(Br)c1OCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M09 compound treatment 165320.0 18400.0 1.26 162880.0 17300.0 1.29 1.7984 0.9999 1179853 CBChromo1_000273 Clc1ccc(NC(=O)c2ccccc2C(=O)OCC#C)c(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M10 compound treatment 187440.0 40500.0 2.76 185680.0 40100.0 2.98 4.0647 0.9993 1463503 CBChromo1_000274 N(C(c1ccccc1)c2ccncc2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M11 compound treatment 214840.0 67900.0 4.63 212560.0 67000.0 4.99 6.8002 0.9993 1913206 CBChromo1_000275 OC(=O)c1ccc(/N=C/c2ccc(O)cc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M12 compound treatment 166080.0 19200.0 1.31 166800.0 21200.0 1.58 2.0413 0.9956 1241870 CBChromo1_000276 COc1cccc(c1)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M13 compound treatment 183480.0 36600.0 2.49 185000.0 39400.0 2.93 3.838 0.9967 1307245 CBChromo1_000277 CCN(CC)c1ccc(cc1)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M14 compound treatment 161160.0 14300.0 0.97 160480.0 14900.0 1.11 1.4715 0.9978 1218208 CBChromo1_000278 COc1ccc(cc1)C(CC(=O)c2ccc(C)cc2)Nc3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M15 compound treatment 162400.0 15500.0 1.06 164200.0 18600.0 1.39 1.7271 0.991 1919544 CBChromo1_000279 [O-][N+](=O)c1cc(ccc1Br)C(=O)Oc2ccc(OC(=O)c3ccc(Br)c(c3)[N+](=O)[O-])c(c2)C(=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M16 compound treatment 173080.0 26200.0 1.78 169280.0 23700.0 1.76 2.5093 1.0 1935088 CBChromo1_000280 Clc1ccc2oc(nc2c1)c3cccc(NS(=O)(=O)c4ccccc4)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M17 compound treatment 167160.0 20300.0 1.38 162600.0 17000.0 1.27 1.8724 0.9991 1915136 CBChromo1_000281 C/C(=N\NC(=O)N)/c1cc(CNC(=O)CCl)cs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M18 compound treatment 159400.0 12500.0 0.85 161440.0 15900.0 1.18 1.4372 0.9872 3624437 CBChromo1_000282 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(Cl)c(Cl)c4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M19 compound treatment 290640.0 144000.0 9.8 322680.0 177000.0 13.18 16.2498 0.9893 1915304 CBChromo1_000283 CC1C=CC(=C(O)C1C(=O)O)N=Nc2ccc(cc2)c3ccc(N=Nc4ccc(C)c(C(=O)O)c4O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M20 compound treatment 158160.0 11300.0 0.77 162520.0 16900.0 1.26 1.4343 0.9717 1614005 CBChromo1_000284 CCc1ccccc1NC(=O)CN(c2ccc(C)cc2)S(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M21 compound treatment 187560.0 40700.0 2.77 185680.0 40100.0 2.98 4.0705 0.9993 1919995 CBChromo1_000285 CCn1c2ccccc2c3cc(/C=N/NC(=O)c4ccccc4O)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M22 compound treatment 194400.0 47500.0 3.24 194560.0 49000.0 3.65 4.8675 0.9983 1925163 CBChromo1_000286 COC(=O)C(=O)/C(=C\c1ccc(o1)c2ccccc2[N+](=O)[O-])/C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M23 mock treatment 154320.0 7420.0 0.51 151400.0 5820.0 0.43 0.6639 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 M24 mock treatment 148840.0 1940.0 0.13 148600.0 3020.0 0.22 0.2524 0.9678 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N01 compound treatment 172000.0 25100.0 1.71 168800.0 23200.0 1.73 2.432 1.0 1369355 CBChromo1_000287 Cc1cc(=O)oc2cc(OC(=O)COc3ccc4c(=O)c(c(C)oc4c3)c5ccc6OCCOc6c5)ccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N02 compound treatment 208440.0 61500.0 4.2 204040.0 58500.0 4.35 6.0433 0.9998 1917291 CBChromo1_000288 O=S1(=O)Nc2cc3nc4ccccc4nc3c5cccc1c25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N03 compound treatment 156400.0 9500.0 0.65 153480.0 7900.0 0.59 0.8737 0.9988 1035127 CBChromo1_000289 O=C(NN=c1c(=O)c2ccccc2c1=O)c3ccncc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N04 compound treatment 171200.0 24300.0 1.66 167040.0 21500.0 1.6 2.3008 0.9998 1975127 CBChromo1_000290 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4cccc5ccccc45)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N05 compound treatment 210840.0 63900.0 4.36 204600.0 59000.0 4.39 6.1885 1.0 1914450 CBChromo1_000291 OC(=O)c1ccc(Nc2nc(Cl)nc(Cl)n2)cc1c3c4ccc(O)cc4oc5cc(=O)ccc35 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N06 compound treatment 184640.0 37700.0 2.57 178440.0 32900.0 2.45 3.5487 0.9997 1734841 CBChromo1_000292 COc1cc(ccc1O)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N07 compound treatment 160720.0 13800.0 0.94 163080.0 17500.0 1.3 1.5872 0.9873 1085540 CBChromo1_000293 O=C(COc1ccccc1)NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N08 compound treatment 165480.0 18600.0 1.27 164480.0 18900.0 1.41 1.8903 0.9986 1361475 CBChromo1_000294 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4cccc(O)c4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N09 compound treatment 165080.0 18200.0 1.24 163160.0 17600.0 1.31 1.8016 0.9996 1920541 CBChromo1_000295 CC(=O)Cc1ccccc1OC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N10 compound treatment 163080.0 16200.0 1.1 164600.0 19000.0 1.42 1.7809 0.9924 3624438 CBChromo1_000296 Fc1cccc(Cl)c1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N11 compound treatment 177280.0 30400.0 2.07 171200.0 25600.0 1.91 2.8128 0.9991 1918269 CBChromo1_000297 O=C(N/N=C\c1c[nH]c2ccccc12)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N12 compound treatment 179520.0 32600.0 2.22 174040.0 28500.0 2.12 3.0703 0.9997 1135840 CBChromo1_000298 CCN(CC)c1ccc(cc1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N13 compound treatment 170240.0 23300.0 1.59 164760.0 19200.0 1.43 2.1345 0.9985 1335771 CBChromo1_000299 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4cccc(F)c4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N14 compound treatment 167600.0 20700.0 1.41 170000.0 24400.0 1.82 2.283 0.9922 1919988 CBChromo1_000300 Oc1[nH]c(SCC(=O)N2CCCCC2)nc(=O)c1C(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N15 compound treatment 161800.0 14900.0 1.02 163120.0 17500.0 1.31 1.6413 0.9923 3624439 CBChromo1_000301 Cc1ccc(COc2cccc(c2)C3C4=C(CC(C)(C)CC4=O)OC5=C3C(=O)CC(C)(C)C5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N16 compound treatment 163440.0 16500.0 1.13 163880.0 18300.0 1.36 1.7604 0.9956 1154816 CBChromo1_000302 CC(NC(=S)c1cccnc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N17 compound treatment 163760.0 16900.0 1.15 167960.0 22400.0 1.67 1.9905 0.9836 1552144 CBChromo1_000303 CN(c1ccccc1)c2ccc(cc2)C3C4=C(CC(C)(C)CC4=O)OC5=C3C(=O)CC(C)(C)C5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N18 compound treatment 158080.0 11200.0 0.76 159000.0 13400.0 1.0 1.2452 0.9911 1924578 CBChromo1_000304 COCCCNC(=O)C(=O)Nc1ccc(Cl)cc1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N19 compound treatment 183640.0 36700.0 2.5 185400.0 39800.0 2.96 3.8668 0.9965 1165782 CBChromo1_000305 CCOc1ccc(NCC(=O)Nc2ccc(C)cc2C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N20 compound treatment 155800.0 8900.0 0.61 156720.0 11100.0 0.83 1.0153 0.9882 529 CBChromo1_000306 Nc1ccccc1NC(=O)c2ccc(CNC(=O)OCc3cccnc3)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N21 compound treatment 164120.0 17200.0 1.17 166760.0 21200.0 1.58 1.9447 0.9895 3624440 CBChromo1_000307 COc1ccc(OC)c(NC(=O)CNc2cccc(C)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N22 compound treatment 151320.0 4420.0 0.3 154160.0 8580.0 0.64 0.6646 0.9412 719 CBChromo1_000308 CN(CC#C)Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N23 mock treatment 146800.0 -103.0 -0.01 145520.0 -58.8 0.0 -0.008 -0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 N24 mock treatment 148320.0 1420.0 0.1 145400.0 -179.0 -0.01 0.0589 0.6041 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O01 compound treatment 175920.0 29000.0 1.98 171320.0 25700.0 1.92 2.7536 0.9999 1921786 CBChromo1_000309 Cc1ccc(/C=N/C(=N\NC(=O)c2ccccc2)/c3ccccc3)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O02 compound treatment 154280.0 7380.0 0.5 153600.0 8020.0 0.6 0.7778 0.9964 1913281 CBChromo1_000310 CN(N=c1c(=O)c2ccccc2c1=O)C(=N)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O03 compound treatment 161240.0 14300.0 0.98 166600.0 21000.0 1.56 1.7975 0.9744 1914260 CBChromo1_000311 CCOc1ccc(cc1)C(Nc2ccc(Br)cc2)P3(=O)OCCCO3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O04 compound treatment 165240.0 18300.0 1.25 161680.0 16100.0 1.2 1.7314 0.9998 1920814 CBChromo1_000312 [O-][N+](=O)c1ccc(NC(NC(=O)c2ccccc2Cl)C(Cl)(Cl)Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O05 compound treatment 153320.0 6420.0 0.44 146160.0 581.0 0.04 0.34 0.7733 1913661 CBChromo1_000313 Oc1ccccc1C(=O)N/N=C/c2ccco2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O06 compound treatment 188160.0 41300.0 2.81 185200.0 39600.0 2.95 4.0741 0.9997 1921127 CBChromo1_000314 C/C(=N\NC(=O)COc1c(C)cc(cc1C)[N+](=O)[O-])/c2cccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O07 compound treatment 159520.0 12600.0 0.86 162760.0 17200.0 1.28 1.5125 0.9814 1921659 CBChromo1_000315 CC(OS(=O)(=O)c1ccccc1)C(F)(F)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O08 compound treatment 165240.0 18300.0 1.25 158760.0 13200.0 0.98 1.5777 0.9928 1474431 CBChromo1_000316 CN1CCN(CC1)C(=O)c2sc3ccccc3c2Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O09 compound treatment 173440.0 26500.0 1.81 169040.0 23500.0 1.75 2.514 0.9998 1036003 CBChromo1_000317 NC(Cc1c[nH]c2ccc(OCc3ccccc3)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O10 compound treatment 165000.0 18100.0 1.23 158200.0 12600.0 0.94 1.5367 0.9909 1919255 CBChromo1_000318 Cc1cc(C)c(C(=O)/C=C/c2ccccc2)c(=O)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O11 compound treatment 157640.0 10700.0 0.73 151480.0 5900.0 0.44 0.8282 0.9701 1920522 CBChromo1_000319 O=C1C(=C(C(=O)c2ccccc12)[n+]3ccc4ccccc4c3)NS(=O)(=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O12 compound treatment 188640.0 41700.0 2.85 182680.0 37100.0 2.76 3.9647 0.9999 3624441 CBChromo1_000320 CCOc1cccc(c1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O13 compound treatment 164640.0 17700.0 1.21 162200.0 16600.0 1.24 1.7298 0.9999 1696710 CBChromo1_000321 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccccc4O)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O14 compound treatment 164320.0 17400.0 1.19 160000.0 14400.0 1.07 1.5986 0.9987 1440513 CBChromo1_000322 COc1ccc(cc1)C(CC(=O)c2ccc(Cl)cc2)Nc3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O15 compound treatment 222000.0 75100.0 5.12 218200.0 72600.0 5.4 7.4422 0.9996 1919154 CBChromo1_000323 Cc1cc(c2cccnc2c1O)C3(OC(=O)c4ccccc43)c5cc(C)c(O)c6ncccc56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O16 compound treatment 164560.0 17700.0 1.2 166840.0 21300.0 1.58 1.9702 0.9909 1262202 CBChromo1_000324 Clc1ccc(Br)cc1c2nc3cc(NS(=O)(=O)c4ccccc4)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O17 compound treatment 153800.0 6900.0 0.47 155360.0 9780.0 0.73 0.8473 0.9776 1569049 CBChromo1_000325 COc1ccc(cc1)C(CC(=O)c2ccccc2)Nc3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O18 compound treatment 161640.0 14700.0 1.0 164120.0 18500.0 1.38 1.6863 0.9878 1924572 CBChromo1_000326 COc1ccc(C/C(=N/OC(=O)c2cccs2)/N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O19 compound treatment 171600.0 24700.0 1.68 177520.0 31900.0 2.38 2.8716 0.9857 1918841 CBChromo1_000327 [O-][N+](=O)c1cc2OCOc2cc1/C=N/NC(=O)C3CC3(c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O20 compound treatment 180760.0 33900.0 2.31 182600.0 37000.0 2.76 3.5806 0.9961 1386229 CBChromo1_000328 CCOc1cc(ccc1OCC=C)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O21 compound treatment 151120.0 4220.0 0.29 159040.0 13500.0 1.0 0.9118 0.8747 1919956 CBChromo1_000329 CCn1c2ccccc2c3cc(/C=N/N=C/c4ccc5n(CC)c6ccccc6c5c4)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O22 compound treatment 152640.0 5740.0 0.39 148160.0 2580.0 0.19 0.4124 0.9464 1973247 CBChromo1_000330 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4cc(Cl)ccc4O)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O23 mock treatment 147600.0 698.0 0.05 145640.0 61.3 0.0 0.0368 0.7714 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 O24 mock treatment 150240.0 3340.0 0.23 144120.0 -1460.0 -0.11 0.0841 0.3337 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P01 compound treatment 159960.0 13100.0 0.89 156440.0 10900.0 0.81 1.2011 0.9988 1915000 CBChromo1_000331 CCc1nnc(NS(=O)(=O)c2ccc(NC(=S)NC(=O)/C=C/c3ccc(OC)c(OC)c3)cc2)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P02 compound treatment 177720.0 30800.0 2.1 177880.0 32300.0 2.4 3.1856 0.9977 1918260 CBChromo1_000332 [O-][n+]1ccc(N/N=C/c2ccccc2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P03 compound treatment 172240.0 25300.0 1.73 175080.0 29500.0 2.2 2.7741 0.993 1913472 CBChromo1_000333 [O-][N+](=O)c1ccc(cc1)S(=O)(=O)NNC(=O)c2ccncc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P04 compound treatment 161760.0 14900.0 1.01 157000.0 11400.0 0.85 1.3173 0.9962 1604763 CBChromo1_000334 CC1(C)CC(=O)C2=C(C1)OC3=C(C2c4ccc(O)cc4)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P05 compound treatment 156560.0 9660.0 0.66 155800.0 10200.0 0.76 1.0035 0.9974 1016032 CBChromo1_000335 COC(=O)C1CC2(CC(CC(C(=O)OC)C2=O)(C(=O)OC)C1=O)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P06 compound treatment 166200.0 19300.0 1.32 160240.0 14700.0 1.09 1.7019 0.9957 1921369 CBChromo1_000336 C/C(=N\NC(=S)N1CCOCC1)/c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P07 compound treatment 167080.0 20200.0 1.38 166840.0 21300.0 1.58 2.0917 0.9976 1362155 CBChromo1_000337 Cc1cccc(OCC(=O)Nc2cccc(O)c2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P08 compound treatment 162360.0 15500.0 1.05 158280.0 12700.0 0.95 1.4136 0.9985 1726183 CBChromo1_000338 Cc1cccc(OCC(=O)Nc2c(C)cccc2C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P09 compound treatment 169040.0 22100.0 1.51 163880.0 18300.0 1.36 2.0304 0.9987 1729379 CBChromo1_000339 ONC(=O)C1(CCCC2CCC1)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P10 compound treatment 157920.0 11000.0 0.75 160320.0 14700.0 1.1 1.3069 0.9829 3624442 CBChromo1_000340 Fc1cccc(F)c1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P11 compound treatment 159440.0 12500.0 0.85 155760.0 10200.0 0.76 1.1402 0.9982 3624443 CBChromo1_000341 CC1(C)CC(=O)C2=C(C1)OC3=C(C2C=C(Cl)Cl)C(=O)CC(C)(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P12 compound treatment 175680.0 28800.0 1.96 172760.0 27200.0 2.02 2.8178 0.9999 1928477 CBChromo1_000342 Clc1ccc(Cl)c(c1)C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P13 compound treatment 183120.0 36200.0 2.47 172200.0 26600.0 1.98 3.147 0.994 3624444 CBChromo1_000343 Cc1ccc2oc(nc2c1)c3cccc(NS(=O)(=O)c4ccc(Cl)cc4)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P14 compound treatment 172720.0 25800.0 1.76 168040.0 22500.0 1.67 2.4267 0.9997 1920301 CBChromo1_000344 C/C(=C/1\C(=NN(C1=O)c2ccc(Br)cc2Br)C)/NCc3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P15 compound treatment 160240.0 13300.0 0.91 161680.0 16100.0 1.2 1.4904 0.9907 3624445 CBChromo1_000345 CCOc1ccc(cc1Cl)C2C3=C(CC(C)(C)CC3=O)OC4=C2C(=O)CC(C)(C)C4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P16 compound treatment 163280.0 16400.0 1.12 155040.0 9460.0 0.7 1.2875 0.9753 1287603 CBChromo1_000346 ONC(=O)CCn1c2ccccc2c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P17 compound treatment 179720.0 32800.0 2.24 177520.0 31900.0 2.38 3.2631 0.9995 3624446 CBChromo1_000347 COc1ccccc1C(=O)n2nnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P18 compound treatment 175520.0 28600.0 1.95 171000.0 25400.0 1.89 2.7175 0.9999 1735115 CBChromo1_000348 Cc1ccc2oc(nc2c1)c3cccc(NS(=O)(=O)c4ccccc4)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P19 compound treatment 160160.0 13300.0 0.9 155720.0 10100.0 0.75 1.1728 0.996 3624447 CBChromo1_000349 COc1ccc(NC(CC(=O)c2ccc(Cl)cc2)c3ccccc3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P20 compound treatment 150920.0 4020.0 0.27 148400.0 2820.0 0.21 0.3422 0.9914 1019 CBChromo1_000350 NC(=O)N1c2ccccc2C=Cc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P21 compound treatment 148240.0 1340.0 0.09 148960.0 3380.0 0.25 0.2424 0.9057 3624448 CBChromo1_000351 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3nc4cc(C)ccc4o3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P22 compound treatment 148760.0 1860.0 0.13 150280.0 4700.0 0.35 0.337 0.9055 3198425 CBChromo1_000352 CC1(C)O[C@@H]2CO[C@@]3(COS(=O)(=O)N)OC(C)(C)O[C@H]3[C@@H]2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P23 mock treatment 146880.0 -22.5 0.0 150080.0 4500.0 0.34 0.2358 0.7039 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2417 P24 mock treatment 144680.0 -2220.0 -0.15 148600.0 3020.0 0.22 0.0519 0.1913 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A01 mock treatment 150480.0 -8270.0 -0.56 152360.0 -2230.0 -0.17 -0.5162 -0.8781 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A02 mock treatment 149480.0 -9270.0 -0.63 150680.0 -3910.0 -0.29 -0.6528 -0.9381 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A03 compound treatment 157800.0 -951.0 -0.06 153880.0 -712.0 -0.05 -0.0833 -0.995 3635560 CMLD6_000001 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/Cc5ccccc5)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A04 compound treatment 158160.0 -591.0 -0.04 153280.0 -1310.0 -0.1 -0.0975 -0.9234 3635562 CMLD6_000002 CN1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A05 compound treatment 153840.0 -4910.0 -0.33 148560.0 -6030.0 -0.45 -0.5542 -0.9896 3635564 CMLD6_000003 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CCOC)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A06 compound treatment 158960.0 209.0 0.01 154640.0 48.2 0.0 0.0126 0.8584 3635566 CMLD6_000004 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(Cc4ccc(cc4)c5ccccc5)[C@H](c6ccccc6)C73CC2(C7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A07 compound treatment 154320.0 -4430.0 -0.3 149240.0 -5350.0 -0.4 -0.4953 -0.9907 3635568 CMLD6_000005 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC5CC5)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A08 compound treatment 160200.0 1450.0 0.1 152880.0 -1710.0 -0.13 -0.0202 -0.1255 3635570 CMLD6_000006 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A09 compound treatment 158320.0 -431.0 -0.03 155800.0 1210.0 0.09 0.0428 0.4525 3635572 CMLD6_000007 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/Cc5ccccc5)C1=O)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A10 compound treatment 172320.0 13600.0 0.93 161000.0 6410.0 0.48 0.9914 0.9525 3635574 CMLD6_000008 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccc(cc7)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A11 compound treatment 148400.0 -10400.0 -0.71 144800.0 -9790.0 -0.73 -1.0143 -0.9999 3635576 CMLD6_000009 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCc5c[nH]c6ccccc56)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A12 compound treatment 173160.0 14400.0 0.98 167320.0 12700.0 0.95 1.3645 0.9998 3635578 CMLD6_000010 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccccc4)C5(CC3(C5)[C@H]2c6ccccc6)c7cccnc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A13 compound treatment 209800.0 51000.0 3.48 186680.0 32100.0 2.39 4.1497 0.9831 3635580 CMLD6_000011 C[C@@H]1[C@H]2[C@@H]([C@@H]3C[C@@H]4[C@H]([C@@H]5C3=C1C(=O)N6C(=O)O/C(=N\CCc7c[nH]c8ccccc78)/[C@]56Cc9ccccc9)C(=O)N(C4=O)c%10ccccc%10)C(=O)N(C2=O)c%11ccccc%11 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A14 compound treatment 157440.0 -1310.0 -0.09 151840.0 -2750.0 -0.2 -0.208 -0.9309 3635582 CMLD6_000012 CN1C[C@@H]2C(c3ccc(cc3)C(F)(F)F)C4(CC2(C4)[C@H]1c5ccccc5)c6ccc(C#N)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A15 compound treatment 152200.0 -6550.0 -0.45 149520.0 -5070.0 -0.38 -0.5827 -0.9965 3635584 CMLD6_000013 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CCOC)C1=O)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A16 compound treatment 156440.0 -2310.0 -0.16 149480.0 -5110.0 -0.38 -0.3804 -0.9239 3635586 CMLD6_000014 Clc1ccc(cn1)C2[C@H]3CN(Cc4ccc(cc4)c5ccccc5)[C@H](c6ccccc6)C73CC2(C7)c8ccc(C#N)cc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A17 compound treatment 153160.0 -5590.0 -0.38 150520.0 -4070.0 -0.3 -0.4838 -0.9935 3635588 CMLD6_000015 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC(=O)OC)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A18 compound treatment 165840.0 7090.0 0.48 159640.0 5050.0 0.38 0.6074 0.9922 3635590 CMLD6_000016 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccc(Cl)nc4)C5(CC3(C5)[C@H]2c6ccccc6)c7cccnc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A19 compound treatment 149080.0 -9670.0 -0.66 149120.0 -5470.0 -0.41 -0.7542 -0.9732 3635592 CMLD6_000017 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CC5CC5)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A20 compound treatment 151000.0 -7750.0 -0.53 149000.0 -5590.0 -0.42 -0.6679 -0.993 3635594 CMLD6_000018 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(C)[C@@H]3c5ccccc5)c6ccc(cc6)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A21 compound treatment 152600.0 -6150.0 -0.42 148200.0 -6390.0 -0.48 -0.6329 -0.998 3635596 CMLD6_000019 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC5CC5)C4=O)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A22 compound treatment 157800.0 -951.0 -0.06 154640.0 48.2 0.0 -0.0433 -0.667 3635598 CMLD6_000020 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccc(Cl)nc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A23 mock treatment 149840.0 -8910.0 -0.61 140520.0 -14100.0 -1.05 -1.1702 -0.9665 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 A24 mock treatment 150240.0 -8510.0 -0.58 143520.0 -11100.0 -0.82 -0.993 -0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B01 mock treatment 147520.0 -11200.0 -0.77 141880.0 -12700.0 -0.95 -1.2104 -0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B02 mock treatment 149880.0 -8870.0 -0.6 144400.0 -10200.0 -0.76 -0.964 -0.9937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B03 compound treatment 179720.0 21000.0 1.43 173040.0 18400.0 1.37 1.9818 0.9998 3635600 CMLD6_000021 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(cc3)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B04 compound treatment 146440.0 -12300.0 -0.84 145600.0 -8990.0 -0.67 -1.0667 -0.9937 3635602 CMLD6_000022 O=C(CC#N)NC(=O)NCC1CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B05 compound treatment 154440.0 -4310.0 -0.29 154800.0 208.0 0.02 -0.1969 -0.6689 3635603 CMLD6_000023 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3cc(F)ccc3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B06 compound treatment 150360.0 -8390.0 -0.57 147520.0 -7070.0 -0.53 -0.7767 -0.9991 1042488 CMLD6_000024 Nc1cc(=O)[nH]c(=O)n1Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B07 compound treatment 147080.0 -11700.0 -0.8 152080.0 -2510.0 -0.19 -0.6948 -0.8501 3635605 CMLD6_000025 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(C)s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B08 compound treatment 145400.0 -13400.0 -0.91 145920.0 -8670.0 -0.65 -1.1 -0.9858 3635607 CMLD6_000026 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC5CC5)C4=O)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B09 compound treatment 155680.0 -3070.0 -0.21 144000.0 -10600.0 -0.79 -0.7055 -0.8649 3635609 CMLD6_000027 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B10 compound treatment 188280.0 29500.0 2.01 176360.0 21800.0 1.62 2.5692 0.9942 3635611 CMLD6_000028 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3c(F)cccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B11 compound treatment 226200.0 67400.0 4.6 223160.0 68600.0 5.1 6.8602 0.9986 3635613 CMLD6_000029 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccco4)c(N)n(Cc5ccccc5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B12 mock treatment 155680.0 -3070.0 -0.21 150240.0 -4350.0 -0.32 -0.3771 -0.9777 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B13 compound treatment 235320.0 76600.0 5.22 215440.0 60800.0 4.53 6.8936 0.9975 3635614 CMLD6_000030 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccco4)c(N)n(CC5CC5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B14 mock treatment 149120.0 -9630.0 -0.66 147000.0 -7590.0 -0.57 -0.8638 -0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B15 compound treatment 149520.0 -9230.0 -0.63 153320.0 -1270.0 -0.09 -0.5119 -0.8044 3635615 CMLD6_000031 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3c(cccc23)C(F)(F)F)C(F)(F)F)c(N)n(Cc4ccccc4)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B16 mock treatment 150560.0 -8190.0 -0.56 144520.0 -10100.0 -0.75 -0.9249 -0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B17 compound treatment 158200.0 -551.0 -0.04 155800.0 1210.0 0.09 0.037 0.3799 3635616 CMLD6_000032 COC(=O)CC1Oc2cc3oc4CC(C)(C)CC(=O)c4c3cc2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B18 mock treatment 154280.0 -4470.0 -0.3 149240.0 -5350.0 -0.4 -0.4972 -0.9913 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B19 compound treatment 172320.0 13600.0 0.93 169520.0 14900.0 1.11 1.4398 0.9959 3635617 CMLD6_000033 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B20 mock treatment 151800.0 -6950.0 -0.47 150080.0 -4510.0 -0.34 -0.5725 -0.9858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B21 compound treatment 150640.0 -8110.0 -0.55 144480.0 -10100.0 -0.75 -0.9232 -0.9885 1057869 CMLD6_000034 NC(=O)NCc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B22 mock treatment 153120.0 -5630.0 -0.38 145720.0 -8870.0 -0.66 -0.7384 -0.9667 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B23 mock treatment 151400.0 -7350.0 -0.5 149200.0 -5390.0 -0.4 -0.6381 -0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 B24 mock treatment 147160.0 -11600.0 -0.79 142920.0 -11700.0 -0.87 -1.173 -0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C01 mock treatment 151480.0 -7270.0 -0.5 150880.0 -3710.0 -0.28 -0.5459 -0.9619 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C02 mock treatment 155520.0 -3230.0 -0.22 154000.0 -592.0 -0.04 -0.1869 -0.832 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C03 compound treatment 159680.0 929.0 0.06 152840.0 -1750.0 -0.13 -0.0474 -0.3271 3635619 CMLD6_000035 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/Cc5ccccc5)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C04 compound treatment 172400.0 13600.0 0.93 160720.0 6130.0 0.46 0.9805 0.9462 3635621 CMLD6_000036 C(C1CCCCC1)N2C[C@@H]3C(c4ccccc4)C5(CC3(C5)[C@H]2c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C05 compound treatment 172960.0 14200.0 0.97 161760.0 7170.0 0.53 1.0622 0.9605 3635623 CMLD6_000037 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)O/C(=N\CCOC)/[C@]4(Cc5ccccc5)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C06 compound treatment 186520.0 27800.0 1.89 181880.0 27300.0 2.03 2.7748 0.9994 3635625 CMLD6_000038 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(Cc4cccnc4)[C@H](c5ccccc5)C63CC2(C6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C07 compound treatment 150480.0 -8270.0 -0.56 152520.0 -2070.0 -0.15 -0.5078 -0.8686 3635627 CMLD6_000039 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC5CC5)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C08 compound treatment 165560.0 6810.0 0.46 162280.0 7690.0 0.57 0.7329 0.9946 3635629 CMLD6_000040 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)C(F)(F)F)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C09 compound treatment 161560.0 2810.0 0.19 150320.0 -4270.0 -0.32 -0.0894 -0.2409 3635631 CMLD6_000041 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC(=O)OC)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C10 compound treatment 175600.0 16800.0 1.15 162600.0 8010.0 0.6 1.2337 0.9533 3635633 CMLD6_000042 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(C)[C@@H]3c5ccccc5)c6ccc(Cl)nc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C11 compound treatment 156560.0 -2190.0 -0.15 150120.0 -4470.0 -0.33 -0.341 -0.9347 3635635 CMLD6_000043 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCc5c[nH]c6ccccc56)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C12 compound treatment 172640.0 13900.0 0.95 159160.0 4570.0 0.34 0.91 0.9045 3635637 CMLD6_000044 C(N1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6cccnc6)c7ccc(cc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C13 compound treatment 181560.0 22800.0 1.56 166760.0 12200.0 0.91 1.74 0.9669 3635639 CMLD6_000045 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C1=O)C(=O)N(C3=O)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C14 compound treatment 167000.0 8250.0 0.56 156160.0 1570.0 0.12 0.4802 0.836 3635641 CMLD6_000046 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(CC4CCCCC4)[C@H](c5ccccc5)C63CC2(C6)c7ccc(C#N)cc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C15 compound treatment 160160.0 1410.0 0.1 152760.0 -1830.0 -0.14 -0.0285 -0.1708 3635643 CMLD6_000047 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCOC)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C16 compound treatment 164800.0 6050.0 0.41 150080.0 -4510.0 -0.34 0.0542 0.1018 3635645 CMLD6_000048 CN1C[C@@H]2C(c3ccc(cc3)C(F)(F)F)C4(CC2(C4)[C@H]1c5ccccc5)c6cccnc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C17 compound treatment 154880.0 -3870.0 -0.26 151360.0 -3230.0 -0.24 -0.3567 -0.9989 3635647 CMLD6_000049 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CC(=O)OC)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C18 compound treatment 162000.0 3250.0 0.22 162760.0 8170.0 0.61 0.5865 0.9064 3635649 CMLD6_000050 Clc1ccc(cn1)C2[C@H]3CN(Cc4ccc(cc4)c5ccccc5)[C@H](c6ccccc6)C73CC2(C7)c8cccnc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C19 compound treatment 155120.0 -3630.0 -0.25 152720.0 -1870.0 -0.14 -0.2736 -0.963 3635651 CMLD6_000051 CCN1C(=O)[C@@H]2C[C@H]3[C@@H]4[C@H]([C@@H](C)C5=C3[C@@H]([C@@H]2C1=O)[C@]/6(C)N(C(=O)O\C6=N/CC7CC7)C5=O)C(=O)N(CC)C4=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C20 compound treatment 154440.0 -4310.0 -0.29 157240.0 2650.0 0.2 -0.0685 -0.1935 3635653 CMLD6_000052 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccc(cc7)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C21 compound treatment 158280.0 -471.0 -0.03 147280.0 -7310.0 -0.54 -0.4075 -0.7475 3635655 CMLD6_000053 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)N(CC5CC5)C(=O)[C@]4(Cc6ccccc6)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C22 compound treatment 156200.0 -2550.0 -0.17 158600.0 4010.0 0.3 0.088 0.2547 3635657 CMLD6_000054 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccc(Cl)nc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C23 mock treatment 146960.0 -11800.0 -0.8 144560.0 -10000.0 -0.75 -1.0964 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 C24 mock treatment 148920.0 -9830.0 -0.67 145640.0 -8950.0 -0.67 -0.9451 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D01 mock treatment 153320.0 -5430.0 -0.37 149440.0 -5150.0 -0.38 -0.5329 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D02 mock treatment 149360.0 -9390.0 -0.64 152480.0 -2110.0 -0.16 -0.5639 -0.8553 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D03 compound treatment 153320.0 -5430.0 -0.37 149600.0 -4990.0 -0.37 -0.5245 -1.0 3635659 CMLD6_000055 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D04 compound treatment 154120.0 -4630.0 -0.32 149080.0 -5510.0 -0.41 -0.5133 -0.9916 3635661 CMLD6_000056 CN(C)/C=N/c1cc(=O)n(Cc2ccccc2)c(=O)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D05 compound treatment 159120.0 369.0 0.03 156640.0 2050.0 0.15 0.1256 0.8128 3635663 CMLD6_000057 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3cc(OC)cc(OC)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D06 compound treatment 156480.0 -2270.0 -0.15 150960.0 -3630.0 -0.27 -0.3006 -0.965 3635665 CMLD6_000058 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCOC)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D07 compound treatment 155640.0 -3110.0 -0.21 151080.0 -3510.0 -0.26 -0.3348 -0.9946 3635667 CMLD6_000059 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3cccc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D08 compound treatment 149560.0 -9190.0 -0.63 150480.0 -4110.0 -0.31 -0.6595 -0.9457 3635669 CMLD6_000060 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC5CC5)C4=O)C1=O)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D09 compound treatment 220560.0 61800.0 4.21 212960.0 58400.0 4.34 6.0515 0.9999 3635671 CMLD6_000061 COc1c(O)c(O)cc2c1oc3c2c(=O)oc4ccc(C)cc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D10 compound treatment 192640.0 33900.0 2.31 186680.0 32100.0 2.39 3.3225 0.9999 3635672 CMLD6_000062 COC(=O)[C@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3c(F)cccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D11 compound treatment 159440.0 689.0 0.05 154640.0 48.2 0.0 0.0357 0.7589 3635673 CMLD6_000063 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)C(F)(F)F)c(=O)n(Cc4ccccc4)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D12 mock treatment 157600.0 -1150.0 -0.08 149920.0 -4670.0 -0.35 -0.3014 -0.8454 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D13 compound treatment 158360.0 -391.0 -0.03 148960.0 -5630.0 -0.42 -0.3152 -0.7506 3635674 CMLD6_000064 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccccc4)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D14 mock treatment 156360.0 -2390.0 -0.16 152680.0 -1910.0 -0.14 -0.2159 -0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D15 compound treatment 233360.0 74600.0 5.09 204480.0 49900.0 3.71 6.2223 0.988 1364812 CMLD6_000065 Oc1cc2oc3c(c(=O)oc4ccccc34)c2cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D16 mock treatment 161040.0 2290.0 0.16 152640.0 -1950.0 -0.15 0.0076 0.0358 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D17 compound treatment 153080.0 -5670.0 -0.39 146040.0 -8550.0 -0.64 -0.7235 -0.9715 3635675 CMLD6_000066 CC(NC(=O)c1ccccc1)C(=O)OC(C)C#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D18 mock treatment 153240.0 -5510.0 -0.38 154760.0 168.0 0.01 -0.2568 -0.6832 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D19 compound treatment 185160.0 26400.0 1.8 180760.0 26200.0 1.95 2.6503 0.9992 3635676 CMLD6_000067 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D20 mock treatment 153160.0 -5590.0 -0.38 151880.0 -2710.0 -0.2 -0.4123 -0.9558 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D21 compound treatment 161480.0 2730.0 0.19 156000.0 1410.0 0.1 0.2057 0.9631 3635678 CMLD6_000068 CN(C)/C=N/c1cc(=O)[nH]c(=O)n1Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D22 mock treatment 149800.0 -8950.0 -0.61 147920.0 -6670.0 -0.5 -0.7826 -0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D23 mock treatment 149200.0 -9550.0 -0.65 146080.0 -8510.0 -0.63 -0.9084 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 D24 mock treatment 152120.0 -6630.0 -0.45 144800.0 -9790.0 -0.73 -0.835 -0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E01 mock treatment 161200.0 2450.0 0.17 156000.0 1410.0 0.1 0.1922 0.9748 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E02 mock treatment 162680.0 3930.0 0.27 157400.0 2810.0 0.21 0.3372 0.9925 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E03 compound treatment 175120.0 16400.0 1.12 166680.0 12100.0 0.9 1.4253 0.9943 3635680 CMLD6_000069 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/Cc5ccccc5)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E04 compound treatment 192400.0 33600.0 2.29 176400.0 21800.0 1.62 2.7699 0.9856 3635682 CMLD6_000070 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccccc4)C5(CC3(C5)[C@H]2c6ccccc6)c7ccccc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E05 compound treatment 169120.0 10400.0 0.71 156000.0 1410.0 0.1 0.574 0.8032 3635684 CMLD6_000071 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CCOC)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E06 compound treatment 191520.0 32800.0 2.23 179480.0 24900.0 1.85 2.8895 0.9957 3635686 CMLD6_000072 CN1C[C@@H]2C(c3ccc(Cl)nc3)C4(CC2(C4)[C@H]1c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E07 compound treatment 163840.0 5090.0 0.35 160000.0 5410.0 0.4 0.53 0.9973 3635688 CMLD6_000073 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC6CC6)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E08 compound treatment 172600.0 13800.0 0.94 167400.0 12800.0 0.95 1.3417 1.0 3635690 CMLD6_000074 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E09 compound treatment 158280.0 -471.0 -0.03 158240.0 3650.0 0.27 0.1693 0.6192 3635692 CMLD6_000075 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CC(=O)OC)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E10 compound treatment 181000.0 22200.0 1.52 169680.0 15100.0 1.12 1.8666 0.9891 3635694 CMLD6_000076 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccc(Cl)nc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E11 compound treatment 164960.0 6210.0 0.42 158960.0 4370.0 0.33 0.5292 0.9915 3635696 CMLD6_000077 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)O/C(=N\CCc5c[nH]c6ccccc56)/[C@]4(C)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E12 compound treatment 200800.0 42000.0 2.87 184280.0 29700.0 2.21 3.5895 0.9917 3635698 CMLD6_000078 C(N1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6cccnc6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E13 compound treatment 188160.0 29400.0 2.01 174000.0 19400.0 1.44 2.4392 0.9871 3635700 CMLD6_000079 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E14 compound treatment 183840.0 25100.0 1.71 170680.0 16100.0 1.2 2.0562 0.9848 3635702 CMLD6_000080 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccc(cc4)C(F)(F)F)C5(CC3(C5)[C@H]2c6ccccc6)c7ccc(C#N)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E15 compound treatment 163320.0 4570.0 0.31 161640.0 7050.0 0.52 0.5912 0.969 3635704 CMLD6_000081 COCC/N=C/1\OC(=O)N2C(=O)C3=C4[C@@H](C[C@@H]5[C@H]([C@H]4[C@]21Cc6ccccc6)C(=O)N(CC(=O)OC)C5=O)[C@@H]7[C@H]([C@H]3C)C(=O)N(CC(=O)OC)C7=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E16 compound treatment 173520.0 14800.0 1.01 163640.0 9050.0 0.67 1.1882 0.9809 3635706 CMLD6_000082 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(CC4CCCCC4)[C@H](c5ccccc5)C63CC2(C6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E17 compound treatment 162440.0 3690.0 0.25 155880.0 1290.0 0.1 0.2456 0.9126 3635708 CMLD6_000083 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CC(=O)OC)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E18 compound treatment 174760.0 16000.0 1.09 174720.0 20100.0 1.5 1.8311 0.9879 3635710 CMLD6_000084 Clc1ccc(cn1)C2[C@H]3CN(Cc4cccnc4)[C@H](c5ccccc5)C63CC2(C6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E19 compound treatment 159000.0 249.0 0.02 155960.0 1370.0 0.1 0.084 0.8137 3635712 CMLD6_000085 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CC5CC5)C1=O)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E20 compound treatment 165920.0 7170.0 0.49 158360.0 3770.0 0.28 0.5439 0.9652 3635714 CMLD6_000086 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)C(F)(F)F)[C@@H]3c6ccccc6)c7ccc(cc7)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E21 compound treatment 158360.0 -391.0 -0.03 152280.0 -2310.0 -0.17 -0.1405 -0.807 3635716 CMLD6_000087 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC5CC5)C4=O)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E22 compound treatment 189840.0 31100.0 2.12 189440.0 34800.0 2.59 3.3327 0.995 3635718 CMLD6_000088 Clc1ccc(cn1)C2[C@H]3CN([C@H](c4ccccc4)C53CC2(C5)c6ccc(C#N)cc6)P(=O)(c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E23 mock treatment 155520.0 -3230.0 -0.22 155640.0 1050.0 0.08 -0.1006 -0.4305 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 E24 mock treatment 155720.0 -3030.0 -0.21 149120.0 -5470.0 -0.41 -0.4341 -0.9505 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F01 mock treatment 160440.0 1690.0 0.12 155480.0 888.0 0.07 0.1282 0.9653 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F02 mock treatment 158760.0 8.93 0.0 152000.0 -2590.0 -0.19 -0.136 -0.7049 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F03 compound treatment 167440.0 8690.0 0.59 163280.0 8690.0 0.65 0.8761 0.999 3635720 CMLD6_000089 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F04 compound treatment 162360.0 3610.0 0.25 158000.0 3410.0 0.25 0.3533 0.9999 3635722 CMLD6_000090 Cn1c(=O)cc(N)n(Cc2ccccc2)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F05 compound treatment 159280.0 529.0 0.04 158640.0 4050.0 0.3 0.2385 0.7861 3635723 CMLD6_000091 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1CC(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F06 compound treatment 159240.0 489.0 0.03 157160.0 2570.0 0.19 0.1587 0.8181 3635725 CMLD6_000092 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CCOC)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F07 compound treatment 160080.0 1330.0 0.09 155880.0 1290.0 0.1 0.1319 0.9996 3635727 CMLD6_000093 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1C/C=C/c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F08 compound treatment 159520.0 769.0 0.05 155200.0 608.0 0.05 0.0691 0.9973 3635607 CMLD6_000094 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC5CC5)C4=O)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F09 compound treatment 166640.0 7890.0 0.54 162480.0 7890.0 0.59 0.7955 0.999 3635729 CMLD6_000095 COC(=O)CC1Oc2cc3oc4c(c(=O)oc5ccccc45)c3cc2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F10 compound treatment 187800.0 29000.0 1.98 186560.0 32000.0 2.38 3.0828 0.9958 3635730 CMLD6_000096 CCCN1[C@@H](C[C@@H]2CC[C@@H](O)C[C@@H]21)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F11 compound treatment 178960.0 20200.0 1.38 173920.0 19300.0 1.44 1.9914 0.9998 3635732 CMLD6_000097 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccccc4)c(=O)n(Cc5ccccc5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F12 mock treatment 162280.0 3530.0 0.24 156320.0 1730.0 0.13 0.2611 0.957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F13 compound treatment 164760.0 6010.0 0.41 149720.0 -4870.0 -0.36 0.0333 0.0608 3635733 CMLD6_000098 CC(C)Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccccc4)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F14 mock treatment 168000.0 9250.0 0.63 161000.0 6410.0 0.48 0.7831 0.9905 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F15 compound treatment 330640.0 172000.0 11.72 306640.0 152000.0 11.32 16.2884 0.9998 3635734 CMLD6_000099 COc1c(O)c(O)cc2c1oc3c2c(=O)oc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F16 mock treatment 167160.0 8410.0 0.57 159280.0 4690.0 0.35 0.6521 0.9717 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F17 compound treatment 160760.0 2010.0 0.14 158680.0 4090.0 0.3 0.312 0.935 3635735 CMLD6_000100 OC(=O)[C@H](Cc1ccccc1)NC(=O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F18 mock treatment 160360.0 1610.0 0.11 154080.0 -512.0 -0.04 0.0506 0.436 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F19 compound treatment 183800.0 25000.0 1.71 174760.0 20200.0 1.5 2.269 0.9979 3635736 CMLD6_000101 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(C)s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F20 mock treatment 160680.0 1930.0 0.13 152800.0 -1790.0 -0.13 -0.0013 -0.007 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F21 compound treatment 158640.0 -111.0 -0.01 151960.0 -2630.0 -0.2 -0.1439 -0.7339 3635738 CMLD6_000102 OC(=O)c1cc(nc2ccccc12)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F22 mock treatment 162640.0 3890.0 0.27 150640.0 -3950.0 -0.29 -0.0205 -0.0518 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F23 mock treatment 155920.0 -2830.0 -0.19 152920.0 -1670.0 -0.12 -0.2245 -0.9774 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 F24 mock treatment 146880.0 -11900.0 -0.81 149640.0 -4950.0 -0.37 -0.8329 -0.9366 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G01 mock treatment 160720.0 1970.0 0.13 157320.0 2730.0 0.2 0.2385 0.9798 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G02 mock treatment 169320.0 10600.0 0.72 164440.0 9850.0 0.73 1.0278 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G03 compound treatment 169920.0 11200.0 0.76 161480.0 6890.0 0.51 0.9009 0.9815 3635739 CMLD6_000103 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/Cc5ccccc5)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G04 compound treatment 173920.0 15200.0 1.03 166000.0 11400.0 0.85 1.3317 0.9952 3635741 CMLD6_000104 C(N1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6ccccc6)c7ccc(cc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G05 compound treatment 173120.0 14400.0 0.98 160960.0 6370.0 0.47 1.0278 0.9445 3635743 CMLD6_000105 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC(=O)OC)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G06 compound treatment 174280.0 15500.0 1.06 170080.0 15500.0 1.15 1.5637 0.9991 3635745 CMLD6_000106 Clc1ccc(cn1)C2[C@H]3CN(CC4CCCCC4)[C@H](c5ccccc5)C63CC2(C6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G07 compound treatment 171360.0 12600.0 0.86 169800.0 15200.0 1.13 1.4082 0.9908 3635747 CMLD6_000107 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC6CC6)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G08 compound treatment 198240.0 39500.0 2.69 186840.0 32200.0 2.4 3.6008 0.9984 3635749 CMLD6_000108 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G09 compound treatment 169440.0 10700.0 0.73 164960.0 10400.0 0.77 1.061 0.9996 3635751 CMLD6_000109 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC(=O)OC)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G10 compound treatment 201040.0 42300.0 2.88 189120.0 34500.0 2.57 3.8558 0.9984 3635753 CMLD6_000110 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)C(F)(F)F)[C@@H]3c6ccccc6)c7ccc(Cl)nc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G11 compound treatment 174200.0 15400.0 1.05 168680.0 14100.0 1.05 1.4862 1.0 3635755 CMLD6_000111 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CCc5c[nH]c6ccccc56)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G12 compound treatment 170240.0 11500.0 0.78 166800.0 12200.0 0.91 1.1964 0.9973 3635757 CMLD6_000112 CN1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6ccc(C#N)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G13 compound treatment 180160.0 21400.0 1.46 178400.0 23800.0 1.77 2.2851 0.9954 3635759 CMLD6_000113 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G14 compound treatment 179440.0 20700.0 1.41 167960.0 13400.0 0.99 1.7009 0.9854 3635761 CMLD6_000114 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(Cc4ccc(cc4)c5ccccc5)[C@H](c6ccccc6)C73CC2(C7)c8ccc(C#N)cc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G15 compound treatment 176440.0 17700.0 1.21 169560.0 15000.0 1.11 1.6405 0.9992 3635763 CMLD6_000115 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCOC)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G16 compound treatment 186600.0 27800.0 1.9 183800.0 29200.0 2.17 2.8797 0.9977 3635765 CMLD6_000116 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccc(cc4)C(F)(F)F)C5(CC3(C5)[C@H]2c6ccccc6)c7cccnc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G17 compound treatment 178280.0 19500.0 1.33 171720.0 17100.0 1.27 1.8429 0.9998 3635767 CMLD6_000117 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)N(Cc5ccccc5)C(=O)[C@]4(Cc6ccccc6)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G18 compound treatment 165880.0 7130.0 0.49 159200.0 4610.0 0.34 0.5862 0.9854 3635769 CMLD6_000118 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(C)[C@@H]3c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G19 compound treatment 170360.0 11600.0 0.79 165000.0 10400.0 0.77 1.1074 0.9999 3635771 CMLD6_000119 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CC6CC6)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G20 compound treatment 171720.0 13000.0 0.88 167600.0 13000.0 0.97 1.3098 0.999 3635773 CMLD6_000120 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccc(cc8)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G21 compound treatment 176600.0 17800.0 1.22 169240.0 14600.0 1.09 1.6314 0.9985 3635775 CMLD6_000121 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(cc3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G22 compound treatment 182240.0 23500.0 1.6 174640.0 20000.0 1.49 2.1875 0.9994 3635777 CMLD6_000122 COC(=O)c1cccc(C#CC(NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G23 mock treatment 159800.0 1050.0 0.07 155640.0 1050.0 0.08 0.1057 0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 G24 mock treatment 156720.0 -2030.0 -0.14 151360.0 -3230.0 -0.24 -0.268 -0.9656 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H01 mock treatment 161040.0 2290.0 0.16 158240.0 3650.0 0.27 0.3023 0.9654 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H02 mock treatment 159080.0 329.0 0.02 158960.0 4370.0 0.33 0.2457 0.7541 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H03 compound treatment 168160.0 9410.0 0.64 164600.0 10000.0 0.74 0.9803 0.9972 3635778 CMLD6_000123 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(cc3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H04 compound treatment 162320.0 3570.0 0.24 161640.0 7050.0 0.52 0.543 0.939 3635780 CMLD6_000124 Nc1cc(=O)[nH]c(=O)n1CC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H05 compound treatment 169120.0 10400.0 0.71 160880.0 6290.0 0.47 0.8308 0.9799 3635781 CMLD6_000125 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H06 compound treatment 169920.0 11200.0 0.76 165000.0 10400.0 0.77 1.0862 1.0 3635782 CMLD6_000126 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCOC)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H07 compound treatment 177240.0 18500.0 1.26 178040.0 23400.0 1.75 2.1253 0.9872 3635784 CMLD6_000127 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3cc(F)ccc3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H08 compound treatment 171600.0 12800.0 0.88 166960.0 12400.0 0.92 1.2703 0.9997 3635785 CMLD6_000128 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(Cc5ccccc5)C4=O)C1=O)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H09 compound treatment 172960.0 14200.0 0.97 168200.0 13600.0 1.01 1.4012 0.9998 3635787 CMLD6_000129 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)C4CC4)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H10 compound treatment 198520.0 39800.0 2.71 195200.0 40600.0 3.02 4.0543 0.9985 3635788 CMLD6_000130 COC(=O)[C@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3c(F)cccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H11 compound treatment 170240.0 11500.0 0.78 159240.0 4650.0 0.35 0.7985 0.9325 3635789 CMLD6_000131 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3c(cccc23)C(F)(F)F)C(F)(F)F)c(N)n(CC4CC4)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H12 mock treatment 166120.0 7370.0 0.5 165680.0 11100.0 0.83 0.9388 0.9717 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H13 compound treatment 254960.0 96200.0 6.56 242120.0 87500.0 6.51 9.2445 1.0 3635790 CMLD6_000132 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccco4)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H14 mock treatment 168480.0 9730.0 0.66 159920.0 5330.0 0.4 0.7494 0.9698 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H15 compound treatment 294520.0 136000.0 9.26 282000.0 127000.0 9.48 13.2504 0.9999 3635791 CMLD6_000133 Cc1c(O)c(O)cc2c1oc3c2c(=O)oc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H16 mock treatment 173440.0 14700.0 1.0 163520.0 8930.0 0.66 1.178 0.9802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H17 compound treatment 193600.0 34800.0 2.38 185120.0 30500.0 2.27 3.2866 0.9998 3635792 CMLD6_000134 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H18 mock treatment 161760.0 3010.0 0.21 159840.0 5250.0 0.39 0.4213 0.9548 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H19 compound treatment 164160.0 5410.0 0.37 165400.0 10800.0 0.8 0.8296 0.9375 3635793 CMLD6_000135 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1CC3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H20 mock treatment 162360.0 3610.0 0.25 155480.0 888.0 0.07 0.2207 0.8664 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H21 compound treatment 216520.0 57800.0 3.94 205840.0 51200.0 3.81 5.482 0.9999 1260538 CMLD6_000136 OC(=O)c1cc(nc2ccccc12)c3ccco3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H22 mock treatment 164280.0 5530.0 0.38 159600.0 5010.0 0.37 0.5301 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H23 mock treatment 156720.0 -2030.0 -0.14 155000.0 408.0 0.03 -0.0764 -0.5391 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 H24 mock treatment 155240.0 -3510.0 -0.24 154680.0 88.2 0.01 -0.1646 -0.6875 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I01 mock treatment 162560.0 3810.0 0.26 157400.0 2810.0 0.21 0.3314 0.9942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I02 mock treatment 163760.0 5010.0 0.34 157080.0 2490.0 0.19 0.3724 0.9587 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I03 compound treatment 164360.0 5610.0 0.38 158960.0 4370.0 0.33 0.5003 0.9967 3635795 CMLD6_000137 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC(=O)OC)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I04 compound treatment 199840.0 41100.0 2.8 183960.0 29400.0 2.19 3.5264 0.9925 3635797 CMLD6_000138 C(N1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6ccccc6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I05 compound treatment 170680.0 11900.0 0.81 167640.0 13000.0 0.97 1.2618 0.9961 3635799 CMLD6_000139 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC(=O)OC)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I06 compound treatment 191160.0 32400.0 2.21 178400.0 23800.0 1.77 2.8154 0.994 3635801 CMLD6_000140 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccc(Cl)nc4)C5(CC3(C5)[C@H]2c6ccccc6)c7ccccc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I07 compound treatment 183440.0 24700.0 1.68 178280.0 23700.0 1.76 2.4369 0.9997 3635803 CMLD6_000141 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC6CC6)C(=O)N(C3=O)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I08 compound treatment 187800.0 29000.0 1.98 174360.0 19800.0 1.47 2.4408 0.9893 3635805 CMLD6_000142 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(C)[C@@H]3c5ccccc5)c6ccc(cc6)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I09 compound treatment 168040.0 9290.0 0.63 159960.0 5370.0 0.4 0.7303 0.9753 3635807 CMLD6_000143 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)O/C(=N\CC(=O)OC)/[C@]4(C)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I10 compound treatment 190640.0 31900.0 2.17 178440.0 23800.0 1.77 2.7924 0.9949 3635809 CMLD6_000144 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccc(Cl)nc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I11 compound treatment 167600.0 8850.0 0.6 162960.0 8370.0 0.62 0.867 0.9999 3635811 CMLD6_000145 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(Cc5ccccc5)C4=O)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I12 compound treatment 182440.0 23700.0 1.62 181240.0 26600.0 1.98 2.5444 0.9948 3635813 CMLD6_000146 N#Cc1ccc(cc1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I13 compound treatment 209880.0 51100.0 3.49 198120.0 43500.0 3.24 4.7556 0.9993 3635815 CMLD6_000147 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I14 compound treatment 208880.0 50100.0 3.42 187120.0 32500.0 2.42 4.1285 0.9857 3635817 CMLD6_000148 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(Cc4cccnc4)[C@H](c5ccccc5)C63CC2(C6)c7ccc(C#N)cc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I15 compound treatment 173520.0 14800.0 1.01 169120.0 14500.0 1.08 1.4766 0.9994 3635819 CMLD6_000149 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCOC)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I16 compound treatment 182440.0 23700.0 1.62 172560.0 18000.0 1.34 2.0876 0.9956 3635821 CMLD6_000150 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(Cc4ccc(cc4)c5ccccc5)[C@H](c6ccccc6)C73CC2(C7)c8cccnc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I17 compound treatment 166880.0 8130.0 0.55 163040.0 8450.0 0.63 0.8365 0.998 3635823 CMLD6_000151 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC5CC5)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I18 compound treatment 174600.0 15800.0 1.08 170960.0 16400.0 1.22 1.6255 0.9982 3635825 CMLD6_000152 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I19 compound treatment 168040.0 9290.0 0.63 162320.0 7730.0 0.58 0.8545 0.9988 3635827 CMLD6_000153 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CC6CC6)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I20 compound treatment 172480.0 13700.0 0.94 166000.0 11400.0 0.85 1.2622 0.9988 3635829 CMLD6_000154 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccc(cc7)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I21 compound treatment 194360.0 35600.0 2.43 184800.0 30200.0 2.25 3.3064 0.9993 3635831 CMLD6_000155 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccccc3OC(=O)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I22 compound treatment 177560.0 18800.0 1.28 169240.0 14600.0 1.09 1.6776 0.9967 3635833 CMLD6_000156 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(cc3)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I23 mock treatment 154480.0 -4270.0 -0.29 151080.0 -3510.0 -0.26 -0.3907 -0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 I24 mock treatment 154720.0 -4030.0 -0.27 148440.0 -6150.0 -0.46 -0.5181 -0.9702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J01 mock treatment 157400.0 -1350.0 -0.09 155960.0 1370.0 0.1 0.0069 0.0501 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J02 mock treatment 160240.0 1490.0 0.1 155000.0 408.0 0.03 0.0933 0.8802 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J03 compound treatment 163600.0 4850.0 0.33 159000.0 4410.0 0.33 0.4658 1.0 3635834 CMLD6_000157 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J04 compound treatment 162160.0 3410.0 0.23 160440.0 5850.0 0.44 0.4721 0.9568 3635836 CMLD6_000158 Cn1c(N)cc(=O)n(Cc2ccccc2)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J05 compound treatment 169000.0 10200.0 0.7 162040.0 7450.0 0.55 0.8861 0.9934 3635837 CMLD6_000159 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J06 compound treatment 166400.0 7650.0 0.52 162520.0 7930.0 0.59 0.786 0.9981 3635838 CMLD6_000160 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CC(=O)OC)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J07 compound treatment 176040.0 17300.0 1.18 170360.0 15800.0 1.17 1.6633 1.0 3635840 CMLD6_000161 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3cc(OC)cc(OC)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J08 compound treatment 166280.0 7530.0 0.51 160120.0 5530.0 0.41 0.6539 0.994 3635841 CMLD6_000162 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)N(CC(=O)OC)C(=O)[C@]4(C)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J09 compound treatment 189160.0 30400.0 2.07 185480.0 30900.0 2.3 3.0915 0.9987 3635843 CMLD6_000163 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccccc4)c(N)n(Cc5ccccc5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J10 compound treatment 173120.0 14400.0 0.98 167440.0 12800.0 0.96 1.3689 0.9999 3635844 CMLD6_000164 CCCN1[C@@H](C[C@]2(O)[C@H]1C[C@H](O)[C@H](O)[C@@H]2O)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J11 compound treatment 178400.0 19600.0 1.34 164200.0 9610.0 0.72 1.4529 0.9568 3635846 CMLD6_000165 Cn1c(N)c(C(=O)COC(=O)c2ccnc3ccccc23)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J12 mock treatment 165280.0 6530.0 0.45 161400.0 6810.0 0.51 0.673 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J13 compound treatment 176040.0 17300.0 1.18 163760.0 9170.0 0.68 1.316 0.9662 3635847 CMLD6_000166 CN(C)/C=N/c1cc(=O)[nH]c(=O)n1CC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J14 mock treatment 165720.0 6970.0 0.48 163120.0 8530.0 0.63 0.7848 0.9898 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J15 compound treatment 272680.0 114000.0 7.77 247880.0 93300.0 6.94 10.4019 0.9984 1951970 CMLD6_000167 Cc1ccc2oc(=O)c3c4cc(O)c(O)cc4oc3c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J16 mock treatment 169760.0 11000.0 0.75 160440.0 5850.0 0.44 0.8385 0.9664 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J17 compound treatment 189960.0 31200.0 2.13 182920.0 28300.0 2.11 2.9954 1.0 3635849 CMLD6_000168 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(cc3)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J18 mock treatment 165480.0 6730.0 0.46 160560.0 5970.0 0.44 0.6385 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J19 compound treatment 167640.0 8890.0 0.61 160360.0 5770.0 0.43 0.7321 0.9857 3635851 CMLD6_000169 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1CC3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J20 mock treatment 160880.0 2130.0 0.15 154720.0 128.0 0.01 0.1094 0.752 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J21 compound treatment 160720.0 1970.0 0.13 153480.0 -1110.0 -0.08 0.0364 0.2309 1191854 CMLD6_000170 OC(=O)c1cc(nc2ccccc12)C3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J22 mock treatment 156040.0 -2710.0 -0.18 152200.0 -2390.0 -0.18 -0.2566 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J23 mock treatment 157680.0 -1070.0 -0.07 151120.0 -3470.0 -0.26 -0.2343 -0.8728 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 J24 mock treatment 149160.0 -9590.0 -0.65 145920.0 -8670.0 -0.65 -0.9187 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K01 mock treatment 157200.0 -1550.0 -0.11 156640.0 2050.0 0.15 0.033 0.178 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K02 mock treatment 165040.0 6290.0 0.43 158280.0 3690.0 0.27 0.4973 0.9768 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K03 compound treatment 171200.0 12400.0 0.85 158680.0 4090.0 0.3 0.8153 0.9043 3635853 CMLD6_000171 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC(=O)OC)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K04 compound treatment 165360.0 6610.0 0.45 158480.0 3890.0 0.29 0.5232 0.9771 3635855 CMLD6_000172 CN1C[C@@H]2C(c3ccc(cc3)C(F)(F)F)C4(CC2(C4)[C@H]1c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K05 compound treatment 177520.0 18800.0 1.28 164640.0 10000.0 0.75 1.4336 0.9673 3635857 CMLD6_000173 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)O/C(=N\Cc5ccccc5)/[C@]4(Cc6ccccc6)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K06 compound treatment 190160.0 31400.0 2.14 180440.0 25800.0 1.92 2.8745 0.9986 3635859 CMLD6_000174 Clc1ccc(cn1)C2[C@H]3CN(Cc4ccc(cc4)c5ccccc5)[C@H](c6ccccc6)C73CC2(C7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K07 compound treatment 174360.0 15600.0 1.06 162840.0 8250.0 0.61 1.1866 0.9658 3635861 CMLD6_000175 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC6CC6)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K08 compound treatment 198640.0 39900.0 2.72 187800.0 33200.0 2.47 3.6707 0.9989 3635863 CMLD6_000176 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccc(cc7)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K09 compound treatment 168960.0 10200.0 0.7 167080.0 12500.0 0.93 1.1494 0.9898 3635865 CMLD6_000177 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CC(=O)OC)C1=O)C(=O)N(C3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K10 compound treatment 190880.0 32100.0 2.19 178760.0 24200.0 1.8 2.8208 0.9952 3635867 CMLD6_000178 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccc(Cl)nc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K11 compound treatment 199600.0 40800.0 2.78 195040.0 40400.0 3.01 4.098 0.9992 3635869 CMLD6_000179 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/Cc6ccccc6)C1=O)C(=O)N(C3=O)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K12 compound treatment 192040.0 33300.0 2.27 176680.0 22100.0 1.64 2.7673 0.9875 3635871 CMLD6_000180 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccccc4)C5(CC3(C5)[C@H]2c6ccccc6)c7ccc(C#N)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K13 compound treatment 194680.0 35900.0 2.45 181640.0 27000.0 2.01 3.1556 0.9953 3635873 CMLD6_000181 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K14 compound treatment 184160.0 25400.0 1.73 181400.0 26800.0 2.0 2.6358 0.9975 3635875 CMLD6_000182 CN1C[C@@H]2C(c3ccc(Cl)nc3)C4(CC2(C4)[C@H]1c5ccccc5)c6ccc(C#N)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K15 compound treatment 170400.0 11600.0 0.79 167040.0 12400.0 0.93 1.2167 0.9971 3635877 CMLD6_000183 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCOC)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K16 compound treatment 200280.0 41500.0 2.83 193600.0 39000.0 2.9 4.055 0.9999 3635879 CMLD6_000184 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(Cc4cccnc4)[C@H](c5ccccc5)C63CC2(C6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K17 compound treatment 167240.0 8490.0 0.58 161640.0 7050.0 0.52 0.7802 0.9988 3635881 CMLD6_000185 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC5CC5)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K18 compound treatment 170000.0 11200.0 0.77 172040.0 17400.0 1.3 1.4606 0.9684 3635883 CMLD6_000186 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)C(F)(F)F)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K19 compound treatment 165200.0 6450.0 0.44 161360.0 6770.0 0.5 0.6671 0.9977 3635885 CMLD6_000187 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)O/C(=N\CC5CC5)/[C@]4(Cc6ccccc6)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K20 compound treatment 168360.0 9610.0 0.66 166880.0 12300.0 0.91 1.1099 0.9866 3635887 CMLD6_000188 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(C)[C@@H]3c5ccccc5)c6ccc(Cl)nc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K21 compound treatment 191360.0 32600.0 2.22 176320.0 21700.0 1.62 2.7155 0.9878 3635889 CMLD6_000189 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccccc3OS(=O)(=O)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K22 compound treatment 182240.0 23500.0 1.6 173280.0 18700.0 1.39 2.1159 0.9975 3635891 CMLD6_000190 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(cc3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K23 mock treatment 156480.0 -2270.0 -0.15 156160.0 1570.0 0.12 -0.027 -0.139 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 K24 mock treatment 154480.0 -4270.0 -0.29 147520.0 -7070.0 -0.53 -0.5781 -0.961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L01 mock treatment 162560.0 3810.0 0.26 154840.0 248.0 0.02 0.1967 0.7555 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L02 mock treatment 161840.0 3090.0 0.21 159880.0 5290.0 0.39 0.4272 0.9571 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L03 compound treatment 174560.0 15800.0 1.08 173840.0 19200.0 1.43 1.7751 0.9902 3635892 CMLD6_000191 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(cc3)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L04 compound treatment 163920.0 5170.0 0.35 163520.0 8930.0 0.66 0.7191 0.956 3635894 CMLD6_000192 CN(C)/C=N/c1cc(=O)n(C)c(=O)n1CC2CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L05 compound treatment 168600.0 9850.0 0.67 163400.0 8810.0 0.66 0.9384 0.9999 3635896 CMLD6_000193 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(cc3)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L06 compound treatment 163720.0 4970.0 0.34 159400.0 4810.0 0.36 0.4926 0.9996 3635897 CMLD6_000194 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC(=O)OC)C4=O)C1=O)C(=O)N(C3=O)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L07 compound treatment 163760.0 5010.0 0.34 164720.0 10100.0 0.75 0.7745 0.9359 3635899 CMLD6_000195 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccccc3OS(=O)(=O)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L08 compound treatment 186320.0 27600.0 1.88 188320.0 33700.0 2.51 3.1041 0.9898 3635901 CMLD6_000196 CCCN1[C@@H](C[C@H]2CC[C@H](O)C[C@H]21)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L09 compound treatment 179320.0 20600.0 1.4 174120.0 19500.0 1.45 2.0193 0.9998 3635902 CMLD6_000197 CC(C)Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)C4CC4)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L10 compound treatment 185000.0 26200.0 1.79 183320.0 28700.0 2.14 2.7773 0.9961 3635903 CMLD6_000198 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(cc3)N4CCN(C)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L11 compound treatment 186880.0 28100.0 1.92 190600.0 36000.0 2.68 3.2511 0.9865 3635905 CMLD6_000199 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3ccccc23)C4CC4)c(N)n(Cc5ccccc5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L12 mock treatment 169000.0 10200.0 0.7 164720.0 10100.0 0.75 1.0271 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L13 compound treatment 164480.0 5730.0 0.39 169440.0 14800.0 1.11 1.0576 0.9023 3635906 CMLD6_000200 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)C(F)(F)F)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L14 mock treatment 168040.0 9290.0 0.63 166760.0 12200.0 0.91 1.0882 0.9847 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L15 compound treatment 289600.0 131000.0 8.92 238040.0 83400.0 6.21 10.6997 0.9843 3635907 CMLD6_000201 Cc1ccc2oc(=O)c3c4cc(O)c(O)c(C)c4oc3c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L16 mock treatment 165800.0 7050.0 0.48 164240.0 9650.0 0.72 0.8476 0.9809 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L17 compound treatment 174920.0 16200.0 1.1 170640.0 16000.0 1.19 1.6241 0.9992 3635908 CMLD6_000202 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L18 mock treatment 165280.0 6530.0 0.45 153840.0 -752.0 -0.06 0.2752 0.6134 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L19 compound treatment 171720.0 13000.0 0.88 165240.0 10600.0 0.79 1.1856 0.9985 3635910 CMLD6_000203 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L20 mock treatment 167120.0 8370.0 0.57 153600.0 -992.0 -0.07 0.3513 0.6105 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L21 compound treatment 162280.0 3530.0 0.24 153760.0 -832.0 -0.06 0.1263 0.5086 3635912 CMLD6_000204 NC(=O)NCC1CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L22 mock treatment 156360.0 -2390.0 -0.16 154120.0 -472.0 -0.04 -0.1401 -0.8401 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L23 mock treatment 153360.0 -5390.0 -0.37 149760.0 -4830.0 -0.36 -0.5142 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 L24 mock treatment 150560.0 -8190.0 -0.56 149600.0 -4990.0 -0.37 -0.6576 -0.9804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M01 mock treatment 165280.0 6530.0 0.45 160520.0 5930.0 0.44 0.6267 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M02 mock treatment 169960.0 11200.0 0.76 166800.0 12200.0 0.91 1.1829 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M03 compound treatment 178000.0 19200.0 1.31 173680.0 19100.0 1.42 1.9325 0.9992 3635913 CMLD6_000205 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CCc5c[nH]c6ccccc56)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M04 compound treatment 193480.0 34700.0 2.37 185800.0 31200.0 2.32 3.3166 1.0 3635915 CMLD6_000206 FC(F)(F)c1ccc(cc1)C2[C@H]3CN(CC4CCCCC4)[C@H](c5ccccc5)C63CC2(C6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M05 compound treatment 174080.0 15300.0 1.05 170840.0 16200.0 1.21 1.5941 0.9974 3635917 CMLD6_000207 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/Cc6ccccc6)C1=O)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M06 compound treatment 201120.0 42400.0 2.89 191960.0 37400.0 2.78 4.0091 0.9998 3635919 CMLD6_000208 Clc1ccc(cn1)C2[C@H]3CN(Cc4cccnc4)[C@H](c5ccccc5)C63CC2(C6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M07 compound treatment 189880.0 31100.0 2.12 175400.0 20800.0 1.55 2.5958 0.988 3635921 CMLD6_000209 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CC6CC6)C1=O)C(=O)N(C3=O)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M08 compound treatment 185400.0 26600.0 1.82 177800.0 23200.0 1.73 2.5061 0.9997 3635923 CMLD6_000210 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)C(F)(F)F)[C@@H]3c6ccccc6)c7ccc(cc7)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M09 compound treatment 171240.0 12500.0 0.85 167720.0 13100.0 0.98 1.293 0.9976 3635925 CMLD6_000211 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/CC(=O)OC)C1=O)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M10 compound treatment 195480.0 36700.0 2.5 188320.0 33700.0 2.51 3.5457 1.0 3635927 CMLD6_000212 CN1C[C@@H]2C(c3ccccc3)C4(CC2(C4)[C@H]1c5ccccc5)c6cccnc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M11 compound treatment 189720.0 31000.0 2.11 181640.0 27000.0 2.01 2.9164 0.9997 3635929 CMLD6_000213 COCC/N=C/1\OC(=O)N2C(=O)C3=C4[C@@H](C[C@@H]5[C@H]([C@H]4[C@]21Cc6ccccc6)C(=O)N(C5=O)c7ccccc7)[C@@H]8[C@H]([C@H]3C)C(=O)N(C8=O)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M12 compound treatment 187320.0 28600.0 1.95 181600.0 27000.0 2.01 2.7986 0.9999 3635931 CMLD6_000214 N#Cc1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M13 compound treatment 178400.0 19600.0 1.34 173760.0 19200.0 1.43 1.956 0.9995 3635933 CMLD6_000215 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N(C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M14 compound treatment 189800.0 31000.0 2.12 181840.0 27200.0 2.03 2.9308 0.9998 3635935 CMLD6_000216 Clc1ccc(cn1)C2[C@H]3CN(CC4CCCCC4)[C@H](c5ccccc5)C63CC2(C6)c7ccc(C#N)cc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M15 compound treatment 186640.0 27900.0 1.9 175440.0 20800.0 1.55 2.4417 0.9949 3635937 CMLD6_000217 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC(=O)OC)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M16 compound treatment 180520.0 21800.0 1.48 173080.0 18500.0 1.38 2.0224 0.9993 3635939 CMLD6_000218 CN1C[C@@H]2C(c3ccc(Cl)nc3)C4(CC2(C4)[C@H]1c5ccccc5)c6cccnc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M17 compound treatment 170840.0 12100.0 0.82 164400.0 9810.0 0.73 1.099 0.9982 3635941 CMLD6_000219 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CC5CC5)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M18 compound treatment 179840.0 21100.0 1.44 169400.0 14800.0 1.1 1.796 0.9914 3635943 CMLD6_000220 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M19 compound treatment 164720.0 5970.0 0.41 168600.0 14000.0 1.04 1.025 0.9158 3635945 CMLD6_000221 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCOC)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M20 compound treatment 171160.0 12400.0 0.85 165320.0 10700.0 0.8 1.1628 0.9996 3635947 CMLD6_000222 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(CC5CCCCC5)[C@@H]3c6ccccc6)c7ccc(Cl)nc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M21 compound treatment 182560.0 23800.0 1.62 171680.0 17100.0 1.27 2.0471 0.9927 3635949 CMLD6_000223 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M22 compound treatment 180280.0 21500.0 1.47 174040.0 19400.0 1.45 2.0614 1.0 3635951 CMLD6_000224 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccccc3OS(=O)(=O)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M23 mock treatment 160520.0 1770.0 0.12 156240.0 1650.0 0.12 0.172 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 M24 mock treatment 157560.0 -1190.0 -0.08 148360.0 -6230.0 -0.46 -0.3854 -0.8185 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N01 mock treatment 164840.0 6090.0 0.42 161000.0 6410.0 0.48 0.6308 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N02 mock treatment 161880.0 3130.0 0.21 166200.0 11600.0 0.86 0.7618 0.856 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N03 compound treatment 165760.0 7010.0 0.48 173280.0 18700.0 1.39 1.3214 0.8985 3635952 CMLD6_000225 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1Cc3ccc(C)s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N04 compound treatment 167680.0 8930.0 0.61 175680.0 21100.0 1.57 1.5403 0.915 3635953 CMLD6_000226 CC(C)Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)C(F)(F)F)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N05 compound treatment 168240.0 9490.0 0.65 162080.0 7490.0 0.56 0.8515 0.9972 3635954 CMLD6_000227 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N06 compound treatment 165200.0 6450.0 0.44 161040.0 6450.0 0.48 0.6502 0.999 3635955 CMLD6_000228 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(C)N(C(=O)N(CC(=O)OC)C4=O)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N07 compound treatment 162440.0 3690.0 0.25 164120.0 9530.0 0.71 0.6793 0.9028 3635957 CMLD6_000229 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1CC(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N08 compound treatment 193040.0 34300.0 2.34 190560.0 36000.0 2.68 3.5459 0.9977 3635958 CMLD6_000230 COC(=O)[C@H]1C[C@H]2CC[C@H](O)C[C@H]2N1CC3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N09 compound treatment 262240.0 103000.0 7.06 247240.0 92600.0 6.9 9.8649 0.9999 3635960 CMLD6_000231 CC(C)Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccco4)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N10 compound treatment 182040.0 23300.0 1.59 187400.0 32800.0 2.44 2.8493 0.9783 3635961 CMLD6_000232 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N11 compound treatment 263840.0 105000.0 7.16 276640.0 122000.0 9.08 11.4893 0.9931 3635962 CMLD6_000233 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)c4ccco4)c(=O)n(Cc5ccccc5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N12 mock treatment 168480.0 9730.0 0.66 170280.0 15700.0 1.17 1.2947 0.9641 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N13 compound treatment 168920.0 10200.0 0.69 168000.0 13400.0 1.0 1.1959 0.9842 3635963 CMLD6_000234 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3c(cccc23)C(F)(F)F)C(F)(F)F)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N14 mock treatment 167240.0 8490.0 0.58 165920.0 11300.0 0.84 1.0054 0.9831 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N15 compound treatment 197600.0 38800.0 2.65 196440.0 41800.0 3.11 4.0752 0.9967 1220814 CMLD6_000235 CC1(C)CC(=O)c2c(C1)oc3cc(O)c(O)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N16 mock treatment 166400.0 7650.0 0.52 164120.0 9530.0 0.71 0.8702 0.9886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N17 compound treatment 174000.0 15200.0 1.04 175240.0 20600.0 1.54 1.8218 0.9819 3635964 CMLD6_000236 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(C)s3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N18 mock treatment 168160.0 9410.0 0.64 163400.0 8810.0 0.66 0.9171 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N19 compound treatment 170960.0 12200.0 0.83 164160.0 9570.0 0.71 1.0921 0.997 3635965 CMLD6_000237 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1CC3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N20 mock treatment 167960.0 9210.0 0.63 159480.0 4890.0 0.36 0.7012 0.9663 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N21 compound treatment 164440.0 5690.0 0.39 161520.0 6930.0 0.52 0.6389 0.9901 3635966 CMLD6_000238 CN(C)/C=N/c1cc(=O)[nH]c(=O)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N22 mock treatment 160480.0 1730.0 0.12 155040.0 448.0 0.03 0.1069 0.8729 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N23 mock treatment 156120.0 -2630.0 -0.18 152120.0 -2470.0 -0.18 -0.2569 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 N24 mock treatment 154200.0 -4550.0 -0.31 151360.0 -3230.0 -0.24 -0.3895 -0.9921 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O01 mock treatment 166960.0 8210.0 0.56 160960.0 6370.0 0.47 0.7309 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O02 mock treatment 161160.0 2410.0 0.16 162160.0 7570.0 0.56 0.5144 0.8768 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O03 compound treatment 160320.0 1570.0 0.11 161280.0 6690.0 0.5 0.4276 0.8399 3635968 CMLD6_000239 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCc5c[nH]c6ccccc56)C(=O)N(CC(=O)OC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O04 compound treatment 179160.0 20400.0 1.39 176400.0 21800.0 1.62 2.1316 0.9971 3635970 CMLD6_000240 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccc(cc4)C(F)(F)F)C5(CC3(C5)[C@H]2c6ccccc6)c7ccccc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O05 compound treatment 166280.0 7530.0 0.51 160200.0 5610.0 0.42 0.6581 0.9947 3635972 CMLD6_000241 CCN1C(=O)[C@@H]2CCC3=C(CC)C(=O)N4C(=O)N(CCOC)C(=O)[C@]4(Cc5ccccc5)[C@@H]3[C@@H]2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O06 compound treatment 180800.0 22000.0 1.5 170320.0 15700.0 1.17 1.8907 0.9924 3635974 CMLD6_000242 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(C)[C@@H]3c5ccccc5)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O07 compound treatment 165920.0 7170.0 0.49 164600.0 10000.0 0.74 0.8723 0.9791 3635976 CMLD6_000243 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N(C(=O)O\C4=N/Cc5ccccc5)C1=O)C(=O)N(C)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O08 compound treatment 177720.0 19000.0 1.29 175600.0 21000.0 1.56 2.0201 0.9956 3635978 CMLD6_000244 COC(=O)c1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)c6ccccc6)[C@@H]3c7ccccc7)c8ccc(cc8)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O09 compound treatment 171440.0 12700.0 0.87 162520.0 7930.0 0.59 1.029 0.9826 3635980 CMLD6_000245 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCc5c[nH]c6ccccc56)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O10 compound treatment 203640.0 44900.0 3.06 187440.0 32800.0 2.44 3.8927 0.9938 3635982 CMLD6_000246 C(C1CCCCC1)N2C[C@@H]3C(c4ccccc4)C5(CC3(C5)[C@H]2c6ccccc6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O11 compound treatment 221160.0 62400.0 4.25 203600.0 49000.0 3.65 5.5878 0.9971 3635984 CMLD6_000247 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C(=O)N(C3=O)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O12 compound treatment 191160.0 32400.0 2.21 178720.0 24100.0 1.8 2.8322 0.9947 3635986 CMLD6_000248 N#Cc1ccc(cc1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O13 compound treatment 195160.0 36400.0 2.48 174320.0 19700.0 1.47 2.7935 0.9686 3635988 CMLD6_000249 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CCc6c[nH]c7ccccc67)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O14 compound treatment 179040.0 20300.0 1.38 174280.0 19700.0 1.47 2.0142 0.9996 3635990 CMLD6_000250 FC(F)(F)c1ccc(CN2C[C@@H]3C(c4ccc(Cl)nc4)C5(CC3(C5)[C@H]2c6ccccc6)c7ccc(C#N)cc7)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O15 compound treatment 165640.0 6890.0 0.47 165760.0 11200.0 0.83 0.9199 0.9635 3635992 CMLD6_000251 COC(=O)C/N=C/1\OC(=O)N2C(=O)C3=C4[C@@H](C[C@@H]5[C@H]([C@H]4[C@]21Cc6ccccc6)C(=O)N(C5=O)c7ccccc7)[C@@H]8[C@H]([C@H]3C)C(=O)N(C8=O)c9ccccc9 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O16 compound treatment 178040.0 19300.0 1.32 176960.0 22400.0 1.66 2.1071 0.9932 3635994 CMLD6_000252 Clc1ccc(cn1)C2[C@H]3CN(CC4CCCCC4)[C@H](c5ccccc5)C63CC2(C6)c7cccnc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O17 compound treatment 173720.0 15000.0 1.02 174360.0 19800.0 1.47 1.762 0.984 3635996 CMLD6_000253 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(Cc5ccccc5)N1C(=O)O\C4=N/CC6CC6)C(=O)NC3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O18 compound treatment 179720.0 21000.0 1.43 174120.0 19500.0 1.45 2.0386 1.0 3635998 CMLD6_000254 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5cccnc5)[C@@H]3c6ccccc6)c7ccccc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O19 compound treatment 166280.0 7530.0 0.51 156160.0 1570.0 0.12 0.4455 0.8463 3636000 CMLD6_000255 CCN(CC)C(=O)OC1=C(CC)C2=CC[C@@H]3[C@H]([C@H]2[C@]/4(C)N1C(=O)O\C4=N/CCOC)C(=O)N(CC)C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O20 compound treatment 169720.0 11000.0 0.75 155680.0 1090.0 0.08 0.5861 0.7791 3636002 CMLD6_000256 COC(=O)c1cccc(c1)C2(CC34C2)C([C@H]4CN(Cc5ccc(cc5)C(F)(F)F)[C@@H]3c6ccccc6)c7ccc(Cl)nc7 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O21 compound treatment 174880.0 16100.0 1.1 165280.0 10700.0 0.8 1.34 0.9874 3636004 CMLD6_000257 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1Cc3ccc(cc3)N4CCN(C)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O22 compound treatment 165040.0 6290.0 0.43 163880.0 9290.0 0.69 0.792 0.9736 3636006 CMLD6_000258 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(cc3)N4CCN(C)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O23 mock treatment 156240.0 -2510.0 -0.17 148640.0 -5950.0 -0.44 -0.4343 -0.9145 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 O24 mock treatment 154360.0 -4390.0 -0.3 145720.0 -8870.0 -0.66 -0.6786 -0.936 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P01 mock treatment 160080.0 1330.0 0.09 160440.0 5850.0 0.44 0.3718 0.8364 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P02 mock treatment 163360.0 4610.0 0.31 161120.0 6530.0 0.49 0.5658 0.9778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P03 compound treatment 163320.0 4570.0 0.31 162000.0 7410.0 0.55 0.6101 0.9635 3636007 CMLD6_000259 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@H](O)[C@H](O)[C@@H]2O)N1C/C=C/c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P04 compound treatment 167560.0 8810.0 0.6 162280.0 7690.0 0.57 0.8293 0.9997 3636008 CMLD6_000260 OC(=O)c1cc(nc2c(cccc12)C(F)(F)F)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P05 compound treatment 164640.0 5890.0 0.4 161520.0 6930.0 0.52 0.6485 0.9923 3636009 CMLD6_000261 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3ccc(cc3)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P06 compound treatment 174080.0 15300.0 1.05 181760.0 27200.0 2.02 2.1688 0.9528 3636010 CMLD6_000262 CCC1=C2CC[C@@H]3[C@H]([C@H]2[C@]4(Cc5ccccc5)N(C(=O)N(CC(=O)OC)C4=O)C1=O)C(=O)N(C3=O)c6ccccc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P07 compound treatment 164840.0 6090.0 0.42 159120.0 4530.0 0.34 0.5318 0.9947 3636012 CMLD6_000263 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1Cc3c(F)cccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P08 compound treatment 188440.0 29700.0 2.02 183880.0 29300.0 2.18 2.9726 0.9993 3636014 CMLD6_000264 COC(=O)[C@@H]1C[C@H]2CC[C@H](O)C[C@H]2N1CC3CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P09 compound treatment 169680.0 10900.0 0.75 166520.0 11900.0 0.89 1.1546 0.9962 3636015 CMLD6_000265 Cn1c(=O)c(C(=O)COC(=O)c2cc(nc3ccccc23)C(F)(F)F)c(N)n(Cc4ccccc4)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P10 compound treatment 184800.0 26000.0 1.78 176920.0 22300.0 1.66 2.4309 0.9994 3636016 CMLD6_000266 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1Cc3ccc(cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P11 compound treatment 174400.0 15600.0 1.07 170760.0 16200.0 1.2 1.6053 0.9982 3636017 CMLD6_000267 Cn1c(N)c(C(=O)COC(=O)c2cc(nc3ccccc23)C4CC4)c(=O)n(Cc5ccccc5)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P12 mock treatment 161640.0 2890.0 0.2 160960.0 6370.0 0.47 0.4744 0.9243 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P13 compound treatment 165640.0 6890.0 0.47 160880.0 6290.0 0.47 0.663 1.0 3636018 CMLD6_000268 CC(C)Cn1c(N)c(C(=O)COC(=O)c2cc(nc3c(cccc23)C(F)(F)F)C(F)(F)F)c(=O)n(C)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P14 mock treatment 164960.0 6210.0 0.42 157680.0 3090.0 0.23 0.4618 0.9588 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P15 compound treatment 174080.0 15300.0 1.05 169320.0 14700.0 1.1 1.5141 0.9997 3636019 CMLD6_000269 CC1(C)CC(=O)c2c(C1)oc3cc4OCOc4cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P16 mock treatment 162720.0 3970.0 0.27 161120.0 6530.0 0.49 0.5349 0.9618 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P17 compound treatment 183240.0 24500.0 1.67 176840.0 22200.0 1.66 2.3514 1.0 3636020 CMLD6_000270 COC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1CC3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P18 mock treatment 159400.0 649.0 0.04 159360.0 4770.0 0.35 0.2822 0.7892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P19 compound treatment 162640.0 3890.0 0.27 159080.0 4490.0 0.33 0.4237 0.9935 3636022 CMLD6_000271 COC(=O)[C@@H]1C[C@]2(O)[C@@H](C[C@@H](O)[C@@H](O)[C@H]2O)N1CC3CCCCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P20 mock treatment 159280.0 529.0 0.04 155000.0 408.0 0.03 0.047 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P21 compound treatment 157880.0 -871.0 -0.06 161920.0 7330.0 0.55 0.3437 0.6264 3636023 CMLD6_000272 CN(C)/C=N/c1cc(=O)n(C)c(=O)n1Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P22 mock treatment 154480.0 -4270.0 -0.29 148440.0 -6150.0 -0.46 -0.5297 -0.9761 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P23 mock treatment 152600.0 -6150.0 -0.42 149880.0 -4710.0 -0.35 -0.5445 -0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2434 P24 mock treatment 155560.0 -3190.0 -0.22 145600.0 -8990.0 -0.67 -0.6271 -0.8911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A01 compound treatment 157480.0 13300.0 0.91 152440.0 8360.0 0.62 1.0805 0.9832 3652636 Neuro1_000001 [O-][N+](=O)c1cccc(c1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A02 compound treatment 145880.0 1690.0 0.11 149480.0 5400.0 0.4 0.3655 0.8743 1542244 Neuro1_000002 CCCOc1ccc(cc1)c2nc(N(CC)CC)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A03 compound treatment 178680.0 34500.0 2.35 179920.0 35800.0 2.67 3.5488 0.998 3652637 Neuro1_000003 [O-][N+](=O)c1cccc(c1)c2nc(Nc3ccccc3F)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A04 compound treatment 146240.0 2050.0 0.14 145240.0 1160.0 0.09 0.1598 0.9735 3652638 Neuro1_000004 CC1CCN(CC1)c2nc(nc3ccccc23)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A05 compound treatment 241120.0 96900.0 6.61 220360.0 76300.0 5.68 8.6872 0.9971 1701346 Neuro1_000005 Cc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A06 compound treatment 183520.0 39300.0 2.68 187160.0 43100.0 3.21 4.1631 0.996 3652639 Neuro1_000006 Oc1ccccc1/C=N/Nc2nc(nc3ccccc23)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A07 compound treatment 217840.0 73600.0 5.02 205960.0 61900.0 4.61 6.807 0.9991 1677893 Neuro1_000007 Fc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A08 compound treatment 146440.0 2250.0 0.15 147400.0 3320.0 0.25 0.2831 0.9735 3652641 Neuro1_000008 COc1cccc2c(NCCCN3CCCC3=O)nc(nc12)C(Cl)(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A09 compound treatment 155920.0 11700.0 0.8 155160.0 11100.0 0.82 1.1485 0.9999 1486822 Neuro1_000009 Cc1ccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A10 compound treatment 141400.0 -2790.0 -0.19 141840.0 -2240.0 -0.17 -0.2525 -0.9978 3652642 Neuro1_000010 COc1ccc(Cl)cc1Nc2nc(N)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A11 compound treatment 273280.0 129000.0 8.8 245680.0 102000.0 7.56 11.5701 0.9971 1143772 Neuro1_000011 COc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A12 compound treatment 150680.0 6490.0 0.44 147800.0 3720.0 0.28 0.5085 0.9746 3652643 Neuro1_000012 C(N1CCN(CC1)c2nc(NC3CCCCC3)c4ccccc4n2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A13 compound treatment 150240.0 6050.0 0.41 150120.0 6040.0 0.45 0.6094 0.9991 1462125 Neuro1_000013 C(Nc1nc(nc2ccccc12)N3CCOCC3)c4ccco4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A14 compound treatment 145760.0 1570.0 0.11 146680.0 2600.0 0.19 0.2124 0.9607 3652644 Neuro1_000014 COc1ccc(Cl)cc1Nc2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A15 compound treatment 183760.0 39600.0 2.7 180400.0 36300.0 2.7 3.8189 1.0 1523378 Neuro1_000015 CCN(CC)c1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A16 compound treatment 258640.0 114000.0 7.8 239520.0 95400.0 7.1 10.5401 0.9989 3652645 Neuro1_000016 Oc1ccccc1Nc2nc(NC3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A17 compound treatment 253400.0 109000.0 7.45 142800.0 -1280.0 -0.1 5.1974 0.698 1312582 Neuro1_000017 Oc1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A18 compound treatment 162560.0 18400.0 1.25 150080.0 6000.0 0.45 1.2012 0.9036 3652646 Neuro1_000018 Fc1ccccc1c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A19 compound treatment 182520.0 38300.0 2.61 183360.0 39300.0 2.92 3.9149 0.9984 1480295 Neuro1_000019 CN(C)c1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A20 compound treatment 166920.0 22700.0 1.55 169280.0 25200.0 1.88 2.4219 0.9955 3652647 Neuro1_000020 CN1CCN(CC1)c2nc(Nc3ccc(Br)cc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A21 compound treatment 150520.0 6330.0 0.43 154080.0 10000.0 0.74 0.8313 0.9663 1670841 Neuro1_000021 COc1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A22 compound treatment 158360.0 14200.0 0.97 155600.0 11500.0 0.86 1.2893 0.9982 3652648 Neuro1_000022 [O-][N+](=O)c1cccc(c1)c2nc(Nc3cccc(Cl)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A23 mock treatment 142240.0 -1950.0 -0.13 142200.0 -1880.0 -0.14 -0.1931 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 A24 mock treatment 141600.0 -2590.0 -0.18 139240.0 -4840.0 -0.36 -0.3797 -0.9464 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B01 compound treatment 138880.0 -5310.0 -0.36 139000.0 -5080.0 -0.38 -0.5235 -0.9998 3652649 Neuro1_000023 CCN(CC)CCNc1nc(nc2ccccc12)c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B02 compound treatment 159240.0 15000.0 1.03 169280.0 25200.0 1.88 2.0516 0.9597 1202518 Neuro1_000024 COc1ccc(cc1)C(=O)Oc2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B03 compound treatment 139080.0 -5110.0 -0.35 140520.0 -3560.0 -0.26 -0.4338 -0.9908 3652650 Neuro1_000025 [O-][N+](=O)c1cccc(c1)c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B04 compound treatment 144320.0 126.0 0.01 139160.0 -4920.0 -0.37 -0.2528 -0.6903 3652651 Neuro1_000026 Fc1ccccc1c2nc(NCCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B05 compound treatment 138880.0 -5310.0 -0.36 137080.0 -7000.0 -0.52 -0.6245 -0.9843 3652652 Neuro1_000027 Cc1cc(C)c2nc(nc(N3CCc4ccccc4C3)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B06 compound treatment 155320.0 11100.0 0.76 152000.0 7920.0 0.59 0.9533 0.9922 1362256 Neuro1_000028 CCOc1ccccc1Nc2ncnc3ccc(I)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B07 compound treatment 170600.0 26400.0 1.8 170440.0 26400.0 1.96 2.6603 0.9991 3652653 Neuro1_000029 Oc1ccc(Nc2nc(NCC3CCCO3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B08 compound treatment 155040.0 10800.0 0.74 148440.0 4360.0 0.32 0.7524 0.9317 1446183 Neuro1_000030 COc1ccc(CCNc2ncnc3ccc(I)cc23)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B09 compound treatment 131720.0 -12500.0 -0.85 134480.0 -9600.0 -0.71 -1.1065 -0.9962 3652654 Neuro1_000031 COc1ccc(CCNc2nc(nc3c(C)cc(C)cc23)C(F)(F)F)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B10 compound treatment 163600.0 19400.0 1.32 164680.0 20600.0 1.53 2.0197 0.9973 3652655 Neuro1_000032 Oc1ccc(cc1Nc2ncnc3ccc(Br)cc23)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B11 compound treatment 145560.0 1370.0 0.09 138560.0 -5520.0 -0.41 -0.2246 -0.5332 3652656 Neuro1_000033 CC(Nc1nc(nc2ccccc12)N3CCCCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B12 compound treatment 140440.0 -3750.0 -0.26 145760.0 1680.0 0.13 -0.0925 -0.3246 3652657 Neuro1_000034 CC(Nc1nc(nc2ccccc12)N3CCN(CCO)CC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B13 compound treatment 138280.0 -5910.0 -0.4 140920.0 -3160.0 -0.24 -0.4513 -0.967 3652658 Neuro1_000035 Clc1cccc(c1)c2nc(NCCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B14 compound treatment 160880.0 16700.0 1.14 158400.0 14300.0 1.07 1.5581 0.9995 1494734 Neuro1_000036 Fc1ccc(cc1)C(=O)Oc2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B15 compound treatment 174560.0 30400.0 2.07 174720.0 30600.0 2.28 3.0765 0.9988 3652659 Neuro1_000037 [O-][N+](=O)c1cccc(Nc2ncnc3ccc(I)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B16 compound treatment 168680.0 24500.0 1.67 166000.0 21900.0 1.63 2.3341 0.9999 3652660 Neuro1_000038 CC(C)OCCCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B17 compound treatment 187560.0 43400.0 2.96 189800.0 45700.0 3.4 4.4968 0.9975 1539522 Neuro1_000039 CN(C)c1ccc(Nc2ncnc3ccc(I)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B18 compound treatment 148920.0 4730.0 0.32 145160.0 1080.0 0.08 0.2847 0.8574 3652661 Neuro1_000040 [O-][N+](=O)c1ccc(NCCNc2nc(nc3ccccc23)N4CCOCC4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B19 compound treatment 141080.0 -3110.0 -0.21 144080.0 1.25 0.0 -0.15 -0.7068 3652662 Neuro1_000041 CCOC(=O)c1nc(Nc2ccc(cc2)S(=O)(=O)Nc3ncccn3)c4ccccc4n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B20 compound treatment 174280.0 30100.0 2.05 171920.0 27800.0 2.07 2.9156 1.0 3652663 Neuro1_000042 OCCNc1nc(Nc2ccc(O)cc2)nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B21 compound treatment 168160.0 24000.0 1.63 165800.0 21700.0 1.62 2.2985 1.0 1395503 Neuro1_000043 Cc1ccc(cc1)C(=O)Oc2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B22 compound treatment 134080.0 -10100.0 -0.69 130680.0 -13400.0 -1.0 -1.1927 -0.9838 3652664 Neuro1_000044 CC1CN(CC(C)O1)c2nc(nc3c(C)cc(C)cc23)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B23 mock treatment 142160.0 -2030.0 -0.14 140040.0 -4040.0 -0.3 -0.3106 -0.9383 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 B24 mock treatment 136760.0 -7430.0 -0.51 137360.0 -6720.0 -0.5 -0.712 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C01 compound treatment 152520.0 8330.0 0.57 153120.0 9040.0 0.67 0.8772 0.9964 3652665 Neuro1_000045 Fc1ccccc1c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C02 compound treatment 152960.0 8770.0 0.6 148240.0 4160.0 0.31 0.6416 0.9532 1476428 Neuro1_000046 Cc1ccc(cc1Nc2ncnc3ccc(Br)cc23)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C03 compound treatment 147440.0 3250.0 0.22 146520.0 2440.0 0.18 0.285 0.9952 3652666 Neuro1_000047 CCOc1ccc(Nc2nc(nc3ccccc23)c4cccc(c4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C04 compound treatment 148120.0 3930.0 0.27 144400.0 321.0 0.02 0.2062 0.7672 3652667 Neuro1_000048 CCN(CC)c1nc(nc2ccccc12)N3CCN(CCO)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C05 compound treatment 162600.0 18400.0 1.25 143400.0 -679.0 -0.05 0.8516 0.6781 1183267 Neuro1_000049 Cc1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C06 compound treatment 147680.0 3490.0 0.24 147720.0 3640.0 0.27 0.3597 0.9979 3652668 Neuro1_000050 Oc1ccccc1/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C07 compound treatment 215160.0 71000.0 4.84 214600.0 70500.0 5.25 7.1325 0.9992 1407411 Neuro1_000051 CCOC(=O)c1ccc(Nc2nc(nc3ccccc23)c4cccnc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C08 compound treatment 143080.0 -1110.0 -0.08 144360.0 281.0 0.02 -0.0389 -0.4938 3652670 Neuro1_000052 Cc1cc(N2CCN(CC2)c3nc(nc4ccccc34)N5CCOCC5)c6ccccc6n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C09 compound treatment 163800.0 19600.0 1.34 152040.0 7960.0 0.59 1.3642 0.933 1627656 Neuro1_000053 Brc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C10 compound treatment 85720.0 -58500.0 -3.99 85000.0 -59100.0 -4.4 -5.9281 -0.9988 3652671 Neuro1_000054 CN(C)c1ccc(Nc2nc(N)c3ccccc3n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C11 compound treatment 234640.0 90400.0 6.17 216040.0 72000.0 5.36 8.1474 0.9975 1165826 Neuro1_000055 Fc1ccc(Nc2nc(NCc3ccccc3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C12 compound treatment 169600.0 25400.0 1.73 166400.0 22300.0 1.66 2.3995 0.9998 3652672 Neuro1_000056 COc1ccc(Cl)cc1Nc2nc(NCCO)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C13 compound treatment 145200.0 1010.0 0.07 142120.0 -1960.0 -0.15 -0.0546 -0.3387 1447299 Neuro1_000057 CCc1ccccc1Nc2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C14 compound treatment 146480.0 2290.0 0.16 145400.0 1320.0 0.1 0.1798 0.9753 3652673 Neuro1_000058 CN1CCN(CC1)c2nc(NC3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C15 compound treatment 171120.0 26900.0 1.84 173960.0 29900.0 2.22 2.8707 0.9955 1577515 Neuro1_000059 Fc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C16 compound treatment 159800.0 15600.0 1.06 157160.0 13100.0 0.97 1.4408 0.999 3652674 Neuro1_000060 COc1ccc(OC)c(Nc2nc(NCC3CCCO3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C17 compound treatment 157200.0 13000.0 0.89 166280.0 22200.0 1.65 1.7954 0.9574 1633041 Neuro1_000061 CCc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C18 compound treatment 144800.0 606.0 0.04 149960.0 5880.0 0.44 0.3387 0.7704 1170803 Neuro1_000062 CCN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(OC)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C19 compound treatment 172280.0 28100.0 1.91 173800.0 29700.0 2.21 2.9182 0.9974 1481237 Neuro1_000063 COc1ccc(C)cc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C20 compound treatment 181640.0 37400.0 2.55 176160.0 32100.0 2.39 3.4936 0.9994 3652675 Neuro1_000064 [O-][N+](=O)c1cccc(c1)c2nc(NC3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C21 compound treatment 146360.0 2170.0 0.15 151440.0 7360.0 0.55 0.4918 0.8668 1141507 Neuro1_000065 CCN(CC)CCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C22 compound treatment 147280.0 3090.0 0.21 146320.0 2240.0 0.17 0.2667 0.9934 3652676 Neuro1_000066 [O-][N+](=O)c1cccc(c1)c2nc(N3CCN(Cc4ccccc4)CC3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C23 mock treatment 137520.0 -6670.0 -0.45 137960.0 -6120.0 -0.46 -0.6437 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 C24 mock treatment 142640.0 -1550.0 -0.11 139800.0 -4280.0 -0.32 -0.3001 -0.8941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D01 compound treatment 146320.0 2130.0 0.14 152000.0 7920.0 0.59 0.5194 0.8555 3652677 Neuro1_000067 COC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccccc4F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D02 compound treatment 143600.0 -594.0 -0.04 147720.0 3640.0 0.27 0.163 0.5949 1128505 Neuro1_000068 CC(C)Oc1ccc(Nc2ncnc3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D03 compound treatment 218720.0 74500.0 5.08 213600.0 69500.0 5.17 7.2515 1.0 3652678 Neuro1_000069 Oc1cccc(Nc2nc(NCc3ccco3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D04 compound treatment 137520.0 -6670.0 -0.45 136840.0 -7240.0 -0.54 -0.7027 -0.9965 3652679 Neuro1_000070 OCCN1CCN(CC1)c2nc(N3CCN(CC3)c4ccc(cc4)[N+](=O)[O-])c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D05 compound treatment 151320.0 7130.0 0.49 144960.0 881.0 0.07 0.3899 0.7954 3086865 Neuro1_000071 OCCNc1nc(nc2ccccc12)N3CCN(CC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D06 compound treatment 154440.0 10200.0 0.7 158000.0 13900.0 1.04 1.2266 0.9816 1371864 Neuro1_000072 CC(=O)Nc1ccc(Nc2ncnc3ccc(I)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D07 compound treatment 145920.0 1730.0 0.12 144120.0 41.3 0.0 0.0854 0.7253 3652680 Neuro1_000073 CCOC(=O)N1CCN(CC1)c2nc(nc3c(C)cc(C)cc23)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D08 compound treatment 155360.0 11200.0 0.76 150800.0 6720.0 0.5 0.892 0.9793 3652681 Neuro1_000074 Ic1ccc2ncnc(NCCCN3CCOCC3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D09 compound treatment 158120.0 13900.0 0.95 151160.0 7080.0 0.53 1.044 0.9614 3652682 Neuro1_000075 CN1CCN(CC1)c2nc(NCCO)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D10 compound treatment 181440.0 37200.0 2.54 171960.0 27900.0 2.08 3.2629 0.995 1228851 Neuro1_000076 Cc1ccc(O)c(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D11 compound treatment 162120.0 17900.0 1.22 160320.0 16200.0 1.21 1.7189 1.0 3652683 Neuro1_000077 CC(Nc1nc(nc2ccccc12)N3CCN(CC3)S(=O)(=O)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D12 compound treatment 186040.0 41800.0 2.85 182640.0 38600.0 2.87 4.0467 1.0 3652684 Neuro1_000078 OC(=O)c1cccc(Nc2nc(nc3ccccc23)C(F)(F)F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D13 compound treatment 155800.0 11600.0 0.79 153800.0 9720.0 0.72 1.0711 0.999 3652685 Neuro1_000079 Clc1cccc(c1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D14 compound treatment 176280.0 32100.0 2.19 174960.0 30900.0 2.3 3.172 0.9997 1555545 Neuro1_000080 N(c1ccccc1)c2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D15 compound treatment 200360.0 56200.0 3.83 203800.0 59700.0 4.44 5.8507 0.9972 1326651 Neuro1_000081 Oc1ccc(Nc2ncnc3ccc(I)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D16 compound treatment 150680.0 6490.0 0.44 152160.0 8080.0 0.6 0.738 0.9886 1553618 Neuro1_000082 O=S(=O)(Nc1ncccn1)c2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D17 compound treatment 172480.0 28300.0 1.93 172680.0 28600.0 2.13 2.8689 0.9988 1414439 Neuro1_000083 Fc1ccc(Nc2ncnc3ccc(I)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D18 compound treatment 165800.0 21600.0 1.47 154240.0 10200.0 0.76 1.5764 0.952 3652686 Neuro1_000084 CC(Nc1nc(nc2ccccc12)N3CCN(CC3)S(=O)(=O)c4ccc(C)cc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D19 compound treatment 187320.0 43100.0 2.94 189040.0 45000.0 3.35 4.4453 0.9979 3652687 Neuro1_000085 CCOC(=O)c1nc(Nc2cc(Cl)ccc2O)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D20 compound treatment 142800.0 -1390.0 -0.1 143000.0 -1080.0 -0.08 -0.124 -0.9965 3652688 Neuro1_000086 Cc1cc(C)c2nc(nc(N3CCN(CC3)c4ccccc4F)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D21 compound treatment 161840.0 17600.0 1.2 164400.0 20300.0 1.51 1.9202 0.9936 3652689 Neuro1_000087 CC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D22 compound treatment 176600.0 32400.0 2.21 185880.0 41800.0 3.11 3.7622 0.9859 3652690 Neuro1_000088 Oc1ccccc1Nc2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D23 mock treatment 138840.0 -5350.0 -0.37 141040.0 -3040.0 -0.23 -0.418 -0.9735 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 D24 mock treatment 137840.0 -6350.0 -0.43 134760.0 -9320.0 -0.69 -0.7967 -0.9743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E01 compound treatment 154120.0 9930.0 0.68 150280.0 6200.0 0.46 0.8049 0.9826 1623881 Neuro1_000089 COc1ccc(cc1)c2nc(NCCO)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E02 compound treatment 169080.0 24900.0 1.7 171680.0 27600.0 2.05 2.6523 0.9955 3652691 Neuro1_000090 OC(=O)C(Nc1nc(nc2ccccc12)C(F)(F)F)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E03 compound treatment 164800.0 20600.0 1.4 160520.0 16400.0 1.22 1.8587 0.9976 1647041 Neuro1_000091 Cc1ccccc1Nc2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E04 compound treatment 176800.0 32600.0 2.22 185880.0 41800.0 3.11 3.7718 0.9864 1935369 Neuro1_000092 CCOc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E05 compound treatment 218480.0 74300.0 5.06 224880.0 80800.0 6.01 7.8336 0.9963 1127286 Neuro1_000093 CCOc1ccccc1Nc2nc(nc3ccccc23)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E06 compound treatment 177600.0 33400.0 2.28 178040.0 34000.0 2.53 3.3978 0.9986 3652692 Neuro1_000094 COc1cccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E07 compound treatment 159880.0 15700.0 1.07 155400.0 11300.0 0.84 1.352 0.993 1515436 Neuro1_000095 C(Nc1nc(nc2ccccc12)N3CCCCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E08 compound treatment 148360.0 4170.0 0.28 149840.0 5760.0 0.43 0.504 0.98 3652694 Neuro1_000096 COc1cccc2c(nc(nc12)C(Cl)(Cl)Cl)N3CC(C)OC(C)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E09 compound treatment 160920.0 16700.0 1.14 161840.0 17800.0 1.32 1.7411 0.9973 1609740 Neuro1_000097 Cc1cccc(Nc2nc(N3CCOCC3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E10 compound treatment 170960.0 26800.0 1.82 171480.0 27400.0 2.04 2.7324 0.9985 3652695 Neuro1_000098 COc1ccc(OC)c(Nc2nc(NCc3ccco3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E11 compound treatment 165720.0 21500.0 1.47 166160.0 22100.0 1.64 2.1998 0.9984 1181771 Neuro1_000099 C(Nc1nc(nc2ccccc12)N3CCN(CC3)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E12 compound treatment 158680.0 14500.0 0.99 153440.0 9360.0 0.7 1.191 0.9854 3652696 Neuro1_000100 COc1ccc(C)cc1Nc2nc(NCCO)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E13 compound treatment 172360.0 28200.0 1.92 170280.0 26200.0 1.95 2.7368 1.0 1643938 Neuro1_000101 Oc1ccccc1c2nc(Nc3ccc(Cl)c(Cl)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E14 compound treatment 170560.0 26400.0 1.8 170960.0 26900.0 2.0 2.6858 0.9986 3652697 Neuro1_000102 Cc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E15 compound treatment 161840.0 17600.0 1.2 159320.0 15200.0 1.13 1.6528 0.9996 3652698 Neuro1_000103 COc1ccccc1N2CCN(CC2)c3nc(nc4ccccc34)c5ccccc5O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E16 compound treatment 183240.0 39000.0 2.66 184480.0 40400.0 3.01 4.0086 0.9982 3652699 Neuro1_000104 COc1ccc(OC)c(Nc2nc(N)c3ccccc3n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E17 compound treatment 184360.0 40200.0 2.74 182680.0 38600.0 2.87 3.9678 0.9997 3652700 Neuro1_000105 CC(=O)c1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E18 compound treatment 173280.0 29100.0 1.98 171320.0 27200.0 2.03 2.8358 0.9999 3652701 Neuro1_000106 [O-][N+](=O)c1cccc(c1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E19 compound treatment 163800.0 19600.0 1.34 162520.0 18400.0 1.37 1.9157 0.9999 1714181 Neuro1_000107 Cc1cc(C)cc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E20 compound treatment 171040.0 26800.0 1.83 172280.0 28200.0 2.1 2.7784 0.9977 3652702 Neuro1_000108 CN1CCN(CC1)c2nc(Nc3cccc(Cl)c3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E21 compound treatment 185920.0 41700.0 2.84 186360.0 42300.0 3.15 4.2367 0.9987 1208363 Neuro1_000109 Brc1ccc2ncnc(N(CC=C)CC=C)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E22 compound treatment 147760.0 3570.0 0.24 147080.0 3000.0 0.22 0.3299 0.9991 1578547 Neuro1_000110 CN(C1CCCCC1)c2nc(nc3ccccc23)c4ccccc4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E23 mock treatment 143720.0 -474.0 -0.03 145400.0 1320.0 0.1 0.0467 0.4511 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 E24 mock treatment 148160.0 3970.0 0.27 146920.0 2840.0 0.21 0.3407 0.9926 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F01 compound treatment 150080.0 5890.0 0.4 149440.0 5360.0 0.4 0.5659 1.0 3652703 Neuro1_000111 COc1ccccc1Nc2nc(nc3ccccc23)c4cccc(c4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F02 compound treatment 146280.0 2090.0 0.14 156120.0 12000.0 0.9 0.7343 0.8092 3652704 Neuro1_000112 OCCCNc1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F03 compound treatment 214960.0 70800.0 4.82 215640.0 71600.0 5.33 7.1776 0.9988 3652705 Neuro1_000113 COC(=O)c1ccc(Nc2nc(NCc3ccccc3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F04 compound treatment 158280.0 14100.0 0.96 159360.0 15300.0 1.14 1.4833 0.9965 3652706 Neuro1_000114 COc1ccc(Nc2nc(nc3ccccc23)N4CCOCC4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F05 compound treatment 148880.0 4690.0 0.32 147520.0 3440.0 0.26 0.407 0.994 3652707 Neuro1_000115 COc1ccccc1N2CCN(CC2)c3nc(nc4c(C)cc(C)cc34)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F06 compound treatment 164240.0 20000.0 1.37 169680.0 25600.0 1.91 2.3137 0.9867 1568958 Neuro1_000116 Ic1ccc2ncnc(NCC3CCCO3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F07 compound treatment 184720.0 40500.0 2.76 198040.0 54000.0 4.02 4.7936 0.9833 3652708 Neuro1_000117 C1CCN(CC1)c2nc(Nc3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F08 compound treatment 170920.0 26700.0 1.82 165800.0 21700.0 1.62 2.4316 0.9982 1676459 Neuro1_000118 COC(=O)c1ccc(Nc2ncnc3ccc(I)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F09 compound treatment 153600.0 9410.0 0.64 152960.0 8880.0 0.66 0.9209 0.9999 1986166 Neuro1_000119 CC(Nc1nc(nc2ccccc12)N3CCN(CC3)S(=O)(=O)C)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F10 compound treatment 161760.0 17600.0 1.2 162560.0 18500.0 1.38 1.8195 0.9976 3652709 Neuro1_000120 Brc1cccc(Nc2ncnc3ccccc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F11 compound treatment 148760.0 4570.0 0.31 149840.0 5760.0 0.43 0.5233 0.9876 3652710 Neuro1_000121 Clc1cccc(c1)c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F12 compound treatment 161960.0 17800.0 1.21 162400.0 18300.0 1.36 1.8207 0.9983 3652711 Neuro1_000122 O=S(=O)(Nc1nccs1)c2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F13 compound treatment 180760.0 36600.0 2.49 171560.0 27500.0 2.05 3.2091 0.9952 3652712 Neuro1_000123 O=C(NCc1ccccc1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F14 compound treatment 199400.0 55200.0 3.76 202120.0 58000.0 4.32 5.716 0.9976 1179362 Neuro1_000124 Cc1ccc(O)c(Nc2nc(nc3ccccc23)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F15 compound treatment 190360.0 46200.0 3.15 192440.0 48400.0 3.6 4.7707 0.9978 3652713 Neuro1_000125 COCCCNc1ncnc2ccc(I)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F16 compound treatment 186040.0 41800.0 2.85 178640.0 34600.0 2.57 3.8362 0.9987 3652714 Neuro1_000126 COc1ccc(cc1Nc2ncnc3ccc(Br)cc23)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F17 compound treatment 168520.0 24300.0 1.66 170840.0 26800.0 1.99 2.5811 0.9959 1600380 Neuro1_000127 CCOC(=O)c1nc(Nc2ccc(C)c(Cl)c2)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F18 compound treatment 155000.0 10800.0 0.74 153400.0 9320.0 0.69 1.0115 0.9995 3652715 Neuro1_000128 CC(Nc1nc(nc2ccccc12)N3CCCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F19 compound treatment 171080.0 26900.0 1.83 170000.0 25900.0 1.93 2.6603 0.9997 3652716 Neuro1_000129 CCOC(=O)c1nc(Nc2ccc(cc2)N3CCOCC3)c4ccccc4n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F20 compound treatment 222720.0 78500.0 5.35 218520.0 74400.0 5.54 7.7033 0.9999 3652717 Neuro1_000130 COc1cccc(Nc2nc(NCC3CCCO3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F21 compound treatment 180680.0 36500.0 2.49 182760.0 38700.0 2.88 3.7946 0.9974 3652718 Neuro1_000131 COc1ccc(cc1Nc2nc(nc3ccccc23)c4ccccc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F22 compound treatment 153120.0 8930.0 0.61 146720.0 2640.0 0.2 0.5693 0.8902 3652719 Neuro1_000132 OCCN1CCN(CC1)c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F23 mock treatment 143360.0 -834.0 -0.06 142800.0 -1280.0 -0.1 -0.1075 -0.9696 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 F24 mock treatment 142800.0 -1390.0 -0.1 143280.0 -799.0 -0.06 -0.1092 -0.9745 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G01 compound treatment 161040.0 16800.0 1.15 152400.0 8320.0 0.62 1.2501 0.958 1201768 Neuro1_000133 CCCNc1nc(nc2ccccc12)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G02 compound treatment 161080.0 16900.0 1.15 158280.0 14200.0 1.06 1.5614 0.9991 3652720 Neuro1_000134 CCN(CC)c1nc(nc2ccccc12)N3CCOCC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G03 compound treatment 174280.0 30100.0 2.05 172840.0 28800.0 2.14 2.964 0.9998 1236128 Neuro1_000135 CCOc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G04 compound treatment 167040.0 22800.0 1.56 161560.0 17500.0 1.3 2.0214 0.996 1935323 Neuro1_000136 Cc1ccc(cc1)c2nc(N/N=C/c3ccccc3O)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G05 compound treatment 162880.0 18700.0 1.27 159880.0 15800.0 1.18 1.7324 0.9992 1614179 Neuro1_000137 CCOc1ccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G06 compound treatment 189120.0 44900.0 3.06 192080.0 48000.0 3.57 4.692 0.9971 3652721 Neuro1_000138 CCOc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G07 compound treatment 258880.0 115000.0 7.82 270880.0 127000.0 9.44 12.2021 0.9956 1257914 Neuro1_000139 COc1cccc(Nc2nc(nc3ccccc23)c4cccnc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G08 compound treatment 162560.0 18400.0 1.25 157680.0 13600.0 1.01 1.6012 0.9944 3652723 Neuro1_000140 COc1cccc2c(nc(nc12)C(Cl)(Cl)Cl)N3CCN(Cc4ccccc4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G09 compound treatment 166280.0 22100.0 1.51 164680.0 20600.0 1.53 2.1489 1.0 1954230 Neuro1_000141 FC(F)(F)c1cccc(Nc2nc(nc3ccccc23)c4cccnc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G10 compound treatment 154320.0 10100.0 0.69 158880.0 14800.0 1.1 1.2671 0.9747 3652724 Neuro1_000142 CCN1CCN(CC1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G11 compound treatment 213480.0 69300.0 4.72 211920.0 67800.0 5.05 6.9105 0.9994 1243756 Neuro1_000143 CCOc1ccc(Nc2nc(nc3ccccc23)c4cccnc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G12 compound treatment 162400.0 18200.0 1.24 160480.0 16400.0 1.22 1.7409 1.0 3652725 Neuro1_000144 COc1ccc(C)cc1Nc2nc(N)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G13 compound treatment 240800.0 96600.0 6.59 253360.0 109000.0 8.13 10.4085 0.9945 1154520 Neuro1_000145 CCN(Cc1ccccc1)c2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G14 compound treatment 215840.0 71600.0 4.88 198440.0 54400.0 4.05 6.3149 0.9956 3652726 Neuro1_000146 OCCNc1nc(Nc2ccc(Cl)c(Cl)c2)nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G15 compound treatment 212960.0 68800.0 4.69 228400.0 84300.0 6.28 7.7527 0.9897 1361807 Neuro1_000147 Cc1ccc(C)c(Nc2nc(nc3ccccc23)c4ccccc4O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G16 compound treatment 160800.0 16600.0 1.13 157960.0 13900.0 1.03 1.5311 0.999 3652727 Neuro1_000148 CCN1CCN(CC1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G17 compound treatment 186560.0 42400.0 2.89 185520.0 41400.0 3.08 4.2234 0.9995 1383741 Neuro1_000149 CC(=O)Nc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G18 compound treatment 183520.0 39300.0 2.68 184280.0 40200.0 2.99 4.0116 0.9985 3652728 Neuro1_000150 COC(=O)c1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G19 compound treatment 173640.0 29400.0 2.01 172920.0 28800.0 2.15 2.9374 0.9994 1379452 Neuro1_000151 CC(C)OC(=O)c1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G20 compound treatment 155760.0 11600.0 0.79 156400.0 12300.0 0.92 1.206 0.9972 3652729 Neuro1_000152 COc1ccc(Cc2nc(NCC3CCCO3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G21 compound treatment 167880.0 23700.0 1.61 158680.0 14600.0 1.09 1.9103 0.9814 1580613 Neuro1_000153 COc1ccc(CCNc2ncnc3ccc(Br)cc23)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G22 compound treatment 177280.0 33100.0 2.26 175440.0 31400.0 2.33 3.2455 0.9999 3652730 Neuro1_000154 Oc1cccc(Nc2nc(N3CCOCC3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G23 mock treatment 153280.0 9090.0 0.62 151280.0 7200.0 0.54 0.817 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 G24 mock treatment 145600.0 1410.0 0.1 146640.0 2560.0 0.19 0.2026 0.9494 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H01 compound treatment 157280.0 13100.0 0.89 149800.0 5720.0 0.43 0.932 0.9427 1141229 Neuro1_000155 Fc1ccccc1c2nc(N3CCN(Cc4ccccc4)CC3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H02 compound treatment 165760.0 21600.0 1.47 168840.0 24800.0 1.84 2.3428 0.9937 1523458 Neuro1_000156 O=C(Oc1ccc(Nc2ncnc3ccccc23)cc1)c4ccncc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H03 compound treatment 160040.0 15800.0 1.08 159920.0 15800.0 1.18 1.5976 0.999 3652731 Neuro1_000157 Cc1ccc(OCCN2CCN(CC2)c3nc(NCc4ccccc4)c5ccccc5n3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H04 compound treatment 174720.0 30500.0 2.08 173200.0 29100.0 2.17 3.0042 0.9998 3652732 Neuro1_000158 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(CC4)c5ccc(cc5)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H05 compound treatment 180160.0 36000.0 2.45 178080.0 34000.0 2.53 3.5233 0.9999 3652733 Neuro1_000159 Oc1ccccc1Nc2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H06 compound treatment 187040.0 42800.0 2.92 183600.0 39500.0 2.94 4.1455 1.0 1329695 Neuro1_000160 Ic1ccc2ncnc(Nc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H07 compound treatment 198200.0 54000.0 3.68 196840.0 52800.0 3.93 5.3803 0.9995 1487640 Neuro1_000161 Oc1ccc(Cl)cc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H08 compound treatment 162080.0 17900.0 1.22 159840.0 15800.0 1.17 1.6917 0.9998 3652734 Neuro1_000162 CN1CCN(CC1)c2nc(NC3CCCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H09 compound treatment 181360.0 37200.0 2.53 180040.0 36000.0 2.68 3.6843 0.9996 3652735 Neuro1_000163 [O-][N+](=O)c1ccc2ncnc(N(Cc3ccccc3)Cc4ccccc4)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H10 compound treatment 169640.0 25400.0 1.73 168000.0 23900.0 1.78 2.4856 0.9999 3652736 Neuro1_000164 Ic1cccc(Nc2ncnc3ccccc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H11 compound treatment 158480.0 14300.0 0.97 159080.0 15000.0 1.12 1.4782 0.9977 3652737 Neuro1_000165 Clc1cccc(c1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H12 compound treatment 167200.0 23000.0 1.57 162400.0 18300.0 1.36 2.0733 0.9976 3652738 Neuro1_000166 Cc1c(Nc2nc(nc3ccccc23)C(F)(F)F)c(=O)n(c4ccccc4)n1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H13 compound treatment 206760.0 62600.0 4.27 200040.0 56000.0 4.17 5.9613 0.9999 1433926 Neuro1_000167 Ic1ccc2ncnc(NC3CCCCC3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H14 compound treatment 179360.0 35200.0 2.4 183520.0 39400.0 2.94 3.771 0.995 3652739 Neuro1_000168 [O-][N+](=O)c1ccc(cc1)C(=O)Oc2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H15 compound treatment 175440.0 31200.0 2.13 169080.0 25000.0 1.86 2.8221 0.9977 1274605 Neuro1_000169 OC(=O)c1cccc(Nc2ncnc3ccc(I)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H16 compound treatment 189080.0 44900.0 3.06 190920.0 46800.0 3.49 4.629 0.9979 1469064 Neuro1_000170 Fc1ccc(Nc2ncnc3ccc(Br)cc23)cc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H17 compound treatment 162640.0 18400.0 1.26 162880.0 18800.0 1.4 1.8787 0.9986 1262527 Neuro1_000171 CCOC(=O)c1nc(Nc2cc(C)cc(C)c2)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H18 compound treatment 160080.0 15900.0 1.08 162400.0 18300.0 1.36 1.7301 0.9935 3119176 Neuro1_000172 CC(Nc1nc(nc2ccccc12)N3CCNCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H19 compound treatment 156240.0 12000.0 0.82 152800.0 8720.0 0.65 1.0397 0.9932 1413519 Neuro1_000173 CCOC(=O)c1nc(Nc2cc(Cl)ccc2OC)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H20 compound treatment 152200.0 8010.0 0.55 157920.0 13800.0 1.03 1.1144 0.9559 3652740 Neuro1_000174 Cc1cc(C)c2nc(nc(N3CCN(CCO)CC3)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H21 compound treatment 160200.0 16000.0 1.09 156640.0 12600.0 0.93 1.4327 0.997 1557489 Neuro1_000175 C(N1CCN(CC1)c2ncnc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H22 compound treatment 164120.0 19900.0 1.36 164520.0 20400.0 1.52 2.0364 0.9984 3652741 Neuro1_000176 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(CC4)S(=O)(=O)C)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H23 mock treatment 148800.0 4610.0 0.31 143120.0 -959.0 -0.07 0.1716 0.5329 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 H24 mock treatment 146720.0 2530.0 0.17 144440.0 361.0 0.03 0.1408 0.8077 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I01 compound treatment 165160.0 21000.0 1.43 167800.0 23700.0 1.77 2.2591 0.9945 1985684 Neuro1_000177 COC(=O)c1ccc(Nc2nc(N3CCN(C)CC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I02 compound treatment 152720.0 8530.0 0.58 153520.0 9440.0 0.7 0.9079 0.9956 3652742 Neuro1_000178 CCN(CC)c1nc(Nc2ccncc2)nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I03 compound treatment 153640.0 9450.0 0.64 156840.0 12800.0 0.95 1.127 0.9821 1983321 Neuro1_000179 C(CNc1nc(nc2ccccc12)c3ccccc3)CN4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I04 compound treatment 180760.0 36600.0 2.49 177920.0 33800.0 2.52 3.5438 1.0 1935653 Neuro1_000180 COc1cccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I05 compound treatment 167720.0 23500.0 1.6 168160.0 24100.0 1.79 2.4015 0.9985 1674338 Neuro1_000181 C1CN(CCO1)c2nc(Nc3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I06 compound treatment 175720.0 31500.0 2.15 175640.0 31600.0 2.35 3.1808 0.999 3652743 Neuro1_000182 Cc1c(O)ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I07 compound treatment 166800.0 22600.0 1.54 166320.0 22200.0 1.66 2.2603 0.9994 1141952 Neuro1_000183 Cc1ccccc1Nc2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I08 compound treatment 159400.0 15200.0 1.04 156120.0 12000.0 0.9 1.3668 0.9974 3652745 Neuro1_000184 CN1CCN(CC1)c2nc(NCCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I09 compound treatment 259160.0 115000.0 7.84 254560.0 110000.0 8.22 11.3567 0.9997 1313914 Neuro1_000185 CCOc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I10 compound treatment 194560.0 50400.0 3.43 191560.0 47500.0 3.53 4.9269 0.9999 3652746 Neuro1_000186 CN(C)c1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I11 compound treatment 159440.0 15200.0 1.04 156960.0 12900.0 0.96 1.4129 0.9992 1591665 Neuro1_000187 OCCN1CCN(CC1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I12 compound treatment 159400.0 15200.0 1.04 159800.0 15700.0 1.17 1.5604 0.9982 3652747 Neuro1_000188 C(Cc1ccccc1)Nc2nc(nc3ccccc23)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I13 compound treatment 159480.0 15300.0 1.04 162600.0 18500.0 1.38 1.7117 0.9905 1382464 Neuro1_000189 CC1CC(C)CN(C1)c2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I14 compound treatment 181760.0 37600.0 2.56 186000.0 41900.0 3.12 4.0172 0.9952 3652748 Neuro1_000190 Cc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I15 compound treatment 173840.0 29600.0 2.02 171560.0 27500.0 2.05 2.8755 1.0 3652749 Neuro1_000191 Oc1ccccc1c2nc(Nc3cccc(c3)C(F)(F)F)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I16 compound treatment 164080.0 19900.0 1.36 173920.0 29800.0 2.22 2.5292 0.972 3652750 Neuro1_000192 COc1ccc(OC)c(Nc2nc(N3CCOCC3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I17 compound treatment 186360.0 42200.0 2.87 186440.0 42400.0 3.15 4.2621 0.9989 1620739 Neuro1_000193 Clc1ccc(Nc2ncnc3ccc(Br)cc23)cc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I18 compound treatment 155120.0 10900.0 0.74 156640.0 12600.0 0.93 1.1878 0.9937 3652751 Neuro1_000194 CC(Nc1nc(nc2ccccc12)c3cccc(c3)[N+](=O)[O-])c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I19 compound treatment 164760.0 20600.0 1.4 163200.0 19100.0 1.42 1.9978 1.0 3652752 Neuro1_000195 CC1CCCN(C1)c2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I20 compound treatment 158760.0 14600.0 0.99 159880.0 15800.0 1.18 1.5338 0.9965 3652753 Neuro1_000196 COc1ccccc1N2CCN(CC2)c3nc(nc4ccccc34)c5cccc(c5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I21 compound treatment 222560.0 78400.0 5.34 218280.0 74200.0 5.52 7.683 0.9999 3652754 Neuro1_000197 CCN1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I22 compound treatment 149160.0 4970.0 0.34 149920.0 5840.0 0.43 0.5468 0.9924 3652755 Neuro1_000198 CN1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I23 mock treatment 147120.0 2930.0 0.2 149200.0 5120.0 0.38 0.4106 0.9544 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 I24 mock treatment 143840.0 -354.0 -0.02 139280.0 -4800.0 -0.36 -0.2696 -0.7531 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J01 compound treatment 156560.0 12400.0 0.84 159240.0 15200.0 1.13 1.3941 0.9897 3652756 Neuro1_000199 Fc1ccccc1Nc2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J02 compound treatment 152720.0 8530.0 0.58 151880.0 7800.0 0.58 0.8216 1.0 3652757 Neuro1_000200 CN1CCN(CC1)c2nc(nc3ccccc23)N4CCN(CC4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J03 compound treatment 170640.0 26400.0 1.8 178080.0 34000.0 2.53 3.0643 0.9862 3652758 Neuro1_000201 CC(C)(C)Nc1nc(nc2ccccc12)c3cccc(c3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J04 compound treatment 162720.0 18500.0 1.26 159000.0 14900.0 1.11 1.6784 0.9979 3209382 Neuro1_000202 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc(NC4CCCC4)c5ccccc5n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J05 compound treatment 201840.0 57600.0 3.93 196480.0 52400.0 3.9 5.5368 1.0 3652759 Neuro1_000203 Oc1ccccc1Nc2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J06 compound treatment 180960.0 36800.0 2.51 175640.0 31600.0 2.35 3.4334 0.9995 1353170 Neuro1_000204 COc1ccc(Nc2ncnc3ccc(I)cc23)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J07 compound treatment 161600.0 17400.0 1.19 158360.0 14300.0 1.06 1.5907 0.9985 3086809 Neuro1_000205 CN1CCN(CC1)c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J08 compound treatment 162320.0 18100.0 1.24 156960.0 12900.0 0.96 1.5517 0.9921 3652760 Neuro1_000206 Cc1c(Cl)cccc1Nc2nc(NCCO)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J09 compound treatment 173720.0 29500.0 2.01 171320.0 27200.0 2.03 2.8571 1.0 3652761 Neuro1_000207 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(CC4)S(=O)(=O)c5ccc(C)cc5)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J10 compound treatment 157160.0 13000.0 0.88 163880.0 19800.0 1.47 1.6672 0.9701 3652762 Neuro1_000208 CC1CN(CC(C)N1)c2nc(nc3ccccc23)N4CCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J11 compound treatment 152680.0 8490.0 0.58 151240.0 7160.0 0.53 0.786 0.9992 3652763 Neuro1_000209 Clc1cccc(c1)c2nc(NCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J12 compound treatment 182640.0 38400.0 2.62 179000.0 34900.0 2.6 3.6913 1.0 1170239 Neuro1_000210 Brc1ccc2ncnc(Nc3cccc(OC(=O)c4cccs4)c3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J13 compound treatment 160920.0 16700.0 1.14 163120.0 19000.0 1.42 1.8084 0.9942 1617762 Neuro1_000211 Ic1ccc2ncnc(NCCN3CCOCC3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J14 compound treatment 177920.0 33700.0 2.3 181240.0 37200.0 2.77 3.5816 0.9958 1523583 Neuro1_000212 Oc1cccc(Nc2nc(nc3ccccc23)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J15 compound treatment 218240.0 74000.0 5.05 212600.0 68500.0 5.1 7.1758 1.0 1234275 Neuro1_000213 Ic1ccc2ncnc(Nc3ccc4OCCOc4c3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J16 compound treatment 165000.0 20800.0 1.42 161800.0 17700.0 1.32 1.9357 0.9993 1985883 Neuro1_000214 COc1ccc(Nc2nc(nc3ccccc23)N4CCCC4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J17 compound treatment 165280.0 21100.0 1.44 164040.0 20000.0 1.49 2.067 0.9999 3652764 Neuro1_000215 CCCOc1ccccc1Nc2nc(nc3ccccc23)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J18 compound treatment 149680.0 5490.0 0.37 149920.0 5840.0 0.43 0.5719 0.9972 3652765 Neuro1_000216 C1CN(CCO1)c2nc(NC3C4CC5CC(C4)CC3C5)c6ccccc6n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J19 compound treatment 170640.0 26400.0 1.8 173080.0 29000.0 2.16 2.8012 0.996 1424113 Neuro1_000217 CC(C)Oc1ccccc1Nc2ncnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J20 compound treatment 159680.0 15500.0 1.06 160040.0 16000.0 1.19 1.5866 0.9983 3652766 Neuro1_000218 OCCNc1nc(Nc2ccc(Cl)cc2)nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J21 compound treatment 168760.0 24600.0 1.67 172480.0 28400.0 2.11 2.679 0.9934 1120309 Neuro1_000219 COc1ccc(OC)c(Nc2ncnc3ccccc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J22 compound treatment 145560.0 1370.0 0.09 151200.0 7120.0 0.53 0.4406 0.8188 1661495 Neuro1_000220 CC(C)CC(Nc1ncnc2ccc(C)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J23 mock treatment 146240.0 2050.0 0.14 149400.0 5320.0 0.4 0.3787 0.9019 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 J24 mock treatment 141800.0 -2390.0 -0.16 142800.0 -1280.0 -0.1 -0.1827 -0.967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K01 compound treatment 154720.0 10500.0 0.72 154440.0 10400.0 0.77 1.0527 0.9994 3652767 Neuro1_000221 CC1CCCCN1c2nc(nc3ccccc23)c4cccc(c4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K02 compound treatment 152360.0 8170.0 0.56 156280.0 12200.0 0.91 1.0358 0.9724 3652768 Neuro1_000222 CCN1CCN(CC1)c2nc(N3CCCC(C)C3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K03 compound treatment 157320.0 13100.0 0.89 158760.0 14700.0 1.09 1.4054 0.9951 1698023 Neuro1_000223 Clc1ccc(cc1)c2nc(Nc3ccc(I)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K04 compound treatment 179720.0 35500.0 2.42 175640.0 31600.0 2.35 3.3737 0.9999 3652769 Neuro1_000224 Cc1ccc(cc1)c2nc(N/N=C/c3cc(Br)ccc3O)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K05 compound treatment 213040.0 68800.0 4.69 199600.0 55500.0 4.13 6.2409 0.998 1623340 Neuro1_000225 Brc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K06 compound treatment 219520.0 75300.0 5.14 211640.0 67600.0 5.03 7.187 0.9999 3652771 Neuro1_000226 Oc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K07 compound treatment 159640.0 15400.0 1.05 155640.0 11600.0 0.86 1.3531 0.995 1447318 Neuro1_000227 COc1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K08 compound treatment 325840.0 182000.0 12.38 313000.0 169000.0 12.57 17.6468 1.0 3652773 Neuro1_000228 C1CCC(C1)Nc2nc(Nc3ccc4OCOc4c3)nc5ccccc25 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K09 compound treatment 222920.0 78700.0 5.37 235400.0 91300.0 6.8 8.6013 0.9932 1143902 Neuro1_000229 Clc1cccc(Nc2nc(NCc3ccco3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K10 compound treatment 188440.0 44200.0 3.02 194400.0 50300.0 3.75 4.7813 0.9942 3652774 Neuro1_000230 CN(C)c1ccc(Nc2nc(NCC3CCCO3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K11 compound treatment 242680.0 98500.0 6.71 258120.0 114000.0 8.49 10.7496 0.9933 1465833 Neuro1_000231 C(Nc1nc(Nc2ccccc2)nc3ccccc13)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K12 compound treatment 219680.0 75500.0 5.15 217680.0 73600.0 5.48 7.5125 0.9995 3652775 Neuro1_000232 Nc1nc(Nc2ccc(Cl)c(Cl)c2)nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K13 compound treatment 177000.0 32800.0 2.24 177200.0 33100.0 2.47 3.3246 0.9988 1154723 Neuro1_000233 Cc1ccc(Nc2ncnc3ccc(Br)cc23)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K14 compound treatment 187160.0 43000.0 2.93 189720.0 45600.0 3.4 4.4733 0.9973 3652776 Neuro1_000234 CN(C)c1ccc(Nc2nc(NCCO)c3ccccc3n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K15 compound treatment 191080.0 46900.0 3.2 192800.0 48700.0 3.63 4.8244 0.998 1458204 Neuro1_000235 Oc1ccccc1c2nc(Nc3ccc(F)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K16 compound treatment 165400.0 21200.0 1.45 164080.0 20000.0 1.49 2.0749 0.9999 3652777 Neuro1_000236 COc1ccc(Cl)cc1Nc2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K17 compound treatment 202840.0 58600.0 4.0 199160.0 55100.0 4.1 5.726 0.9999 1601387 Neuro1_000237 Oc1ccccc1c2nc(Nc3ccccc3Cl)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K18 compound treatment 170280.0 26100.0 1.78 161480.0 17400.0 1.3 2.1734 0.9879 1495821 Neuro1_000238 COc1ccc(cc1)c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K19 compound treatment 188600.0 44400.0 3.03 189440.0 45400.0 3.38 4.528 0.9985 1322048 Neuro1_000239 COC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccccc4O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K20 compound treatment 155240.0 11000.0 0.75 154600.0 10500.0 0.78 1.0862 0.9998 1153244 Neuro1_000240 COc1ccc(cc1)c2nc(NCC=C)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K21 compound treatment 211320.0 67100.0 4.58 216480.0 72400.0 5.39 7.0464 0.9967 1320708 Neuro1_000241 Brc1ccc2ncnc(Nc3ccc(cc3)N4CCCC4)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K22 compound treatment 151760.0 7570.0 0.52 154840.0 10800.0 0.8 0.9311 0.9774 3652778 Neuro1_000242 COc1ccccc1Nc2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K23 mock treatment 146840.0 2650.0 0.18 144160.0 81.3 0.01 0.1318 0.7304 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 K24 mock treatment 144280.0 86.3 0.01 145520.0 1440.0 0.11 0.08 0.7448 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L01 compound treatment 190800.0 46600.0 3.18 194440.0 50400.0 3.75 4.8972 0.9966 3652779 Neuro1_000243 CN1CCN(CC1)c2nc(Nc3ccc(O)cc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L02 compound treatment 261960.0 118000.0 8.03 259120.0 115000.0 8.56 11.7317 0.9995 3652780 Neuro1_000244 Oc1cccc(Nc2nc(NCc3ccccc3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L03 compound treatment 154440.0 10200.0 0.7 155960.0 11900.0 0.88 1.1192 0.9932 3652781 Neuro1_000245 CN(Cc1ccccc1)c2nc(nc3ccccc23)c4cccc(c4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L04 compound treatment 154360.0 10200.0 0.69 157520.0 13400.0 1.0 1.1975 0.9839 3652782 Neuro1_000246 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(CCO)CC4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L05 compound treatment 167880.0 23700.0 1.61 167800.0 23700.0 1.77 2.3903 0.999 3652783 Neuro1_000247 Fc1cccc(Nc2nc(NCC3CCCO3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L06 compound treatment 177040.0 32800.0 2.24 177520.0 33400.0 2.49 3.3434 0.9986 3652784 Neuro1_000248 CC(=O)c1cccc(Nc2ncnc3ccc(I)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L07 compound treatment 174240.0 30000.0 2.05 155760.0 11700.0 0.87 2.0632 0.9272 3652785 Neuro1_000249 COc1ccc(cc1)N2CCN(CC2)c3nc(nc4c(C)cc(C)cc34)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L08 compound treatment 163040.0 18800.0 1.28 159720.0 15600.0 1.16 1.7317 0.9988 3652786 Neuro1_000250 CCN1CCN(CC1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L09 compound treatment 168440.0 24200.0 1.65 169760.0 25700.0 1.91 2.5204 0.9974 3652787 Neuro1_000251 CN1CCN(CC1)c2nc(NCCNc3ccc(cc3)[N+](=O)[O-])c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L10 compound treatment 161480.0 17300.0 1.18 165040.0 21000.0 1.56 1.9365 0.9904 3652788 Neuro1_000252 Cc1ccc2ncnc(Nc3cccc(c3)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L11 compound treatment 159280.0 15100.0 1.03 156720.0 12600.0 0.94 1.3926 0.999 3652789 Neuro1_000253 COCCNc1nc(nc2ccccc12)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L12 compound treatment 183240.0 39000.0 2.66 185960.0 41900.0 3.12 4.0865 0.9969 1418789 Neuro1_000254 CC1CCN(CC1)c2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L13 compound treatment 187800.0 43600.0 2.97 176000.0 31900.0 2.38 3.7821 0.9938 1599005 Neuro1_000255 COc1ccccc1Nc2ncnc3ccc(I)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L14 compound treatment 153600.0 9410.0 0.64 149880.0 5800.0 0.43 0.7588 0.9815 1165430 Neuro1_000256 CC(=O)Nc1ccc(Nc2nc(nc3ccccc23)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L15 compound treatment 336400.0 192000.0 13.1 334920.0 191000.0 14.2 19.3095 0.9992 1624986 Neuro1_000257 Oc1cccc(Nc2ncnc3ccc(I)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L16 compound treatment 208320.0 64100.0 4.37 188880.0 44800.0 3.33 5.4492 0.9911 1706455 Neuro1_000258 O=C(CCc1ccccc1)Oc2ccc(Nc3ncnc4ccccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L17 compound treatment 171000.0 26800.0 1.83 169480.0 25400.0 1.89 2.6291 0.9999 3652790 Neuro1_000259 CCOC(=O)c1nc(Nc2cc(ccc2O)[N+](=O)[O-])c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L18 compound treatment 154680.0 10500.0 0.71 158240.0 14200.0 1.05 1.2508 0.9821 3211569 Neuro1_000260 CC(Nc1nc(nc2ccccc12)N3CCOCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L19 compound treatment 169000.0 24800.0 1.69 174440.0 30400.0 2.26 2.7937 0.9898 1534926 Neuro1_000261 CC(C)C(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L20 compound treatment 154880.0 10700.0 0.73 155520.0 11400.0 0.85 1.1173 0.997 3652791 Neuro1_000262 C(Nc1nc(nc2ccccc12)N3CCOCC3)C4CCCO4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L21 compound treatment 159840.0 15600.0 1.07 152400.0 8320.0 0.62 1.1922 0.9666 1624571 Neuro1_000263 O=C(Oc1ccc(Nc2ncnc3ccccc23)cc1)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L22 compound treatment 155640.0 11400.0 0.78 154520.0 10400.0 0.78 1.1013 1.0 1447467 Neuro1_000264 COc1ccc(CCNc2ncnc3ccccc23)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L23 mock treatment 149360.0 5170.0 0.35 146040.0 1960.0 0.15 0.3523 0.924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 L24 mock treatment 141760.0 -2430.0 -0.17 146800.0 2720.0 0.2 0.0259 0.0989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M01 compound treatment 267600.0 123000.0 8.41 196240.0 52200.0 3.88 8.6943 0.9383 3652792 Neuro1_000265 Oc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M02 compound treatment 158520.0 14300.0 0.98 158480.0 14400.0 1.07 1.4486 0.9989 3652793 Neuro1_000266 CCN(CC)c1nc(nc2ccccc12)N3CCN(C)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M03 compound treatment 195120.0 50900.0 3.47 201720.0 57600.0 4.29 5.4886 0.9945 1304107 Neuro1_000267 CCOC(=O)c1cccc(Nc2nc(nc3ccccc23)c4cccnc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M04 compound treatment 180160.0 36000.0 2.45 173840.0 29800.0 2.22 3.3001 0.9987 3652794 Neuro1_000268 Cc1ccc(cc1)c2nc(N/N=C/c3c(O)ccc4ccccc34)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M05 compound treatment 313520.0 169000.0 11.54 311600.0 168000.0 12.47 16.9792 0.9993 1282699 Neuro1_000269 CC(Nc1nc(nc2ccccc12)c3cccnc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M06 compound treatment 176320.0 32100.0 2.19 165640.0 21600.0 1.6 2.6835 0.9883 3652796 Neuro1_000270 COc1cc2ncnc(Nc3c(C)n(C)n(c4ccccc4)c3=O)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M07 compound treatment 199800.0 55600.0 3.79 190360.0 46300.0 3.44 5.1164 0.9989 1294207 Neuro1_000271 Clc1cccc(Nc2nc(N3CCOCC3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M08 compound treatment 169280.0 25100.0 1.71 171280.0 27200.0 2.02 2.6409 0.9965 3652797 Neuro1_000272 Cc1ccc(Nc2nc(NCCO)c3ccccc3n2)cc1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M09 compound treatment 164880.0 20700.0 1.41 158400.0 14300.0 1.07 1.7509 0.9905 1726085 Neuro1_000273 OCCN1CCN(CC1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M10 compound treatment 171240.0 27000.0 1.84 177640.0 33600.0 2.5 3.0701 0.9888 3652798 Neuro1_000274 COc1ccc(OC)c(Nc2nc(N3CCCCC3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M11 compound treatment 174360.0 30200.0 2.06 176160.0 32100.0 2.39 3.1426 0.9972 1627384 Neuro1_000275 C(CN1CCOCC1)Nc2nc(nc3ccccc23)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M12 compound treatment 173280.0 29100.0 1.98 172000.0 27900.0 2.08 2.8716 0.9997 3652799 Neuro1_000276 COc1ccc(OC)c(Nc2nc(NCCO)c3ccccc3n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M13 compound treatment 191560.0 47400.0 3.23 187920.0 43800.0 3.26 4.5907 1.0 1298176 Neuro1_000277 CCCOc1ccccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M14 compound treatment 160000.0 15800.0 1.08 155880.0 11800.0 0.88 1.3831 0.9948 3652800 Neuro1_000278 CCN1CCN(CC1)c2nc(NCCO)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M15 compound treatment 178000.0 33800.0 2.3 179840.0 35800.0 2.66 3.5118 0.9974 1359384 Neuro1_000279 CC(Nc1ncnc2ccc(Br)cc12)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M16 compound treatment 170720.0 26500.0 1.81 169920.0 25800.0 1.92 2.6388 0.9995 3652801 Neuro1_000280 Cc1ccccc1Nc2nc(nc3ccccc23)c4cccc(c4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M17 compound treatment 179040.0 34800.0 2.38 185920.0 41800.0 3.11 3.8819 0.9911 3652802 Neuro1_000281 Oc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M18 compound treatment 155880.0 11700.0 0.8 156960.0 12900.0 0.96 1.2413 0.9958 3652803 Neuro1_000282 Clc1ccc2nc(nc(N3CCCCC3)c2c1)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M19 compound treatment 161640.0 17400.0 1.19 159080.0 15000.0 1.12 1.6305 0.9995 1533661 Neuro1_000283 CCCOc1ccc(cc1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M20 compound treatment 168320.0 24100.0 1.64 160240.0 16200.0 1.2 2.0136 0.9882 3652804 Neuro1_000284 [O-][N+](=O)c1cccc(c1)c2nc(N3CCN(CC3)c4ccccc4)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M21 compound treatment 168840.0 24600.0 1.68 171600.0 27500.0 2.05 2.6365 0.9952 1672231 Neuro1_000285 CCOc1ccccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M22 compound treatment 195680.0 51500.0 3.51 183720.0 39600.0 2.95 4.5683 0.9963 3652805 Neuro1_000286 [O-][N+](=O)c1cccc(c1)c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M23 mock treatment 149480.0 5290.0 0.36 155520.0 11400.0 0.85 0.857 0.9268 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 M24 mock treatment 146960.0 2770.0 0.19 149640.0 5560.0 0.41 0.426 0.9366 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N01 compound treatment 166080.0 21900.0 1.49 168280.0 24200.0 1.8 2.3288 0.9956 3652806 Neuro1_000287 [O-][N+](=O)c1cccc(c1)c2nc(Nc3ccc(F)c(F)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N02 compound treatment 164160.0 20000.0 1.36 156320.0 12200.0 0.91 1.6068 0.9809 3652807 Neuro1_000288 CCN(CC)CCCNc1nc(nc2ccccc12)c3ccc(OC)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N03 compound treatment 155680.0 11500.0 0.78 156040.0 12000.0 0.89 1.1832 0.998 3652808 Neuro1_000289 OCCNc1nc(nc2ccccc12)N3CCN(Cc4ccccc4)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N04 compound treatment 154880.0 10700.0 0.73 155040.0 11000.0 0.82 1.092 0.9984 3652809 Neuro1_000290 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc(NC4CCCC4)c5ccccc5n3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N05 compound treatment 155520.0 11300.0 0.77 154800.0 10700.0 0.8 1.1103 0.9999 3652810 Neuro1_000291 Cc1cc(C)c2nc(nc(NCc3ccc4OCOc4c3)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N06 compound treatment 207640.0 63400.0 4.33 174000.0 29900.0 2.23 4.6333 0.9523 3652811 Neuro1_000292 OCCOCCNc1ncnc2ccc(I)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N07 compound treatment 169680.0 25500.0 1.74 159640.0 15600.0 1.16 2.0476 0.9806 3652812 Neuro1_000293 Cc1cc(C)c2nc(nc(NCCCN3CCOCC3)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N08 compound treatment 217280.0 73100.0 4.98 208280.0 64200.0 4.78 6.9021 0.9998 1144684 Neuro1_000294 Cc1ccc(O)c(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N09 compound treatment 172840.0 28600.0 1.95 172520.0 28400.0 2.12 2.8778 0.9992 3652813 Neuro1_000295 C1CN(CCO1)c2ccc(Nc3nc(nc4ccccc34)N5CCOCC5)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N10 compound treatment 175840.0 31600.0 2.16 168000.0 23900.0 1.78 2.7845 0.9954 3652814 Neuro1_000296 OC(=O)C1CCCN1c2nc(nc3ccccc23)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N11 compound treatment 173200.0 29000.0 1.98 159800.0 15700.0 1.17 2.2257 0.9686 3652815 Neuro1_000297 CCN(CC)CCNc1nc(nc2ccccc12)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N12 compound treatment 177160.0 33000.0 2.25 179480.0 35400.0 2.63 3.4523 0.9969 1650814 Neuro1_000298 N(c1ccc(Oc2ccccc2)cc1)c3ncnc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N13 compound treatment 182240.0 38000.0 2.59 182920.0 38800.0 2.89 3.8783 0.9985 3652816 Neuro1_000299 CC(=O)c1ccc(Nc2ncnc3ccc(I)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N14 compound treatment 168200.0 24000.0 1.64 162040.0 18000.0 1.34 2.1026 0.995 3652817 Neuro1_000300 COc1ccc(Nc2nc(nc3ccccc23)N4CCCCC4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N15 compound treatment 182280.0 38100.0 2.6 184160.0 40100.0 2.98 3.9455 0.9976 3652818 Neuro1_000301 CC(Nc1nc(nc2ccccc12)N3CCN(CC3)C(=O)c4ccc(Cl)cc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N16 compound treatment 160720.0 16500.0 1.13 161520.0 17400.0 1.3 1.7146 0.9975 1426920 Neuro1_000302 CN(C1CCN(C)CC1)c2nc(nc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N17 compound treatment 167080.0 22900.0 1.56 164600.0 20500.0 1.53 2.1833 0.9999 1368755 Neuro1_000303 CCOC(=O)c1nc(Nc2ccc(F)cc2)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N18 compound treatment 166760.0 22600.0 1.54 169880.0 25800.0 1.92 2.4457 0.994 3652819 Neuro1_000304 [O-][N+](=O)c1cc(ccc1NCCCNc2nc(nc3ccccc23)N4CCOCC4)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N19 compound treatment 180000.0 35800.0 2.44 180080.0 36000.0 2.68 3.6208 0.9989 1549121 Neuro1_000305 COc1ccc(Cl)cc1Nc2ncnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N20 compound treatment 146080.0 1890.0 0.13 147840.0 3760.0 0.28 0.2889 0.9377 3652820 Neuro1_000306 Cc1cc(C)c2nc(nc(N3CCN(Cc4ccccc4)CC3)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N21 compound treatment 170640.0 26400.0 1.8 167880.0 23800.0 1.77 2.5275 1.0 1173401 Neuro1_000307 O=C(Oc1ccc(Nc2ncnc3ccccc23)cc1)C4CCCCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N22 compound treatment 150920.0 6730.0 0.46 155280.0 11200.0 0.83 0.9138 0.9604 1191667 Neuro1_000308 Fc1ccccc1c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N23 mock treatment 145880.0 1690.0 0.11 146200.0 2120.0 0.16 0.1929 0.9879 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 N24 mock treatment 143240.0 -954.0 -0.07 141880.0 -2200.0 -0.16 -0.1617 -0.9182 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O01 compound treatment 162000.0 17800.0 1.21 152360.0 8280.0 0.62 1.2942 0.9506 1510828 Neuro1_000309 Fc1ccccc1c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O02 compound treatment 156800.0 12600.0 0.86 151400.0 7320.0 0.54 0.993 0.9758 3652821 Neuro1_000310 CC(Nc1nc(nc2ccccc12)N3CCN(C)CC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O03 compound treatment 161920.0 17700.0 1.21 156840.0 12800.0 0.95 1.5261 0.9929 1168079 Neuro1_000311 C1CN(CCO1)c2nc(nc3ccccc23)N4CCN(CC4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O04 compound treatment 173120.0 28900.0 1.97 169520.0 25400.0 1.89 2.7334 0.9998 3652822 Neuro1_000312 COc1cccc(/C=N/Nc2nc(nc3ccccc23)c4cccnc4)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O05 compound treatment 143360.0 -834.0 -0.06 145640.0 1560.0 0.12 0.042 0.3245 1975084 Neuro1_000313 CC(C)(C)c1ccc(cc1)c2nc(NCCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O06 compound treatment 161320.0 17100.0 1.17 163800.0 19700.0 1.47 1.8635 0.9936 3652824 Neuro1_000314 COc1ccc(CNc2nc(nc3c(OC)cccc23)C(Cl)(Cl)Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O07 compound treatment 264600.0 120000.0 8.21 260720.0 117000.0 8.68 11.9432 0.9996 1535722 Neuro1_000315 CN(C)c1ccc(Nc2nc(nc3ccccc23)c4cccnc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O08 compound treatment 156480.0 12300.0 0.84 163880.0 19800.0 1.47 1.6344 0.9642 3652825 Neuro1_000316 CCN1CCN(CC1)c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O09 compound treatment 152200.0 8010.0 0.55 155960.0 11900.0 0.88 1.0113 0.9731 1201288 Neuro1_000317 Cc1c(Cl)cccc1Nc2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O10 compound treatment 149800.0 5610.0 0.38 144400.0 321.0 0.02 0.2872 0.7499 3652826 Neuro1_000318 Cc1ccc(Nc2nc(N)c3ccccc3n2)cc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O11 compound treatment 156320.0 12100.0 0.83 153320.0 9240.0 0.69 1.0709 0.9958 1556983 Neuro1_000319 OCCN1CCN(CC1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O12 compound treatment 157640.0 13400.0 0.92 151280.0 7200.0 0.54 1.0272 0.9673 3652827 Neuro1_000320 C1CCC(CC1)Nc2nc(nc3ccccc23)N4CCOCC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O13 compound treatment 181640.0 37400.0 2.55 184320.0 40200.0 3.0 3.923 0.9968 1641717 Neuro1_000321 COc1ccc(OC)c(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O14 compound treatment 300600.0 156000.0 10.66 297520.0 153000.0 11.42 15.6154 0.9994 3652828 Neuro1_000322 CN(C)c1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O15 compound treatment 159040.0 14800.0 1.01 157400.0 13300.0 0.99 1.4168 0.9999 3652829 Neuro1_000323 CCCOc1ccc(cc1)c2nc(N3CCN(Cc4ccccc4)CC3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O16 compound treatment 162800.0 18600.0 1.27 168960.0 24900.0 1.85 2.2064 0.983 3652830 Neuro1_000324 Cc1ccc(OCCN2CCN(CC2)c3nc(NCc4ccco4)c5ccccc5n3)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O17 compound treatment 204760.0 60600.0 4.13 207240.0 63200.0 4.7 6.2438 0.9979 1330225 Neuro1_000325 CCCN(CCC)c1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O18 compound treatment 164760.0 20600.0 1.4 167520.0 23400.0 1.74 2.2251 0.9941 3652831 Neuro1_000326 COc1ccc(OC)c(Nc2nc(nc3ccccc23)c4cccc(c4)[N+](=O)[O-])c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O19 compound treatment 166600.0 22400.0 1.53 161640.0 17600.0 1.31 2.0044 0.997 1494026 Neuro1_000327 CC1CCCCN1c2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O20 compound treatment 152520.0 8330.0 0.57 154880.0 10800.0 0.8 0.9698 0.9855 1736348 Neuro1_000328 COc1ccc(OC)c(Nc2nc(nc3ccccc23)c4ccccc4F)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O21 compound treatment 186280.0 42100.0 2.87 186840.0 42800.0 3.18 4.2793 0.9987 1492306 Neuro1_000329 COc1ccc(Cl)cc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O22 compound treatment 152560.0 8370.0 0.57 150440.0 6360.0 0.47 0.7381 0.9957 3652832 Neuro1_000330 Fc1ccc(Nc2nc(nc3ccccc23)c4ccccc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O23 mock treatment 148760.0 4570.0 0.31 149640.0 5560.0 0.41 0.5128 0.9901 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 O24 mock treatment 140360.0 -3830.0 -0.26 140960.0 -3120.0 -0.23 -0.349 -0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P01 compound treatment 159360.0 15200.0 1.03 153280.0 9200.0 0.68 1.2154 0.98 3652833 Neuro1_000331 [O-][N+](=O)c1cccc(c1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P02 compound treatment 173680.0 29500.0 2.01 173520.0 29400.0 2.19 2.9709 0.9991 3652834 Neuro1_000332 Oc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P03 compound treatment 158160.0 14000.0 0.95 155960.0 11900.0 0.88 1.2986 0.9993 3652835 Neuro1_000333 Cc1cc(C)c2nc(nc(NCCCN3CCCC3=O)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P04 compound treatment 162080.0 17900.0 1.22 159120.0 15000.0 1.12 1.6539 0.9991 3652836 Neuro1_000334 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(CC4)S(=O)(=O)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P05 compound treatment 167520.0 23300.0 1.59 169080.0 25000.0 1.86 2.4403 0.9969 3652837 Neuro1_000335 OCCNc1nc(Nc2ccc(Br)cc2)nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P06 compound treatment 157000.0 12800.0 0.87 174680.0 30600.0 2.28 2.2278 0.9134 1442987 Neuro1_000336 CC(O)CNc1ncnc2ccc(I)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P07 compound treatment 170000.0 25800.0 1.76 164320.0 20200.0 1.51 2.3093 0.997 3652838 Neuro1_000337 Cc1cc(C)c2nc(nc(N3CCN(CC3)C(=O)c4ccco4)c2c1)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P08 compound treatment 221320.0 77100.0 5.26 232560.0 88500.0 6.59 8.3747 0.9938 1685272 Neuro1_000338 Oc1ccc(Cl)cc1Nc2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P09 compound treatment 164400.0 20200.0 1.38 159960.0 15900.0 1.18 1.8099 0.9971 3652839 Neuro1_000339 [O-][N+](=O)c1ccc(NCCNc2nc(nc3ccccc23)N4CCCC4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P10 compound treatment 155400.0 11200.0 0.76 167080.0 23000.0 1.71 1.7507 0.9339 3652840 Neuro1_000340 OC(=O)C1CCN(CC1)c2nc(nc3ccccc23)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P11 compound treatment 155440.0 11200.0 0.77 153320.0 9240.0 0.69 1.0285 0.9985 3652841 Neuro1_000341 CN(C)CCCNc1nc(nc2ccccc12)c3cccc(Cl)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P12 compound treatment 169640.0 25400.0 1.73 170840.0 26800.0 1.99 2.6351 0.9976 3652842 Neuro1_000342 CCCCOc1ccccc1Nc2ncnc3ccccc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P13 compound treatment 198600.0 54400.0 3.71 197760.0 53700.0 4.0 5.448 0.9993 1617765 Neuro1_000343 Ic1ccc2ncnc(NCc3ccco3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P14 compound treatment 175360.0 31200.0 2.12 174880.0 30800.0 2.29 3.1235 0.9993 1544623 Neuro1_000344 O=C(Oc1ccc(Nc2ncnc3ccccc23)cc1)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P15 compound treatment 197080.0 52900.0 3.61 198200.0 54100.0 4.03 5.3978 0.9985 1134738 Neuro1_000345 Ic1ccc2ncnc(NCCc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P16 compound treatment 152520.0 8330.0 0.57 153200.0 9120.0 0.68 0.8814 0.996 1366684 Neuro1_000346 C1CN(CCN1c2ncnc3ccccc23)c4ncnc5ccccc45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P17 compound treatment 159840.0 15600.0 1.07 159080.0 15000.0 1.12 1.5438 0.9997 3652843 Neuro1_000347 CCOC(=O)c1cccc(Nc2nc(nc3ccccc23)C(=O)OCC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P18 compound treatment 150200.0 6010.0 0.41 153080.0 9000.0 0.67 0.7633 0.9721 3652844 Neuro1_000348 Cc1ccc(C)c(Nc2nc(NCCO)c3ccccc3n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P19 compound treatment 151160.0 6970.0 0.47 157520.0 13400.0 1.0 1.0432 0.942 1361396 Neuro1_000349 C(N1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P20 compound treatment 155640.0 11400.0 0.78 152640.0 8560.0 0.64 1.0024 0.9949 3652845 Neuro1_000350 COc1ccc(Nc2nc(NCC3CCCO3)c4ccccc4n2)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P21 compound treatment 153560.0 9370.0 0.64 155280.0 11200.0 0.83 1.041 0.9913 1450719 Neuro1_000351 CCCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P22 compound treatment 153920.0 9730.0 0.66 154600.0 10500.0 0.78 1.0226 0.9966 3652846 Neuro1_000352 CN(C)CCCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P23 mock treatment 147320.0 3130.0 0.21 145800.0 1720.0 0.13 0.2413 0.9703 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2435 P24 mock treatment 138920.0 -5270.0 -0.36 141400.0 -2680.0 -0.2 -0.3952 -0.9613 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A01 compound treatment 143960.0 -293.0 -0.02 142240.0 383.0 0.03 0.006 0.1735 3652847 Neuro1_000353 COc1ccc(cc1OC)/C(=N/Nc2nc(nc3ccccc23)c4cccnc4)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A02 compound treatment 152320.0 8070.0 0.55 150880.0 9020.0 0.67 0.8638 0.9951 1407528 Neuro1_000354 Oc1ccccc1c2nc(N3CCN(CC3)c4ccccc4)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A03 compound treatment 50640.0 -93600.0 -6.38 48640.0 -93200.0 -6.94 -9.4187 -0.9991 3652849 Neuro1_000355 Brc1ccc(cc1)c2nc(N/N=C/c3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A04 compound treatment 147960.0 3710.0 0.25 149000.0 7140.0 0.53 0.5546 0.9422 3652851 Neuro1_000356 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A05 compound treatment 157960.0 13700.0 0.93 154920.0 13100.0 0.97 1.3483 0.9998 3652853 Neuro1_000357 Cc1cc(C)n(n1)c2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A06 compound treatment 136880.0 -7370.0 -0.5 134880.0 -6980.0 -0.52 -0.7226 -0.9999 3652854 Neuro1_000358 Cc1ccc(cc1)c2nc(N/N=C/c3ccccc3[N+](=O)[O-])c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A07 compound treatment 152800.0 8550.0 0.58 148680.0 6820.0 0.51 0.7711 0.9976 1558498 Neuro1_000359 COC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A08 compound treatment 153040.0 8790.0 0.6 153280.0 11400.0 0.85 1.0248 0.9853 3652856 Neuro1_000360 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(I)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A09 compound treatment 144320.0 67.5 0.0 146320.0 4460.0 0.33 0.2381 0.7168 1168208 Neuro1_000361 CC(C)Nc1nc(nc2ccccc12)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A10 compound treatment 129520.0 -14700.0 -1.0 123000.0 -18900.0 -1.4 -1.7027 -0.9865 1935975 Neuro1_000362 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A11 compound treatment 144720.0 468.0 0.03 138480.0 -3380.0 -0.25 -0.1552 -0.6125 1506528 Neuro1_000363 Clc1ccc(cc1Cl)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A12 compound treatment 167480.0 23200.0 1.58 173880.0 32000.0 2.38 2.805 0.9803 1321517 Neuro1_000364 Clc1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A13 compound treatment 144200.0 -52.5 0.0 145920.0 4060.0 0.3 0.2113 0.6987 1653294 Neuro1_000365 Clc1ccccc1c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A14 compound treatment 156200.0 11900.0 0.81 151840.0 9980.0 0.74 1.1013 0.9989 1226926 Neuro1_000366 OC(=O)CCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A15 compound treatment 183480.0 39200.0 2.67 181920.0 40100.0 2.98 3.9995 0.9985 1318548 Neuro1_000367 COc1ccc(Nc2nc(nc3ccccc23)c4ccccc4O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A16 compound treatment 143080.0 -1170.0 -0.08 139520.0 -2340.0 -0.17 -0.1795 -0.9378 1974909 Neuro1_000368 COCCN(CCOC)c1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A17 compound treatment 143160.0 -1090.0 -0.07 145120.0 3260.0 0.24 0.119 0.4687 1706867 Neuro1_000369 CC1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A18 compound treatment 152080.0 7830.0 0.53 151560.0 9700.0 0.72 0.888 0.9889 3652858 Neuro1_000370 Fc1ccc(Nc2nc(/C=C/c3ccccc3)nc4ccccc24)cc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A19 compound treatment 151760.0 7510.0 0.51 147120.0 5260.0 0.39 0.6389 0.9913 3652860 Neuro1_000371 OC(=O)CCCCCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A20 compound treatment 156680.0 12400.0 0.85 161720.0 19900.0 1.48 1.6444 0.9651 3652861 Neuro1_000372 C1CCC(CC1)Nc2nc(/C=C/c3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A21 compound treatment 127160.0 -17100.0 -1.17 130720.0 -11100.0 -0.83 -1.4101 -0.9861 1917968 Neuro1_000373 CCN(CC)CCCC(C)Nc1nc(/C=C/c2ccc(Br)cc2)nc3cc(Cl)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A22 compound treatment 141000.0 -3250.0 -0.22 139720.0 -2140.0 -0.16 -0.2693 -0.9867 1415981 Neuro1_000374 CCN1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A23 mock treatment 141320.0 -2930.0 -0.2 139840.0 -2020.0 -0.15 -0.2475 -0.99 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 A24 mock treatment 140400.0 -3850.0 -0.26 138080.0 -3780.0 -0.28 -0.3845 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B01 compound treatment 136560.0 -7690.0 -0.52 134240.0 -7620.0 -0.57 -0.7717 -0.9992 1974596 Neuro1_000375 [O-][N+](=O)c1ccc(cc1)c2nc(NCCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B02 compound treatment 167160.0 22900.0 1.56 174400.0 32500.0 2.42 2.817 0.9775 1532266 Neuro1_000376 Oc1ccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B03 compound treatment 183160.0 38900.0 2.65 187520.0 45700.0 3.4 4.2788 0.9925 1864017 Neuro1_000377 [O-][N+](=O)c1ccc(cc1)c2nc(Nc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B04 compound treatment 141680.0 -2570.0 -0.18 138960.0 -2900.0 -0.22 -0.2765 -0.9947 1337812 Neuro1_000378 OC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B05 compound treatment 143560.0 -693.0 -0.05 146360.0 4500.0 0.34 0.2036 0.6015 1974637 Neuro1_000379 COCCN(CCOC)c1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B06 compound treatment 189960.0 45700.0 3.12 222000.0 80100.0 5.96 6.4212 0.9542 1606595 Neuro1_000380 Cc1ccc(C)c(Nc2nc(NCc3ccco3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B07 compound treatment 178360.0 34100.0 2.33 180840.0 39000.0 2.9 3.6958 0.994 1864021 Neuro1_000381 Cc1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B08 compound treatment 174640.0 30400.0 2.07 174360.0 32500.0 2.42 3.1755 0.997 1472713 Neuro1_000382 Cc1cccc(c1)c2nc(Nc3ccc(cc3)N4CCOCC4)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B09 compound treatment 245480.0 101000.0 6.9 218160.0 76300.0 5.68 8.8956 0.9953 1628280 Neuro1_000383 Clc1ccc(Nc2nc(NCc3ccco3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B10 compound treatment 150200.0 5950.0 0.41 155240.0 13400.0 1.0 0.991 0.9215 1326862 Neuro1_000384 Cc1ccccc1C(=O)Oc2cccc(Nc3ncnc4ccccc34)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B11 compound treatment 151200.0 6950.0 0.47 143320.0 1460.0 0.11 0.4119 0.8475 1864058 Neuro1_000385 CCN(CC)c1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B12 compound treatment 148920.0 4670.0 0.32 140280.0 -1580.0 -0.12 0.142 0.4186 1482064 Neuro1_000386 Cc1ccc(cc1)c2nc(NCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B13 compound treatment 162080.0 17800.0 1.22 159760.0 17900.0 1.33 1.8016 0.9989 1418455 Neuro1_000387 Clc1ccc(c(Cl)c1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B14 compound treatment 180040.0 35800.0 2.44 171080.0 29200.0 2.17 3.2632 0.9984 3652863 Neuro1_000388 [O-][N+](=O)c1ccc(cc1)C(=O)Oc2cccc(Nc3ncnc4ccccc34)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B15 compound treatment 144640.0 388.0 0.03 140880.0 -978.0 -0.07 -0.0328 -0.4233 1974602 Neuro1_000389 COCCN(CCOC)c1nc(nc2ccccc12)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B16 compound treatment 177920.0 33700.0 2.3 178600.0 36700.0 2.73 3.5567 0.9962 1348023 Neuro1_000390 Brc1ccc2ncnc(Nc3ccc(cc3)N4CCCCC4)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B17 compound treatment 143720.0 -533.0 -0.04 138280.0 -3580.0 -0.27 -0.2139 -0.7962 1864057 Neuro1_000391 OCCNc1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B18 compound treatment 197200.0 52900.0 3.61 194360.0 52500.0 3.91 5.3156 0.9992 1384325 Neuro1_000392 Oc1ccccc1c2nc(Nc3ccccc3F)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B19 compound treatment 157800.0 13500.0 0.92 163800.0 21900.0 1.63 1.8079 0.9636 1223663 Neuro1_000393 Clc1ccccc1c2nc(Nc3ccc4OCCOc4c3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B20 compound treatment 157960.0 13700.0 0.93 157520.0 15700.0 1.17 1.4851 0.994 1123336 Neuro1_000394 Cc1cc(Cl)ccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B21 compound treatment 156280.0 12000.0 0.82 168840.0 27000.0 2.01 1.9999 0.9219 1238844 Neuro1_000395 Cc1ccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B22 compound treatment 142800.0 -1450.0 -0.1 139880.0 -1980.0 -0.15 -0.1741 -0.9814 1561925 Neuro1_000396 CC1CCCN(C1)c2nc(nc3ccccc23)c4ccccc4F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B23 mock treatment 138560.0 -5690.0 -0.39 132560.0 -9300.0 -0.69 -0.7637 -0.9626 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 B24 mock treatment 136840.0 -7410.0 -0.51 134480.0 -7380.0 -0.55 -0.7456 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C01 compound treatment 82240.0 -62000.0 -4.23 68720.0 -73100.0 -5.44 -6.8386 -0.9922 3652864 Neuro1_000397 N(/N=C/c1cccnc1)c2nc(nc3ccccc23)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C02 compound treatment 149640.0 5390.0 0.37 151440.0 9580.0 0.71 0.764 0.9524 3652866 Neuro1_000398 Oc1ccccc1c2nc(N/N=C/c3ccccc3Cl)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C03 compound treatment 119200.0 -25100.0 -1.71 119880.0 -22000.0 -1.64 -2.3644 -0.9998 3652868 Neuro1_000399 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(Br)cc3)/c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C04 compound treatment 30400.0 -114000.0 -7.76 27200.0 -115000.0 -8.53 -11.5228 -0.9989 2115809 Neuro1_000400 Cc1ccc(cc1)c2nc(N/N=C/c3ccc(O)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C05 compound treatment 146960.0 2710.0 0.18 142600.0 743.0 0.06 0.1696 0.8802 1691530 Neuro1_000401 CC1CCN(CC1)c2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C06 compound treatment 158600.0 14300.0 0.98 152200.0 10300.0 0.77 1.236 0.993 1935368 Neuro1_000402 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(N)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C07 compound treatment 151200.0 6950.0 0.47 147400.0 5540.0 0.41 0.6266 0.9976 1673689 Neuro1_000403 Brc1ccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C08 compound treatment 99400.0 -44900.0 -3.06 91800.0 -50100.0 -3.73 -4.7967 -0.9952 1935618 Neuro1_000404 Cc1ccc(cc1)c2nc(N/N=C/c3cccc(F)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C09 compound treatment 157520.0 13300.0 0.9 161160.0 19300.0 1.44 1.6555 0.9751 3652870 Neuro1_000405 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(Br)cc3)/c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C10 compound treatment 158880.0 14600.0 1.0 159480.0 17600.0 1.31 1.6326 0.9909 3652872 Neuro1_000406 COc1ccccc1/C=N/Nc2nc(nc3ccccc23)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C11 compound treatment 145560.0 1310.0 0.09 145560.0 3700.0 0.28 0.2579 0.8904 1460559 Neuro1_000407 Clc1ccc(cc1)c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C12 compound treatment 180120.0 35900.0 2.45 178840.0 37000.0 2.75 3.6754 0.9983 1438608 Neuro1_000408 Brc1ccc2ncnc(Nc3cccc4ccccc34)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C13 compound treatment 153760.0 9510.0 0.65 150440.0 8580.0 0.64 0.91 1.0 1174599 Neuro1_000409 CCN(CC)c1nc(nc2ccccc12)c3ccccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C14 compound treatment 233960.0 89700.0 6.12 239880.0 98000.0 7.3 9.4834 0.9962 1677801 Neuro1_000410 CN(Cc1ccccc1)c2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C15 compound treatment 225520.0 81300.0 5.54 233320.0 91500.0 6.81 8.7312 0.9948 1492426 Neuro1_000411 CC(Nc1nc(nc2ccccc12)c3ccccc3O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C16 compound treatment 147840.0 3590.0 0.24 147840.0 5980.0 0.45 0.4878 0.9602 1324336 Neuro1_000412 CN(C)CCNc1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C17 compound treatment 157520.0 13300.0 0.9 159080.0 17200.0 1.28 1.546 0.9854 1335943 Neuro1_000413 Cc1ccc2ncnc(Nc3ccc(I)cc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C18 compound treatment 151800.0 7550.0 0.51 148240.0 6380.0 0.48 0.6997 0.9992 3652874 Neuro1_000414 Fc1ccc(Nc2nc(/C=C/c3ccccc3)nc4ccccc24)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C19 compound treatment 160960.0 16700.0 1.14 161720.0 19900.0 1.48 1.8508 0.9917 1254761 Neuro1_000415 COc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C20 compound treatment 148200.0 3950.0 0.27 149840.0 7980.0 0.59 0.6104 0.9359 3652876 Neuro1_000416 CC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(cc4)C(C)(C)C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C21 compound treatment 152600.0 8350.0 0.57 150640.0 8780.0 0.65 0.8646 0.9976 1915748 Neuro1_000417 CCN(CC)CCCC(C)Nc1nc(C)nc2cc(Cl)ccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C22 compound treatment 154360.0 10100.0 0.69 157760.0 15900.0 1.18 1.3242 0.9669 1864052 Neuro1_000418 [O-][N+](=O)c1ccc(cc1)c2nc(NCC3CCCO3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C23 mock treatment 136040.0 -8210.0 -0.56 131520.0 -10300.0 -0.77 -0.94 -0.9878 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 C24 mock treatment 141560.0 -2690.0 -0.18 133840.0 -8020.0 -0.6 -0.5517 -0.8838 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D01 compound treatment 159800.0 15500.0 1.06 155080.0 13200.0 0.98 1.4454 0.9993 1864024 Neuro1_000419 [O-][N+](=O)c1ccc(cc1)c2nc(Nc3ccc(cc3)N4CCOCC4)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D02 compound treatment 145920.0 1670.0 0.11 149320.0 7460.0 0.56 0.4731 0.8345 1736515 Neuro1_000420 C(Nc1nc(nc2ccccc12)N3CCOCC3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D03 compound treatment 141320.0 -2930.0 -0.2 144360.0 2500.0 0.19 -0.0097 -0.0354 1403547 Neuro1_000421 Clc1ccc(cc1)c2nc(N(CC=C)CC=C)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D04 compound treatment 202920.0 58700.0 4.0 216000.0 74100.0 5.52 6.7302 0.9875 3652877 Neuro1_000422 Ic1ccc(Nc2nc(nc3ccccc23)c4cccnc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D05 compound treatment 153000.0 8750.0 0.6 154080.0 12200.0 0.91 1.0649 0.979 3652878 Neuro1_000423 COCCNc1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D06 compound treatment 162160.0 17900.0 1.22 159280.0 17400.0 1.3 1.7802 0.9995 1382426 Neuro1_000424 C(Nc1nc(nc2ccccc12)N3CCN(CC3)c4ccccc4)c5ccco5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D07 compound treatment 159040.0 14800.0 1.01 171880.0 30000.0 2.23 2.2929 0.9353 3652879 Neuro1_000425 [O-][N+](=O)c1ccc(cc1)c2nc(Nc3cccc(c3)C(F)(F)F)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D08 compound treatment 154720.0 10500.0 0.71 155400.0 13500.0 1.01 1.2173 0.9857 1875932 Neuro1_000426 Cc1ccc(cc1)c2nc(Nc3cccc(c3)[N+](=O)[O-])c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D09 compound treatment 190800.0 46500.0 3.17 185720.0 43900.0 3.26 4.5524 0.9999 3652880 Neuro1_000427 CC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D10 compound treatment 160720.0 16500.0 1.12 170560.0 28700.0 2.14 2.3044 0.9549 3652881 Neuro1_000428 CC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(C)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D11 compound treatment 150320.0 6070.0 0.41 146160.0 4300.0 0.32 0.5189 0.992 1864075 Neuro1_000429 CCN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D12 compound treatment 148040.0 3790.0 0.26 144440.0 2580.0 0.19 0.3185 0.9894 1698173 Neuro1_000430 Cc1cccc(c1)c2nc(Nc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D13 compound treatment 150360.0 6110.0 0.42 154800.0 12900.0 0.96 0.9756 0.9296 1864064 Neuro1_000431 CN(Cc1ccccc1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D14 compound treatment 149160.0 4910.0 0.33 150560.0 8700.0 0.65 0.6946 0.9528 1722222 Neuro1_000432 Cc1ccc(cc1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D15 compound treatment 155760.0 11500.0 0.78 157480.0 15600.0 1.16 1.3769 0.9817 1864048 Neuro1_000433 CC(Nc1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-])c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D16 compound treatment 159880.0 15600.0 1.07 158280.0 16400.0 1.22 1.6177 0.9977 1346578 Neuro1_000434 CC(C)Oc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D17 compound treatment 149400.0 5150.0 0.35 144960.0 3100.0 0.23 0.4114 0.9794 1864074 Neuro1_000435 CN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D18 compound treatment 165120.0 20900.0 1.42 161760.0 19900.0 1.48 2.0534 0.9998 3652882 Neuro1_000436 CCCCOc1ccccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D19 compound treatment 156680.0 12400.0 0.85 147920.0 6060.0 0.45 0.9182 0.9565 1698013 Neuro1_000437 COC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D20 compound treatment 152640.0 8390.0 0.57 156880.0 15000.0 1.12 1.1949 0.9515 3652883 Neuro1_000438 CCCCOc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D21 compound treatment 162480.0 18200.0 1.24 163760.0 21900.0 1.63 2.0314 0.991 3652884 Neuro1_000439 CC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D22 compound treatment 144640.0 388.0 0.03 172400.0 30500.0 2.27 1.6261 0.7153 3652885 Neuro1_000440 CCOc1ccc(Nc2nc(N3CCN(C)CC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D23 mock treatment 139440.0 -4810.0 -0.33 137080.0 -4780.0 -0.36 -0.4834 -0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 D24 mock treatment 140840.0 -3410.0 -0.23 136880.0 -4980.0 -0.37 -0.4265 -0.9749 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E01 compound treatment 148360.0 4110.0 0.28 249600.0 108000.0 8.02 5.8683 0.7314 1476399 Neuro1_000441 COc1ccc(Nc2nc(nc3ccccc23)c4cccnc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E02 compound treatment 162760.0 18500.0 1.26 160120.0 18300.0 1.36 1.8533 0.9993 1934925 Neuro1_000442 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4cccc(c4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E03 compound treatment 151840.0 7590.0 0.52 150000.0 8140.0 0.61 0.7943 0.9969 1331650 Neuro1_000443 Brc1ccc(cc1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E04 compound treatment 153520.0 9270.0 0.63 160440.0 18600.0 1.38 1.4247 0.937 3652886 Neuro1_000444 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(Cl)c(Cl)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E05 compound treatment 76840.0 -67400.0 -4.6 79160.0 -62700.0 -4.67 -6.5495 -1.0 3652888 Neuro1_000445 Oc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E06 compound treatment 152560.0 8310.0 0.57 147840.0 5980.0 0.45 0.7153 0.9929 3652890 Neuro1_000446 Cc1ccc(cc1)c2nc(Nc3cccc(F)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E07 compound treatment 158760.0 14500.0 0.99 164120.0 22300.0 1.66 1.871 0.9696 1651398 Neuro1_000447 Fc1ccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E08 compound treatment 71160.0 -73100.0 -4.98 78120.0 -63700.0 -4.74 -6.878 -0.9997 1935777 Neuro1_000448 Cc1ccc(cc1)c2nc(N/N=C/c3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E09 compound treatment 177360.0 33100.0 2.26 174160.0 32300.0 2.4 3.2961 0.9995 3652891 Neuro1_000449 NNc1nc(nc2ccccc12)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E10 compound treatment 178840.0 34600.0 2.36 179120.0 37300.0 2.77 3.6284 0.9967 1431459 Neuro1_000450 Clc1ccccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E11 compound treatment 156280.0 12000.0 0.82 153280.0 11400.0 0.85 1.181 0.9998 1523927 Neuro1_000451 Clc1ccccc1c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E12 compound treatment 192680.0 48400.0 3.3 194880.0 53000.0 3.95 5.1251 0.9961 1941178 Neuro1_000452 [O-][N+](=O)c1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E13 compound treatment 166720.0 22500.0 1.53 164200.0 22300.0 1.66 2.259 0.9992 1565218 Neuro1_000453 Clc1ccccc1c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E14 compound treatment 163080.0 18800.0 1.28 162960.0 21100.0 1.57 2.0182 0.995 1305930 Neuro1_000454 OCC(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E15 compound treatment 168880.0 24600.0 1.68 166840.0 25000.0 1.86 2.502 0.9987 1345839 Neuro1_000455 Oc1ccccc1c2nc(N3CCCCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E16 compound treatment 152120.0 7870.0 0.54 150840.0 8980.0 0.67 0.852 0.994 1137633 Neuro1_000456 CCN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E17 compound treatment 171040.0 26800.0 1.83 173080.0 31200.0 2.32 2.9346 0.9929 1164201 Neuro1_000457 Clc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E18 compound treatment 178320.0 34100.0 2.32 183400.0 41500.0 3.09 3.8286 0.9901 3652892 Neuro1_000458 C1CCCN(CC1)c2nc(/C=C/c3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E19 compound treatment 175360.0 31100.0 2.12 179400.0 37500.0 2.79 3.4754 0.9907 1711587 Neuro1_000459 Cc1c(Cl)cccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E20 compound treatment 152800.0 8550.0 0.58 154160.0 12300.0 0.92 1.0595 0.9762 3652894 Neuro1_000460 CCC1CCCCN1c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E21 compound treatment 201520.0 57300.0 3.9 205520.0 63700.0 4.74 6.1112 0.9954 1358947 Neuro1_000461 Cc1ccc(Nc2nc(nc3ccccc23)c4ccccc4O)c(C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E22 compound treatment 152000.0 7750.0 0.53 149520.0 7660.0 0.57 0.7768 0.9993 1316921 Neuro1_000462 CC(C)(C)c1ccc(cc1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E23 mock treatment 146240.0 1990.0 0.14 140880.0 -978.0 -0.07 0.0444 0.2885 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 E24 mock treatment 141440.0 -2810.0 -0.19 146200.0 4340.0 0.32 0.093 0.2473 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F01 compound treatment 158560.0 14300.0 0.98 159200.0 17300.0 1.29 1.6024 0.9905 1667500 Neuro1_000463 COc1ccc(Cl)cc1Nc2nc(nc3ccccc23)c4ccc(Cl)cc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F02 compound treatment 166400.0 22100.0 1.51 165440.0 23600.0 1.76 2.3088 0.9972 1461219 Neuro1_000464 Fc1ccccc1Nc2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F03 compound treatment 160520.0 16300.0 1.11 154000.0 12100.0 0.9 1.4233 0.9948 1864063 Neuro1_000465 CN(C1CCCCC1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F04 compound treatment 174120.0 29900.0 2.04 164240.0 22400.0 1.67 2.6178 0.995 1609272 Neuro1_000466 COc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F05 compound treatment 153960.0 9710.0 0.66 152360.0 10500.0 0.78 1.0207 0.9966 1731031 Neuro1_000467 C(Cc1ccccc1)Nc2nc(nc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F06 compound treatment 169920.0 25700.0 1.75 165000.0 23100.0 1.72 2.4553 1.0 1165915 Neuro1_000468 CCOC(=O)c1cccc(Nc2ncnc3ccccc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F07 compound treatment 173600.0 29300.0 2.0 163600.0 21700.0 1.62 2.5591 0.9945 1654363 Neuro1_000469 Cc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F08 compound treatment 162520.0 18300.0 1.25 158880.0 17000.0 1.27 1.7765 1.0 1875933 Neuro1_000470 Cc1cccc(c1)c2nc(Nc3cccc(c3)[N+](=O)[O-])c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F09 compound treatment 270000.0 126000.0 8.57 263400.0 122000.0 9.05 12.4586 0.9996 1692238 Neuro1_000471 CCOc1ccc(Nc2nc(NCc3ccccc3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F10 compound treatment 146880.0 2630.0 0.18 148960.0 7100.0 0.53 0.5005 0.8966 1663781 Neuro1_000472 CC1CN(CC(C)O1)c2nc(nc3ccccc23)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F11 compound treatment 162440.0 18200.0 1.24 175240.0 33400.0 2.48 2.6336 0.9484 1864073 Neuro1_000473 CC1CN(CC(C)O1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F12 compound treatment 153680.0 9430.0 0.64 154360.0 12500.0 0.93 1.1125 0.9837 1197549 Neuro1_000474 Cc1cccc(c1)c2nc(NCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F13 compound treatment 158080.0 13800.0 0.94 158200.0 16300.0 1.22 1.5267 0.9921 1864050 Neuro1_000475 [O-][N+](=O)c1ccc(cc1)c2nc(NCCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F14 compound treatment 175400.0 31100.0 2.12 171280.0 29400.0 2.19 3.05 0.9999 1123686 Neuro1_000476 O=C(Oc1cccc(Nc2ncnc3ccccc23)c1)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F15 compound treatment 166920.0 22700.0 1.55 172360.0 30500.0 2.27 2.698 0.9824 1863996 Neuro1_000477 [O-][N+](=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F16 compound treatment 153600.0 9350.0 0.64 153240.0 11400.0 0.85 1.0497 0.9902 1983310 Neuro1_000478 C(CNc1ncnc2ccccc12)CNc3ncnc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F17 compound treatment 167600.0 23300.0 1.59 159400.0 17500.0 1.31 2.0488 0.9952 1974998 Neuro1_000479 COCCNc1nc(nc2ccccc12)c3ccc(cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F18 compound treatment 157360.0 13100.0 0.89 164960.0 23100.0 1.72 1.8477 0.9535 1209891 Neuro1_000480 CN(C1CCN(C)CC1)c2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F19 compound treatment 177000.0 32700.0 2.23 176200.0 34300.0 2.56 3.3861 0.9977 1420188 Neuro1_000481 Cc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F20 compound treatment 165000.0 20700.0 1.41 163080.0 21200.0 1.58 2.1171 0.9985 1637647 Neuro1_000482 Cc1ccc(Nc2ncnc3ccc(Br)cc23)cc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F21 compound treatment 157560.0 13300.0 0.91 152920.0 11100.0 0.82 1.2237 0.9988 1665278 Neuro1_000483 Clc1ccccc1c2nc(Nc3ccc(I)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F22 compound treatment 156960.0 12700.0 0.87 146960.0 5100.0 0.38 0.8811 0.9315 3652895 Neuro1_000484 CC(=C)CN1CCN(CC1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F23 mock treatment 152200.0 7950.0 0.54 141000.0 -858.0 -0.06 0.338 0.6195 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 F24 mock treatment 139040.0 -5210.0 -0.36 146120.0 4260.0 0.32 -0.027 -0.0566 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G01 compound treatment 161840.0 17600.0 1.2 161480.0 19600.0 1.46 1.8806 0.9952 3652896 Neuro1_000485 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4cccnc4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G02 compound treatment 17960.0 -126000.0 -8.61 16200.0 -126000.0 -9.35 -12.7014 -0.9991 1935032 Neuro1_000486 Cc1ccc(cc1)c2nc(N/N=C/c3ccncc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G03 compound treatment 164840.0 20600.0 1.4 159560.0 17700.0 1.32 1.9241 0.9995 1580403 Neuro1_000487 OCCNc1nc(nc2ccccc12)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G04 compound treatment 161280.0 17000.0 1.16 164640.0 22800.0 1.7 2.0199 0.9829 1487118 Neuro1_000488 Cc1cc(C)n(n1)c2nc(nc3ccccc23)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G05 compound treatment 47880.0 -96400.0 -6.57 52560.0 -89300.0 -6.65 -9.3455 -1.0 3652898 Neuro1_000489 COc1cc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G06 compound treatment 167040.0 22800.0 1.55 160920.0 19100.0 1.42 2.1018 0.999 1935415 Neuro1_000490 CN(C)c1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G07 compound treatment 164760.0 20500.0 1.4 166400.0 24500.0 1.83 2.2802 0.9913 1639473 Neuro1_000491 Clc1cccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G08 compound treatment 74200.0 -70100.0 -4.78 79320.0 -62500.0 -4.65 -6.6683 -0.9999 1935724 Neuro1_000492 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G09 compound treatment 161640.0 17400.0 1.19 158360.0 16500.0 1.23 1.7067 0.9998 1626806 Neuro1_000493 CCN(CC)c1nc(nc2ccccc12)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G10 compound treatment 156840.0 12600.0 0.86 155400.0 13500.0 1.01 1.3195 0.9968 1617513 Neuro1_000494 CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G11 compound treatment 161800.0 17500.0 1.2 160160.0 18300.0 1.36 1.8092 0.9979 1726213 Neuro1_000495 Clc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G12 compound treatment 175320.0 31100.0 2.12 170040.0 28200.0 2.1 2.9809 1.0 1171304 Neuro1_000496 CCOC(=O)c1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G13 compound treatment 177360.0 33100.0 2.26 176000.0 34100.0 2.54 3.3929 0.9983 1733773 Neuro1_000497 COc1ccc(Nc2nc(nc3ccccc23)c4ccncc4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G14 compound treatment 188040.0 43800.0 2.99 189000.0 47100.0 3.51 4.5919 0.9968 1263689 Neuro1_000498 Brc1ccc2ncnc(NCc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G15 compound treatment 165160.0 20900.0 1.43 164160.0 22300.0 1.66 2.1816 0.9971 1925712 Neuro1_000499 Brc1ccc(cc1)c2nc(NCCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G16 compound treatment 161400.0 17100.0 1.17 164440.0 22600.0 1.68 2.0151 0.9843 1233473 Neuro1_000500 Clc1ccc(cc1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G17 compound treatment 159440.0 15200.0 1.04 160640.0 18800.0 1.4 1.7206 0.9891 1203567 Neuro1_000501 CC(C)CC(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G18 compound treatment 166160.0 21900.0 1.49 165440.0 23600.0 1.76 2.2972 0.9968 3652900 Neuro1_000502 CC1CCN(CC1)c2nc(/C=C/c3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G19 compound treatment 158320.0 14100.0 0.96 158720.0 16900.0 1.26 1.5656 0.9912 1941232 Neuro1_000503 FC(F)(F)c1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G20 compound treatment 154400.0 10100.0 0.69 152200.0 10300.0 0.77 1.0335 0.9986 1558452 Neuro1_000504 Clc1ccc(c(Cl)c1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G21 compound treatment 179440.0 35200.0 2.4 195200.0 53300.0 3.97 4.5036 0.9709 1278774 Neuro1_000505 Oc1ccccc1c2nc(Nc3cccc(F)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G22 compound treatment 163240.0 19000.0 1.29 165520.0 23700.0 1.76 2.1607 0.9885 1864051 Neuro1_000506 [O-][N+](=O)c1ccc(cc1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G23 mock treatment 149720.0 5470.0 0.37 146400.0 4540.0 0.34 0.5026 0.9988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 G24 mock treatment 148200.0 3950.0 0.27 146440.0 4580.0 0.34 0.4315 0.9931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H01 compound treatment 192040.0 47800.0 3.26 181440.0 39600.0 2.95 4.3869 0.9987 3652902 Neuro1_000507 CC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H02 compound treatment 182400.0 38100.0 2.6 173880.0 32000.0 2.38 3.5243 0.999 1413336 Neuro1_000508 Clc1ccccc1Nc2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H03 compound treatment 152280.0 8030.0 0.55 151800.0 9940.0 0.74 0.9102 0.989 1155824 Neuro1_000509 CC1CN(CC(C)O1)c2nc(nc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H04 compound treatment 151440.0 7190.0 0.49 152840.0 11000.0 0.82 0.9245 0.9701 1392884 Neuro1_000510 CN1CCN(CC1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H05 compound treatment 189760.0 45500.0 3.1 178000.0 36100.0 2.69 4.0959 0.9975 1864023 Neuro1_000511 Cc1cc(Cl)ccc1Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H06 compound treatment 173240.0 29000.0 1.98 168120.0 26300.0 1.95 2.7796 1.0 1864032 Neuro1_000512 COc1ccccc1Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H07 compound treatment 179920.0 35700.0 2.43 172760.0 30900.0 2.3 3.3458 0.9996 1411828 Neuro1_000513 Clc1ccc(cc1)c2nc(Nc3ccc4OCCOc4c3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H08 compound treatment 159680.0 15400.0 1.05 158640.0 16800.0 1.25 1.627 0.9963 1556370 Neuro1_000514 CN(C1CCN(C)CC1)c2nc(nc3ccccc23)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H09 compound treatment 295560.0 151000.0 10.32 273680.0 132000.0 9.81 14.2318 0.9997 1224552 Neuro1_000515 Cc1cccc(Nc2nc(NCc3ccco3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H10 compound treatment 151600.0 7350.0 0.5 149960.0 8100.0 0.6 0.7806 0.9957 3118214 Neuro1_000516 Cc1cccc(c1)c2nc(NCCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H11 compound treatment 154720.0 10500.0 0.71 157160.0 15300.0 1.14 1.31 0.9746 1864067 Neuro1_000517 [O-][N+](=O)c1ccc(cc1)c2nc(N3CCCCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H12 compound treatment 160360.0 16100.0 1.1 149840.0 7980.0 0.59 1.1966 0.9584 1166424 Neuro1_000518 Cc1cccc(c1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H13 compound treatment 173600.0 29300.0 2.0 167760.0 25900.0 1.93 2.778 0.9998 1864035 Neuro1_000519 CCOc1ccccc1Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H14 compound treatment 175680.0 31400.0 2.14 176800.0 34900.0 2.6 3.354 0.9954 1440212 Neuro1_000520 Clc1ccccc1C(=O)Oc2cccc(Nc3ncnc4ccccc34)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H15 compound treatment 166600.0 22300.0 1.52 161480.0 19600.0 1.46 2.11 0.9998 1864072 Neuro1_000521 [O-][N+](=O)c1ccc(cc1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H16 compound treatment 159520.0 15300.0 1.04 157960.0 16100.0 1.2 1.5835 0.9975 1317715 Neuro1_000522 Cc1ccccc1Nc2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H17 compound treatment 150200.0 5950.0 0.41 145520.0 3660.0 0.27 0.4795 0.9813 1718575 Neuro1_000523 CC(C)(C)c1ccc(cc1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H18 compound treatment 169240.0 25000.0 1.7 166640.0 24800.0 1.84 2.5089 0.9992 1423155 Neuro1_000524 CCCOC(=O)c1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H19 compound treatment 174000.0 29700.0 2.03 167560.0 25700.0 1.91 2.7867 0.9996 3652903 Neuro1_000525 CCC(CC)c1nc(Nc2cccc(c2)C(=O)C)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H20 compound treatment 193240.0 49000.0 3.34 178320.0 36500.0 2.71 4.2805 0.9947 3652904 Neuro1_000526 Oc1ccccc1c2nc(Nc3cccc(Cl)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H21 compound treatment 160760.0 16500.0 1.13 157520.0 15700.0 1.17 1.6201 0.9998 1520301 Neuro1_000527 CCCOC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H22 compound treatment 145720.0 1470.0 0.1 149800.0 7940.0 0.59 0.4887 0.8152 3652905 Neuro1_000528 Cc1ccc(C)c(Nc2nc(NCC3CCCO3)c4ccccc4n2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H23 mock treatment 147320.0 3070.0 0.21 146560.0 4700.0 0.35 0.3954 0.9697 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 H24 mock treatment 149120.0 4870.0 0.33 141720.0 -138.0 -0.01 0.2274 0.685 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I01 compound treatment 177960.0 33700.0 2.3 169480.0 27600.0 2.06 3.0787 0.9985 1333707 Neuro1_000529 CCN1CCN(CC1)c2ccc(Nc3nc(C)nc4cc(Cl)ccc34)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I02 compound treatment 151400.0 7150.0 0.49 158080.0 16200.0 1.21 1.1983 0.9204 1304777 Neuro1_000530 COc1ccc(Nc2nc(nc3ccccc23)c4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I03 compound treatment 171880.0 27600.0 1.88 188160.0 46300.0 3.45 3.7687 0.9596 3652906 Neuro1_000531 Clc1ccccc1Nc2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I04 compound treatment 155040.0 10800.0 0.74 158520.0 16700.0 1.24 1.397 0.9689 3652907 Neuro1_000532 CCCCCOc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I05 compound treatment 114160.0 -30100.0 -2.05 109120.0 -32700.0 -2.44 -3.1736 -0.9963 3652909 Neuro1_000533 COc1cccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I06 compound treatment 145840.0 1590.0 0.11 151360.0 9500.0 0.71 0.5766 0.8059 1935362 Neuro1_000534 Cc1ccc(cc1)c2nc(N/N=C/c3cccc(c3)[N+](=O)[O-])c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I07 compound treatment 154200.0 9950.0 0.68 150560.0 8700.0 0.65 0.9375 0.9997 1724591 Neuro1_000535 Brc1ccc(cc1)c2nc(Nc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I08 compound treatment 80560.0 -63700.0 -4.34 66840.0 -75000.0 -5.58 -7.0185 -0.9923 1935729 Neuro1_000536 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I09 compound treatment 92280.0 -52000.0 -3.54 98120.0 -43700.0 -3.26 -4.8073 -0.9991 3652911 Neuro1_000537 Fc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I10 compound treatment 171720.0 27500.0 1.87 169440.0 27600.0 2.05 2.7758 0.9989 1473263 Neuro1_000538 Cc1ccccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I11 compound treatment 158560.0 14300.0 0.98 156520.0 14700.0 1.09 1.4614 0.9984 1589310 Neuro1_000539 CN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I12 compound treatment 174000.0 29700.0 2.03 168960.0 27100.0 2.02 2.8604 1.0 1411301 Neuro1_000540 Cc1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I13 compound treatment 168280.0 24000.0 1.64 165680.0 23800.0 1.77 2.4121 0.9992 1928846 Neuro1_000541 FC(F)(F)c1cccc(Nc2nc(nc3ccccc23)c4ccncc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I14 compound treatment 177320.0 33100.0 2.25 179680.0 37800.0 2.82 3.5846 0.9939 1560672 Neuro1_000542 COc1ccccc1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I15 compound treatment 212760.0 68500.0 4.67 212360.0 70500.0 5.25 7.013 0.9983 1553258 Neuro1_000543 CN1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I16 compound treatment 155200.0 10900.0 0.75 152280.0 10400.0 0.78 1.0763 0.9998 1219300 Neuro1_000544 CC1CN(CC(C)O1)c2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I17 compound treatment 168960.0 24700.0 1.68 165960.0 24100.0 1.79 2.4596 0.9995 1566980 Neuro1_000545 Cc1cccc(C)c1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I18 compound treatment 168480.0 24200.0 1.65 163720.0 21900.0 1.63 2.3185 1.0 3652913 Neuro1_000546 C1CN(CCO1)c2nc(/C=C/c3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I19 compound treatment 184800.0 40500.0 2.76 172960.0 31100.0 2.31 3.5916 0.9961 1715482 Neuro1_000547 COC(=O)c1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I20 compound treatment 170320.0 26100.0 1.78 166200.0 24300.0 1.81 2.5378 1.0 1864065 Neuro1_000548 [O-][N+](=O)c1ccc(cc1)c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I21 compound treatment 51680.0 -92600.0 -6.31 46960.0 -94900.0 -7.06 -9.457 -0.9984 3652915 Neuro1_000549 CCOc1ccc(Nc2nc(N)c3ccccc3n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I22 compound treatment 150440.0 6190.0 0.42 147000.0 5140.0 0.38 0.5689 0.9988 1864070 Neuro1_000550 CC1CCN(CC1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I23 mock treatment 144320.0 67.5 0.0 146000.0 4140.0 0.31 0.2213 0.7176 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 I24 mock treatment 145640.0 1390.0 0.09 140200.0 -1660.0 -0.12 -0.0203 -0.1309 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J01 compound treatment 151800.0 7550.0 0.51 152680.0 10800.0 0.81 0.9334 0.9766 3652916 Neuro1_000551 COCCCNc1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J02 compound treatment 155000.0 10700.0 0.73 153360.0 11500.0 0.86 1.1235 0.997 1610139 Neuro1_000552 C(Nc1nc(nc2ccccc12)N3CCN(Cc4ccccc4)CC3)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J03 compound treatment 183920.0 39700.0 2.7 187080.0 45200.0 3.37 4.2923 0.9941 1864038 Neuro1_000553 CN(C)c1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J04 compound treatment 166760.0 22500.0 1.53 164440.0 22600.0 1.68 2.2735 0.999 1691758 Neuro1_000554 Fc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J05 compound treatment 162720.0 18500.0 1.26 155120.0 13300.0 0.99 1.5883 0.9927 3652917 Neuro1_000555 OCCCNc1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J06 compound treatment 155160.0 10900.0 0.74 153360.0 11500.0 0.86 1.1312 0.9975 1347171 Neuro1_000556 Cc1ccc(cc1)c2nc(Nc3ccc(cc3)C(=O)O)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J07 compound treatment 166720.0 22500.0 1.53 168280.0 26400.0 1.97 2.4737 0.9924 1387715 Neuro1_000557 C(Nc1nc(nc2ccccc12)N3CCN(Cc4ccccc4)CC3)c5ccco5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J08 compound treatment 165600.0 21300.0 1.46 160000.0 18100.0 1.35 1.9839 0.9993 1259981 Neuro1_000558 Cc1ccc(cc1)c2nc(Nc3ccc(O)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J09 compound treatment 150640.0 6390.0 0.44 150560.0 8700.0 0.65 0.7659 0.9813 1864055 Neuro1_000559 CN(C)CCNc1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J10 compound treatment 161600.0 17300.0 1.18 162560.0 20700.0 1.54 1.9258 0.9915 1386535 Neuro1_000560 Cc1cccc(c1)c2nc(Nc3ccc(O)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J11 compound treatment 193480.0 49200.0 3.36 190960.0 49100.0 3.65 4.9573 0.9991 1864019 Neuro1_000561 Cc1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J12 compound treatment 164760.0 20500.0 1.4 165160.0 23300.0 1.73 2.215 0.9943 1252547 Neuro1_000562 Cc1ccc(cc1)c2nc(Nc3cccc(O)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J13 compound treatment 164560.0 20300.0 1.38 155640.0 13800.0 1.03 1.7043 0.9891 1864062 Neuro1_000563 [O-][N+](=O)c1ccc(cc1)c2nc(N(CC=C)CC=C)c3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J14 compound treatment 205120.0 60900.0 4.15 200040.0 58200.0 4.33 5.9963 0.9998 1517067 Neuro1_000564 Oc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J15 compound treatment 176880.0 32600.0 2.22 175400.0 33500.0 2.5 3.3382 0.9983 1864042 Neuro1_000565 OC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J16 compound treatment 251760.0 108000.0 7.33 252120.0 110000.0 8.21 10.9856 0.9984 1121498 Neuro1_000566 COc1ccc(Nc2nc(NCc3ccccc3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J17 compound treatment 162560.0 18300.0 1.25 160400.0 18500.0 1.38 1.8584 0.9987 1444843 Neuro1_000567 CC(C)(C)c1ccc(cc1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J18 compound treatment 184720.0 40500.0 2.76 187760.0 45900.0 3.42 4.3666 0.9944 1176544 Neuro1_000568 Oc1ccccc1c2nc(NCCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J19 compound treatment 171480.0 27200.0 1.86 165000.0 23100.0 1.72 2.5305 0.9993 1233327 Neuro1_000569 CCC(CC)c1nc(Nc2cccc(OC)c2)c3ccccc3n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J20 compound treatment 201480.0 57200.0 3.9 204920.0 63100.0 4.69 6.0777 0.9958 1274473 Neuro1_000570 Oc1ccccc1c2nc(Nc3ccc(Br)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J21 compound treatment 158000.0 13700.0 0.94 154880.0 13000.0 0.97 1.3481 0.9999 1193123 Neuro1_000571 COc1cccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J22 compound treatment 157720.0 13500.0 0.92 155360.0 13500.0 1.0 1.3599 0.999 1261607 Neuro1_000572 Fc1ccccc1c2nc(N3CCN(CC3)c4ccccc4)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J23 mock treatment 144160.0 -92.5 -0.01 143000.0 1140.0 0.09 0.0557 0.6529 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 J24 mock treatment 144880.0 628.0 0.04 141520.0 -338.0 -0.03 0.0125 0.2517 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K01 compound treatment 98080.0 -46200.0 -3.15 87520.0 -54300.0 -4.04 -5.0856 -0.9923 3652918 Neuro1_000573 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K02 compound treatment 139000.0 -5250.0 -0.36 135640.0 -6220.0 -0.46 -0.5804 -0.992 3652920 Neuro1_000574 Cc1ccc(cc1)c2nc(N/N=C/c3ccccc3Cl)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K03 compound treatment 163920.0 19700.0 1.34 161760.0 19900.0 1.48 1.9956 0.9988 1554183 Neuro1_000575 Clc1ccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K04 compound treatment 17280.0 -127000.0 -8.66 17520.0 -124000.0 -9.25 -12.6647 -0.9994 1935257 Neuro1_000576 Cc1ccc(cc1)c2nc(N/N=C/c3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K05 compound treatment 156440.0 12200.0 0.83 153240.0 11400.0 0.85 1.1866 1.0 1246914 Neuro1_000577 COc1ccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K06 compound treatment 167360.0 23100.0 1.58 163720.0 21900.0 1.63 2.2645 0.9999 1935637 Neuro1_000578 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K07 compound treatment 157520.0 13300.0 0.9 163120.0 21300.0 1.58 1.7586 0.9648 1271420 Neuro1_000579 CN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K08 compound treatment 168520.0 24300.0 1.65 168120.0 26300.0 1.95 2.552 0.9966 3652922 Neuro1_000580 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K09 compound treatment 161320.0 17100.0 1.16 159000.0 17100.0 1.28 1.725 0.9989 1434003 Neuro1_000581 COc1ccc(CNc2nc(nc3ccccc23)c4ccccc4)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K10 compound treatment 163240.0 19000.0 1.29 161600.0 19700.0 1.47 1.9544 0.998 1941166 Neuro1_000582 Brc1ccc2ncnc(NCCCN3CCOCC3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K11 compound treatment 156160.0 11900.0 0.81 156760.0 14900.0 1.11 1.3583 0.9882 1372612 Neuro1_000583 Clc1ccc(c(Cl)c1)c2nc(N3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K12 compound treatment 186440.0 42200.0 2.88 180240.0 38400.0 2.86 4.0538 1.0 1941168 Neuro1_000584 CC(=O)c1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K13 compound treatment 202200.0 57900.0 3.95 197240.0 55400.0 4.12 5.7082 0.9998 1267611 Neuro1_000585 Clc1ccc(Nc2nc(nc3ccccc23)c4ccncc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K14 compound treatment 165200.0 20900.0 1.43 159760.0 17900.0 1.33 1.952 0.9994 1659533 Neuro1_000586 Cc1ccc2ncnc(NC(CC(=O)O)C(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K15 compound treatment 192560.0 48300.0 3.29 187160.0 45300.0 3.37 4.713 0.9999 1172751 Neuro1_000587 Brc1ccc(Nc2nc(nc3ccccc23)c4ccncc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K16 compound treatment 160320.0 16100.0 1.1 152200.0 10300.0 0.77 1.3189 0.9851 1941548 Neuro1_000588 COCCNc1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K17 compound treatment 165440.0 21200.0 1.44 162680.0 20800.0 1.55 2.1173 0.9994 3652924 Neuro1_000589 CCN(CC)CCCNc1ncnc2ccc(Br)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K18 compound treatment 172120.0 27900.0 1.9 166680.0 24800.0 1.85 2.6498 0.9999 3652925 Neuro1_000590 C(Cc1ccccc1)Nc2nc(/C=C/c3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K19 compound treatment 200440.0 56200.0 3.83 190680.0 48800.0 3.63 5.2781 0.9997 1401934 Neuro1_000591 Brc1ccc2ncnc(NCCc3ccccc3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K20 compound treatment 197560.0 53300.0 3.63 198040.0 56200.0 4.18 5.5266 0.9976 1864031 Neuro1_000592 Oc1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K21 compound treatment 154400.0 10100.0 0.69 155360.0 13500.0 1.0 1.1998 0.9834 3027313 Neuro1_000593 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(C)CC4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K22 compound treatment 163400.0 19100.0 1.31 159440.0 17600.0 1.31 1.8484 1.0 1184905 Neuro1_000594 COC(=O)c1ccc(Nc2ncnc3ccccc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K23 mock treatment 147920.0 3670.0 0.25 146880.0 5020.0 0.37 0.4411 0.9809 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 K24 mock treatment 146440.0 2190.0 0.15 139160.0 -2700.0 -0.2 -0.0365 -0.146 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L01 compound treatment 151600.0 7350.0 0.5 148240.0 6380.0 0.48 0.6901 0.9996 3652927 Neuro1_000595 Clc1ccc(c(Cl)c1)c2nc(Nc3ccc(I)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L02 compound treatment 158000.0 13700.0 0.94 155920.0 14100.0 1.05 1.4028 0.9985 1201460 Neuro1_000596 CN1CCN(CC1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L03 compound treatment 170760.0 26500.0 1.81 170040.0 28200.0 2.1 2.7611 0.9972 1155180 Neuro1_000597 Oc1ccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L04 compound treatment 179120.0 34900.0 2.38 206040.0 64200.0 4.78 5.0587 0.9481 1356650 Neuro1_000598 Fc1ccccc1Nc2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L05 compound treatment 168880.0 24600.0 1.68 158240.0 16400.0 1.22 2.0494 0.9877 1589346 Neuro1_000599 Clc1ccc(c(Cl)c1)c2nc(Nc3ccc4OCCOc4c3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L06 compound treatment 179160.0 34900.0 2.38 182840.0 41000.0 3.05 3.8397 0.9925 1371105 Neuro1_000600 Fc1ccc(cc1)C(=O)Oc2cccc(Nc3ncnc4ccccc34)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L07 compound treatment 179760.0 35500.0 2.42 175320.0 33500.0 2.49 3.4728 0.9999 1441651 Neuro1_000601 Fc1ccccc1Nc2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L08 compound treatment 158280.0 14000.0 0.96 151280.0 9420.0 0.7 1.1721 0.9884 1491367 Neuro1_000602 COc1cccc(Nc2nc(nc3ccccc23)c4ccc(C)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L09 compound treatment 160480.0 16200.0 1.11 161240.0 19400.0 1.44 1.8024 0.9914 1864056 Neuro1_000603 [O-][N+](=O)c1ccc(cc1)c2nc(NCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L10 compound treatment 160360.0 16100.0 1.1 161360.0 19500.0 1.45 1.8029 0.9905 1488897 Neuro1_000604 Cc1ccc(cc1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L11 compound treatment 157440.0 13200.0 0.9 155680.0 13800.0 1.03 1.3632 0.9977 1864069 Neuro1_000605 CC1CCCN(C1)c2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L12 compound treatment 155840.0 11600.0 0.79 154360.0 12500.0 0.93 1.2166 0.9967 1589550 Neuro1_000606 COc1ccccc1Nc2nc(nc3ccccc23)c4ccc(C)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L13 compound treatment 180760.0 36500.0 2.49 178520.0 36700.0 2.73 3.6894 0.9989 1864030 Neuro1_000607 Oc1cccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L14 compound treatment 178080.0 33800.0 2.31 178080.0 36200.0 2.7 3.5371 0.997 1438155 Neuro1_000608 CCCOc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L15 compound treatment 151640.0 7390.0 0.5 149080.0 7220.0 0.54 0.7362 0.9995 1228044 Neuro1_000609 CN(C)CCNc1nc(nc2ccccc12)c3ccc(cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L16 compound treatment 192280.0 48000.0 3.27 195480.0 53600.0 3.99 5.1374 0.9952 1241988 Neuro1_000610 Clc1ccc(Nc2nc(N3CCOCC3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L17 compound treatment 167240.0 23000.0 1.57 165160.0 23300.0 1.73 2.3345 0.9987 1650752 Neuro1_000611 CC(C)(C)c1ccc(cc1)c2nc(Nc3ccc(cc3)C(=O)O)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L18 compound treatment 270560.0 126000.0 8.61 269640.0 128000.0 9.51 12.814 0.9988 3652928 Neuro1_000612 Oc1ccccc1c2nc(NCC3CCOC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L19 compound treatment 169880.0 25600.0 1.75 169520.0 27700.0 2.06 2.6913 0.9967 1615698 Neuro1_000613 CCOC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L20 compound treatment 174200.0 29900.0 2.04 167240.0 25400.0 1.89 2.7795 0.9992 1457150 Neuro1_000614 COc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L21 compound treatment 155680.0 11400.0 0.78 155440.0 13600.0 1.01 1.2657 0.9917 1608866 Neuro1_000615 CCOc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L22 compound treatment 148080.0 3830.0 0.26 145800.0 3940.0 0.29 0.392 0.9983 1445378 Neuro1_000616 COc1ccccc1Nc2nc(nc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L23 mock treatment 148760.0 4510.0 0.31 143800.0 1940.0 0.14 0.3195 0.9409 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 L24 mock treatment 145480.0 1230.0 0.08 140320.0 -1540.0 -0.11 -0.0217 -0.1533 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M01 compound treatment 139880.0 -4370.0 -0.3 140120.0 -1740.0 -0.13 -0.3022 -0.9301 3652929 Neuro1_000617 Fc1ccccc1/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M02 compound treatment 152760.0 8510.0 0.58 153960.0 12100.0 0.9 1.0471 0.9773 3652931 Neuro1_000618 C/C(=N\Nc1nc(nc2ccccc12)c3ccc(C)cc3)/c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M03 compound treatment 134000.0 -10300.0 -0.7 132800.0 -9060.0 -0.67 -0.9709 -0.9998 3652933 Neuro1_000619 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M04 compound treatment 128960.0 -15300.0 -1.04 123480.0 -18400.0 -1.37 -1.7044 -0.991 1935343 Neuro1_000620 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M05 compound treatment 163000.0 18700.0 1.28 159840.0 18000.0 1.34 1.8502 0.9997 1590843 Neuro1_000621 Brc1ccc(cc1)c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M06 compound treatment 174960.0 30700.0 2.09 169360.0 27500.0 2.05 2.9278 0.9999 3652935 Neuro1_000622 CCCCCc1ccc(cc1)/C(=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M07 compound treatment 128080.0 -16200.0 -1.1 114240.0 -27600.0 -2.06 -2.2331 -0.9574 3652937 Neuro1_000623 COc1ccccc1/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M08 compound treatment 172800.0 28500.0 1.95 169720.0 27900.0 2.07 2.8426 0.9995 1935891 Neuro1_000624 Cc1ccc(cc1)c2nc(N/N=C/c3ccc(cc3)[N+](=O)[O-])c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M09 compound treatment 168280.0 24000.0 1.64 160720.0 18900.0 1.4 2.151 0.997 1505815 Neuro1_000625 CCOC(=O)C1CCN(CC1)c2nc(nc3ccccc23)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M10 compound treatment 162560.0 18300.0 1.25 158920.0 17100.0 1.27 1.7805 1.0 1578334 Neuro1_000626 OC(=O)CC(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M11 compound treatment 159120.0 14900.0 1.01 159360.0 17500.0 1.3 1.6379 0.9923 1608315 Neuro1_000627 CC(C)Nc1nc(nc2ccccc12)c3ccc(Cl)cc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M12 compound treatment 183840.0 39600.0 2.7 181240.0 39400.0 2.93 3.9811 0.9992 1597755 Neuro1_000628 Cc1ccc(Nc2ncnc3ccc(Br)cc23)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M13 compound treatment 179960.0 35700.0 2.43 178400.0 36500.0 2.72 3.6445 0.9985 1195961 Neuro1_000629 Cc1ccc(C)c(Nc2nc(nc3ccccc23)c4ccncc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M14 compound treatment 161560.0 17300.0 1.18 157560.0 15700.0 1.17 1.6608 1.0 1466687 Neuro1_000630 CC(C)CNc1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M15 compound treatment 163200.0 18900.0 1.29 161080.0 19200.0 1.43 1.9251 0.9987 1483149 Neuro1_000631 COC(=O)CCNc1nc(nc2ccccc12)c3ccc(Br)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M16 compound treatment 165560.0 21300.0 1.45 160800.0 18900.0 1.41 2.0241 0.9999 1738379 Neuro1_000632 CCOC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M17 compound treatment 201920.0 57700.0 3.93 200120.0 58300.0 4.34 5.8463 0.9988 1164820 Neuro1_000633 CC1CCCCC1Nc2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M18 compound treatment 166520.0 22300.0 1.52 164760.0 22900.0 1.7 2.2788 0.9983 3652939 Neuro1_000634 COC(=O)c1cccc(Nc2nc(/C=C/c3ccccc3)nc4ccccc24)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M19 compound treatment 205280.0 61000.0 4.16 201040.0 59200.0 4.4 6.0567 0.9996 1330942 Neuro1_000635 Brc1ccc2ncnc(Nc3ccc4OCCOc4c3)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M20 compound treatment 210000.0 65700.0 4.48 207720.0 65900.0 4.9 6.6358 0.999 1864046 Neuro1_000636 [O-][N+](=O)c1ccc(cc1)c2nc(NC3CCCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M21 compound treatment 175320.0 31100.0 2.12 170720.0 28900.0 2.15 3.0167 1.0 1681263 Neuro1_000637 Cc1ccc(Nc2nc(nc3ccccc23)c4ccccc4O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M22 compound treatment 155920.0 11700.0 0.8 156320.0 14500.0 1.08 1.3236 0.9889 1864071 Neuro1_000638 CC1(CC2CC(C)(C)C1)CN2c3nc(nc4ccccc34)c5ccc(cc5)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M23 mock treatment 149800.0 5550.0 0.38 145360.0 3500.0 0.26 0.4518 0.9835 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 M24 mock treatment 147960.0 3710.0 0.25 148000.0 6140.0 0.46 0.502 0.961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N01 compound treatment 175640.0 31400.0 2.14 182680.0 40800.0 3.04 3.6615 0.9853 1864018 Neuro1_000639 Cc1ccccc1Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N02 compound treatment 154680.0 10400.0 0.71 153360.0 11500.0 0.86 1.108 0.9957 1118945 Neuro1_000640 C(N1CCN(CC1)c2nc(N3CCOCC3)c4ccccc4n2)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N03 compound treatment 156160.0 11900.0 0.81 157000.0 15100.0 1.13 1.371 0.987 1864029 Neuro1_000641 COc1ccc(Cl)cc1Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N04 compound treatment 187280.0 43000.0 2.93 188760.0 46900.0 3.49 4.5427 0.9963 1677576 Neuro1_000642 CN(C)CCNc1nc(nc2ccccc12)c3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N05 compound treatment 171520.0 27300.0 1.86 175400.0 33500.0 2.5 3.0798 0.9895 1864025 Neuro1_000643 [O-][N+](=O)c1ccc(cc1)c2nc(Nc3cccc(Cl)c3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N06 compound treatment 166920.0 22700.0 1.55 160600.0 18700.0 1.39 2.0791 0.9987 1573616 Neuro1_000644 Cc1cccc(c1)c2nc(N3CC4(C)CC3CC(C)(C)C4)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N07 compound treatment 165440.0 21200.0 1.44 162120.0 20300.0 1.51 2.0878 0.9998 1432761 Neuro1_000645 CCOc1ccccc1Nc2nc(nc3ccccc23)c4ccc(Cl)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N08 compound treatment 158520.0 14300.0 0.97 150480.0 8620.0 0.64 1.1416 0.9796 1314067 Neuro1_000646 Cc1ccc(cc1)c2nc(Nc3cccc(c3)C(=O)O)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N09 compound treatment 165240.0 21000.0 1.43 160800.0 18900.0 1.41 2.0087 1.0 1560212 Neuro1_000647 CC(C)(C)c1ccc(cc1)c2nc(N3CCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N10 compound treatment 151640.0 7390.0 0.5 154200.0 12300.0 0.92 1.0057 0.96 1393428 Neuro1_000648 COc1ccccc1Nc2nc(nc3ccccc23)c4cccc(C)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N11 compound treatment 193880.0 49600.0 3.38 195720.0 53900.0 4.01 5.2271 0.9964 1874117 Neuro1_000649 COC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N12 compound treatment 161360.0 17100.0 1.17 160480.0 18600.0 1.39 1.8048 0.9963 1309268 Neuro1_000650 COC(=O)c1cccc(Nc2nc(nc3ccccc23)c4cccc(C)c4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N13 compound treatment 237680.0 93400.0 6.37 241800.0 99900.0 7.44 9.7637 0.997 1864036 Neuro1_000651 CCOc1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N14 compound treatment 171320.0 27100.0 1.85 169960.0 28100.0 2.09 2.7839 0.9981 1368813 Neuro1_000652 COc1ccc(Nc2ncnc3ccc(Br)cc23)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N15 compound treatment 211240.0 67000.0 4.57 202400.0 60500.0 4.51 6.4156 1.0 1864039 Neuro1_000653 COC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N16 compound treatment 174760.0 30500.0 2.08 166480.0 24600.0 1.83 2.7665 0.998 1523724 Neuro1_000654 COc1ccc(OC)c(Nc2nc(nc3ccccc23)c4ccccc4O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N17 compound treatment 155160.0 10900.0 0.74 153760.0 11900.0 0.89 1.1522 0.9962 1975030 Neuro1_000655 COCCCNc1nc(nc2ccccc12)c3ccc(cc3)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N18 compound treatment 163040.0 18800.0 1.28 167160.0 25300.0 1.88 2.2373 0.9824 3652941 Neuro1_000656 Oc1ccccc1c2nc(N3CCN(CC3)C(c4ccccc4)c5ccccc5)c6ccccc6n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N19 compound treatment 161480.0 17200.0 1.17 158160.0 16300.0 1.21 1.6885 0.9999 1421575 Neuro1_000657 OC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N20 compound treatment 160640.0 16400.0 1.12 159720.0 17900.0 1.33 1.7301 0.9963 1371006 Neuro1_000658 Cc1cccc(Nc2ncnc3ccc(Br)cc23)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N21 compound treatment 160880.0 16600.0 1.13 168360.0 26500.0 1.97 2.1964 0.9654 1371117 Neuro1_000659 Oc1cccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N22 compound treatment 160360.0 16100.0 1.1 161600.0 19700.0 1.47 1.8155 0.9897 3652942 Neuro1_000660 Fc1ccc(Nc2nc(NCC3CCCO3)c4ccccc4n2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N23 mock treatment 145280.0 1030.0 0.07 143400.0 1540.0 0.11 0.1307 0.9719 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 N24 mock treatment 140360.0 -3890.0 -0.27 142720.0 863.0 0.06 -0.1423 -0.521 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O01 compound treatment 87400.0 -56900.0 -3.88 63440.0 -78400.0 -5.84 -6.8677 -0.9802 3652943 Neuro1_000661 COc1ccc(/C=N/Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O02 compound treatment 152080.0 7830.0 0.53 151800.0 9940.0 0.74 0.9006 0.9871 3652945 Neuro1_000662 CCCCc1ccc(cc1)/C(=N/Nc2nc(nc3ccccc23)c4ccc(C)cc4)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O03 compound treatment 168760.0 24500.0 1.67 172720.0 30900.0 2.3 2.8057 0.9878 1145689 Neuro1_000663 COC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O04 compound treatment 154960.0 10700.0 0.73 164320.0 22500.0 1.67 1.6983 0.931 3652947 Neuro1_000664 Cc1ccc(cc1)c2nc(N/N=C/c3c(F)c(F)c(F)c(F)c3F)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O05 compound treatment 153880.0 9630.0 0.66 153960.0 12100.0 0.9 1.1011 0.9879 3652949 Neuro1_000665 Fc1ccc(Nc2nc(nc3ccccc23)c4ccc(Br)cc4)cc1F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O06 compound treatment 157920.0 13700.0 0.93 147480.0 5620.0 0.42 0.9548 0.9347 1458048 Neuro1_000666 Cc1ccc(Nc2nc(nc3ccccc23)c4ccc(C)cc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O07 compound treatment 158600.0 14300.0 0.98 150120.0 8260.0 0.61 1.1265 0.975 1191448 Neuro1_000667 Brc1ccc(cc1)c2nc(N3CCCCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O08 compound treatment 155320.0 11100.0 0.75 151160.0 9300.0 0.69 1.0231 0.9991 3652950 Neuro1_000668 Cc1ccc(cc1)c2nc(N/N=C/c3ccc(Br)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O09 compound treatment 184480.0 40200.0 2.74 191960.0 50100.0 3.73 4.5761 0.9886 3652952 Neuro1_000669 CC(=O)c1ccc(cc1)N2CCN(CC2)c3nc(nc4ccccc34)c5ccccc5 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O10 compound treatment 174520.0 30300.0 2.06 166480.0 24600.0 1.83 2.755 0.9982 1476095 Neuro1_000670 COC(=O)c1cccc(Nc2ncnc3ccc(Br)cc23)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O11 compound treatment 152120.0 7870.0 0.54 152760.0 10900.0 0.81 0.9531 0.9798 1384871 Neuro1_000671 CN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(Cl)c(Cl)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O12 compound treatment 174800.0 30500.0 2.08 172360.0 30500.0 2.27 3.0779 0.9991 1260329 Neuro1_000672 CCC(Nc1ncnc2ccc(Br)cc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O13 compound treatment 195040.0 50800.0 3.46 187480.0 45600.0 3.4 4.8494 1.0 1616520 Neuro1_000673 COc1ccc(Nc2nc(nc3ccccc23)c4ccncc4)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O14 compound treatment 157240.0 13000.0 0.89 159840.0 18000.0 1.34 1.5725 0.9799 1565343 Neuro1_000674 OC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccccc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O15 compound treatment 201600.0 57300.0 3.91 204320.0 62500.0 4.65 6.0519 0.9963 1630999 Neuro1_000675 C(Cc1ccccc1)Nc2nc(nc3ccccc23)c4cccnc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O16 compound treatment 149200.0 4950.0 0.34 150120.0 8260.0 0.61 0.6733 0.96 1141931 Neuro1_000676 Clc1ccc(cc1)c2nc(NCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O17 compound treatment 179240.0 35000.0 2.39 176280.0 34400.0 2.56 3.4983 0.9994 1165000 Neuro1_000677 Cc1ccc(Nc2ncnc3ccc(Br)cc23)cc1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O18 compound treatment 165000.0 20700.0 1.41 170760.0 28900.0 2.15 2.5213 0.9793 3652953 Neuro1_000678 CN1CCN(CC1)c2nc(/C=C/c3ccccc3)nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O19 compound treatment 157520.0 13300.0 0.9 155640.0 13800.0 1.03 1.3649 0.998 1194253 Neuro1_000679 CCN1CCN(CC1)c2ncnc3ccc(Br)cc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O20 compound treatment 165240.0 21000.0 1.43 163240.0 21400.0 1.59 2.1371 0.9986 1974698 Neuro1_000680 COCCCNc1nc(nc2ccccc12)c3ccc(cc3)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O21 compound treatment 198160.0 53900.0 3.68 195480.0 53600.0 3.99 5.4208 0.9992 1933893 Neuro1_000681 CC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccccc4O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O22 compound treatment 176480.0 32200.0 2.2 169520.0 27700.0 2.06 3.0094 0.9995 1864034 Neuro1_000682 COc1ccc(Nc2nc(nc3ccccc23)c4ccc(cc4)[N+](=O)[O-])cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O23 mock treatment 142560.0 -1690.0 -0.12 151760.0 9900.0 0.74 0.4396 0.5892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 O24 mock treatment 141800.0 -2450.0 -0.17 140720.0 -1140.0 -0.08 -0.1781 -0.9503 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P01 compound treatment 182200.0 37900.0 2.59 177640.0 35800.0 2.66 3.7125 0.9999 3652955 Neuro1_000683 CC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P02 compound treatment 152640.0 8390.0 0.57 152040.0 10200.0 0.76 0.9402 0.9904 1419363 Neuro1_000684 CCOC(=O)c1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P03 compound treatment 166120.0 21900.0 1.49 169720.0 27900.0 2.07 2.5205 0.9869 1618578 Neuro1_000685 COC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P04 compound treatment 146760.0 2510.0 0.17 148400.0 6540.0 0.49 0.4652 0.9014 1276280 Neuro1_000686 Cc1cccc(Nc2nc(nc3ccccc23)c4ccc(Cl)cc4)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P05 compound treatment 217080.0 72800.0 4.97 207920.0 66100.0 4.92 6.9876 1.0 1864053 Neuro1_000687 [O-][N+](=O)c1ccc(cc1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P06 compound treatment 176040.0 31800.0 2.17 173960.0 32100.0 2.39 3.2219 0.9988 1334348 Neuro1_000688 O=C(Oc1cccc(Nc2ncnc3ccccc23)c1)c4cccs4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P07 compound treatment 156400.0 12100.0 0.83 153480.0 11600.0 0.87 1.1973 0.9998 1287828 Neuro1_000689 CN1CCN(CC1)c2nc(NCc3ccco3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P08 compound treatment 155160.0 10900.0 0.74 158120.0 16300.0 1.21 1.3817 0.9726 1652815 Neuro1_000690 CN(Cc1ccccc1)c2nc(nc3ccccc23)c4cccc(C)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P09 compound treatment 247760.0 104000.0 7.06 260840.0 119000.0 8.86 11.2517 0.9937 1864049 Neuro1_000691 [O-][N+](=O)c1ccc(cc1)c2nc(NCc3ccccc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P10 compound treatment 179040.0 34800.0 2.37 179360.0 37500.0 2.79 3.6507 0.9967 1329450 Neuro1_000692 COc1cc(cc(OC)c1OC)C(=O)Oc2cccc(Nc3ncnc4ccccc34)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P11 compound treatment 171760.0 27500.0 1.88 173400.0 31500.0 2.35 2.9861 0.9938 3652956 Neuro1_000693 [O-][N+](=O)c1ccc(cc1)c2nc(Nc3ccc4OCCOc4c3)c5ccccc5n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P12 compound treatment 163920.0 19700.0 1.34 159640.0 17800.0 1.32 1.884 1.0 1481183 Neuro1_000694 Cc1cccc(c1)c2nc(NCc3cccnc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P13 compound treatment 158520.0 14300.0 0.97 156080.0 14200.0 1.06 1.4363 0.9991 1974536 Neuro1_000695 CCN(CC)CCCNc1nc(nc2ccccc12)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P14 compound treatment 418600.0 274000.0 18.7 418920.0 277000.0 20.62 27.807 0.9988 3652957 Neuro1_000696 CN(C)CCCNc1nc(nc2ccccc12)c3ccccc3O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P15 compound treatment 183840.0 39600.0 2.7 181800.0 39900.0 2.97 4.0105 0.9988 1864026 Neuro1_000697 [O-][N+](=O)c1ccc(cc1)c2nc(Nc3ccc(Cl)cc3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P16 compound treatment 168920.0 24700.0 1.68 169400.0 27500.0 2.05 2.6387 0.9952 1227490 Neuro1_000698 COc1ccc(Nc2nc(nc3ccccc23)c4ccccc4O)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P17 compound treatment 140480.0 -3770.0 -0.26 140000.0 -1860.0 -0.14 -0.2796 -0.9576 1672057 Neuro1_000699 CC(C)(C)c1ccc(cc1)c2nc(NCCN3CCOCC3)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P18 compound treatment 173080.0 28800.0 1.97 173560.0 31700.0 2.36 3.0582 0.9959 1204793 Neuro1_000700 COc1ccc(Nc2ncnc3ccc(Br)cc23)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P19 compound treatment 172680.0 28400.0 1.94 171840.0 30000.0 2.23 2.9484 0.9975 1864298 Neuro1_000701 [O-][N+](=O)c1cccc(Nc2nc(nc3ccccc23)c4ccccc4Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P20 compound treatment 177720.0 33500.0 2.28 169520.0 27700.0 2.06 3.0692 0.9987 1679198 Neuro1_000702 CC(C)(C)c1ccc(cc1)c2nc(Nc3cccc(c3)C(=O)O)c4ccccc4n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P21 compound treatment 167440.0 23200.0 1.58 162720.0 20900.0 1.55 2.2158 1.0 1267483 Neuro1_000703 Cc1c(Cl)cccc1Nc2nc(nc3ccccc23)c4ccccc4Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P22 compound treatment 160760.0 16500.0 1.13 158080.0 16200.0 1.21 1.6496 0.9994 3652958 Neuro1_000704 COC(=O)c1ccc(Nc2nc(nc3ccccc23)c4ccccc4F)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P23 mock treatment 147160.0 2910.0 0.2 146560.0 4700.0 0.35 0.3876 0.9638 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2436 P24 mock treatment 145280.0 1030.0 0.07 140440.0 -1420.0 -0.11 -0.0251 -0.1979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A01 mock treatment 142840.0 -3440.0 -0.23 145600.0 -2860.0 -0.21 -0.3163 -0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A02 mock treatment 137760.0 -8520.0 -0.58 145440.0 -3020.0 -0.22 -0.5696 -0.9147 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A03 compound treatment 139400.0 -6880.0 -0.47 148440.0 -21.0 0.0 -0.3327 -0.7095 1023 BSPBio_003201 CN[C@H](CC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A04 compound treatment 199000.0 52700.0 3.59 215120.0 66700.0 4.96 6.0498 0.9875 1053060 BSPBio_003202 COc1ccc(cc1OC)c2oc3ccccc3c(=O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A05 compound treatment 141920.0 -4360.0 -0.3 142840.0 -5620.0 -0.42 -0.5059 -0.9859 1496 BSPBio_003203 CSc1ccc2Sc3ccccc3CC(N4CCN(C)CC4)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A06 compound treatment 140720.0 -5560.0 -0.38 144120.0 -4340.0 -0.32 -0.4964 -0.9969 3198541 BSPBio_003204 CC(CCC=C(C)C)C1CC[C@@]2(C)C3=C(CC[C@]12C)C4(C)CC[C@H](OC(=O)C)C(C)(C)C4CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A07 compound treatment 139160.0 -7120.0 -0.49 145680.0 -2780.0 -0.21 -0.4895 -0.9278 1280 BSPBio_003205 NCCNC(=O)c1ccc(Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A08 compound treatment 138400.0 -7880.0 -0.54 144160.0 -4300.0 -0.32 -0.6061 -0.9694 1001518 BSPBio_003206 CCC[C@H](N[C@@H](C)C(=O)N1[C@@H](C[C@@H]2CCCC[C@@H]21)C(=O)O)C(=O)OCC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A09 compound treatment 138080.0 -8200.0 -0.56 145280.0 -3180.0 -0.24 -0.5626 -0.9269 924 BSPBio_003207 NC(=N)NC(=N)Nc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A10 compound treatment 142720.0 -3560.0 -0.24 148960.0 499.0 0.04 -0.1452 -0.5919 1003535 BSPBio_003208 ONC(=O)Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A11 compound treatment 145560.0 -718.0 -0.05 146520.0 -1940.0 -0.14 -0.1367 -0.8965 3174610 BSPBio_003209 COc1cc(cc(OC)c1OC)C(=O)O[C@H]2CC[C@@]3(C)[C@@H]4CC[C@@H]5[C@@]3(C[C@@]6(O)[C@@H]7CN8C[C@@H](C)CC[C@H]8[C@@](C)(O)[C@@]7(O)[C@@H](O)C[C@@]56O)O[C@@]42O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A12 compound treatment 170720.0 24400.0 1.67 169600.0 21100.0 1.57 2.2908 0.9996 3079280 BSPBio_003210 O[C@@H]1Cc2c(O)cc(O)cc2O[C@@H]1c3ccc(O)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A13 compound treatment 150520.0 4240.0 0.29 148120.0 -341.0 -0.03 0.1866 0.6426 1384 BSPBio_003211 COC(=O)[C@@H](N1CCc2sccc2C1)c3ccccc3Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A14 compound treatment 144640.0 -1640.0 -0.11 143520.0 -4940.0 -0.37 -0.339 -0.882 1110410 BSPBio_003212 COc1ccc(C(=O)C)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A15 compound treatment 173800.0 27500.0 1.88 175080.0 26600.0 1.98 2.7277 0.9996 3198436 BSPBio_003213 CO[C@H]1CC(O[C@H]/2[C@@H](C)\C=C\C=C\3/CO[C@@H]4\C(=N/O)\C(=C[C@@H](C(=O)O[C@H]5C[C@@H](C\C=C2/C)O[C@@]6(CC[C@H](C)[C@H](O6)C7CCCCC7)C5)[C@@]43O)C)O[C@@H](C)C1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A16 compound treatment 144280.0 -2000.0 -0.14 147320.0 -1140.0 -0.08 -0.1563 -0.9742 3079389 BSPBio_003214 COc1cc(OC)c(C(=O)c2ccc(O)cc2)c(OC)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A17 compound treatment 222080.0 75800.0 5.17 245360.0 96900.0 7.21 8.7539 0.9866 1950 BSPBio_003215 Oc1cc2oc(cc(=O)c2c(O)c1O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A18 compound treatment 239680.0 93400.0 6.37 269760.0 121000.0 9.03 10.8865 0.9854 2069327 BSPBio_003216 COC/1=CC(=O)C(=C\C1=C/C=C/c2ccccc2)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A19 compound treatment 159240.0 13000.0 0.88 172600.0 24100.0 1.8 1.8953 0.9466 3172852 BSPBio_003217 CC1(C)CC[C@@]2(CC[C@]3(C)C(=CCC4[C@@]5(C)CC[C@H](O)[C@@](C)(CO)C5CC[C@]43C)C2C1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A20 compound treatment 147960.0 1680.0 0.11 149560.0 1100.0 0.08 0.139 0.9863 3054572 BSPBio_003218 CC(=O)O[C@@H]1CC[C@@]2(C)C(CC[C@]3(C)C2CC=C4C5CC(C)(C)CC[C@@]5(CC[C@]43C)C(=O)O)C1(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A21 compound treatment 141000.0 -5280.0 -0.36 141960.0 -6500.0 -0.48 -0.5966 -0.9894 3650214 BSPBio_003219 C[C@H]1O[C@H](O[C@H]2[C@H](O)[C@H](O)CO[C@@H]2O[C@H]3CC[C@@]4(C)C(CC[C@]5(C)C4CC=C6[C@@H]7CC(C)(C)CC[C@@]7(CC[C@]65C)C(=O)O)[C@]3(C)CO)[C@@H](O)[C@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A22 compound treatment 174800.0 28500.0 1.94 177400.0 28900.0 2.15 2.898 0.9987 3081175 BSPBio_003220 CCOC(=O)c1c(C)c(Cl)c(O)c(Cl)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A23 mock treatment 140000.0 -6280.0 -0.43 141240.0 -7220.0 -0.54 -0.6827 -0.9936 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 A24 mock treatment 135600.0 -10700.0 -0.73 138240.0 -10200.0 -0.76 -1.0527 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B01 mock treatment 140640.0 -5640.0 -0.38 138040.0 -10400.0 -0.78 -0.8202 -0.9475 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B02 mock treatment 137520.0 -8760.0 -0.6 174800.0 26300.0 1.96 0.964 0.4704 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B03 compound treatment 134840.0 -11400.0 -0.78 140080.0 -8380.0 -0.62 -0.9925 -0.9939 1000115 BSPBio_003221 COC(=O)[C@@H]1[C@@H](O)CC[C@@H]2CN3CCc4c([nH]c5ccccc45)[C@@H]3C[C@H]12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B04 compound treatment 142920.0 -3360.0 -0.23 148680.0 219.0 0.02 -0.1503 -0.6551 1864491 BSPBio_003222 COc1ccc(cc1)c2coc3cc(OC)cc(OC)c3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B05 compound treatment 149800.0 3520.0 0.24 149080.0 619.0 0.05 0.2024 0.8277 1258696 BSPBio_003223 Cc1c(Cl)cccc1Nc2ccccc2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B06 compound treatment 252400.0 106000.0 7.24 263760.0 115000.0 8.58 11.1839 0.9964 1119359 BSPBio_003224 COc1cc2ccc(=O)oc2c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B07 compound treatment 149040.0 2760.0 0.19 152600.0 4140.0 0.31 0.351 0.9721 1865 BSPBio_003225 Clc1cccc(Nc2nnc(c3ccccc3)c4ccccc24)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B08 compound treatment 135880.0 -10400.0 -0.71 143000.0 -5460.0 -0.41 -0.7886 -0.9651 907087 BSPBio_003226 CCN(CC)CCNC(=O)c1ccc(NC(=O)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B09 compound treatment 138480.0 -7800.0 -0.53 139360.0 -9100.0 -0.68 -0.8549 -0.9928 1271 BSPBio_003227 CC(=O)OC(CC(=O)O)[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B10 compound treatment 216880.0 70600.0 4.81 223200.0 74700.0 5.56 7.337 0.9974 1329 BSPBio_003228 NC(Cc1cc(I)c(Oc2ccc(O)c(I)c2)c(I)c1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B11 compound treatment 140800.0 -5480.0 -0.37 142880.0 -5580.0 -0.42 -0.5578 -0.9986 3198548 BSPBio_003229 OC(=O)CCC/C=C\C[C@@H]1CO[C@@H](O[C@@H]1c2ccccc2O)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B12 compound treatment 142720.0 -3560.0 -0.24 147000.0 -1460.0 -0.11 -0.2484 -0.9345 1269 BSPBio_003230 CC(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B13 compound treatment 147200.0 923.0 0.06 147320.0 -1140.0 -0.08 -0.0156 -0.1474 1458 BSPBio_003231 NC(Cc1ccc(Cl)cc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B14 compound treatment 139000.0 -7280.0 -0.5 143080.0 -5380.0 -0.4 -0.634 -0.9944 1001907 BSPBio_003232 C[C@](N)(Cc1ccc(O)cc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B15 compound treatment 151080.0 4800.0 0.33 149080.0 619.0 0.05 0.2641 0.7987 1502 BSPBio_003233 OC(=O)c1c2ccccc2cc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B16 compound treatment 139720.0 -6560.0 -0.45 138040.0 -10400.0 -0.78 -0.8646 -0.9657 2060343 BSPBio_003234 CCCc1occc(=O)c1/C=C/O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B17 compound treatment 150480.0 4200.0 0.29 155400.0 6940.0 0.52 0.5678 0.9614 440 BSPBio_003235 COC(=O)Nc1nc2cc(ccc2[nH]1)C(=O)c3cccs3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B18 compound treatment 139200.0 -7080.0 -0.48 142040.0 -6420.0 -0.48 -0.6791 -1.0 1429 BSPBio_003236 CCCCOC(=O)c1ccc(N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B19 compound treatment 167920.0 21600.0 1.48 176000.0 27500.0 2.05 2.4927 0.987 2069318 BSPBio_003237 C[C@@H](NC(=O)/C(=C\c1ccc(O)c(O)c1)/C#N)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B20 compound treatment 141360.0 -4920.0 -0.34 145440.0 -3020.0 -0.22 -0.3961 -0.9811 1008566 BSPBio_003238 Cc1cc(c(O)c(c1)C(C)(C)C)C(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B21 compound treatment 151120.0 4840.0 0.33 152480.0 4020.0 0.3 0.445 0.9988 3480197 BSPBio_003239 CCC(NC(C)C)C(O)c1ccc(O)c2[nH]c(=O)ccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B22 compound treatment 138160.0 -8120.0 -0.55 143520.0 -4940.0 -0.37 -0.6514 -0.9803 1000287 BSPBio_003240 OC(=O)CC(O)(CC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B23 mock treatment 138640.0 -7640.0 -0.52 140160.0 -8300.0 -0.62 -0.8051 -0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 B24 mock treatment 140280.0 -6000.0 -0.41 139800.0 -8660.0 -0.64 -0.7449 -0.9759 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C01 mock treatment 141400.0 -4880.0 -0.33 140040.0 -8420.0 -0.63 -0.6783 -0.956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C02 mock treatment 147160.0 883.0 0.06 146040.0 -2420.0 -0.18 -0.0849 -0.4467 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C03 compound treatment 139600.0 -6680.0 -0.46 144760.0 -3700.0 -0.28 -0.5167 -0.971 3172862 BSPBio_003241 O=c1cccc2C3CNC[C@@H](C3)Cn21 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C04 compound treatment 145280.0 -998.0 -0.07 151480.0 3020.0 0.22 0.1108 0.472 3081176 BSPBio_003242 COc1ccccc1c2coc3cc(OC)c(OC)c(OC)c3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C05 compound treatment 148240.0 1960.0 0.13 153800.0 5340.0 0.4 0.3756 0.8958 1024517 BSPBio_003243 COc1cc2CCNC(C)c2cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C06 compound treatment 88360.0 -57900.0 -3.95 84440.0 -64000.0 -4.76 -6.1614 -0.9956 2559 BSPBio_003244 CC(=O)O[Cd]OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C07 compound treatment 174960.0 28700.0 1.96 168920.0 20500.0 1.52 2.4594 0.9923 2060328 BSPBio_003245 CC(C)CC(=O)c1c(O)c(C)c(O)c2c1oc3c(C(=O)CC(C)C)c(O)c(C)c(O)c32 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C08 compound treatment 146840.0 563.0 0.04 147320.0 -1140.0 -0.08 -0.0329 -0.3534 BSPBio_003246 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C09 compound treatment 142880.0 -3400.0 -0.23 139440.0 -9020.0 -0.67 -0.6385 -0.8991 2060287 BSPBio_003247 Cc1c(O)c(O)cc2c1CC=C3[C@@]2(C)CC[C@@]4(C)C5C[C@@](C)(CC[C@]5(C)CC[C@]34C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C10 compound treatment 158000.0 11700.0 0.8 153520.0 5060.0 0.38 0.8314 0.941 2561 BSPBio_003248 Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C11 compound treatment 148240.0 1960.0 0.13 148680.0 219.0 0.02 0.1061 0.7874 2060298 BSPBio_003249 CCCCCC1C(CC(=O)O)CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C12 compound treatment 152080.0 5800.0 0.4 156600.0 8140.0 0.61 0.7081 0.9787 2558 BSPBio_003250 c1ccc2c(c1)cc3ccc4cccc5ccc2c3c45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C13 compound treatment 367640.0 221000.0 15.09 372720.0 224000.0 16.69 22.4738 0.9987 BSPBio_003251 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C14 compound treatment 162040.0 15800.0 1.07 160120.0 11700.0 0.87 1.3735 0.9944 1152 BSPBio_003252 CN(C)CCN(Cc1ccccc1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C15 compound treatment 191640.0 45400.0 3.09 207760.0 59300.0 4.41 5.3076 0.9849 2060454 BSPBio_003253 Oc1cc(O)c2c(=O)cc(oc2c1)c3cc(O)c(O)c(O)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C16 compound treatment 147400.0 1120.0 0.08 145800.0 -2660.0 -0.2 -0.0859 -0.4047 840 BSPBio_003254 CCOc1ccc2ccccc2c1NC(=O)[C@H]3[C@H]4SC(C)(C)C(N4C3=O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C17 compound treatment 143160.0 -3120.0 -0.21 148640.0 179.0 0.01 -0.1409 -0.6615 3173493 BSPBio_003255 CC1=C2CCC3C4CCC(=O)[C@@]4(C)CCC3[C@@]2(C)CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C18 compound treatment 164360.0 18100.0 1.23 170120.0 21700.0 1.61 2.0116 0.9912 3174105 BSPBio_003256 CN(C)c1ccc2[n+](C)c(/C=C/c3cc(C)n(c3C)c4ccccc4)ccc2c1.OC(=O)c1cc2ccccc2c(Cc3c(O)c(cc4ccccc34)C(=O)O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C19 compound treatment 158640.0 12400.0 0.84 160480.0 12000.0 0.89 1.2285 0.9996 2060271 BSPBio_003257 CCC(C)C(=O)c1c(O)c(C)c2oc3c(C)c(O)c(C(=O)C(C)CC)c(O)c3c2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C20 compound treatment 145720.0 -558.0 -0.04 146800.0 -1660.0 -0.12 -0.1143 -0.8837 3173091 BSPBio_003258 NC[C@@H]1O[C@H](O[C@H]2[C@@H](O)C(O[C@@H]3[C@@H](O)[C@H](N)C[C@H](N)[C@H]3OC4O[C@H](CN)[C@@H](O)[C@H](O)[C@H]4N)O[C@@H]2CO)[C@H](N)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C21 compound treatment 172280.0 26000.0 1.77 172840.0 24400.0 1.81 2.5366 0.9999 2060482 BSPBio_003259 CC(C)c1cc2CCC3C(C)(C)CCC[C@]3(C(=O)O)c2c(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C22 compound treatment 139120.0 -7160.0 -0.49 143800.0 -4660.0 -0.35 -0.5903 -0.986 934 BSPBio_003260 Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C23 mock treatment 139680.0 -6600.0 -0.45 146120.0 -2340.0 -0.17 -0.4413 -0.9148 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 C24 mock treatment 135520.0 -10800.0 -0.73 143960.0 -4500.0 -0.33 -0.7555 -0.937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D01 mock treatment 141920.0 -4360.0 -0.3 142160.0 -6300.0 -0.47 -0.5417 -0.9757 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D02 mock treatment 142840.0 -3440.0 -0.23 145040.0 -3420.0 -0.25 -0.3458 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D03 compound treatment 147080.0 803.0 0.05 143560.0 -4900.0 -0.36 -0.2192 -0.5944 1000118 BSPBio_003261 CN[C@@H](C)[C@@H](O)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D04 compound treatment 141720.0 -4560.0 -0.31 145480.0 -2980.0 -0.22 -0.3766 -0.9864 3198649 BSPBio_003262 COc1c(oc2c(CC=C(C)C)c3OC(C)(C)C=Cc3c(OC)c2c1=O)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D05 compound treatment 141880.0 -4400.0 -0.3 146520.0 -1940.0 -0.14 -0.3141 -0.944 1010471 BSPBio_003263 O=c1ccc2ccccc2o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D06 compound treatment 146840.0 563.0 0.04 151520.0 3060.0 0.23 0.1881 0.8147 3055306 BSPBio_003264 C[C@@H]1CC[C@]2(CO)CC[C@]3(C)C(=CCC4[C@@]5(C)CC[C@H](O)C(C)(C)C5CC[C@]43C)[C@@H]2[C@H]1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D07 compound treatment 144640.0 -1640.0 -0.11 150040.0 1580.0 0.12 0.0042 0.0257 867 BSPBio_003265 Nc1ccc(cc1)S(=O)(=O)Nc2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D08 compound treatment 148960.0 2680.0 0.18 148360.0 -101.0 -0.01 0.124 0.6775 957 BSPBio_003266 NC(COC(=O)C=[N+]=[N-])C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D09 compound treatment 148560.0 2280.0 0.16 151320.0 2860.0 0.21 0.2605 0.9882 1009654 BSPBio_003267 COc1ccc(cc1OC)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D10 compound treatment 144920.0 -1360.0 -0.09 153560.0 5100.0 0.38 0.2029 0.5194 2577 BSPBio_003268 OC(=O)c1nn(Cc2ccc(Cl)c(Cl)c2)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D11 compound treatment 159840.0 13600.0 0.92 163720.0 15300.0 1.14 1.4569 0.9948 2060316 BSPBio_003269 COc1c2C=CC(C)(C)Oc2cc3occ(c4ccc5OCOc5c4)c(=O)c13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D12 compound treatment 141240.0 -5040.0 -0.34 140880.0 -7580.0 -0.56 -0.6418 -0.9717 1000411 BSPBio_003270 CCCCCNC(=N)N/N=C/c1c[nH]c2ccc(OC)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D13 compound treatment 150000.0 3720.0 0.25 148560.0 99.0 0.01 0.1847 0.7273 3650215 BSPBio_003271 CC1(C)CC2/C(=C/C=C/[C@@](C)(O)CC[C@]21O)/CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D14 compound treatment 129800.0 -16500.0 -1.12 133320.0 -15100.0 -1.13 -1.5912 -1.0 3077177 BSPBio_003272 CC(=O)OCC(O)CC(=O)CCCCCCCCCCCC#C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D15 compound treatment 144120.0 -2160.0 -0.15 151400.0 2940.0 0.22 0.0507 0.1922 1050602 BSPBio_003273 COc1ccc(CC(=O)c2ccc(O)cc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D16 compound treatment 144320.0 -1960.0 -0.13 148160.0 -301.0 -0.02 -0.1102 -0.8144 1279 BSPBio_003274 N[C@@H]([C@@H]1CC(=NO1)Cl)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D17 compound treatment 157520.0 11200.0 0.77 162920.0 14500.0 1.08 1.3029 0.9862 1250 BSPBio_003275 COc1cc(C)c2c(=O)cc(oc2c1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D18 compound treatment 160000.0 13700.0 0.94 166400.0 17900.0 1.34 1.6056 0.9849 3173761 BSPBio_003276 N[C@@H](C(=O)N[C@H]1[C@H]2SCC(=C(N2C1=O)C(=O)O)Cl)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D19 compound treatment 148600.0 2320.0 0.16 146080.0 -2380.0 -0.18 -0.0133 -0.0561 1041649 BSPBio_003277 CC(C)c1ccc(C)c(C(=O)O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D20 compound treatment 144720.0 -1560.0 -0.11 148280.0 -181.0 -0.01 -0.0846 -0.7905 2060315 BSPBio_003278 C[N+]1(C)C[C@H](O)[C@@H](C1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D21 compound treatment 143880.0 -2400.0 -0.16 141760.0 -6700.0 -0.5 -0.4682 -0.8922 1547 BSPBio_003279 CN1C(=O)CN=C(c2ccccc2)c3cc(Cl)ccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D22 compound treatment 147800.0 1520.0 0.1 147920.0 -541.0 -0.04 0.0449 0.4035 3198650 BSPBio_003280 COc1cc(NS(=O)(=O)C)ccc1Cc2c3ccccc3nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D23 mock treatment 140200.0 -6080.0 -0.41 144560.0 -3900.0 -0.29 -0.4983 -0.9849 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 D24 mock treatment 136520.0 -9760.0 -0.67 137680.0 -10800.0 -0.8 -1.0378 -0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E01 mock treatment 148800.0 2520.0 0.17 151040.0 2580.0 0.19 0.2573 0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E02 mock treatment 148000.0 1720.0 0.12 153200.0 4740.0 0.35 0.3324 0.8943 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E03 compound treatment 169680.0 23400.0 1.6 175560.0 27100.0 2.02 2.5544 0.9933 2060432 BSPBio_003281 CC[C@@]1(O)C(=O)OCc2c1cc3-c4nc5ccc(O)cc5cc4Cn3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E04 compound treatment 151680.0 5400.0 0.37 152840.0 4380.0 0.33 0.4909 0.9981 1259 BSPBio_003282 CCc1nc(N)nc(N)c1c2ccc(Cl)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E05 compound treatment 152400.0 6120.0 0.42 152600.0 4140.0 0.31 0.513 0.9888 2060497 BSPBio_003283 CC(C)(O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)C#N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E06 compound treatment 153880.0 7600.0 0.52 156920.0 8460.0 0.63 0.8117 0.9953 3054523 BSPBio_003284 C[C@@H]1CC[C@@]2(CC[C@]3(C)C(=CCC4[C@@]5(C)CC[C@H](O)C(C)(C)C5CC[C@]43C)C2[C@H]1C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E07 compound treatment 263880.0 118000.0 8.02 276520.0 128000.0 9.53 12.4089 0.9963 1386109 BSPBio_003285 Oc1ccc2c(=O)c(O)c(oc2c1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E08 compound treatment 154680.0 8400.0 0.57 152760.0 4300.0 0.32 0.6313 0.9621 2565 BSPBio_003286 COC1=CC(=O)OC1(O)C(=C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E09 compound treatment 164520.0 18200.0 1.24 161840.0 13400.0 1.0 1.5835 0.9939 2060144 BSPBio_003287 COc1cccc(c1)c2cc(=O)c3cc(OC)ccc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E10 compound treatment 153000.0 6720.0 0.46 156080.0 7620.0 0.57 0.7251 0.9944 1506 BSPBio_003288 OCc1cc(=O)c(O)co1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E11 compound treatment 149120.0 2840.0 0.19 153640.0 5180.0 0.39 0.4096 0.9494 2060456 BSPBio_003289 C[C@@H]1CC(Cl)CC[C@H]1C(=O)OC(C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E12 compound treatment 161880.0 15600.0 1.06 158000.0 9540.0 0.71 1.2542 0.9807 2060349 BSPBio_003290 CCC[C@H]1CC2=C(C[C@@H](CC)CC3=C1C(=O)OC3=O)C(=O)OC2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E13 compound treatment 160560.0 14300.0 0.97 153520.0 5060.0 0.38 0.9548 0.9145 907120 BSPBio_003291 CC(N)C(=O)OC(C)(C)Cc1ccc(Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E14 compound treatment 156320.0 10000.0 0.68 154280.0 5820.0 0.43 0.7904 0.9756 1001994 BSPBio_003292 C[C@@H](N)[C@@H](O)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E15 compound treatment 157520.0 11200.0 0.77 155120.0 6660.0 0.5 0.8924 0.9777 2060459 BSPBio_003293 OC[C@H]1OC2[C@@H](Oc3nc(=N)ccn23)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E16 compound treatment 148120.0 1840.0 0.13 146280.0 -2180.0 -0.16 -0.026 -0.1265 1393 BSPBio_003294 CN(C)CCCN1c2ccccc2CCc3ccc(Cl)cc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E17 compound treatment 150920.0 4640.0 0.32 151640.0 3180.0 0.24 0.3911 0.9897 2060471 BSPBio_003295 C[C@H]1[C@H]2[C@H](OC1=O)[C@@H]3C(=CC(=O)C3=C(C)C[C@@H]2O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E18 compound treatment 156960.0 10700.0 0.73 156280.0 7820.0 0.58 0.9265 0.9938 1190 BSPBio_003296 Nc1c2C(O)CCCc2nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E19 compound treatment 152000.0 5720.0 0.39 153280.0 4820.0 0.36 0.5295 0.9991 3474314 BSPBio_003297 CN1CCCCC1C(=O)Nc2c(C)cccc2C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E20 compound treatment 158480.0 12200.0 0.83 157960.0 9500.0 0.71 1.0882 0.9967 1516 BSPBio_003298 Nc1c2CCCCc2nc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E21 compound treatment 154160.0 7880.0 0.54 153400.0 4940.0 0.37 0.6399 0.9828 1001314 BSPBio_003299 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]3O[C@H](C)C[C@@H]([C@H]3O)N(C)C)[C@](C)(O)C[C@@H](C)[C@@H]4N[C@@H](COCCOC)O[C@H]([C@H]4C)[C@]1(C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E22 compound treatment 148600.0 2320.0 0.16 153600.0 5140.0 0.38 0.3824 0.9238 3172849 BSPBio_003300 CN1CCC[C@H]1c2cccnc2.OC(C(O)C(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E23 mock treatment 145440.0 -838.0 -0.06 147560.0 -901.0 -0.07 -0.0878 -0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 E24 mock treatment 146480.0 203.0 0.01 141560.0 -6900.0 -0.51 -0.3534 -0.6879 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F01 mock treatment 148680.0 2400.0 0.16 148320.0 -141.0 -0.01 0.1084 0.6605 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F02 mock treatment 148960.0 2680.0 0.18 151960.0 3500.0 0.26 0.3135 0.985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F03 compound treatment 154040.0 7760.0 0.53 149760.0 1300.0 0.1 0.4426 0.8227 1573 BSPBio_003301 CCCC(C)C1(CC)C(=O)NC(=NC1=O)S 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F04 compound treatment 152280.0 6000.0 0.41 151400.0 2940.0 0.22 0.444 0.9569 1008 BSPBio_003302 OC1CCCCC1N2CCC(CC2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F05 compound treatment 156520.0 10200.0 0.7 157800.0 9340.0 0.7 0.9853 1.0 1570 BSPBio_003303 CCCC(C)C1(CC=C)C(=O)NC(=NC1=O)S 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F06 compound treatment 154080.0 7800.0 0.53 157920.0 9460.0 0.7 0.874 0.9904 3474312 BSPBio_003304 Cc1ccc(cc1)S(=O)(=O)NC(=O)NN2CC3CCCC3C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F07 compound treatment 154760.0 8480.0 0.58 158120.0 9660.0 0.72 0.9173 0.9942 1572 BSPBio_003305 CCCC(C)C1(CC)C(=O)NC(=NC1=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F08 compound treatment 152760.0 6480.0 0.44 154520.0 6060.0 0.45 0.6314 0.9999 2069347 BSPBio_003306 CCC1(Cc2ccccc2O1)C3=NCCN3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F09 compound treatment 162560.0 16300.0 1.11 162840.0 14400.0 1.07 1.5417 0.9998 3055245 BSPBio_003307 CCC[C@@H]1CCCCN1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F10 compound treatment 173720.0 27400.0 1.87 185360.0 36900.0 2.75 3.2649 0.9825 2118912 BSPBio_003308 Oc1ccc(/C=C/C(=O)c2ccccc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F11 compound treatment 149760.0 3480.0 0.24 153200.0 4740.0 0.35 0.4173 0.9814 1304 BSPBio_003309 ClC1=C(Cl)C2(Cl)C3C4CC(C5OC54)C3C1(Cl)C2(Cl)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F12 compound treatment 147800.0 1520.0 0.1 154520.0 6060.0 0.45 0.3923 0.8477 1014978 BSPBio_003310 OCC(O)C(O)C(O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F13 compound treatment 178640.0 32400.0 2.21 176240.0 27800.0 2.07 3.0221 0.9995 2069281 BSPBio_003311 C[C@@]12CCC3C(CCc4cc(OC(=O)c5ccccc5)ccc34)C2CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F14 compound treatment 177960.0 31700.0 2.16 178040.0 29600.0 2.2 3.084 1.0 1003115 BSPBio_003312 COc1cc(cc(OC)c1O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F15 compound treatment 169440.0 23200.0 1.58 175560.0 27100.0 2.02 2.5428 0.9927 2060499 BSPBio_003313 OC[C@H]1O[C@@H](Oc2cc(O)c3c(=O)cc(oc3c2)c4ccc(O)cc4)[C@H](O[C@@H]5OC[C@](O)(CO)[C@H]5O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F16 compound treatment 148800.0 2520.0 0.17 151560.0 3100.0 0.23 0.2847 0.9895 3104621 BSPBio_003314 CC[C@H]/1CC[C@H]2O[C@@]3(CC[C@@H](C)[C@@H](C[C@H](C)O)O3)[C@H](C)[C@@H](OC(=O)/C=C/[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@H](C)[C@H](O)[C@@H](C)C(=O)[C@@](C)(O)[C@H](O)[C@@H](C)C\C=C\C=C1)[C@H]2C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F17 compound treatment 154960.0 8680.0 0.59 151720.0 3260.0 0.24 0.5901 0.9224 1010 BSPBio_003315 COc1ccc(CN(CCN(C)C)c2ncccn2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F18 compound treatment 151120.0 4840.0 0.33 151160.0 2700.0 0.2 0.3755 0.9716 1113 BSPBio_003316 COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)OCC(=O)O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F19 compound treatment 166320.0 20000.0 1.37 158840.0 10400.0 0.77 1.5124 0.9635 3177324 BSPBio_003317 C[C@@]12CC(=O)C3C(CC[C@@H]4C[C@H](O)CC[C@@]43C)C2CC[C@]1(O)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F20 compound treatment 150920.0 4640.0 0.32 153560.0 5100.0 0.38 0.4922 0.9959 774 BSPBio_003318 OC(=O)C1=CCNCC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F21 compound treatment 148680.0 2400.0 0.16 153760.0 5300.0 0.39 0.3947 0.9242 2069306 BSPBio_003319 C[C@@]12CCC3C(CCC4=CC(=O)C=C[C@]34C)C2CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F22 compound treatment 145480.0 -798.0 -0.05 148280.0 -181.0 -0.01 -0.048 -0.8564 3081181 BSPBio_003320 C[C@H]1CCC2=C1C[C@@H](CC[C@@H]2C)C(C)(C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F23 mock treatment 154800.0 8520.0 0.58 146840.0 -1620.0 -0.12 0.3255 0.5486 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 F24 mock treatment 142600.0 -3680.0 -0.25 145480.0 -2980.0 -0.22 -0.3342 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G01 mock treatment 151880.0 5600.0 0.38 159600.0 11100.0 0.83 0.8563 0.9381 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G02 mock treatment 157520.0 11200.0 0.77 158040.0 9580.0 0.71 1.0461 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G03 compound treatment 159600.0 13300.0 0.91 157720.0 9260.0 0.69 1.1295 0.9907 2060476 BSPBio_003321 C[C@H]1[C@@H]2CCC(=C3[C@@H]([C@H]2OC1=O)C(=CC3=O)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G04 compound treatment 158960.0 12700.0 0.86 161480.0 13000.0 0.97 1.2966 0.9984 718 BSPBio_003322 Cn1c(=O)n(C)c2ncn(CCO)c2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G05 compound treatment 159200.0 12900.0 0.88 160840.0 12400.0 0.92 1.2745 0.9997 1089854 BSPBio_003323 Cc1ncc(CNC(=O)N(CCCl)N=O)c(N)n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G06 compound treatment 154080.0 7800.0 0.53 161040.0 12600.0 0.94 1.0382 0.9641 806 BSPBio_003324 OC(=O)C1CCCNC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G07 compound treatment 157960.0 11700.0 0.8 155200.0 6740.0 0.5 0.9179 0.9751 1765 BSPBio_003325 CC1(C)NC(=O)N(C1=O)c2ccc([N+](=O)[O-])c(c2)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G08 compound treatment 157840.0 11600.0 0.79 156800.0 8340.0 0.62 0.9963 0.993 1055442 BSPBio_003326 Nc1nc(O)c2nc(cnc2n1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G09 compound treatment 163880.0 17600.0 1.2 161960.0 13500.0 1.0 1.559 0.9961 1013144 BSPBio_003327 O=C1OC(=O)C2C3CCC(O3)C21 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G10 compound treatment 163440.0 17200.0 1.17 161400.0 12900.0 0.96 1.5083 0.9953 1464728 BSPBio_003328 Cn1c(=O)[nH]c2nc[nH]c2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G11 compound treatment 162840.0 16600.0 1.13 164200.0 15700.0 1.17 1.6268 0.9998 1734308 BSPBio_003329 Oc1cc(O)c2C(=O)C[C@H](Oc2c1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G12 compound treatment 157560.0 11300.0 0.77 155400.0 6940.0 0.52 0.9091 0.9812 370 BSPBio_003330 O=C1N(C2CCC(=O)NC2=O)C(=O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G13 compound treatment 167080.0 20800.0 1.42 160360.0 11900.0 0.89 1.6291 0.9743 3059440 BSPBio_003331 OC(=O)C1CC(CN2CCCCC12)[C@@H]3CCCCN3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G14 compound treatment 167560.0 21300.0 1.45 163880.0 15400.0 1.15 1.8375 0.9933 1049467 BSPBio_003332 COC(=O)c1c(C)cc(OC(=O)c2c(C)cc(O)c(C=O)c2O)c(C)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G15 compound treatment 167680.0 21400.0 1.46 163120.0 14700.0 1.09 1.8033 0.9897 1307902 BSPBio_003333 CN1CCCCC1c2ccc(nc2)c3cccnc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G16 compound treatment 161080.0 14800.0 1.01 157800.0 9340.0 0.7 1.2051 0.9834 986 BSPBio_003334 CN1CC(=O)NC1=N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G17 compound treatment 160920.0 14600.0 1.0 160000.0 11500.0 0.86 1.3132 0.9972 1216977 BSPBio_003335 CC1(C)Oc2ccc3ccc(=O)oc3c2CC1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G18 compound treatment 154280.0 8000.0 0.55 152360.0 3900.0 0.29 0.591 0.9563 1029490 BSPBio_003336 COc1cc(O)c(C)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G19 compound treatment 158520.0 12200.0 0.83 162680.0 14200.0 1.06 1.3385 0.9931 2060489 BSPBio_003337 C/C=C(/C)\C(=O)O[C@@H]1Cc2c(OC1(C)C)ccc3ccc(=O)oc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G20 compound treatment 158440.0 12200.0 0.83 158560.0 10100.0 0.75 1.1178 0.9988 1060118 BSPBio_003338 COc1cc(OC)c2c(=O)c(OC)c(oc2c1)c3ccc(OC)c(OC)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G21 compound treatment 162240.0 16000.0 1.09 156640.0 8180.0 0.61 1.2 0.9623 2060490 BSPBio_003339 C/C=C(\C)/C(=O)O[C@H]1[C@@H](OC(=O)C)C(C)(C)Oc2ccc3ccc(=O)oc3c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G22 compound treatment 155880.0 9600.0 0.65 154040.0 5580.0 0.42 0.7565 0.9759 1024489 BSPBio_003340 Cc1cc(O)cc(=O)o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G23 mock treatment 147280.0 1000.0 0.07 149520.0 1060.0 0.08 0.1041 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 G24 mock treatment 146840.0 563.0 0.04 147440.0 -1020.0 -0.08 -0.0266 -0.3127 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H01 mock treatment 154480.0 8200.0 0.56 148240.0 -221.0 -0.02 0.3838 0.686 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H02 mock treatment 153320.0 7040.0 0.48 154880.0 6420.0 0.48 0.6773 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H03 compound treatment 153200.0 6920.0 0.47 150760.0 2300.0 0.17 0.4547 0.9058 749 BSPBio_003341 NC(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H04 compound treatment 172840.0 26600.0 1.81 174360.0 25900.0 1.93 2.6435 0.9995 1275 BSPBio_003342 CC(=O)NCCc1c[nH]c2ccc(O)cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H05 compound treatment 157080.0 10800.0 0.74 167800.0 19300.0 1.44 1.5385 0.9516 3046992 BSPBio_003343 CO[C@]12[C@@H]3NC3CN2C4=C([C@@H]1COC(=O)N)C(=O)C(=C(C)C4=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H06 compound treatment 156400.0 10100.0 0.69 159880.0 11400.0 0.85 1.0889 0.9947 757 BSPBio_003344 OC(=O)c1cn(C2CC2)c3cc(N4CCNCC4)c(F)cc3c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H07 compound treatment 151400.0 5120.0 0.35 156320.0 7860.0 0.58 0.6606 0.9696 1000009 BSPBio_003345 C/C(=C\C=C\C(=C/C(=O)O)\C)/C=C/C1=C(C)CCCC1(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H08 compound treatment 154240.0 7960.0 0.54 155560.0 7100.0 0.53 0.7575 0.9999 1607 BSPBio_003346 CC[C@H](C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@@H]12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H09 compound treatment 156680.0 10400.0 0.71 159240.0 10800.0 0.8 1.0688 0.9981 3177651 BSPBio_003347 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N2[C@@H](C[C@@H]3CCC[C@@H]32)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H10 compound treatment 155160.0 8880.0 0.61 157840.0 9380.0 0.7 0.9218 0.9975 839 BSPBio_003348 Nc1nc2n(COCCO)cnc2c(=O)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H11 compound treatment 168880.0 22600.0 1.54 168800.0 20300.0 1.51 2.16 1.0 2060352 BSPBio_003349 O=C(O[C@H]1Cc2c(OC(=O)c3ccccc3)cc(OC(=O)c4ccccc4)cc2O[C@@H]1c5ccc(OC(=O)c6ccccc6)c(OC(=O)c7ccccc7)c5)c8ccccc8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H12 compound treatment 153360.0 7080.0 0.48 161200.0 12700.0 0.95 1.0119 0.951 3055308 BSPBio_003350 COC(=O)C1=CO[C@@H](O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)[C@@H]3[C@@H](C)[C@@H](O)C[C@@H]31 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H13 compound treatment 296480.0 150000.0 10.24 295040.0 147000.0 10.91 14.9551 0.9995 2060100 BSPBio_003351 OC(=O)c1cc(O)c(=O)c2c(O)c(O)ccc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H14 compound treatment 170160.0 23900.0 1.63 170600.0 22100.0 1.65 2.3165 1.0 1380 BSPBio_003352 NC(=O)c1ncn(n1)[C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H15 compound treatment 185520.0 39200.0 2.68 184680.0 36200.0 2.7 3.7979 1.0 3173763 BSPBio_003353 O[C@@H]1C[C@](O)(C[C@@H](OC(=O)/C=C/c2ccc(O)c(O)c2)[C@@H]1O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H16 compound treatment 160360.0 14100.0 0.96 163840.0 15400.0 1.14 1.4883 0.9962 2080198 BSPBio_003354 CC(=O)C1=C(O)C2C3C(Cc4cccc5[nH]cc3c45)C(C)(C)N2C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H17 compound treatment 153720.0 7440.0 0.51 158960.0 10500.0 0.78 0.9113 0.9781 2060377 BSPBio_003355 COc1c(ccc2OC(C)(C)CCc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H18 compound treatment 149960.0 3680.0 0.25 158880.0 10400.0 0.78 0.7259 0.8905 1537 BSPBio_003356 NC(Cc1ccc(F)cc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H19 compound treatment 148800.0 2520.0 0.17 153640.0 5180.0 0.39 0.3942 0.9339 2060217 BSPBio_003357 COc1c(ccc2OC(C)(C)CCc12)C3COc4cc5OC(C)(C)C(O)Cc5cc4C3=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H20 compound treatment 156560.0 10300.0 0.7 157200.0 8740.0 0.65 0.9556 0.9993 1672652 BSPBio_003358 COc1ccc(cc1)c2cc(=O)c3ccc(OC)cc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H21 compound treatment 422520.0 276000.0 18.83 419000.0 271000.0 20.14 27.5551 0.9994 2060169 BSPBio_003359 Oc1cc(O)c2C[C@@H](OC(=O)c3cc(O)c(O)c(O)c3)[C@H](Oc2c1)c4cc(O)c(O)c(O)c4c5c(O)c(O)c(O)cc5[C@H]6Oc7cc(O)cc(O)c7C[C@H]6OC(=O)c8cc(O)c(O)c(O)c8 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H22 compound treatment 147880.0 1600.0 0.11 153520.0 5060.0 0.38 0.3435 0.8761 790507 BSPBio_003360 OC(=O)CN1C(=O)c2cccc3cccc(C1=O)c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H23 mock treatment 146560.0 283.0 0.02 148840.0 379.0 0.03 0.0336 0.9827 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 H24 mock treatment 143240.0 -3040.0 -0.21 146680.0 -1780.0 -0.13 -0.2402 -0.9768 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I01 mock treatment 152120.0 5840.0 0.4 151880.0 3420.0 0.25 0.4616 0.9766 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I02 mock treatment 149880.0 3600.0 0.25 152240.0 3780.0 0.28 0.3726 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I03 compound treatment 155240.0 8960.0 0.61 157520.0 9060.0 0.67 0.9088 0.9988 2060491 BSPBio_003361 CC(C)CC(=O)O[C@@H]1[C@H](OC(=O)C)c2c(OC1(C)C)ccc3ccc(=O)oc23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I04 compound treatment 171560.0 25300.0 1.72 170280.0 21800.0 1.62 2.3671 0.9996 2060467 BSPBio_003362 COc1ccc2C(=O)/C(=C\c3ccc(OC)c(OC)c3)/COc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I05 compound treatment 163240.0 17000.0 1.16 165640.0 17200.0 1.28 1.7218 0.9987 3055383 BSPBio_003363 CC(C)(O)[C@@H]1Cc2cc3ccc(=O)oc3cc2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I06 compound treatment 169480.0 23200.0 1.58 173120.0 24700.0 1.84 2.4163 0.9973 2060448 BSPBio_003364 COc1ccc2[C@H](O)[C@H](Cc3ccc(OC)c(OC)c3)COc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I07 compound treatment 157400.0 11100.0 0.76 161280.0 12800.0 0.95 1.2108 0.9935 3055445 BSPBio_003365 CC(=O)OC(C)(C)[C@@H]1Cc2cc3ccc(=O)oc3cc2O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I08 compound treatment 190520.0 44200.0 3.02 197440.0 49000.0 3.65 4.7105 0.9956 2060258 BSPBio_003366 CC(=O)O[C@H]1Cc2c(OC(=O)C)cc(OC(=O)C)cc2O[C@@H]1c3ccc(OC(=O)C)c(OC(=O)C)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I09 compound treatment 169240.0 23000.0 1.57 173240.0 24800.0 1.84 2.411 0.9967 2060501 BSPBio_003367 CC(C)(OC(=O)c1ccccc1)[C@@H]2Cc3cc4ccc(=O)oc4cc3O2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I10 compound treatment 185800.0 39500.0 2.69 188440.0 40000.0 2.98 4.0093 0.9988 2060260 BSPBio_003368 COc1ccc(cc1)C2CC(=O)c3ccc(OC)cc3O2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I11 compound treatment 162840.0 16600.0 1.13 162200.0 13700.0 1.02 1.5215 0.9988 1023016 BSPBio_003369 COc1ccc2ccc(=O)oc2c1CC=C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I12 compound treatment 163520.0 17200.0 1.18 165960.0 17500.0 1.3 1.7522 0.9987 2060417 BSPBio_003370 CC(=C)C1Cc2c(O1)ccc(C(=O)O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I13 compound treatment 157560.0 11300.0 0.77 162800.0 14300.0 1.07 1.2985 0.9871 1296906 BSPBio_003371 COc1ccc(C(=O)CC(=O)O)c2OC(C)(C)C=Cc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I14 compound treatment 177840.0 31600.0 2.15 180240.0 31800.0 2.37 3.194 0.9989 791 BSPBio_003372 CC(C)Oc1ccc2c(=O)cc(oc2c1)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I15 compound treatment 161960.0 15700.0 1.07 165240.0 16800.0 1.25 1.6391 0.997 1204574 BSPBio_003373 COc1c(oc2cc3oc(=O)ccc3cc12)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I16 compound treatment 294360.0 148000.0 10.1 245640.0 97200.0 7.23 12.2531 0.9866 2069329 BSPBio_003374 COc1cc(O)c2c(=O)cc(oc2c1)c3ccc(OC)c(c3)c4c(O)cc(O)c5c(=O)cc(oc45)c6ccc(O)cc6 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I17 compound treatment 162720.0 16400.0 1.12 157640.0 9180.0 0.68 1.2757 0.9718 1095093 BSPBio_003375 CNCCC(Oc1ccc(cc1)C(F)(F)F)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I18 compound treatment 156200.0 9920.0 0.68 152640.0 4180.0 0.31 0.6983 0.9378 1192 BSPBio_003376 Cc1noc(NS(=O)(=O)c2ccc(N)cc2)c1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I19 compound treatment 159600.0 13300.0 0.91 164240.0 15800.0 1.17 1.4727 0.9919 1091368 BSPBio_003377 CNc1ccccc1C(=O)N2CCc3c([nH]c4ccccc34)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I20 compound treatment 154760.0 8480.0 0.58 156840.0 8380.0 0.62 0.8499 0.9993 1175 BSPBio_003378 Nc1ccc(cc1)S(=O)(=O)Nc2nccs2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I21 compound treatment 155960.0 9680.0 0.66 157160.0 8700.0 0.65 0.9246 1.0 2321 BSPBio_003379 COc1ccc2CC3N(CCc4cc(OC)c(OC)cc34)Cc2c1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I22 compound treatment 148200.0 1920.0 0.13 145760.0 -2700.0 -0.2 -0.0495 -0.2061 960 BSPBio_003380 C1N2CN3CN1CN(C2)C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I23 mock treatment 145440.0 -838.0 -0.06 145120.0 -3340.0 -0.25 -0.2162 -0.8474 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 I24 mock treatment 144560.0 -1720.0 -0.12 146560.0 -1900.0 -0.14 -0.1828 -0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J01 mock treatment 147400.0 1120.0 0.08 151480.0 3020.0 0.22 0.213 0.8973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J02 mock treatment 151600.0 5320.0 0.36 152400.0 3940.0 0.29 0.4639 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J03 compound treatment 158800.0 12500.0 0.85 156720.0 8260.0 0.61 1.0383 0.987 3045136 BSPBio_003381 CC[C@H](C)C(=O)O[C@H]1CCC=C2C=C[C@H](C)C(CCC3C[C@@H](O)CC(=O)O3)[C@@H]12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J04 compound treatment 160560.0 14300.0 0.97 161800.0 13300.0 0.99 1.3905 1.0 2060354 BSPBio_003382 COc1ccc(cc1)c2coc3cc(OC(=O)C)cc(OC(=O)C)c3c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J05 compound treatment 175680.0 29400.0 2.0 170320.0 21900.0 1.63 2.5678 0.9946 2060359 BSPBio_003383 COc1ccc(cc1)c2c(O)c3c(OC)c4C=CC(C)(C)Oc4cc3oc2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J06 compound treatment 286960.0 141000.0 9.59 271400.0 123000.0 9.15 13.2521 0.9997 360 BSPBio_003384 Oc1ccc(cc1)c2cc(=O)c3c(O)cc(O)cc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J07 compound treatment 158920.0 12600.0 0.86 157960.0 9500.0 0.71 1.1094 0.9952 2060284 BSPBio_003385 COc1cc(OC)c(c(OC)c1)c2c(OC)cc(OC)cc2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J08 compound treatment 170800.0 24500.0 1.67 173920.0 25500.0 1.89 2.522 0.9981 3077174 BSPBio_003386 CC(=O)Oc1ccc(cc1)c2cc(=O)c3c(OC(=O)C)cc(OC(=O)C)cc3o2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J09 compound treatment 166680.0 20400.0 1.39 172520.0 24100.0 1.79 2.2497 0.9922 2060302 BSPBio_003387 CC(C)CCC[C@@H](C)CCC[C@@H](C)CC/C(=C/CO)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J10 compound treatment 200000.0 53700.0 3.66 205240.0 56800.0 4.23 5.578 0.9975 1013706 BSPBio_003388 O=c1c2ccccc2oc3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J11 compound treatment 176800.0 30500.0 2.08 180560.0 32100.0 2.39 3.1607 0.9976 907381 BSPBio_003389 CC(=CCC/C(=C/C=C/C(=C/C=C/C(=C/C=C/C=C(\C)/C=C/C=C(\C)/C=C/C=C(\C)/CCC=C(C)C)/C)/C)/C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J12 compound treatment 175480.0 29200.0 1.99 179280.0 30800.0 2.29 3.0297 0.9975 3077175 BSPBio_003390 COc1ccc2C(=O)/C(=C\c3ccc(O)c(O)c3)/COc2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J13 compound treatment 158280.0 12000.0 0.82 160400.0 11900.0 0.89 1.2069 0.9992 1461 BSPBio_003391 CN1CCCN=C1COC(=O)C(O)(C2CCCCC2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J14 compound treatment 159240.0 13000.0 0.88 159280.0 10800.0 0.81 1.1943 0.9989 1045 BSPBio_003392 C[C@@H]1CC2C3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J15 compound treatment 156440.0 10200.0 0.69 158120.0 9660.0 0.72 0.9983 0.9998 3080396 BSPBio_003393 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)C(C)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J16 compound treatment 223200.0 76900.0 5.24 221840.0 73400.0 5.46 7.5701 0.9998 1000323 BSPBio_003394 N[C@@H](Cc1cc(I)c(Oc2ccc(O)c(I)c2)c(I)c1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J17 compound treatment 154480.0 8200.0 0.56 155560.0 7100.0 0.53 0.769 0.9996 1095029 BSPBio_003395 CCCCCCCCCCCCCCCCCCOP(=O)(O)OCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J18 compound treatment 165040.0 18800.0 1.28 163400.0 14900.0 1.11 1.6907 0.9976 810 BSPBio_003396 CCCCC[C@@H]1[C@@H](OC(=O)CC(C)C)[C@H](C)OC(=O)[C@@H](NC(=O)c2cccc(NC=O)c2O)[C@@H](C)OC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J19 compound treatment 176320.0 30000.0 2.05 175680.0 27200.0 2.03 2.8808 1.0 3176939 BSPBio_003397 ClCC(=O)[C@H](Cc1ccccc1)NC(=O)OCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J20 compound treatment 156040.0 9760.0 0.67 151240.0 2780.0 0.21 0.6169 0.8851 3198426 BSPBio_003398 NCC(CC(=O)O)c1ccc(Cl)s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J21 compound treatment 155400.0 9120.0 0.62 147600.0 -861.0 -0.06 0.3945 0.6309 3079212 BSPBio_003399 NCCCN.OC(C(O)C(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J22 compound treatment 149000.0 2720.0 0.19 151640.0 3180.0 0.24 0.2986 0.9928 1450 BSPBio_003400 NCCc1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J23 mock treatment 144480.0 -1800.0 -0.12 148120.0 -341.0 -0.03 -0.1046 -0.8358 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 J24 mock treatment 141520.0 -4760.0 -0.32 140320.0 -8140.0 -0.61 -0.6578 -0.9571 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K01 mock treatment 154880.0 8600.0 0.59 158080.0 9620.0 0.72 0.9209 0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K02 mock treatment 152840.0 6560.0 0.45 157960.0 9500.0 0.71 0.8163 0.9756 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K03 compound treatment 248680.0 102000.0 6.98 249360.0 101000.0 7.51 10.2467 0.9993 3172984 BSPBio_003401 COC(=O)[C@]1(C)CC[C@]2(C)CC[C@]3(C)C4=CC=C5C(=C(O)C(=O)C=C5[C@]4(C)CC[C@@]3(C)[C@@H]2C1)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K04 compound treatment 180960.0 34700.0 2.36 172560.0 24100.0 1.79 2.9403 0.9907 912 BSPBio_003402 CCCc1cc(=O)[nH]c(=S)[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K05 compound treatment 160680.0 14400.0 0.98 158520.0 10100.0 0.75 1.2237 0.991 3173234 BSPBio_003403 Cn1c(=O)[nH]c(=O)c2nc[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K06 compound treatment 164560.0 18300.0 1.25 170640.0 22200.0 1.65 2.0486 0.9904 967 BSPBio_003404 C/C(=C\C=C\C=C(/C)\C=C\C=C(/C)\C=C\C1=C(C)CCCC1(C)C)/C=C/C=C(\C)/C=C/C2=C(C)CCCC2(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K07 compound treatment 159680.0 13400.0 0.91 163840.0 15400.0 1.14 1.4555 0.9938 1001642 BSPBio_003405 OC[C@H]1OC(C[C@@H]1O)n2cc(c(=O)[nH]c2=O)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K08 compound treatment 159560.0 13300.0 0.91 158920.0 10500.0 0.78 1.1908 0.9972 471 BSPBio_003406 CCCC(CCC)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K09 compound treatment 159840.0 13600.0 0.92 163000.0 14500.0 1.08 1.419 0.9969 1015899 BSPBio_003407 NCC(=O)CCC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K10 compound treatment 161680.0 15400.0 1.05 169320.0 20900.0 1.55 1.8403 0.9819 2060105 BSPBio_003408 CC1(C)Oc2cc3occ(c4ccc5OCOc5c4)c(=O)c3c(O)c2C=C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K11 compound treatment 156400.0 10100.0 0.69 159360.0 10900.0 0.81 1.0616 0.9968 907463 BSPBio_003409 Cc1nc2ccccn2c(=O)c1CCN3CCC(CC3)C(=O)c4ccc(F)cc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K12 compound treatment 175520.0 29200.0 1.99 168720.0 20300.0 1.51 2.4759 0.9905 1213 BSPBio_003410 CNCCc1ccccn1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K13 compound treatment 225240.0 79000.0 5.38 224520.0 76100.0 5.66 7.8095 0.9997 831758 BSPBio_003411 Oc1ccc(/C=C/C(=O)c2ccc(O)cc2O)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K14 compound treatment 163200.0 16900.0 1.15 157640.0 9180.0 0.68 1.2989 0.9687 89599 BSPBio_003412 OC(=O)c1cc(O)c2c(Cl)cc(Cl)cc2n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K15 compound treatment 163280.0 17000.0 1.16 159360.0 10900.0 0.81 1.3933 0.9848 2060386 BSPBio_003413 CCN1C[C@]2(C)CC[C@H](OC)[C@@]34C2[C@H](O)[C@]5(OCO[C@]65C[C@H](OC)[C@H]7C[C@]4(O)C6[C@H]7O)C13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K16 compound treatment 166240.0 20000.0 1.36 163880.0 15400.0 1.15 1.7738 0.9964 831 BSPBio_003414 Nc1nccs1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K17 compound treatment 220880.0 74600.0 5.09 216200.0 67700.0 5.04 7.1614 1.0 3055171 BSPBio_003415 COC(=O)[C@]1(C)CC[C@]2(C)CC[C@]3(C)C4=CCc5c(C)c(O)c(O)cc5[C@]4(C)CC[C@@]3(C)C2C1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K18 compound treatment 160160.0 13900.0 0.95 157560.0 9100.0 0.68 1.1481 0.9865 1202 BSPBio_003416 COc1ccc2CN(C)CC[C@]34C=C[C@H](O)C[C@@H]4Oc1c23 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K19 compound treatment 155800.0 9520.0 0.65 154280.0 5820.0 0.43 0.7653 0.9806 4480 BSPBio_003417 CC(C)NC(=N)NC(=N)Nc1ccc(Cl)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K20 compound treatment 163600.0 17300.0 1.18 158120.0 9660.0 0.72 1.3434 0.9717 3198647 BSPBio_003418 CC1(C)[C@H](O)C[C@H](O)[C@@]2(C)C1CC(=O)[C@]3(C)C2CC[C@@]4(C)[C@@H](OC(=O)C=C43)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K21 compound treatment 361760.0 215000.0 14.69 348040.0 200000.0 14.85 20.8915 1.0 1010201 BSPBio_003419 ClC1=C(Cl)C(=O)C(=C(Cl)C1=O)Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K22 compound treatment 156960.0 10700.0 0.73 153320.0 4860.0 0.36 0.7707 0.9478 3045298 BSPBio_003420 C[C@@H]1CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K23 mock treatment 145800.0 -478.0 -0.03 150960.0 2500.0 0.19 0.1085 0.5746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 K24 mock treatment 144920.0 -1360.0 -0.09 145640.0 -2820.0 -0.21 -0.2139 -0.9323 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L01 mock treatment 147800.0 1520.0 0.1 153400.0 4940.0 0.37 0.3333 0.8727 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L02 mock treatment 148400.0 2120.0 0.14 152400.0 3940.0 0.29 0.3096 0.947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L03 compound treatment 152040.0 5760.0 0.39 157800.0 9340.0 0.7 0.7693 0.9635 3079213 BSPBio_003421 N[C@@H](CCC(=O)N[C@@H](CCSC(CC(=O)O)C(=O)O)C(=O)NCC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L04 compound treatment 157720.0 11400.0 0.78 156040.0 7580.0 0.56 0.9505 0.9873 1526 BSPBio_003422 CC1CCCC(C)N1NC(=O)c2ccc(Cl)c(c2)S(=O)(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L05 compound treatment 153000.0 6720.0 0.46 152600.0 4140.0 0.31 0.5419 0.9813 3198431 BSPBio_003423 CC(C)[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L06 compound treatment 158840.0 12600.0 0.86 157640.0 9180.0 0.68 1.0887 0.9937 1835 BSPBio_003424 CCCc1nn(C)c2c(=O)[nH]c(nc12)c3cc(ccc3OCC)S(=O)(=O)N4CCN(C)CC4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L07 compound treatment 156040.0 9760.0 0.67 157400.0 8940.0 0.67 0.9411 1.0 3198435 BSPBio_003425 N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L08 compound treatment 174040.0 27800.0 1.89 170320.0 21900.0 1.63 2.4888 0.9972 3173357 BSPBio_003426 CC(=C)[C@@H]1CC[C@@]2(CCC3[C@H](CCC4[C@@]3(C)CCC5C(C)(C)[C@H](O)CC[C@@]54C)C12)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L09 compound treatment 156640.0 10400.0 0.71 158400.0 9940.0 0.74 1.0226 0.9997 3198434 BSPBio_003427 NCCCC[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L10 compound treatment 157000.0 10700.0 0.73 160840.0 12400.0 0.92 1.1684 0.9934 1493 BSPBio_003428 CCC(=O)O[C@@]1([C@@H](C)CC2C3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C)C(=O)CCl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L11 compound treatment 148880.0 2600.0 0.18 150080.0 1620.0 0.12 0.2107 0.9822 1000377 BSPBio_003429 CC(C)c1nc(nc(c1/C=C/[C@@H](O)C[C@@H](O)CC(=O)O)c2ccc(F)cc2)N(C)S(=O)(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L12 compound treatment 154640.0 8360.0 0.57 153320.0 4860.0 0.36 0.6589 0.9759 1431 BSPBio_003430 Clc1ccc(cc1)C(OCCN2CCCCC2)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L13 compound treatment 157320.0 11000.0 0.75 162440.0 14000.0 1.04 1.268 0.9874 1032444 BSPBio_003431 CC(=O)Oc1c(C)cccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L14 compound treatment 160160.0 13900.0 0.95 161360.0 12900.0 0.96 1.3481 1.0 2060453 BSPBio_003432 Clc1c(Cl)c(C#N)c(Cl)c(C#N)c1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L15 compound treatment 175120.0 28800.0 1.97 176760.0 28300.0 2.11 2.8798 0.9994 3079222 BSPBio_003433 CC(=O)OC[C@H]1O[C@@H](Oc2cc(OC(=O)C)c3c(=O)cc(oc3c2)c4ccc(OC(=O)C)cc4)[C@H](OC(=O)C)[C@@H](OC(=O)C)[C@@H]1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L16 compound treatment 113240.0 -33000.0 -2.25 112640.0 -35800.0 -2.67 -3.4779 -0.9965 1419 BSPBio_003434 NCCSSCCN 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L17 compound treatment 170800.0 24500.0 1.67 172080.0 23600.0 1.76 2.4252 0.9997 3079224 BSPBio_003435 COC1=C(O)C(=O)c2c(O)c3c(O)c(oc3cc2C1=O)C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L18 compound treatment 185440.0 39200.0 2.67 180320.0 31900.0 2.37 3.5646 0.9982 1000697 BSPBio_003436 COc1cc(cc(OC)c1O)[C@H]2[C@@H]3C(COC3=O)C(O[C@@H]4O[C@@H]5CO[C@H](OC5[C@H](O)[C@H]4O)c6cccs6)c7cc8OCOc8cc27 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L19 compound treatment 171960.0 25700.0 1.75 172720.0 24300.0 1.81 2.5148 0.9999 3078331 BSPBio_003437 OC(=O)c1cccc(O)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L20 compound treatment 162800.0 16500.0 1.13 167080.0 18600.0 1.39 1.7764 0.9947 2060442 BSPBio_003438 CCC(N)C(O)c1ccc(O)c(O)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L21 compound treatment 151360.0 5080.0 0.35 153760.0 5300.0 0.39 0.5239 0.9979 1331 BSPBio_003439 CC(=O)CCCCn1c(=O)n(C)c2ncn(C)c2c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L22 compound treatment 145280.0 -998.0 -0.07 152000.0 3540.0 0.26 0.1382 0.5079 1316 BSPBio_003440 CC(C)(C)NCC(O)c1ccccc1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L23 mock treatment 144400.0 -1880.0 -0.13 148240.0 -221.0 -0.02 -0.1021 -0.7914 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 L24 mock treatment 141280.0 -5000.0 -0.34 145280.0 -3180.0 -0.24 -0.4083 -0.9842 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M01 mock treatment 151720.0 5440.0 0.37 157480.0 9020.0 0.67 0.737 0.9609 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M02 mock treatment 153120.0 6840.0 0.47 157360.0 8900.0 0.66 0.7982 0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M03 compound treatment 153360.0 7080.0 0.48 158200.0 9740.0 0.72 0.854 0.9805 2060483 BSPBio_003441 CC(=O)N[C@@H](CC(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M04 compound treatment 158800.0 12500.0 0.85 163320.0 14900.0 1.11 1.3857 0.9918 944 BSPBio_003442 Nc1ccc(cc1)S(=O)(=O)Nc2ccnn2c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M05 compound treatment 169360.0 23100.0 1.57 175240.0 26800.0 1.99 2.5221 0.9932 907181 BSPBio_003443 NC(=N)NC(=O)c1nc(Cl)c(nc1N)N2CCCCCC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M06 compound treatment 154440.0 8160.0 0.56 156000.0 7540.0 0.56 0.7903 1.0 1401 BSPBio_003444 CN(C)CCCN1c2ccccc2Sc3ccc(cc13)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M07 compound treatment 215560.0 69300.0 4.72 221760.0 73300.0 5.46 7.1976 0.9974 3173242 BSPBio_003445 Nc1nc2cc(Cl)ccc2o1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M08 compound treatment 159240.0 13000.0 0.88 163640.0 15200.0 1.13 1.4237 0.9926 930 BSPBio_003446 CC(CN1CCCCC1)C(=O)c2ccc(C)cc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M09 compound treatment 163560.0 17300.0 1.18 167240.0 18800.0 1.4 1.8215 0.9964 1002855 BSPBio_003447 CCC(C(=O)O)c1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M10 compound treatment 170920.0 24600.0 1.68 168320.0 19900.0 1.48 2.2331 0.998 3173213 BSPBio_003448 COc1ccc(C[C@H](N)C(=O)N[C@H]2[C@@H](O)C(O[C@@H]2CO)n3cnc4c(ncnc34)N(C)C)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M11 compound treatment 192560.0 46300.0 3.16 201000.0 52500.0 3.91 4.9962 0.9943 2060416 BSPBio_003449 Sc1nc2ccccc2s1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M12 compound treatment 158160.0 11900.0 0.81 168200.0 19700.0 1.47 1.6117 0.9607 1000122 BSPBio_003450 O[C@@H]([C@@H]1C[C@@H]2CCN1C[C@@H]2C=C)c3ccnc4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M13 compound treatment 169680.0 23400.0 1.6 160960.0 12500.0 0.93 1.786 0.967 1001451 BSPBio_003451 Cc1cc(C)cc(OCC2CNC(=O)O2)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M14 compound treatment 162280.0 16000.0 1.09 158320.0 9860.0 0.73 1.2903 0.9814 1462 BSPBio_003452 CC1C(CCC(C)(C)N1C)OC(=O)C(O)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M15 compound treatment 163120.0 16800.0 1.15 158680.0 10200.0 0.76 1.3498 0.98 3172732 BSPBio_003453 CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]3O[C@H](C)C[C@@H]([C@H]3O)N(C)C)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M16 compound treatment 159240.0 13000.0 0.88 165640.0 17200.0 1.28 1.529 0.9837 3177385 BSPBio_003454 CC1(C)O[C@@H]2CC3C4C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M17 compound treatment 187160.0 40900.0 2.79 187720.0 39300.0 2.92 4.037 0.9997 2060378 BSPBio_003455 Oc1nc2cc(Cl)c(Cl)cc2nc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M18 compound treatment 153920.0 7640.0 0.52 156120.0 7660.0 0.57 0.7715 0.999 1302 BSPBio_003456 CC(C)CC1N2C(=O)[C@](NC(=O)C3CN(C)[C@@H]4Cc5c(Br)[nH]c6cccc(C4=C3)c56)(OC2(O)[C@@H]7CCCN7C1=O)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M19 compound treatment 155120.0 8840.0 0.6 156480.0 8020.0 0.6 0.8483 1.0 1001496 BSPBio_003457 NC(=O)N1c2ccccc2CC(=O)c3ccccc13 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M20 compound treatment 165800.0 19500.0 1.33 167320.0 18900.0 1.4 1.9337 0.9996 1000054 BSPBio_003458 CC(C)CC1NC(=O)C(CCCN)NC(=O)C(NC(=O)C2CCCN2C(=O)C(Cc3ccccc3)NC(=O)C(CC(C)C)NC(=O)C(CCCN)NC(=O)C(NC(=O)C4CCCN4C(=O)C(Cc5ccccc5)NC1=O)C(C)C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M21 compound treatment 174160.0 27900.0 1.9 183360.0 34900.0 2.6 3.1808 0.9882 3059445 BSPBio_003459 CCCCCCCCCCC[C@@H](C[C@H]1OC(=O)[C@H]1CCCCCC)OC(=O)[C@@H](CC(C)C)NC=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M22 compound treatment 149600.0 3320.0 0.23 152640.0 4180.0 0.31 0.3801 0.9879 1021 BSPBio_003460 CO[C@@H]1[C@@H](O)[C@H](C)O[C@@H](O[C@H]2CC[C@@]3(C)[C@H](CCC4C3CC[C@]5(C)C(CC[C@]45O)C6=CC(=O)OC6)C2)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M23 mock treatment 146760.0 483.0 0.03 149480.0 1020.0 0.08 0.0769 0.9301 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 M24 mock treatment 147800.0 1520.0 0.1 147560.0 -901.0 -0.07 0.026 0.2103 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N01 mock treatment 153720.0 7440.0 0.51 156680.0 8220.0 0.61 0.7913 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N02 mock treatment 154000.0 7720.0 0.53 159720.0 11300.0 0.84 0.9648 0.9749 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N03 compound treatment 193080.0 46800.0 3.19 202520.0 54100.0 4.02 5.1013 0.9934 2269 BSPBio_003461 Oc1ccc(/C=C/c2cc(O)cc(O)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N04 compound treatment 154800.0 8520.0 0.58 166080.0 17600.0 1.31 1.3381 0.9329 3045655 BSPBio_003462 CC(=O)[C@@]1(O)CCC2C3C=C(Cl)C4=CC(=O)[C@@H]5CC5[C@]4(C)C3CC[C@@]21C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N05 compound treatment 167560.0 21300.0 1.45 175880.0 27400.0 2.04 2.469 0.986 2060255 BSPBio_003463 CC(=O)Oc1ccc(/C=C/c2cc(OC(=O)C)cc(OC(=O)C)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N06 compound treatment 156600.0 10300.0 0.7 159720.0 11300.0 0.84 1.0902 0.9962 1510 BSPBio_003464 CN(C)CCN(Cc1cccs1)c2ccccn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N07 compound treatment 164880.0 18600.0 1.27 167480.0 19000.0 1.42 1.8977 0.9985 3103678 BSPBio_003465 N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)/NCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N08 compound treatment 169600.0 23300.0 1.59 173000.0 24500.0 1.83 2.4158 0.9976 2060303 BSPBio_003466 Cc1occc(=O)c1/C=C/O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N09 compound treatment 158840.0 12600.0 0.86 161280.0 12800.0 0.95 1.2803 0.9985 1494 BSPBio_003467 C1CN(CCN1)c2ccc3ccccc3n2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N10 compound treatment 161560.0 15300.0 1.04 172800.0 24300.0 1.81 2.0177 0.9655 3060195 BSPBio_003468 COC(C)(C)CCC[C@H](C)C/C=C/C(=C/C(=O)OC(C)C)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N11 compound treatment 161640.0 15400.0 1.05 164200.0 15700.0 1.17 1.5689 0.9984 1002022 BSPBio_003469 NC(CCC(=O)O)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N12 compound treatment 162800.0 16500.0 1.13 160040.0 11600.0 0.86 1.4059 0.9913 1489 BSPBio_003470 CCCNCC(O)COc1ccccc1C(=O)CCc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N13 compound treatment 158760.0 12500.0 0.85 163960.0 15500.0 1.15 1.4174 0.9888 2270 BSPBio_003471 CCCCOc1cc(CC2CNC(=O)N2)ccc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N14 compound treatment 156520.0 10200.0 0.7 162680.0 14200.0 1.06 1.2421 0.9796 1442 BSPBio_003472 CC(=O)NC1SCCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N15 compound treatment 154320.0 8040.0 0.55 160400.0 11900.0 0.89 1.016 0.9731 3173760 BSPBio_003473 COc1cc2CCN(C)[C@@H]3Cc4cccc(Oc5ccc(C[C@@H]6N(C)CCc7cc(OC)c(Oc(c1OC)c32)cc67)c(O)c5)c4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N16 compound treatment 152760.0 6480.0 0.44 155840.0 7380.0 0.55 0.7009 0.9942 1507 BSPBio_003474 CC(N)CCCC(C)(C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N17 compound treatment 154240.0 7960.0 0.54 162040.0 13600.0 1.01 1.0985 0.9575 417 BSPBio_003475 CN1CCN(CC1)C2=Nc3cc(Cl)ccc3Nc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N18 compound treatment 152920.0 6640.0 0.45 153680.0 5220.0 0.39 0.5949 0.9971 1524 BSPBio_003476 CC(C)Nc1c(C)n(C)n(c2ccccc2)c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N19 compound treatment 168840.0 22600.0 1.54 168000.0 19500.0 1.45 2.116 0.9996 1090658 BSPBio_003477 COc1cc(O)c2C(=O)c3c(O)cc(C)cc3C(=O)c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N20 compound treatment 153240.0 6960.0 0.47 153680.0 5220.0 0.39 0.6103 0.995 860 BSPBio_003478 CN(C)C(=O)Oc1ccc[n+](C)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N21 compound treatment 147240.0 963.0 0.07 151320.0 2860.0 0.21 0.1969 0.8841 4362 BSPBio_003479 CN1CCN(CC1)C2=Nc3ccccc3Oc4ccc(Cl)cc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N22 compound treatment 226360.0 80100.0 5.46 229880.0 81400.0 6.06 8.1455 0.9986 2060342 BSPBio_003480 O[C@@H]1[C@H](Oc2cc(O)ccc2C1=O)c3cc(O)c(O)c(O)c3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N23 mock treatment 145760.0 -518.0 -0.04 148480.0 19.0 0.0 -0.0239 -0.6781 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 N24 mock treatment 145880.0 -398.0 -0.03 146560.0 -1900.0 -0.14 -0.1192 -0.8275 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O01 mock treatment 151600.0 5320.0 0.36 155640.0 7180.0 0.53 0.6344 0.9822 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O02 mock treatment 152960.0 6680.0 0.46 157400.0 8940.0 0.67 0.7926 0.9829 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O03 compound treatment 162720.0 16400.0 1.12 167760.0 19300.0 1.44 1.8083 0.9925 2069291 BSPBio_003481 COc1cc(cc(OC)c1OC)[C@H]2[C@H]3[C@H](COC3=O)[C@@H](O)c4cc5OCOc5cc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O04 compound treatment 153040.0 6760.0 0.46 148920.0 459.0 0.03 0.3502 0.7574 1318 BSPBio_003482 CN(C(=O)CN(CCO)CC(=O)N(C)C(C)(C)Cc1ccccc1)C(C)(C)Cc2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O05 compound treatment 182880.0 36600.0 2.5 171400.0 22900.0 1.71 2.9718 0.9829 3177591 BSPBio_003483 COc1cc(cc(OC)c1OC)[C@H]2[C@@H]3[C@H](COC3=O)[C@@H](OC(=O)C)c4cc5OCOc5cc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O06 compound treatment 156400.0 10100.0 0.69 158400.0 9940.0 0.74 1.0111 0.9994 3198648 BSPBio_003484 CC(CCC(=O)O)[C@H]1CCC2C3CC=C4C[C@@H](O)CC[C@]4(C)C3CC[C@]12C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O07 compound treatment 162440.0 16200.0 1.1 160000.0 11500.0 0.86 1.3864 0.9924 3060196 BSPBio_003485 COc1c(CN2CC[C@@H]3CCCN[C@@H]3C2)c(F)cc4c(=O)c(cn(C5CC5)c14)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O08 compound treatment 274320.0 128000.0 8.73 267040.0 119000.0 8.83 12.4133 1.0 996 BSPBio_003486 NCCc1cc(O)c(O)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O09 compound treatment 160080.0 13800.0 0.94 153720.0 5260.0 0.39 0.9422 0.9244 1000322 BSPBio_003487 CCOC(=O)[C@H](CCc1ccccc1)N[C@H]2CCc3ccccc3N(CC(=O)O)C2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O10 compound treatment 154600.0 8320.0 0.57 159600.0 11100.0 0.83 0.9874 0.9829 2060458 BSPBio_003488 CC(=O)Oc1cccc(C(=O)O)c1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O11 compound treatment 161960.0 15700.0 1.07 168440.0 20000.0 1.49 1.8075 0.9869 1696 BSPBio_003489 CC(=O)OCC(CCn1cnc2cnc(N)nc12)COC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O12 compound treatment 157400.0 11100.0 0.76 155920.0 7460.0 0.56 0.9288 0.9882 1421 BSPBio_003490 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O13 compound treatment 160040.0 13800.0 0.94 159960.0 11500.0 0.86 1.2686 0.9989 1001491 BSPBio_003491 CCCc1nc(c(C(=O)OCc2oc(=O)oc2C)n1Cc3ccc(cc3)c4ccccc4c5nn[nH]n5)C(C)(C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O14 compound treatment 157080.0 10800.0 0.74 154120.0 5660.0 0.42 0.8186 0.9649 2060310 BSPBio_003492 CC(C)C1=CC2=CC[C@H]3[C@](C)(CO)CCC[C@]3(C)C2CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O15 compound treatment 155960.0 9680.0 0.66 159640.0 11200.0 0.83 1.0551 0.9934 3198315 BSPBio_003493 COc1ccc(cc1F)c2cc(nn2c3ccc(cc3)S(=O)(=O)N)C(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O16 compound treatment 153680.0 7400.0 0.5 157160.0 8700.0 0.65 0.8147 0.9924 857 BSPBio_003494 O=C(OCc1ccccc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O17 compound treatment 156440.0 10200.0 0.69 159680.0 11200.0 0.83 1.0804 0.9957 1592184 BSPBio_003495 O=C1CCCC2C3CC(CN21)[C@@H]4CCCCN4C3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O18 compound treatment 152680.0 6400.0 0.44 157600.0 9140.0 0.68 0.7896 0.977 3177322 BSPBio_003496 CC(=O)[C@@]1(O)CCC2C3CCC4=CC(=O)CC[C@]4(C)C3CC[C@@]21C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O19 compound treatment 150520.0 4240.0 0.29 155720.0 7260.0 0.54 0.5866 0.9571 3198437 BSPBio_003497 C[N+](C)(C)CCOP(=O)(O)OP(=O)(O)OC[C@H]1OC([C@H](O)[C@@H]1O)n2ccc(N)nc2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O20 compound treatment 151640.0 5360.0 0.37 150640.0 2180.0 0.16 0.3732 0.9331 3173755 BSPBio_003498 C[C@@]12CC(=O)C3C(CCC4=CC(=O)CC[C@]34C)C2CC[C@]1(O)C(=O)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O21 compound treatment 188480.0 42200.0 2.88 189560.0 41100.0 3.06 4.1975 0.9995 1005991 BSPBio_003499 O=C1c2ccccc2-c3cccc4cccc1c34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O22 compound treatment 141840.0 -4440.0 -0.3 143840.0 -4620.0 -0.34 -0.4571 -0.998 3081177 BSPBio_003500 CC(C)CCCC(C)C1CCC2C3C(CC[C@]12C)[C@@]4(C)CC[C@@H](CC4=CC3=O)OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O23 mock treatment 143880.0 -2400.0 -0.16 144240.0 -4220.0 -0.31 -0.3377 -0.9537 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 O24 mock treatment 144200.0 -2080.0 -0.14 142120.0 -6340.0 -0.47 -0.4339 -0.8805 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P01 mock treatment 153760.0 7480.0 0.51 154960.0 6500.0 0.48 0.7027 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P02 mock treatment 151680.0 5400.0 0.37 154240.0 5780.0 0.43 0.5646 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P03 compound treatment 153400.0 7120.0 0.49 154200.0 5740.0 0.43 0.6454 0.998 3059817 BSPBio_003501 CCCCC(=O)N(Cc1ccc(cc1)c2ccccc2c3nn[nH]n3)[C@@H](C(C)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P04 compound treatment 153040.0 6760.0 0.46 156240.0 7780.0 0.58 0.7354 0.9936 2060318 BSPBio_003502 C/C(=C\C=C\C=C(/C)\C=C\C=C(/C)\C=C\[C@]12O[C@]2(C)C[C@@H](O)CC1(C)C)/C=C/C=C(\C)/C=C/C3=C(C)C[C@@H](O)CC3(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P05 compound treatment 152960.0 6680.0 0.46 153440.0 4980.0 0.37 0.5842 0.9947 1001638 BSPBio_003503 CC(C)NC(=O)NS(=O)(=O)c1cnccc1Nc2cccc(C)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P06 compound treatment 154600.0 8320.0 0.57 156480.0 8020.0 0.6 0.8232 0.9997 1605 BSPBio_003504 OC(Cn1cncn1)(Cn2cncn2)c3ccc(F)cc3F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P07 compound treatment 149640.0 3360.0 0.23 156920.0 8460.0 0.63 0.6073 0.9064 2060333 BSPBio_003505 COc1ccc(/C=C/c2cc(O)cc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P08 compound treatment 157640.0 11400.0 0.77 160920.0 12500.0 0.93 1.2035 0.996 3616563 BSPBio_003506 C[C@H](N)[C@H](O)c1cccc(O)c1.O[C@H]([C@@H](O)C(=O)O)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P09 compound treatment 156120.0 9840.0 0.67 156200.0 7740.0 0.58 0.8818 0.9971 2971 BSPBio_003507 CCCn1cnc2n(C)c(=O)n(CCCCC(=O)C)c(=O)c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P10 compound treatment 161320.0 15000.0 1.03 166760.0 18300.0 1.36 1.6882 0.9902 3069629 BSPBio_003508 CC(=O)/N=c/1\sc(nn1C)S(=O)(=O)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P11 compound treatment 155840.0 9560.0 0.65 156720.0 8260.0 0.61 0.8956 0.9996 1439 BSPBio_003509 CSCCC(N)C(=O)NC(CC(C)C)C(=O)NC(Cc1ccccc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P12 compound treatment 159120.0 12800.0 0.88 156720.0 8260.0 0.61 1.0538 0.985 1457 BSPBio_003510 CC(=O)OCC(=O)[C@]12OC3(CCCC3)O[C@@H]2CC4C5CCC6=CC(=O)C=C[C@]6(C)[C@@]5(F)[C@@H](O)C[C@@]41C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P13 compound treatment 153400.0 7120.0 0.49 160280.0 11800.0 0.88 0.9654 0.9608 1434 BSPBio_003511 CN1CCN2C(C1)c3ccccc3Cc4ccccc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P14 compound treatment 433000.0 287000.0 19.55 434000.0 286000.0 21.25 28.8497 0.9991 3081192 BSPBio_003512 CC(=O)OC1Cc2c(OC(=O)C)cc(OC(=O)C)cc2O[C@@H]1c3cc(OC(=O)C)c(OC(=O)C)c4c(=O)c(OC(=O)C)cc(cc34)[C@H]5Oc6cc(OC(=O)C)cc(OC(=O)C)c6C[C@H]5OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P15 compound treatment 141960.0 -4320.0 -0.29 147440.0 -1020.0 -0.08 -0.2619 -0.8614 3174224 BSPBio_003513 CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C2=O)c4c(O)c(\C=N/N5CCN(C)CC5)c(NC(=O)/C(=C\C=C\C(C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@@H](OC(=O)C)[C@@H]1C)/C)c(O)c4c(O)c3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P16 compound treatment 147520.0 1240.0 0.08 152040.0 3580.0 0.27 0.2483 0.8881 3174220 BSPBio_003514 CO[C@@H]1C[C@@H](C[C@H]2CC[C@H](C)[C@@H](O2)[C@@H](C)C(=O)O)O[C@]3(O[C@@](C)(C[C@H]3C)[C@H]4CC[C@](C)(O4)C5O[C@H](C[C@@H]5C)C6O[C@@](O)(CO)[C@H](C)C[C@@H]6C)[C@@H]1C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P17 compound treatment 149880.0 3600.0 0.25 152960.0 4500.0 0.33 0.4104 0.9884 3198954 BSPBio_003515 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@H]1C(=O)N[C@@H]([C@@H](C)CC)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P18 compound treatment 150360.0 4080.0 0.28 158440.0 9980.0 0.74 0.722 0.9103 191 BSPBio_003516 CCCc1c(O)c(ccc1OCCCCc2nnn[nH]2)C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P19 compound treatment 153240.0 6960.0 0.47 160040.0 11600.0 0.86 0.945 0.9605 907526 BSPBio_003517 CN1CCN(CC(=O)N2c3c(C)scc3C(=O)Nc4ccccc24)CC1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P20 compound treatment 184360.0 38100.0 2.6 202840.0 54400.0 4.05 4.6977 0.977 3173485 BSPBio_003518 OC[C@H]1O[C@H](Oc2cccc3[C@H]([C@@H]4c5cccc(O[C@H]6O[C@H](CO)[C@@H](O)[C@H](O)[C@H]6O)c5C(=O)c7c(O)cc(cc47)C(=O)O)c8cc(cc(O)c8C(=O)c23)C(=O)O)[C@H](O)[C@@H](O)[C@@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P21 compound treatment 153240.0 6960.0 0.47 156800.0 8340.0 0.62 0.7745 0.9912 3081180 BSPBio_003519 CN1[C@@H]2CC[C@@H]1CC(O)C2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P22 compound treatment 145840.0 -438.0 -0.03 151800.0 3340.0 0.25 0.1546 0.6178 2060321 BSPBio_003520 C[C@@H]1O[C@@H](O[C@@H]2[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]2Oc3cc(O)c4c(=O)cc(oc4c3)c5ccc(O)cc5)[C@H](O)[C@H](O)[C@H]1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P23 mock treatment 141400.0 -4880.0 -0.33 143960.0 -4500.0 -0.33 -0.472 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2463 P24 mock treatment 142800.0 -3480.0 -0.24 143760.0 -4700.0 -0.35 -0.415 -0.982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A01 mock treatment 145640.0 -4580.0 -0.31 143320.0 -6030.0 -0.45 -0.5384 -0.9843 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A02 mock treatment 142080.0 -8140.0 -0.56 143840.0 -5510.0 -0.41 -0.6827 -0.9889 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A03 compound treatment 140800.0 -9420.0 -0.64 137760.0 -11600.0 -0.86 -1.0644 -0.9895 3480106 BSPBio_003521 CC(C)(C(=O)O)c1ccc(cc1)C(O)CCCN2CCC(CC2)C(O)(c3ccccc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A04 mock treatment 145280.0 -4940.0 -0.34 141920.0 -7430.0 -0.55 -0.6295 -0.9718 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A05 compound treatment 144360.0 -5860.0 -0.4 142800.0 -6550.0 -0.49 -0.6275 -0.9951 BSPBio_003522 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A06 mock treatment 141440.0 -8780.0 -0.6 139560.0 -9790.0 -0.73 -0.9388 -0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A07 compound treatment 142680.0 -7540.0 -0.51 140960.0 -8390.0 -0.62 -0.8053 -0.9954 3054095 BSPBio_003523 CCC(/C=C/[C@@H](C)[C@H]1CCC2C3CC=C4C[C@@H](O)CC[C@]4(C)C3CC[C@]12C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A08 mock treatment 141600.0 -8620.0 -0.59 138720.0 -10600.0 -0.79 -0.9753 -0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A09 compound treatment 140680.0 -9540.0 -0.65 140520.0 -8830.0 -0.66 -0.9249 -1.0 2069287 BSPBio_003524 CCCCCC1C(CC(=O)OC)CCC1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A10 mock treatment 144200.0 -6020.0 -0.41 145680.0 -3670.0 -0.27 -0.4837 -0.9804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A11 compound treatment 179840.0 29600.0 2.02 177160.0 27800.0 2.07 2.8912 0.9999 2069289 BSPBio_003525 CC(=O)Oc1cc2c(CC3OC34[C@@]2(C)CC[C@@]5(C)C6C[C@@](C)(CC[C@]6(C)CC[C@]45C)C(=O)O)c(C)c1OC(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A12 mock treatment 142160.0 -8060.0 -0.55 143240.0 -6110.0 -0.45 -0.7104 -0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A13 compound treatment 147760.0 -2460.0 -0.17 142720.0 -6630.0 -0.49 -0.4678 -0.8973 2475 BSPBio_003526 CC(=CC1C(C(=O)O)C1(C)C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A14 mock treatment 145000.0 -5220.0 -0.36 142720.0 -6630.0 -0.49 -0.6009 -0.9872 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A15 compound treatment 166760.0 16500.0 1.13 165560.0 16200.0 1.21 1.6502 0.9994 2060112 BSPBio_003527 COc1ccc(/C=C/c2cc(O)cc(O)c2)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A16 mock treatment 146680.0 -3540.0 -0.24 141120.0 -8230.0 -0.61 -0.6041 -0.9172 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A17 compound treatment 144760.0 -5460.0 -0.37 137720.0 -11600.0 -0.87 -0.8756 -0.929 2060338 BSPBio_003528 CC(C)c1ccc2c(CC[C@H]3C4=C(CC[C@@]32C)C(=O)OC4)c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A18 mock treatment 138560.0 -11700.0 -0.8 143480.0 -5870.0 -0.44 -0.8713 -0.9602 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A19 compound treatment 138720.0 -11500.0 -0.78 140080.0 -9270.0 -0.69 -1.0426 -0.998 3174115 BSPBio_003529 CC[C@H](CCC(C)[C@H]1CCC2C3CCC4C[C@@H](O)CC[C@]4(C)C3CC[C@]12C)C(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A20 mock treatment 139520.0 -10700.0 -0.73 143760.0 -5590.0 -0.42 -0.8103 -0.9645 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A21 compound treatment 154840.0 4620.0 0.31 150200.0 848.0 0.06 0.2672 0.8324 2060334 BSPBio_003530 C[C@H]1[C@@H](O)C[C@H]2[C@@H]1[C@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)OC=C2C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A22 mock treatment 144600.0 -5620.0 -0.38 141040.0 -8310.0 -0.62 -0.7086 -0.9736 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A23 mock treatment 142400.0 -7820.0 -0.53 140520.0 -8830.0 -0.66 -0.842 -0.9946 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 A24 mock treatment 142080.0 -8140.0 -0.56 140480.0 -8870.0 -0.66 -0.8595 -0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B01 mock treatment 138200.0 -12000.0 -0.82 134600.0 -14800.0 -1.1 -1.356 -0.9896 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B02 mock treatment 134520.0 -15700.0 -1.07 132560.0 -16800.0 -1.25 -1.6408 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B03 mock treatment 137120.0 -13100.0 -0.89 135920.0 -13400.0 -1.0 -1.3386 -0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B04 mock treatment 145240.0 -4980.0 -0.34 137440.0 -11900.0 -0.89 -0.8672 -0.9134 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B05 mock treatment 143560.0 -6660.0 -0.45 140280.0 -9070.0 -0.68 -0.7987 -0.9814 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B06 mock treatment 152280.0 2060.0 0.14 146840.0 -2510.0 -0.19 -0.0331 -0.1416 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B07 mock treatment 144120.0 -6100.0 -0.42 140800.0 -8550.0 -0.64 -0.7443 -0.9788 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B08 mock treatment 140200.0 -10000.0 -0.68 141440.0 -7910.0 -0.59 -0.8996 -0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B09 mock treatment 141440.0 -8780.0 -0.6 138720.0 -10600.0 -0.79 -0.983 -0.9906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B10 mock treatment 143560.0 -6660.0 -0.45 137680.0 -11700.0 -0.87 -0.9355 -0.9543 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B11 mock treatment 144720.0 -5500.0 -0.38 140720.0 -8630.0 -0.64 -0.7196 -0.9672 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B12 mock treatment 145520.0 -4700.0 -0.32 136080.0 -13300.0 -0.99 -0.9253 -0.8909 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B13 mock treatment 145880.0 -4340.0 -0.3 136240.0 -13100.0 -0.98 -0.8995 -0.882 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B14 mock treatment 142280.0 -7940.0 -0.54 141680.0 -7670.0 -0.57 -0.7867 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B15 mock treatment 136720.0 -13500.0 -0.92 138960.0 -10400.0 -0.77 -1.1979 -0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B16 mock treatment 135200.0 -15000.0 -1.02 138320.0 -11000.0 -0.82 -1.3049 -0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B17 mock treatment 141720.0 -8500.0 -0.58 138360.0 -11000.0 -0.82 -0.9885 -0.9858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B18 mock treatment 139720.0 -10500.0 -0.72 136400.0 -13000.0 -0.96 -1.188 -0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B19 mock treatment 142280.0 -7940.0 -0.54 140320.0 -9030.0 -0.67 -0.8583 -0.9943 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B20 mock treatment 139120.0 -11100.0 -0.76 141240.0 -8110.0 -0.6 -0.9622 -0.9937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B21 mock treatment 141600.0 -8620.0 -0.59 134640.0 -14700.0 -1.09 -1.19 -0.9575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B22 mock treatment 136240.0 -14000.0 -0.95 136560.0 -12800.0 -0.95 -1.3474 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B23 mock treatment 135520.0 -14700.0 -1.0 138320.0 -11000.0 -0.82 -1.2895 -0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 B24 mock treatment 135440.0 -14800.0 -1.01 138800.0 -10600.0 -0.79 -1.268 -0.9924 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C01 mock treatment 142880.0 -7340.0 -0.5 143200.0 -6150.0 -0.46 -0.6778 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C02 mock treatment 140400.0 -9820.0 -0.67 138320.0 -11000.0 -0.82 -1.0542 -0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C03 compound treatment 205160.0 54900.0 3.75 200400.0 51000.0 3.8 5.3349 1.0 854065 BSPBio_003531 CCCCCCCCCCCC1=C(O)C(=O)C=C(O)C1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C04 mock treatment 154200.0 3980.0 0.27 142640.0 -6710.0 -0.5 -0.1616 -0.2843 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C05 compound treatment 173560.0 23300.0 1.59 169840.0 20500.0 1.52 2.2032 0.9998 2060337 BSPBio_003532 COc1ccc(cc1O)c2oc3cc(O[C@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)c(OC)c(O)c3c(=O)c2OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C06 mock treatment 146480.0 -3740.0 -0.26 140240.0 -9110.0 -0.68 -0.66 -0.9109 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C07 compound treatment 147960.0 -2260.0 -0.15 146920.0 -2430.0 -0.18 -0.2371 -0.9969 783 BSPBio_003533 CO[C@@]12C[C@@H](COC(=O)c3cncc(Br)c3)CN(C)[C@@H]2Cc4cn(C)c5cccc1c45 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C08 mock treatment 150680.0 455.0 0.03 140760.0 -8590.0 -0.64 -0.4302 -0.672 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C09 compound treatment 146000.0 -4220.0 -0.29 143600.0 -5750.0 -0.43 -0.5064 -0.9814 3079215 BSPBio_003534 CC(C)C[C@H](N)C(=O)N[C@@H](C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C10 mock treatment 143400.0 -6820.0 -0.47 147640.0 -1710.0 -0.13 -0.4191 -0.8687 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C11 compound treatment 146280.0 -3940.0 -0.27 149520.0 168.0 0.01 -0.1813 -0.6734 3198430 BSPBio_003535 CC(C)C(NC(=O)C(Cc1ccc(O)cc1)NC(=O)C(NC(=O)C(F)(F)F)C(C)C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C12 mock treatment 148320.0 -1900.0 -0.13 145480.0 -3870.0 -0.29 -0.2956 -0.9352 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C13 compound treatment 155920.0 5700.0 0.39 148720.0 -632.0 -0.05 0.2413 0.617 3079214 BSPBio_003536 CC(C)CC(NC(=O)CN)C(=O)NC(Cc1ccccc1)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C14 mock treatment 141840.0 -8380.0 -0.57 144520.0 -4830.0 -0.36 -0.6585 -0.975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C15 compound treatment 155920.0 5700.0 0.39 141800.0 -7550.0 -0.56 -0.1229 -0.1798 3081193 BSPBio_003537 C/N=C(\N)/NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C16 mock treatment 143720.0 -6500.0 -0.44 143520.0 -5830.0 -0.43 -0.6205 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C17 compound treatment 153400.0 3180.0 0.22 146040.0 -3310.0 -0.25 -0.0212 -0.0646 3198433 BSPBio_003538 NC(Cc1c[nH]cn1)C(=O)Nc2ccc3ccccc3c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C18 mock treatment 140160.0 -10100.0 -0.69 148560.0 -792.0 -0.06 -0.5269 -0.765 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C19 compound treatment 144360.0 -5860.0 -0.4 144000.0 -5350.0 -0.4 -0.5644 -1.0 3198432 BSPBio_003539 CSC(=N)NCCC[C@@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C20 mock treatment 146520.0 -3700.0 -0.25 141400.0 -7950.0 -0.59 -0.5971 -0.9279 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C21 compound treatment 153400.0 3180.0 0.22 146040.0 -3310.0 -0.25 -0.0212 -0.0646 1466 BSPBio_003540 NCCCCC(N)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)NC(CCCCN)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C22 mock treatment 139320.0 -10900.0 -0.74 142760.0 -6590.0 -0.49 -0.8726 -0.9796 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C23 mock treatment 138360.0 -11900.0 -0.81 138080.0 -11300.0 -0.84 -1.1652 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 C24 mock treatment 140200.0 -10000.0 -0.68 140520.0 -8830.0 -0.66 -0.9481 -0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D01 mock treatment 136360.0 -13900.0 -0.95 145720.0 -3630.0 -0.27 -0.8595 -0.8743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D02 mock treatment 142280.0 -7940.0 -0.54 139520.0 -9830.0 -0.73 -0.9004 -0.989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D03 mock treatment 148640.0 -1580.0 -0.11 144960.0 -4390.0 -0.33 -0.3075 -0.8933 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D04 mock treatment 147880.0 -2340.0 -0.16 142720.0 -6630.0 -0.49 -0.462 -0.8906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D05 mock treatment 149600.0 -625.0 -0.04 144760.0 -4590.0 -0.34 -0.2718 -0.7891 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D06 mock treatment 154560.0 4340.0 0.3 143280.0 -6070.0 -0.45 -0.1105 -0.2047 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D07 mock treatment 145760.0 -4460.0 -0.3 147040.0 -2310.0 -0.17 -0.3369 -0.9635 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D08 mock treatment 149760.0 -465.0 -0.03 145120.0 -4230.0 -0.31 -0.2451 -0.7743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D09 mock treatment 142680.0 -7540.0 -0.51 146520.0 -2830.0 -0.21 -0.5127 -0.9224 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D10 mock treatment 146400.0 -3820.0 -0.26 147880.0 -1470.0 -0.11 -0.2618 -0.9258 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D11 mock treatment 148120.0 -2100.0 -0.14 140920.0 -8430.0 -0.63 -0.5452 -0.8469 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D12 mock treatment 145920.0 -4300.0 -0.29 148720.0 -632.0 -0.05 -0.2408 -0.81 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D13 mock treatment 148120.0 -2100.0 -0.14 141240.0 -8110.0 -0.6 -0.5284 -0.8514 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D14 mock treatment 147640.0 -2580.0 -0.18 147640.0 -1710.0 -0.13 -0.2147 -0.9873 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D15 mock treatment 150960.0 735.0 0.05 144120.0 -5230.0 -0.39 -0.2399 -0.611 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D16 mock treatment 139600.0 -10600.0 -0.72 145400.0 -3950.0 -0.29 -0.7202 -0.9212 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D17 mock treatment 139800.0 -10400.0 -0.71 145440.0 -3910.0 -0.29 -0.7084 -0.9224 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D18 mock treatment 144160.0 -6060.0 -0.41 143760.0 -5590.0 -0.42 -0.5866 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D19 mock treatment 138000.0 -12200.0 -0.83 143560.0 -5790.0 -0.43 -0.8941 -0.9529 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D20 mock treatment 144200.0 -6020.0 -0.41 143080.0 -6270.0 -0.47 -0.6205 -0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D21 mock treatment 143240.0 -6980.0 -0.48 143800.0 -5550.0 -0.41 -0.6289 -0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D22 mock treatment 140720.0 -9500.0 -0.65 145960.0 -3390.0 -0.25 -0.6367 -0.9155 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D23 mock treatment 143440.0 -6780.0 -0.46 143120.0 -6230.0 -0.46 -0.655 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 D24 mock treatment 136680.0 -13500.0 -0.92 140080.0 -9270.0 -0.69 -1.1409 -0.9897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E01 mock treatment 150480.0 255.0 0.02 148480.0 -872.0 -0.06 -0.0336 -0.4996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E02 mock treatment 148120.0 -2100.0 -0.14 148080.0 -1270.0 -0.09 -0.1684 -0.9796 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E03 compound treatment 294480.0 144000.0 9.83 286440.0 137000.0 10.2 14.169 0.9998 1538 BSPBio_003541 Oc1ccc(c(O)c1)c2oc3cc(O)cc(O)c3c(=O)c2O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E04 mock treatment 151000.0 775.0 0.05 152360.0 3010.0 0.22 0.1957 0.8507 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E05 compound treatment 155760.0 5540.0 0.38 147200.0 -2150.0 -0.16 0.1536 0.3747 873168 BSPBio_003542 OC(=O)c1cc(O)c2ccc(Cl)cc2n1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E06 mock treatment 148000.0 -2220.0 -0.15 151920.0 2570.0 0.19 0.0279 0.1144 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E07 compound treatment 156440.0 6220.0 0.42 154440.0 5090.0 0.38 0.5674 0.9984 1452 BSPBio_003543 CCCCN(CCCC)CCCOC(=O)c1ccc(N)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E08 mock treatment 149920.0 -305.0 -0.02 152680.0 3330.0 0.25 0.1605 0.6456 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E09 compound treatment 150160.0 -64.6 0.0 148280.0 -1070.0 -0.08 -0.0595 -0.745 3079387 BSPBio_003544 CN(/C=N/c1ccc(C)cc1C)/C=N/c2ccc(C)cc2C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E10 mock treatment 151720.0 1500.0 0.1 148280.0 -1070.0 -0.08 0.0157 0.1213 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E11 compound treatment 159520.0 9300.0 0.63 167360.0 18000.0 1.34 1.3959 0.9415 3199905 BSPBio_003545 CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C2=O)c4c5nc6cc(C)ccn6c5c(NC(=O)/C(=C\C=C\[C@H](C)[C@H](O)[C@@H](C)C(O)[C@@H](C)[C@H](OC(=O)C)[C@@H]1C)/C)c(O)c4c(O)c3C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E12 mock treatment 154880.0 4660.0 0.32 151520.0 2170.0 0.16 0.3385 0.9508 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E13 compound treatment 126080.0 -24100.0 -1.65 124040.0 -25300.0 -1.88 -2.4961 -0.9977 3198427 BSPBio_003546 CCCCCCCCCc1ccc(OCCOCCOCCOCCOCCOCCOCCOCCOCCO)cc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E14 mock treatment 150720.0 495.0 0.03 154880.0 5530.0 0.41 0.3148 0.7626 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E15 compound treatment 266960.0 117000.0 7.96 273440.0 124000.0 9.24 12.1581 0.9973 1007083 BSPBio_003547 Oc1cc(O)c2C(=O)c3ccccc3C(=O)c2c1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E16 mock treatment 153800.0 3580.0 0.24 155440.0 6090.0 0.45 0.4928 0.9577 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E17 compound treatment 151560.0 1340.0 0.09 151320.0 1970.0 0.15 0.168 0.9738 3199906 BSPBio_003548 CC[C@H]1OC(=O)C[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)[C@@H](O[C@H]3C[C@@](C)(O)[C@@H](O)[C@H](C)O3)[C@@H]([C@H]2O)N(C)C)[C@@H](CC=O)C[C@@H](C)C(=O)/C=C/C(=C/[C@@H]1CO[C@@H]4O[C@H](C)[C@@H](O)[C@@H](OC)[C@H]4OC)/C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E18 mock treatment 148520.0 -1700.0 -0.12 150680.0 1330.0 0.1 -0.0123 -0.0804 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E19 compound treatment 145520.0 -4700.0 -0.32 152000.0 2650.0 0.2 -0.0874 -0.2322 832325 BSPBio_003549 COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CC(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E20 mock treatment 150720.0 495.0 0.03 148680.0 -672.0 -0.05 -0.0115 -0.19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E21 compound treatment 159320.0 9100.0 0.62 163200.0 13800.0 1.03 1.1673 0.9704 1008492 BSPBio_003550 O=C(CC(=O)c1ccccc1)c2ccccc2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E22 mock treatment 148360.0 -1860.0 -0.13 151800.0 2450.0 0.18 0.039 0.1754 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E23 mock treatment 144280.0 -5940.0 -0.41 147520.0 -1830.0 -0.14 -0.383 -0.8956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 E24 mock treatment 138920.0 -11300.0 -0.77 144080.0 -5270.0 -0.39 -0.8224 -0.9509 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F01 mock treatment 146000.0 -4220.0 -0.29 151400.0 2050.0 0.15 -0.0959 -0.2941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F02 mock treatment 148440.0 -1780.0 -0.12 147880.0 -1470.0 -0.11 -0.1635 -0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F03 mock treatment 152520.0 2300.0 0.16 151520.0 2170.0 0.16 0.2248 0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F04 mock treatment 155240.0 5020.0 0.34 147120.0 -2230.0 -0.17 0.1243 0.3271 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F05 mock treatment 152880.0 2660.0 0.18 148120.0 -1230.0 -0.09 0.0632 0.3114 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F06 mock treatment 149040.0 -1180.0 -0.08 147600.0 -1750.0 -0.13 -0.1493 -0.9735 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F07 mock treatment 151960.0 1740.0 0.12 149800.0 448.0 0.03 0.1073 0.8725 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F08 mock treatment 155000.0 4780.0 0.33 148160.0 -1190.0 -0.09 0.1675 0.4964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F09 mock treatment 148520.0 -1700.0 -0.12 152920.0 3570.0 0.27 0.1056 0.3643 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F10 mock treatment 151840.0 1620.0 0.11 150840.0 1490.0 0.11 0.1562 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F11 mock treatment 151560.0 1340.0 0.09 152800.0 3450.0 0.26 0.2459 0.9028 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F12 mock treatment 151680.0 1460.0 0.1 149560.0 208.0 0.02 0.0811 0.8078 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F13 mock treatment 147800.0 -2420.0 -0.17 151240.0 1890.0 0.14 -0.0175 -0.0807 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F14 mock treatment 152400.0 2180.0 0.15 154680.0 5330.0 0.4 0.3853 0.91 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F15 mock treatment 155200.0 4980.0 0.34 153000.0 3650.0 0.27 0.4319 0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F16 mock treatment 149120.0 -1100.0 -0.08 152040.0 2690.0 0.2 0.0882 0.4127 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F17 mock treatment 151520.0 1300.0 0.09 150000.0 648.0 0.05 0.0966 0.9596 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F18 mock treatment 149320.0 -905.0 -0.06 148520.0 -832.0 -0.06 -0.0874 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F19 mock treatment 151720.0 1500.0 0.1 147560.0 -1790.0 -0.13 -0.0222 -0.1322 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F20 mock treatment 152040.0 1820.0 0.12 146640.0 -2710.0 -0.2 -0.0552 -0.2331 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F21 mock treatment 145160.0 -5060.0 -0.35 146760.0 -2590.0 -0.19 -0.3805 -0.9622 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F22 mock treatment 146360.0 -3860.0 -0.26 142560.0 -6790.0 -0.51 -0.5437 -0.9539 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F23 mock treatment 142600.0 -7620.0 -0.52 149760.0 408.0 0.03 -0.3461 -0.6646 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 F24 mock treatment 139600.0 -10600.0 -0.72 146640.0 -2710.0 -0.2 -0.6549 -0.8709 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G01 mock treatment 152000.0 1780.0 0.12 149920.0 568.0 0.04 0.1155 0.9008 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G02 mock treatment 153120.0 2900.0 0.2 151720.0 2370.0 0.18 0.2642 0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G03 compound treatment 169720.0 19500.0 1.33 169920.0 20600.0 1.53 2.0223 0.9975 758 BSPBio_003551 CCCOc1ccc2nc(NC(=O)OC)[nH]c2c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G04 mock treatment 158720.0 8500.0 0.58 156480.0 7130.0 0.53 0.7847 0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G05 compound treatment 156160.0 5940.0 0.4 163160.0 13800.0 1.03 1.0128 0.917 1090918 BSPBio_003552 Cc1nc(C)c(Cl)c(O)c1Cl 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G06 mock treatment 156800.0 6580.0 0.45 150080.0 728.0 0.05 0.3553 0.7869 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G07 compound treatment 158640.0 8420.0 0.57 158800.0 9450.0 0.7 0.9029 0.9949 3199907 BSPBio_003553 OC(=O)c1cn(c2ccc(F)cc2)c3cc(N4CCNCC4)c(F)cc3c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G08 mock treatment 155800.0 5580.0 0.38 156680.0 7330.0 0.55 0.6545 0.9844 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G09 compound treatment 161160.0 10900.0 0.75 157720.0 8370.0 0.62 0.9676 0.996 3078276 BSPBio_003554 COC(=O)N/N=C/c1c[n+]([O-])c2ccccc2[n+]1[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G10 mock treatment 156000.0 5780.0 0.39 156480.0 7130.0 0.53 0.6536 0.9892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G11 compound treatment 251280.0 101000.0 6.89 245240.0 95900.0 7.14 9.9181 0.9998 3198533 BSPBio_003555 CCc1c(C)c2=Cc3c(C=C)c(C)c4C=c5c(C)c(CCC(=O)O)c6=C7C(C(=O)O)C(=O)c8c(C)c9C=c1n2[Cu](n9c78)(n43)n56 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G12 mock treatment 157560.0 7340.0 0.5 160560.0 11200.0 0.83 0.9435 0.9701 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G13 compound treatment 154360.0 4140.0 0.28 152880.0 3530.0 0.26 0.3851 0.9994 3077147 BSPBio_003556 CC(O)Cn1c(C)ncc1[N+](=O)[O-] 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G14 mock treatment 164080.0 13900.0 0.94 159120.0 9770.0 0.73 1.182 0.9916 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G15 compound treatment 158800.0 8580.0 0.58 155480.0 6130.0 0.46 0.7359 0.9925 907420 BSPBio_003557 CNC(=N)NCCC[C@H](N)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G16 mock treatment 154960.0 4740.0 0.32 151600.0 2250.0 0.17 0.3466 0.9532 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G17 compound treatment 156160.0 5940.0 0.4 160480.0 11100.0 0.83 0.8718 0.9457 435 BSPBio_003558 CC(C)Cn1c(=O)n(C)c(=O)c2nc[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G18 mock treatment 157600.0 7380.0 0.5 155600.0 6250.0 0.47 0.6844 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G19 compound treatment 157120.0 6900.0 0.47 161880.0 12500.0 0.93 0.9918 0.9497 3480338 BSPBio_003559 OC(=O)C(Cc1cc(=O)[nH]c2ccccc12)NC(=O)c3ccc(Cl)cc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G20 mock treatment 149400.0 -825.0 -0.06 154240.0 4890.0 0.36 0.2175 0.5908 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G21 compound treatment 154280.0 4060.0 0.28 156560.0 7210.0 0.54 0.5749 0.9525 2801 BSPBio_003560 CCCCCCNC(=O)n1cc(F)c(=O)[nH]c1=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G22 mock treatment 154720.0 4500.0 0.31 150040.0 688.0 0.05 0.2529 0.814 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G23 mock treatment 145680.0 -4540.0 -0.31 152120.0 2770.0 0.21 -0.0734 -0.1972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 G24 mock treatment 149440.0 -785.0 -0.05 143080.0 -6270.0 -0.47 -0.3679 -0.783 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H01 mock treatment 150480.0 255.0 0.02 149840.0 488.0 0.04 0.038 0.9432 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H02 mock treatment 153280.0 3060.0 0.21 148920.0 -432.0 -0.03 0.1246 0.5911 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H03 mock treatment 155280.0 5060.0 0.34 151360.0 2010.0 0.15 0.3494 0.9301 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H04 mock treatment 152600.0 2380.0 0.16 152440.0 3090.0 0.23 0.2771 0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H05 mock treatment 154760.0 4540.0 0.31 149880.0 528.0 0.04 0.2465 0.7907 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H06 mock treatment 155080.0 4860.0 0.33 154360.0 5010.0 0.37 0.4977 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H07 mock treatment 158000.0 7780.0 0.53 157360.0 8010.0 0.6 0.7963 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H08 mock treatment 157120.0 6900.0 0.47 154400.0 5050.0 0.38 0.5981 0.9938 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H09 mock treatment 159320.0 9100.0 0.62 148200.0 -1150.0 -0.09 0.3779 0.6036 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H10 mock treatment 154880.0 4660.0 0.32 155640.0 6290.0 0.47 0.5554 0.9821 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H11 mock treatment 151120.0 895.0 0.06 156640.0 7290.0 0.54 0.4267 0.7817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H12 mock treatment 156200.0 5980.0 0.41 155200.0 5850.0 0.44 0.5959 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H13 mock treatment 173560.0 23300.0 1.59 161080.0 11700.0 0.87 1.7422 0.9601 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H14 mock treatment 155680.0 5460.0 0.37 151680.0 2330.0 0.17 0.3855 0.9396 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H15 mock treatment 170720.0 20500.0 1.4 163080.0 13700.0 1.02 1.7105 0.9882 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H16 mock treatment 151680.0 1460.0 0.1 152800.0 3450.0 0.26 0.2516 0.9145 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H17 mock treatment 155840.0 5620.0 0.38 159240.0 9890.0 0.74 0.7911 0.9536 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H18 mock treatment 153760.0 3540.0 0.24 152360.0 3010.0 0.22 0.3288 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H19 mock treatment 148000.0 -2220.0 -0.15 148840.0 -512.0 -0.04 -0.1342 -0.858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H20 mock treatment 150280.0 55.4 0.0 152080.0 2730.0 0.2 0.1463 0.7201 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H21 mock treatment 166960.0 16700.0 1.14 154640.0 5290.0 0.39 1.0851 0.899 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H22 mock treatment 148960.0 -1260.0 -0.09 142920.0 -6430.0 -0.48 -0.3994 -0.8213 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H23 mock treatment 146000.0 -4220.0 -0.29 147320.0 -2030.0 -0.15 -0.3106 -0.9548 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 H24 mock treatment 142800.0 -7420.0 -0.51 143720.0 -5630.0 -0.42 -0.6543 -0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I01 mock treatment 152880.0 2660.0 0.18 147440.0 -1910.0 -0.14 0.0274 0.119 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I02 mock treatment 149560.0 -665.0 -0.05 147240.0 -2110.0 -0.16 -0.1432 -0.8753 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I03 compound treatment 155160.0 4940.0 0.34 158240.0 8890.0 0.66 0.7057 0.9508 2335 BSPBio_003561 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)O)cc1OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I04 mock treatment 151360.0 1140.0 0.08 155160.0 5810.0 0.43 0.3604 0.8207 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I05 compound treatment 152200.0 1980.0 0.13 153000.0 3650.0 0.27 0.2872 0.9477 1099044 BSPBio_003562 CC(C)(C)C(=O)C(Oc1ccc(Cl)cc1)n2cncn2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I06 mock treatment 157680.0 7460.0 0.51 152880.0 3530.0 0.26 0.5451 0.9528 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I07 compound treatment 164680.0 14500.0 0.99 164120.0 14800.0 1.1 1.4741 0.9985 1000069 BSPBio_003563 COc1ccc2C[C@H]3N(C)CCc4cc(OC)c(Oc5c6OCOc6cc7CCN(C)[C@@H](Cc8ccc(Oc1c2)cc8)c75)cc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I08 mock treatment 158880.0 8660.0 0.59 159880.0 10500.0 0.78 0.9713 0.9902 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I09 compound treatment 169240.0 19000.0 1.3 160120.0 10800.0 0.8 1.4834 0.9733 3182 BSPBio_003564 CCCc1cc(ccn1)C(=S)N 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I10 mock treatment 159160.0 8940.0 0.61 157600.0 8250.0 0.61 0.8649 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I11 compound treatment 182440.0 32200.0 2.2 184560.0 35200.0 2.62 3.406 0.9961 3077356 BSPBio_003565 COc1cc(cc(OC)c1O)[C@H]2C3C(COC3=O)[C@H](O)c4cc5OCOc5cc24 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I12 mock treatment 154160.0 3940.0 0.27 155720.0 6370.0 0.47 0.5249 0.9637 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I13 compound treatment 155800.0 5580.0 0.38 156960.0 7610.0 0.57 0.6692 0.9812 1078453 BSPBio_003566 Fc1ccc(cc1)C(=O)CCCN2CCN(CC2)c3ccccn3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I14 mock treatment 155520.0 5300.0 0.36 158280.0 8930.0 0.66 0.7252 0.9589 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I15 compound treatment 153400.0 3180.0 0.22 157400.0 8050.0 0.6 0.5767 0.9053 3077146 BSPBio_003567 CN[C@@H]1[C@@H](O)C(OC2[C@@H](N)C[C@@H](N)[C@H](O[C@H]3O[C@H](C(C)O)[C@@H](O)[C@H](O)[C@H]3N)[C@H]2O)OC[C@]1(C)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I16 mock treatment 153720.0 3500.0 0.24 153760.0 4410.0 0.33 0.4005 0.9877 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I17 compound treatment 161240.0 11000.0 0.75 159400.0 10000.0 0.75 1.0599 1.0 3069053 BSPBio_003568 CCOC(=O)n1ccn(C)c1=S 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I18 mock treatment 154200.0 3980.0 0.27 150680.0 1330.0 0.1 0.2616 0.9066 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I19 compound treatment 152320.0 2100.0 0.14 151680.0 2330.0 0.17 0.2236 0.9954 3078275 BSPBio_003569 C[C@@H](N)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I20 mock treatment 151200.0 975.0 0.07 152600.0 3250.0 0.24 0.218 0.8693 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I21 compound treatment 173240.0 23000.0 1.57 167280.0 17900.0 1.33 2.0531 0.9967 3480340 BSPBio_003570 c1cn(cn1)C(c2ccccc2)c3ccc(cc3)c4ccccc4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I22 mock treatment 152200.0 1980.0 0.13 144840.0 -4510.0 -0.34 -0.1422 -0.3931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I23 mock treatment 144840.0 -5380.0 -0.37 146240.0 -3110.0 -0.23 -0.4233 -0.9753 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 I24 mock treatment 143440.0 -6780.0 -0.46 144720.0 -4630.0 -0.34 -0.5708 -0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J01 mock treatment 149720.0 -505.0 -0.03 147560.0 -1790.0 -0.13 -0.1186 -0.8613 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J02 mock treatment 151880.0 1660.0 0.11 153000.0 3650.0 0.27 0.2718 0.9243 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J03 mock treatment 157240.0 7020.0 0.48 150640.0 1290.0 0.1 0.406 0.8323 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J04 mock treatment 150800.0 575.0 0.04 151440.0 2090.0 0.16 0.1376 0.8586 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J05 mock treatment 153800.0 3580.0 0.24 150520.0 1170.0 0.09 0.2339 0.9036 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J06 mock treatment 153360.0 3140.0 0.21 155400.0 6050.0 0.45 0.4695 0.9421 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J07 mock treatment 153600.0 3380.0 0.23 152880.0 3530.0 0.26 0.3484 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J08 mock treatment 153440.0 3220.0 0.22 157080.0 7730.0 0.58 0.5617 0.9126 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J09 mock treatment 157000.0 6780.0 0.46 158160.0 8810.0 0.66 0.7902 0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J10 mock treatment 153280.0 3060.0 0.21 156120.0 6770.0 0.5 0.5035 0.9236 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J11 mock treatment 156120.0 5900.0 0.4 159520.0 10200.0 0.76 0.8193 0.9562 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J12 mock treatment 153720.0 3500.0 0.24 158280.0 8930.0 0.66 0.6384 0.9043 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J13 mock treatment 154280.0 4060.0 0.28 154360.0 5010.0 0.37 0.4591 0.9892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J14 mock treatment 157120.0 6900.0 0.47 152760.0 3410.0 0.25 0.5118 0.9581 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J15 mock treatment 153520.0 3300.0 0.22 156880.0 7530.0 0.56 0.5551 0.9195 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J16 mock treatment 156720.0 6500.0 0.44 152680.0 3330.0 0.25 0.4883 0.9623 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J17 mock treatment 153360.0 3140.0 0.21 148560.0 -792.0 -0.06 0.1095 0.4938 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J18 mock treatment 151920.0 1700.0 0.12 150720.0 1370.0 0.1 0.1537 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J19 mock treatment 154920.0 4700.0 0.32 150320.0 968.0 0.07 0.2773 0.8452 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J20 mock treatment 151600.0 1380.0 0.09 147840.0 -1510.0 -0.11 -0.0132 -0.0904 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J21 mock treatment 148960.0 -1260.0 -0.09 146160.0 -3190.0 -0.24 -0.2289 -0.9059 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J22 mock treatment 144560.0 -5660.0 -0.39 143320.0 -6030.0 -0.45 -0.5905 -0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J23 mock treatment 145920.0 -4300.0 -0.29 144040.0 -5310.0 -0.4 -0.4871 -0.9892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 J24 mock treatment 145120.0 -5100.0 -0.35 142360.0 -6990.0 -0.52 -0.614 -0.9809 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K01 mock treatment 154720.0 4500.0 0.31 147680.0 -1670.0 -0.12 0.1287 0.3892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K02 mock treatment 151800.0 1580.0 0.11 148560.0 -792.0 -0.06 0.0343 0.2799 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K03 compound treatment 157800.0 7580.0 0.52 161760.0 12400.0 0.92 1.0182 0.9623 1461079 BSPBio_003571 CCn1cc(C(=O)O)c(=O)c2cc(F)c(cc12)N3CCN(C)CC3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K04 mock treatment 152920.0 2700.0 0.18 153800.0 4450.0 0.33 0.3641 0.9614 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K05 compound treatment 172600.0 22400.0 1.53 163000.0 13600.0 1.02 1.797 0.9805 3198532 BSPBio_003572 COC(=O)Nc1nc2ccc(cc2[nH]1)S(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K06 mock treatment 156200.0 5980.0 0.41 156320.0 6970.0 0.52 0.6548 0.9929 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K07 compound treatment 153200.0 2980.0 0.2 155400.0 6050.0 0.45 0.4618 0.9352 2109 BSPBio_003573 OCc1c[nH]c2ccccc12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K08 mock treatment 155400.0 5180.0 0.35 155400.0 6050.0 0.45 0.5678 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K09 compound treatment 161720.0 11500.0 0.78 162560.0 13200.0 0.98 1.2493 0.9937 1117560 BSPBio_003574 CC(=C)C1CCC(=CC1)CO 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K10 mock treatment 152280.0 2060.0 0.14 156240.0 6890.0 0.51 0.4616 0.8685 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K11 compound treatment 155400.0 5180.0 0.35 153760.0 4410.0 0.33 0.4815 0.9993 3172846 BSPBio_003575 NC(CO)(CO)CO.OC(=O)C1CCn2c(ccc12)C(=O)c3ccccc3 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K12 mock treatment 160680.0 10500.0 0.71 155240.0 5890.0 0.44 0.8139 0.9727 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K13 compound treatment 165000.0 14800.0 1.01 157680.0 8330.0 0.62 1.1506 0.9728 1017318 BSPBio_003576 NC(=O)c1ccc(N)nc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K14 mock treatment 161520.0 11300.0 0.77 154200.0 4850.0 0.36 0.7997 0.9403 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K15 compound treatment 160880.0 10700.0 0.73 155920.0 6570.0 0.49 0.8594 0.9814 3198319 BSPBio_003577 O=C1O[C@]2(C[C@H]3C=CC2=C1)[C@H]4CCCCN34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K16 mock treatment 153000.0 2780.0 0.19 154720.0 5370.0 0.4 0.4163 0.9417 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K17 compound treatment 155320.0 5100.0 0.35 158000.0 8650.0 0.64 0.7008 0.9581 3078274 BSPBio_003578 N[C@H](CO)Cc1ccccc1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K18 mock treatment 157720.0 7500.0 0.51 150480.0 1130.0 0.08 0.4207 0.8124 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K19 compound treatment 157200.0 6980.0 0.48 151160.0 1810.0 0.13 0.4314 0.8729 3078461 BSPBio_003579 NCCc1ccccc1S(=O)(=O)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K20 mock treatment 157640.0 7420.0 0.51 147760.0 -1590.0 -0.12 0.2737 0.5271 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K21 compound treatment 157080.0 6860.0 0.47 153000.0 3650.0 0.27 0.5225 0.9666 1912 BSPBio_003580 [O-][N+](=O)c1cccc2cn[nH]c12 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K22 mock treatment 147760.0 -2460.0 -0.17 147200.0 -2150.0 -0.16 -0.232 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K23 mock treatment 146440.0 -3780.0 -0.26 145800.0 -3550.0 -0.26 -0.3694 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 K24 mock treatment 144200.0 -6020.0 -0.41 141440.0 -7910.0 -0.59 -0.7068 -0.9845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L01 mock treatment 151000.0 775.0 0.05 153760.0 4410.0 0.33 0.2694 0.8106 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L02 mock treatment 154960.0 4740.0 0.32 153200.0 3850.0 0.29 0.4308 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L03 mock treatment 157040.0 6820.0 0.46 154120.0 4770.0 0.35 0.5795 0.9912 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L04 mock treatment 151600.0 1380.0 0.09 157720.0 8370.0 0.62 0.5067 0.8045 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L05 mock treatment 153640.0 3420.0 0.23 154160.0 4810.0 0.36 0.4177 0.9783 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L06 mock treatment 157440.0 7220.0 0.49 155560.0 6210.0 0.46 0.6746 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L07 mock treatment 150400.0 175.0 0.01 152080.0 2730.0 0.2 0.152 0.7475 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L08 mock treatment 157920.0 7700.0 0.52 152760.0 3410.0 0.25 0.5504 0.9444 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L09 mock treatment 153960.0 3740.0 0.25 156520.0 7170.0 0.53 0.5573 0.9427 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L10 mock treatment 156560.0 6340.0 0.43 154520.0 5170.0 0.38 0.5774 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L11 mock treatment 155360.0 5140.0 0.35 159840.0 10500.0 0.78 0.7996 0.9346 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L12 mock treatment 152760.0 2540.0 0.17 160480.0 11100.0 0.83 0.7079 0.8367 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L13 mock treatment 153240.0 3020.0 0.21 159320.0 9970.0 0.74 0.67 0.8702 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L14 mock treatment 155160.0 4940.0 0.34 156240.0 6890.0 0.51 0.6004 0.9791 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L15 mock treatment 155760.0 5540.0 0.38 153080.0 3730.0 0.28 0.4631 0.9886 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L16 mock treatment 154760.0 4540.0 0.31 152760.0 3410.0 0.25 0.398 0.9952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L17 mock treatment 150320.0 95.4 0.01 150200.0 848.0 0.06 0.0492 0.7758 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L18 mock treatment 154280.0 4060.0 0.28 153240.0 3890.0 0.29 0.4001 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L19 mock treatment 151760.0 1540.0 0.1 151080.0 1730.0 0.13 0.165 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L20 mock treatment 151800.0 1580.0 0.11 145520.0 -3830.0 -0.29 -0.1257 -0.4125 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L21 mock treatment 147160.0 -3060.0 -0.21 147520.0 -1830.0 -0.14 -0.2441 -0.9786 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L22 mock treatment 142240.0 -7980.0 -0.54 145880.0 -3470.0 -0.26 -0.5676 -0.942 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L23 mock treatment 148200.0 -2020.0 -0.14 141800.0 -7550.0 -0.56 -0.495 -0.8553 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 L24 mock treatment 139920.0 -10300.0 -0.7 142320.0 -7030.0 -0.52 -0.8668 -0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M01 mock treatment 152560.0 2340.0 0.16 156400.0 7050.0 0.52 0.4835 0.882 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M02 mock treatment 154440.0 4220.0 0.29 157560.0 8210.0 0.61 0.6352 0.9408 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M03 compound treatment 305120.0 155000.0 10.56 320160.0 171000.0 12.71 16.4565 0.9958 3198318 BSPBio_003581 C[C@H]1CCCC(=O)CCC/C=C/c2cc(O)cc(O)c2C(=O)O1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M04 mock treatment 164720.0 14500.0 0.99 164600.0 15200.0 1.13 1.5013 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M05 compound treatment 192000.0 41800.0 2.85 197280.0 47900.0 3.57 4.5363 0.9938 3198320 BSPBio_003582 Clc1ccc(CO/N=C(\Cn2ccnc2)/c3ccc(Cl)cc3Cl)c(Cl)c1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M06 mock treatment 156760.0 6540.0 0.45 159400.0 10000.0 0.75 0.8439 0.9694 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M07 compound treatment 159480.0 9260.0 0.63 164160.0 14800.0 1.1 1.2255 0.965 3077148 BSPBio_003583 CCCCC(=O)Oc1ccccc1C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M08 mock treatment 161160.0 10900.0 0.75 158920.0 9570.0 0.71 1.0307 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M09 compound treatment 158160.0 7940.0 0.54 160840.0 11500.0 0.86 0.9872 0.9756 3480341 BSPBio_003584 CN1CCCC(CC1)n2nc(Cc3ccc(Cl)cc3)c4ccccc4c2=O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M10 mock treatment 161400.0 11200.0 0.76 160400.0 11000.0 0.82 1.1202 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M11 compound treatment 153640.0 3420.0 0.23 165680.0 16300.0 1.22 1.024 0.8275 3081194 BSPBio_003585 CC(=O)O[C@@H]1CC(=O)OC(C)(C)C2CC(=O)[C@]3(C)C(CC[C@@]4(C)[C@@H](OC(=O)[C@H]5O[C@]543)c6ccoc6)[C@]21C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M12 mock treatment 157400.0 7180.0 0.49 162600.0 13200.0 0.99 1.0431 0.9477 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M13 compound treatment 253560.0 103000.0 7.05 256720.0 107000.0 7.99 10.6322 0.998 1907763 BSPBio_003586 Oc1ccc(/C=C/C(=O)OCCc2ccccc2)cc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M14 mock treatment 161960.0 11700.0 0.8 158080.0 8730.0 0.65 1.0251 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M15 compound treatment 138560.0 -11700.0 -0.8 137920.0 -11400.0 -0.85 -1.1639 -0.9994 3198321 BSPBio_003587 CCCCCCCC/C=C/CCCCCCCCOP(=O)(O)OCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M16 mock treatment 159440.0 9220.0 0.63 157760.0 8410.0 0.63 0.8868 1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M17 compound treatment 160880.0 10700.0 0.73 159760.0 10400.0 0.77 1.0615 0.9995 2097 BSPBio_003588 CCCCCCCCCCCCCCCCOP(=O)(O)OCC[N+](C)(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M18 mock treatment 155840.0 5620.0 0.38 160560.0 11200.0 0.83 0.8606 0.9376 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M19 compound treatment 210120.0 59900.0 4.08 205600.0 56200.0 4.19 5.8477 0.9999 122 BSPBio_003589 C(c1c[nH]c2ccccc12)c3c[nH]c4ccccc34 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M20 mock treatment 158000.0 7780.0 0.53 152480.0 3130.0 0.23 0.5395 0.9318 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M21 compound treatment 200160.0 49900.0 3.4 195880.0 46500.0 3.46 4.856 1.0 3055363 BSPBio_003590 COc1cc(/C=C/C(=C/C(=O)\C=C\c2ccc(O)c(OC)c2)/O)ccc1O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M22 mock treatment 156840.0 6620.0 0.45 148520.0 -832.0 -0.06 0.2752 0.6044 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M23 mock treatment 151760.0 1540.0 0.1 149440.0 88.4 0.01 0.0787 0.7501 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 M24 mock treatment 146640.0 -3580.0 -0.24 147440.0 -1910.0 -0.14 -0.2734 -0.9669 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N01 mock treatment 157240.0 7020.0 0.48 155000.0 5650.0 0.42 0.6355 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N02 mock treatment 156720.0 6500.0 0.44 154840.0 5490.0 0.41 0.602 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N03 mock treatment 155720.0 5500.0 0.37 150800.0 1450.0 0.11 0.3412 0.8751 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N04 mock treatment 157840.0 7620.0 0.52 152760.0 3410.0 0.25 0.5465 0.9457 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N05 mock treatment 154280.0 4060.0 0.28 155480.0 6130.0 0.46 0.518 0.9712 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N06 mock treatment 153760.0 3540.0 0.24 153960.0 4610.0 0.34 0.413 0.9851 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N07 mock treatment 155840.0 5620.0 0.38 156560.0 7210.0 0.54 0.6501 0.9863 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N08 mock treatment 161360.0 11100.0 0.76 153120.0 3770.0 0.28 0.7351 0.9083 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N09 mock treatment 163960.0 13700.0 0.94 154280.0 4930.0 0.37 0.9215 0.9163 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N10 mock treatment 158320.0 8100.0 0.55 162240.0 12900.0 0.96 1.0686 0.9655 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N11 mock treatment 156680.0 6460.0 0.44 155840.0 6490.0 0.48 0.6527 0.9989 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N12 mock treatment 162280.0 12100.0 0.82 163840.0 14500.0 1.08 1.3437 0.991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N13 mock treatment 157400.0 7180.0 0.49 159880.0 10500.0 0.78 0.9 0.9743 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N14 mock treatment 156080.0 5860.0 0.4 160040.0 10700.0 0.8 0.8448 0.9491 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N15 mock treatment 154000.0 3780.0 0.26 151080.0 1730.0 0.13 0.273 0.9486 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N16 mock treatment 154720.0 4500.0 0.31 152040.0 2690.0 0.2 0.3582 0.9786 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N17 mock treatment 152200.0 1980.0 0.13 158920.0 9570.0 0.71 0.5988 0.8262 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N18 mock treatment 150120.0 -105.0 -0.01 152560.0 3210.0 0.24 0.1638 0.6857 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N19 mock treatment 153680.0 3460.0 0.24 151760.0 2410.0 0.18 0.2933 0.9909 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N20 mock treatment 154400.0 4180.0 0.28 149320.0 -31.6 0.0 0.1996 0.7012 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N21 mock treatment 151000.0 775.0 0.05 146280.0 -3070.0 -0.23 -0.1243 -0.5296 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N22 mock treatment 155560.0 5340.0 0.36 147800.0 -1550.0 -0.12 0.1756 0.46 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N23 mock treatment 153040.0 2820.0 0.19 142080.0 -7270.0 -0.54 -0.247 -0.4301 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 N24 mock treatment 141120.0 -9100.0 -0.62 144520.0 -4830.0 -0.36 -0.6932 -0.9663 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O01 mock treatment 154920.0 4700.0 0.32 149000.0 -352.0 -0.03 0.2079 0.6471 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O02 mock treatment 150040.0 -185.0 -0.01 149880.0 528.0 0.04 0.0189 0.4579 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O03 compound treatment 153000.0 2780.0 0.19 150480.0 1130.0 0.08 0.1932 0.9332 1017172 BSPBio_003591 C=CCSCC=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O04 mock treatment 151040.0 815.0 0.06 156000.0 6650.0 0.49 0.3892 0.7816 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O05 compound treatment 161680.0 11500.0 0.78 161120.0 11800.0 0.88 1.1716 0.9984 3081195 BSPBio_003592 CC(=O)O[C@@]1(CCC2C3C=C(Cl)C4=CC(=O)CC[C@]4(C)C3CC[C@@]21C)C(=O)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O06 mock treatment 149120.0 -1100.0 -0.08 153720.0 4370.0 0.33 0.1766 0.5293 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O07 compound treatment 152640.0 2420.0 0.16 152960.0 3610.0 0.27 0.3063 0.9724 1029168 BSPBio_003593 CC(=O)c1ccc[nH]1 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O08 mock treatment 156680.0 6460.0 0.44 151640.0 2290.0 0.17 0.4316 0.9147 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O09 compound treatment 149640.0 -585.0 -0.04 151120.0 1770.0 0.13 0.0649 0.4718 3198420 BSPBio_003594 CC[C@]1(O)CC2CN(C1)CCc3c([nH]c4ccccc34)[C@@](C2)(C(=O)OC)c5cc6c(cc5OC)N(C)[C@@H]7[C@@]86CCN9CC=C[C@](CC)([C@H]98)[C@@H](OC(=O)C)[C@]7(O)C(=O)OC 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O10 mock treatment 152920.0 2700.0 0.18 152240.0 2890.0 0.21 0.282 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O11 compound treatment 259160.0 109000.0 7.43 261080.0 112000.0 8.32 11.1316 0.9984 2272 BSPBio_003595 OC(=O)C(Cc1ccc(O)c(O)c1)OC(=O)/C=C/c2ccc(O)c(O)c2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O12 mock treatment 149480.0 -745.0 -0.05 151200.0 1850.0 0.14 0.0614 0.4186 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O13 compound treatment 150320.0 95.4 0.01 149440.0 88.4 0.01 0.0093 1.0 1478 BSPBio_003596 Cc1ccc(cc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)N)C(F)(F)F 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O14 mock treatment 150600.0 375.0 0.03 155640.0 6290.0 0.47 0.349 0.7447 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O15 compound treatment 154920.0 4700.0 0.32 151760.0 2410.0 0.18 0.3531 0.9624 2777 BSPBio_003597 COc1cc(N)c(Cl)cc1C(=O)NC2CCN(Cc3ccccc3)CC2 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O16 mock treatment 149000.0 -1220.0 -0.08 155000.0 5650.0 0.42 0.2382 0.5558 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O17 compound treatment 148880.0 -1340.0 -0.09 153480.0 4130.0 0.31 0.1524 0.4754 3173083 BSPBio_003598 CO[C@H]1[C@H](O)CC(=O)O[C@@H](C)C/C=C/C=C/[C@H](O[C@H]2CC[C@@H]([C@@H](C)O2)N(C)C)[C@H](C)C[C@H](CC=O)[C@@H]1O[C@@H]3O[C@H](C)[C@@H](O[C@H]4C[C@@](C)(O)[C@H](O)[C@H](C)O4)[C@@H]([C@H]3O)N(C)C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O18 mock treatment 149880.0 -345.0 -0.02 147880.0 -1470.0 -0.11 -0.0941 -0.8397 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O19 compound treatment 148040.0 -2180.0 -0.15 145880.0 -3470.0 -0.26 -0.288 -0.9657 1383 BSPBio_003599 CC[C@H]([C@H]1CC[C@H](C)[C@@H](O1)[C@@H](C)[C@H](O)[C@H](C)C(=O)[C@H](CC)[C@H]2OC3(O[C@@]4(CC[C@](C)(O4)[C@H]5CC[C@](O)(CC)[C@H](C)O5)[C@H](O)C=C3)[C@H](C)C[C@@H]2C)C(=O)O 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O20 mock treatment 147600.0 -2620.0 -0.18 145240.0 -4110.0 -0.31 -0.3429 -0.9673 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O21 compound treatment 143560.0 -6660.0 -0.45 145920.0 -3430.0 -0.26 -0.5019 -0.9629 1000112 BSPBio_003600 CC(=O)O[C@H]1[C@@H](O)C2C(C)(C)CC[C@H](O)[C@]2(C)[C@@]3(O)C(=O)C[C@@](C)(O[C@]13C)C=C 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O22 mock treatment 145680.0 -4540.0 -0.31 144960.0 -4390.0 -0.33 -0.4502 -0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O23 mock treatment 141640.0 -8580.0 -0.59 139160.0 -10200.0 -0.76 -0.9502 -0.9918 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 O24 mock treatment 142120.0 -8100.0 -0.55 139360.0 -9990.0 -0.74 -0.9165 -0.9893 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P01 mock treatment 150280.0 55.4 0.0 153240.0 3890.0 0.29 0.2073 0.7163 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P02 mock treatment 150840.0 615.0 0.04 148080.0 -1270.0 -0.09 -0.0373 -0.3599 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P03 mock treatment 150200.0 -24.6 0.0 148600.0 -752.0 -0.06 -0.0407 -0.728 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P04 mock treatment 151360.0 1140.0 0.08 150640.0 1290.0 0.1 0.1225 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P05 mock treatment 154600.0 4380.0 0.3 150200.0 848.0 0.06 0.2556 0.8382 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P06 mock treatment 150000.0 -225.0 -0.02 152720.0 3370.0 0.25 0.1664 0.6627 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P07 mock treatment 152680.0 2460.0 0.17 150800.0 1450.0 0.11 0.1946 0.9773 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P08 mock treatment 149640.0 -585.0 -0.04 155720.0 6370.0 0.47 0.307 0.6454 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P09 mock treatment 155240.0 5020.0 0.34 151760.0 2410.0 0.18 0.3685 0.9546 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P10 mock treatment 146920.0 -3300.0 -0.23 148200.0 -1150.0 -0.09 -0.2199 -0.9123 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P11 mock treatment 147240.0 -2980.0 -0.2 152880.0 3530.0 0.26 0.0418 0.1259 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P12 mock treatment 154520.0 4300.0 0.29 149640.0 288.0 0.02 0.2223 0.7569 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P13 mock treatment 153960.0 3740.0 0.25 152560.0 3210.0 0.24 0.3489 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P14 mock treatment 154280.0 4060.0 0.28 153920.0 4570.0 0.34 0.4359 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P15 mock treatment 150760.0 535.0 0.04 158600.0 9250.0 0.69 0.5125 0.7436 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P16 mock treatment 147240.0 -2980.0 -0.2 150920.0 1570.0 0.12 -0.0613 -0.2615 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P17 mock treatment 150600.0 375.0 0.03 147520.0 -1830.0 -0.14 -0.0783 -0.5645 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P18 mock treatment 151880.0 1660.0 0.11 148600.0 -752.0 -0.06 0.0402 0.3195 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P19 mock treatment 150360.0 135.0 0.01 149400.0 48.4 0.0 0.0091 0.9158 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P20 mock treatment 146160.0 -4060.0 -0.28 144360.0 -4990.0 -0.37 -0.4586 -0.9896 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P21 mock treatment 145440.0 -4780.0 -0.33 142880.0 -6470.0 -0.48 -0.5712 -0.982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P22 mock treatment 147120.0 -3100.0 -0.21 144160.0 -5190.0 -0.39 -0.4229 -0.9599 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P23 mock treatment 141360.0 -8860.0 -0.6 137440.0 -11900.0 -0.89 -1.0542 -0.9826 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.2464 P24 mock treatment 138720.0 -11500.0 -0.78 164240.0 14900.0 1.11 0.2289 0.1686 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A01 mock treatment 206640.0 2630.0 0.18 144400.0 -4740.0 -0.35 -0.1228 -0.3102 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A02 mock treatment 212160.0 8150.0 0.56 141840.0 -7300.0 -0.54 0.0086 0.0111 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A03 mock treatment 217680.0 13700.0 0.93 141920.0 -7220.0 -0.54 0.2789 0.2593 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A04 mock treatment 202400.0 -1610.0 -0.11 144120.0 -5020.0 -0.37 -0.3419 -0.8778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A05 mock treatment 208680.0 4670.0 0.32 141800.0 -7340.0 -0.55 -0.1612 -0.255 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A06 mock treatment 205360.0 1350.0 0.09 140960.0 -8180.0 -0.61 -0.3655 -0.5935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A07 mock treatment 203800.0 -211.0 -0.01 145560.0 -3580.0 -0.27 -0.1986 -0.7441 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A08 mock treatment 197840.0 -6170.0 -0.42 140160.0 -8980.0 -0.67 -0.7701 -0.9751 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A09 mock treatment 208720.0 4710.0 0.32 142840.0 -6300.0 -0.47 -0.1046 -0.184 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A10 mock treatment 201600.0 -2410.0 -0.16 141480.0 -7660.0 -0.57 -0.5194 -0.8753 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A11 mock treatment 200480.0 -3530.0 -0.24 141360.0 -7780.0 -0.58 -0.5797 -0.9243 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A12 mock treatment 195080.0 -8930.0 -0.61 139040.0 -10100.0 -0.75 -0.9621 -0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A13 mock treatment 197320.0 -6690.0 -0.46 139360.0 -9780.0 -0.73 -0.8373 -0.9746 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A14 mock treatment 196120.0 -7890.0 -0.54 139240.0 -9900.0 -0.74 -0.9015 -0.988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A15 mock treatment 193720.0 -10300.0 -0.7 143960.0 -5180.0 -0.39 -0.7688 -0.9603 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A16 mock treatment 188400.0 -15600.0 -1.06 142080.0 -7060.0 -0.53 -1.1242 -0.9471 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A17 mock treatment 195800.0 -8210.0 -0.56 140640.0 -8500.0 -0.63 -0.8432 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A18 mock treatment 196160.0 -7850.0 -0.54 140640.0 -8500.0 -0.63 -0.8259 -0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A19 mock treatment 198520.0 -5490.0 -0.37 140960.0 -8180.0 -0.61 -0.6952 -0.9727 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A20 mock treatment 196440.0 -7570.0 -0.52 142800.0 -6340.0 -0.47 -0.6987 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A21 mock treatment 195800.0 -8210.0 -0.56 144720.0 -4420.0 -0.33 -0.6285 -0.9679 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A22 mock treatment 190400.0 -13600.0 -0.93 140040.0 -9100.0 -0.68 -1.1351 -0.988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A23 mock treatment 191400.0 -12600.0 -0.86 141800.0 -7340.0 -0.55 -0.9943 -0.9761 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base A24 mock treatment 185160.0 -18900.0 -1.29 137520.0 -11600.0 -0.86 -1.5203 -0.9814 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B01 mock treatment 177320.0 -26700.0 -1.82 137120.0 -12000.0 -0.89 -1.9194 -0.9465 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B02 mock treatment 184560.0 -19500.0 -1.33 140240.0 -8900.0 -0.66 -1.4061 -0.9486 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B03 mock treatment 183320.0 -20700.0 -1.41 142560.0 -6580.0 -0.49 -1.3438 -0.8999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B04 mock treatment 186760.0 -17300.0 -1.18 138520.0 -10600.0 -0.79 -1.3906 -0.9813 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B05 mock treatment 184680.0 -19300.0 -1.32 142960.0 -6180.0 -0.46 -1.2572 -0.9006 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B06 mock treatment 185120.0 -18900.0 -1.29 146960.0 -2180.0 -0.16 -1.0255 -0.79 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B07 mock treatment 184480.0 -19500.0 -1.33 137840.0 -11300.0 -0.84 -1.5363 -0.9755 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B08 mock treatment 183960.0 -20100.0 -1.37 138000.0 -11100.0 -0.83 -1.5529 -0.9713 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B09 mock treatment 181000.0 -23000.0 -1.57 139240.0 -9900.0 -0.74 -1.6304 -0.9406 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B10 mock treatment 186880.0 -17100.0 -1.17 138880.0 -10300.0 -0.76 -1.3659 -0.9788 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B11 mock treatment 186520.0 -17500.0 -1.19 142120.0 -7020.0 -0.52 -1.2127 -0.9315 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B12 mock treatment 196360.0 -7650.0 -0.52 138400.0 -10700.0 -0.8 -0.9341 -0.9786 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B13 mock treatment 189560.0 -14500.0 -0.99 137120.0 -12000.0 -0.89 -1.3293 -0.9988 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B14 mock treatment 191040.0 -13000.0 -0.88 139640.0 -9500.0 -0.71 -1.1253 -0.9939 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B15 mock treatment 182440.0 -21600.0 -1.47 140200.0 -8940.0 -0.67 -1.5104 -0.9357 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B16 mock treatment 183640.0 -20400.0 -1.39 135200.0 -13900.0 -1.04 -1.7157 -0.9897 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B17 mock treatment 185400.0 -18600.0 -1.27 136360.0 -12800.0 -0.95 -1.5698 -0.9899 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B18 mock treatment 189920.0 -14100.0 -0.96 138200.0 -10900.0 -0.81 -1.2551 -0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B19 mock treatment 196960.0 -7050.0 -0.48 137400.0 -11700.0 -0.87 -0.9578 -0.9604 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B20 mock treatment 190480.0 -13500.0 -0.92 136640.0 -12500.0 -0.93 -1.3102 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B21 mock treatment 186760.0 -17300.0 -1.18 139960.0 -9180.0 -0.68 -1.3148 -0.9666 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B22 mock treatment 192560.0 -11500.0 -0.78 139880.0 -9260.0 -0.69 -1.0394 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B23 mock treatment 189720.0 -14300.0 -0.97 141320.0 -7820.0 -0.58 -1.1005 -0.9697 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base B24 mock treatment 181800.0 -22200.0 -1.51 133560.0 -15600.0 -1.16 -1.8907 -0.9913 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C01 mock treatment 207640.0 3630.0 0.25 145200.0 -3940.0 -0.29 -0.0324 -0.0845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C02 mock treatment 198840.0 -5170.0 -0.35 144400.0 -4740.0 -0.35 -0.4988 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C03 mock treatment 200640.0 -3370.0 -0.23 150000.0 859.0 0.06 -0.1173 -0.4917 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C04 mock treatment 205160.0 1150.0 0.08 148720.0 -421.0 -0.03 0.0332 0.394 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C05 mock treatment 204480.0 469.0 0.03 146680.0 -2460.0 -0.18 -0.1069 -0.5749 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C06 mock treatment 200440.0 -3570.0 -0.24 143320.0 -5820.0 -0.43 -0.4785 -0.9628 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C07 mock treatment 206520.0 2510.0 0.17 140680.0 -8460.0 -0.63 -0.3243 -0.497 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C08 mock treatment 198400.0 -5610.0 -0.38 144400.0 -4740.0 -0.35 -0.52 -0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C09 mock treatment 196720.0 -7290.0 -0.5 139920.0 -9220.0 -0.69 -0.8368 -0.9875 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C10 mock treatment 209000.0 4990.0 0.34 156480.0 7340.0 0.55 0.6268 0.974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C11 mock treatment 203600.0 -411.0 -0.03 141560.0 -7580.0 -0.56 -0.4188 -0.7413 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C12 mock treatment 208560.0 4550.0 0.31 147120.0 -2020.0 -0.15 0.113 0.3277 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C13 mock treatment 204360.0 349.0 0.02 143680.0 -5460.0 -0.41 -0.2706 -0.6645 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C14 mock treatment 210960.0 6950.0 0.47 142720.0 -6420.0 -0.48 -0.0029 -0.0043 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C15 mock treatment 203160.0 -851.0 -0.06 141360.0 -7780.0 -0.58 -0.4505 -0.774 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C16 mock treatment 202160.0 -1850.0 -0.13 136960.0 -12200.0 -0.91 -0.7303 -0.7978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C17 mock treatment 201920.0 -2090.0 -0.14 140000.0 -9140.0 -0.68 -0.5819 -0.8371 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C18 mock treatment 205360.0 1350.0 0.09 140720.0 -8420.0 -0.63 -0.3781 -0.5969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C19 mock treatment 200000.0 -4010.0 -0.27 138320.0 -10800.0 -0.81 -0.7628 -0.8969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C20 mock treatment 204520.0 509.0 0.03 135520.0 -13600.0 -1.01 -0.6923 -0.6825 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C21 mock treatment 202480.0 -1530.0 -0.1 141760.0 -7380.0 -0.55 -0.4622 -0.8266 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C22 mock treatment 193400.0 -10600.0 -0.72 140400.0 -8740.0 -0.65 -0.9715 -0.9986 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C23 mock treatment 191360.0 -12700.0 -0.86 138520.0 -10600.0 -0.79 -1.1688 -0.9991 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base C24 mock treatment 184600.0 -19400.0 -1.32 139640.0 -9500.0 -0.71 -1.4358 -0.9569 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D01 mock treatment 183520.0 -20500.0 -1.4 139400.0 -9740.0 -0.72 -1.5005 -0.9533 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D02 mock treatment 193680.0 -10300.0 -0.7 141800.0 -7340.0 -0.55 -0.8844 -0.9921 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D03 mock treatment 184400.0 -19600.0 -1.34 143200.0 -5940.0 -0.44 -1.2581 -0.8934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D04 mock treatment 190760.0 -13300.0 -0.9 144240.0 -4900.0 -0.36 -0.8967 -0.9204 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D05 mock treatment 188840.0 -15200.0 -1.03 143760.0 -5380.0 -0.4 -1.0145 -0.9147 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D06 mock treatment 189000.0 -15000.0 -1.02 142840.0 -6300.0 -0.47 -1.0552 -0.9374 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D07 mock treatment 191720.0 -12300.0 -0.84 139840.0 -9300.0 -0.69 -1.082 -0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D08 mock treatment 194840.0 -9170.0 -0.63 142720.0 -6420.0 -0.48 -0.78 -0.9912 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D09 mock treatment 188920.0 -15100.0 -1.03 141280.0 -7860.0 -0.59 -1.1412 -0.9642 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D10 mock treatment 191520.0 -12500.0 -0.85 145600.0 -3540.0 -0.26 -0.7885 -0.8846 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D11 mock treatment 194440.0 -9570.0 -0.65 144120.0 -5020.0 -0.37 -0.7256 -0.965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D12 mock treatment 195920.0 -8090.0 -0.55 144080.0 -5060.0 -0.38 -0.6564 -0.9827 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D13 mock treatment 200760.0 -3250.0 -0.22 146120.0 -3020.0 -0.22 -0.3157 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D14 mock treatment 197000.0 -7010.0 -0.48 143640.0 -5500.0 -0.41 -0.6275 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D15 mock treatment 193440.0 -10600.0 -0.72 146720.0 -2420.0 -0.18 -0.637 -0.8575 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D16 mock treatment 194080.0 -9930.0 -0.68 140480.0 -8660.0 -0.64 -0.9346 -0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D17 mock treatment 192040.0 -12000.0 -0.82 142920.0 -6220.0 -0.46 -0.9045 -0.9639 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D18 mock treatment 205600.0 1590.0 0.11 143360.0 -5780.0 -0.43 -0.2276 -0.513 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D19 mock treatment 198880.0 -5130.0 -0.35 137960.0 -11200.0 -0.83 -0.8358 -0.9259 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D20 mock treatment 199680.0 -4330.0 -0.3 142040.0 -7100.0 -0.53 -0.5825 -0.9622 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D21 mock treatment 192200.0 -11800.0 -0.81 139040.0 -10100.0 -0.75 -1.101 -0.9994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D22 mock treatment 195360.0 -8650.0 -0.59 136400.0 -12700.0 -0.95 -1.0876 -0.9739 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D23 mock treatment 190560.0 -13500.0 -0.92 136840.0 -12300.0 -0.92 -1.2958 -1.0 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base D24 mock treatment 184160.0 -19900.0 -1.35 135440.0 -13700.0 -1.02 -1.678 -0.9903 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E01 mock treatment 210920.0 6910.0 0.47 148720.0 -421.0 -0.03 0.3109 0.6586 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E02 mock treatment 216960.0 12900.0 0.88 151360.0 2220.0 0.17 0.741 0.8251 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E03 mock treatment 213760.0 9750.0 0.66 152320.0 3180.0 0.24 0.6373 0.9033 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E04 mock treatment 205200.0 1190.0 0.08 153200.0 4060.0 0.3 0.2709 0.8662 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E05 mock treatment 216960.0 12900.0 0.88 148000.0 -1140.0 -0.08 0.5642 0.6362 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E06 mock treatment 213840.0 9830.0 0.67 161240.0 12100.0 0.9 1.1106 0.9894 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E07 mock treatment 228480.0 24500.0 1.67 151240.0 2100.0 0.16 1.2901 0.77 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E08 mock treatment 208800.0 4790.0 0.33 149040.0 -101.0 -0.01 0.2256 0.6906 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E09 mock treatment 207280.0 3270.0 0.22 145440.0 -3700.0 -0.28 -0.0372 -0.1049 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E10 mock treatment 213200.0 9190.0 0.63 151080.0 1940.0 0.14 0.545 0.8478 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E11 mock treatment 211880.0 7870.0 0.54 148760.0 -381.0 -0.03 0.3593 0.6688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E12 mock treatment 227880.0 23900.0 1.63 152200.0 3060.0 0.23 1.3117 0.7983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E13 mock treatment 208400.0 4390.0 0.3 145800.0 -3340.0 -0.25 0.0358 0.0919 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E14 mock treatment 212720.0 8710.0 0.59 152160.0 3020.0 0.22 0.5787 0.9116 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E15 mock treatment 210760.0 6750.0 0.46 150840.0 1700.0 0.13 0.4148 0.8692 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E16 mock treatment 205720.0 1710.0 0.12 146120.0 -3020.0 -0.22 -0.0766 -0.3024 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E17 mock treatment 205120.0 1110.0 0.08 148360.0 -781.0 -0.06 0.0124 0.1297 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E18 mock treatment 204040.0 29.3 0.0 153440.0 4300.0 0.32 0.2277 0.7115 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E19 mock treatment 200480.0 -3530.0 -0.24 148920.0 -221.0 -0.02 -0.1818 -0.7537 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E20 mock treatment 208640.0 4630.0 0.32 147600.0 -1540.0 -0.11 0.1421 0.4231 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E21 mock treatment 202360.0 -1650.0 -0.11 147760.0 -1380.0 -0.1 -0.1523 -0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E22 mock treatment 199000.0 -5010.0 -0.34 146960.0 -2180.0 -0.16 -0.3563 -0.9422 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E23 mock treatment 195680.0 -8330.0 -0.57 146080.0 -3060.0 -0.23 -0.5627 -0.9195 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base E24 mock treatment 190200.0 -13800.0 -0.94 143760.0 -5380.0 -0.4 -0.949 -0.9275 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F01 mock treatment 192320.0 -11700.0 -0.8 147600.0 -1540.0 -0.11 -0.6447 -0.8006 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F02 mock treatment 200800.0 -3210.0 -0.22 149240.0 99.0 0.01 -0.1496 -0.6829 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F03 mock treatment 195560.0 -8450.0 -0.58 148000.0 -1140.0 -0.08 -0.4674 -0.8027 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F04 mock treatment 193880.0 -10100.0 -0.69 150240.0 1100.0 0.08 -0.4305 -0.619 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F05 mock treatment 198200.0 -5810.0 -0.4 149040.0 -101.0 -0.01 -0.2854 -0.7204 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F06 mock treatment 201080.0 -2930.0 -0.2 150160.0 1020.0 0.08 -0.0877 -0.4102 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F07 mock treatment 200680.0 -3330.0 -0.23 155440.0 6300.0 0.47 0.1709 0.3281 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F08 mock treatment 195600.0 -8410.0 -0.57 152520.0 3380.0 0.25 -0.2276 -0.3636 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F09 mock treatment 198280.0 -5730.0 -0.39 146360.0 -2780.0 -0.21 -0.4226 -0.9559 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F10 mock treatment 199640.0 -4370.0 -0.3 151320.0 2180.0 0.16 -0.096 -0.2831 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F11 mock treatment 200760.0 -3250.0 -0.22 149160.0 19.0 0.0 -0.1557 -0.7026 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F12 mock treatment 199800.0 -4210.0 -0.29 151000.0 1860.0 0.14 -0.1052 -0.33 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F13 mock treatment 199400.0 -4610.0 -0.31 149920.0 779.0 0.06 -0.1813 -0.5671 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F14 mock treatment 203320.0 -691.0 -0.05 149040.0 -101.0 -0.01 -0.0386 -0.8098 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F15 mock treatment 201360.0 -2650.0 -0.18 149680.0 539.0 0.04 -0.0994 -0.5371 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F16 mock treatment 207440.0 3430.0 0.23 147800.0 -1340.0 -0.1 0.0947 0.3727 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F17 mock treatment 208240.0 4230.0 0.29 147320.0 -1820.0 -0.14 0.1081 0.3391 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F18 mock treatment 209240.0 5230.0 0.36 148120.0 -1020.0 -0.08 0.1984 0.5442 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F19 mock treatment 200720.0 -3290.0 -0.22 145920.0 -3220.0 -0.24 -0.3282 -0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F20 mock treatment 203160.0 -851.0 -0.06 145040.0 -4100.0 -0.31 -0.2568 -0.8267 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F21 mock treatment 199240.0 -4770.0 -0.33 144040.0 -5100.0 -0.38 -0.4984 -0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F22 mock treatment 194320.0 -9690.0 -0.66 145840.0 -3300.0 -0.25 -0.6409 -0.9092 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F23 mock treatment 196480.0 -7530.0 -0.51 146120.0 -3020.0 -0.22 -0.522 -0.9314 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base F24 mock treatment 197200.0 -6810.0 -0.46 145040.0 -4100.0 -0.31 -0.5442 -0.9793 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G01 mock treatment 210280.0 6270.0 0.43 147480.0 -1660.0 -0.12 0.2148 0.4828 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G02 mock treatment 218360.0 14300.0 0.98 155520.0 6380.0 0.47 1.0275 0.9449 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G03 mock treatment 223880.0 19900.0 1.35 157480.0 8340.0 0.62 1.3967 0.9374 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G04 mock treatment 220720.0 16700.0 1.14 154680.0 5540.0 0.41 1.097 0.9055 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G05 mock treatment 222960.0 18900.0 1.29 159320.0 10200.0 0.76 1.4492 0.9677 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G06 mock treatment 217280.0 13300.0 0.9 153880.0 4740.0 0.35 0.8891 0.9157 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G07 mock treatment 214560.0 10500.0 0.72 152840.0 3700.0 0.28 0.7032 0.9132 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G08 mock treatment 214640.0 10600.0 0.72 156360.0 7220.0 0.54 0.8923 0.9892 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G09 mock treatment 213040.0 9030.0 0.62 153560.0 4420.0 0.33 0.6678 0.9569 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G10 mock treatment 210640.0 6630.0 0.45 158000.0 8860.0 0.66 0.7858 0.983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G11 mock treatment 210600.0 6590.0 0.45 158280.0 9140.0 0.68 0.7986 0.9797 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G12 mock treatment 208440.0 4430.0 0.3 160320.0 11200.0 0.83 0.8019 0.9059 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G13 mock treatment 212920.0 8910.0 0.61 159120.0 9980.0 0.74 0.9547 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G14 mock treatment 215000.0 11000.0 0.75 152480.0 3340.0 0.25 0.7055 0.8938 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G15 mock treatment 220000.0 16000.0 1.09 152320.0 3180.0 0.24 0.9381 0.841 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G16 mock treatment 215600.0 11600.0 0.79 149680.0 539.0 0.04 0.5871 0.742 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G17 mock treatment 212560.0 8550.0 0.58 156000.0 6860.0 0.51 0.7731 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G18 mock treatment 214000.0 9990.0 0.68 158640.0 9500.0 0.71 0.9815 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G19 mock treatment 211520.0 7510.0 0.51 151800.0 2660.0 0.2 0.5019 0.9145 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G20 mock treatment 212280.0 8270.0 0.56 151520.0 2380.0 0.18 0.5238 0.8865 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G21 mock treatment 204360.0 349.0 0.02 153320.0 4180.0 0.31 0.2368 0.759 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G22 mock treatment 201440.0 -2570.0 -0.18 151280.0 2140.0 0.16 -0.0114 -0.048 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G23 mock treatment 200080.0 -3930.0 -0.27 149440.0 299.0 0.02 -0.1738 -0.6462 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base G24 mock treatment 202200.0 -1810.0 -0.12 147600.0 -1540.0 -0.11 -0.1684 -0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H01 mock treatment 191440.0 -12600.0 -0.86 148000.0 -1140.0 -0.08 -0.6661 -0.7734 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H02 mock treatment 201720.0 -2290.0 -0.16 149880.0 739.0 0.05 -0.0715 -0.4321 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H03 mock treatment 197840.0 -6170.0 -0.42 153160.0 4020.0 0.3 -0.086 -0.1665 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H04 mock treatment 197400.0 -6610.0 -0.45 156760.0 7620.0 0.57 0.0823 0.1136 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H05 mock treatment 200840.0 -3170.0 -0.22 153560.0 4420.0 0.33 0.0797 0.2025 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H06 mock treatment 202320.0 -1690.0 -0.12 151800.0 2660.0 0.2 0.0584 0.2551 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H07 mock treatment 212040.0 8030.0 0.55 154200.0 5060.0 0.38 0.6533 0.9833 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H08 mock treatment 206120.0 2110.0 0.14 150040.0 899.0 0.07 0.149 0.9394 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H09 mock treatment 205080.0 1070.0 0.07 152360.0 3220.0 0.24 0.221 0.8823 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H10 mock treatment 204320.0 309.0 0.02 155480.0 6340.0 0.47 0.3485 0.738 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H11 mock treatment 204720.0 709.0 0.05 150240.0 1100.0 0.08 0.092 0.9686 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H12 mock treatment 205160.0 1150.0 0.08 153920.0 4780.0 0.36 0.3069 0.8427 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H13 mock treatment 204680.0 669.0 0.05 155280.0 6140.0 0.46 0.3553 0.7739 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H14 mock treatment 204280.0 269.0 0.02 157960.0 8820.0 0.66 0.4771 0.7266 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H15 mock treatment 212880.0 8870.0 0.6 156840.0 7700.0 0.57 0.8328 0.9996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H16 mock treatment 203000.0 -1010.0 -0.07 149960.0 819.0 0.06 -0.0056 -0.0611 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H17 mock treatment 204760.0 749.0 0.05 151800.0 2660.0 0.2 0.1761 0.8614 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H18 mock treatment 205680.0 1670.0 0.11 153120.0 3980.0 0.3 0.2899 0.9137 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H19 mock treatment 205320.0 1310.0 0.09 152040.0 2900.0 0.22 0.2157 0.9237 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H20 mock treatment 203280.0 -731.0 -0.05 147600.0 -1540.0 -0.11 -0.1163 -0.9303 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H21 mock treatment 200240.0 -3770.0 -0.26 146280.0 -2860.0 -0.21 -0.3323 -0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H22 mock treatment 205000.0 989.0 0.07 147800.0 -1340.0 -0.1 -0.0229 -0.19 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H23 mock treatment 197480.0 -6530.0 -0.45 149240.0 99.0 0.01 -0.3096 -0.6953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base H24 mock treatment 200720.0 -3290.0 -0.22 146800.0 -2340.0 -0.17 -0.2818 -0.9922 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I01 mock treatment 213680.0 9670.0 0.66 150520.0 1380.0 0.1 0.5387 0.8075 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I02 mock treatment 212240.0 8230.0 0.56 147320.0 -1820.0 -0.14 0.3009 0.5213 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I03 mock treatment 216080.0 12100.0 0.82 155160.0 6020.0 0.45 0.8986 0.9591 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I04 mock treatment 213280.0 9270.0 0.63 149400.0 259.0 0.02 0.4605 0.7283 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I05 mock treatment 216720.0 12700.0 0.87 153120.0 3980.0 0.3 0.8221 0.8978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I06 mock treatment 210720.0 6710.0 0.46 151680.0 2540.0 0.19 0.4571 0.9235 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I07 mock treatment 209280.0 5270.0 0.36 151360.0 2220.0 0.17 0.3708 0.9378 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I08 mock treatment 216080.0 12100.0 0.82 150920.0 1780.0 0.13 0.6755 0.8105 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I09 mock treatment 217200.0 13200.0 0.9 150120.0 979.0 0.07 0.6874 0.7619 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I10 mock treatment 214480.0 10500.0 0.71 152720.0 3580.0 0.27 0.6931 0.9097 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I11 mock treatment 217840.0 13800.0 0.94 150560.0 1420.0 0.11 0.7414 0.7814 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I12 mock treatment 217600.0 13600.0 0.93 151960.0 2820.0 0.21 0.8035 0.8458 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I13 mock treatment 216360.0 12300.0 0.84 150960.0 1820.0 0.14 0.6911 0.8104 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I14 mock treatment 212720.0 8710.0 0.59 153960.0 4820.0 0.36 0.6735 0.9709 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I15 mock treatment 211840.0 7830.0 0.53 152960.0 3820.0 0.28 0.5784 0.9565 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I16 mock treatment 216440.0 12400.0 0.85 149760.0 619.0 0.05 0.6318 0.7444 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I17 mock treatment 213280.0 9270.0 0.63 148920.0 -221.0 -0.02 0.4352 0.6885 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I18 mock treatment 213360.0 9350.0 0.64 147880.0 -1260.0 -0.09 0.3843 0.5966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I19 mock treatment 214400.0 10400.0 0.71 150480.0 1340.0 0.1 0.5713 0.7987 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I20 mock treatment 207840.0 3830.0 0.26 150560.0 1420.0 0.11 0.2593 0.9207 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I21 mock treatment 200720.0 -3290.0 -0.22 148640.0 -501.0 -0.04 -0.185 -0.8135 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I22 mock treatment 202120.0 -1890.0 -0.13 141960.0 -7180.0 -0.53 -0.4691 -0.8532 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I23 mock treatment 195920.0 -8090.0 -0.55 146080.0 -3060.0 -0.23 -0.5511 -0.9235 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base I24 mock treatment 207600.0 3590.0 0.24 142120.0 -7020.0 -0.52 -0.1965 -0.3405 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J01 mock treatment 194680.0 -9330.0 -0.64 146840.0 -2300.0 -0.17 -0.5709 -0.8666 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J02 mock treatment 197920.0 -6090.0 -0.42 148880.0 -261.0 -0.02 -0.3074 -0.7394 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J03 mock treatment 200520.0 -3490.0 -0.24 147760.0 -1380.0 -0.1 -0.241 -0.9295 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J04 mock treatment 207800.0 3790.0 0.26 152360.0 3220.0 0.24 0.3521 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J05 mock treatment 204000.0 -10.7 0.0 149440.0 299.0 0.02 0.0152 0.6836 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J06 mock treatment 204000.0 -10.7 0.0 147560.0 -1580.0 -0.12 -0.0837 -0.7115 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J07 mock treatment 203400.0 -611.0 -0.04 156880.0 7740.0 0.58 0.3778 0.6543 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J08 mock treatment 203960.0 -50.7 0.0 154640.0 5500.0 0.41 0.287 0.7011 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J09 mock treatment 208960.0 4950.0 0.34 157160.0 8020.0 0.6 0.6606 0.9635 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J10 mock treatment 209400.0 5390.0 0.37 152440.0 3300.0 0.25 0.4334 0.9808 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J11 mock treatment 207240.0 3230.0 0.22 155000.0 5860.0 0.44 0.464 0.9499 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J12 mock treatment 205960.0 1950.0 0.13 150600.0 1460.0 0.11 0.1708 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J13 mock treatment 205760.0 1750.0 0.12 154080.0 4940.0 0.37 0.3443 0.8908 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J14 mock treatment 205600.0 1590.0 0.11 156680.0 7540.0 0.56 0.4734 0.8284 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J15 mock treatment 203800.0 -211.0 -0.01 150480.0 1340.0 0.1 0.0603 0.599 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J16 mock treatment 204480.0 469.0 0.03 148640.0 -501.0 -0.04 -0.0037 -0.0762 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J17 mock treatment 203440.0 -571.0 -0.04 150560.0 1420.0 0.11 0.0472 0.4191 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J18 mock treatment 209880.0 5870.0 0.4 149040.0 -101.0 -0.01 0.2776 0.6937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J19 mock treatment 203760.0 -251.0 -0.02 148080.0 -1060.0 -0.08 -0.0679 -0.8407 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J20 mock treatment 204240.0 229.0 0.02 148080.0 -1060.0 -0.08 -0.0448 -0.5563 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J21 mock treatment 201800.0 -2210.0 -0.15 145320.0 -3820.0 -0.28 -0.3077 -0.9559 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J22 mock treatment 198480.0 -5530.0 -0.38 146320.0 -2820.0 -0.21 -0.4151 -0.9618 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J23 mock treatment 196040.0 -7970.0 -0.54 142920.0 -6220.0 -0.46 -0.7117 -0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base J24 mock treatment 192440.0 -11600.0 -0.79 140120.0 -9020.0 -0.67 -1.0326 -0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K01 mock treatment 218640.0 14600.0 1.0 148920.0 -221.0 -0.02 0.6936 0.6953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K02 mock treatment 225680.0 21700.0 1.48 150600.0 1460.0 0.11 1.1214 0.757 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K03 mock treatment 211400.0 7390.0 0.5 153760.0 4620.0 0.34 0.5993 0.9826 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K04 mock treatment 218760.0 14700.0 1.01 153600.0 4460.0 0.33 0.9457 0.8931 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K05 mock treatment 217200.0 13200.0 0.9 153080.0 3940.0 0.29 0.8431 0.8915 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K06 mock treatment 212960.0 8950.0 0.61 153960.0 4820.0 0.36 0.685 0.9679 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K07 mock treatment 221160.0 17100.0 1.17 155520.0 6380.0 0.47 1.1624 0.9212 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K08 mock treatment 212880.0 8870.0 0.6 153840.0 4700.0 0.35 0.6749 0.9661 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K09 mock treatment 216720.0 12700.0 0.87 154760.0 5620.0 0.42 0.9084 0.9442 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K10 mock treatment 216520.0 12500.0 0.85 153840.0 4700.0 0.35 0.8503 0.9225 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K11 mock treatment 217200.0 13200.0 0.9 152800.0 3660.0 0.27 0.8284 0.8817 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K12 mock treatment 214840.0 10800.0 0.74 153400.0 4260.0 0.32 0.7462 0.9287 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K13 mock treatment 214760.0 10700.0 0.73 155080.0 5940.0 0.44 0.8308 0.9707 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K14 mock treatment 218640.0 14600.0 1.0 151600.0 2460.0 0.18 0.8347 0.8231 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K15 mock treatment 215640.0 11600.0 0.79 155280.0 6140.0 0.46 0.8837 0.9657 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K16 mock treatment 211920.0 7910.0 0.54 151720.0 2580.0 0.19 0.517 0.9033 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K17 mock treatment 208200.0 4190.0 0.29 152000.0 2860.0 0.21 0.3524 0.9895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K18 mock treatment 214480.0 10500.0 0.71 148280.0 -861.0 -0.06 0.4594 0.641 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K19 mock treatment 210560.0 6550.0 0.45 147600.0 -1540.0 -0.11 0.2346 0.509 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K20 mock treatment 214000.0 9990.0 0.68 150160.0 1020.0 0.08 0.5352 0.781 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K21 mock treatment 204280.0 269.0 0.02 149440.0 299.0 0.02 0.0287 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K22 mock treatment 202680.0 -1330.0 -0.09 147760.0 -1380.0 -0.1 -0.1368 -0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K23 mock treatment 198640.0 -5370.0 -0.37 155360.0 6220.0 0.46 0.0684 0.1159 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base K24 mock treatment 211040.0 7030.0 0.48 144160.0 -4980.0 -0.37 0.0767 0.1266 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L01 mock treatment 191760.0 -12300.0 -0.84 149280.0 139.0 0.01 -0.5833 -0.6983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L02 mock treatment 195600.0 -8410.0 -0.57 151760.0 2620.0 0.19 -0.2676 -0.4419 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L03 mock treatment 200880.0 -3130.0 -0.21 147600.0 -1540.0 -0.11 -0.232 -0.9576 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L04 mock treatment 200480.0 -3530.0 -0.24 151520.0 2380.0 0.18 -0.045 -0.1506 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L05 mock treatment 202800.0 -1210.0 -0.08 150320.0 1180.0 0.09 0.0037 0.0306 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L06 mock treatment 208120.0 4110.0 0.28 152520.0 3380.0 0.25 0.3759 0.9985 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L07 mock treatment 204320.0 309.0 0.02 153880.0 4740.0 0.35 0.2643 0.748 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L08 mock treatment 202200.0 -1810.0 -0.12 152080.0 2940.0 0.22 0.0674 0.2683 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L09 mock treatment 204280.0 269.0 0.02 153200.0 4060.0 0.3 0.2266 0.7487 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L10 mock treatment 207360.0 3350.0 0.23 157200.0 8060.0 0.6 0.5856 0.9124 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L11 mock treatment 209440.0 5430.0 0.37 157600.0 8460.0 0.63 0.7069 0.9679 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L12 mock treatment 207280.0 3270.0 0.22 151440.0 2300.0 0.17 0.2786 0.9915 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L13 mock treatment 204720.0 709.0 0.05 153720.0 4580.0 0.34 0.2752 0.7994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L14 mock treatment 212680.0 8670.0 0.59 152120.0 2980.0 0.22 0.5747 0.9104 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L15 mock treatment 206640.0 2630.0 0.18 149680.0 539.0 0.04 0.1551 0.8445 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L16 mock treatment 210000.0 5990.0 0.41 151360.0 2220.0 0.17 0.4055 0.9206 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L17 mock treatment 199120.0 -4890.0 -0.33 148880.0 -261.0 -0.02 -0.2495 -0.747 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L18 mock treatment 206040.0 2030.0 0.14 146840.0 -2300.0 -0.17 -0.0233 -0.1057 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L19 mock treatment 206240.0 2230.0 0.15 150560.0 1420.0 0.11 0.1821 0.9842 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L20 mock treatment 206120.0 2110.0 0.14 144800.0 -4340.0 -0.32 -0.1268 -0.3585 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L21 mock treatment 204160.0 149.0 0.01 148440.0 -701.0 -0.05 -0.0297 -0.5586 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L22 mock treatment 200800.0 -3210.0 -0.22 144040.0 -5100.0 -0.38 -0.4232 -0.9658 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L23 mock treatment 198160.0 -5850.0 -0.4 145720.0 -3420.0 -0.25 -0.4621 -0.9765 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base L24 mock treatment 196720.0 -7290.0 -0.5 145960.0 -3180.0 -0.24 -0.5189 -0.9425 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M01 mock treatment 231320.0 27300.0 1.86 152600.0 3460.0 0.26 1.4986 0.7973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M02 mock treatment 219240.0 15200.0 1.04 156400.0 7260.0 0.54 1.1162 0.9537 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M03 mock treatment 219560.0 15500.0 1.06 156680.0 7540.0 0.56 1.1464 0.9558 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M04 mock treatment 215360.0 11300.0 0.77 161560.0 12400.0 0.92 1.2007 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M05 mock treatment 228040.0 24000.0 1.64 155640.0 6500.0 0.48 1.5004 0.8784 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M06 mock treatment 219520.0 15500.0 1.06 157560.0 8420.0 0.63 1.1907 0.9688 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M07 mock treatment 226200.0 22200.0 1.51 158280.0 9140.0 0.68 1.5507 0.9349 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M08 mock treatment 219080.0 15100.0 1.03 156680.0 7540.0 0.56 1.1232 0.9595 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M09 mock treatment 215600.0 11600.0 0.79 156720.0 7580.0 0.56 0.9576 0.9864 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M10 mock treatment 220880.0 16900.0 1.15 166040.0 16900.0 1.26 1.7026 0.999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M11 mock treatment 220280.0 16300.0 1.11 158800.0 9660.0 0.72 1.2926 0.978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M12 mock treatment 214880.0 10900.0 0.74 158360.0 9220.0 0.69 1.0092 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M13 mock treatment 215040.0 11000.0 0.75 157160.0 8020.0 0.6 0.9537 0.9935 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M14 mock treatment 214120.0 10100.0 0.69 157040.0 7900.0 0.59 0.9031 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M15 mock treatment 213560.0 9550.0 0.65 157480.0 8340.0 0.62 0.8992 0.9997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M16 mock treatment 213200.0 9190.0 0.63 158640.0 9500.0 0.71 0.9429 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M17 mock treatment 213360.0 9350.0 0.64 154600.0 5460.0 0.41 0.738 0.9763 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M18 mock treatment 217800.0 13800.0 0.94 157200.0 8060.0 0.6 1.0889 0.9764 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M19 mock treatment 212120.0 8110.0 0.55 154960.0 5820.0 0.43 0.6972 0.9927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M20 mock treatment 209520.0 5510.0 0.38 154880.0 5740.0 0.43 0.5676 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M21 mock treatment 213880.0 9870.0 0.67 150880.0 1740.0 0.13 0.5673 0.8279 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M22 mock treatment 205520.0 1510.0 0.1 150080.0 939.0 0.07 0.1222 0.9822 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M23 mock treatment 214440.0 10400.0 0.71 153920.0 4780.0 0.36 0.7543 0.9487 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base M24 mock treatment 195080.0 -8930.0 -0.61 149040.0 -101.0 -0.01 -0.4359 -0.7158 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N01 mock treatment 197160.0 -6850.0 -0.47 148920.0 -221.0 -0.02 -0.3419 -0.7316 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N02 mock treatment 201320.0 -2690.0 -0.18 158040.0 8900.0 0.66 0.3386 0.4927 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N03 mock treatment 202200.0 -1810.0 -0.12 152440.0 3300.0 0.25 0.0863 0.3141 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N04 mock treatment 207480.0 3470.0 0.24 152120.0 2980.0 0.22 0.324 0.9995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N05 mock treatment 212960.0 8950.0 0.61 156720.0 7580.0 0.56 0.8303 0.9992 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N06 mock treatment 203960.0 -50.7 0.0 157000.0 7860.0 0.58 0.4112 0.7029 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N07 mock treatment 206440.0 2430.0 0.17 155240.0 6100.0 0.45 0.4381 0.9066 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N08 mock treatment 205760.0 1750.0 0.12 155520.0 6380.0 0.47 0.42 0.8581 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N09 mock treatment 206560.0 2550.0 0.17 158120.0 8980.0 0.67 0.5954 0.8623 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N10 mock treatment 212080.0 8070.0 0.55 163360.0 14200.0 1.06 1.1373 0.9535 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N11 mock treatment 207360.0 3350.0 0.23 159160.0 10000.0 0.75 0.6887 0.8832 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N12 mock treatment 206520.0 2510.0 0.17 153800.0 4660.0 0.35 0.3662 0.947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N13 mock treatment 212040.0 8030.0 0.55 158240.0 9100.0 0.68 0.8659 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N14 mock treatment 211280.0 7270.0 0.5 157040.0 7900.0 0.59 0.7661 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N15 mock treatment 218120.0 14100.0 0.96 154760.0 5620.0 0.42 0.9759 0.9304 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N16 mock treatment 209960.0 5950.0 0.41 155800.0 6660.0 0.5 0.6373 0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N17 mock treatment 208440.0 4430.0 0.3 155720.0 6580.0 0.49 0.5598 0.973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N18 mock treatment 212680.0 8670.0 0.59 162360.0 13200.0 0.98 1.1136 0.9703 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N19 mock treatment 208040.0 4030.0 0.27 157480.0 8340.0 0.62 0.6331 0.9328 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N20 mock treatment 206000.0 1990.0 0.14 150720.0 1580.0 0.12 0.179 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N21 mock treatment 206560.0 2550.0 0.17 149200.0 59.0 0.0 0.126 0.7247 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N22 mock treatment 199440.0 -4570.0 -0.31 145040.0 -4100.0 -0.31 -0.4362 -0.9999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N23 mock treatment 201200.0 -2810.0 -0.19 148640.0 -501.0 -0.04 -0.1619 -0.8292 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base N24 mock treatment 192200.0 -11800.0 -0.81 145520.0 -3620.0 -0.27 -0.7599 -0.895 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O01 mock treatment 223600.0 19600.0 1.34 149400.0 259.0 0.02 0.958 0.7172 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O02 mock treatment 218560.0 14500.0 0.99 156640.0 7500.0 0.56 1.0961 0.963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O03 mock treatment 215520.0 11500.0 0.78 154000.0 4860.0 0.36 0.8106 0.9382 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O04 mock treatment 214200.0 10200.0 0.69 157160.0 8020.0 0.6 0.9132 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O05 mock treatment 215600.0 11600.0 0.79 155240.0 6100.0 0.45 0.8797 0.9654 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O06 mock treatment 210160.0 6150.0 0.42 155200.0 6060.0 0.45 0.6153 0.9993 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O07 mock treatment 210120.0 6110.0 0.42 153480.0 4340.0 0.32 0.5229 0.9921 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O08 mock treatment 214760.0 10700.0 0.73 155360.0 6220.0 0.46 0.8455 0.9754 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O09 mock treatment 214400.0 10400.0 0.71 158320.0 9180.0 0.68 0.9839 0.9998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O10 mock treatment 217400.0 13400.0 0.91 156960.0 7820.0 0.58 1.057 0.9764 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O11 mock treatment 209920.0 5910.0 0.4 160240.0 11100.0 0.83 0.869 0.9455 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O12 mock treatment 213760.0 9750.0 0.66 153640.0 4500.0 0.33 0.7068 0.9496 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O13 mock treatment 209400.0 5390.0 0.37 156640.0 7500.0 0.56 0.6545 0.9794 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O14 mock treatment 205040.0 1030.0 0.07 154240.0 5100.0 0.38 0.318 0.8239 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O15 mock treatment 208040.0 4030.0 0.27 157760.0 8620.0 0.64 0.6478 0.9284 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O16 mock treatment 208000.0 3990.0 0.27 157560.0 8420.0 0.63 0.6354 0.9302 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O17 mock treatment 206240.0 2230.0 0.15 153560.0 4420.0 0.33 0.34 0.9385 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O18 mock treatment 206080.0 2070.0 0.14 154600.0 5460.0 0.41 0.3871 0.8999 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O19 mock treatment 201760.0 -2250.0 -0.15 151200.0 2060.0 0.15 -1.0E-4 -7.0E-4 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O20 mock treatment 204920.0 909.0 0.06 147600.0 -1540.0 -0.11 -0.0373 -0.2858 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O21 mock treatment 201840.0 -2170.0 -0.15 146800.0 -2340.0 -0.17 -0.2278 -0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O22 mock treatment 194480.0 -9530.0 -0.65 145320.0 -3820.0 -0.28 -0.6606 -0.9313 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O23 mock treatment 196080.0 -7930.0 -0.54 147360.0 -1780.0 -0.13 -0.4761 -0.8551 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base O24 mock treatment 187920.0 -16100.0 -1.1 143360.0 -5780.0 -0.43 -1.0799 -0.9165 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P01 mock treatment 191840.0 -12200.0 -0.83 151280.0 2140.0 0.16 -0.4742 -0.5612 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P02 mock treatment 200840.0 -3170.0 -0.22 152960.0 3820.0 0.28 0.0481 0.1348 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P03 mock treatment 201840.0 -2170.0 -0.15 152480.0 3340.0 0.25 0.0711 0.2457 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P04 mock treatment 196680.0 -7330.0 -0.5 149720.0 579.0 0.04 -0.3229 -0.6438 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P05 mock treatment 195880.0 -8130.0 -0.55 151040.0 1900.0 0.14 -0.292 -0.5105 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P06 mock treatment 195160.0 -8850.0 -0.6 152320.0 3180.0 0.24 -0.2594 -0.4002 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P07 mock treatment 196160.0 -7850.0 -0.54 152160.0 3020.0 0.22 -0.2196 -0.3783 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P08 mock treatment 197640.0 -6370.0 -0.43 152840.0 3700.0 0.28 -0.1125 -0.2187 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P09 mock treatment 197000.0 -7010.0 -0.48 155520.0 6380.0 0.47 -0.0023 -0.0034 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P10 mock treatment 198720.0 -5290.0 -0.36 151480.0 2340.0 0.17 -0.132 -0.3295 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P11 mock treatment 200200.0 -3810.0 -0.26 154760.0 5620.0 0.42 0.112 0.2275 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P12 mock treatment 202840.0 -1170.0 -0.08 152680.0 3540.0 0.26 0.1298 0.4717 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P13 mock treatment 198920.0 -5090.0 -0.35 147240.0 -1900.0 -0.14 -0.3455 -0.9217 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P14 mock treatment 203360.0 -651.0 -0.04 152080.0 2940.0 0.22 0.1233 0.5525 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P15 mock treatment 198600.0 -5410.0 -0.37 150800.0 1660.0 0.12 -0.1735 -0.4461 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P16 mock treatment 196800.0 -7210.0 -0.49 149320.0 179.0 0.01 -0.3382 -0.6877 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P17 mock treatment 200280.0 -3730.0 -0.25 151440.0 2300.0 0.17 -0.0589 -0.192 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P18 mock treatment 197800.0 -6210.0 -0.42 149320.0 179.0 0.01 -0.29 -0.6845 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P19 mock treatment 192760.0 -11300.0 -0.77 149560.0 419.0 0.03 -0.5203 -0.6778 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P20 mock treatment 191800.0 -12200.0 -0.83 146440.0 -2700.0 -0.2 -0.7308 -0.8533 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P21 mock treatment 191720.0 -12300.0 -0.84 145520.0 -3620.0 -0.27 -0.7831 -0.8896 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P22 mock treatment 193680.0 -10300.0 -0.7 144600.0 -4540.0 -0.34 -0.737 -0.9434 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P23 mock treatment 187400.0 -16600.0 -1.13 143240.0 -5900.0 -0.44 -1.1113 -0.9149 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Base P24 mock treatment 189720.0 -14300.0 -0.97 142640.0 -6500.0 -0.48 -1.0311 -0.9478 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A01 positive control 605600.0 402000.0 27.38 472280.0 323000.0 24.05 36.366 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A02 positive control 588080.0 384000.0 26.18 461000.0 312000.0 23.21 34.9278 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A03 positive control 599600.0 396000.0 26.97 459560.0 310000.0 23.1 35.4074 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A04 positive control 598320.0 394000.0 26.88 467440.0 318000.0 23.69 35.7604 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A05 positive control 597760.0 394000.0 26.84 468040.0 319000.0 23.73 35.7649 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A06 positive control 594120.0 390000.0 26.6 455960.0 307000.0 22.84 34.9537 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A07 positive control 598120.0 394000.0 26.87 458520.0 309000.0 23.03 35.2813 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A08 positive control 599760.0 396000.0 26.98 460360.0 311000.0 23.16 35.4572 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A09 positive control 596520.0 393000.0 26.76 458680.0 310000.0 23.04 35.2126 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A10 positive control 599440.0 395000.0 26.96 464880.0 316000.0 23.5 35.6796 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A11 positive control 600000.0 396000.0 27.0 464080.0 315000.0 23.44 35.6645 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A12 positive control 609080.0 405000.0 27.62 468760.0 320000.0 23.79 36.3485 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A13 positive control 601320.0 397000.0 27.09 457200.0 308000.0 22.93 35.3661 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A14 positive control 599120.0 395000.0 26.94 460200.0 311000.0 23.15 35.4179 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A15 positive control 596600.0 393000.0 26.77 463480.0 314000.0 23.4 35.469 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A16 positive control 597160.0 393000.0 26.8 460880.0 312000.0 23.2 35.3592 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A17 positive control 594560.0 391000.0 26.63 466160.0 317000.0 23.59 35.5117 0.9982 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A18 positive control 602520.0 399000.0 27.17 463280.0 314000.0 23.38 35.7439 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A19 positive control 602080.0 398000.0 27.14 466320.0 317000.0 23.61 35.8827 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A20 positive control 602080.0 398000.0 27.14 468080.0 319000.0 23.74 35.9753 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A21 positive control 604680.0 401000.0 27.32 469680.0 321000.0 23.86 36.1849 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A22 positive control 606040.0 402000.0 27.41 461720.0 313000.0 23.26 35.8315 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A23 positive control 606040.0 402000.0 27.41 468040.0 319000.0 23.73 36.1641 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos A24 positive control 607240.0 403000.0 27.49 478440.0 329000.0 24.51 36.7693 0.9984 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B01 positive control 590520.0 387000.0 26.35 458120.0 309000.0 23.0 34.8938 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B02 positive control 592000.0 388000.0 26.45 457920.0 309000.0 22.98 34.9547 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B03 positive control 592520.0 389000.0 26.49 453200.0 304000.0 22.63 34.7313 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B04 positive control 593120.0 389000.0 26.53 453280.0 304000.0 22.64 34.7645 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B05 positive control 601440.0 397000.0 27.1 450960.0 302000.0 22.46 35.0435 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B06 positive control 594680.0 391000.0 26.63 445200.0 296000.0 22.03 34.4144 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B07 positive control 595000.0 391000.0 26.66 447640.0 298000.0 22.22 34.5583 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B08 positive control 592880.0 389000.0 26.51 438760.0 290000.0 21.56 33.9887 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B09 positive control 589000.0 385000.0 26.25 445120.0 296000.0 22.03 34.1364 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B10 positive control 588760.0 385000.0 26.23 451520.0 302000.0 22.51 34.4617 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B11 positive control 592720.0 389000.0 26.5 451960.0 303000.0 22.54 34.6757 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B12 positive control 600160.0 396000.0 27.01 452000.0 303000.0 22.54 35.0365 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B13 positive control 598760.0 395000.0 26.91 451680.0 303000.0 22.52 34.9522 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B14 positive control 598120.0 394000.0 26.87 451440.0 302000.0 22.5 34.9087 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B15 positive control 599720.0 396000.0 26.98 442040.0 293000.0 21.8 34.4911 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B16 positive control 593680.0 390000.0 26.57 451240.0 302000.0 22.48 34.6841 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B17 positive control 592040.0 388000.0 26.45 454440.0 305000.0 22.72 34.7734 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B18 positive control 597800.0 394000.0 26.85 450680.0 302000.0 22.44 34.8532 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B19 positive control 599480.0 395000.0 26.96 440320.0 291000.0 21.67 34.389 0.9941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B20 positive control 595920.0 392000.0 26.72 453760.0 305000.0 22.67 34.9247 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B21 positive control 594040.0 390000.0 26.59 453320.0 304000.0 22.64 34.8109 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B22 positive control 601160.0 397000.0 27.08 452920.0 304000.0 22.61 35.1331 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B23 positive control 591000.0 387000.0 26.38 456280.0 307000.0 22.86 34.8201 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos B24 positive control 603360.0 399000.0 27.23 472720.0 324000.0 24.08 36.2812 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C01 positive control 606600.0 403000.0 27.45 471160.0 322000.0 23.97 36.3553 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C02 positive control 601440.0 397000.0 27.1 453920.0 305000.0 22.68 35.1992 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C03 positive control 608520.0 405000.0 27.58 443120.0 294000.0 21.88 34.9722 0.9934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C04 positive control 606600.0 403000.0 27.45 458080.0 309000.0 22.99 35.6669 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C05 positive control 612680.0 409000.0 27.86 457560.0 308000.0 22.95 35.9327 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C06 positive control 597880.0 394000.0 26.85 444520.0 295000.0 21.98 34.5329 0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C07 positive control 603440.0 399000.0 27.23 459480.0 310000.0 23.1 35.5883 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C08 positive control 602880.0 399000.0 27.19 449680.0 301000.0 22.37 35.0455 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C09 positive control 598760.0 395000.0 26.91 452360.0 303000.0 22.57 34.9879 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C10 positive control 600120.0 396000.0 27.01 461880.0 313000.0 23.28 35.5545 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C11 positive control 601040.0 397000.0 27.07 460040.0 311000.0 23.14 35.502 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C12 positive control 612240.0 408000.0 27.83 467480.0 318000.0 23.69 36.4335 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C13 positive control 608320.0 404000.0 27.56 450920.0 302000.0 22.46 35.373 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C14 positive control 609200.0 405000.0 27.62 454320.0 305000.0 22.71 35.5944 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C15 positive control 607000.0 403000.0 27.47 449640.0 300000.0 22.37 35.242 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C16 positive control 602960.0 399000.0 27.2 463320.0 314000.0 23.38 35.7672 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C17 positive control 602280.0 398000.0 27.15 448040.0 299000.0 22.25 34.9303 0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C18 positive control 602080.0 398000.0 27.14 452160.0 303000.0 22.55 35.1375 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C19 positive control 603600.0 400000.0 27.24 456960.0 308000.0 22.91 35.4634 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C20 positive control 602400.0 398000.0 27.16 445560.0 296000.0 22.06 34.8056 0.9947 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C21 positive control 600800.0 397000.0 27.05 460600.0 311000.0 23.18 35.5199 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C22 positive control 595320.0 391000.0 26.68 446640.0 297000.0 22.14 34.5211 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C23 positive control 605120.0 401000.0 27.35 456000.0 307000.0 22.84 35.4861 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos C24 positive control 604600.0 401000.0 27.31 470600.0 321000.0 23.93 36.2294 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D01 positive control 602000.0 398000.0 27.13 463080.0 314000.0 23.37 35.7083 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D02 positive control 605960.0 402000.0 27.4 445000.0 296000.0 22.02 34.9477 0.9941 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D03 positive control 621640.0 418000.0 28.47 433600.0 284000.0 21.17 35.1037 0.9894 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D04 positive control 617000.0 413000.0 28.16 445040.0 296000.0 22.02 35.482 0.9926 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D05 positive control 604840.0 401000.0 27.33 440200.0 291000.0 21.66 34.6411 0.9934 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D06 positive control 604000.0 400000.0 27.27 441080.0 292000.0 21.73 34.6469 0.9937 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D07 positive control 603800.0 400000.0 27.26 440640.0 291000.0 21.7 34.6141 0.9936 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D08 positive control 603440.0 399000.0 27.23 445920.0 297000.0 22.09 34.8746 0.9946 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D09 positive control 601480.0 397000.0 27.1 450160.0 301000.0 22.4 35.0033 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D10 positive control 605720.0 402000.0 27.39 470440.0 321000.0 23.91 36.275 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D11 positive control 606800.0 403000.0 27.46 450800.0 302000.0 22.45 35.2934 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D12 positive control 611320.0 407000.0 27.77 451360.0 302000.0 22.49 35.5408 0.9945 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D13 positive control 609160.0 405000.0 27.62 454360.0 305000.0 22.72 35.5946 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D14 positive control 606560.0 403000.0 27.44 452000.0 303000.0 22.54 35.345 0.9952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D15 positive control 594880.0 391000.0 26.65 450920.0 302000.0 22.46 34.7251 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D16 positive control 597080.0 393000.0 26.8 448040.0 299000.0 22.25 34.6796 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D17 positive control 602720.0 399000.0 27.18 457800.0 309000.0 22.97 35.4651 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D18 positive control 604080.0 400000.0 27.28 458080.0 309000.0 22.99 35.5454 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D19 positive control 594200.0 390000.0 26.6 446000.0 297000.0 22.09 34.4334 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D20 positive control 604640.0 401000.0 27.31 447760.0 299000.0 22.23 35.0293 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D21 positive control 599480.0 395000.0 26.96 442080.0 293000.0 21.8 34.4816 0.9944 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D22 positive control 606240.0 402000.0 27.42 450240.0 301000.0 22.41 35.237 0.995 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D23 positive control 601800.0 398000.0 27.12 451680.0 303000.0 22.52 35.0987 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos D24 positive control 609520.0 406000.0 27.65 458600.0 309000.0 23.03 35.8351 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E01 positive control 618320.0 414000.0 28.25 469240.0 320000.0 23.82 36.8193 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E02 positive control 612640.0 409000.0 27.86 465560.0 316000.0 23.55 36.3518 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E03 positive control 612560.0 409000.0 27.85 467880.0 319000.0 23.72 36.47 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E04 positive control 614480.0 410000.0 27.98 467320.0 318000.0 23.68 36.5331 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E05 positive control 619960.0 416000.0 28.36 465000.0 316000.0 23.51 36.6752 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E06 positive control 611680.0 408000.0 27.79 467360.0 318000.0 23.68 36.4002 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E07 positive control 616680.0 413000.0 28.13 467240.0 318000.0 23.68 36.6349 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E08 positive control 622520.0 419000.0 28.53 464600.0 315000.0 23.48 36.7775 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E09 positive control 610280.0 406000.0 27.7 473080.0 324000.0 24.11 36.6338 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E10 positive control 616720.0 413000.0 28.14 476360.0 327000.0 24.35 37.1168 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E11 positive control 608480.0 404000.0 27.58 468520.0 319000.0 23.77 36.307 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E12 positive control 616760.0 413000.0 28.14 472800.0 324000.0 24.09 36.9314 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E13 positive control 615640.0 412000.0 28.06 472120.0 323000.0 24.04 36.8416 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E14 positive control 622120.0 418000.0 28.51 470560.0 321000.0 23.92 37.0719 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E15 positive control 619240.0 415000.0 28.31 470240.0 321000.0 23.9 36.9162 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E16 positive control 615560.0 412000.0 28.06 469360.0 320000.0 23.83 36.6925 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E17 positive control 613520.0 410000.0 27.92 468240.0 319000.0 23.75 36.5352 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E18 positive control 613680.0 410000.0 27.93 458240.0 309000.0 23.01 36.0167 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E19 positive control 617160.0 413000.0 28.17 463160.0 314000.0 23.37 36.4434 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E20 positive control 616680.0 413000.0 28.13 472440.0 323000.0 24.06 36.9086 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E21 positive control 612640.0 409000.0 27.86 463280.0 314000.0 23.38 36.2318 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E22 positive control 618800.0 415000.0 28.28 464960.0 316000.0 23.51 36.6171 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E23 positive control 616080.0 412000.0 28.09 467440.0 318000.0 23.69 36.6165 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos E24 positive control 608600.0 405000.0 27.58 466640.0 317000.0 23.63 36.2138 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F01 positive control 612120.0 408000.0 27.82 463480.0 314000.0 23.4 36.2172 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F02 positive control 617160.0 413000.0 28.17 457600.0 308000.0 22.96 36.1507 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F03 positive control 613720.0 410000.0 27.93 450040.0 301000.0 22.39 35.587 0.994 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F04 positive control 619120.0 415000.0 28.3 466240.0 317000.0 23.6 36.6999 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F05 positive control 615440.0 411000.0 28.05 460040.0 311000.0 23.14 36.1962 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F06 positive control 611600.0 408000.0 27.79 460640.0 311000.0 23.18 36.0427 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F07 positive control 611000.0 407000.0 27.75 463120.0 314000.0 23.37 36.1443 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F08 positive control 616840.0 413000.0 28.15 467400.0 318000.0 23.69 36.6511 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F09 positive control 610760.0 407000.0 27.73 456920.0 308000.0 22.91 35.8064 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F10 positive control 613520.0 410000.0 27.92 471000.0 322000.0 23.95 36.6805 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F11 positive control 608960.0 405000.0 27.61 467160.0 318000.0 23.67 36.2586 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F12 positive control 609320.0 405000.0 27.63 470720.0 322000.0 23.93 36.4633 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F13 positive control 614720.0 411000.0 28.0 469640.0 320000.0 23.85 36.6668 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F14 positive control 609720.0 406000.0 27.66 466160.0 317000.0 23.59 36.2426 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F15 positive control 615240.0 411000.0 28.04 465720.0 317000.0 23.56 36.4855 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F16 positive control 613920.0 410000.0 27.95 468000.0 319000.0 23.73 36.5419 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F17 positive control 608160.0 404000.0 27.55 467720.0 319000.0 23.71 36.2495 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F18 positive control 609920.0 406000.0 27.67 459000.0 310000.0 23.06 35.8754 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F19 positive control 610760.0 407000.0 27.73 459320.0 310000.0 23.09 35.9327 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F20 positive control 619920.0 416000.0 28.36 464880.0 316000.0 23.5 36.6669 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F21 positive control 607840.0 404000.0 27.53 464720.0 316000.0 23.49 36.0762 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F22 positive control 606960.0 403000.0 27.47 456000.0 307000.0 22.84 35.5748 0.9958 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F23 positive control 605680.0 402000.0 27.38 465000.0 316000.0 23.51 35.9868 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos F24 positive control 602720.0 399000.0 27.18 459040.0 310000.0 23.06 35.5304 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G01 positive control 620880.0 417000.0 28.42 487040.0 338000.0 25.15 37.8794 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G02 positive control 625800.0 422000.0 28.76 480320.0 331000.0 24.65 37.763 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G03 positive control 622400.0 418000.0 28.52 483720.0 335000.0 24.9 37.778 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G04 positive control 631400.0 427000.0 29.14 476640.0 327000.0 24.37 37.8393 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G05 positive control 629840.0 426000.0 29.03 482280.0 333000.0 24.79 38.0609 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G06 positive control 626600.0 423000.0 28.81 479400.0 330000.0 24.58 37.7531 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G07 positive control 624920.0 421000.0 28.7 472320.0 323000.0 24.05 37.2995 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G08 positive control 619480.0 415000.0 28.33 481120.0 332000.0 24.71 37.5004 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G09 positive control 628840.0 425000.0 28.96 484240.0 335000.0 24.94 38.1158 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G10 positive control 623000.0 419000.0 28.57 480840.0 332000.0 24.69 37.6554 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G11 positive control 628680.0 425000.0 28.95 483200.0 334000.0 24.86 38.0534 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G12 positive control 628240.0 424000.0 28.92 482680.0 334000.0 24.82 38.0048 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G13 positive control 628880.0 425000.0 28.97 483800.0 335000.0 24.91 38.0946 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G14 positive control 629320.0 425000.0 29.0 479920.0 331000.0 24.62 37.9116 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G15 positive control 630160.0 426000.0 29.05 482280.0 333000.0 24.79 38.0763 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G16 positive control 620640.0 417000.0 28.4 482600.0 333000.0 24.82 37.6342 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G17 positive control 626880.0 423000.0 28.83 478560.0 329000.0 24.52 37.7224 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G18 positive control 613400.0 409000.0 27.91 479120.0 330000.0 24.56 37.102 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G19 positive control 624720.0 421000.0 28.68 470320.0 321000.0 23.9 37.1846 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G20 positive control 628240.0 424000.0 28.92 475200.0 326000.0 24.27 37.6111 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G21 positive control 618200.0 414000.0 28.24 469880.0 321000.0 23.87 36.8472 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G22 positive control 622360.0 418000.0 28.52 471720.0 323000.0 24.01 37.1445 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G23 positive control 620800.0 417000.0 28.42 470680.0 322000.0 23.93 37.0146 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos G24 positive control 611960.0 408000.0 27.81 472840.0 324000.0 24.09 36.7021 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H01 positive control 616720.0 413000.0 28.14 470400.0 321000.0 23.91 36.8032 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H02 positive control 624160.0 420000.0 28.64 483120.0 334000.0 24.86 37.8313 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H03 positive control 624800.0 421000.0 28.69 476120.0 327000.0 24.34 37.4937 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H04 positive control 624480.0 420000.0 28.67 477920.0 329000.0 24.47 37.573 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H05 positive control 630440.0 426000.0 29.07 482000.0 333000.0 24.77 38.0751 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H06 positive control 629040.0 425000.0 28.98 481640.0 332000.0 24.75 37.9886 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H07 positive control 621200.0 417000.0 28.44 483920.0 335000.0 24.92 37.7307 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H08 positive control 614760.0 411000.0 28.0 466560.0 317000.0 23.62 36.5066 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H09 positive control 621040.0 417000.0 28.43 479760.0 331000.0 24.61 37.504 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H10 positive control 625000.0 421000.0 28.7 482880.0 334000.0 24.84 37.8591 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H11 positive control 617880.0 414000.0 28.22 481280.0 332000.0 24.72 37.4317 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H12 positive control 626640.0 423000.0 28.81 481960.0 333000.0 24.77 37.8898 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H13 positive control 626760.0 423000.0 28.82 481080.0 332000.0 24.71 37.8492 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H14 positive control 616960.0 413000.0 28.15 472880.0 324000.0 24.09 36.9453 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H15 positive control 620680.0 417000.0 28.41 475400.0 326000.0 24.28 37.2572 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H16 positive control 624520.0 421000.0 28.67 477680.0 329000.0 24.45 37.5623 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H17 positive control 618280.0 414000.0 28.24 484320.0 335000.0 24.95 37.611 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H18 positive control 614880.0 411000.0 28.01 476520.0 327000.0 24.37 37.0365 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H19 positive control 621240.0 417000.0 28.45 474840.0 326000.0 24.24 37.2547 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H20 positive control 618160.0 414000.0 28.24 468560.0 319000.0 23.77 36.7758 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H21 positive control 617600.0 414000.0 28.2 466040.0 317000.0 23.59 36.6161 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H22 positive control 613440.0 409000.0 27.91 465120.0 316000.0 23.52 36.3672 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H23 positive control 612680.0 409000.0 27.86 467040.0 318000.0 23.66 36.4316 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos H24 positive control 601240.0 397000.0 27.08 467320.0 318000.0 23.68 35.8948 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I01 positive control 621680.0 418000.0 28.48 480000.0 331000.0 24.62 37.5475 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I02 positive control 617000.0 413000.0 28.16 471440.0 322000.0 23.99 36.8714 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I03 positive control 619760.0 416000.0 28.34 475680.0 327000.0 24.3 37.2276 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I04 positive control 621720.0 418000.0 28.48 469680.0 321000.0 23.86 37.0063 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I05 positive control 625960.0 422000.0 28.77 479960.0 331000.0 24.62 37.7517 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I06 positive control 619400.0 415000.0 28.32 473200.0 324000.0 24.12 37.0797 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I07 positive control 627880.0 424000.0 28.9 472440.0 323000.0 24.06 37.4485 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I08 positive control 623040.0 419000.0 28.57 474880.0 326000.0 24.24 37.3436 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I09 positive control 620120.0 416000.0 28.37 474960.0 326000.0 24.25 37.2071 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I10 positive control 625160.0 421000.0 28.71 473200.0 324000.0 24.12 37.3574 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I11 positive control 618560.0 415000.0 28.26 475000.0 326000.0 24.25 37.134 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I12 positive control 619520.0 416000.0 28.33 477360.0 328000.0 24.43 37.3044 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I13 positive control 610560.0 407000.0 27.72 478480.0 329000.0 24.51 36.9314 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I14 positive control 621040.0 417000.0 28.43 479120.0 330000.0 24.56 37.4703 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I15 positive control 622720.0 419000.0 28.55 483600.0 334000.0 24.89 37.7871 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I16 positive control 615000.0 411000.0 28.02 472880.0 324000.0 24.09 36.8508 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I17 positive control 621160.0 417000.0 28.44 469680.0 321000.0 23.86 36.9793 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I18 positive control 616680.0 413000.0 28.13 474520.0 325000.0 24.22 37.0181 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I19 positive control 617440.0 413000.0 28.19 471640.0 322000.0 24.0 36.9031 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I20 positive control 613960.0 410000.0 27.95 472800.0 324000.0 24.09 36.7964 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I21 positive control 615520.0 412000.0 28.06 467920.0 319000.0 23.73 36.6148 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I22 positive control 607560.0 404000.0 27.51 465280.0 316000.0 23.53 36.0921 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I23 positive control 612720.0 409000.0 27.86 462240.0 313000.0 23.3 36.1809 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos I24 positive control 612320.0 408000.0 27.84 465960.0 317000.0 23.58 36.3574 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J01 positive control 620320.0 416000.0 28.38 479800.0 331000.0 24.61 37.4714 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J02 positive control 614400.0 410000.0 27.98 476840.0 328000.0 24.39 37.0302 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J03 positive control 620120.0 416000.0 28.37 468600.0 319000.0 23.78 36.8723 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J04 positive control 628240.0 424000.0 28.92 476120.0 327000.0 24.34 37.6596 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J05 positive control 620080.0 416000.0 28.37 466560.0 317000.0 23.62 36.7631 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J06 positive control 620000.0 416000.0 28.36 475440.0 326000.0 24.29 37.2265 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J07 positive control 628920.0 425000.0 28.97 477400.0 328000.0 24.43 37.7597 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J08 positive control 629920.0 426000.0 29.04 479240.0 330000.0 24.57 37.9047 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J09 positive control 623600.0 420000.0 28.61 467840.0 319000.0 23.72 37.0001 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J10 positive control 624920.0 421000.0 28.7 477160.0 328000.0 24.41 37.5542 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J11 positive control 630640.0 427000.0 29.09 478880.0 330000.0 24.54 37.9205 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J12 positive control 622200.0 418000.0 28.51 482080.0 333000.0 24.78 37.682 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J13 positive control 626600.0 423000.0 28.81 484120.0 335000.0 24.93 38.0015 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J14 positive control 618320.0 414000.0 28.25 474280.0 325000.0 24.2 37.0845 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J15 positive control 612560.0 409000.0 27.85 476000.0 327000.0 24.33 36.8973 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J16 positive control 608920.0 405000.0 27.61 477160.0 328000.0 24.41 36.7829 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J17 positive control 614560.0 411000.0 27.99 473320.0 324000.0 24.13 36.8527 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J18 positive control 612960.0 409000.0 27.88 465680.0 317000.0 23.56 36.3735 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J19 positive control 610680.0 407000.0 27.73 469320.0 320000.0 23.83 36.4552 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J20 positive control 610640.0 407000.0 27.72 468160.0 319000.0 23.74 36.3922 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J21 positive control 608000.0 404000.0 27.54 459080.0 310000.0 23.07 35.787 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J22 positive control 607640.0 404000.0 27.52 461440.0 312000.0 23.24 35.8939 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J23 positive control 602680.0 399000.0 27.18 459640.0 310000.0 23.11 35.5601 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos J24 positive control 601240.0 397000.0 27.08 464360.0 315000.0 23.46 35.739 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K01 positive control 620320.0 416000.0 28.38 477040.0 328000.0 24.4 37.3262 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K02 positive control 622600.0 419000.0 28.54 474400.0 325000.0 24.21 37.2971 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K03 positive control 631240.0 427000.0 29.13 476800.0 328000.0 24.39 37.84 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K04 positive control 627400.0 423000.0 28.87 478680.0 330000.0 24.53 37.7538 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K05 positive control 630640.0 427000.0 29.09 479320.0 330000.0 24.57 37.9437 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K06 positive control 626680.0 423000.0 28.82 474280.0 325000.0 24.2 37.4875 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K07 positive control 635120.0 431000.0 29.39 483240.0 334000.0 24.87 38.3659 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K08 positive control 621240.0 417000.0 28.45 481000.0 332000.0 24.7 37.5789 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K09 positive control 628680.0 425000.0 28.95 473520.0 324000.0 24.14 37.5439 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K10 positive control 627160.0 423000.0 28.85 482360.0 333000.0 24.8 37.9359 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K11 positive control 629080.0 425000.0 28.98 485440.0 336000.0 25.03 38.1905 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K12 positive control 634000.0 430000.0 29.32 477160.0 328000.0 24.41 37.992 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K13 positive control 628920.0 425000.0 28.97 482600.0 333000.0 24.82 38.0334 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K14 positive control 627240.0 423000.0 28.85 468480.0 319000.0 23.77 37.2093 0.9954 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K15 positive control 623440.0 419000.0 28.6 482280.0 333000.0 24.79 37.7523 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K16 positive control 615760.0 412000.0 28.07 473080.0 324000.0 24.11 36.8979 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K17 positive control 625120.0 421000.0 28.71 479120.0 330000.0 24.56 37.667 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K18 positive control 628600.0 425000.0 28.95 478760.0 330000.0 24.53 37.8159 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K19 positive control 618720.0 415000.0 28.27 471800.0 323000.0 24.01 36.9733 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K20 positive control 620600.0 417000.0 28.4 472600.0 323000.0 24.07 37.106 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K21 positive control 611680.0 408000.0 27.79 467680.0 319000.0 23.71 36.4171 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K22 positive control 612760.0 409000.0 27.87 457360.0 308000.0 22.94 35.926 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K23 positive control 610640.0 407000.0 27.72 468960.0 320000.0 23.8 36.4343 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos K24 positive control 611680.0 408000.0 27.79 458480.0 309000.0 23.02 35.9329 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L01 positive control 625000.0 421000.0 28.7 474040.0 325000.0 24.18 37.3939 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L02 positive control 625600.0 422000.0 28.74 464040.0 315000.0 23.44 36.8965 0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L03 positive control 626240.0 422000.0 28.79 482880.0 334000.0 24.84 37.9189 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L04 positive control 626640.0 423000.0 28.81 469600.0 320000.0 23.85 37.2393 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L05 positive control 628200.0 424000.0 28.92 469120.0 320000.0 23.82 37.2892 0.9953 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L06 positive control 630320.0 426000.0 29.06 478800.0 330000.0 24.54 37.9009 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L07 positive control 622200.0 418000.0 28.51 477280.0 328000.0 24.42 37.4294 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L08 positive control 626440.0 422000.0 28.8 482960.0 334000.0 24.85 37.9328 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L09 positive control 625840.0 422000.0 28.76 476680.0 328000.0 24.38 37.5733 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L10 positive control 629600.0 426000.0 29.02 479560.0 330000.0 24.59 37.9062 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L11 positive control 631560.0 428000.0 29.15 475840.0 327000.0 24.32 37.8049 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L12 positive control 621320.0 417000.0 28.45 483720.0 335000.0 24.9 37.7259 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L13 positive control 628080.0 424000.0 28.91 475320.0 326000.0 24.28 37.6097 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L14 positive control 627240.0 423000.0 28.85 476240.0 327000.0 24.34 37.6177 0.9964 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L15 positive control 620680.0 417000.0 28.41 469840.0 321000.0 23.87 36.9646 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L16 positive control 620720.0 417000.0 28.41 468600.0 319000.0 23.78 36.9013 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L17 positive control 624920.0 421000.0 28.7 469320.0 320000.0 23.83 37.1416 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L18 positive control 610880.0 407000.0 27.74 471520.0 322000.0 23.99 36.5806 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L19 positive control 617560.0 414000.0 28.19 459680.0 311000.0 23.11 36.2795 0.9951 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L20 positive control 616800.0 413000.0 28.14 462840.0 314000.0 23.35 36.4092 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L21 positive control 617760.0 414000.0 28.21 462640.0 313000.0 23.33 36.4449 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L22 positive control 612000.0 408000.0 27.82 457920.0 309000.0 22.98 35.9188 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L23 positive control 609120.0 405000.0 27.62 460560.0 311000.0 23.18 35.9189 0.9962 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos L24 positive control 604880.0 401000.0 27.33 455760.0 307000.0 22.82 35.4619 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M01 positive control 629560.0 426000.0 29.01 479040.0 330000.0 24.55 37.8769 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M02 positive control 633120.0 429000.0 29.26 486760.0 338000.0 25.13 38.4548 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M03 positive control 638400.0 434000.0 29.62 479360.0 330000.0 24.58 38.3199 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M04 positive control 628120.0 424000.0 28.91 486520.0 337000.0 25.11 38.2011 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M05 positive control 629720.0 426000.0 29.02 475960.0 327000.0 24.32 37.7225 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M06 positive control 630600.0 427000.0 29.08 483640.0 334000.0 24.9 38.1691 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M07 positive control 635040.0 431000.0 29.39 471560.0 322000.0 24.0 37.7474 0.9949 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M08 positive control 630720.0 427000.0 29.09 486960.0 338000.0 25.14 38.3496 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M09 positive control 624920.0 421000.0 28.7 485920.0 337000.0 25.07 38.0153 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M10 positive control 631160.0 427000.0 29.12 484360.0 335000.0 24.95 38.234 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M11 positive control 639960.0 436000.0 29.72 492920.0 344000.0 25.59 39.1087 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M12 positive control 634280.0 430000.0 29.33 492280.0 343000.0 25.54 38.8012 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M13 positive control 637640.0 434000.0 29.56 489960.0 341000.0 25.37 38.8411 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M14 positive control 635920.0 432000.0 29.45 491800.0 343000.0 25.5 38.855 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M15 positive control 631720.0 428000.0 29.16 488120.0 339000.0 25.23 38.4589 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M16 positive control 626080.0 422000.0 28.78 483200.0 334000.0 24.86 37.928 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M17 positive control 623600.0 420000.0 28.61 476400.0 327000.0 24.36 37.4506 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M18 positive control 625840.0 422000.0 28.76 480720.0 332000.0 24.68 37.7859 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M19 positive control 625440.0 421000.0 28.73 474120.0 325000.0 24.19 37.4193 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M20 positive control 620600.0 417000.0 28.4 471960.0 323000.0 24.03 37.0723 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M21 positive control 623720.0 420000.0 28.61 471040.0 322000.0 23.96 37.1743 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M22 positive control 621040.0 417000.0 28.43 464680.0 316000.0 23.48 36.7104 0.9955 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M23 positive control 616840.0 413000.0 28.15 468760.0 320000.0 23.79 36.7226 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos M24 positive control 608360.0 404000.0 27.57 473320.0 324000.0 24.13 36.5538 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N01 positive control 629640.0 426000.0 29.02 482640.0 333000.0 24.82 38.0702 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N02 positive control 632400.0 428000.0 29.21 486840.0 338000.0 25.13 38.4243 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N03 positive control 632400.0 428000.0 29.21 471400.0 322000.0 23.98 37.6117 0.9952 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N04 positive control 623920.0 420000.0 28.63 485560.0 336000.0 25.04 37.9481 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N05 positive control 632080.0 428000.0 29.18 477280.0 328000.0 24.42 37.9057 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N06 positive control 633960.0 430000.0 29.31 470080.0 321000.0 23.89 37.6174 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N07 positive control 635680.0 432000.0 29.43 486400.0 337000.0 25.1 38.5592 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N08 positive control 632240.0 428000.0 29.2 477800.0 329000.0 24.46 37.9408 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N09 positive control 634800.0 431000.0 29.37 486880.0 338000.0 25.14 38.5421 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N10 positive control 635600.0 432000.0 29.42 479640.0 330000.0 24.6 38.1996 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N11 positive control 634200.0 430000.0 29.33 476440.0 327000.0 24.36 37.9637 0.9957 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N12 positive control 639520.0 436000.0 29.69 490480.0 341000.0 25.4 38.9591 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N13 positive control 629040.0 425000.0 28.98 478040.0 329000.0 24.48 37.7992 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N14 positive control 634520.0 431000.0 29.35 486320.0 337000.0 25.1 38.4991 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N15 positive control 629880.0 426000.0 29.03 488160.0 339000.0 25.23 38.3723 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N16 positive control 629440.0 425000.0 29.0 480080.0 331000.0 24.63 37.9258 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N17 positive control 625520.0 422000.0 28.74 479160.0 330000.0 24.56 37.6884 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N18 positive control 619760.0 416000.0 28.34 466880.0 318000.0 23.65 36.7645 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N19 positive control 611120.0 407000.0 27.76 470480.0 321000.0 23.92 36.5374 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N20 positive control 624080.0 420000.0 28.64 470200.0 321000.0 23.9 37.1475 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N21 positive control 617760.0 414000.0 28.21 469960.0 321000.0 23.88 36.8302 0.9966 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N22 positive control 608680.0 405000.0 27.59 465800.0 317000.0 23.57 36.1735 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N23 positive control 612680.0 409000.0 27.86 453760.0 305000.0 22.67 35.7327 0.9948 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos N24 positive control 606080.0 402000.0 27.41 460080.0 311000.0 23.14 35.7471 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O01 positive control 622840.0 419000.0 28.55 488080.0 339000.0 25.23 38.0287 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O02 positive control 619920.0 416000.0 28.36 484320.0 335000.0 24.95 37.69 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O03 positive control 621880.0 418000.0 28.49 482480.0 333000.0 24.81 37.6877 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O04 positive control 626200.0 422000.0 28.78 469280.0 320000.0 23.83 37.2012 0.9956 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O05 positive control 624520.0 421000.0 28.67 482960.0 334000.0 24.85 37.8402 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O06 positive control 629480.0 425000.0 29.01 474600.0 325000.0 24.22 37.6393 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O07 positive control 624640.0 421000.0 28.68 479400.0 330000.0 24.58 37.6586 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O08 positive control 620440.0 416000.0 28.39 467600.0 318000.0 23.7 36.8351 0.996 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O09 positive control 626240.0 422000.0 28.79 482360.0 333000.0 24.8 37.8915 0.9972 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O10 positive control 620880.0 417000.0 28.42 476640.0 327000.0 24.37 37.3321 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O11 positive control 623560.0 420000.0 28.6 477240.0 328000.0 24.42 37.4929 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O12 positive control 618360.0 414000.0 28.25 478040.0 329000.0 24.48 37.2843 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O13 positive control 622440.0 418000.0 28.53 478320.0 329000.0 24.5 37.4957 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O14 positive control 620520.0 417000.0 28.4 468360.0 319000.0 23.76 36.879 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O15 positive control 615560.0 412000.0 28.06 467480.0 318000.0 23.69 36.5936 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O16 positive control 625920.0 422000.0 28.76 476000.0 327000.0 24.33 37.5414 0.9965 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O17 positive control 625440.0 421000.0 28.73 479520.0 330000.0 24.59 37.7035 0.997 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O18 positive control 629960.0 426000.0 29.04 475920.0 327000.0 24.32 37.732 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O19 positive control 612400.0 408000.0 27.84 470200.0 321000.0 23.9 36.5844 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O20 positive control 614120.0 410000.0 27.96 463920.0 315000.0 23.43 36.3368 0.9961 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O21 positive control 614040.0 410000.0 27.95 462480.0 313000.0 23.32 36.2572 0.9959 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O22 positive control 607600.0 404000.0 27.52 460120.0 311000.0 23.15 35.8225 0.9963 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O23 positive control 608240.0 404000.0 27.56 468360.0 319000.0 23.76 36.287 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos O24 positive control 603720.0 400000.0 27.25 465840.0 317000.0 23.57 35.9365 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P01 positive control 623640.0 420000.0 28.61 488000.0 339000.0 25.22 38.063 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P02 positive control 627800.0 424000.0 28.89 478880.0 330000.0 24.54 37.7836 0.9967 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P03 positive control 629920.0 426000.0 29.04 483760.0 335000.0 24.9 38.1426 0.9971 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P04 positive control 622440.0 418000.0 28.53 483360.0 334000.0 24.87 37.761 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P05 positive control 619600.0 416000.0 28.33 478960.0 330000.0 24.55 37.3925 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P06 positive control 617760.0 414000.0 28.21 482800.0 334000.0 24.83 37.5059 0.998 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P07 positive control 620760.0 417000.0 28.41 481040.0 332000.0 24.7 37.5579 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P08 positive control 625920.0 422000.0 28.76 482800.0 334000.0 24.83 37.8993 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P09 positive control 627240.0 423000.0 28.85 489080.0 340000.0 25.3 38.2934 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P10 positive control 624800.0 421000.0 28.69 482200.0 333000.0 24.79 37.8137 0.9974 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P11 positive control 623680.0 420000.0 28.61 485360.0 336000.0 25.02 37.926 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P12 positive control 617440.0 413000.0 28.19 483560.0 334000.0 24.89 37.5305 0.9981 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P13 positive control 624120.0 420000.0 28.64 487360.0 338000.0 25.17 38.0525 0.9979 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P14 positive control 626560.0 423000.0 28.81 421760.0 273000.0 20.29 34.7177 0.9853 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P15 positive control 625040.0 421000.0 28.7 485480.0 336000.0 25.03 37.9979 0.9977 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P16 positive control 619080.0 415000.0 28.3 480360.0 331000.0 24.65 37.4411 0.9976 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P17 positive control 617120.0 413000.0 28.16 479920.0 331000.0 24.62 37.3235 0.9978 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P18 positive control 616440.0 412000.0 28.12 476560.0 327000.0 24.37 37.1139 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P19 positive control 611560.0 408000.0 27.79 471240.0 322000.0 23.97 36.5986 0.9973 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P20 positive control 612200.0 408000.0 27.83 468040.0 319000.0 23.73 36.4611 0.9969 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P21 positive control 606440.0 402000.0 27.44 462920.0 314000.0 23.35 35.9139 0.9968 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P22 positive control 607000.0 403000.0 27.47 469800.0 321000.0 23.87 36.303 0.9975 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P23 positive control 595240.0 391000.0 26.67 467680.0 319000.0 23.71 35.6245 0.9983 1132.0002 KinaseGlo(1132.0002) FAKInhibition 1132.0002.Pos P24 positive control 599520.0 396000.0 26.96 468640.0 319000.0 23.78 35.8814 0.998