ASSAY_ID ASSAY PROJECT PLATE WELL WELL_TYPE RAW_VALUE_A BSUB_VALUE_A Z_SCORE_A RAW_VALUE_B BSUB_VALUE_B Z_SCORE_B COMPOSITE_Z REPRODUCIBILITY CHEMBANK_ID VIRTUAL_ID SMILES 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A01 compound treatment 480.0 -966.0 -0.34 360.0 -291.0 -0.22 -0.4002 -0.9784 1487428 ChemDiv3_000705 CCOC(=O)C1=C(CC)NC2=C(C1c3ccc(Cl)cc3)C(=O)CCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A02 compound treatment 200.0 -1250.0 -0.44 600.0 -50.7 -0.04 -0.3401 -0.7664 1295860 ChemDiv3_000706 Ic1ccc(NC(=O)COc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A03 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1077646 ChemDiv3_000707 Clc1ccc2Sc3ccccc3N(CCC#N)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A04 compound treatment 960.0 -486.0 -0.17 200.0 -451.0 -0.35 -0.3666 -0.9483 3117740 ChemDiv3_000708 FC(F)(F)Oc1ccc(cc1)N2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A05 compound treatment 280.0 -1170.0 -0.41 440.0 -211.0 -0.16 -0.4069 -0.916 3020717 ChemDiv3_000709 NC(=S)N1C(CCN1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A06 compound treatment 1600.0 154.0 0.05 320.0 -331.0 -0.25 -0.1409 -0.5428 1443291 ChemDiv3_000710 OCCc1ccc(s1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A07 compound treatment 240.0 -1210.0 -0.43 360.0 -291.0 -0.22 -0.4604 -0.9539 3117741 ChemDiv3_000711 CCN(N(CC)S(=O)(=O)c1ccc(C)cc1)C2=NS(=O)(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A08 compound treatment 1760.0 314.0 0.11 3360.0 2710.0 2.08 1.5495 0.7439 3020718 ChemDiv3_000712 COc1ccccc1/N=C/c2ccsc2S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A09 compound treatment 400.0 -1050.0 -0.37 280.0 -371.0 -0.28 -0.4637 -0.9914 1233664 ChemDiv3_000713 O=C(CCN1C(=O)c2ccccc2C1=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A10 compound treatment 2600.0 1150.0 0.41 360.0 -291.0 -0.22 0.1316 0.2823 1914325 ChemDiv3_000714 NC(=N)SCCS(=O)(=O)c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A11 compound treatment 2480.0 1030.0 0.37 240.0 -411.0 -0.32 0.0364 0.0752 1506625 ChemDiv3_000715 COC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A12 compound treatment 320.0 -1130.0 -0.4 400.0 -251.0 -0.19 -0.4186 -0.9439 1069326 ChemDiv3_000716 FC(F)(F)c1ccccc1NC(=O)c2ccccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A13 compound treatment 280.0 -1170.0 -0.41 200.0 -451.0 -0.35 -0.5372 -0.996 1446136 ChemDiv3_000717 COc1ccc(NC(=O)C2CSC(C)(C)N2C=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A14 compound treatment 5280.0 3830.0 1.36 480.0 -171.0 -0.13 0.869 0.636 3020719 ChemDiv3_000718 COc1ccc(/C=N/c2nc3ccccc3n2Cc4ccc(Cl)cc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A15 compound treatment 5840.0 4390.0 1.56 280.0 -371.0 -0.28 0.9009 0.5686 1718021 ChemDiv3_000719 COC(=O)c1cc(Cl)c(NC(=S)NC(=O)C(C)(C)C)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A16 compound treatment 320.0 -1130.0 -0.4 400.0 -251.0 -0.19 -0.4186 -0.9439 3117742 ChemDiv3_000720 CN(C)c1ccc(/C=N/c2nc3ccccc3n2Cc4ccc(C)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A17 compound treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 1339224 ChemDiv3_000721 COC(=O)C(Cc1c[nH]c2ccccc12)NS(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A18 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1054488 ChemDiv3_000722 Cc1cc(C)n(n1)S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A19 compound treatment 240.0 -1210.0 -0.43 360.0 -291.0 -0.22 -0.4604 -0.9539 1779183 ChemDiv3_000723 CC(C)COC(=O)CNc1n[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A20 compound treatment 1560.0 114.0 0.04 3040.0 2390.0 1.83 1.3256 0.7225 3117743 ChemDiv3_000724 CCOc1cc(/C=C/2\Sc3ccccc3C2=O)cc(I)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A21 compound treatment 200.0 -1250.0 -0.44 400.0 -251.0 -0.19 -0.4487 -0.9306 1646638 ChemDiv3_000725 COC(=O)C(Cc1ccc(O)cc1)NC(=O)c2ccccc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A22 compound treatment 680.0 -766.0 -0.27 240.0 -411.0 -0.32 -0.4151 -0.9973 1624682 ChemDiv3_000726 COC(=O)c1ccccc1NC(=O)CCCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A23 mock treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 A24 mock treatment 520.0 -926.0 -0.33 240.0 -411.0 -0.32 -0.4553 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B01 compound treatment 280.0 -1170.0 -0.41 760.0 109.0 0.08 -0.2332 -0.5524 1725673 ChemDiv3_000727 CCc1ccc(cc1)C2C(=C(C)NC3=C2C(=O)CCC3)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B02 compound treatment 400.0 -1050.0 -0.37 200.0 -451.0 -0.35 -0.5071 -0.9994 3117744 ChemDiv3_000728 CN1C(=O)/C(=C\2/SC(=S)N(NC(=O)C)C2=O)/c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B03 compound treatment 4600.0 3150.0 1.12 1160.0 509.0 0.39 1.0676 0.9008 3020720 ChemDiv3_000729 Cc1cccc(c1)C(=O)Oc2ccc(C)c(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B04 compound treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 1254173 ChemDiv3_000730 Cc1ccccc1OCCn2c(SCc3nc4ccccc4[nH]3)nc5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B05 compound treatment 320.0 -1130.0 -0.4 360.0 -291.0 -0.22 -0.4403 -0.9621 3020816 ChemDiv3_000731 C1CCC2CC(OCC2C1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B06 compound treatment 320.0 -1130.0 -0.4 200.0 -451.0 -0.35 -0.5272 -0.9974 3117745 ChemDiv3_000732 Cc1ccc(cc1)S(=O)(=O)/N=C(/NC(=S)Nc2ccccc2)\c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B07 compound treatment 5240.0 3790.0 1.35 440.0 -211.0 -0.16 0.8373 0.6177 3020817 ChemDiv3_000733 CCN(CC)C(=O)CSc1nnc(o1)c2ccccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B08 compound treatment 200.0 -1250.0 -0.44 440.0 -211.0 -0.16 -0.427 -0.907 3117746 ChemDiv3_000734 CC(=O)NC(=O)c/1cc2c(ccc3ccccc32)o\c1=N/c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B09 compound treatment 760.0 -686.0 -0.24 280.0 -371.0 -0.28 -0.3734 -0.997 1423328 ChemDiv3_000735 OC(CNCc1ccccc1)Cn2c3ccc(Cl)cc3c4cc(Cl)ccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B10 compound treatment 280.0 -1170.0 -0.41 160.0 -491.0 -0.38 -0.5589 -0.9989 1240251 ChemDiv3_000736 Cc1c(Cl)cccc1NC(=O)c2cccnc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B11 compound treatment 680.0 -766.0 -0.27 240.0 -411.0 -0.32 -0.4151 -0.9973 3020818 ChemDiv3_000737 CCOc1ccc-2c(c1)C(=O)c3cc(OCC)ccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B12 compound treatment 160.0 -1290.0 -0.46 200.0 -451.0 -0.35 -0.5673 -0.9907 1727003 ChemDiv3_000738 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc3sc(SC)nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B13 compound treatment 400.0 -1050.0 -0.37 280.0 -371.0 -0.28 -0.4637 -0.9914 1740255 ChemDiv3_000739 Cc1ccc(cc1)S(=O)(=O)N2CCN(C2c3ccccc3)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B14 compound treatment 800.0 -646.0 -0.23 200.0 -451.0 -0.35 -0.4068 -0.98 3020819 ChemDiv3_000740 CC1(C)CC(=S)C=C(C1)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B15 compound treatment 3120.0 1670.0 0.59 800.0 149.0 0.11 0.5009 0.8283 1741101 ChemDiv3_000741 Clc1cc2sc(=O)oc2cc1OC(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B16 compound treatment 280.0 -1170.0 -0.41 360.0 -291.0 -0.22 -0.4503 -0.958 3117538 ChemDiv3_000742 COc1ccc(OC)c(/N=C/c2cc(I)cc(C)c2O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B17 compound treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 3117539 ChemDiv3_000743 CCOc1ccc(cc1)N2C(=O)S/C(=C/3\C(=O)Nc4ccccc34)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B18 compound treatment 400.0 -1050.0 -0.37 280.0 -371.0 -0.28 -0.4637 -0.9914 1455599 ChemDiv3_000744 CC(C)c1cc(C(C)C)c(c(c1)C(C)C)S(=O)(=O)Nc2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B19 compound treatment 1640.0 194.0 0.07 240.0 -411.0 -0.32 -0.1743 -0.5403 1507311 ChemDiv3_000745 CC(C)CN(CC(C)C)C(=O)c1cc2ccccc2oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B20 compound treatment 280.0 -1170.0 -0.41 6480.0 5830.0 4.48 2.872 0.639 3117540 ChemDiv3_000746 CCN1C(=O)/C(=C/Nc2ccccc2)/OC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B21 compound treatment 600.0 -846.0 -0.3 360.0 -291.0 -0.22 -0.3701 -0.9893 1429235 ChemDiv3_000747 CCOc1ccc(NC(=O)CCOc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B22 compound treatment 1440.0 -6.25 0.0 480.0 -171.0 -0.13 -0.0942 -0.719 1159158 ChemDiv3_000748 O=C1CC(CC(=C1)NCc2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B23 mock treatment 240.0 -1210.0 -0.43 360.0 -291.0 -0.22 -0.4604 -0.9539 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 B24 mock treatment 280.0 -1170.0 -0.41 280.0 -371.0 -0.28 -0.4938 -0.9833 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C01 compound treatment 440.0 -1010.0 -0.36 320.0 -331.0 -0.25 -0.4319 -0.9861 1611722 ChemDiv3_000749 CCOC(=O)C1=C(CC)NC2=C(C1c3ccccc3OCC)C(=O)CCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C02 compound treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 1332565 ChemDiv3_000750 CCOC(=O)c1ccc(NC(=O)c2ccc(C)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C03 compound treatment 3040.0 1590.0 0.57 280.0 -371.0 -0.28 0.1986 0.3137 1451908 ChemDiv3_000751 CCOC(=O)Nc1ccc2Sc3ccccc3N(C(=O)CCN(C)C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C04 compound treatment 1280.0 -166.0 -0.06 240.0 -411.0 -0.32 -0.2646 -0.8251 2112223 ChemDiv3_000752 O=c1oc2ccccc2cc1c3cn4c(n3)sc5ccccc54 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C05 compound treatment 200.0 -1250.0 -0.44 280.0 -371.0 -0.28 -0.5138 -0.9773 1471012 ChemDiv3_000753 S=C(Nc1ccccc1)N2CCCN2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C06 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1915139 ChemDiv3_000754 NC(C(=O)O)c1ccc(CCCC(=O)O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C07 compound treatment 360.0 -1090.0 -0.39 280.0 -371.0 -0.28 -0.4737 -0.9889 1351042 ChemDiv3_000755 O=C(Nc1ccccc1)Nc2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C08 compound treatment 480.0 -966.0 -0.34 320.0 -331.0 -0.25 -0.4219 -0.9891 3020820 ChemDiv3_000756 CN(/C=C\1/C=C(C)SC1=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C09 compound treatment 720.0 -726.0 -0.26 280.0 -371.0 -0.28 -0.3834 -0.9988 3117541 ChemDiv3_000757 Clc1ccc(C(=O)OCCCN2C(=O)c3ccccc3C2=O)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C10 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1673647 ChemDiv3_000758 O=C1CC(OC21CCCCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C11 compound treatment 320.0 -1130.0 -0.4 160.0 -491.0 -0.38 -0.5489 -0.9996 1920609 ChemDiv3_000759 FC(F)(F)c1ccccc1NC(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C12 compound treatment 240.0 -1210.0 -0.43 120.0 -531.0 -0.41 -0.5907 -0.9997 1187258 ChemDiv3_000760 O=C(N(CC#N)CC#N)c1ccc(cc1)C(=O)N(CC#N)CC#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C13 compound treatment 200.0 -1250.0 -0.44 240.0 -411.0 -0.32 -0.5355 -0.9863 1351252 ChemDiv3_000761 CC(C)C(=O)Oc1ccc2c(c1)oc(=O)c3ccccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C14 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 3117542 ChemDiv3_000762 Clc1ccc(Cn2c(/N=C/c3ccc4OCOc4c3)nc5ccccc25)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C15 compound treatment 360.0 -1090.0 -0.39 280.0 -371.0 -0.28 -0.4737 -0.9889 1648199 ChemDiv3_000763 Nc1c(C#N)c2nc3ccccc3nc2n1c4ccc(O)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C16 compound treatment 3760.0 2310.0 0.82 280.0 -371.0 -0.28 0.3792 0.4365 3117543 ChemDiv3_000764 Cc1ccc(Cn2c(/N=C/c3ccc(Br)cc3)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C17 compound treatment 360.0 -1090.0 -0.39 280.0 -371.0 -0.28 -0.4737 -0.9889 3020844 ChemDiv3_000765 CN(Cc1ccccc1)C(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C18 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1586578 ChemDiv3_000766 Brc1ccc(cc1)C(=O)COC(=O)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C19 compound treatment 2920.0 1470.0 0.52 400.0 -251.0 -0.19 0.2336 0.4193 1919025 ChemDiv3_000767 FC(F)(F)c1cccc(NC(=O)COc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C20 compound treatment 4360.0 2910.0 1.03 240.0 -411.0 -0.32 0.508 0.47 3020845 ChemDiv3_000768 NNC(=O)c1ccc(/C=N\O)nc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C21 compound treatment 2840.0 1390.0 0.49 240.0 -411.0 -0.32 0.1267 0.216 3020846 ChemDiv3_000769 Brc1ccc(NC(=O)/C=C/c2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C22 compound treatment 2720.0 1270.0 0.45 560.0 -90.7 -0.07 0.2703 0.5912 1510082 ChemDiv3_000770 OC(=O)CCC(=O)NCc1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C23 mock treatment 360.0 -1090.0 -0.39 800.0 149.0 0.11 -0.1914 -0.4761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 C24 mock treatment 200.0 -1250.0 -0.44 240.0 -411.0 -0.32 -0.5355 -0.9863 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D01 compound treatment 2960.0 1510.0 0.54 320.0 -331.0 -0.25 0.2002 0.3371 1123230 ChemDiv3_000771 Oc1ccccc1N2C(=O)C3CC=CCC3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D02 compound treatment 1720.0 274.0 0.1 280.0 -371.0 -0.28 -0.1326 -0.4408 1485584 ChemDiv3_000772 CCN(CC)c1ccc(NC(=O)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D03 compound treatment 360.0 -1090.0 -0.39 400.0 -251.0 -0.19 -0.4086 -0.9485 3020847 ChemDiv3_000773 O=C(NN1C(=O)CSC1=S)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D04 compound treatment 320.0 -1130.0 -0.4 200.0 -451.0 -0.35 -0.5272 -0.9974 3117544 ChemDiv3_000774 C(CSc1nc2ccccc2[nH]1)CN3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D05 compound treatment 1040.0 -406.0 -0.14 800.0 149.0 0.11 -0.0208 -0.1132 1778456 ChemDiv3_000775 OC(=O)CC(Sc1nc2sc3CCCCc3c2c(=O)[nH]1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D06 compound treatment 320.0 -1130.0 -0.4 320.0 -331.0 -0.25 -0.462 -0.976 3020848 ChemDiv3_000776 FC(F)(F)c1cccc(NC(=O)c2ccc3ccccc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D07 compound treatment 320.0 -1130.0 -0.4 280.0 -371.0 -0.28 -0.4837 -0.9862 3020849 ChemDiv3_000777 Cc1sc(Nc2ccccc2F)nc1c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D08 compound treatment 160.0 -1290.0 -0.46 320.0 -331.0 -0.25 -0.5022 -0.9617 1364991 ChemDiv3_000778 Brc1cccc(c1)c2nnc(o2)c3cc4ccccc4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D09 compound treatment 200.0 -1250.0 -0.44 240.0 -411.0 -0.32 -0.5355 -0.9863 3117545 ChemDiv3_000779 CCOC(=O)c1c(/N=c/2\oc3ccc4ccccc4c3cc2C(=O)N)sc5CCCCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D10 compound treatment 200.0 -1250.0 -0.44 200.0 -451.0 -0.35 -0.5573 -0.9926 1665286 ChemDiv3_000780 CN1CCN(CC1)NC(=O)c2ccc(cc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D11 compound treatment 200.0 -1250.0 -0.44 280.0 -371.0 -0.28 -0.5138 -0.9773 1652224 ChemDiv3_000781 COC(=O)COc1ccc-2c(c1)C(=NO)c3cc(OCC(=O)OC)ccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D12 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1235358 ChemDiv3_000782 CCC1Nc2ccccc2-c3nnc(SC)nc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D13 compound treatment 200.0 -1250.0 -0.44 240.0 -411.0 -0.32 -0.5355 -0.9863 1443634 ChemDiv3_000783 OC(=O)C1C2CC=CC2c3cc(Cl)cc4C5C=CCC5CN1c43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D14 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 3020850 ChemDiv3_000784 Fc1cccc(c1)C2=N/C(=C\c3cccc4ccccc34)/C(=O)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D15 compound treatment 160.0 -1290.0 -0.46 240.0 -411.0 -0.32 -0.5456 -0.9837 1569541 ChemDiv3_000785 CCOC(=O)c1cnn(c1N(C(=O)c2ccccc2F)C(=O)c3ccccc3F)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D16 compound treatment 480.0 -966.0 -0.34 320.0 -331.0 -0.25 -0.4219 -0.9891 3020851 ChemDiv3_000786 CC(=O)Nc1cccc(/N=C/c2cc(I)cc(C)c2O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D17 compound treatment 320.0 -1130.0 -0.4 160.0 -491.0 -0.38 -0.5489 -0.9996 1355069 ChemDiv3_000787 CS(=O)(=O)Nc1ccc(Cl)cc1C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D18 compound treatment 160.0 -1290.0 -0.46 200.0 -451.0 -0.35 -0.5673 -0.9907 1626307 ChemDiv3_000788 CC(C)c1cc(C(C)C)c(c(c1)C(C)C)S(=O)(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D19 compound treatment 400.0 -1050.0 -0.37 480.0 -171.0 -0.13 -0.3551 -0.9022 3117546 ChemDiv3_000789 Cc1cc(C)c(C(=O)NCC=C)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D20 compound treatment 2120.0 674.0 0.24 200.0 -451.0 -0.35 -0.0756 -0.1799 3117547 ChemDiv3_000790 CCN1/C(=C\2/C(=NN(C2=O)c3ccccc3)C)/C=Cc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D21 compound treatment 3440.0 1990.0 0.71 200.0 -451.0 -0.35 0.2555 0.3245 1388884 ChemDiv3_000791 O=C(CCOc1ccccc1)NCc2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D22 compound treatment 6680.0 5230.0 1.86 280.0 -371.0 -0.28 1.1116 0.5918 3117548 ChemDiv3_000792 COc1ccccc1/C=C/2\SC(=O)N(CCC(=O)N3c4ccccc4Sc5ccccc35)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D23 mock treatment 2440.0 994.0 0.35 200.0 -451.0 -0.35 0.0046 0.0094 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 D24 mock treatment 320.0 -1130.0 -0.4 160.0 -491.0 -0.38 -0.5489 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E01 compound treatment 1160.0 -286.0 -0.1 3600.0 2950.0 2.26 1.5293 0.6747 1583492 ChemDiv3_000793 COC(=O)C1=C(C)NC2=C(C1c3ccc(cc3)N(C)C)C(=O)CC(C2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E02 compound treatment 280.0 -1170.0 -0.41 2280.0 1630.0 1.25 0.592 0.4493 1432876 ChemDiv3_000794 CCc1ccc(OCC(=O)Nc2ccc(OC)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E03 compound treatment 1000.0 -446.0 -0.16 440.0 -211.0 -0.16 -0.2263 -0.9999 3117549 ChemDiv3_000795 COc1cccc(/C=C/C(=O)C2C(=O)c3ccccc3C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E04 compound treatment 7240.0 5790.0 2.06 320.0 -331.0 -0.25 1.2738 0.6151 1606983 ChemDiv3_000796 Oc1cccc(NC(=O)c2c(O)c3ccccc3n(CC=C)c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E05 compound treatment 320.0 -1130.0 -0.4 1960.0 1310.0 1.01 0.4283 0.3959 1715553 ChemDiv3_000797 Cc1[nH]c2ccc(CN3C(=O)c4ccccc4C3=O)cc2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E06 compound treatment 320.0 -1130.0 -0.4 680.0 29.3 0.02 -0.2666 -0.6662 3020853 ChemDiv3_000798 COC(=O)c1cc(N)c(Cl)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E07 compound treatment 240.0 -1210.0 -0.43 4840.0 4190.0 3.22 1.9716 0.6077 1915335 ChemDiv3_000799 FC(F)(F)c1cccc(NC(=O)Nc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E08 compound treatment 360.0 -1090.0 -0.39 320.0 -331.0 -0.25 -0.452 -0.9795 1289585 ChemDiv3_000800 CC1(OC(=O)C2C1C3CCCCC3=C4CCCCC24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E09 compound treatment 4680.0 3230.0 1.15 3200.0 2550.0 1.96 2.1951 0.9676 1304126 ChemDiv3_000801 O=C(N1CC(=O)Nc2ccccc12)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E10 compound treatment 480.0 -966.0 -0.34 800.0 149.0 0.11 -0.1613 -0.4463 1265761 ChemDiv3_000802 COc1cc(nc(OC)n1)N2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E11 compound treatment 240.0 -1210.0 -0.43 320.0 -331.0 -0.25 -0.4821 -0.9689 1735414 ChemDiv3_000803 COC(=O)c1ccc(OC(=O)CCN2C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E12 compound treatment 2200.0 754.0 0.27 760.0 109.0 0.08 0.2484 0.8864 3020873 ChemDiv3_000804 CN(c1ccccc1)S(=O)(=O)c2c(C)cc(C)cc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E13 compound treatment 240.0 -1210.0 -0.43 560.0 -90.7 -0.07 -0.3518 -0.8115 1517748 ChemDiv3_000805 CN(C1CCCCC1)C(=O)COc2ccc(Cl)c(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E14 compound treatment 2040.0 594.0 0.21 880.0 229.0 0.18 0.2734 0.996 1467248 ChemDiv3_000806 Cc1nc2n(Cc3ccccc3)c4ccccc4n2c1C(=S)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E15 compound treatment 360.0 -1090.0 -0.39 1080.0 429.0 0.33 -0.0394 -0.0777 1918958 ChemDiv3_000807 Clc1cccc(CC2SC(=N)NC2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E16 compound treatment 1480.0 33.8 0.01 520.0 -131.0 -0.1 -0.0625 -0.6183 3020874 ChemDiv3_000808 CC(/N=C/c1nc2ccccc2n1C)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E17 compound treatment 320.0 -1130.0 -0.4 520.0 -131.0 -0.1 -0.3534 -0.858 3117550 ChemDiv3_000809 Cc1ccc(cc1)C(=O)Nc2cccc(c2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E18 compound treatment 320.0 -1130.0 -0.4 800.0 149.0 0.11 -0.2014 -0.4846 3117551 ChemDiv3_000810 COc1ccc(O)c(/C=N/CC(C)\N=C\c2cc(OC)ccc2O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E19 compound treatment 320.0 -1130.0 -0.4 2240.0 1590.0 1.22 0.5803 0.452 1413824 ChemDiv3_000811 COC(=O)c1ccccc1NC(=O)COc2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E20 compound treatment 1400.0 -46.3 -0.02 6120.0 5470.0 4.2 2.9575 0.7043 1629872 ChemDiv3_000812 COc1ccccc1C(=O)Nc2ccc3oc(nc3c2)c4ccc5ccccc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E21 compound treatment 2480.0 1030.0 0.37 720.0 69.3 0.05 0.2969 0.8013 1625558 ChemDiv3_000813 COC(=O)c1cccc(NC(=O)c2ccccc2C(=O)O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E22 compound treatment 920.0 -526.0 -0.19 440.0 -211.0 -0.16 -0.2464 -0.9974 1326899 ChemDiv3_000814 COc1ccccc1N2CCN(CC2)C(=O)CCCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E23 mock treatment 1120.0 -326.0 -0.12 1960.0 1310.0 1.01 0.6289 0.6216 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 E24 mock treatment 1640.0 194.0 0.07 1200.0 549.0 0.42 0.3468 0.8116 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F01 compound treatment 1040.0 -406.0 -0.14 1840.0 1190.0 0.91 0.5437 0.5882 1373507 ChemDiv3_000815 OC(=O)C1CC=CCC1C(=O)Nc2ccc(Cc3ccncc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F02 compound treatment 960.0 -486.0 -0.17 1600.0 949.0 0.73 0.3934 0.5252 3020875 ChemDiv3_000816 O=C(NC1CCCC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F03 compound treatment 2360.0 914.0 0.32 440.0 -211.0 -0.16 0.1148 0.317 1442394 ChemDiv3_000817 O=C(NCCc1ccccc1)c2ccccc2CN3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F04 compound treatment 1160.0 -286.0 -0.1 280.0 -371.0 -0.28 -0.273 -0.9036 3020876 ChemDiv3_000818 FC(F)(F)c1nc2ccccc2n1CCOc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F05 compound treatment 2200.0 754.0 0.27 1080.0 429.0 0.33 0.4221 0.9946 3117552 ChemDiv3_000819 O=C(N/C(=C/c1ccccc1)/S(=O)(=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F06 compound treatment 280.0 -1170.0 -0.41 2440.0 1790.0 1.37 0.6788 0.4732 3020877 ChemDiv3_000820 CCOc1ccc(cc1Br)C(=O)Nc2cccc(NC(=O)c3ccccc3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F07 compound treatment 640.0 -806.0 -0.29 1080.0 429.0 0.33 0.0308 0.0706 3117553 ChemDiv3_000821 O=C(Nc1ccccc1)c2cnc[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F08 compound treatment 2360.0 914.0 0.32 960.0 309.0 0.24 0.3971 0.9883 1673072 ChemDiv3_000822 OC(C(=O)Nc1cc(Cl)ccc1Cl)(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F09 compound treatment 1960.0 514.0 0.18 1240.0 589.0 0.45 0.4488 0.9201 3020878 ChemDiv3_000823 CCN(CC)c1ccc2cc(C(=O)N)/c(=N/c3cccc(C)c3)/oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F10 compound treatment 320.0 -1130.0 -0.4 2160.0 1510.0 1.16 0.5368 0.438 3117554 ChemDiv3_000824 Fc1ccc(NC(=O)c2cnccn2)c(F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F11 compound treatment 440.0 -1010.0 -0.36 1520.0 869.0 0.67 0.2195 0.29 1470949 ChemDiv3_000825 COc1ccc(cc1)c2ccc(OC)cc2C(=O)NN 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F12 compound treatment 2880.0 1430.0 0.51 760.0 109.0 0.08 0.419 0.8128 1687536 ChemDiv3_000826 CCN(CC)S(=O)(=O)c1ccc(Cl)c(c1)C(=O)Oc2ccc(C)cc2n3nc4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F13 compound treatment 400.0 -1050.0 -0.37 2680.0 2030.0 1.56 0.8392 0.524 1365314 ChemDiv3_000827 Clc1ccc2NC(C3CC=CC3c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F14 compound treatment 320.0 -1130.0 -0.4 360.0 -291.0 -0.22 -0.4403 -0.9621 1517186 ChemDiv3_000828 Cc1cccc(c1)C(=O)Nc2ccc(NC(=O)c3ccco3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F15 compound treatment 240.0 -1210.0 -0.43 1760.0 1110.0 0.85 0.2996 0.3144 1513840 ChemDiv3_000829 COC(=O)C1=C(C)N(C(=C(C1c2ccccc2)C(=O)OC)C)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F16 compound treatment 1040.0 -406.0 -0.14 1560.0 909.0 0.7 0.3917 0.5495 3117555 ChemDiv3_000830 COc1cccc(/C=C\2/C(=O)NN(C2=O)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F17 compound treatment 800.0 -646.0 -0.23 760.0 109.0 0.08 -0.1028 -0.4209 3020879 ChemDiv3_000831 CS(=O)(=O)NCCc1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F18 compound treatment 3040.0 1590.0 0.57 1280.0 629.0 0.48 0.7414 0.9969 1468720 ChemDiv3_000832 OC(=O)c1ccccc1C(=O)NC=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F19 compound treatment 1560.0 114.0 0.04 7080.0 6430.0 4.94 3.5188 0.7129 3117556 ChemDiv3_000833 CC(C)c1ccc(/C=C/C(=O)NCC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F20 compound treatment 280.0 -1170.0 -0.41 840.0 189.0 0.15 -0.1898 -0.4327 3117557 ChemDiv3_000834 CC(C)CNC=C1C(=O)CC(C)(C)CC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F21 compound treatment 280.0 -1170.0 -0.41 1040.0 389.0 0.3 -0.0812 -0.1591 1393505 ChemDiv3_000835 Cc1cc(C)cc(NC(=O)c2cc3ccccc3o2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F22 compound treatment 240.0 -1210.0 -0.43 2440.0 1790.0 1.37 0.6688 0.4648 3117558 ChemDiv3_000836 CN1CCN(CC1)C(=O)CCN2C(=O)/C(=C/c3ccc(Cl)cc3)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F23 mock treatment 280.0 -1170.0 -0.41 2880.0 2230.0 1.71 0.9177 0.5212 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 F24 mock treatment 320.0 -1130.0 -0.4 4200.0 3550.0 2.72 1.6443 0.597 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G01 compound treatment 1280.0 -166.0 -0.06 3120.0 2470.0 1.9 1.2988 0.6848 1690924 ChemDiv3_000837 COC(=O)C1=C(C)NC2=C(C1c3ccccc3)C(=O)CCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G02 compound treatment 360.0 -1090.0 -0.39 1920.0 1270.0 0.97 0.4166 0.3975 1254482 ChemDiv3_000838 Cc1ccc(OCC(=O)NCc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G03 compound treatment 640.0 -806.0 -0.29 440.0 -211.0 -0.16 -0.3166 -0.9636 1006818 ChemDiv3_000839 OC(=O)CCCC(=O)c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G04 compound treatment 1520.0 73.8 0.03 400.0 -251.0 -0.19 -0.1176 -0.6054 3117559 ChemDiv3_000840 CC(C)(C)c1ccc(cc1)C(=O)N2CCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G05 compound treatment 1440.0 -6.25 0.0 720.0 69.3 0.05 0.0361 0.6771 1344674 ChemDiv3_000841 Clc1ccccc1C(=O)c2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G06 compound treatment 720.0 -726.0 -0.26 1720.0 1070.0 0.82 0.3983 0.4629 1914993 ChemDiv3_000842 COC(=O)CCC(=O)c1cc(sc1C(C)(C)C)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G07 compound treatment 2080.0 634.0 0.22 2800.0 2150.0 1.65 1.3258 0.7961 1342176 ChemDiv3_000843 CC1CCN(Cn2c(=S)oc3ccccc23)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G08 compound treatment 4560.0 3110.0 1.1 560.0 -90.7 -0.07 0.7318 0.6612 1917056 ChemDiv3_000844 FC(F)(F)COc1nc(nc(n1)N2CCCCC2)N(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G09 compound treatment 600.0 -846.0 -0.3 560.0 -90.7 -0.07 -0.2615 -0.8485 1584064 ChemDiv3_000845 Cc1ccccc1OCC(=O)NC(c2ccccc2)c3c(O)ccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G10 compound treatment 1640.0 194.0 0.07 1000.0 349.0 0.27 0.2382 0.8605 1318907 ChemDiv3_000846 CCCc1nc(N)c(C#N)c(c1CC)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G11 compound treatment 3400.0 1950.0 0.69 960.0 309.0 0.24 0.658 0.8981 1607665 ChemDiv3_000847 O=C(NCCc1ccccc1)c2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G12 compound treatment 1600.0 154.0 0.05 1240.0 589.0 0.45 0.3585 0.7867 1316192 ChemDiv3_000848 CCN(Cc1ccccc1)S(=O)(=O)c2cc(Cl)ccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G13 compound treatment 2120.0 674.0 0.24 480.0 -171.0 -0.13 0.0764 0.2801 3117560 ChemDiv3_000849 Clc1ccc(/C=C/C(=O)Nc2nccs2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G14 compound treatment 2160.0 714.0 0.25 520.0 -131.0 -0.1 0.1081 0.3969 1342653 ChemDiv3_000850 Clc1ccc2[nH]c(nc2c1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G15 compound treatment 880.0 -566.0 -0.2 480.0 -171.0 -0.13 -0.2347 -0.9786 1360061 ChemDiv3_000851 CCOc1ccccc1C(=O)Nc2cccc(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G16 compound treatment 4600.0 3150.0 1.12 560.0 -90.7 -0.07 0.7419 0.6618 1160846 ChemDiv3_000852 CC1CN(CC(C)O1)S(=O)(=O)c2ccc(NC(=O)C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G17 compound treatment 2240.0 794.0 0.28 920.0 269.0 0.21 0.3453 0.9885 3020907 ChemDiv3_000853 Cc1ccc(NC(=O)c2ccc(F)cc2)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G18 compound treatment 680.0 -766.0 -0.27 480.0 -171.0 -0.13 -0.2849 -0.944 1569529 ChemDiv3_000854 Cc1ccc(NC(=O)c2nc[nH]c2C(=O)N3CCCCC3)c(c1)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G19 compound treatment 400.0 -1050.0 -0.37 640.0 -10.7 -0.01 -0.2682 -0.7225 1657157 ChemDiv3_000855 CC(C)(C)C(=O)NC(c1ccccc1)c2c(O)ccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G20 compound treatment 320.0 -1130.0 -0.4 2520.0 1870.0 1.44 0.7323 0.4916 1709867 ChemDiv3_000856 COc1cccc(c1)C(=O)Nc2ccc3oc(nc3c2)c4cccc(I)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G21 compound treatment 320.0 -1130.0 -0.4 760.0 109.0 0.08 -0.2232 -0.5466 1083894 ChemDiv3_000857 Clc1ccc(cc1)C(=O)NCCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G22 compound treatment 1880.0 434.0 0.15 2560.0 1910.0 1.47 1.1453 0.7771 3117561 ChemDiv3_000858 COc1cccc(c1)C(C(F)(F)F)P(=O)(C)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G23 mock treatment 1920.0 474.0 0.17 440.0 -211.0 -0.16 0.0045 0.0192 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 G24 mock treatment 3280.0 1830.0 0.65 480.0 -171.0 -0.13 0.3673 0.5536 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H01 compound treatment 1160.0 -286.0 -0.1 1400.0 749.0 0.58 0.335 0.5734 1366343 ChemDiv3_000859 CC(=O)N(CN1C(=O)C2CC=CCC2C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H02 compound treatment 1480.0 33.8 0.01 760.0 109.0 0.08 0.0678 0.7999 1584378 ChemDiv3_000860 CCOC(=O)Cc1csc(NC(=O)c2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H03 compound treatment 1840.0 394.0 0.14 680.0 29.3 0.02 0.1147 0.8106 3117562 ChemDiv3_000861 CC(C)c1ccc(C)cc1OCC(=O)/C=C/2\Sc3ccccc3N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H04 compound treatment 5480.0 4030.0 1.43 720.0 69.3 0.05 1.0495 0.7329 1622162 ChemDiv3_000862 Cc1ccccc1C(=O)Nc2ccc(NC(=O)c3ccc(cc3)C(C)(C)C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H05 compound treatment 5680.0 4230.0 1.5 6480.0 5830.0 4.48 4.2265 0.8953 3117563 ChemDiv3_000863 Cc1ccc(cc1)S(=O)(=O)NN2C(=O)S/C(=C/c3ccccc3)/C2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H06 compound treatment 600.0 -846.0 -0.3 440.0 -211.0 -0.16 -0.3266 -0.9579 3020908 ChemDiv3_000864 CSc1ccc(/C=C\2/SC(=O)N(CNc3ccccc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H07 compound treatment 960.0 -486.0 -0.17 1320.0 669.0 0.51 0.2414 0.4453 1912608 ChemDiv3_000865 Oc1ccc(/N=C/c2c[nH]c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H08 compound treatment 1400.0 -46.3 -0.02 520.0 -131.0 -0.1 -0.0825 -0.812 1623791 ChemDiv3_000866 Cc1ccc(NC(=O)c2ccc(cc2)c3ccccc3)nc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H09 compound treatment 1400.0 -46.3 -0.02 4160.0 3510.0 2.69 1.8935 0.7028 3117564 ChemDiv3_000867 COc1cccc2cc(c3csc(Nc4cccc(c4)C(F)(F)F)n3)c(=O)oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H10 compound treatment 1680.0 234.0 0.08 360.0 -291.0 -0.22 -0.0992 -0.4165 3020909 ChemDiv3_000868 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H11 compound treatment 1360.0 -86.3 -0.03 440.0 -211.0 -0.16 -0.136 -0.8262 1919894 ChemDiv3_000869 CCS(=O)(=O)C(=C(Nc1ccccc1)Nc2ccccc2)S(=O)(=O)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H12 compound treatment 6720.0 5270.0 1.87 600.0 -50.7 -0.04 1.2954 0.6923 1361150 ChemDiv3_000870 COC(=O)C(C(C)C)N1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H13 compound treatment 1680.0 234.0 0.08 1160.0 509.0 0.39 0.3351 0.8384 1526618 ChemDiv3_000871 Cc1c(Cl)cccc1NC(=O)c2ccc(cc2)N3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H14 compound treatment 960.0 -486.0 -0.17 960.0 309.0 0.24 0.046 0.1566 3118161 ChemDiv3_000872 O=C(Nc1ccc(cc1)c2nc3c(ccc4ccccc34)o2)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H15 compound treatment 1080.0 -366.0 -0.13 1040.0 389.0 0.3 0.1195 0.3666 1157871 ChemDiv3_000873 O=C(COc1ccc2c(cc(=O)oc2c1)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H16 compound treatment 800.0 -646.0 -0.23 400.0 -251.0 -0.19 -0.2982 -0.9962 3118162 ChemDiv3_000874 Nc1nnnn1/N=C\c2ccc(O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H17 compound treatment 1160.0 -286.0 -0.1 4520.0 3870.0 2.97 2.0287 0.6825 1288630 ChemDiv3_000875 CCOC(=O)c1ccccc1NS(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H18 compound treatment 920.0 -526.0 -0.19 640.0 -10.7 -0.01 -0.1378 -0.7374 1696480 ChemDiv3_000876 Cc1ccc(NCC(O)Cn2c3ccccc3c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H19 compound treatment 1600.0 154.0 0.05 1160.0 509.0 0.39 0.3151 0.798 1434081 ChemDiv3_000877 CC(C)c1ccc(OCC(=O)NCC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H20 compound treatment 960.0 -486.0 -0.17 560.0 -90.7 -0.07 -0.1712 -0.9203 3020910 ChemDiv3_000878 CC1(C)CC(=O)C(=CNCc2ccco2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H21 compound treatment 1840.0 394.0 0.14 3720.0 3070.0 2.36 1.765 0.7477 1350794 ChemDiv3_000879 COc1ccc(OC(=O)c2cc3ccccc3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H22 compound treatment 480.0 -966.0 -0.34 1120.0 469.0 0.36 0.0124 0.0249 3020911 ChemDiv3_000880 O=c1[nH]nc(N2CCOCC2)c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H23 mock treatment 720.0 -726.0 -0.26 600.0 -50.7 -0.04 -0.2097 -0.8047 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 H24 mock treatment 4000.0 2550.0 0.91 640.0 -10.7 -0.01 0.6348 0.7007 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I01 compound treatment 6240.0 4790.0 1.7 520.0 -131.0 -0.1 1.1315 0.6642 1682167 ChemDiv3_000881 CCOC(=O)C1=C(NC(=O)NC1c2ccc(OC)cc2)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I02 compound treatment 680.0 -766.0 -0.27 840.0 189.0 0.15 -0.0894 -0.2901 3020912 ChemDiv3_000882 C1CN(CCO1)c2ccc(C=Nn3cncn3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I03 compound treatment 1200.0 -246.0 -0.09 560.0 -90.7 -0.07 -0.111 -0.9937 1588286 ChemDiv3_000883 CCOc1ccccc1N2C(=O)C3C(C(C=CC3c4ccccc4)c5ccccc5)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I04 compound treatment 520.0 -926.0 -0.33 760.0 109.0 0.08 -0.173 -0.5101 3118163 ChemDiv3_000884 Cc1ccc(C)c(c1)S(=O)(=O)NCCCn2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I05 compound treatment 320.0 -1130.0 -0.4 1280.0 629.0 0.48 0.0591 0.0943 1319250 ChemDiv3_000885 O=C(Nc1ccc2-c3ccc(NC(=O)C4CCCCC4)cc3S(=O)(=O)c2c1)C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I06 compound treatment 320.0 -1130.0 -0.4 800.0 149.0 0.11 -0.2014 -0.4846 3020913 ChemDiv3_000886 CC1NC(=O)NC1CCCCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I07 compound treatment 360.0 -1090.0 -0.39 280.0 -371.0 -0.28 -0.4737 -0.9889 1370690 ChemDiv3_000887 CCC1CCCCN1C(=O)CN2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I08 compound treatment 1280.0 -166.0 -0.06 360.0 -291.0 -0.22 -0.1995 -0.8643 3020914 ChemDiv3_000888 CCC1(CC)Cc2ccccc2/C(=N/c3c(C)n(C)n(c4ccccc4)c3=O)/N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I09 compound treatment 240.0 -1210.0 -0.43 920.0 269.0 0.21 -0.1564 -0.329 3118164 ChemDiv3_000889 CC(C)CC(N1C(=O)c2ccccc2C1=O)C(=O)Nc3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I10 compound treatment 280.0 -1170.0 -0.41 280.0 -371.0 -0.28 -0.4938 -0.9833 3118165 ChemDiv3_000890 COc1ccc(Cl)cc1NC(=O)c2nc3nc(cc(n3n2)C(F)(F)F)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I11 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1696086 ChemDiv3_000891 CCc1ccc(OCC(=O)N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I12 compound treatment 360.0 -1090.0 -0.39 240.0 -411.0 -0.32 -0.4954 -0.995 1643226 ChemDiv3_000892 OC(=O)CP(=O)(O)c1ccc(Cl)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I13 compound treatment 960.0 -486.0 -0.17 1040.0 389.0 0.3 0.0894 0.259 3118166 ChemDiv3_000893 Clc1ccccc1/C=C/C(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I14 compound treatment 240.0 -1210.0 -0.43 3080.0 2430.0 1.87 1.0162 0.5311 3020915 ChemDiv3_000894 COc1ccccc1/C=N\c2ccc3n(Cc4ccccc4)c(C)nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I15 compound treatment 280.0 -1170.0 -0.41 520.0 -131.0 -0.1 -0.3635 -0.8538 1438926 ChemDiv3_000895 COC(=O)c1ccccc1NC(=O)c2ccccc2Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I16 compound treatment 240.0 -1210.0 -0.43 320.0 -331.0 -0.25 -0.4821 -0.9689 1126074 ChemDiv3_000896 O=S(=O)(Cc1ccccc1)Nc2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I17 compound treatment 280.0 -1170.0 -0.41 360.0 -291.0 -0.22 -0.4503 -0.958 3118167 ChemDiv3_000897 Clc1ccc(/C=C/C(=O)NCc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I18 compound treatment 280.0 -1170.0 -0.41 3720.0 3070.0 2.36 1.3737 0.5742 3118168 ChemDiv3_000898 O=C1CS/C(=N\c2ccccc2)/N1Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I19 compound treatment 280.0 -1170.0 -0.41 3000.0 2350.0 1.8 0.9828 0.5311 1496753 ChemDiv3_000899 CC(=O)n1cc(c2ccncc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I20 compound treatment 240.0 -1210.0 -0.43 320.0 -331.0 -0.25 -0.4821 -0.9689 3118169 ChemDiv3_000900 CC(=O)NC(=O)c/1cc2ccccc2o\c1=N/c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I21 compound treatment 960.0 -486.0 -0.17 240.0 -411.0 -0.32 -0.3449 -0.9597 1085397 ChemDiv3_000901 Clc1ccccc1NC(=O)COc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I22 compound treatment 320.0 -1130.0 -0.4 320.0 -331.0 -0.25 -0.462 -0.976 3020938 ChemDiv3_000902 CP(=O)(O)C(c1cccc(Cl)c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I23 mock treatment 760.0 -686.0 -0.24 320.0 -331.0 -0.25 -0.3516 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 I24 mock treatment 360.0 -1090.0 -0.39 320.0 -331.0 -0.25 -0.452 -0.9795 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J01 compound treatment 304800.0 303000.0 107.61 32720.0 32100.0 24.62 93.5034 0.847 3118170 ChemDiv3_000903 O=C1NC(=O)/C(=C\c2c3ccccc3cc4ccccc24)/C(=O)N1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J02 compound treatment 2760.0 1310.0 0.47 880.0 229.0 0.18 0.454 0.9114 1538193 ChemDiv3_000904 Cc1cccc(Nc2nc(C)cc(C)c2C#N)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J03 compound treatment 480.0 -966.0 -0.34 2160.0 1510.0 1.16 0.577 0.4775 3020939 ChemDiv3_000905 CC(C)C(=O)/C=C\1/Sc2ccccc2N1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J04 compound treatment 360.0 -1090.0 -0.39 520.0 -131.0 -0.1 -0.3434 -0.8624 1399642 ChemDiv3_000906 CC(C)(C#CC(O)(c1ccccc1)c2ccccc2)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J05 compound treatment 480.0 -966.0 -0.34 1920.0 1270.0 0.97 0.4467 0.4324 3118171 ChemDiv3_000907 Clc1ccc(/C=C\2/SC(=O)N(NC(=O)c3ccccc3Cl)C2=S)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J06 compound treatment 16000.0 14600.0 5.16 19120.0 18500.0 14.18 13.677 0.9064 1545446 ChemDiv3_000908 OC(=O)c1ccccc1n2c(=O)c3cc4c(=O)n(c5ccccc5C(=O)O)c(=O)c4cc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J07 compound treatment 480.0 -966.0 -0.34 440.0 -211.0 -0.16 -0.3567 -0.9412 1642929 ChemDiv3_000909 C(N1CCN(Cc2ccccc2)C1c3c[nH]c4ccccc34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J08 compound treatment 280.0 -1170.0 -0.41 720.0 69.3 0.05 -0.2549 -0.6111 3118172 ChemDiv3_000910 FC(F)(F)c1cccc(NC(=O)c2ccc(cc2)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J09 compound treatment 680.0 -766.0 -0.27 440.0 -211.0 -0.16 -0.3066 -0.9692 3020940 ChemDiv3_000911 Ic1cccc(/C=N/N2C(=O)C3C4C=CC(C3C2=O)C54CC5)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J10 compound treatment 360.0 -1090.0 -0.39 280.0 -371.0 -0.28 -0.4737 -0.9889 3118173 ChemDiv3_000912 Cc1cc(I)ccc1NC(=O)c2ccc(cc2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J11 compound treatment 320.0 -1130.0 -0.4 280.0 -371.0 -0.28 -0.4837 -0.9862 1477505 ChemDiv3_000913 CCCS(=O)(=O)c1c(C(=O)OC)n2ccccc2c1S(=O)(=O)CCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J12 compound treatment 440.0 -1010.0 -0.36 600.0 -50.7 -0.04 -0.2799 -0.7795 1130176 ChemDiv3_000914 Cc1cccc(NCN2C(=O)C3C4CC(C=C4)C3C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J13 compound treatment 5400.0 3950.0 1.4 720.0 69.3 0.05 1.0294 0.7334 3020941 ChemDiv3_000915 O=C/1OC(=N\C1=C/Nc2ccccn2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J14 compound treatment 400.0 -1050.0 -0.37 360.0 -291.0 -0.22 -0.4202 -0.9704 1478515 ChemDiv3_000916 CCCOc1ccc(cc1)C(=O)Nc2ccc(cc2)c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J15 compound treatment 280.0 -1170.0 -0.41 360.0 -291.0 -0.22 -0.4503 -0.958 3118174 ChemDiv3_000917 CC(C)(C)NC(=O)CCCN1C(=O)/C(=C/c2ccccc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J16 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 3020942 ChemDiv3_000918 Brc1ccc(cc1)C2=N/C(=C\Nc3ccccc3)/C(=O)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J17 compound treatment 280.0 -1170.0 -0.41 480.0 -171.0 -0.13 -0.3852 -0.8876 3118175 ChemDiv3_000919 OC(=O)CCCNc1n[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J18 compound treatment 320.0 -1130.0 -0.4 720.0 69.3 0.05 -0.2449 -0.6075 1721267 ChemDiv3_000920 O=C1N(CN2CCCCC2)C(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J19 compound treatment 280.0 -1170.0 -0.41 360.0 -291.0 -0.22 -0.4503 -0.958 1065790 ChemDiv3_000921 COc1ccc(NC(=S)NC2CCCCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J20 compound treatment 440.0 -1010.0 -0.36 280.0 -371.0 -0.28 -0.4536 -0.9937 1923178 ChemDiv3_000922 CC1(C)CC(=O)C(=CNCC2CCCO2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J21 compound treatment 1480.0 33.8 0.01 280.0 -371.0 -0.28 -0.1928 -0.6768 1623304 ChemDiv3_000923 Cc1ccc(OC(=O)c2cc3ccccc3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J22 compound treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 3118176 ChemDiv3_000924 CCOCc1c[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J23 mock treatment 720.0 -726.0 -0.26 320.0 -331.0 -0.25 -0.3617 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 J24 mock treatment 4640.0 3190.0 1.13 5000.0 4350.0 3.34 3.1622 0.8968 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K01 compound treatment 3320.0 1870.0 0.66 640.0 -10.7 -0.01 0.4642 0.6983 1216806 ChemDiv3_000925 CC(=O)OCCn1c(=O)[nH]c(=O)c2nsnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K02 compound treatment 1200.0 -246.0 -0.09 560.0 -90.7 -0.07 -0.111 -0.9937 3118177 ChemDiv3_000926 CC(C)(C)c1cc(Cl)c(O)c(/N=C/c2ccccc2O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K03 compound treatment 480.0 -966.0 -0.34 360.0 -291.0 -0.22 -0.4002 -0.9784 1915945 ChemDiv3_000927 CCOC(=O)/C=C(\C)/N1N=C2C(CCc3cc(OC)ccc23)C1c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K04 compound treatment 1240.0 -206.0 -0.07 320.0 -331.0 -0.25 -0.2312 -0.8753 1496403 ChemDiv3_000928 Cc1cn(cn1)S(=O)(=O)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K05 compound treatment 1400.0 -46.3 -0.02 3160.0 2510.0 1.93 1.3506 0.7011 1637460 ChemDiv3_000929 CCOc1cc(ccc1O)c2cc(C)c3c(ccc4ccccc43)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K06 compound treatment 480.0 -966.0 -0.34 680.0 29.3 0.02 -0.2265 -0.6592 3020943 ChemDiv3_000930 CCC1=C/C(=C/N(C)c2ccccc2)/C(=O)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K07 compound treatment 720.0 -726.0 -0.26 480.0 -171.0 -0.13 -0.2748 -0.9508 1083865 ChemDiv3_000931 FC(F)(F)c1cccc(NC(=O)c2ccco2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K08 compound treatment 800.0 -646.0 -0.23 320.0 -331.0 -0.25 -0.3416 -0.9987 1678628 ChemDiv3_000932 NCCCc1nc2cc3ccccc3cc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K09 compound treatment 6720.0 5270.0 1.87 440.0 -211.0 -0.16 1.2085 0.6436 3118178 ChemDiv3_000933 CN(C)c1n[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K10 compound treatment 1920.0 474.0 0.17 440.0 -211.0 -0.16 0.0045 0.0192 1535139 ChemDiv3_000934 NC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K11 compound treatment 360.0 -1090.0 -0.39 560.0 -90.7 -0.07 -0.3217 -0.8215 3020944 ChemDiv3_000935 NN1C(=O)/C(=C\c2ccccc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K12 compound treatment 1160.0 -286.0 -0.1 280.0 -371.0 -0.28 -0.273 -0.9036 1729835 ChemDiv3_000936 C(Cn1c(Cc2ccccc2)nc3ccccc13)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K13 compound treatment 1360.0 -86.3 -0.03 360.0 -291.0 -0.22 -0.1794 -0.7966 3020945 ChemDiv3_000937 CC1CCN(CC1)C(=O)/C=C/c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K14 compound treatment 1120.0 -326.0 -0.12 600.0 -50.7 -0.04 -0.1093 -0.8955 3118311 ChemDiv3_000938 Cc1nc2cc(/N=C\c3ccc(Cl)cc3)ccc2n1Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K15 compound treatment 400.0 -1050.0 -0.37 400.0 -251.0 -0.19 -0.3985 -0.9532 3020946 ChemDiv3_000939 CCCCc1ccc(NC(=O)CC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K16 compound treatment 600.0 -846.0 -0.3 320.0 -331.0 -0.25 -0.3918 -0.9965 1129901 ChemDiv3_000940 O=S(=O)(Cc1ccccc1)Nn2cnnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K17 compound treatment 720.0 -726.0 -0.26 480.0 -171.0 -0.13 -0.2748 -0.9508 3020947 ChemDiv3_000941 CC(NC(=O)/C=C/c1ccccc1Cl)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K18 compound treatment 1840.0 394.0 0.14 360.0 -291.0 -0.22 -0.059 -0.2242 3020310 ChemDiv3_000942 CCOc1ccc(OCCSc2nc3ccccc3n2Cc4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K19 compound treatment 9080.0 7630.0 2.71 480.0 -171.0 -0.13 1.8222 0.6721 1632334 ChemDiv3_000943 CCOC(=O)c1ccccc1NC(=O)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K20 compound treatment 7120.0 5670.0 2.01 280.0 -371.0 -0.28 1.222 0.6012 3118312 ChemDiv3_000944 CCOc1cccc2cc(C(=O)N)/c(=N/Cc3ccccc3)/oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K21 compound treatment 800.0 -646.0 -0.23 360.0 -291.0 -0.22 -0.3199 -0.9999 1564768 ChemDiv3_000945 COC(=O)c1cccc(NC(=O)COc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K22 compound treatment 2720.0 1270.0 0.45 600.0 -50.7 -0.04 0.292 0.6439 1122886 ChemDiv3_000946 COC(=O)C1=C(C)NC(=O)CC1c2ccccc2I 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K23 mock treatment 560.0 -886.0 -0.31 480.0 -171.0 -0.13 -0.315 -0.9247 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 K24 mock treatment 840.0 -606.0 -0.22 1920.0 1270.0 0.97 0.537 0.5381 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L01 compound treatment 1840.0 394.0 0.14 1160.0 509.0 0.39 0.3753 0.9038 1725902 ChemDiv3_000947 CCOC(=O)CSc1nc2ccccc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L02 compound treatment 1480.0 33.8 0.01 440.0 -211.0 -0.16 -0.1059 -0.653 3118313 ChemDiv3_000948 Clc1cccc(c1)C2OCC3(CO2)COC(OC3)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L03 compound treatment 1800.0 354.0 0.13 520.0 -131.0 -0.1 0.0178 0.1108 3020311 ChemDiv3_000949 Clc1ccc(/C=C\2/C=C(OC2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L04 compound treatment 1120.0 -326.0 -0.12 280.0 -371.0 -0.28 -0.2831 -0.9214 1215566 ChemDiv3_000950 COc1ccc(cc1)C2Nc3ccccc3C(=O)N2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L05 compound treatment 400.0 -1050.0 -0.37 240.0 -411.0 -0.32 -0.4854 -0.9967 1482448 ChemDiv3_000951 Clc1ccc(OCC(=O)NC2CCS(=O)(=O)C2)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L06 compound treatment 800.0 -646.0 -0.23 720.0 69.3 0.05 -0.1245 -0.5289 3118314 ChemDiv3_000952 O=C1CCC(=O)N1c2nccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L07 compound treatment 4280.0 2830.0 1.01 400.0 -251.0 -0.19 0.5748 0.5615 1240764 ChemDiv3_000953 Oc1ccccc1C2N(Cc3ccccc3)CCN2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L08 compound treatment 440.0 -1010.0 -0.36 520.0 -131.0 -0.1 -0.3233 -0.872 1351151 ChemDiv3_000954 Clc1c(sc2ccccc12)C(=O)NCc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L09 compound treatment 1120.0 -326.0 -0.12 320.0 -331.0 -0.25 -0.2613 -0.9367 1921190 ChemDiv3_000955 Nc1nnc(CCS(=O)(=O)c2ccc(Br)cc2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L10 compound treatment 480.0 -966.0 -0.34 520.0 -131.0 -0.1 -0.3133 -0.8773 1668007 ChemDiv3_000956 O=C(Nc1cccnc1)c2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L11 compound treatment 440.0 -1010.0 -0.36 360.0 -291.0 -0.22 -0.4102 -0.9744 3118315 ChemDiv3_000957 CN1CNC(=NS(=O)(=O)c2ccc(C)cc2)NC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L12 compound treatment 1040.0 -406.0 -0.14 280.0 -371.0 -0.28 -0.3031 -0.9503 1733849 ChemDiv3_000958 COC(=O)c1ccc(NC(=O)C2C(C3CCC2C3)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L13 compound treatment 480.0 -966.0 -0.34 640.0 -10.7 -0.01 -0.2482 -0.7238 3020312 ChemDiv3_000959 O=C/1OC(=N\C1=C/N2CCCCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L14 compound treatment 480.0 -966.0 -0.34 480.0 -171.0 -0.13 -0.335 -0.913 1222654 ChemDiv3_000960 CCCOc1ccc(cc1)C(=O)Nc2ccc-3c(Cc4ccccc43)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L15 compound treatment 360.0 -1090.0 -0.39 2120.0 1470.0 1.13 0.5252 0.4406 3020313 ChemDiv3_000961 Cc1cccc(/N=C/2\SCC(=O)N2c3cccc(C)c3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L16 compound treatment 440.0 -1010.0 -0.36 320.0 -331.0 -0.25 -0.4319 -0.9861 3118316 ChemDiv3_000962 COC(=O)CNC(c1ccccc1)c2cc(Br)ccc2NC(=O)CCN3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L17 compound treatment 920.0 -526.0 -0.19 360.0 -291.0 -0.22 -0.2898 -0.9961 3020314 ChemDiv3_000963 CCCOC(=O)c1ccc(NC(=O)/C=C/c2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L18 compound treatment 1000.0 -446.0 -0.16 440.0 -211.0 -0.16 -0.2263 -0.9999 3118317 ChemDiv3_000964 CCCCN1C(=O)/C(=C/N(C(=O)C)c2ccccc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L19 compound treatment 4360.0 2910.0 1.03 1480.0 829.0 0.64 1.1811 0.9729 1677249 ChemDiv3_000965 CCc1cccc(C)c1NC(=O)C2COc3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L20 compound treatment 920.0 -526.0 -0.19 360.0 -291.0 -0.22 -0.2898 -0.9961 3118318 ChemDiv3_000966 COc1ccc(CNC=C2C(=O)CC(C)(C)CC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L21 compound treatment 1760.0 314.0 0.11 2760.0 2110.0 1.62 1.2238 0.7539 3118319 ChemDiv3_000967 Clc1ccc(/C=C/2\SC(=O)N(CC(=O)Nc3cccnc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L22 compound treatment 1000.0 -446.0 -0.16 520.0 -131.0 -0.1 -0.1829 -0.9758 3020315 ChemDiv3_000968 CN(/C(=N\S(=O)(=O)c1ccc(C)cc1)/c2ccccc2)c3ccc(O)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L23 mock treatment 480.0 -966.0 -0.34 400.0 -251.0 -0.19 -0.3785 -0.9627 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 L24 mock treatment 3560.0 2110.0 0.75 400.0 -251.0 -0.19 0.3941 0.5091 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M01 compound treatment 960.0 -486.0 -0.17 2160.0 1510.0 1.16 0.6974 0.5953 3118320 ChemDiv3_000969 OC(=O)c1ccc(/N=C/c2cn(Cc3ccccc3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M02 compound treatment 440.0 -1010.0 -0.36 240.0 -411.0 -0.32 -0.4753 -0.9981 3020316 ChemDiv3_000970 Fc1ccc(cc1)c2nc3cc(/N=C/C=C/c4ccc5OCOc5c4)ccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M03 compound treatment 3280.0 1830.0 0.65 280.0 -371.0 -0.28 0.2588 0.3644 3118321 ChemDiv3_000971 COc1ccc2CC/C(=C\c3ccc(cc3)N(C)C)/C(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M04 compound treatment 360.0 -1090.0 -0.39 240.0 -411.0 -0.32 -0.4954 -0.995 1918339 ChemDiv3_000972 CC(C)(C)S(=O)(=O)c1ccc(s1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M05 compound treatment 3320.0 1870.0 0.66 640.0 -10.7 -0.01 0.4642 0.6983 1679374 ChemDiv3_000973 CCc1ccc(cc1)C2C3=C(CCCC3=O)OC4=C2C(=O)CCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M06 compound treatment 1440.0 -6.25 0.0 2160.0 1510.0 1.16 0.8178 0.7058 3118322 ChemDiv3_000974 CCC1=C/C(=C\c2ccc3OCOc3c2)/C(=O)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M07 compound treatment 2960.0 1510.0 0.54 1880.0 1230.0 0.94 1.0471 0.9643 3118323 ChemDiv3_000975 Brc1ccc2NC(=O)/C(=C/3\SC(=S)N(C3=O)c4cccc(Br)c4)/c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M08 compound treatment 6280.0 4830.0 1.71 360.0 -291.0 -0.22 1.0547 0.6099 1260425 ChemDiv3_000976 OC(=O)c1cncc(OC(=O)OCc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M09 compound treatment 4400.0 2950.0 1.05 200.0 -451.0 -0.35 0.4963 0.4497 1445337 ChemDiv3_000977 O=C(CCN1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)S(=O)(=O)Nc4nccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M10 compound treatment 1720.0 274.0 0.1 320.0 -331.0 -0.25 -0.1108 -0.4078 1228370 ChemDiv3_000978 COc1ccc(cc1)S(=O)(=O)N2CCCCC2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M11 compound treatment 680.0 -766.0 -0.27 1360.0 709.0 0.54 0.1929 0.3169 1353970 ChemDiv3_000979 CCS(=O)(=O)c1ccc(O)c(NC(=O)COc2ccc(OC)cc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M12 compound treatment 1360.0 -86.3 -0.03 760.0 109.0 0.08 0.0377 0.4222 3020317 ChemDiv3_000980 Brc1ccc(/C=N/c2nc3ccccc3n2CCN4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M13 compound treatment 800.0 -646.0 -0.23 880.0 229.0 0.18 -0.0376 -0.1301 1731333 ChemDiv3_000981 CCOC(=O)c1cccc(NC(=O)c2ccccc2Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M14 compound treatment 320.0 -1130.0 -0.4 440.0 -211.0 -0.16 -0.3969 -0.9208 3020318 ChemDiv3_000982 CN(C)c1ccc(/C=N/c2ccc3n(cnc3c2)c4ccc(C)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M15 compound treatment 880.0 -566.0 -0.2 1440.0 789.0 0.61 0.2865 0.4487 1678613 ChemDiv3_000983 CCOc1ccccc1C(=O)Nc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M16 compound treatment 1280.0 -166.0 -0.06 4000.0 3350.0 2.57 1.7765 0.6907 1685159 ChemDiv3_000984 CC1CC(C)CN(C1)C(=O)c2c(C)onc2c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M17 compound treatment 200.0 -1250.0 -0.44 1600.0 949.0 0.73 0.2027 0.2378 3020319 ChemDiv3_000985 CC(NC(=O)/C=C/c1ccc2OCOc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M18 compound treatment 320.0 -1130.0 -0.4 320.0 -331.0 -0.25 -0.462 -0.976 3118324 ChemDiv3_000986 CCOc1ccc(OCCSc2nc(=O)cc(C)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M19 compound treatment 1960.0 514.0 0.18 1400.0 749.0 0.58 0.5357 0.8876 1635077 ChemDiv3_000987 NC(=O)CCN1C(=O)c2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M20 compound treatment 280.0 -1170.0 -0.41 200.0 -451.0 -0.35 -0.5372 -0.996 1419414 ChemDiv3_000988 C(CN1CCOCC1)Cc2ccc(COc3ccccc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M21 compound treatment 4920.0 3470.0 1.23 1000.0 349.0 0.27 1.061 0.8413 1606786 ChemDiv3_000989 COC(=O)c1ccccc1NC(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M22 compound treatment 2080.0 634.0 0.22 320.0 -331.0 -0.25 -0.0205 -0.0606 1273253 ChemDiv3_000990 CNS(=O)(=O)c1ccc-2c(c1)C(=NO)c3cc(ccc32)S(=O)(=O)NC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M23 mock treatment 7080.0 5630.0 2.0 640.0 -10.7 -0.01 1.4074 0.7042 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 M24 mock treatment 5280.0 3830.0 1.36 440.0 -211.0 -0.16 0.8473 0.6187 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N01 compound treatment 1800.0 354.0 0.13 4600.0 3950.0 3.03 2.2327 0.7357 1426304 ChemDiv3_000991 Cc1cc(C)cc(OC(=O)CCN2C(=O)c3ccccc3C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N02 compound treatment 280.0 -1170.0 -0.41 4000.0 3350.0 2.57 1.5257 0.5858 3020320 ChemDiv3_000992 Brc1ccc(cc1)C2OCC(CO2)OC(=O)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N03 compound treatment 320.0 -1130.0 -0.4 560.0 -90.7 -0.07 -0.3317 -0.818 1721013 ChemDiv3_000993 Clc1ccc(cc1Cl)C(=O)NCCc2nc3ccccc3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N04 compound treatment 1200.0 -246.0 -0.09 960.0 309.0 0.24 0.1062 0.4195 3020321 ChemDiv3_000994 Brc1ccc(cc1)S(=O)(=O)/N=C(\Nc2ccccc2)/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N05 compound treatment 320.0 -1130.0 -0.4 480.0 -171.0 -0.13 -0.3752 -0.8922 1559580 ChemDiv3_000995 CCOC(=O)C1=C(C)N(C)C(=O)NC1c2ccccc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N06 compound treatment 1240.0 -206.0 -0.07 1360.0 709.0 0.54 0.3333 0.6067 3020344 ChemDiv3_000996 CSc1ccc(/C=c\2/sc3nc4c(C)c(C)ccc4n3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N07 compound treatment 5000.0 3550.0 1.26 1120.0 469.0 0.36 1.1462 0.8742 1921413 ChemDiv3_000997 CC(=O)Nc1ccc(NC(=O)/C=C/c2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N08 compound treatment 920.0 -526.0 -0.19 400.0 -251.0 -0.19 -0.2681 -0.9999 1649360 ChemDiv3_000998 CC(C)c1ccc(NC(=O)c2cccnc2Cl)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N09 compound treatment 240.0 -1210.0 -0.43 160.0 -491.0 -0.38 -0.5689 -0.998 1551746 ChemDiv3_000999 CC(=O)Nc1nnc(CCS(=O)(=O)c2ccc(C)cc2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N10 compound treatment 5000.0 3550.0 1.26 880.0 229.0 0.18 1.0159 0.7981 3118325 ChemDiv3_001000 Oc1ccccc1NC(=S)NC(=O)/C=C/c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N11 compound treatment 5480.0 4030.0 1.43 200.0 -451.0 -0.35 0.7672 0.5211 3118597 ChemDiv3_001001 NC(=NS(=O)(=O)c1ccc(NC(=O)OC2CCCC2)cc1)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N12 compound treatment 2000.0 554.0 0.2 280.0 -371.0 -0.28 -0.0623 -0.1802 1270195 ChemDiv3_001002 CC(N1C(=O)C2C3CC(C=C3)C2C1=O)C(=O)OCC(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N13 compound treatment 2720.0 1270.0 0.45 1240.0 589.0 0.45 0.6394 1.0 3118453 ChemDiv3_001003 O=S(=O)(/N=C(\OC1CCCCC1)/c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N14 compound treatment 6600.0 5150.0 1.83 720.0 69.3 0.05 1.3304 0.7274 1241887 ChemDiv3_001004 CCCOc1cccc(c1)C(=O)Nc2ccc(cc2)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N15 compound treatment 240.0 -1210.0 -0.43 800.0 149.0 0.11 -0.2215 -0.5 3020346 ChemDiv3_001005 COc1ccccc1N2C(=O)S/C(=C\c3ccccc3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N16 compound treatment 1600.0 154.0 0.05 1200.0 549.0 0.42 0.3368 0.792 1373892 ChemDiv3_001006 CC(=C)Cn1c(SCC(=O)NN)nc2ccccc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N17 compound treatment 160.0 -1290.0 -0.46 1880.0 1230.0 0.94 0.3447 0.3288 1493653 ChemDiv3_001007 CC(C)c1ccccc1NC(=O)c2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N18 compound treatment 480.0 -966.0 -0.34 640.0 -10.7 -0.01 -0.2482 -0.7238 3118454 ChemDiv3_001008 CC(=O)N(/C=C/1\SC(=S)N(Cc2ccccc2)C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N19 compound treatment 280.0 -1170.0 -0.41 920.0 269.0 0.21 -0.1463 -0.3164 1232650 ChemDiv3_001009 CCOC(=O)c1cccc(NC(=O)CCOc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N20 compound treatment 360.0 -1090.0 -0.39 760.0 109.0 0.08 -0.2131 -0.5404 3118455 ChemDiv3_001010 CC1(C)CC(=O)C(=CNCc2cccnc2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N21 compound treatment 680.0 -766.0 -0.27 1640.0 989.0 0.76 0.3449 0.4275 3118456 ChemDiv3_001011 CN1CCN(CC1)NC(=O)CN2C(=O)S/C(=C/c3ccc(Cl)cc3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N22 compound treatment 520.0 -926.0 -0.33 600.0 -50.7 -0.04 -0.2598 -0.7853 1118985 ChemDiv3_001012 COc1ccccc1NC(=O)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N23 mock treatment 1040.0 -406.0 -0.14 640.0 -10.7 -0.01 -0.1077 -0.7461 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 N24 mock treatment 640.0 -806.0 -0.29 1760.0 1110.0 0.85 0.4 0.4452 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O01 compound treatment 1960.0 514.0 0.18 360.0 -291.0 -0.22 -0.0289 -0.1004 3118457 ChemDiv3_001013 COC(=O)CNC(c1ccccc1)c2cc(Br)ccc2NC(=O)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O02 compound treatment 2120.0 674.0 0.24 320.0 -331.0 -0.25 -0.0105 -0.0301 3020347 ChemDiv3_001014 OC(=O)c1ccc(cc1)c2ccc(/C=C/3\Sc4ccccc4C3=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O03 compound treatment 360.0 -1090.0 -0.39 160.0 -491.0 -0.38 -0.5388 -0.9999 1433689 ChemDiv3_001015 COc1ccc(cc1OC)C2CC(=NN2C=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O04 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1216374 ChemDiv3_001016 CC1(C)CC(=CC(C)(C)N1)c2ccc(s2)C3=CC(C)(C)NC(C)(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O05 compound treatment 2160.0 714.0 0.25 320.0 -331.0 -0.25 -5.0E-4 -0.0013 1687051 ChemDiv3_001017 Oc1cccc(c1)c2nc3ccc4ccccc4c3c5CCCCc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O06 compound treatment 320.0 -1130.0 -0.4 160.0 -491.0 -0.38 -0.5489 -0.9996 3020348 ChemDiv3_001018 CCc1cc2c[n+](sc2s1)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O07 compound treatment 1920.0 474.0 0.17 240.0 -411.0 -0.32 -0.1041 -0.2914 1282936 ChemDiv3_001019 Cc1cc(=O)oc2cc(OCC(=O)O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O08 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1606633 ChemDiv3_001020 CC(=O)Oc1cncc(c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O09 compound treatment 280.0 -1170.0 -0.41 280.0 -371.0 -0.28 -0.4938 -0.9833 1192059 ChemDiv3_001021 O=C(NCc1ccccc1)C(Cc2ccccc2)N3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O10 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1475559 ChemDiv3_001022 COc1ccc(cc1)C(=O)NCC#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O11 compound treatment 240.0 -1210.0 -0.43 280.0 -371.0 -0.28 -0.5038 -0.9804 1080178 ChemDiv3_001023 Clc1ccc(cc1)C(=O)NC(=S)Nc2ccccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O12 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 3118458 ChemDiv3_001024 Clc1ccc(/C=N/c2nc3ccccc3n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O13 compound treatment 320.0 -1130.0 -0.4 320.0 -331.0 -0.25 -0.462 -0.976 1649330 ChemDiv3_001025 O=C(CNC(=O)c1ccccc1)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O14 compound treatment 400.0 -1050.0 -0.37 160.0 -491.0 -0.38 -0.5288 -1.0 3118459 ChemDiv3_001026 COc1ccccc1n2cnc3cc(/N=C/c4ccccc4O)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O15 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1328150 ChemDiv3_001027 Cc1ccc(cc1)N(C2CS(=O)(=O)CC2OC(=O)c3ccccc3)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O16 compound treatment 200.0 -1250.0 -0.44 360.0 -291.0 -0.22 -0.4704 -0.9499 1283075 ChemDiv3_001028 COc1ccc(NC(=O)CN2C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O17 compound treatment 280.0 -1170.0 -0.41 280.0 -371.0 -0.28 -0.4938 -0.9833 3118460 ChemDiv3_001029 Cc1ccccc1NC(=O)/C=C/c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O18 compound treatment 320.0 -1130.0 -0.4 2280.0 1630.0 1.25 0.602 0.4584 1317231 ChemDiv3_001030 NNC(=O)CNC(=O)C1COc2ccccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O19 compound treatment 680.0 -766.0 -0.27 320.0 -331.0 -0.25 -0.3717 -0.9994 1195157 ChemDiv3_001031 COc1ccc(CCNC(=O)C(C(C)C)N2C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O20 compound treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 3020350 ChemDiv3_001032 OC(=O)C/1=NN(C(=O)\C1=C/c2c[nH]c3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O21 compound treatment 320.0 -1130.0 -0.4 200.0 -451.0 -0.35 -0.5272 -0.9974 1154870 ChemDiv3_001033 COc1ccc(NC(=O)COc2ccc(C)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O22 compound treatment 320.0 -1130.0 -0.4 280.0 -371.0 -0.28 -0.4837 -0.9862 1195792 ChemDiv3_001034 CCNS(=O)(=O)c1ccc-2c(c1)C(=O)c3cc(ccc32)S(=O)(=O)NCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O23 mock treatment 320.0 -1130.0 -0.4 480.0 -171.0 -0.13 -0.3752 -0.8922 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 O24 mock treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P01 compound treatment 200.0 -1250.0 -0.44 240.0 -411.0 -0.32 -0.5355 -0.9863 1266216 ChemDiv3_001035 Cc1cccc(C)c1OC(=O)CN2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P02 compound treatment 240.0 -1210.0 -0.43 320.0 -331.0 -0.25 -0.4821 -0.9689 3118461 ChemDiv3_001036 Cc1ccccc1OCCn2c(S)nc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P03 compound treatment 3160.0 1710.0 0.61 880.0 229.0 0.18 0.5544 0.8759 1270060 ChemDiv3_001037 O=C(NC1CCCC1)c2cc3nc(cc(c4ccccc4)n3n2)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P04 compound treatment 200.0 -1250.0 -0.44 240.0 -411.0 -0.32 -0.5355 -0.9863 3020351 ChemDiv3_001038 Cc1ccccc1N/C(=N\S(=O)(=O)c2ccccc2)/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P05 compound treatment 920.0 -526.0 -0.19 240.0 -411.0 -0.32 -0.3549 -0.9687 1725017 ChemDiv3_001039 COc1ccc(CC(C)CC(=O)Nc2ccc(I)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P06 compound treatment 400.0 -1050.0 -0.37 280.0 -371.0 -0.28 -0.4637 -0.9914 1202851 ChemDiv3_001040 Nc1c(C#N)c(c(C#N)c2nc3ccccc3n12)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P07 compound treatment 1760.0 314.0 0.11 280.0 -371.0 -0.28 -0.1225 -0.401 1528263 ChemDiv3_001041 COc1ccc(NCC(O)Cn2c3ccc(Cl)cc3c4cc(Cl)ccc24)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P08 compound treatment 360.0 -1090.0 -0.39 240.0 -411.0 -0.32 -0.4954 -0.995 1730700 ChemDiv3_001042 Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3ccccc3Br)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P09 compound treatment 240.0 -1210.0 -0.43 200.0 -451.0 -0.35 -0.5472 -0.9944 3020380 ChemDiv3_001043 COc1ccc-2c(c1)C(=NN)c3cc(OC)ccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P10 compound treatment 240.0 -1210.0 -0.43 320.0 -331.0 -0.25 -0.4821 -0.9689 3118462 ChemDiv3_001044 OC(=O)CCN1C(=O)/C(=C/c2ccc(o2)c3ccc(Cl)cc3Cl)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P11 compound treatment 240.0 -1210.0 -0.43 1040.0 389.0 0.3 -0.0912 -0.1748 1544835 ChemDiv3_001045 CC(C)OC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P12 compound treatment 240.0 -1210.0 -0.43 280.0 -371.0 -0.28 -0.5038 -0.9804 3118463 ChemDiv3_001046 CCN1/C(=C\2/SC(=S)N(N)C2=O)/C=Cc3cc(C)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P13 compound treatment 520.0 -926.0 -0.33 120.0 -531.0 -0.41 -0.5204 -0.9943 3118464 ChemDiv3_001047 CCS(=O)(=O)CCc1nnc(NC(=O)Nc2cccc(c2)C(F)(F)F)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P14 compound treatment 240.0 -1210.0 -0.43 240.0 -411.0 -0.32 -0.5255 -0.9887 1403310 ChemDiv3_001048 CCOc1ccc(NC(=O)c2cc3ccccc3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P15 compound treatment 160.0 -1290.0 -0.46 280.0 -371.0 -0.28 -0.5239 -0.9742 3118465 ChemDiv3_001049 COc1ccc(/C=C/2\SC(=O)N(C2=O)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P16 compound treatment 200.0 -1250.0 -0.44 280.0 -371.0 -0.28 -0.5138 -0.9773 3020381 ChemDiv3_001050 CN(C)c1ccc(/C=C/c2ccncc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P17 compound treatment 280.0 -1170.0 -0.41 240.0 -411.0 -0.32 -0.5155 -0.991 1724755 ChemDiv3_001051 CCc1ccc(NC(=O)c2cc3ccccc3oc2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P18 compound treatment 720.0 -726.0 -0.26 320.0 -331.0 -0.25 -0.3617 -1.0 3020382 ChemDiv3_001052 CN1C(=O)/C(=C/Nc2ccccc2)/OC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P19 compound treatment 160.0 -1290.0 -0.46 280.0 -371.0 -0.28 -0.5239 -0.9742 1157486 ChemDiv3_001053 Cc1cccc(NC(=O)CCOc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P20 compound treatment 280.0 -1170.0 -0.41 200.0 -451.0 -0.35 -0.5372 -0.996 1218521 ChemDiv3_001054 CCOP(=S)(OCC)SCSn1c(=O)oc2cc(Cl)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P21 compound treatment 2880.0 1430.0 0.51 160.0 -491.0 -0.38 0.0933 0.1474 3118466 ChemDiv3_001055 O=C/1N(C(=S)S\C1=C\c2cccs2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P22 compound treatment 1440.0 -6.25 0.0 200.0 -451.0 -0.35 -0.2462 -0.7116 3020383 ChemDiv3_001056 CC(Oc1ccc(Br)cc1)C(=O)NN 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P23 mock treatment 1480.0 33.8 0.01 200.0 -451.0 -0.35 -0.2362 -0.6822 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2003 P24 mock treatment 320.0 -1130.0 -0.4 240.0 -411.0 -0.32 -0.5054 -0.9931 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A01 compound treatment 4440.0 3070.0 1.09 3760.0 2520.0 1.93 2.1366 0.9632 1172919 ChemDiv3_001409 COc1ccc(cc1OC)C(=O)Nc2ccc(cc2)c3nc4cc(C)cc(C)c4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A02 compound treatment 2840.0 1470.0 0.52 360.0 -883.0 -0.68 -0.1104 -0.1291 1360520 ChemDiv3_001410 CC(C)C1C(NC(CC1=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A03 compound treatment 5440.0 4070.0 1.44 440.0 -803.0 -0.62 0.5852 0.3728 1912544 ChemDiv3_001411 OC(=O)CSCCc1ccncc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A04 compound treatment 440.0 -930.0 -0.33 440.0 -803.0 -0.62 -0.669 -0.9571 1141661 ChemDiv3_001412 Clc1cccc2n(c3ccc(Br)cc3)c4nc(=O)[nH]c(=O)c4cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A05 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 3021166 ChemDiv3_001413 CC1(C)CC(=O)C(=CNCCN2CCOCC2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A06 compound treatment 240.0 -1130.0 -0.4 240.0 -1000.0 -0.77 -0.8278 -0.9538 3119497 ChemDiv3_001414 CC(O)c1cccc(NC(=O)c2cnn3C(CC(Nc23)c4cccs4)C(F)(F)F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A07 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1556247 ChemDiv3_001415 COc1cccc(c1)C(=O)Nc2ccc(cc2)c3cn4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A08 compound treatment 240.0 -1130.0 -0.4 200.0 -1040.0 -0.8 -0.8495 -0.9489 1464561 ChemDiv3_001416 CC(=O)Nc1cc2ccc(OC(=O)C)cc2oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A09 compound treatment 320.0 -1050.0 -0.37 200.0 -1040.0 -0.8 -0.8294 -0.9394 3021167 ChemDiv3_001417 Cc1cc(c(C#N)c(=S)[nH]1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A10 compound treatment 400.0 -970.0 -0.34 1080.0 -163.0 -0.12 -0.3316 -0.9059 1216127 ChemDiv3_001418 CC(=O)N(Cc1ccccc1)C2CCCc3c2[nH]c4ccc(C)cc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A11 compound treatment 240.0 -1130.0 -0.4 360.0 -883.0 -0.68 -0.7626 -0.9686 1428104 ChemDiv3_001419 O=C(Nn1cnc2ccccc2c1=O)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A12 compound treatment 440.0 -930.0 -0.33 240.0 -1000.0 -0.77 -0.7776 -0.9285 3119498 ChemDiv3_001420 CCOc1cc(/C=C\2/SC(=O)NC2=O)ccc1OCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A13 compound treatment 320.0 -1050.0 -0.37 280.0 -963.0 -0.74 -0.786 -0.9497 3021168 ChemDiv3_001421 O=C1CC(CC(=O)C1=CNCc2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A14 compound treatment 240.0 -1130.0 -0.4 200.0 -1040.0 -0.8 -0.8495 -0.9489 3119499 ChemDiv3_001422 CC(C)c1ccc(/C=C\2/N(C(=O)C)C(=S)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A15 compound treatment 120.0 -1250.0 -0.44 160.0 -1080.0 -0.83 -0.9013 -0.9567 1202793 ChemDiv3_001423 Cn1c(NC(=O)c2ccccc2NC(=O)c3ccccc3)nc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A16 compound treatment 240.0 -1130.0 -0.4 720.0 -523.0 -0.4 -0.5672 -1.0 1785399 ChemDiv3_001424 CCC(Nc1n[nH]c(=O)[nH]c1=O)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A17 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1694993 ChemDiv3_001425 Clc1c(cnn(c2ccccc2)c1=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A18 compound treatment 280.0 -1090.0 -0.39 200.0 -1040.0 -0.8 -0.8394 -0.9443 3119500 ChemDiv3_001426 O=C1/C(=C\NCc2ccccc2)/Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A19 compound treatment 200.0 -1170.0 -0.42 320.0 -923.0 -0.71 -0.7944 -0.9676 1385512 ChemDiv3_001427 O=C(Nc1ccc2nn(nc2c1)c3ccccc3)C(c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A20 compound treatment 240.0 -1130.0 -0.4 240.0 -1000.0 -0.77 -0.8278 -0.9538 3021169 ChemDiv3_001428 Brc1ccccc1c2nc3sc4CCCc4c3c(=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A21 compound treatment 240.0 -1130.0 -0.4 240.0 -1000.0 -0.77 -0.8278 -0.9538 1737060 ChemDiv3_001429 CN1CCc2c(C1)sc3NC(NC(=O)c23)c4ccc(OC(=O)c5ccccc5Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A22 compound treatment 360.0 -1010.0 -0.36 560.0 -683.0 -0.52 -0.6239 -0.9828 3021170 ChemDiv3_001430 CCOC(=O)c1c(N/C=C\2/C(=O)N(C)c3ccccc23)scc1c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A23 mock treatment 200.0 -1170.0 -0.42 200.0 -1040.0 -0.8 -0.8595 -0.9532 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 A24 mock treatment 800.0 -570.0 -0.2 3040.0 1800.0 1.38 0.8327 0.5971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B01 compound treatment 640.0 -730.0 -0.26 600.0 -643.0 -0.49 -0.532 -0.9547 3119501 ChemDiv3_001431 CCOc1ccc(/C=N\n2c(C)nnc2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B02 compound treatment 480.0 -890.0 -0.32 640.0 -603.0 -0.46 -0.5504 -0.9826 3119502 ChemDiv3_001432 CCOc1ccc(/C=C/2\SC(=NC2=O)Nc3cccc(C)c3C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B03 compound treatment 4200.0 2830.0 1.0 1360.0 117.0 0.09 0.7736 0.7675 3021171 ChemDiv3_001433 Cc1ccc(CN2CCN(CC2)/N=C\C=C\c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B04 compound treatment 280.0 -1090.0 -0.39 1480.0 237.0 0.18 -0.1446 -0.3382 3119503 ChemDiv3_001434 Cn1/c(=N/C(=O)CCSc2ccccc2)/sc3cc(Cl)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B05 compound treatment 200.0 -1170.0 -0.42 280.0 -963.0 -0.74 -0.8161 -0.9628 1384175 ChemDiv3_001435 Cc1cc(C)n(n1)C(=O)CNC(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B06 compound treatment 360.0 -1010.0 -0.36 320.0 -923.0 -0.71 -0.7542 -0.9501 3119504 ChemDiv3_001436 CC(C)(C)n1nc2CSCc2c1NC(=O)/C=C/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B07 compound treatment 240.0 -1130.0 -0.4 320.0 -923.0 -0.71 -0.7843 -0.9637 1576625 ChemDiv3_001437 Cc1ccc(C)c(c1)C(=O)COC(=O)c2cccc(n2)C(=O)OCC(=O)c3cc(C)ccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B08 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 1569810 ChemDiv3_001438 Clc1ccc(COc2ccc3c4CCCc4c(=O)oc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B09 compound treatment 1280.0 -90.0 -0.03 480.0 -763.0 -0.59 -0.4366 -0.7446 1294258 ChemDiv3_001439 Brc1cc(Br)c2cccnc2c1OC(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B10 compound treatment 520.0 -850.0 -0.3 320.0 -923.0 -0.71 -0.7141 -0.9276 3119505 ChemDiv3_001440 COc1cc([o+]c2ccccc12)c3ccc(cc3)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B11 compound treatment 320.0 -1050.0 -0.37 320.0 -923.0 -0.71 -0.7643 -0.955 3119506 ChemDiv3_001441 C(N1C2=NCCCN2c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B12 compound treatment 400.0 -970.0 -0.34 320.0 -923.0 -0.71 -0.7442 -0.945 3021172 ChemDiv3_001442 Clc1ccc2sc(cc(=O)c2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B13 compound treatment 320.0 -1050.0 -0.37 240.0 -1000.0 -0.77 -0.8077 -0.9445 1656193 ChemDiv3_001443 CC(C)(C)c1ccc(Cn2c(=N)n(CCO)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B14 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1367556 ChemDiv3_001444 Cc1nn(C(=O)C2(CC3CC4CC(C3)C2)C4)c(C)c1Sc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B15 compound treatment 160.0 -1210.0 -0.43 400.0 -843.0 -0.65 -0.761 -0.9801 3119507 ChemDiv3_001445 O=C1OC2(CCCC2)OC(=O)C1=Cc3c[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B16 compound treatment 200.0 -1170.0 -0.42 200.0 -1040.0 -0.8 -0.8595 -0.9532 1164014 ChemDiv3_001446 COc1ccc(Cn2c3ccccc3c4nc5ccccc5nc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B17 compound treatment 960.0 -410.0 -0.15 200.0 -1040.0 -0.8 -0.6689 -0.8221 1193371 ChemDiv3_001447 CN(C)c1ccc(CNc2ccc3n(cnc3c2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B18 compound treatment 160.0 -1210.0 -0.43 240.0 -1000.0 -0.77 -0.8478 -0.962 3119508 ChemDiv3_001448 CCN(CC)c1nc2c(C)cccn2c(=O)c1/C=N/O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B19 compound treatment 440.0 -930.0 -0.33 200.0 -1040.0 -0.8 -0.7993 -0.9232 3021173 ChemDiv3_001449 CCCOc1ccc(/C=C/C(=O)Nc2nccs2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B20 compound treatment 320.0 -1050.0 -0.37 280.0 -963.0 -0.74 -0.786 -0.9497 1665994 ChemDiv3_001450 C=CCN(CC=C)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccccc2c3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B21 compound treatment 360.0 -1010.0 -0.36 3400.0 2160.0 1.66 0.9178 0.5416 1144767 ChemDiv3_001451 Cn1cc(C(=O)c2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B22 compound treatment 960.0 -410.0 -0.15 1640.0 397.0 0.31 0.1129 0.3339 1499357 ChemDiv3_001452 CC(=O)N1CCN(CC1)C(=S)c2ccc(o2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B23 mock treatment 280.0 -1090.0 -0.39 800.0 -443.0 -0.34 -0.5137 -0.9979 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 B24 mock treatment 200.0 -1170.0 -0.42 400.0 -843.0 -0.65 -0.7509 -0.977 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C01 compound treatment 520.0 -850.0 -0.3 280.0 -963.0 -0.74 -0.7358 -0.9218 1424763 ChemDiv3_001453 Ic1ccc(Nc2nc3nonc3nc2N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C02 compound treatment 800.0 -570.0 -0.2 1400.0 157.0 0.12 -0.0576 -0.2444 3021226 ChemDiv3_001454 CCN/1CCS\C1=C/C=C/C2=[N+](CC)CCS2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C03 compound treatment 97160.0 95800.0 33.98 147600.0 146000.0 112.36 103.4797 0.8815 1048602 ChemDiv3_001455 CCCCc1oc2ccccc2c1C(=O)c3ccc(O)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C04 compound treatment 1000.0 -370.0 -0.13 1480.0 237.0 0.18 0.036 0.1604 1647191 ChemDiv3_001456 CC(C)(C)C1CCc2nc(N)c3c(=O)oc4ccccc4c3c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C05 compound treatment 320.0 -1050.0 -0.37 360.0 -883.0 -0.68 -0.7425 -0.9603 1247277 ChemDiv3_001457 COc1cccc(c1)C2N(C(=O)C)c3ccccc3NC4=C2C(=O)CC(C)(C)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C06 compound treatment 280.0 -1090.0 -0.39 3960.0 2720.0 2.09 1.2017 0.5664 3119509 ChemDiv3_001458 CCC(C)NC(=O)c1nn2C(CC(Nc2c1Cl)c3ccc(OC)cc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C07 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1174490 ChemDiv3_001459 COc1ccc(cc1)C2CC(=NN2S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C08 compound treatment 200.0 -1170.0 -0.42 160.0 -1080.0 -0.83 -0.8812 -0.9485 3021227 ChemDiv3_001460 O=C/1SC(=N\C1=C\c2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C09 compound treatment 280.0 -1090.0 -0.39 360.0 -883.0 -0.68 -0.7526 -0.9646 1606754 ChemDiv3_001461 COc1ccc(Nc2cc(C)c(C#N)c3nc4ccccc4n23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C10 compound treatment 480.0 -890.0 -0.32 240.0 -1000.0 -0.77 -0.7676 -0.9225 3021228 ChemDiv3_001462 CN(C)/C=C\1/Nc2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C11 compound treatment 5280.0 3910.0 1.39 160.0 -1080.0 -0.83 0.3931 0.2431 3119510 ChemDiv3_001463 Clc1ccccc1/C=C/C(=O)Nn2cnc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C12 compound treatment 480.0 -890.0 -0.32 400.0 -843.0 -0.65 -0.6807 -0.9456 3021229 ChemDiv3_001464 C/C(=C\c1ccccc1)/C=C\2/SC(=O)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C13 compound treatment 1080.0 -290.0 -0.1 280.0 -963.0 -0.74 -0.5953 -0.7978 3119511 ChemDiv3_001465 CC(C)CCNC=C1C(=O)CC(CC1=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C14 compound treatment 280.0 -1090.0 -0.39 320.0 -923.0 -0.71 -0.7743 -0.9595 3119512 ChemDiv3_001466 CC(=O)N/1C(=S)NC(=O)\C1=C/c2c(Cl)cccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C15 compound treatment 480.0 -890.0 -0.32 280.0 -963.0 -0.74 -0.7458 -0.928 1388103 ChemDiv3_001467 COc1ccc(cc1)n2c(nc3ccccc3c2=O)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C16 compound treatment 320.0 -1050.0 -0.37 240.0 -1000.0 -0.77 -0.8077 -0.9445 3119513 ChemDiv3_001468 CN1CCN(Cc2c(O)ccc3c(=O)c(c4ccc(Cl)cc4Cl)c(oc23)C(F)(F)F)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C17 compound treatment 280.0 -1090.0 -0.39 200.0 -1040.0 -0.8 -0.8394 -0.9443 1040451 ChemDiv3_001469 Clc1c(cnn(c2ccccc2)c1=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C18 compound treatment 320.0 -1050.0 -0.37 320.0 -923.0 -0.71 -0.7643 -0.955 3119818 ChemDiv3_001470 CCC(=O)Oc1ccc(Br)cc1/C=C/2\Sc3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C19 compound treatment 200.0 -1170.0 -0.42 240.0 -1000.0 -0.77 -0.8378 -0.958 1725871 ChemDiv3_001471 CC(C)(C)c1ccc(OCC(=O)Nc2ccc3c(c2)oc4ccccc43)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C20 compound treatment 280.0 -1090.0 -0.39 320.0 -923.0 -0.71 -0.7743 -0.9595 3021230 ChemDiv3_001472 CCOC(=O)c1c(C)n(CC)c2ccc(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C21 compound treatment 280.0 -1090.0 -0.39 2120.0 877.0 0.67 0.2028 0.2612 1698973 ChemDiv3_001473 Nc1ccc2nc(SCc3cccc(F)c3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C22 compound treatment 320.0 -1050.0 -0.37 400.0 -843.0 -0.65 -0.7208 -0.9656 3119657 ChemDiv3_001474 CN1C(=O)/C(=C/Nc2cccc3ccccc23)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C23 mock treatment 2880.0 1510.0 0.54 2920.0 1680.0 1.29 1.2893 0.9245 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 C24 mock treatment 400.0 -970.0 -0.34 3600.0 2360.0 1.81 1.0364 0.5626 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D01 compound treatment 320.0 -1050.0 -0.37 400.0 -843.0 -0.65 -0.7208 -0.9656 3021231 ChemDiv3_001475 CCc1ccc(/C=N/N2CCN(Cc3ccccc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D02 compound treatment 440.0 -930.0 -0.33 440.0 -803.0 -0.62 -0.669 -0.9571 3119658 ChemDiv3_001476 COC(=O)CCN1C(=O)/C(=C\c2cccs2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D03 compound treatment 1400.0 30.0 0.01 1680.0 437.0 0.34 0.2449 0.7292 3119659 ChemDiv3_001477 Clc1ccc(CN2CCN(CC2)/N=C\3/C(=O)Nc4ccccc34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D04 compound treatment 320.0 -1050.0 -0.37 400.0 -843.0 -0.65 -0.7208 -0.9656 1518636 ChemDiv3_001478 CCOC(=O)C1CCN(CC1)C(=S)NC2Cc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D05 compound treatment 280.0 -1090.0 -0.39 320.0 -923.0 -0.71 -0.7743 -0.9595 1671796 ChemDiv3_001479 Cc1cc(C)n(n1)C(=O)CNC(=O)COc2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D06 compound treatment 200.0 -1170.0 -0.42 360.0 -883.0 -0.68 -0.7727 -0.9723 1229552 ChemDiv3_001480 Cc1ccc(cc1)C(=O)Nc2c3CSCc3nn2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D07 compound treatment 320.0 -1050.0 -0.37 200.0 -1040.0 -0.8 -0.8294 -0.9394 1448199 ChemDiv3_001481 O=C(c1ccccc1)c2ccc(Oc3cc(C#N)c4ccccc4n3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D08 compound treatment 280.0 -1090.0 -0.39 320.0 -923.0 -0.71 -0.7743 -0.9595 1186512 ChemDiv3_001482 OC(=O)COc1cc2oc(=O)c3CCCc3c2cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D09 compound treatment 3280.0 1910.0 0.68 320.0 -923.0 -0.71 -0.0218 -0.0222 1377235 ChemDiv3_001483 CCCCn1c(N)nc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D10 compound treatment 200.0 -1170.0 -0.42 240.0 -1000.0 -0.77 -0.8378 -0.958 1023460 ChemDiv3_001484 Cc1cc(cc([o+]1)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D11 compound treatment 400.0 -970.0 -0.34 280.0 -963.0 -0.74 -0.7659 -0.9395 3021232 ChemDiv3_001485 Brc1ccc(s1)C(=O)CN2C3=NCCCN3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D12 compound treatment 760.0 -610.0 -0.22 640.0 -603.0 -0.46 -0.4802 -0.9401 1192182 ChemDiv3_001486 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(N2CCCC2)c3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D13 compound treatment 920.0 -450.0 -0.16 320.0 -923.0 -0.71 -0.6138 -0.8453 1376656 ChemDiv3_001487 CCCCn1c(=N)n(CCOc2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D14 compound treatment 280.0 -1090.0 -0.39 200.0 -1040.0 -0.8 -0.8394 -0.9443 1598019 ChemDiv3_001488 CC(=O)Oc1ccc2c(=O)c(c(C)oc2c1C)c3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D15 compound treatment 240.0 -1130.0 -0.4 200.0 -1040.0 -0.8 -0.8495 -0.9489 3119660 ChemDiv3_001489 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)c3cccc(Cl)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D16 compound treatment 200.0 -1170.0 -0.42 280.0 -963.0 -0.74 -0.8161 -0.9628 1618279 ChemDiv3_001490 Cc1ccc2nc(Cl)c(CC3CC(=NN3C(=O)CCCC(=O)O)c4ccccc4)cc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D17 compound treatment 240.0 -1130.0 -0.4 200.0 -1040.0 -0.8 -0.8495 -0.9489 1508458 ChemDiv3_001491 Cc1ccc(cc1)n2cnc3cc(NC(=O)c4ccccc4)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D18 compound treatment 320.0 -1050.0 -0.37 200.0 -1040.0 -0.8 -0.8294 -0.9394 1297401 ChemDiv3_001492 Cc1cc(OCc2c(F)cccc2Cl)c3c4CCCCc4c(=O)oc3c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D19 compound treatment 200.0 -1170.0 -0.42 440.0 -803.0 -0.62 -0.7292 -0.9815 1442148 ChemDiv3_001493 Cc1cccc(c1)N2COc3ccc4ccccc4c3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D20 compound treatment 280.0 -1090.0 -0.39 280.0 -963.0 -0.74 -0.796 -0.9543 1177599 ChemDiv3_001494 COc1ccccc1C(=O)Nc2c3CSCc3nn2c4ccc(Oc5ccccc5)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D21 compound treatment 240.0 -1130.0 -0.4 1640.0 397.0 0.31 -0.0678 -0.1345 1313552 ChemDiv3_001495 O=C(Cn1c2ncnn2c3ccccc13)c4ccc(cc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D22 compound treatment 360.0 -1010.0 -0.36 720.0 -523.0 -0.4 -0.5371 -0.9984 1124488 ChemDiv3_001496 CSc1nc2ccc3nc(NC(=O)c4ccccc4C)sc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D23 mock treatment 360.0 -1010.0 -0.36 840.0 -403.0 -0.31 -0.4719 -0.9973 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 D24 mock treatment 240.0 -1130.0 -0.4 5480.0 4240.0 3.25 2.0168 0.6153 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E01 compound treatment 2560.0 1190.0 0.42 760.0 -483.0 -0.37 0.0365 0.065 1465681 ChemDiv3_001497 Brc1ccc(NC(=O)c2ccc3nsnc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E02 compound treatment 1800.0 430.0 0.15 3120.0 1880.0 1.44 1.127 0.7776 1437302 ChemDiv3_001498 Clc1nc(NCCN2CCOCC2)nc(NC3CCCCC3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E03 compound treatment 2320.0 950.0 0.34 600.0 -643.0 -0.49 -0.1106 -0.1851 1173233 ChemDiv3_001499 S=C(Nc1ccccc1)Nc2ccc3c(c2)oc4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E04 compound treatment 2840.0 1470.0 0.52 440.0 -803.0 -0.62 -0.067 -0.083 1598038 ChemDiv3_001500 CCOc1cccc(c1)C(=O)Oc2cccc3ccc(C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E05 compound treatment 320.0 -1050.0 -0.37 1840.0 597.0 0.46 0.0609 0.1031 1192729 ChemDiv3_001501 CC(C)OC(=O)C1=C(C)OC23OC(=C(C#N)C31C(=O)c4ccccc42)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E06 compound treatment 600.0 -770.0 -0.27 320.0 -923.0 -0.71 -0.694 -0.9142 1490936 ChemDiv3_001502 CCC(C)C1NC(=O)NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E07 compound treatment 560.0 -810.0 -0.29 1000.0 -243.0 -0.19 -0.3349 -0.978 3119661 ChemDiv3_001503 Cc1ccc2nc(O)c(C3=NN(C(C3)c4ccccc4)C(=O)CCC(=O)O)c(c5ccccc5)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E08 compound treatment 1560.0 190.0 0.07 320.0 -923.0 -0.71 -0.4532 -0.6369 1449149 ChemDiv3_001504 CCC(=O)Nc1ccc(cc1NC(=O)CC)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E09 compound treatment 1920.0 550.0 0.2 3200.0 1960.0 1.5 1.2005 0.7923 1579424 ChemDiv3_001505 Cc1c(Cc2ccccc2)c(Cl)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E10 compound treatment 360.0 -1010.0 -0.36 240.0 -1000.0 -0.77 -0.7977 -0.9395 3119662 ChemDiv3_001506 CCN1C(=O)/C(=C\C=C\c2ccccc2Cl)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E11 compound treatment 4760.0 3390.0 1.2 6240.0 5000.0 3.84 3.5632 0.8862 1182144 ChemDiv3_001507 Cc1cc(N2CCOCC2)c3c(N)cc(C)c(C)c3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E12 compound treatment 78560.0 77200.0 27.38 27360.0 26100.0 20.05 33.5406 0.9883 3021233 ChemDiv3_001508 COc1cc(/C=C\2/SC(=S)NC2=O)ccc1OC(=O)c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E13 compound treatment 1080.0 -290.0 -0.1 600.0 -643.0 -0.49 -0.4216 -0.8366 1369185 ChemDiv3_001509 CCNCC(O)c1cccc(OC(=O)c2ccccc2C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E14 compound treatment 1400.0 30.0 0.01 4880.0 3640.0 2.79 1.9821 0.7098 3119663 ChemDiv3_001510 CCN1C(=O)/C(=C/2\NC(=S)NC2=O)/c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E15 compound treatment 1120.0 -250.0 -0.09 280.0 -963.0 -0.74 -0.5853 -0.7863 1448713 ChemDiv3_001511 CC(=O)Nc1ccccc1C(=O)N(Cc2ccccc2)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E16 compound treatment 1880.0 510.0 0.18 520.0 -723.0 -0.55 -0.2644 -0.453 3119664 ChemDiv3_001512 Cc1ccccc1/N=C/2\C(=O)N(CN3CCCCC3)c4ccc(Br)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E17 compound treatment 1000.0 -370.0 -0.13 1160.0 -82.7 -0.06 -0.1377 -0.9444 3021234 ChemDiv3_001513 Clc1c(cn[nH]c1=O)N2CCCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E18 compound treatment 2720.0 1350.0 0.48 800.0 -443.0 -0.34 0.0983 0.1675 3119665 ChemDiv3_001514 C/C(=C/1\Sc2ccccc2C1=O)/Nc3ccc(C)cc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E19 compound treatment 1320.0 -50.0 -0.02 6440.0 5200.0 3.99 2.8089 0.704 1455795 ChemDiv3_001515 O=C(COc1ccc2ccccc2c1)Nc3cccc(c3)c4nc5ncccc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E20 compound treatment 5280.0 3910.0 1.39 720.0 -523.0 -0.4 0.6971 0.4828 1548836 ChemDiv3_001516 CCOC(=O)c1c(C)n(c2ccc(OC)cc2)c3ccc(OC)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E21 compound treatment 1040.0 -330.0 -0.12 1160.0 -82.7 -0.06 -0.1277 -0.9586 3021235 ChemDiv3_001517 Nc1ccc2nc(SCc3ccccc3Cl)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E22 compound treatment 5720.0 4350.0 1.54 1200.0 -42.7 -0.03 1.068 0.6919 3119666 ChemDiv3_001518 O=C/1OC(=N\C1=C/Nc2ccccc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E23 mock treatment 5600.0 4230.0 1.5 1400.0 157.0 0.12 1.1465 0.7616 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 E24 mock treatment 1320.0 -50.0 -0.02 1640.0 397.0 0.31 0.2032 0.6649 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F01 compound treatment 320.0 -1050.0 -0.37 280.0 -963.0 -0.74 -0.786 -0.9497 3119667 ChemDiv3_001519 Clc1cccc(/C=N/N2CCN(Cc3ccccc3)CC2)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F02 compound treatment 320.0 -1050.0 -0.37 1360.0 117.0 0.09 -0.1997 -0.5211 3021236 ChemDiv3_001520 Brc1cccc(/C=C/2\SC(=S)N(CC(=O)N3CCCc4ccccc34)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F03 compound treatment 280.0 -1090.0 -0.39 3640.0 2400.0 1.84 1.028 0.5466 3119668 ChemDiv3_001521 C(N1CCN(CC1)/N=C/C=C/c2ccccc2)c3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F04 compound treatment 1080.0 -290.0 -0.1 2880.0 1640.0 1.26 0.8161 0.6471 1686599 ChemDiv3_001522 O=C(NCc1n[nH]c(=S)n1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F05 compound treatment 2200.0 830.0 0.29 480.0 -763.0 -0.59 -0.2058 -0.314 1371196 ChemDiv3_001523 CCOc1ccc(cc1)C(=O)NCC(=O)n2nc(C)cc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F06 compound treatment 3320.0 1950.0 0.69 1680.0 437.0 0.34 0.7266 0.9449 1292858 ChemDiv3_001524 Clc1ccc(cc1)n2nc3CSCc3c2NC(=O)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F07 compound treatment 880.0 -490.0 -0.17 1760.0 517.0 0.4 0.1579 0.3643 1135980 ChemDiv3_001525 COc1cccc(c1)C(=O)Nc2ccc(Cc3ccc(NC(=O)c4cccc(OC)c4)cc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F08 compound treatment 400.0 -970.0 -0.34 1720.0 477.0 0.37 0.0158 0.0314 3021237 ChemDiv3_001526 CC(C)C(N1C(=O)/C(=C/c2ccc(C)cc2)/SC1=S)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F09 compound treatment 840.0 -530.0 -0.19 10320.0 9080.0 6.97 4.7948 0.6878 1387806 ChemDiv3_001527 Nc1nc2ccccc2n1CCN3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F10 compound treatment 360.0 -1010.0 -0.36 3560.0 2320.0 1.78 1.0046 0.5536 3119819 ChemDiv3_001528 Cc1ccccc1C2CC(=O)NC(=C2C#N)SCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F11 compound treatment 6160.0 4790.0 1.7 1360.0 117.0 0.09 1.2652 0.7435 1175819 ChemDiv3_001529 CCn1c2nc(C)c(C(=O)OC)n2c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F12 compound treatment 2160.0 790.0 0.28 2160.0 917.0 0.7 0.6961 0.9184 3021293 ChemDiv3_001530 COc1cc(/C=C/2\SC(=S)N(C(C(C)C)C(=O)O)C2=O)cc(OC)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F13 compound treatment 560.0 -810.0 -0.29 760.0 -483.0 -0.37 -0.4652 -0.9921 1207608 ChemDiv3_001531 Cc1ccc(OCCn2c(N)nc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F14 compound treatment 1760.0 390.0 0.14 960.0 -283.0 -0.22 -0.0556 -0.2161 3021294 ChemDiv3_001532 CC(=O)Oc1ccc2c(=O)c(c3ccccc3)c(oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F15 compound treatment 1640.0 270.0 0.1 9360.0 8120.0 6.23 4.4743 0.7179 1429215 ChemDiv3_001533 Brc1cccc(NC(=O)C2C(=C2c3ccccc3)c4ccccc4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F16 compound treatment 1920.0 550.0 0.2 1240.0 -2.67 0.0 0.1365 0.6996 1221702 ChemDiv3_001534 COc1ccc(cc1)C2=NN(C(C2)c3cc4ccccc4nc3Cl)C(=O)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F17 compound treatment 1640.0 270.0 0.1 1880.0 637.0 0.49 0.4137 0.8298 1912856 ChemDiv3_001535 Clc1ccccc1S(=O)(=O)NC(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F18 compound treatment 2080.0 710.0 0.25 4120.0 2880.0 2.21 1.7401 0.7827 3021295 ChemDiv3_001536 COC(=O)C1=C(C)N(C)C(=S)NC1c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F19 compound treatment 3000.0 1630.0 0.58 1840.0 597.0 0.46 0.7331 0.9934 3021296 ChemDiv3_001537 C=CCn1c(=S)n(CC=C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F20 compound treatment 640.0 -730.0 -0.26 1440.0 197.0 0.15 -0.076 -0.2533 1512592 ChemDiv3_001538 CC(C)C(=O)Nc1c2CSCc2nn1c3ccc(Oc4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F21 compound treatment 480.0 -890.0 -0.32 1760.0 517.0 0.4 0.0576 0.1135 1573297 ChemDiv3_001539 c1coc(c1)c2cn3ccc4ccccc4c3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F22 compound treatment 360.0 -1010.0 -0.36 3840.0 2600.0 1.99 1.1566 0.5709 1238343 ChemDiv3_001540 CSc1nc2ccc3nc(NC(=O)c4ccccc4Cl)sc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F23 mock treatment 2520.0 1150.0 0.41 3800.0 2560.0 1.96 1.6767 0.8362 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 F24 mock treatment 800.0 -570.0 -0.2 1880.0 637.0 0.49 0.203 0.3834 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G01 compound treatment 720.0 -650.0 -0.23 4120.0 2880.0 2.21 1.3989 0.6299 3119820 ChemDiv3_001541 COC(=O)c1cc(ccc1Cl)c2ccc(/C=C\3/C(=C(C#N)C(=O)N=C3O)C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G02 compound treatment 1160.0 -210.0 -0.07 2720.0 1480.0 1.13 0.7493 0.6592 3021297 ChemDiv3_001542 COc1nc(Nc2ccc3OCOc3c2)nc(OC)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G03 compound treatment 1520.0 150.0 0.05 5000.0 3760.0 2.88 2.0773 0.72 1468410 ChemDiv3_001543 CC1(C)CC(=O)C=C(C1)NCC2CCN(CC2)C(=S)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G04 compound treatment 1400.0 30.0 0.01 520.0 -723.0 -0.55 -0.3848 -0.6934 3119821 ChemDiv3_001544 CCOC(=O)c1cc2NC(CC(n2n1)C(F)(F)F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G05 compound treatment 760.0 -610.0 -0.22 2040.0 797.0 0.61 0.2798 0.431 3021298 ChemDiv3_001545 CC(C)OC(=O)CSc1nc2ccccc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G06 compound treatment 360.0 -1010.0 -0.36 360.0 -883.0 -0.68 -0.7325 -0.9556 3119822 ChemDiv3_001546 CCc1ccc(cc1)N2N(O)c3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G07 compound treatment 360.0 -1010.0 -0.36 920.0 -323.0 -0.25 -0.4285 -0.9838 1165154 ChemDiv3_001547 Cc1cc(C)cc(CC2CC(=O)N(CCc3ccc4OCOc4c3)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G08 compound treatment 680.0 -690.0 -0.24 1320.0 77.3 0.06 -0.1311 -0.5205 1431964 ChemDiv3_001548 CC(=O)N1CC2(NC(=O)c3ccccc3N2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G09 compound treatment 360.0 -1010.0 -0.36 4680.0 3440.0 2.64 1.6126 0.6055 1737262 ChemDiv3_001549 Cc1cc(NCCO)n2c3ccccc3nc2c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G10 compound treatment 400.0 -970.0 -0.34 1000.0 -243.0 -0.19 -0.3751 -0.9585 3119823 ChemDiv3_001550 CCN1C(=O)/C(=C\c2ccsc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G11 compound treatment 360.0 -1010.0 -0.36 440.0 -803.0 -0.62 -0.6891 -0.9667 3119824 ChemDiv3_001551 O=C1CC(CC(=O)C1=CNCc2ccncc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G12 compound treatment 1040.0 -330.0 -0.12 600.0 -643.0 -0.49 -0.4317 -0.8512 3021299 ChemDiv3_001552 COc1ccc(cc1)N2C(=O)/C(=C\C=C\c3ccccc3)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G13 compound treatment 6760.0 5390.0 1.91 8760.0 7520.0 5.77 5.4329 0.8936 3119825 ChemDiv3_001553 COc1ccc(/C=c/2\oc3cccc4c(OC)ccc(c2=O)c34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G14 compound treatment 560.0 -810.0 -0.29 640.0 -603.0 -0.46 -0.5303 -0.9737 1172050 ChemDiv3_001554 CCOC(=O)c1ccc(Nc2ncnc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G15 compound treatment 2800.0 1430.0 0.51 1920.0 677.0 0.52 0.7264 0.9999 3119826 ChemDiv3_001555 COc1cc(/C=C/2\SC(=S)NC2=O)ccc1OCc3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G16 compound treatment 480.0 -890.0 -0.32 680.0 -563.0 -0.43 -0.5287 -0.9881 3119827 ChemDiv3_001556 O=C/1N(CN2CCOCC2)c3ccccc3\C1=N\c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G17 compound treatment 1040.0 -330.0 -0.12 4640.0 3400.0 2.61 1.7615 0.6747 3021300 ChemDiv3_001557 CC1=C(C(NC(=S)N1)c2ccc(F)cc2)C(=O)Nc3cccc(Cl)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G18 compound treatment 5880.0 4510.0 1.6 4360.0 3120.0 2.39 2.8236 0.9808 3119828 ChemDiv3_001558 CC(=O)N(/N=C/1\Sc2ccccc2C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G19 compound treatment 3600.0 2230.0 0.79 1280.0 37.3 0.03 0.5796 0.7322 1604755 ChemDiv3_001559 O=C(COc1ccc2ccccc2c1)Nc3ccc4nn(nc4c3)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G20 compound treatment 560.0 -810.0 -0.29 600.0 -643.0 -0.49 -0.5521 -0.9669 1447009 ChemDiv3_001560 CCOC(=O)c1c(C)n(Cc2ccccc2)c3ccc(OC(=O)C)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G21 compound treatment 1560.0 190.0 0.07 2640.0 1400.0 1.07 0.8062 0.7501 3119829 ChemDiv3_001561 CCc1ccc(cc1)N2NC(=O)/C(=C\c3c(C)c(C#N)c4nc5ccccc5n4c3O)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G22 compound treatment 1520.0 150.0 0.05 3080.0 1840.0 1.41 1.035 0.7333 3021301 ChemDiv3_001562 CC/1=NN(C(=S)\C1=C\Nc2cccc(Br)c2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G23 mock treatment 1640.0 270.0 0.1 2040.0 797.0 0.61 0.5006 0.8079 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 G24 mock treatment 1320.0 -50.0 -0.02 560.0 -683.0 -0.52 -0.3831 -0.7306 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H01 compound treatment 240.0 -1130.0 -0.4 360.0 -883.0 -0.68 -0.7626 -0.9686 3119830 ChemDiv3_001563 Oc1ccc2ccccc2c1/C=N/N3CCN(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H02 compound treatment 920.0 -450.0 -0.16 640.0 -603.0 -0.46 -0.44 -0.8991 1322139 ChemDiv3_001564 CCOC(=O)c1c(C)n(c2ccccc2)c3ccc(OC(=O)c4ccccc4NC(=O)CC)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H03 compound treatment 760.0 -610.0 -0.22 920.0 -323.0 -0.25 -0.3282 -0.9977 3119831 ChemDiv3_001565 C1CN(CCN1/N=C\c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H04 compound treatment 320.0 -1050.0 -0.37 840.0 -403.0 -0.31 -0.482 -0.9957 3119832 ChemDiv3_001566 CCOc1ccc2n(C)/c(=N/C(=O)c3cc4ccccc4cc3OC)/sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H05 compound treatment 1240.0 -130.0 -0.05 560.0 -683.0 -0.52 -0.4032 -0.7664 1575164 ChemDiv3_001567 O=C(Sc1ccc(Oc2ccc(SC(=O)c3ccco3)cc2)cc1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H06 compound treatment 520.0 -850.0 -0.3 1320.0 77.3 0.06 -0.1712 -0.5572 1615009 ChemDiv3_001568 CC(C)(C)n1nc2CSCc2c1NC(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H07 compound treatment 600.0 -770.0 -0.27 560.0 -683.0 -0.52 -0.5637 -0.9539 1373227 ChemDiv3_001569 OC(=O)C1CCCCC1C(=O)Nc2cccc(c2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H08 compound treatment 4720.0 3350.0 1.19 960.0 -283.0 -0.22 0.6869 0.5686 1684031 ChemDiv3_001570 OCc1cc(=O)c(O)c(o1)C(Nc2ccccn2)c3ccccc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H09 compound treatment 2800.0 1430.0 0.51 680.0 -563.0 -0.43 0.0533 0.0799 1601378 ChemDiv3_001571 OC(Cn1c(=N)n(Cc2ccccc2)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H10 compound treatment 880.0 -490.0 -0.17 840.0 -403.0 -0.31 -0.3415 -0.9629 3119833 ChemDiv3_001572 CCOc1ccc(cc1)c2c(C#N)c(N)nc(SCC(=O)c3ccc(Cl)cc3)c2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H11 compound treatment 360.0 -1010.0 -0.36 600.0 -643.0 -0.49 -0.6022 -0.9877 1449806 ChemDiv3_001573 COc1ccc(cc1)C(=O)Cn2c(=N)n(CC=C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H12 compound treatment 600.0 -770.0 -0.27 1320.0 77.3 0.06 -0.1512 -0.5408 3119834 ChemDiv3_001574 Cc1ccc(Sc2c(nc3sccn23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H13 compound treatment 320.0 -1050.0 -0.37 760.0 -483.0 -0.37 -0.5254 -1.0 1668029 ChemDiv3_001575 Nc1nc2ccccc2n1CCOc3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H14 compound treatment 360.0 -1010.0 -0.36 1760.0 517.0 0.4 0.0275 0.0514 3119835 ChemDiv3_001576 COc1ccc2c(=O)c(c3ccccc3C)c(oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H15 compound treatment 920.0 -450.0 -0.16 840.0 -403.0 -0.31 -0.3315 -0.9527 3021302 ChemDiv3_001577 Brc1cccc(c1)N2C(=O)C3C(C(C=CC3c4ccccc4)c5ccccc5)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H16 compound treatment 320.0 -1050.0 -0.37 720.0 -523.0 -0.4 -0.5471 -0.9993 3119836 ChemDiv3_001578 Cc1ccc(cc1)C2CC(=NN2C(=O)c3ccc(Br)o3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H17 compound treatment 960.0 -410.0 -0.15 840.0 -403.0 -0.31 -0.3214 -0.9409 1123601 ChemDiv3_001579 CCOC(=O)CNc1ccc(cc1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H18 compound treatment 2280.0 910.0 0.32 920.0 -323.0 -0.25 0.0531 0.1305 3119837 ChemDiv3_001580 Clc1ccc(cc1)C(=O)/C=C/C=C/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H19 compound treatment 600.0 -770.0 -0.27 680.0 -563.0 -0.43 -0.4986 -0.9756 3119838 ChemDiv3_001581 Cc1ccc(O)c(c1)c2cc(nc(n2)c3ccccc3)C(F)(F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H20 compound treatment 3840.0 2470.0 0.88 880.0 -363.0 -0.28 0.4227 0.4598 3021303 ChemDiv3_001582 Cc1ccc(c(C)c1)n2nc3CSCc3c2NC(=O)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H21 compound treatment 560.0 -810.0 -0.29 5240.0 4000.0 3.07 1.9668 0.6381 1718858 ChemDiv3_001583 Cc1nc2n(CCN3CCOCC3)c4ccccc4n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H22 compound treatment 800.0 -570.0 -0.2 1640.0 397.0 0.31 0.0727 0.1987 1657446 ChemDiv3_001584 O=C(Nc1ccc(cc1)c2nc3ccccc3o2)c4ccc(Oc5ccccc5)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H23 mock treatment 1040.0 -330.0 -0.12 880.0 -363.0 -0.28 -0.2797 -0.9259 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 H24 mock treatment 360.0 -1010.0 -0.36 640.0 -603.0 -0.46 -0.5805 -0.992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I01 compound treatment 440.0 -930.0 -0.33 280.0 -963.0 -0.74 -0.7559 -0.9339 1538533 ChemDiv3_001585 COc1ccc(cc1)C2NC(=S)NC(=C2C(=O)N)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I02 compound treatment 320.0 -1050.0 -0.37 320.0 -923.0 -0.71 -0.7643 -0.955 3119978 ChemDiv3_001586 Cc1cccc(CSCc2nnc(NC(=O)/C=C/c3ccccc3)s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I03 compound treatment 200.0 -1170.0 -0.42 720.0 -523.0 -0.4 -0.5772 -0.9999 3021304 ChemDiv3_001587 CC1(C)CC(=O)C(=CNCCN2CCN(CC2)C(=O)Nc3ccc(Cl)c(Cl)c3)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I04 compound treatment 360.0 -1010.0 -0.36 240.0 -1000.0 -0.77 -0.7977 -0.9395 3119979 ChemDiv3_001588 FC(F)(F)c1c2CCc3ccccc3-c2nc4cc(nn14)C(=O)Nc5ccc(Cl)cc5Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I05 compound treatment 320.0 -1050.0 -0.37 240.0 -1000.0 -0.77 -0.8077 -0.9445 1590870 ChemDiv3_001589 CCOc1ccc2c(=O)c(Oc3ccc(OC)cc3)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I06 compound treatment 360.0 -1010.0 -0.36 280.0 -963.0 -0.74 -0.7759 -0.9447 3119980 ChemDiv3_001590 CC(C)N1C(=O)/C(=C/c2cccc(Br)c2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I07 compound treatment 360.0 -1010.0 -0.36 280.0 -963.0 -0.74 -0.7759 -0.9447 3119981 ChemDiv3_001591 OC(=O)C(CC(=O)Nc1cccc(c1)C(F)(F)F)Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I08 compound treatment 360.0 -1010.0 -0.36 160.0 -1080.0 -0.83 -0.8411 -0.9293 3427363 ChemDiv3_001592 COc1cc2CCN3CC4N(CCc5cc(OC)c(OC)cc45)CC3c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I09 compound treatment 280.0 -1090.0 -0.39 200.0 -1040.0 -0.8 -0.8394 -0.9443 1494132 ChemDiv3_001593 N#Cc1c2CCCc2c(Nc3ccccc3)n4c5ccccc5nc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I10 compound treatment 320.0 -1050.0 -0.37 280.0 -963.0 -0.74 -0.786 -0.9497 3119982 ChemDiv3_001594 C/C(=C\c1ccccc1)/C=C\2/SC(=S)N(C3CCCCC3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I11 compound treatment 280.0 -1090.0 -0.39 680.0 -563.0 -0.43 -0.5789 -0.9985 3021305 ChemDiv3_001595 O=C1CC(CC(=O)C1=CNCCN2CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I12 compound treatment 400.0 -970.0 -0.34 280.0 -963.0 -0.74 -0.7659 -0.9395 3119983 ChemDiv3_001596 O=C/1N\C(=N/c2ccccc2)\S\C1=C\c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I13 compound treatment 560.0 -810.0 -0.29 1520.0 277.0 0.21 -0.0526 -0.1472 3021306 ChemDiv3_001597 COc1ccc2c(=O)/c(=C/c3ccc4OCOc4c3)/oc5cccc1c52 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I14 compound treatment 320.0 -1050.0 -0.37 360.0 -883.0 -0.68 -0.7425 -0.9603 1203947 ChemDiv3_001598 CC(C)Nc1nc(nc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I15 compound treatment 200.0 -1170.0 -0.42 1440.0 197.0 0.15 -0.1864 -0.4218 3021307 ChemDiv3_001599 COc1cc(/C=c\2/sc3nc4ccccc4n3c2=O)cc(OC)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I16 compound treatment 480.0 -890.0 -0.32 800.0 -443.0 -0.34 -0.4636 -0.9993 3119984 ChemDiv3_001600 CN(C)CN1C(=O)/C(=N\c2ccc3ccccc3c2)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I17 compound treatment 760.0 -610.0 -0.22 1400.0 157.0 0.12 -0.0676 -0.2728 1726741 ChemDiv3_001601 O=C(NCc1ccncc1)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I18 compound treatment 360.0 -1010.0 -0.36 280.0 -963.0 -0.74 -0.7759 -0.9447 3021308 ChemDiv3_001602 CCOc1ccc(cc1)N(/C=C/2\Sc3ccccc3C2=O)C(=O)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I19 compound treatment 280.0 -1090.0 -0.39 200.0 -1040.0 -0.8 -0.8394 -0.9443 1339625 ChemDiv3_001603 Fc1ccccc1C(=O)Nc2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I20 compound treatment 4600.0 3230.0 1.15 1680.0 437.0 0.34 1.0476 0.8774 1713175 ChemDiv3_001604 COc1ccc2n(c(C)c(C(=O)O)c2c1)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I21 compound treatment 400.0 -970.0 -0.34 480.0 -763.0 -0.59 -0.6573 -0.9679 3119985 ChemDiv3_001605 OC(=O)c1ccc(cc1)n2nnnc2SCC(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I22 compound treatment 400.0 -970.0 -0.34 2920.0 1680.0 1.29 0.6672 0.5006 3119986 ChemDiv3_001606 CCOC(=O)c1ccc(NC=C2C(=O)NC(=O)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I23 mock treatment 480.0 -890.0 -0.32 240.0 -1000.0 -0.77 -0.7676 -0.9225 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 I24 mock treatment 2920.0 1550.0 0.55 360.0 -883.0 -0.68 -0.0904 -0.1035 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J01 compound treatment 360.0 -1010.0 -0.36 360.0 -883.0 -0.68 -0.7325 -0.9556 3021309 ChemDiv3_001607 Cc1ccc(/C=N/N2CCN(Cc3ccccc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J02 compound treatment 440.0 -930.0 -0.33 480.0 -763.0 -0.59 -0.6473 -0.9632 1644734 ChemDiv3_001608 C=CCNC(=O)c1cc(=O)c2ccccc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J03 compound treatment 440.0 -930.0 -0.33 1000.0 -243.0 -0.19 -0.365 -0.9634 3021310 ChemDiv3_001609 COc1ccccc1/C=C/C=N\N2CCN(CC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J04 compound treatment 280.0 -1090.0 -0.39 680.0 -563.0 -0.43 -0.5789 -0.9985 1423874 ChemDiv3_001610 O=C(CCOc1ccccc1)Nc2nc3c(ccc4ccccc34)s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J05 compound treatment 280.0 -1090.0 -0.39 160.0 -1080.0 -0.83 -0.8612 -0.9394 1201781 ChemDiv3_001611 O=C(COC(=O)c1ccccc1Nc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J06 compound treatment 360.0 -1010.0 -0.36 280.0 -963.0 -0.74 -0.7759 -0.9447 1685020 ChemDiv3_001612 CC(C)(C)c1ccc(cc1)C(=O)Nc2c3CSCc3nn2c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J07 compound treatment 320.0 -1050.0 -0.37 280.0 -963.0 -0.74 -0.786 -0.9497 1369848 ChemDiv3_001613 COc1ccc(NC(=O)c2ccc(cc2)N3C(=O)c4ccccc4C3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J08 compound treatment 920.0 -450.0 -0.16 360.0 -883.0 -0.68 -0.592 -0.8504 3021370 ChemDiv3_001614 CC(N1C(=O)/C(=C\c2ccc(C)o2)/SC1=S)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J09 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 1352921 ChemDiv3_001615 COC(=O)Cn1c(=N)n(C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J10 compound treatment 200.0 -1170.0 -0.42 600.0 -643.0 -0.49 -0.6424 -0.9963 1463142 ChemDiv3_001616 COC(=O)C1C(C(=C(NC1=O)SCc2ccccc2)C#N)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J11 compound treatment 200.0 -1170.0 -0.42 1360.0 117.0 0.09 -0.2298 -0.541 1215092 ChemDiv3_001617 C=CCn1c(=N)n(CC(=O)c2ccc(cc2)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J12 compound treatment 280.0 -1090.0 -0.39 280.0 -963.0 -0.74 -0.796 -0.9543 3021371 ChemDiv3_001618 COc1ccc(cc1)C(=O)On2c(cc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J13 compound treatment 680.0 -690.0 -0.24 2000.0 757.0 0.58 0.238 0.3773 1340086 ChemDiv3_001619 O=C(Nc1ccccc1C(=O)NC2CCCCC2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J14 compound treatment 360.0 -1010.0 -0.36 200.0 -1040.0 -0.8 -0.8194 -0.9343 3021372 ChemDiv3_001620 Oc1ccccc1/C=C/2\N=C3CCCCCN3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J15 compound treatment 240.0 -1130.0 -0.4 240.0 -1000.0 -0.77 -0.8278 -0.9538 1558867 ChemDiv3_001621 Cc1cc(C)cc(NC(=O)Nc2ccccc2C(=O)Nc3cc(C)cc(C)c3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J16 compound treatment 160.0 -1210.0 -0.43 240.0 -1000.0 -0.77 -0.8478 -0.962 1137505 ChemDiv3_001622 Cc1ccc(cc1)C2=NN(C(C2)c3cn(nc3c4ccc(C)cc4)c5ccccc5)C(=O)CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J17 compound treatment 440.0 -930.0 -0.33 320.0 -923.0 -0.71 -0.7342 -0.9395 1319284 ChemDiv3_001623 Cc1cc(O)ccc1n2c(=O)c3cc4c(=O)n(c5ccc(O)cc5C)c(=O)c4cc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J18 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1596958 ChemDiv3_001624 CC1CCc2nc(NC(=O)c3ccc(cc3)S(=O)(=O)N(CC=C)CC=C)sc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J19 compound treatment 640.0 -730.0 -0.26 240.0 -1000.0 -0.77 -0.7274 -0.8957 3021373 ChemDiv3_001625 FC(F)(F)C1(CC(=O)c2ccco2)NCCN1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J20 compound treatment 560.0 -810.0 -0.29 560.0 -683.0 -0.52 -0.5738 -0.96 3119987 ChemDiv3_001626 Cc1ccc(cc1)n2nc3CSCc3c2NC(=O)/C=C\c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J21 compound treatment 800.0 -570.0 -0.2 480.0 -763.0 -0.59 -0.557 -0.8992 3021374 ChemDiv3_001627 O=C(CCCN1C(=O)/C(=C\c2cccs2)/SC1=S)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J22 compound treatment 360.0 -1010.0 -0.36 320.0 -923.0 -0.71 -0.7542 -0.9501 3119988 ChemDiv3_001628 Cn1/c(=N\C(=O)c2ccc(cc2)S(=O)(=O)N3CCCCC3)/sc4c1ccc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J23 mock treatment 360.0 -1010.0 -0.36 240.0 -1000.0 -0.77 -0.7977 -0.9395 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 J24 mock treatment 5880.0 4510.0 1.6 520.0 -723.0 -0.55 0.739 0.4364 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K01 compound treatment 1320.0 -50.0 -0.02 280.0 -963.0 -0.74 -0.5351 -0.7239 1467244 ChemDiv3_001629 CC(C)(C)c1cc(cc(c1)S(=O)(=O)CCc2ccccn2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K02 compound treatment 720.0 -650.0 -0.23 360.0 -883.0 -0.68 -0.6422 -0.8972 3021375 ChemDiv3_001630 Fc1ccccc1CSCc2nnc(NC(=O)/C=C/c3ccccc3)s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K03 compound treatment 520.0 -850.0 -0.3 1680.0 437.0 0.34 0.0242 0.0536 3119989 ChemDiv3_001631 CCCC/1=NN(C(=O)\C1=C\N(C)C)c2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K04 compound treatment 240.0 -1130.0 -0.4 400.0 -843.0 -0.65 -0.7409 -0.9735 3119990 ChemDiv3_001632 CC(C)OC(=O)c1cnn2c(cc(nc12)c3ccc(C)cc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K05 compound treatment 480.0 -890.0 -0.32 360.0 -883.0 -0.68 -0.7024 -0.9396 1566112 ChemDiv3_001633 COC(=O)COc1ccc2c(=O)c(Oc3ccc(OC)cc3)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K06 compound treatment 760.0 -610.0 -0.22 1120.0 -123.0 -0.09 -0.2196 -0.9305 3119991 ChemDiv3_001634 O=S(=O)(NCc1ccccc1)c2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K07 compound treatment 600.0 -770.0 -0.27 360.0 -883.0 -0.68 -0.6723 -0.9202 1513154 ChemDiv3_001635 OC(=O)CN1C(=O)CC(Cc2ccc(Cl)cc2)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K08 compound treatment 320.0 -1050.0 -0.37 800.0 -443.0 -0.34 -0.5037 -0.999 1680762 ChemDiv3_001636 COC(CN(C1CCCc2c1[nH]c3ccc(C)cc23)C(=O)C)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K09 compound treatment 4640.0 3270.0 1.16 2560.0 1320.0 1.01 1.5354 0.9977 1379664 ChemDiv3_001637 CCc1c(C)c(C#N)c2nc3ccccc3n2c1n4ccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K10 compound treatment 560.0 -810.0 -0.29 920.0 -323.0 -0.25 -0.3783 -0.9973 3119992 ChemDiv3_001638 CN(C)c1ccc(/C=C/C=C\2/SC(=S)N(C)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K11 compound treatment 400.0 -970.0 -0.34 7040.0 5800.0 4.45 2.9038 0.6505 3119993 ChemDiv3_001639 Cc1ccc(SCC/2=NN(C(=O)\C2=C\NCc3ccco3)c4nc5ccccc5s4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K12 compound treatment 1960.0 590.0 0.21 880.0 -363.0 -0.28 -0.0489 -0.1403 3021376 ChemDiv3_001640 OC(=O)COc1ccc(/C=C\2/NC(=S)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K13 compound treatment 320.0 -1050.0 -0.37 1440.0 197.0 0.15 -0.1563 -0.3886 3021377 ChemDiv3_001641 COc1ccc(cc1)C(=O)C(=C2Nc3ccccc3N2)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K14 compound treatment 280.0 -1090.0 -0.39 440.0 -803.0 -0.62 -0.7092 -0.9748 3119994 ChemDiv3_001642 Oc1ccc2c(=O)c(c3ccc(Cl)cc3Cl)c(oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K15 compound treatment 760.0 -610.0 -0.22 440.0 -803.0 -0.62 -0.5887 -0.9015 1190196 ChemDiv3_001643 COc1cc(OC)cc(c1)c2nc3ccccc3c(=O)n2OC(=O)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K16 compound treatment 400.0 -970.0 -0.34 640.0 -603.0 -0.46 -0.5705 -0.9894 3021378 ChemDiv3_001644 O=C(CCN1C(=O)c2ccccc2C1=O)C(=C3Nc4ccccc4N3)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K17 compound treatment 280.0 -1090.0 -0.39 1080.0 -163.0 -0.12 -0.3617 -0.8902 1229182 ChemDiv3_001645 Cc1onc(c1C(=O)n2cnc3cc(C)c(C)cc23)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K18 compound treatment 600.0 -770.0 -0.27 440.0 -803.0 -0.62 -0.6289 -0.933 1396504 ChemDiv3_001646 CCOC(=O)c1c(NC=O)scc1c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K19 compound treatment 440.0 -930.0 -0.33 4760.0 3520.0 2.7 1.6761 0.6161 1614792 ChemDiv3_001647 COc1cc2ccccc2cc1C(=O)Nc3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K20 compound treatment 2560.0 1190.0 0.42 760.0 -483.0 -0.37 0.0365 0.065 3021379 ChemDiv3_001648 CN1C(=O)/C(=C\NN2CCOCC2)/c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K21 compound treatment 640.0 -730.0 -0.26 1240.0 -2.67 0.0 -0.1846 -0.7127 3120138 ChemDiv3_001649 CCN(CC)c1ccc(/C=C\2/C(=O)NN(C2=O)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K22 compound treatment 920.0 -450.0 -0.16 1200.0 -42.7 -0.03 -0.136 -0.8348 1271860 ChemDiv3_001650 O=c1n(cnc2sc3CCCCc3c12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K23 mock treatment 920.0 -450.0 -0.16 400.0 -843.0 -0.65 -0.5703 -0.8559 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 K24 mock treatment 960.0 -410.0 -0.15 1160.0 -82.7 -0.06 -0.1477 -0.9309 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L01 compound treatment 360.0 -1010.0 -0.36 640.0 -603.0 -0.46 -0.5805 -0.992 3120139 ChemDiv3_001651 CCOc1ccccc1/C=N\n2cnnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L02 compound treatment 1000.0 -370.0 -0.13 880.0 -363.0 -0.28 -0.2897 -0.9411 3120140 ChemDiv3_001652 COC(=O)c1ccccc1NC=C2C(=O)NC(=S)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L03 compound treatment 4280.0 2910.0 1.03 280.0 -963.0 -0.74 0.2074 0.1633 3021380 ChemDiv3_001653 Cc1ccc(cc1)N2CCN(CC2)/N=C\C=C\c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L04 compound treatment 640.0 -730.0 -0.26 280.0 -963.0 -0.74 -0.7057 -0.9012 3120141 ChemDiv3_001654 CCOc1ccc2n(C)/c(=N\C(=O)CCOc3ccccc3)/sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L05 compound treatment 960.0 -410.0 -0.15 520.0 -723.0 -0.55 -0.4952 -0.8633 1125649 ChemDiv3_001655 CNc1ccccc1C(=O)OCC(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L06 compound treatment 640.0 -730.0 -0.26 640.0 -603.0 -0.46 -0.5103 -0.9624 1333133 ChemDiv3_001656 Clc1ccc(cc1)n2nc3CSCc3c2NC(=O)c4ccc(cc4)C(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L07 compound treatment 520.0 -850.0 -0.3 560.0 -683.0 -0.52 -0.5838 -0.9655 3021381 ChemDiv3_001657 CC(=O)N1N=C(N)SC21CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L08 compound treatment 880.0 -490.0 -0.17 440.0 -803.0 -0.62 -0.5586 -0.8725 3120142 ChemDiv3_001658 COc1cccc(/C=C/2\SC(=S)N(C(Cc3ccccc3)C(=O)O)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L09 compound treatment 600.0 -770.0 -0.27 400.0 -843.0 -0.65 -0.6506 -0.9265 1735087 ChemDiv3_001659 Cc1ccc(Cn2c(=N)n(CC(=O)O)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L10 compound treatment 280.0 -1090.0 -0.39 520.0 -723.0 -0.55 -0.6657 -0.9844 1873281 ChemDiv3_001660 CCOC(=O)CSC1=C(C#N)C(C(C(=O)OC)C(=O)N1)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L11 compound treatment 360.0 -1010.0 -0.36 320.0 -923.0 -0.71 -0.7542 -0.9501 3021382 ChemDiv3_001661 C=CCn1c2nc(cn2c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L12 compound treatment 320.0 -1050.0 -0.37 400.0 -843.0 -0.65 -0.7208 -0.9656 1591933 ChemDiv3_001662 Cc1[nH]c2ccccc2c1CN3CCC(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L13 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1237818 ChemDiv3_001663 O=C(NCc1ccccc1)c2ccccc2NC(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L14 compound treatment 640.0 -730.0 -0.26 1280.0 37.3 0.03 -0.1628 -0.625 1564490 ChemDiv3_001664 COc1ccc(C)cc1S(=O)(=O)N2CCN(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L15 compound treatment 400.0 -970.0 -0.34 840.0 -403.0 -0.31 -0.4619 -0.9986 1447061 ChemDiv3_001665 COc1ccc(OC)c(Nc2nc3nonc3nc2N4CCC(C)CC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L16 compound treatment 320.0 -1050.0 -0.37 760.0 -483.0 -0.37 -0.5254 -1.0 1193553 ChemDiv3_001666 CC(C)c1cc(NS(=O)(=O)c2ccccc2)c(O)c(c1)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L17 compound treatment 680.0 -690.0 -0.24 480.0 -763.0 -0.59 -0.5871 -0.9251 1642809 ChemDiv3_001667 O=C(OCc1nc2ccccc2[nH]1)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L18 compound treatment 400.0 -970.0 -0.34 840.0 -403.0 -0.31 -0.4619 -0.9986 3021383 ChemDiv3_001668 CCOC(=O)c1s/c(=N\C(=O)c2ccc(OCC)cc2)/n(C)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L19 compound treatment 440.0 -930.0 -0.33 1320.0 77.3 0.06 -0.1913 -0.5707 3120143 ChemDiv3_001669 COc1ccccc1NC(=O)c2cc3ccccc3c(/C=N/c4ccc(NC(=O)C)cc4)c2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L20 compound treatment 560.0 -810.0 -0.29 920.0 -323.0 -0.25 -0.3783 -0.9973 1201425 ChemDiv3_001670 COc1ccc(CC(=O)Nc2c3CSCc3nn2c4ccc(C)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L21 compound treatment 840.0 -530.0 -0.19 2640.0 1400.0 1.07 0.6256 0.5744 3120144 ChemDiv3_001671 O=C(CCCN1C(=O)/C(=C/c2cccs2)/SC1=S)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L22 compound treatment 2480.0 1110.0 0.39 1600.0 357.0 0.27 0.4724 0.9844 3021384 ChemDiv3_001672 Cc1cccc(NC(=S)NCCCN2CCOCC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L23 mock treatment 1560.0 190.0 0.07 600.0 -643.0 -0.49 -0.3012 -0.6049 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 L24 mock treatment 1680.0 310.0 0.11 1280.0 37.3 0.03 0.098 0.8626 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M01 compound treatment 520.0 -850.0 -0.3 1480.0 237.0 0.18 -0.0844 -0.2395 1915602 ChemDiv3_001673 CC(C)c1ccc(cc1)S(=O)(=O)CCc2ccc(C)[n+](C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M02 compound treatment 360.0 -1010.0 -0.36 2040.0 797.0 0.61 0.1795 0.2531 3120145 ChemDiv3_001674 CC(C)(C)C(=O)Nc1nnc(SCc2ccc(Cl)cc2Cl)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M03 compound treatment 400.0 -970.0 -0.34 1360.0 117.0 0.09 -0.1796 -0.505 1626138 ChemDiv3_001675 CC(=C1C(=O)CC(C)(C)CC1=O)NCC2CCNCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M04 compound treatment 1680.0 310.0 0.11 720.0 -523.0 -0.4 -0.206 -0.4951 3021385 ChemDiv3_001676 CC1CCCCN1C(=O)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M05 compound treatment 96600.0 95200.0 33.78 16720.0 15500.0 11.88 32.2898 0.9017 3120146 ChemDiv3_001677 CC(C)(C)c1cc(/C=C/2\SC(=S)NC2=O)cc(c1O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M06 compound treatment 1600.0 230.0 0.08 1240.0 -2.67 0.0 0.0562 0.6891 1369956 ChemDiv3_001678 OC(=O)c1ccccc1C(=O)Nc2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M07 compound treatment 320.0 -1050.0 -0.37 1640.0 397.0 0.31 -0.0477 -0.0991 3021386 ChemDiv3_001679 CC(C(Cc1cc(C)cc(C)c1)C(=O)O)C(=O)Nc2cccc(c2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M08 compound treatment 960.0 -410.0 -0.15 400.0 -843.0 -0.65 -0.5603 -0.845 1367959 ChemDiv3_001680 CCOC(=O)c1c(C)sc2Sc3ccc(Cl)cc3Nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M09 compound treatment 1160.0 -210.0 -0.07 760.0 -483.0 -0.37 -0.3147 -0.8326 1584915 ChemDiv3_001681 CCc1c(C)c(C#N)c2[nH]c3ccccc3n2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M10 compound treatment 1720.0 350.0 0.12 2480.0 1240.0 0.95 0.7595 0.7928 3120147 ChemDiv3_001682 CN1C(=O)/C(=C\c2ccc(o2)c3ccc(C)c(Cl)c3)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M11 compound treatment 680.0 -690.0 -0.24 320.0 -923.0 -0.71 -0.674 -0.8993 1579702 ChemDiv3_001683 CCC(=O)N1C(C2=C(CC(CC2=O)c3ccccc3)Nc4ccccc14)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M12 compound treatment 1640.0 270.0 0.1 320.0 -923.0 -0.71 -0.4332 -0.606 1133651 ChemDiv3_001684 C(Cc1cccs1)Nc2ncnc3sc4CCCc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M13 compound treatment 2120.0 750.0 0.27 560.0 -683.0 -0.52 -0.1825 -0.3104 3120148 ChemDiv3_001685 O=C(COc1ccccc1)C(=C2Nc3ccccc3N2)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M14 compound treatment 1480.0 110.0 0.04 280.0 -963.0 -0.74 -0.495 -0.6688 3021387 ChemDiv3_001686 OC(=O)c1ccc(/N=C/2\SC(Cc3cccc(Cl)c3)C(=O)N2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M15 compound treatment 5760.0 4390.0 1.56 400.0 -843.0 -0.65 0.6438 0.3817 1726607 ChemDiv3_001687 Cc1cccc(c1)c2nc3ccccc3c(=O)n2OC(=O)c4ccc(C)c(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M16 compound treatment 400.0 -970.0 -0.34 720.0 -523.0 -0.4 -0.5271 -0.9971 3120149 ChemDiv3_001688 CC1CN(CC(C)O1)C(=O)c2sc3cc(C)ccc3c2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M17 compound treatment 280.0 -1090.0 -0.39 480.0 -763.0 -0.59 -0.6874 -0.9797 1427209 ChemDiv3_001689 CC(C)CCNC(=O)C1c2ccccc2Oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M18 compound treatment 2520.0 1150.0 0.41 1080.0 -163.0 -0.12 0.2002 0.4692 1691429 ChemDiv3_001690 CCOC(=O)c1c(C)c(C)sc1NC(=O)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M19 compound treatment 560.0 -810.0 -0.29 560.0 -683.0 -0.52 -0.5738 -0.96 1389933 ChemDiv3_001691 Cc1ccc2cc(C(=O)N)c(=N)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M20 compound treatment 1120.0 -250.0 -0.09 880.0 -363.0 -0.28 -0.2596 -0.8884 3120150 ChemDiv3_001692 CCOC(=O)c1c(N/C=C\2/C(=O)N(C)c3ccccc23)sc4CCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M21 compound treatment 11520.0 10200.0 3.6 32640.0 31400.0 24.1 19.5904 0.8038 3021478 ChemDiv3_001693 CC/1=NN(C(=O)\C1=C\c2ccc(o2)c3cccc(Cl)c3C)c4cccc(c4)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M22 compound treatment 246120.0 245000.0 86.82 141360.0 140000.0 107.57 137.4578 0.9944 3120151 ChemDiv3_001694 Cc1cccc(OCCOc2ccc(Br)cc2/C=C/3\SC(=S)NC3=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M23 mock treatment 2640.0 1270.0 0.45 1600.0 357.0 0.27 0.5126 0.9717 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 M24 mock treatment 840.0 -530.0 -0.19 1800.0 557.0 0.43 0.1696 0.3629 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N01 compound treatment 640.0 -730.0 -0.26 400.0 -843.0 -0.65 -0.6406 -0.9192 3021479 ChemDiv3_001695 C(=N/n1cnnc1)\c2cccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N02 compound treatment 840.0 -530.0 -0.19 8120.0 6880.0 5.28 3.6005 0.6815 3118032 ChemDiv3_001696 COc1ccc(cc1)n2nc3CSCc3c2NC(=O)c4ccccc4C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N03 compound treatment 920.0 -450.0 -0.16 680.0 -563.0 -0.43 -0.4183 -0.9084 3021480 ChemDiv3_001697 Clc1ccccc1CN2CCN(CC2)/N=C/C=C\c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N04 compound treatment 5240.0 3870.0 1.37 360.0 -883.0 -0.68 0.4916 0.3211 3117871 ChemDiv3_001698 Cn1/c(=N\C(=O)CCOc2ccccc2)/sc3cc(Br)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N05 compound treatment 1760.0 390.0 0.14 1160.0 -82.7 -0.06 0.053 0.3479 1590935 ChemDiv3_001699 CCC(=O)c1ccc(OC(=O)C2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N06 compound treatment 480.0 -890.0 -0.32 520.0 -723.0 -0.55 -0.6156 -0.9643 1201811 ChemDiv3_001700 Cc1cccc(COc2ccc3c(C)cc(=O)oc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N07 compound treatment 640.0 -730.0 -0.26 280.0 -963.0 -0.74 -0.7057 -0.9012 1923213 ChemDiv3_001701 OCCN1CCN(CC#CCn2c3ccccc3c4ccccc24)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N08 compound treatment 280.0 -1090.0 -0.39 920.0 -323.0 -0.25 -0.4486 -0.9768 1578316 ChemDiv3_001702 O=C(CC(C1CCCCC1=O)c2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N09 compound treatment 520.0 -850.0 -0.3 400.0 -843.0 -0.65 -0.6707 -0.9396 1582025 ChemDiv3_001703 CCN(CC)CCCn1c(cn2c1nc3ccccc32)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N10 compound treatment 840.0 -530.0 -0.19 720.0 -523.0 -0.4 -0.4167 -0.9403 1873341 ChemDiv3_001704 COC(=O)C1C(C(=C(NC1=O)SCC=C)C#N)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N11 compound treatment 320.0 -1050.0 -0.37 440.0 -803.0 -0.62 -0.6991 -0.9709 1619409 ChemDiv3_001705 OCCn1c(=N)n(CC=C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N12 compound treatment 400.0 -970.0 -0.34 400.0 -843.0 -0.65 -0.7008 -0.9563 1130658 ChemDiv3_001706 O=c1c2ccccc2nc3c4ccccc4c(nn13)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N13 compound treatment 1040.0 -330.0 -0.12 7600.0 6360.0 4.88 3.3684 0.6899 1508826 ChemDiv3_001707 CCOC(=O)c1c(C)nn(Cc2cccc(Cl)c2)c1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N14 compound treatment 400.0 -970.0 -0.34 440.0 -803.0 -0.62 -0.6791 -0.9621 1777814 ChemDiv3_001708 C/C(=C(\C#N)/c1nc2ccccc2[nH]1)/O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N15 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1709331 ChemDiv3_001709 Cn1c(Sc2nnc(N)s2)nc3n(C)c(=O)n(C)c(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N16 compound treatment 400.0 -970.0 -0.34 640.0 -603.0 -0.46 -0.5705 -0.9894 3117873 ChemDiv3_001710 COc1ccc(Nc2nc3c(C)cccn3c(=O)c2/C=N/Cc4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N17 compound treatment 400.0 -970.0 -0.34 360.0 -883.0 -0.68 -0.7225 -0.9506 3117874 ChemDiv3_001711 COCc1cc(C)nc(SCC(=O)c2ccc(O)c(O)c2)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N18 compound treatment 720.0 -650.0 -0.23 640.0 -603.0 -0.46 -0.4902 -0.9483 3021481 ChemDiv3_001712 CCOc1ccc2n(C)/c(=N\C(=O)c3ccc(cc3)S(=O)(=O)N4CCc5ccccc45)/sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N19 compound treatment 720.0 -650.0 -0.23 640.0 -603.0 -0.46 -0.4902 -0.9483 3117875 ChemDiv3_001713 CCCN1C/C(=C\c2ccc(OC)cc2)/C(=O)\C(=C/c3ccc(OC)cc3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N20 compound treatment 640.0 -730.0 -0.26 360.0 -883.0 -0.68 -0.6623 -0.9129 1525047 ChemDiv3_001714 Cc1ccc(c(C)c1)n2nc3CSCc3c2NC(=O)COc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N21 compound treatment 4960.0 3590.0 1.27 5560.0 4320.0 3.31 3.2442 0.9137 3021482 ChemDiv3_001715 Cc1cccc(NC2=NC(=O)/C(=C/c3ccc(F)cc3)/S2)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N22 compound treatment 4720.0 3350.0 1.19 2120.0 877.0 0.67 1.3166 0.9638 1667814 ChemDiv3_001716 CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)N4CCc5ccccc5C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N23 mock treatment 760.0 -610.0 -0.22 6200.0 4960.0 3.81 2.5381 0.6658 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 N24 mock treatment 1320.0 -50.0 -0.02 2440.0 1200.0 0.92 0.6374 0.6933 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O01 compound treatment 240.0 -1130.0 -0.4 120.0 -1120.0 -0.86 -0.8929 -0.9394 3021483 ChemDiv3_001717 OC(=O)C/1=NN(C(=O)\C1=C\c2cccs2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O02 compound treatment 280.0 -1090.0 -0.39 280.0 -963.0 -0.74 -0.796 -0.9543 3117876 ChemDiv3_001718 CCOc1cc(C=C2C(=O)NC(=S)NC2=O)ccc1OCCOc3ccc(cc3)C(C)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O03 compound treatment 360.0 -1010.0 -0.36 400.0 -843.0 -0.65 -0.7108 -0.9612 3021484 ChemDiv3_001719 CC1(C)CC(=O)C=C(C1)NCCCn2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O04 compound treatment 400.0 -970.0 -0.34 200.0 -1040.0 -0.8 -0.8093 -0.9289 3117877 ChemDiv3_001720 CC(C)NC(=O)c1cc2NC(CC(n2n1)C(F)(F)F)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O05 compound treatment 280.0 -1090.0 -0.39 280.0 -963.0 -0.74 -0.796 -0.9543 3021485 ChemDiv3_001721 CCOc1cc(/C=c\2/sc3nc4ccccc4n3c2=O)ccc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O06 compound treatment 2360.0 990.0 0.35 280.0 -963.0 -0.74 -0.2743 -0.3352 3117878 ChemDiv3_001722 CC(C)(C)C(O)(CC#CCN1CCCC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O07 compound treatment 280.0 -1090.0 -0.39 240.0 -1000.0 -0.77 -0.8177 -0.9493 1383847 ChemDiv3_001723 CCOc1ccc(NC(=O)C(C)C(Cc2ccc(C)cc2)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O08 compound treatment 2600.0 1230.0 0.44 280.0 -963.0 -0.74 -0.2141 -0.2494 1624938 ChemDiv3_001724 O=C1CCCN1CCNC(=S)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O09 compound treatment 360.0 -1010.0 -0.36 240.0 -1000.0 -0.77 -0.7977 -0.9395 1249695 ChemDiv3_001725 CCC1(CC)Cc2ccccc2-c3[nH]c(=S)n(Cc4ccccc4)c(=O)c31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O10 compound treatment 2360.0 990.0 0.35 280.0 -963.0 -0.74 -0.2743 -0.3352 3117879 ChemDiv3_001726 CN1C(=O)/C(=C\c2ccncc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O11 compound treatment 320.0 -1050.0 -0.37 240.0 -1000.0 -0.77 -0.8077 -0.9445 1610336 ChemDiv3_001727 CC(=O)Nc1ncc2C(=O)CC(Cc2n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O12 compound treatment 240.0 -1130.0 -0.4 760.0 -483.0 -0.37 -0.5455 -0.9992 1305118 ChemDiv3_001728 CCOc1ccc2c(=O)c(Oc3ccccc3Br)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O13 compound treatment 320.0 -1050.0 -0.37 400.0 -843.0 -0.65 -0.7208 -0.9656 3117880 ChemDiv3_001729 CC(N1C(=O)c2ccccc2C1=O)C(=O)C(=C3Nc4ccccc4N3)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O14 compound treatment 200.0 -1170.0 -0.42 280.0 -963.0 -0.74 -0.8161 -0.9628 3021518 ChemDiv3_001730 Cc1ccc(cc1)n/2c(cs\c2=N\C(=O)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O15 compound treatment 240.0 -1130.0 -0.4 320.0 -923.0 -0.71 -0.7843 -0.9637 1281278 ChemDiv3_001731 Clc1c(cnn(c2ccccc2)c1=O)N3CCN(CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O16 compound treatment 120.0 -1250.0 -0.44 240.0 -1000.0 -0.77 -0.8579 -0.9657 3021519 ChemDiv3_001732 COc1ccc(N/C=C\2/Sc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O17 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 1330175 ChemDiv3_001733 CCC(C)c1ccc(NC(=O)c2cc3ccccc3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O18 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 1220991 ChemDiv3_001734 CCOC(=O)c1c(CC(C)C)csc1NC(=O)c2ccccc2OC(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O19 compound treatment 280.0 -1090.0 -0.39 320.0 -923.0 -0.71 -0.7743 -0.9595 3117881 ChemDiv3_001735 N/C(=N\O)/CCCN1CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O20 compound treatment 320.0 -1050.0 -0.37 320.0 -923.0 -0.71 -0.7643 -0.955 3117882 ChemDiv3_001736 CCOC(=O)c1c(C)c(C)sc1N/C=C\2/C(=O)N(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O21 compound treatment 680.0 -690.0 -0.24 400.0 -843.0 -0.65 -0.6305 -0.9116 1915686 ChemDiv3_001737 O=C(CSc1nnnn1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O22 compound treatment 400.0 -970.0 -0.34 240.0 -1000.0 -0.77 -0.7876 -0.9341 3021520 ChemDiv3_001738 Cc1nnc(C)n1/N=C\c2cccc(OCc3ccccc3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O23 mock treatment 2280.0 910.0 0.32 440.0 -803.0 -0.62 -0.2075 -0.2982 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 O24 mock treatment 520.0 -850.0 -0.3 280.0 -963.0 -0.74 -0.7358 -0.9218 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P01 compound treatment 1680.0 310.0 0.11 320.0 -923.0 -0.71 -0.4231 -0.5903 3021521 ChemDiv3_001739 C(=N/n1cnnc1)\c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P02 compound treatment 400.0 -970.0 -0.34 160.0 -1080.0 -0.83 -0.8311 -0.9238 1680808 ChemDiv3_001740 CC1CC(C)CN(C1)S(=O)(=O)c2ccc(cc2)C(=O)Nc3ccc(C)cc3C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P03 compound treatment 2400.0 1030.0 0.37 360.0 -883.0 -0.68 -0.2208 -0.2868 3021522 ChemDiv3_001741 Cc1nnc(C)n1/N=C/c2cc(Br)cc(Br)c2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P04 compound treatment 200.0 -1170.0 -0.42 320.0 -923.0 -0.71 -0.7944 -0.9676 3117883 ChemDiv3_001742 O=C(CN1C(=O)/C(=C/c2ccccc2)/SC1=S)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P05 compound treatment 280.0 -1090.0 -0.39 320.0 -923.0 -0.71 -0.7743 -0.9595 1137126 ChemDiv3_001743 Cc1cc(C)c(C)c(C(=O)COC(=O)c2cc(O)nc3ccccc23)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P06 compound treatment 280.0 -1090.0 -0.39 880.0 -363.0 -0.28 -0.4703 -0.987 1455967 ChemDiv3_001744 CCCc1cc(=O)oc2cc(OCC(=O)OCc3ccccc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P07 compound treatment 240.0 -1130.0 -0.4 360.0 -883.0 -0.68 -0.7626 -0.9686 1311949 ChemDiv3_001745 OC(CN1CCCCC1)CN2c3ccccc3Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P08 compound treatment 960.0 -410.0 -0.15 200.0 -1040.0 -0.8 -0.6689 -0.8221 3021523 ChemDiv3_001746 CN1/C(=C\C=C/2\C(=O)Oc3ccccc3C2=O)/C(C)(C)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P09 compound treatment 5240.0 3870.0 1.37 240.0 -1000.0 -0.77 0.4265 0.2709 3117884 ChemDiv3_001747 Clc1ccc(cc1)c2cn3c(nc4ccccc43)n2CCCNC5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P10 compound treatment 3280.0 1910.0 0.68 240.0 -1000.0 -0.77 -0.0652 -0.0636 3021524 ChemDiv3_001748 Cc1cccn2c(=O)c(/C=N/O)c(nc12)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P11 compound treatment 480.0 -890.0 -0.32 240.0 -1000.0 -0.77 -0.7676 -0.9225 1157071 ChemDiv3_001749 OCCn1c(=N)n(Cc2ccc(Cl)cc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P12 compound treatment 280.0 -1090.0 -0.39 280.0 -963.0 -0.74 -0.796 -0.9543 3117885 ChemDiv3_001750 Cc1ccc(cc1)c2cnc(o2)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P13 compound treatment 880.0 -490.0 -0.17 2920.0 1680.0 1.29 0.7876 0.6062 3021525 ChemDiv3_001751 C=CCn1cc(C=C2C(=O)OC3(CCCC3)OC2=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P14 compound treatment 240.0 -1130.0 -0.4 400.0 -843.0 -0.65 -0.7409 -0.9735 3117886 ChemDiv3_001752 O/C(=C(/C#N)\c1nc2ccccc2[nH]1)/C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P15 compound treatment 280.0 -1090.0 -0.39 200.0 -1040.0 -0.8 -0.8394 -0.9443 1689476 ChemDiv3_001753 Cn1c(CCN)nc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P16 compound treatment 200.0 -1170.0 -0.42 160.0 -1080.0 -0.83 -0.8812 -0.9485 3118033 ChemDiv3_001754 CCN(CC)c1nc2c(C)cccn2c(=O)c1C=C3C(=O)NC(=O)NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P17 compound treatment 200.0 -1170.0 -0.42 160.0 -1080.0 -0.83 -0.8812 -0.9485 1463531 ChemDiv3_001755 CCc1ccc(OCC(=O)Nc2sc3CCCCc3c2C(=O)OC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P18 compound treatment 240.0 -1130.0 -0.4 200.0 -1040.0 -0.8 -0.8495 -0.9489 1302503 ChemDiv3_001756 Cc1nc2c(ccc3nc(NC(=O)c4cccc(Oc5ccccc5)c4)sc32)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P19 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 3118034 ChemDiv3_001757 CCC(=O)N1N=C(CC1c2ccc(cc2)N(C)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P20 compound treatment 240.0 -1130.0 -0.4 280.0 -963.0 -0.74 -0.806 -0.9587 1354491 ChemDiv3_001758 O=C(Nc1c2CSCc2nn1c3ccc(Oc4ccccc4)cc3)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P21 compound treatment 960.0 -410.0 -0.15 320.0 -923.0 -0.71 -0.6037 -0.8349 3118035 ChemDiv3_001759 Cc1cccc(NC2=NC(=O)/C(=C\3/C(=O)N(CC(=O)O)c4ccccc34)/S2)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P22 compound treatment 960.0 -410.0 -0.15 360.0 -883.0 -0.68 -0.582 -0.8398 3021526 ChemDiv3_001760 CCC(C)(C)n1c(=O)[nH]c2CCCc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P23 mock treatment 360.0 -1010.0 -0.36 1080.0 -163.0 -0.12 -0.3417 -0.9004 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2005 P24 mock treatment 400.0 -970.0 -0.34 200.0 -1040.0 -0.8 -0.8093 -0.9289 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A01 compound treatment 3240.0 2360.0 0.84 280.0 -348.0 -0.27 0.4036 0.4591 1658490 ChemDiv3_001761 Cc1cc(=O)[nH]c(Nc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A02 compound treatment 2960.0 2080.0 0.74 200.0 -428.0 -0.33 0.2899 0.3588 1465213 ChemDiv3_001762 CCOc1ccc2nc(Nc3nc(O)cc(O)n3)nc(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A03 compound treatment 360.0 -519.0 -0.18 360.0 -268.0 -0.21 -0.2754 -0.9985 3118036 ChemDiv3_001763 COc1cccc2s/c(=N/C(=O)Cc3cccc4ccccc34)/n(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A04 compound treatment 680.0 -199.0 -0.07 600.0 -27.6 -0.02 -0.0648 -0.8806 3118037 ChemDiv3_001764 NC1=NC(=O)CC(S1)C(=O)Nc2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A05 compound treatment 280.0 -599.0 -0.21 360.0 -268.0 -0.21 -0.2955 -0.9999 1135271 ChemDiv3_001765 Oc1cc(Cc2nc3ccccc3s2)c(O)cc1Cc4nc5ccccc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A06 compound treatment 240.0 -639.0 -0.23 200.0 -428.0 -0.33 -0.3923 -0.9836 1132838 ChemDiv3_001766 O=C(CSC#N)n1c2ccccc2c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A07 compound treatment 320.0 -559.0 -0.2 320.0 -308.0 -0.24 -0.3071 -0.9962 3118038 ChemDiv3_001767 O=S(=O)(/N=C(/NC(=S)OC1CCCCC1)\c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A08 compound treatment 160.0 -719.0 -0.25 3680.0 3050.0 2.34 1.4767 0.6265 3021527 ChemDiv3_001768 CC(C)COc1ccc(cc1)C(=S)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A09 compound treatment 320.0 -559.0 -0.2 400.0 -228.0 -0.17 -0.2637 -0.998 3021563 ChemDiv3_001769 COc1ccc(/C=C/C(=O)O)cc1S(=O)(=O)N(C)CCO 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A10 compound treatment 280.0 -599.0 -0.21 1880.0 1250.0 0.96 0.5297 0.5379 3021564 ChemDiv3_001770 Cc1cc(C(=O)O)c(=O)[nH]c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A11 compound treatment 200.0 -679.0 -0.24 240.0 -388.0 -0.3 -0.3807 -0.9945 1689022 ChemDiv3_001771 Cc1ccc2n(CC(O)CNCc3ccco3)c(c(c4ccccc4)c2c1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A12 compound treatment 320.0 -559.0 -0.2 720.0 92.4 0.07 -0.09 -0.4275 3118039 ChemDiv3_001772 NNC(=O)CN1C(c2ccccc2)c3cc(Cl)ccc3N=C1c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A13 compound treatment 280.0 -599.0 -0.21 560.0 -67.6 -0.05 -0.1869 -0.8547 1296978 ChemDiv3_001773 C=CCNC(=O)c1cc2ccccc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A14 compound treatment 320.0 -559.0 -0.2 240.0 -388.0 -0.3 -0.3506 -0.9805 3021565 ChemDiv3_001774 CCOC(=O)/C(=C/1\Nc2ccccc2C1=O)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A15 compound treatment 240.0 -639.0 -0.23 280.0 -348.0 -0.27 -0.3489 -0.9967 1549910 ChemDiv3_001775 CC(=O)Nc1ccc(NC(=O)C2(CCCC2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A16 compound treatment 240.0 -639.0 -0.23 200.0 -428.0 -0.33 -0.3923 -0.9836 3021566 ChemDiv3_001776 Clc1ccc(cc1)N2C(=O)C3CC=CCC3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A17 compound treatment 240.0 -639.0 -0.23 2040.0 1410.0 1.08 0.6065 0.5475 3118040 ChemDiv3_001777 NC(=O)/C(=C/c1ccc2OCOc2c1)/NC(=O)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A18 compound treatment 160.0 -719.0 -0.25 280.0 -348.0 -0.27 -0.369 -0.9997 3021567 ChemDiv3_001778 O=C1C=C(N2CCOCC2)C(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A19 compound treatment 320.0 -559.0 -0.2 760.0 132.0 0.1 -0.0683 -0.3065 1179633 ChemDiv3_001779 COc1cc(CN2CCN(CC2)C(=O)COc3ccccc3)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A20 compound treatment 440.0 -439.0 -0.16 320.0 -308.0 -0.24 -0.277 -0.9795 3118041 ChemDiv3_001780 CC(C)(C)c1n[nH]c2OC(=C(C#N)C(c12)c3ccc(OC(=O)c4ccccc4Cl)cc3)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A21 compound treatment 320.0 -559.0 -0.2 200.0 -428.0 -0.33 -0.3723 -0.9708 3021568 ChemDiv3_001781 Cc1ccc(cc1)C2C3=C(NC4=C2C(=O)CC(C)(C)C4)c5ccccc5C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A22 compound treatment 200.0 -679.0 -0.24 200.0 -428.0 -0.33 -0.4024 -0.9884 3118042 ChemDiv3_001782 COc1cccc(c1)N2C(=O)/C(=C/c3ccsc3)/C(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A23 mock treatment 560.0 -319.0 -0.11 320.0 -308.0 -0.24 -0.2469 -0.9431 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 A24 mock treatment 400.0 -479.0 -0.17 320.0 -308.0 -0.24 -0.2871 -0.9869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B01 compound treatment 1200.0 321.0 0.11 240.0 -388.0 -0.3 -0.1298 -0.4074 1408187 ChemDiv3_001783 Cc1ccc(NC(=O)CSc2nnc(s2)N3C(=O)c4ccccc4C3=O)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B02 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 1465544 ChemDiv3_001784 S=C(Nc1ccccc1)N2CCC(=N2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B03 compound treatment 240.0 -639.0 -0.23 280.0 -348.0 -0.27 -0.3489 -0.9967 3118043 ChemDiv3_001785 Cc1cc(C)c(N2C(=O)NC(=O)/C(=C\Nc3cccc(O)c3)/C2=O)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B04 compound treatment 280.0 -599.0 -0.21 400.0 -228.0 -0.17 -0.2737 -0.9953 1229641 ChemDiv3_001786 CCOC(=O)C(Cc1ccccc1)C(=O)Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B05 compound treatment 1080.0 201.0 0.07 200.0 -428.0 -0.33 -0.1816 -0.5407 3021569 ChemDiv3_001787 CCN1C(=O)C(=Cc2ccc(o2)c3ccccc3F)C(=O)N(CC)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B06 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 1193124 ChemDiv3_001788 Cc1oc2ccc(O)cc2c1C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B07 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 3021570 ChemDiv3_001789 CC(C)(C)N(CCO)C(=O)CN1C(=O)/C(=C/c2cccc(Br)c2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B08 compound treatment 360.0 -519.0 -0.18 360.0 -268.0 -0.21 -0.2754 -0.9985 1231195 ChemDiv3_001790 COC(=O)COc1cccc2c1ccc3c4CCCCc4c(=O)oc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B09 compound treatment 320.0 -559.0 -0.2 240.0 -388.0 -0.3 -0.3506 -0.9805 3118044 ChemDiv3_001791 CCCCn1c-2c(CCc3nonc32)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B10 compound treatment 200.0 -679.0 -0.24 280.0 -348.0 -0.27 -0.359 -0.9987 1442608 ChemDiv3_001792 COc1ccc(cc1OC)C2CC(=O)c3cnc(N)nc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B11 compound treatment 320.0 -559.0 -0.2 240.0 -388.0 -0.3 -0.3506 -0.9805 1122476 ChemDiv3_001793 Clc1ccc(cc1)c2nc(N3CCCCC3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B12 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 3118045 ChemDiv3_001794 CN1C(=O)/C(=C/2\SC(=S)N(C3CCS(=O)(=O)C3)C2=O)/c4cc(Br)ccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B13 compound treatment 1520.0 641.0 0.23 280.0 -348.0 -0.27 -0.0278 -0.0794 1382733 ChemDiv3_001795 Oc1ccc(I)nc1CCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B14 compound treatment 560.0 -319.0 -0.11 240.0 -388.0 -0.3 -0.2904 -0.9122 1453546 ChemDiv3_001796 CN(C)c1ccc(cc1)N2C(=O)C3CC(=C(C)CC3C2=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B15 compound treatment 360.0 -519.0 -0.18 240.0 -388.0 -0.3 -0.3405 -0.9733 1593282 ChemDiv3_001797 COc1ccc2N(C(=O)Nc3ccc(Cl)cc3)C(C)(C)CC(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B16 compound treatment 440.0 -439.0 -0.16 1680.0 1050.0 0.81 0.4613 0.5606 3021571 ChemDiv3_001798 CCCCC1(C)OC(=O)C(=Cc2ccc(SC)cc2)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B17 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 1026532 ChemDiv3_001799 Cc1ccc(cc1)C(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B18 compound treatment 360.0 -519.0 -0.18 280.0 -348.0 -0.27 -0.3188 -0.9835 3021572 ChemDiv3_001800 O=C1C=CC2(CC3(CCCCC3)N=C2SCc4ccccc4)C=C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B19 compound treatment 4440.0 3560.0 1.26 14360.0 13700.0 10.54 8.3481 0.7862 1698847 ChemDiv3_001801 O=c1n(Cc2ccccc2)c(=S)[nH]c3sc4CCCCCc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B20 compound treatment 600.0 -279.0 -0.1 400.0 -228.0 -0.17 -0.1935 -0.9637 1202827 ChemDiv3_001802 Cc1nc2ccccc2c(=O)n1NCc3ccccc3Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B21 compound treatment 520.0 -359.0 -0.13 1560.0 932.0 0.72 0.4162 0.5724 1391827 ChemDiv3_001803 CNC(=O)c1c(c2ccccc2)c3cc(OC)ccc3n1CCN(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B22 compound treatment 2920.0 2040.0 0.72 280.0 -348.0 -0.27 0.3233 0.419 3118046 ChemDiv3_001804 CCOC(=O)c1c(C)oc2ccc(OCC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B23 mock treatment 320.0 -559.0 -0.2 320.0 -308.0 -0.24 -0.3071 -0.9962 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 B24 mock treatment 520.0 -359.0 -0.13 280.0 -348.0 -0.27 -0.2787 -0.9426 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C01 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 3118047 ChemDiv3_001805 COc1ccc(cc1OC)C(CC(=O)c2ccco2)Sc3cccc4cccnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C02 compound treatment 280.0 -599.0 -0.21 200.0 -428.0 -0.33 -0.3823 -0.9778 1315783 ChemDiv3_001806 Cn1ccnc1SCC(=O)N2c3ccccc3C(C)(CC2(C)C)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C03 compound treatment 240.0 -639.0 -0.23 2000.0 1370.0 1.05 0.5848 0.5426 3118179 ChemDiv3_001807 COc1cccc2s/c(=N/C(=O)COc3ccc(Cl)cc3Cl)/n(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C04 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 3021573 ChemDiv3_001808 CCOC(=O)CCSc1nc(C)c2ccccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C05 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 1356071 ChemDiv3_001809 CP(=O)(O)c1nccn1c2ccc(Cl)nn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C06 compound treatment 280.0 -599.0 -0.21 200.0 -428.0 -0.33 -0.3823 -0.9778 3118180 ChemDiv3_001810 COCc1cc(=O)nc(Sc2c(O)nc3cc(Cl)ccc3c2c4ccccc4)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C07 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 3021574 ChemDiv3_001811 Cc1n(C)c2ccccc2[n+]1CC(=O)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C08 compound treatment 1640.0 761.0 0.27 160.0 -468.0 -0.36 -0.0629 -0.14 1515483 ChemDiv3_001812 S=C(N1CCCCC1)c2cccc(OCc3ccccc3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C09 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 1633788 ChemDiv3_001813 COc1ccc(cc1OC)C2CC(=O)n3nc(nc3S2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C10 compound treatment 200.0 -679.0 -0.24 400.0 -228.0 -0.17 -0.2938 -0.9876 3118181 ChemDiv3_001814 C/C(=C\C=C\c1ccccc1)/C(=O)c2c(C)cc(C)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C11 compound treatment 240.0 -639.0 -0.23 320.0 -308.0 -0.24 -0.3272 -0.9998 1558595 ChemDiv3_001815 Cc1ccc2n(CC(O)Cn3c(C)cc(C)nc3=O)c(c(c4ccccc4)c2c1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C12 compound treatment 440.0 -439.0 -0.16 240.0 -388.0 -0.3 -0.3205 -0.9543 3021616 ChemDiv3_001816 COC(=O)CN1C(c2ccccc2)c3cc(Cl)ccc3N=C1c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C13 compound treatment 240.0 -639.0 -0.23 200.0 -428.0 -0.33 -0.3923 -0.9836 1164199 ChemDiv3_001817 COc1ccc(CNc2ncn[nH]2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C14 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 1183780 ChemDiv3_001818 Cc1ccc(cc1C)C(=O)c2cc(F)c(cc2Cl)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C15 compound treatment 200.0 -679.0 -0.24 320.0 -308.0 -0.24 -0.3372 -1.0 1590710 ChemDiv3_001819 Clc1ccccc1C(=O)NCCc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C16 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 3118182 ChemDiv3_001820 COc1ccccc1N2C(=O)NC(=O)/C(=C\C=C\c3ccco3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C17 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 3021617 ChemDiv3_001821 OC(=O)/C(=C/c1ccc2OCOc2c1)/NC(=O)c3ccccc3Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C18 compound treatment 200.0 -679.0 -0.24 280.0 -348.0 -0.27 -0.359 -0.9987 3118183 ChemDiv3_001822 Ic1ccc(Nc2nc(Nc3ccccc3)nc(n2)N4CCOCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C19 compound treatment 320.0 -559.0 -0.2 440.0 -188.0 -0.14 -0.242 -0.9877 1705372 ChemDiv3_001823 CCn1c2ccccc2c3cc(CN4CCN(Cc5cccc(C)c5)CC4)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C20 compound treatment 320.0 -559.0 -0.2 240.0 -388.0 -0.3 -0.3506 -0.9805 1427498 ChemDiv3_001824 Clc1ccc(CN2CCNCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C21 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 1410682 ChemDiv3_001825 CC1CC(Nc2ccccc2)c3ccccc3N1S(=O)(=O)c4ccc(Br)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C22 compound treatment 400.0 -479.0 -0.17 240.0 -388.0 -0.3 -0.3305 -0.9646 3021618 ChemDiv3_001826 COc1cccc(/C=C/2\C(=O)NC(=O)N(C)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C23 mock treatment 320.0 -559.0 -0.2 3680.0 3050.0 2.34 1.5169 0.645 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 C24 mock treatment 240.0 -639.0 -0.23 440.0 -188.0 -0.14 -0.2621 -0.9761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D01 compound treatment 720.0 -159.0 -0.06 240.0 -388.0 -0.3 -0.2502 -0.8263 3021619 ChemDiv3_001827 CCOC(=O)c1nc2ccccc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D02 compound treatment 360.0 -519.0 -0.18 280.0 -348.0 -0.27 -0.3188 -0.9835 1548078 ChemDiv3_001828 O=C(c1c(oc2C(=O)c3ccccc3C(=O)c12)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D03 compound treatment 360.0 -519.0 -0.18 280.0 -348.0 -0.27 -0.3188 -0.9835 3118184 ChemDiv3_001829 Oc1ccc(/C=C/2\C(=O)NC(=O)N(CC=C)C2=O)cc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D04 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 1159195 ChemDiv3_001830 O=C(CCC1CCCCC1)Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D05 compound treatment 600.0 -279.0 -0.1 120.0 -508.0 -0.39 -0.3455 -0.8593 3021621 ChemDiv3_001831 Clc1ccc(cc1)c2ccc(=S)n(n2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D06 compound treatment 240.0 -639.0 -0.23 400.0 -228.0 -0.17 -0.2838 -0.9917 1463047 ChemDiv3_001832 Cc1ccc(OC(=O)c2cc(ccc2C)S(=O)(=O)N3CCCC3)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D07 compound treatment 320.0 -559.0 -0.2 360.0 -268.0 -0.21 -0.2854 -0.9998 3021622 ChemDiv3_001833 CCOC(=O)C1C(NC(=S)NC1(O)C(F)(F)F)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D08 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 1242363 ChemDiv3_001834 CCOC(=O)C(C)Oc1cc2oc(=O)c3CCCCc3c2cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D09 compound treatment 280.0 -599.0 -0.21 200.0 -428.0 -0.33 -0.3823 -0.9778 3021623 ChemDiv3_001835 CCOC(=O)c1c(C)n(OCc2ccccc2)c3ccc4nonc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D10 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 1388539 ChemDiv3_001836 COc1ccc(cc1)C2CC(=O)C3=C(C2)Nc4ccccc4N(C3c5ccccc5)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D11 compound treatment 360.0 -519.0 -0.18 240.0 -388.0 -0.3 -0.3405 -0.9733 3021624 ChemDiv3_001837 CCOc1nc(nc2ccccc12)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D12 compound treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 3118185 ChemDiv3_001838 Cc1cccn2c(=O)c(/C=C/3\SC(=S)NC3=O)c(NCC=C)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D13 compound treatment 360.0 -519.0 -0.18 240.0 -388.0 -0.3 -0.3405 -0.9733 3021625 ChemDiv3_001839 CC1(C)CC(=O)/C(=C/c2ccco2)/CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D14 compound treatment 440.0 -439.0 -0.16 240.0 -388.0 -0.3 -0.3205 -0.9543 1476666 ChemDiv3_001840 Brc1ccccc1C(=O)Nc2cccc(c2)c3nc4ccccc4c(=O)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D15 compound treatment 200.0 -679.0 -0.24 320.0 -308.0 -0.24 -0.3372 -1.0 3118186 ChemDiv3_001841 CCOc1ccc(Nc2nc(Nc3ccc(OCC)cc3)nc(SC4=NCCS4)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D16 compound treatment 1200.0 321.0 0.11 600.0 -27.6 -0.02 0.0656 0.566 3021626 ChemDiv3_001842 O=C1OC(OC(=O)C1=Cc2cccc(OCc3ccccc3)c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D17 compound treatment 320.0 -559.0 -0.2 400.0 -228.0 -0.17 -0.2637 -0.998 1107247 ChemDiv3_001843 CC1CCCC(C)N1C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D18 compound treatment 280.0 -599.0 -0.21 160.0 -468.0 -0.36 -0.404 -0.9686 3021627 ChemDiv3_001844 COc1cc2CC(C)(C)N=C(Nc3nc(cs3)c4ccccc4)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D19 compound treatment 440.0 -439.0 -0.16 280.0 -348.0 -0.27 -0.2987 -0.9671 3118187 ChemDiv3_001845 CCCCc1nc2ccccc2c(=O)n1c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D20 compound treatment 3080.0 2200.0 0.78 280.0 -348.0 -0.27 0.3635 0.4405 1507247 ChemDiv3_001846 Clc1c(sc2ccccc12)C(=O)NCCC3=CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D21 compound treatment 360.0 -519.0 -0.18 280.0 -348.0 -0.27 -0.3188 -0.9835 3021628 ChemDiv3_001847 COC(=O)Cn1c2CCCCc2c3cc(C)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D22 compound treatment 240.0 -639.0 -0.23 280.0 -348.0 -0.27 -0.3489 -0.9967 1488517 ChemDiv3_001848 COC(=O)c1c(C)oc2ccc(OCC#N)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D23 mock treatment 160.0 -719.0 -0.25 360.0 -268.0 -0.21 -0.3256 -0.9943 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 D24 mock treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E01 compound treatment 200.0 -679.0 -0.24 1240.0 612.0 0.47 0.1622 0.3071 1575197 ChemDiv3_001849 O=C(Nc1ccc(cc1)c2nc3ccccc3o2)c4ccc(cc4)C(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E02 compound treatment 400.0 -479.0 -0.17 2800.0 2170.0 1.67 1.0592 0.6318 1324387 ChemDiv3_001850 Cc1ccc(cc1)C(=O)N2C(=O)C(Oc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E03 compound treatment 240.0 -639.0 -0.23 320.0 -308.0 -0.24 -0.3272 -0.9998 3118188 ChemDiv3_001851 COc1cccc2s/c(=N/C(=S)NC(=O)c3ccc(C)cc3)/n(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E04 compound treatment 1240.0 361.0 0.13 360.0 -268.0 -0.21 -0.0546 -0.2257 3021629 ChemDiv3_001852 CCOC(=O)CSc1nc(C)c2cc(C)c(C)cc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E05 compound treatment 560.0 -319.0 -0.11 240.0 -388.0 -0.3 -0.2904 -0.9122 1633868 ChemDiv3_001853 O=C(Nc1ccccc1c2nc3ccccc3s2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E06 compound treatment 400.0 -479.0 -0.17 240.0 -388.0 -0.3 -0.3305 -0.9646 1479197 ChemDiv3_001854 Oc1nc2cc(Cl)ccc2c(c1SC3=NCCS3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E07 compound treatment 800.0 -78.8 -0.03 1000.0 372.0 0.29 0.1824 0.635 1403729 ChemDiv3_001855 COc1ccc(cc1)S(=O)(=O)N2Cc3ccccc3CC2C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E08 compound treatment 280.0 -599.0 -0.21 1160.0 532.0 0.41 0.1388 0.3014 1609478 ChemDiv3_001856 COc1ccc(cc1OC)C(=S)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E09 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 3118189 ChemDiv3_001857 Cc1ccc(c(C)c1)n2c(C)cc(=O)cc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E10 compound treatment 240.0 -639.0 -0.23 2600.0 1970.0 1.51 0.9105 0.5947 1627173 ChemDiv3_001858 OC(=O)CCCC(=O)Nc1cccc2cccnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E11 compound treatment 400.0 -479.0 -0.17 840.0 212.0 0.16 -0.0048 -0.0203 3021676 ChemDiv3_001859 Cc1cc(O)nc(SCC(=O)c2cccs2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E12 compound treatment 360.0 -519.0 -0.18 920.0 292.0 0.22 0.0286 0.0986 3118190 ChemDiv3_001860 Cc1ccc2[nH]c(=O)c(c(c3ccccc3)c2c1)[n+]4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E13 compound treatment 14600.0 13700.0 4.87 2760.0 2130.0 1.64 4.5995 0.8956 3118191 ChemDiv3_001861 C/C(=C/1\SC(=S)NC1=O)/C\C(=C/2\SC(=S)NC2=O)\C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E14 compound treatment 880.0 1.25 0.0 960.0 332.0 0.26 0.1808 0.7083 1418462 ChemDiv3_001862 O=C(Oc1ccc2ccc(=O)oc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E15 compound treatment 960.0 81.3 0.03 880.0 252.0 0.19 0.1574 0.8034 1307975 ChemDiv3_001863 CCOC(=O)c1ccc(Nc2cc(C)nc(n2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E16 compound treatment 440.0 -439.0 -0.16 760.0 132.0 0.1 -0.0382 -0.2054 3021677 ChemDiv3_001864 COc1cccc(/C=C/2\C(=O)NC(=O)N(C2=O)c3cccc(OC)c3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E17 compound treatment 1000.0 121.0 0.04 3000.0 2370.0 1.82 1.3183 0.7236 3118326 ChemDiv3_001865 Clc1ccccc1C(=O)N/C(=C\c2ccc3OCOc3c2)/C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E18 compound treatment 4640.0 3760.0 1.33 680.0 52.4 0.04 0.9719 0.7281 1535987 ChemDiv3_001866 CC1CCN(Cn2c(=S)n(CN3CCC(C)CC3)c4ccccc24)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E19 compound treatment 5840.0 4960.0 1.76 1360.0 732.0 0.56 1.6421 0.8888 1155262 ChemDiv3_001867 COc1ccccc1CN2CCN(Cc3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E20 compound treatment 680.0 -199.0 -0.07 920.0 292.0 0.22 0.1089 0.4627 1640740 ChemDiv3_001868 CCCC1=C(C(C(=C(N1)SC)C#N)c2ccccc2Cl)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E21 compound treatment 2640.0 1760.0 0.62 320.0 -308.0 -0.24 0.2748 0.4115 1272136 ChemDiv3_001869 CC1=CC(C)(C)N(C(=O)CN2C(=O)c3ccccc3C2=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E22 compound treatment 1520.0 641.0 0.23 360.0 -268.0 -0.21 0.0156 0.0509 3118327 ChemDiv3_001870 CN1C(=O)NC(=O)/C(=C\c2ccc(O)cc2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E23 mock treatment 560.0 -319.0 -0.11 5240.0 4610.0 3.54 2.4239 0.6842 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 E24 mock treatment 320.0 -559.0 -0.2 880.0 252.0 0.19 -0.0031 -0.0113 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F01 compound treatment 1480.0 601.0 0.21 2240.0 1610.0 1.24 1.0261 0.8169 1132984 ChemDiv3_001871 COc1ccc(NC(=S)NCC2CCCO2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F02 compound treatment 1640.0 761.0 0.27 800.0 172.0 0.13 0.2846 0.9462 3118328 ChemDiv3_001872 O=C1c2oc(c(C#N)c2C(=O)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F03 compound treatment 1640.0 761.0 0.27 1760.0 1130.0 0.87 0.8057 0.885 3021678 ChemDiv3_001873 CCN1C(=O)/C(=C/c2ccc[nH]2)/C(=O)NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F04 compound treatment 2480.0 1600.0 0.57 2480.0 1850.0 1.42 1.4073 0.919 3118329 ChemDiv3_001874 COc1ccc(cc1OC)C2CC(=NN2)c3cc(Cl)ccc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F05 compound treatment 3840.0 2960.0 1.05 1560.0 932.0 0.72 1.249 0.9825 1704441 ChemDiv3_001875 CCSc1ccc(NC(=O)CC2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F06 compound treatment 680.0 -199.0 -0.07 1000.0 372.0 0.29 0.1523 0.5172 1175553 ChemDiv3_001876 Cc1ccc(cc1S(=O)(=O)N2CCCCC2)C(=O)NCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F07 compound treatment 2280.0 1400.0 0.5 6520.0 5890.0 4.52 3.5502 0.7801 3118330 ChemDiv3_001877 CCCCN(C)Cc1c(O)ccc2c(=O)c(c3ccccc3OC)c(oc12)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F08 compound treatment 1960.0 1080.0 0.38 600.0 -27.6 -0.02 0.2562 0.667 1437891 ChemDiv3_001878 Cc1cn2c(n1)n(Cc3ccc(C)cc3)c4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F09 compound treatment 1600.0 721.0 0.26 2280.0 1650.0 1.27 1.0779 0.8329 3118331 ChemDiv3_001879 [O-][n+]1c(c2ccccc2)c(=O)n(OCc3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F10 compound treatment 2760.0 1880.0 0.67 2600.0 1970.0 1.51 1.5426 0.9322 1724763 ChemDiv3_001880 CCNC(=S)N1C(C2=C(CC(C)(C)CC2=O)Nc3ccccc13)c4ccc(cc4)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F11 compound treatment 2040.0 1160.0 0.41 1920.0 1290.0 0.99 0.9929 0.9242 1445265 ChemDiv3_001881 C1CCN(C1)c2nc3ccccc3n4cnnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F12 compound treatment 6960.0 6080.0 2.16 680.0 52.4 0.04 1.5539 0.7202 1581689 ChemDiv3_001882 Cc1ccc(cc1)c2nnc(Sc3nc4ccccc4o3)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F13 compound treatment 4320.0 3440.0 1.22 880.0 252.0 0.19 1.0002 0.8092 1785410 ChemDiv3_001883 CC(C)N1CC2(N3CC4(C)CN2CC(C)(C3)C4=O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F14 compound treatment 4400.0 3520.0 1.25 1440.0 812.0 0.62 1.3243 0.9485 1701789 ChemDiv3_001884 CS(=O)(=O)N(Cc1ccc(Cl)cc1)c2ccc(cc2)C(=O)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F15 compound treatment 6600.0 5720.0 2.03 2560.0 1930.0 1.48 2.4842 0.9881 3118332 ChemDiv3_001885 NC(=N)/N=c/1\[nH]c(=O)c2ccccc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F16 compound treatment 2360.0 1480.0 0.53 1240.0 612.0 0.47 0.704 0.9985 3118333 ChemDiv3_001886 CC(C)(C)C1(C)OC(=O)C(=Cc2ccccc2Cl)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F17 compound treatment 4160.0 3280.0 1.16 1120.0 492.0 0.38 1.0904 0.8909 1472344 ChemDiv3_001887 O=C(OCCN1C(=O)c2ccccc2C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F18 compound treatment 2760.0 1880.0 0.67 1040.0 412.0 0.32 0.6958 0.9419 1671379 ChemDiv3_001888 COc1ccc(OC)c2C(=NC(C)(C)Cc12)SC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F19 compound treatment 1200.0 321.0 0.11 280.0 -348.0 -0.27 -0.1081 -0.3726 3021679 ChemDiv3_001889 CCOC(=O)c1c(C)c2/C(=N/O)/CCCc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F20 compound treatment 840.0 -38.8 -0.01 2360.0 1730.0 1.33 0.9307 0.6998 1637847 ChemDiv3_001890 CC(=O)Oc1ccc2cc(c3nc4ccccc4n3C)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F21 compound treatment 1600.0 721.0 0.26 4080.0 3450.0 2.65 2.0551 0.7718 3021680 ChemDiv3_001891 N#CCc1nnc2CCCCCn12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F22 compound treatment 1680.0 801.0 0.28 3440.0 2810.0 2.16 1.7277 0.7933 1388136 ChemDiv3_001892 COC(=O)c1c(C)oc2ccc(OCc3ccccc3C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F23 mock treatment 1680.0 801.0 0.28 5280.0 4650.0 3.57 2.7266 0.761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 F24 mock treatment 480.0 -399.0 -0.14 760.0 132.0 0.1 -0.0281 -0.1616 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G01 compound treatment 600.0 -279.0 -0.1 2480.0 1850.0 1.42 0.9357 0.6564 3021681 ChemDiv3_001893 Cn1/c(=N/C(=O)c2cccc(c2)C(F)(F)F)/sc3c1ccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G02 compound treatment 600.0 -279.0 -0.1 800.0 172.0 0.13 0.0237 0.1433 1418652 ChemDiv3_001894 COc1ccc(OCC(=O)N2c3ccccc3Sc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G03 compound treatment 2280.0 1400.0 0.5 480.0 -148.0 -0.11 0.2714 0.5323 1381191 ChemDiv3_001895 Nc1c(C(=O)c2ccccc2)n3ccccc3c1c4nc(cs4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G04 compound treatment 640.0 -239.0 -0.08 1080.0 452.0 0.35 0.1857 0.5195 1522414 ChemDiv3_001896 Cc1ccc(SCc2cc(O)nc(Nc3nc4ccccc4o3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G05 compound treatment 2440.0 1560.0 0.55 440.0 -188.0 -0.14 0.2898 0.5064 1650593 ChemDiv3_001897 CCCCC1CCC(CC1)C(=O)ON2C(=O)c3cccc4cccc(C2=O)c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G06 compound treatment 480.0 -399.0 -0.14 2400.0 1770.0 1.36 0.8621 0.6302 1442367 ChemDiv3_001898 S=c1[nH]nc(c2cccnc2)n1C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G07 compound treatment 680.0 -199.0 -0.07 440.0 -188.0 -0.14 -0.1517 -0.946 1200273 ChemDiv3_001899 CC1(C)CC(=O)C2=C(C1)Nc3[nH]c(=S)[nH]c(=O)c3C2c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G08 compound treatment 440.0 -439.0 -0.16 1000.0 372.0 0.29 0.0921 0.283 3020977 ChemDiv3_001900 Clc1ccc(cc1)C(=S)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G09 compound treatment 2000.0 1120.0 0.4 440.0 -188.0 -0.14 0.1794 0.4241 3020978 ChemDiv3_001901 CCCCn1c(nc(=S)c2CCCCc21)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G10 compound treatment 440.0 -439.0 -0.16 1320.0 692.0 0.53 0.2658 0.4799 1183988 ChemDiv3_001902 CC(C)c1cc(C(C)C)c(c(c1)C(C)C)S(=O)(=O)NCCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G11 compound treatment 920.0 41.3 0.01 560.0 -67.6 -0.05 -0.0263 -0.4886 3020979 ChemDiv3_001903 Nc1cc(O)nc(SCC(=O)c2cccs2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G12 compound treatment 560.0 -319.0 -0.11 800.0 172.0 0.13 0.0136 0.0784 1644588 ChemDiv3_001904 CCCc1c(O)nc(SCc2ccccc2)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G13 compound treatment 960.0 81.3 0.03 600.0 -27.6 -0.02 0.0054 0.1511 3118334 ChemDiv3_001905 C/N=C(\c1ccc(C)cc1)/n2c(=S)nc(c3ccc(C)cc3)n(C)c2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G14 compound treatment 720.0 -159.0 -0.06 360.0 -268.0 -0.21 -0.1851 -0.8689 3020980 ChemDiv3_001906 CCC(=O)NC(Nc1cccnc1Cl)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G15 compound treatment 1320.0 441.0 0.16 440.0 -188.0 -0.14 0.0089 0.0416 1404360 ChemDiv3_001907 Cc1sc(NC(=O)C(Cc2ccccc2)Cc3ccccc3)c(C#N)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G16 compound treatment 400.0 -479.0 -0.17 720.0 92.4 0.07 -0.0699 -0.3799 1312332 ChemDiv3_001908 Cc1ccc(NC(=O)c2cc3ccccc3oc2=N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G17 compound treatment 920.0 41.3 0.01 1840.0 1210.0 0.93 0.6685 0.7181 3118335 ChemDiv3_001909 COc1ccccc1C(=O)N/C(=C\c2ccccc2)/C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G18 compound treatment 480.0 -399.0 -0.14 1120.0 492.0 0.38 0.1673 0.4145 1265569 ChemDiv3_001910 CC1(C)C(C(=O)N2CCN(CC2)c3ccc(Cl)cc3)C1(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G19 compound treatment 520.0 -359.0 -0.13 560.0 -67.6 -0.05 -0.1267 -0.9217 1567377 ChemDiv3_001911 COc1ccc(CNC2C3CC4CC(C3)CC2C4)c(OC)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G20 compound treatment 480.0 -399.0 -0.14 1520.0 892.0 0.69 0.3844 0.5495 1616500 ChemDiv3_001912 CC(C)OC(=O)CSC1=C(C#N)C(CC(=O)N1)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G21 compound treatment 840.0 -38.8 -0.01 360.0 -268.0 -0.21 -0.155 -0.7527 1342244 ChemDiv3_001913 O=C(CN1C(=O)c2ccccc2C1=O)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G22 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 3020981 ChemDiv3_001914 Cc1ccc(cc1)c2nc(no2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G23 mock treatment 1160.0 281.0 0.1 1240.0 612.0 0.47 0.403 0.8385 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 G24 mock treatment 720.0 -159.0 -0.06 440.0 -188.0 -0.14 -0.1417 -0.9161 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H01 compound treatment 560.0 -319.0 -0.11 2360.0 1730.0 1.33 0.8605 0.6447 1224823 ChemDiv3_001915 CC(Oc1ccc(Cl)c(C)c1)C(=O)Nc2sc3CCCCCCc3c2C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H02 compound treatment 1000.0 121.0 0.04 560.0 -67.6 -0.05 -0.0063 -0.0931 1608454 ChemDiv3_001916 O=C1OC(Oc2cccc3cccnc23)(c4ccccc14)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H03 compound treatment 2680.0 1800.0 0.64 520.0 -108.0 -0.08 0.3934 0.6106 3020982 ChemDiv3_001917 CCc1n[nH]c2OC(=C(C#N)C(c12)c3cccc(OC(=O)N4CCOCC4)c3)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H04 compound treatment 1240.0 361.0 0.13 440.0 -188.0 -0.14 -0.0112 -0.0582 1208340 ChemDiv3_001918 N(c1ccc2ccccc2c1)c3ncnc4[nH]ncc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H05 compound treatment 720.0 -159.0 -0.06 520.0 -108.0 -0.08 -0.0982 -0.9826 3118467 ChemDiv3_001919 Clc1ccccc1OCCNC(=O)CC2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H06 compound treatment 1000.0 121.0 0.04 560.0 -67.6 -0.05 -0.0063 -0.0931 1533326 ChemDiv3_001920 OC(=O)c1cccc(NC(=O)c2cccc(c2)S(=O)(=O)N3CCCCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H07 compound treatment 440.0 -439.0 -0.16 520.0 -108.0 -0.08 -0.1685 -0.9561 3118468 ChemDiv3_001921 COC(=O)CN1C(=O)/C(=C\c2ccc(O)cc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H08 compound treatment 1000.0 121.0 0.04 920.0 292.0 0.22 0.1892 0.8275 3118469 ChemDiv3_001922 CC(C)CCOc1ccc(/C=N/c2nc3ccccc3n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H09 compound treatment 3400.0 2520.0 0.89 680.0 52.4 0.04 0.6609 0.7382 1416640 ChemDiv3_001923 CCOn1c(=O)c(=O)n(OC)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H10 compound treatment 600.0 -279.0 -0.1 560.0 -67.6 -0.05 -0.1066 -0.9547 3020983 ChemDiv3_001924 O=C1C(=CNCCN2CCOCC2)C(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H11 compound treatment 1760.0 881.0 0.31 520.0 -108.0 -0.08 0.1627 0.503 3118470 ChemDiv3_001925 C(Nc1ccccc1)C2OCc3ccccc3CO2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H12 compound treatment 1720.0 841.0 0.3 1000.0 372.0 0.29 0.4132 0.9998 1432963 ChemDiv3_001926 COc1ccc(cc1)c2nnc(Nc3ccc(Cl)cc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H13 compound treatment 920.0 41.3 0.01 1920.0 1290.0 0.99 0.7119 0.7175 3020985 ChemDiv3_001927 Oc1ccc(/C=N/CC2OCCc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H14 compound treatment 480.0 -399.0 -0.14 440.0 -188.0 -0.14 -0.2019 -1.0 1651658 ChemDiv3_001928 CS(=O)(=O)N(CC(=O)NCc1ccco1)c2ccccc2Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H15 compound treatment 1560.0 681.0 0.24 640.0 12.4 0.01 0.1776 0.7344 3020986 ChemDiv3_001929 CC(=O)/N=C(/Nc1cc(C)cc(C)c1)\Nc2nc(C)cc(C)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H16 compound treatment 680.0 -199.0 -0.07 1760.0 1130.0 0.87 0.5649 0.6476 3118471 ChemDiv3_001930 CCOc1ccc(C=C2C(=O)OC(OC2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H17 compound treatment 560.0 -319.0 -0.11 2280.0 1650.0 1.27 0.8171 0.6415 1104705 ChemDiv3_001931 OC(=O)c1ccc2[n+]([O-])onc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H18 compound treatment 880.0 1.25 0.0 3440.0 2810.0 2.16 1.5271 0.7073 1710057 ChemDiv3_001932 COc1ccc(OC)c2-c3nnc(c4ccc(Cl)cc4)n3C(C)(C)Cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H19 compound treatment 520.0 -359.0 -0.13 680.0 52.4 0.04 -0.0615 -0.461 1559608 ChemDiv3_001933 CCOC(=O)c1c(C)sc2c3CCCCc3[nH]c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H20 compound treatment 1120.0 241.0 0.09 520.0 -108.0 -0.08 0.0021 0.0178 1736634 ChemDiv3_001934 CCc1cc2c(=O)c(coc2cc1OC(=O)C)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H21 compound treatment 720.0 -159.0 -0.06 960.0 332.0 0.26 0.1406 0.5381 1604867 ChemDiv3_001935 O=c1cc(Nc2ccccc2)cc[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H22 compound treatment 840.0 -38.8 -0.01 400.0 -228.0 -0.17 -0.1333 -0.7604 1199255 ChemDiv3_001936 CC(C)OC(=O)c1c(C)oc2cc(Br)c(OC(=O)c3ccco3)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H23 mock treatment 760.0 -119.0 -0.04 360.0 -268.0 -0.21 -0.175 -0.8347 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 H24 mock treatment 1240.0 361.0 0.13 920.0 292.0 0.22 0.2494 0.9646 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I01 compound treatment 320.0 -559.0 -0.2 680.0 52.4 0.04 -0.1117 -0.5523 3020987 ChemDiv3_001937 CCN(CC)c1ccc(cc1)C(=O)/N=c/2\sc3c(ccc4ccccc34)n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I02 compound treatment 320.0 -559.0 -0.2 4320.0 3690.0 2.83 1.8643 0.6561 3118472 ChemDiv3_001938 COc1ccccc1C(=O)/N=C(\N)/Nc2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I03 compound treatment 360.0 -519.0 -0.18 520.0 -108.0 -0.08 -0.1885 -0.9347 1156027 ChemDiv3_001939 CC1CCN(CC(O)COc2ccc(C)cc2C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I04 compound treatment 400.0 -479.0 -0.17 440.0 -188.0 -0.14 -0.2219 -0.9966 3020988 ChemDiv3_001940 Cc1ccc(cc1)C(=O)/N=C(\N)/Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I05 compound treatment 240.0 -639.0 -0.23 3760.0 3130.0 2.4 1.5402 0.6377 1061384 ChemDiv3_001941 CCOC(=O)c1c2C(=O)c3ccccc3C(=O)c2n4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I06 compound treatment 320.0 -559.0 -0.2 360.0 -268.0 -0.21 -0.2854 -0.9998 1323512 ChemDiv3_001942 O=C(NC(Cc1ccccc1)C(=O)OCc2cnc(o2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I07 compound treatment 480.0 -399.0 -0.14 400.0 -228.0 -0.17 -0.2236 -0.9945 3020989 ChemDiv3_001943 CC1(C)C/C(=N\O)/c2c(C1)nc(c3[nH]c4ccccc4c23)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I08 compound treatment 360.0 -519.0 -0.18 280.0 -348.0 -0.27 -0.3188 -0.9835 3020990 ChemDiv3_001944 Oc1ccc(cc1)C(=S)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I09 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 3118473 ChemDiv3_001945 CCN(CC)c1ccc(/C=N/CCc2ccccc2)c(O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I10 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 1727202 ChemDiv3_001946 CCOC(=O)CSc1nc2CCCCc2cc1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I11 compound treatment 400.0 -479.0 -0.17 280.0 -348.0 -0.27 -0.3088 -0.9762 1682537 ChemDiv3_001947 Cc1ccc(cc1)S(=O)(=O)N2N=C(CC2c3ccc(Cl)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I12 compound treatment 1760.0 881.0 0.31 440.0 -188.0 -0.14 0.1192 0.3464 1023355 ChemDiv3_001948 O=C1NC(=S)NC(=O)C1c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I13 compound treatment 1160.0 281.0 0.1 360.0 -268.0 -0.21 -0.0747 -0.3271 3118474 ChemDiv3_001949 O/N=C(/CC1(O)C(=O)Nc2ccccc21)\c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I14 compound treatment 6120.0 5240.0 1.86 1480.0 852.0 0.65 1.7775 0.9018 1292612 ChemDiv3_001950 CC(C)(C)NC(=O)CSc1nc2ccccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I15 compound treatment 640.0 -239.0 -0.08 720.0 92.4 0.07 -0.0097 -0.088 1268842 ChemDiv3_001951 COc1ccc(CN(CCC(c2ccc3OCOc3c2)c4ccccc4OC)C(=O)c5ccco5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I16 compound treatment 1440.0 561.0 0.2 360.0 -268.0 -0.21 -0.0045 -0.0156 3021034 ChemDiv3_001952 COC(=O)c1c(NC(=S)NC(=O)c2ccccc2)sc3CCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I17 compound treatment 760.0 -119.0 -0.04 640.0 12.4 0.01 -0.023 -0.5337 3118475 ChemDiv3_001953 COc1ccccc1C(=O)N/C(=C\c2ccccc2)/C(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I18 compound treatment 320.0 -559.0 -0.2 240.0 -388.0 -0.3 -0.3506 -0.9805 1441672 ChemDiv3_001954 O=C(NC1CCCCCC1)c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I19 compound treatment 360.0 -519.0 -0.18 320.0 -308.0 -0.24 -0.2971 -0.9924 1243149 ChemDiv3_001955 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3csc(n3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I20 compound treatment 680.0 -199.0 -0.07 360.0 -268.0 -0.21 -0.1951 -0.8984 3021035 ChemDiv3_001956 Cn1cccc1/C=C/2\C(=O)NC(=S)N(C2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I21 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 3118476 ChemDiv3_001957 FC(F)(F)c1ccc2Sc3ccccc3N(c2c1)S(=O)(=O)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I22 compound treatment 200.0 -679.0 -0.24 320.0 -308.0 -0.24 -0.3372 -1.0 1013814 ChemDiv3_001958 O=C(N1CN(CN(C1)C(=O)c2ccccc2)C(=O)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I23 mock treatment 280.0 -599.0 -0.21 400.0 -228.0 -0.17 -0.2737 -0.9953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 I24 mock treatment 2840.0 1960.0 0.7 1560.0 932.0 0.72 0.9981 0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J01 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 3021036 ChemDiv3_001959 CCC(C)NC=C1C(=O)NC(=O)NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J02 compound treatment 280.0 -599.0 -0.21 640.0 12.4 0.01 -0.1435 -0.6747 3118477 ChemDiv3_001960 CCOC(=O)C(C1CCCCC1)C(=O)Nc2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J03 compound treatment 360.0 -519.0 -0.18 240.0 -388.0 -0.3 -0.3405 -0.9733 3021037 ChemDiv3_001961 COc1ccc(cc1OC)/C(=C/c2ccc3OCOc3c2)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J04 compound treatment 320.0 -559.0 -0.2 320.0 -308.0 -0.24 -0.3071 -0.9962 1193383 ChemDiv3_001962 Cc1cccc(c1)n2ncc3c(Nc4ccc(cc4)c5ccccc5)ncnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J05 compound treatment 240.0 -639.0 -0.23 320.0 -308.0 -0.24 -0.3272 -0.9998 3118478 ChemDiv3_001963 CC1(C)CC(=C(C2C3=C(CC(C)(C)CC3=O)Oc4ccc(Br)cc24)C(=O)C1)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J06 compound treatment 240.0 -639.0 -0.23 320.0 -308.0 -0.24 -0.3272 -0.9998 1079134 ChemDiv3_001964 OC1(CC(=O)CC2(O)C(=O)Nc3ccccc32)C(=O)Nc4ccccc41 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J07 compound treatment 560.0 -319.0 -0.11 200.0 -428.0 -0.33 -0.3121 -0.8988 3021006 ChemDiv3_001965 COC(=O)CN1C(=O)/C(=C/c2ccc(cc2)N(C)C)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J08 compound treatment 120.0 -759.0 -0.27 280.0 -348.0 -0.27 -0.379 -1.0 3021008 ChemDiv3_001966 COc1ccc(/C=N/c2nc3ccccc3n2C)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J09 compound treatment 160.0 -719.0 -0.25 280.0 -348.0 -0.27 -0.369 -0.9997 3118479 ChemDiv3_001967 CC1(C)NC(=[N+]([O-])C1(C)O)C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J10 compound treatment 560.0 -319.0 -0.11 240.0 -388.0 -0.3 -0.2904 -0.9122 3118608 ChemDiv3_001968 O=C1C(=CNCCc2c[nH]c3ccccc23)C(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J11 compound treatment 320.0 -559.0 -0.2 360.0 -268.0 -0.21 -0.2854 -0.9998 3021012 ChemDiv3_001969 CCN(CC)c1nc(Cl)nc(n1)N(C)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J12 compound treatment 440.0 -439.0 -0.16 400.0 -228.0 -0.17 -0.2336 -0.9983 1214793 ChemDiv3_001970 Cc1ccccc1Nc2nnc(c3ccc(cc3)C(=O)NCCO)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J13 compound treatment 720.0 -159.0 -0.06 880.0 252.0 0.19 0.0972 0.4817 1120090 ChemDiv3_001971 CCc1ccc(NC2=CC(=O)CC(C2)c3ccco3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J14 compound treatment 760.0 -119.0 -0.04 560.0 -67.6 -0.05 -0.0665 -0.9947 1659923 ChemDiv3_001972 O=C(NCc1ccccc1)c2ccc(CN3CCC(Cc4ccccc4)CC3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J15 compound treatment 720.0 -159.0 -0.06 440.0 -188.0 -0.14 -0.1417 -0.9161 1418748 ChemDiv3_001973 CC(=O)NC(c1ccccc1)c2ccc3cccnc3c2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J16 compound treatment 520.0 -359.0 -0.13 320.0 -308.0 -0.24 -0.257 -0.9579 1553968 ChemDiv3_001974 COc1cc(OC)cc(c1)C(=O)Nc2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J17 compound treatment 720.0 -159.0 -0.06 320.0 -308.0 -0.24 -0.2068 -0.8519 1597222 ChemDiv3_001975 CN(C)c1ccc(cc1)C(=S)N2CCN(CC2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J18 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 1631516 ChemDiv3_001976 COC(=O)Cn1c(SCc2ccccc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J19 compound treatment 440.0 -439.0 -0.16 320.0 -308.0 -0.24 -0.277 -0.9795 1261544 ChemDiv3_001977 CCn1c2C(=O)CCCc2c3cc(ccc13)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J20 compound treatment 320.0 -559.0 -0.2 560.0 -67.6 -0.05 -0.1768 -0.8631 1370635 ChemDiv3_001978 O=C(Oc1ccc2cc(c3nc4ccccc4s3)c(=O)oc2c1)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J21 compound treatment 280.0 -599.0 -0.21 4440.0 3810.0 2.93 1.9194 0.6541 1921265 ChemDiv3_001979 CC(=O)n1c(C)c(c2ccccc2)c3cc(Cl)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J22 compound treatment 480.0 -399.0 -0.14 360.0 -268.0 -0.21 -0.2453 -0.9834 1050374 ChemDiv3_001980 O=C1NC(=S)NC(=O)C1=Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J23 mock treatment 280.0 -599.0 -0.21 240.0 -388.0 -0.3 -0.3606 -0.9863 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 J24 mock treatment 3680.0 2800.0 0.99 1040.0 412.0 0.32 0.9266 0.8884 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K01 compound treatment 2480.0 1600.0 0.57 1000.0 372.0 0.29 0.6038 0.9495 1285843 ChemDiv3_001981 COC(=O)c1sc2ccccc2c1NC(=O)c3ccc(cc3)S(=O)(=O)N(C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K02 compound treatment 1440.0 561.0 0.2 480.0 -148.0 -0.11 0.0607 0.2648 1506924 ChemDiv3_001982 COc1ccc(OCC(=O)N2c3ccccc3C(C)(CC2(C)C)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K03 compound treatment 360.0 -519.0 -0.18 360.0 -268.0 -0.21 -0.2754 -0.9985 1117809 ChemDiv3_001983 CC1CCCC(C)N1CC(O)COc2ccc(C)cc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K04 compound treatment 240.0 -639.0 -0.23 200.0 -428.0 -0.33 -0.3923 -0.9836 3118609 ChemDiv3_001984 COc1ccc(/C=C/C(=O)N2c3ccccc3Sc4ccccc24)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K05 compound treatment 320.0 -559.0 -0.2 800.0 172.0 0.13 -0.0466 -0.1954 1720319 ChemDiv3_001985 CCOC(=O)N1CCN(CC(O)COc2c(OC)cccc2OC)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K06 compound treatment 920.0 41.3 0.01 1320.0 692.0 0.53 0.3862 0.7263 1677632 ChemDiv3_001986 O=C(Oc1ccc(cc1)C(=S)N2CCCCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K07 compound treatment 600.0 -279.0 -0.1 1040.0 412.0 0.32 0.154 0.4642 1191436 ChemDiv3_001987 O=C(CCN1C(=O)c2ccccc2C1=O)N(C3CCCCC3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K08 compound treatment 960.0 81.3 0.03 440.0 -188.0 -0.14 -0.0815 -0.5546 3021061 ChemDiv3_001988 O=C(Oc1ccccc1)c2ccc(=O)oc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K09 compound treatment 320.0 -559.0 -0.2 400.0 -228.0 -0.17 -0.2637 -0.998 1177858 ChemDiv3_001989 O=S(=O)(N(Cc1ccccc1)Cc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K10 compound treatment 4640.0 3760.0 1.33 360.0 -268.0 -0.21 0.7982 0.5913 1319852 ChemDiv3_001990 CCC(=O)Nc1cc2c(C)cc(=O)oc2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K11 compound treatment 320.0 -559.0 -0.2 400.0 -228.0 -0.17 -0.2637 -0.998 1184848 ChemDiv3_001991 Cc1ccc(cc1)S(=O)(=O)NCCC(=O)N2CCOCCOCCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K12 compound treatment 800.0 -78.8 -0.03 1000.0 372.0 0.29 0.1824 0.635 1733832 ChemDiv3_001992 CC(=C)c1cccc(c1)C(C)(C)NC(=O)Nc2ccc3c(c2)oc4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K13 compound treatment 3000.0 2120.0 0.75 1240.0 612.0 0.47 0.8646 0.9744 3021100 ChemDiv3_001993 C1CC(SC(C1)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K14 compound treatment 4200.0 3320.0 1.18 3520.0 2890.0 2.22 2.4033 0.956 3118610 ChemDiv3_001994 Cc1ccccc1N2C(=O)NC(=O)/C(=C\C=C\c3ccco3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K15 compound treatment 1400.0 521.0 0.18 1640.0 1010.0 0.78 0.6803 0.8516 1633163 ChemDiv3_001995 O=C(NN1C(=O)C2C3CC(C=C3)C2C1=O)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K16 compound treatment 920.0 41.3 0.01 960.0 332.0 0.26 0.1908 0.7464 1547041 ChemDiv3_001996 OC(=O)c1ccc(Nc2ccnc3cc(Cl)ccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K17 compound treatment 640.0 -239.0 -0.08 4280.0 3650.0 2.8 1.9229 0.6854 1254558 ChemDiv3_001997 CCn1c2ccccc2c3cc(CN4CCN(CC4)C(=O)c5c(OC)cccc5OC)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K18 compound treatment 5640.0 4760.0 1.69 320.0 -308.0 -0.24 1.0274 0.6024 3021103 ChemDiv3_001998 N#Cc1ccc(CSc2nc3ccccc3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K19 compound treatment 520.0 -359.0 -0.13 280.0 -348.0 -0.27 -0.2787 -0.9426 1375332 ChemDiv3_001999 COc1ccccc1C(=O)Nc2cccc(c2)c3csc(n3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K20 compound treatment 4520.0 3640.0 1.29 960.0 332.0 0.26 1.0938 0.8307 3118611 ChemDiv3_002000 O=C/1NC(=S)N(C(=O)\C1=C\C=C\c2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K21 compound treatment 400.0 -479.0 -0.17 600.0 -27.6 -0.02 -0.1351 -0.7892 1417257 ChemDiv3_002001 O=C(CSc1nc2ccccc2s1)n3c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K22 compound treatment 800.0 -78.8 -0.03 320.0 -308.0 -0.24 -0.1867 -0.7853 1162359 ChemDiv3_002002 CC(=O)Nc1cccc(Oc2ccc3C(=O)N(C(=O)c3c2)c4cccc(Cl)c4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K23 mock treatment 560.0 -319.0 -0.11 320.0 -308.0 -0.24 -0.2469 -0.9431 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 K24 mock treatment 3680.0 2800.0 0.99 1040.0 412.0 0.32 0.9266 0.8884 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L01 compound treatment 1120.0 241.0 0.09 1120.0 492.0 0.38 0.3278 0.8458 3118612 ChemDiv3_002003 Cc1ccccc1N2C(=O)NC(=O)/C(=C\Nc3nccs3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L02 compound treatment 440.0 -439.0 -0.16 360.0 -268.0 -0.21 -0.2553 -0.9906 3021107 ChemDiv3_002004 CCOC(=O)C(C1CCCCC1)C(=O)Nc2cccc(c2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L03 compound treatment 200.0 -679.0 -0.24 480.0 -148.0 -0.11 -0.2504 -0.9409 3118613 ChemDiv3_002005 Cc1cc(nc(SCC(=O)NCc2cccc(c2)C(F)(F)F)n1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L04 compound treatment 280.0 -599.0 -0.21 1160.0 532.0 0.41 0.1388 0.3014 1175222 ChemDiv3_002006 C(c1ccccc1)n2ncc3c(Nc4ccc5ccccc5c4)ncnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L05 compound treatment 400.0 -479.0 -0.17 600.0 -27.6 -0.02 -0.1351 -0.7892 1331687 ChemDiv3_002007 CC1(C)CC(=O)C2=C(C1)c3c(NC2C4CCC=CC4)ccc5ncccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L06 compound treatment 320.0 -559.0 -0.2 360.0 -268.0 -0.21 -0.2854 -0.9998 1043898 ChemDiv3_002008 CN(C)Cc1ccc(O)c(CN(C)C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L07 compound treatment 2720.0 1840.0 0.65 320.0 -308.0 -0.24 0.2949 0.4246 3118614 ChemDiv3_002009 COC(=O)CN1C(=O)/C(=C/c2ccc(OCc3ccccc3)c(OC)c2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L08 compound treatment 360.0 -519.0 -0.18 440.0 -188.0 -0.14 -0.232 -0.9926 3021145 ChemDiv3_002010 CN(C)c1ccc(/C=N/c2nc3ccccc3n2Cc4ccc(Cl)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L09 compound treatment 480.0 -399.0 -0.14 920.0 292.0 0.22 0.0587 0.2213 3118615 ChemDiv3_002011 CC12CCCCC2(O)[N+](=C(N1)C(=O)c3ccccc3)[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L10 compound treatment 480.0 -399.0 -0.14 440.0 -188.0 -0.14 -0.2019 -1.0 3021148 ChemDiv3_002012 Cc1ccsc1/C=C(\C#N)/S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L11 compound treatment 600.0 -279.0 -0.1 320.0 -308.0 -0.24 -0.2369 -0.9254 1334871 ChemDiv3_002013 CCOC(=O)CSc1nc(NC#N)nc(n1)N(CC)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L12 compound treatment 720.0 -159.0 -0.06 760.0 132.0 0.1 0.0321 0.2759 1265403 ChemDiv3_002014 COc1ccc(cc1OC)C(=O)c2nc3ccccc3n2C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L13 compound treatment 3720.0 2840.0 1.01 3320.0 2690.0 2.07 2.1743 0.9455 1205179 ChemDiv3_002015 O=C1CC(CC(=C1)NCCc2ccccc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L14 compound treatment 644880.0 644000.0 228.46 453520.0 453000.0 347.69 407.4001 0.9792 3021152 ChemDiv3_002016 O=C1OC(OC(=O)C1=C/C=C/c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L15 compound treatment 4880.0 4000.0 1.42 3840.0 3210.0 2.47 2.7476 0.9656 1493360 ChemDiv3_002017 CCC(=O)NC(c1ccco1)c2c(OC(=O)C)ccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L16 compound treatment 2760.0 1880.0 0.67 2840.0 2210.0 1.7 1.6729 0.9167 1179677 ChemDiv3_002018 CC(C)(C)c1ccc(OCC(=O)Nc2cccc3nsnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L17 compound treatment 760.0 -119.0 -0.04 600.0 -27.6 -0.02 -0.0448 -0.9494 3118616 ChemDiv3_002019 COc1ccccc1OCCn2cc(/C=C\3/SC(=S)NC3=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L18 compound treatment 520.0 -359.0 -0.13 280.0 -348.0 -0.27 -0.2787 -0.9426 1728260 ChemDiv3_002020 O=C1c2ccccc2-c3nc(cc4cccc1c34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L19 compound treatment 480.0 -399.0 -0.14 240.0 -388.0 -0.3 -0.3104 -0.9422 1780366 ChemDiv3_002021 CCOC(=O)CCn1cc(F)c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L20 compound treatment 360.0 -519.0 -0.18 440.0 -188.0 -0.14 -0.232 -0.9926 1567440 ChemDiv3_002022 CCOC(=O)COc1cc2oc(C)c(c3nc4ccccc4s3)c(=O)c2cc1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L21 compound treatment 1920.0 1040.0 0.37 720.0 92.4 0.07 0.3114 0.8278 1579324 ChemDiv3_002023 COC(=O)c1c(N)c(C#N)c2CCCn12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L22 compound treatment 1240.0 361.0 0.13 440.0 -188.0 -0.14 -0.0112 -0.0582 3118756 ChemDiv3_002024 Cc1ccc(C=C2C(=O)NC(=O)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L23 mock treatment 3440.0 2560.0 0.91 680.0 52.4 0.04 0.6709 0.7377 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 L24 mock treatment 840.0 -38.8 -0.01 720.0 92.4 0.07 0.0404 0.5597 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M01 compound treatment 5200.0 4320.0 1.53 880.0 252.0 0.19 1.221 0.7902 1553903 ChemDiv3_002025 COC(=O)c1ccc(cc1)C(=O)NC(=S)Nc2nc3CCCCc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M02 compound treatment 2560.0 1680.0 0.6 1960.0 1330.0 1.02 1.145 0.967 1287477 ChemDiv3_002026 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2c3ccccc3CCc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M03 compound treatment 400.0 -479.0 -0.17 240.0 -388.0 -0.3 -0.3305 -0.9646 1572495 ChemDiv3_002027 Cc1cc(OCC(O)CNC(C)(C)C)ccc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M04 compound treatment 2440.0 1560.0 0.55 600.0 -27.6 -0.02 0.3767 0.6796 3021223 ChemDiv3_002028 Cc1ccc(SCc2cc(O)nc(Nc3nc(C)c4ccccc4n3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M05 compound treatment 2080.0 1200.0 0.43 2440.0 1810.0 1.39 1.2852 0.8832 3118757 ChemDiv3_002029 CCN(CC)/C(=N/S(=O)(=O)c1ccc(Cl)cc1)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M06 compound treatment 4640.0 3760.0 1.33 5120.0 4490.0 3.45 3.3822 0.9146 1719295 ChemDiv3_002030 O=C(Oc1ccccc1C(=S)N2CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M07 compound treatment 5560.0 4680.0 1.66 440.0 -188.0 -0.14 1.0724 0.6434 1588037 ChemDiv3_002031 COc1ccc(cc1)n2c(SCC(=O)c3ccc(Cl)cc3)nc4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M08 compound treatment 5440.0 4560.0 1.62 7920.0 7290.0 5.6 5.1029 0.8756 1217270 ChemDiv3_002032 CC(=O)Nc1cc2c(ccc3ccccc32)oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M09 compound treatment 360.0 -519.0 -0.18 1200.0 572.0 0.44 0.1806 0.3791 1402210 ChemDiv3_002033 COc1ccc(cc1)c2cc3ccccc3n2CC(O)CN(CC=C)CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M10 compound treatment 840.0 -38.8 -0.01 360.0 -268.0 -0.21 -0.155 -0.7527 1306235 ChemDiv3_002034 CC(=O)Nc1cc2nc(N)sc2cc1NC(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M11 compound treatment 3640.0 2760.0 0.98 680.0 52.4 0.04 0.7211 0.7355 3118758 ChemDiv3_002035 COc1ccc(/C=N/c2nc3ccccc3n2CCN4CCCCC4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M12 compound treatment 400.0 -479.0 -0.17 1520.0 892.0 0.69 0.3644 0.5162 3021285 ChemDiv3_002036 CCOC(=O)c1sc(c(C#N)c1C)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M13 compound treatment 960.0 81.3 0.03 920.0 292.0 0.22 0.1791 0.7914 1367535 ChemDiv3_002037 Brc1ccc(cc1)C(=O)NCC2OCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M14 compound treatment 5200.0 4320.0 1.53 6560.0 5930.0 4.55 4.3044 0.8957 3118759 ChemDiv3_002038 CN1C(=O)NC(=O)/C(=C\C=C\c2ccco2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M15 compound treatment 5240.0 4360.0 1.55 1320.0 692.0 0.53 1.4699 0.8985 1234318 ChemDiv3_002039 CCOC(=O)c1c(NC(=S)NCC=C)sc2CCCCCc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M16 compound treatment 680.0 -199.0 -0.07 2200.0 1570.0 1.21 0.8037 0.6647 1416446 ChemDiv3_002040 O=C1C2C3CC(C=C3)C2C(=O)N1CN4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M17 compound treatment 480.0 -399.0 -0.14 360.0 -268.0 -0.21 -0.2453 -0.9834 1311577 ChemDiv3_002041 O=C(N1CCN(Cc2ccc3OCOc3c2)CC1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M18 compound treatment 320.0 -559.0 -0.2 320.0 -308.0 -0.24 -0.3071 -0.9962 3118760 ChemDiv3_002042 COC(=O)/C(=C/c1c[nH]c2ccccc12)/NC(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M19 compound treatment 480.0 -399.0 -0.14 280.0 -348.0 -0.27 -0.2887 -0.9559 1397577 ChemDiv3_002043 Nc1c(nc2ccccn12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M20 compound treatment 600.0 -279.0 -0.1 600.0 -27.6 -0.02 -0.0849 -0.8395 3021354 ChemDiv3_002044 CCN1C(=O)/C(=C/C=C/c2ccco2)/C(=O)NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M21 compound treatment 560.0 -319.0 -0.11 800.0 172.0 0.13 0.0136 0.0784 1484277 ChemDiv3_002045 O=C(C1CC1)N2c3ccccc3CCc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M22 compound treatment 320.0 -559.0 -0.2 2560.0 1930.0 1.48 0.9089 0.6072 3118761 ChemDiv3_002046 Cc1cccc2c1nc3s/c(=C/c4c[nH]nc4c5ccccc5)/c(=O)n32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M23 mock treatment 1000.0 121.0 0.04 1040.0 412.0 0.32 0.2543 0.7959 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 M24 mock treatment 520.0 -359.0 -0.13 2360.0 1730.0 1.33 0.8505 0.6365 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N01 compound treatment 320.0 -559.0 -0.2 1720.0 1090.0 0.84 0.4529 0.5255 3021358 ChemDiv3_002047 Fc1ccccc1N2C(=O)NC(=O)/C(=C\NCCC3=CCCCC3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N02 compound treatment 4160.0 3280.0 1.16 480.0 -148.0 -0.11 0.743 0.6353 1546469 ChemDiv3_002048 OC(=O)c1ccccc1C(=O)OCCN2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N03 compound treatment 1800.0 921.0 0.33 200.0 -428.0 -0.33 -0.001 -0.0022 3021361 ChemDiv3_002049 Cn1cnnc1SCC(=O)NCc2cccc(c2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N04 compound treatment 1280.0 401.0 0.14 800.0 172.0 0.13 0.1942 0.9993 1201390 ChemDiv3_002050 CC1C(NC(C(C)C1=O)c2ccc(cc2)N(C)C)c3ccc(cc3)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N05 compound treatment 400.0 -479.0 -0.17 280.0 -348.0 -0.27 -0.3088 -0.9762 1193866 ChemDiv3_002051 OC(=O)c1c2CCCCc2nc3ccc(Br)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N06 compound treatment 520.0 -359.0 -0.13 1240.0 612.0 0.47 0.2425 0.4978 3118762 ChemDiv3_002052 CC(=O)OC1CCC2C3CCc4cc(OC(=O)C)c(Br)cc4C3CCC12C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N07 compound treatment 840.0 -38.8 -0.01 360.0 -268.0 -0.21 -0.155 -0.7527 1701950 ChemDiv3_002053 Fc1ccc(cc1)N2CCN(CC2)C(=O)Cc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N08 compound treatment 360.0 -519.0 -0.18 480.0 -148.0 -0.11 -0.2102 -0.9729 3118763 ChemDiv3_002054 Cn1c(/N=C/c2cc(c(O)c(c2)C(C)(C)C)C(C)(C)C)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N09 compound treatment 280.0 -599.0 -0.21 1720.0 1090.0 0.84 0.4428 0.5119 3118764 ChemDiv3_002055 Cc1ccc(cc1)C2OCC3(CO2)COC(OC3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N10 compound treatment 680.0 -199.0 -0.07 1280.0 652.0 0.5 0.3043 0.6016 3021365 ChemDiv3_002056 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(o2)c3ccc(Cl)cc3)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N11 compound treatment 720.0 -159.0 -0.06 640.0 12.4 0.01 -0.0331 -0.5792 1540197 ChemDiv3_002057 COc1ccc2oc(C)c(C(=O)CSc3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N12 compound treatment 1000.0 121.0 0.04 1240.0 612.0 0.47 0.3629 0.7686 1543540 ChemDiv3_002058 CCCn1c(nc2ccccc12)C(O)c3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N13 compound treatment 1080.0 201.0 0.07 1440.0 812.0 0.62 0.4915 0.7829 3118765 ChemDiv3_002059 CC(=O)/N=C(\N)/Nc1nc2ccccc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N14 compound treatment 2200.0 1320.0 0.47 1280.0 652.0 0.5 0.6856 0.9995 3021368 ChemDiv3_002060 O=C1OC(OC(=O)C1=Cc2cccs2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N15 compound treatment 1520.0 641.0 0.23 760.0 132.0 0.1 0.2327 0.9341 1445360 ChemDiv3_002061 CN1c2ccccc2C(C)(C)C31Cc4cc(NS(=O)(=O)c5ccc(Cl)cc5)ccc4O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N16 compound treatment 400.0 -479.0 -0.17 2240.0 1610.0 1.24 0.7552 0.6044 3021615 ChemDiv3_002062 COc1cc2CC(C)(C)N/C(=N\N)/c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N17 compound treatment 520.0 -359.0 -0.13 440.0 -188.0 -0.14 -0.1918 -0.9981 3118766 ChemDiv3_002063 COc1ccccc1OCCn2cc(/C=C\3/SC(=S)N(CC=C)C3=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N18 compound treatment 320.0 -559.0 -0.2 680.0 52.4 0.04 -0.1117 -0.5523 1141689 ChemDiv3_002064 Nc1ccc2nc(NC(=O)C3(CC4CC5CC(C4)C3)C5)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N19 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 3021663 ChemDiv3_002065 COc1ccc(/N=C/2\CCCc3ccccc3N2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N20 compound treatment 1040.0 161.0 0.06 520.0 -108.0 -0.08 -0.018 -0.1787 1293367 ChemDiv3_002066 COC(=O)c1c(C)oc2ccc(OC(=O)c3ccc(OC)cc3)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N21 compound treatment 520.0 -359.0 -0.13 1120.0 492.0 0.38 0.1773 0.4445 1917815 ChemDiv3_002067 Clc1ccc(CSc2cn3CCCc3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N22 compound treatment 360.0 -519.0 -0.18 600.0 -27.6 -0.02 -0.1451 -0.7833 3021666 ChemDiv3_002068 CC(C)c1ccc(C=C2C(=O)NC(=O)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N23 mock treatment 200.0 -679.0 -0.24 360.0 -268.0 -0.21 -0.3155 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 N24 mock treatment 280.0 -599.0 -0.21 640.0 12.4 0.01 -0.1435 -0.6747 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O01 compound treatment 200.0 -679.0 -0.24 240.0 -388.0 -0.3 -0.3807 -0.9945 3118767 ChemDiv3_002069 COc1cccc2s/c(=N/C(=O)c3ccccc3)/n(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O02 compound treatment 240.0 -639.0 -0.23 360.0 -268.0 -0.21 -0.3055 -0.9988 1397032 ChemDiv3_002070 Oc1cc(O)nc(SCC(=O)N2c3ccccc3Sc4ccccc24)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O03 compound treatment 360.0 -519.0 -0.18 360.0 -268.0 -0.21 -0.2754 -0.9985 3118768 ChemDiv3_002071 COc1cc(/C=C/C(=O)O)cc(c1OC)S(=O)(=O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O04 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 3021669 ChemDiv3_002072 O=C(/N=c/1\[nH]c(=O)c2ccccc2s1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O05 compound treatment 240.0 -639.0 -0.23 320.0 -308.0 -0.24 -0.3272 -0.9998 3118769 ChemDiv3_002073 CN(C)/C(=N/S(=O)(=O)c1cc(C)ccc1C)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O06 compound treatment 440.0 -439.0 -0.16 240.0 -388.0 -0.3 -0.3205 -0.9543 3021673 ChemDiv3_002074 COc1ccc(cc1)C(=S)N2CCC(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O07 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 3118916 ChemDiv3_002075 Cc1ccc(/C=C/C(=O)O)cc1S(=O)(=O)N2CCC(CC2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O08 compound treatment 240.0 -639.0 -0.23 280.0 -348.0 -0.27 -0.3489 -0.9967 3118917 ChemDiv3_002076 O=C/1N(C2=C(CCCC2)C(=O)\C1=C\Nc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O09 compound treatment 400.0 -479.0 -0.17 240.0 -388.0 -0.3 -0.3305 -0.9646 1215882 ChemDiv3_002077 NNC(=O)CCn1c(c(c2ccccc2)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O10 compound treatment 280.0 -599.0 -0.21 280.0 -348.0 -0.27 -0.3389 -0.9936 1725909 ChemDiv3_002078 CC(=O)Nc1cc(NC(=O)C)c2nc(N)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O11 compound treatment 480.0 -399.0 -0.14 360.0 -268.0 -0.21 -0.2453 -0.9834 3020973 ChemDiv3_002079 COc1cc(cc(OC)c1OC)C(=O)NN2CCN(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O12 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 1397238 ChemDiv3_002080 COc1cccc(c1)c2nc([nH]c2c3cccc(OC)c3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O13 compound treatment 280.0 -599.0 -0.21 440.0 -188.0 -0.14 -0.252 -0.9821 1464925 ChemDiv3_002081 Cc1ccc(cc1)S(=O)(=O)NCC2OCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O14 compound treatment 360.0 -519.0 -0.18 320.0 -308.0 -0.24 -0.2971 -0.9924 1524063 ChemDiv3_002082 CC1(C)CC(=O)C2=C(C1)Oc3ccccc3C2CC(=O)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O15 compound treatment 360.0 -519.0 -0.18 320.0 -308.0 -0.24 -0.2971 -0.9924 1607555 ChemDiv3_002083 CC(C)Oc1ccc(Cc2c(O)nc(SCc3ccccc3)nc2O)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O16 compound treatment 400.0 -479.0 -0.17 440.0 -188.0 -0.14 -0.2219 -0.9966 1471552 ChemDiv3_002084 Oc1ccc(NCN2C(=O)C3C4CC(C=C4)C3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O17 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 1326920 ChemDiv3_002085 Brc1ccccc1CN2CCN(CC2)C(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O18 compound treatment 200.0 -679.0 -0.24 280.0 -348.0 -0.27 -0.359 -0.9987 3021020 ChemDiv3_002086 Nc1ccc2oc(=O)c(cc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O19 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 1185960 ChemDiv3_002087 CCCCc1nn2c(=O)cc(O)nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O20 compound treatment 280.0 -599.0 -0.21 200.0 -428.0 -0.33 -0.3823 -0.9778 1185069 ChemDiv3_002088 CSc1ccc(cc1)C2Nc3ccccc3C(=O)N2c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O21 compound treatment 200.0 -679.0 -0.24 280.0 -348.0 -0.27 -0.359 -0.9987 3021024 ChemDiv3_002089 COc1ccc2c(C)nc(NC(=N)/N=C(\C)/c3ccccc3C(=O)O)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O22 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 3442330 ChemDiv3_002090 O=C1C2CC=CCC2C(=O)N1CNc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O23 mock treatment 160.0 -719.0 -0.25 240.0 -388.0 -0.3 -0.3907 -0.997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 O24 mock treatment 360.0 -519.0 -0.18 320.0 -308.0 -0.24 -0.2971 -0.9924 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P01 compound treatment 200.0 -679.0 -0.24 200.0 -428.0 -0.33 -0.4024 -0.9884 3118918 ChemDiv3_002091 CCN(CC)CCN/C=C/1\C(=O)NC(=O)N(C1=O)c2ccccc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P02 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 1679160 ChemDiv3_002092 CCOC(=O)C(C1CCCCC1)C(=O)Nc2ccc(cc2)N(CC)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P03 compound treatment 320.0 -559.0 -0.2 280.0 -348.0 -0.27 -0.3288 -0.9893 3118919 ChemDiv3_002093 Fc1ccc(CN2C(=O)c3cccc4cccc2c34)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P04 compound treatment 200.0 -679.0 -0.24 200.0 -428.0 -0.33 -0.4024 -0.9884 3021032 ChemDiv3_002094 CCN(CC)CCSc1nc2ccccc2c(=S)n1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P05 compound treatment 240.0 -639.0 -0.23 280.0 -348.0 -0.27 -0.3489 -0.9967 3118920 ChemDiv3_002095 Brc1cccc(/C=C/2\SC(=S)N(CC(=O)NCCc3ccccc3)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P06 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 3118921 ChemDiv3_002096 Oc1ccccc1c2nc(no2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P07 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 1122737 ChemDiv3_002097 C(c1ccccc1)n2c-3c(CCc4nonc43)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P08 compound treatment 240.0 -639.0 -0.23 280.0 -348.0 -0.27 -0.3489 -0.9967 3118922 ChemDiv3_002098 CCOc1ccc2n(C)c(S)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P09 compound treatment 240.0 -639.0 -0.23 1840.0 1210.0 0.93 0.4979 0.5198 1696348 ChemDiv3_002099 Ic1cn(Cc2ccccc2)c(=O)n(Cc3ccccc3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P10 compound treatment 240.0 -639.0 -0.23 1080.0 452.0 0.35 0.0854 0.2059 3021064 ChemDiv3_002100 C=CCN1C(=O)/C(=C/2\SC(=NC2=O)N3CCCCC3)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P11 compound treatment 280.0 -599.0 -0.21 2280.0 1650.0 1.27 0.7468 0.5806 1341945 ChemDiv3_002101 CC(=O)Oc1ccc(cc1)C(=O)N(C(=O)c2ccc(OC(=O)C)cc2)c3cc(C)ccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P12 compound treatment 280.0 -599.0 -0.21 1000.0 372.0 0.29 0.052 0.1459 1706099 ChemDiv3_002102 Brc1ccc(CNc2ccc3n(cnc3c2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P13 compound treatment 280.0 -599.0 -0.21 360.0 -268.0 -0.21 -0.2955 -0.9999 3118923 ChemDiv3_002103 Cc1ccc(cc1)C(=O)/N=C(\N)/Nc2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P14 compound treatment 320.0 -559.0 -0.2 560.0 -67.6 -0.05 -0.1768 -0.8631 3118924 ChemDiv3_002104 Brc1cccc(c1)c2ccc(C=C3C(=O)OC(OC3=O)c4ccccc4)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P15 compound treatment 240.0 -639.0 -0.23 360.0 -268.0 -0.21 -0.3055 -0.9988 1477399 ChemDiv3_002105 Oc1ccc(NS(=O)(=O)c2ccccc2)cc1Sc3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P16 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 3118925 ChemDiv3_002106 CCOC(=O)/C(=N\O)/C1=NC2(CCCC2)Cc3cc(OC)c(OC)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P17 compound treatment 240.0 -639.0 -0.23 320.0 -308.0 -0.24 -0.3272 -0.9998 3021069 ChemDiv3_002107 Fc1ccccc1CNn2c(nc3ccccc3c2=O)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P18 compound treatment 200.0 -679.0 -0.24 200.0 -428.0 -0.33 -0.4024 -0.9884 1607792 ChemDiv3_002108 Cc1nc2ccccc2c(=O)n1NCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P19 compound treatment 280.0 -599.0 -0.21 320.0 -308.0 -0.24 -0.3172 -0.9986 3021070 ChemDiv3_002109 COc1ccc(CC/N=C\2/CCc3ccccc3N2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P20 compound treatment 320.0 -559.0 -0.2 240.0 -388.0 -0.3 -0.3506 -0.9805 1449139 ChemDiv3_002110 CCC1CCCCN1Cc2c(O)ccc3cc(c4nc5ccccc5[nH]4)c(=O)oc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P21 compound treatment 280.0 -599.0 -0.21 200.0 -428.0 -0.33 -0.3823 -0.9778 3118926 ChemDiv3_002111 FC(F)(F)c1cccc(CNC=C2C(=O)CC(CC2=O)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P22 compound treatment 240.0 -639.0 -0.23 240.0 -388.0 -0.3 -0.3706 -0.991 1566538 ChemDiv3_002112 Cc1c(C)c2ccccc2n1CC(O)CNC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P23 mock treatment 160.0 -719.0 -0.25 200.0 -428.0 -0.33 -0.4124 -0.9922 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2006 P24 mock treatment 160.0 -719.0 -0.25 160.0 -468.0 -0.36 -0.4341 -0.986 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A01 compound treatment 200.0 -891.0 -0.32 200.0 -396.0 -0.3 -0.4386 -0.9998 3118927 ChemDiv3_002113 OC(=O)/C=C/c1ccc(cc1)N2C(=O)CC(Cc3ccccc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A02 compound treatment 280.0 -811.0 -0.29 440.0 -156.0 -0.12 -0.2883 -0.9246 3021074 ChemDiv3_002114 CN1C(=O)C(=Cc2ccccc2OCc3ccccc3)C(=O)N(C)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A03 compound treatment 200.0 -891.0 -0.32 240.0 -356.0 -0.27 -0.4169 -0.9974 1510568 ChemDiv3_002115 OCCN(CCO)S(=O)(=O)c1ccc2NC(=O)c3cccc1c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A04 compound treatment 400.0 -691.0 -0.25 200.0 -396.0 -0.3 -0.3884 -0.9943 1149803 ChemDiv3_002116 COc1cccc(c1)C(CC(=O)Nc2sc3CCCCc3c2C#N)NC(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A05 compound treatment 240.0 -851.0 -0.3 680.0 83.9 0.06 -0.168 -0.5441 1377802 ChemDiv3_002117 Clc1ccc2n(CCN(Cc3ccccc3)Cc4ccccc4)c5C(=O)CCCc5c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A06 compound treatment 240.0 -851.0 -0.3 960.0 364.0 0.28 -0.016 -0.0389 1433002 ChemDiv3_002118 OC1=C(N(CC(=O)c2ccccc2)S(=O)(=O)c3ccccc13)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A07 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 1633409 ChemDiv3_002119 Cc1ccc2nc(oc2c1)c3cccc(NC(=O)C4CCCCC4)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A08 compound treatment 160.0 -931.0 -0.33 880.0 284.0 0.22 -0.0795 -0.2009 1233960 ChemDiv3_002120 CC1=C(C(C2=C(CCCC2=O)N1)c3ccsc3)C(=O)Nc4cccc(C)n4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A09 compound treatment 280.0 -811.0 -0.29 2560.0 1960.0 1.51 0.8626 0.562 1227263 ChemDiv3_002121 Cc1cc2nn(nc2cc1NC(=O)c3ccco3)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A10 compound treatment 240.0 -851.0 -0.3 320.0 -276.0 -0.21 -0.3634 -0.985 3021113 ChemDiv3_002122 Cc1ccccc1C(=O)Nc2cccc(NC(=O)c3ccc(o3)c4ccc(Cl)cc4Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A11 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 1332760 ChemDiv3_002123 CCC(C)C1NC(=S)N(C2CCCCC2)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A12 compound treatment 320.0 -771.0 -0.27 480.0 -116.0 -0.09 -0.2565 -0.8914 3021114 ChemDiv3_002124 COc1ccc(/C=C/2\SC(=N)N(C2=O)c3ccc(OC)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A13 compound treatment 600.0 -491.0 -0.17 240.0 -356.0 -0.27 -0.3166 -0.9763 1163749 ChemDiv3_002125 CCOC(=O)c1ccc(Nc2c(cnc3ccccc23)C(=O)OCC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A14 compound treatment 280.0 -811.0 -0.29 720.0 124.0 0.1 -0.1363 -0.4495 1674789 ChemDiv3_002126 CNC(=S)N1N=C(CC1c2cc3ccc(C)cc3nc2Cl)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A15 compound treatment 600.0 -491.0 -0.17 240.0 -356.0 -0.27 -0.3166 -0.9763 1554243 ChemDiv3_002127 Nc1c2CCN(C3CCCCC3)c2nc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A16 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 1450773 ChemDiv3_002128 COc1ccc(Nc2cc(C)nc(n2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A17 compound treatment 280.0 -811.0 -0.29 400.0 -196.0 -0.15 -0.31 -0.9543 3119066 ChemDiv3_002129 CCC(CC)C(=O)N1c2ccccc2CCc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A18 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 3021118 ChemDiv3_002130 CCOC(=O)C1=C(Nc2ccccc2)S/C(=C\c3cccs3)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A19 compound treatment 200.0 -891.0 -0.32 280.0 -316.0 -0.24 -0.3952 -0.9915 3119067 ChemDiv3_002131 CCc1cccc(C)c1n2c(C)cc(/C=C/3\C(=O)NC(=S)N(C3=O)c4ccccc4F)c2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A20 compound treatment 240.0 -851.0 -0.3 320.0 -276.0 -0.21 -0.3634 -0.985 1725478 ChemDiv3_002132 COC(=O)c1c(C)c(C)sc1NC(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A21 compound treatment 240.0 -851.0 -0.3 1120.0 524.0 0.4 0.0709 0.1409 1568777 ChemDiv3_002133 Cc1ccccc1NC2SC(=O)N(Cc3ccccc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A22 compound treatment 320.0 -771.0 -0.27 240.0 -356.0 -0.27 -0.3868 -1.0 1274453 ChemDiv3_002134 O=C(CSc1nc2ccccc2[nH]1)n3c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A23 mock treatment 160.0 -931.0 -0.33 240.0 -356.0 -0.27 -0.4269 -0.9956 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 A24 mock treatment 160.0 -931.0 -0.33 200.0 -396.0 -0.3 -0.4486 -0.9991 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B01 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 1368128 ChemDiv3_002135 COc1ccc(cc1)S(=O)(=O)N2CCC(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B02 compound treatment 200.0 -891.0 -0.32 320.0 -276.0 -0.21 -0.3735 -0.9811 1240761 ChemDiv3_002136 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2C(=O)c3cccc4cccc2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B03 compound treatment 360.0 -731.0 -0.26 360.0 -236.0 -0.18 -0.3116 -0.9846 1428491 ChemDiv3_002137 Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2cccnc2)c3cc(C)cc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B04 compound treatment 5000.0 3910.0 1.39 280.0 -316.0 -0.24 0.8089 0.5746 3119068 ChemDiv3_002138 CN(C)/C=C\1/C=C(N(C)C1=S)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B05 compound treatment 960.0 -131.0 -0.05 600.0 3.87 0.0 -0.0308 -0.6606 3021126 ChemDiv3_002139 CN1CCN(CC1)C(=O)CCN2C(=O)/C(=C/C(=C/c3ccccc3)/C)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B06 compound treatment 360.0 -731.0 -0.26 280.0 -316.0 -0.24 -0.355 -0.9994 1461034 ChemDiv3_002140 CCOc1ccc(OC(=O)c2sc3ncn(CC)c(=O)c3c2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B07 compound treatment 240.0 -851.0 -0.3 320.0 -276.0 -0.21 -0.3634 -0.985 1139126 ChemDiv3_002141 CCOc1ccc(cc1)C2Nc3ccccc3NC4=C2C(=O)CCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B08 compound treatment 200.0 -891.0 -0.32 280.0 -316.0 -0.24 -0.3952 -0.9915 3021956 ChemDiv3_002142 CCn1c(C(=O)O)c(CC(=O)NC2CCCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B09 compound treatment 440.0 -651.0 -0.23 320.0 -276.0 -0.21 -0.3133 -0.9991 1733689 ChemDiv3_002143 CC(=O)Nc1ccc(cc1)n2sc3c(-c4cc(C)ccc4NC3(C)C)c2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B10 compound treatment 640.0 -451.0 -0.16 360.0 -236.0 -0.18 -0.2414 -0.9981 1697535 ChemDiv3_002144 OC(=O)CCNc1nc(c2ccccc2)c3cc(Br)ccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B11 compound treatment 400.0 -691.0 -0.25 1920.0 1320.0 1.02 0.5453 0.5215 3021957 ChemDiv3_002145 OC1(CC(=O)/C=C/C=C/c2ccccc2)C(=O)Nc3ccc(Br)cc31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B12 compound treatment 280.0 -811.0 -0.29 280.0 -316.0 -0.24 -0.3751 -0.9964 3119069 ChemDiv3_002146 CC(=O)N1N=C(CC1c2ccco2)c3c(c4ccccc4)c5cc(Cl)ccc5[nH]c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B13 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 3021958 ChemDiv3_002147 CCn1c(SCCOc2ccc(OC)cc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B14 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 3119070 ChemDiv3_002148 C(/N=C\c1cn(nc1c2cccs2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B15 compound treatment 200.0 -891.0 -0.32 240.0 -356.0 -0.27 -0.4169 -0.9974 1197683 ChemDiv3_002149 Fc1ccc(CN2C(=O)C3C4C=CC(C3C2=O)C54CC5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B16 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 3021959 ChemDiv3_002150 CC[n+]1c(C)n(c2ccccc2)c3ccc(N)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B17 compound treatment 160.0 -931.0 -0.33 200.0 -396.0 -0.3 -0.4486 -0.9991 3021960 ChemDiv3_002151 CCC1(O)CC(=NN1C(=O)c2ccccc2)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B18 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 3119071 ChemDiv3_002152 CNC(=O)CSc1nc2ccccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B19 compound treatment 280.0 -811.0 -0.29 400.0 -196.0 -0.15 -0.31 -0.9543 3119072 ChemDiv3_002153 NS(=O)(=O)c1ccc(cc1)n2cccc2/C=C\3/C(=O)NN(C3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B20 compound treatment 200.0 -891.0 -0.32 240.0 -356.0 -0.27 -0.4169 -0.9974 3021961 ChemDiv3_002154 COc1cccc(/C=C\2/S\C(=N\c3ccccc3)\N(CCc4ccccc4)C2=O)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B21 compound treatment 240.0 -851.0 -0.3 200.0 -396.0 -0.3 -0.4286 -1.0 3119073 ChemDiv3_002155 S=C1NCCN1CCOc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B22 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 3119074 ChemDiv3_002156 Cc1ccc(cc1)C2(CC/N=C/c3ccccc3)CCOC(C)(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B23 mock treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 B24 mock treatment 880.0 -211.0 -0.07 720.0 124.0 0.1 0.0143 0.1177 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C01 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 1621129 ChemDiv3_002157 Clc1ccc(CC2CC(=O)N(C2=O)c3ccccn3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C02 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 3119075 ChemDiv3_002158 Brc1ccc(cc1)N2C(=O)/C(=C/c3ccsc3)/C(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C03 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 3021962 ChemDiv3_002159 C/N=C\1/S/C(=C/c2cccc(F)c2)/C(=O)N1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C04 compound treatment 400.0 -691.0 -0.25 320.0 -276.0 -0.21 -0.3233 -0.9974 1725073 ChemDiv3_002160 CC(C)c1nnc(NC(=O)CC(NC(=O)c2ccccc2)c3ccccc3)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C05 compound treatment 280.0 -811.0 -0.29 280.0 -316.0 -0.24 -0.3751 -0.9964 3021963 ChemDiv3_002161 Cc1cc(C=C2C(=O)c3ccccc3C2=O)c(C)n1c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C06 compound treatment 360.0 -731.0 -0.26 240.0 -356.0 -0.27 -0.3768 -0.9997 1564247 ChemDiv3_002162 CCN1C(=C(O)c2ccccc2S1(=O)=O)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C07 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 1559748 ChemDiv3_002163 O=C(NC(=S)Nc1ccc(Nc2ccccc2)cc1)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C08 compound treatment 200.0 -891.0 -0.32 320.0 -276.0 -0.21 -0.3735 -0.9811 3119076 ChemDiv3_002164 Cc1ccc(cc1)C(=O)C2=C(N)OC3=C(C2c4ccccc4)C(=O)CC(C)(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C09 compound treatment 200.0 -891.0 -0.32 280.0 -316.0 -0.24 -0.3952 -0.9915 1631117 ChemDiv3_002165 CCOc1ccc(cc1Br)C(=O)Nc2c(C)ccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C10 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 1544235 ChemDiv3_002166 COc1ccc(NC(=O)c2ccc3OCCOc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C11 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 3119077 ChemDiv3_002167 CCC(C)C1NC(=S)N(CC=C)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C12 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 1523871 ChemDiv3_002168 Cc1ccccc1OCC(=O)Nc2ccc(NC(=O)c3cccs3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C13 compound treatment 360.0 -731.0 -0.26 400.0 -196.0 -0.15 -0.2899 -0.9665 1635423 ChemDiv3_002169 CCOC(=O)c1cnc2ccccc2c1NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C14 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 3021964 ChemDiv3_002170 O=C(CSc1nnc[nH]1)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C15 compound treatment 240.0 -851.0 -0.3 320.0 -276.0 -0.21 -0.3634 -0.985 1920176 ChemDiv3_002171 CN(C)/C(=N/c1c2CCN(C)c2nc3ccccc13)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C16 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 1612181 ChemDiv3_002172 Cc1ccc(cc1)c2nc3n(ncc3c(=O)n2c4cccc(C)c4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C17 compound treatment 320.0 -771.0 -0.27 160.0 -436.0 -0.33 -0.4302 -0.995 1493219 ChemDiv3_002173 Cc1ncc(NS(=O)(=O)c2ccc(NC(=O)NC3CCCCC3)cc2)c(C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C18 compound treatment 320.0 -771.0 -0.27 240.0 -356.0 -0.27 -0.3868 -1.0 3021965 ChemDiv3_002174 Brc1cccc(c1)C2Nc3ccccc3NC4=C2C(=O)CCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C19 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 3119078 ChemDiv3_002175 C=CCNS(=O)(=O)c1cccc2nonc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C20 compound treatment 240.0 -851.0 -0.3 200.0 -396.0 -0.3 -0.4286 -1.0 3021966 ChemDiv3_002176 Cc1ccc(cc1)c2onc3ccc(Cl)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C21 compound treatment 320.0 -771.0 -0.27 600.0 3.87 0.0 -0.1914 -0.6994 1656889 ChemDiv3_002177 COc1ccc(NC2SC(=O)N(Cc3ccccc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C22 compound treatment 240.0 -851.0 -0.3 360.0 -236.0 -0.18 -0.3417 -0.9702 1674086 ChemDiv3_002178 CC1CC(N(c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C23 mock treatment 360.0 -731.0 -0.26 200.0 -396.0 -0.3 -0.3985 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 C24 mock treatment 5760.0 4670.0 1.66 280.0 -316.0 -0.24 0.9995 0.5971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D01 compound treatment 3600.0 2510.0 0.89 200.0 -396.0 -0.3 0.4143 0.4405 1647021 ChemDiv3_002179 COc1ccc(OCC(=O)NCc2ccco2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D02 compound treatment 360.0 -731.0 -0.26 360.0 -236.0 -0.18 -0.3116 -0.9846 3021967 ChemDiv3_002180 Brc1ccc(cc1)S(=O)(=O)N2C(=O)c3cccc4cccc2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D03 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 1147332 ChemDiv3_002181 CCC(=O)Nc1cccc(NC(=O)c2ccccc2Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D04 compound treatment 280.0 -811.0 -0.29 280.0 -316.0 -0.24 -0.3751 -0.9964 1364711 ChemDiv3_002182 OC(=O)CC1N(COC1=O)C(=O)OCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D05 compound treatment 8360.0 7270.0 2.58 3120.0 2520.0 1.94 3.1934 0.9901 3119079 ChemDiv3_002183 C/C(=C\c1ccccc1)/C=C/2\SC(=S)N(CCC(=O)Nc3ccc(O)c(c3)C(=O)O)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D06 compound treatment 2480.0 1390.0 0.49 400.0 -196.0 -0.15 0.2419 0.4695 1738589 ChemDiv3_002184 CCOC(=O)c1sc2nc(C)nc(N3CCC(C)CC3)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D07 compound treatment 440.0 -651.0 -0.23 280.0 -316.0 -0.24 -0.335 -0.9997 1640618 ChemDiv3_002185 CCCCC(=O)N1C(C2=C(CCCC2=O)Nc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D08 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 3119215 ChemDiv3_002186 CCCN(C(=O)Cc1c(C(=O)O)n(CC)c2ccccc12)c3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D09 compound treatment 200.0 -891.0 -0.32 200.0 -396.0 -0.3 -0.4386 -0.9998 1463910 ChemDiv3_002187 O=C(COc1cccc2ccccc12)N3c4ccccc4CCc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D10 compound treatment 200.0 -891.0 -0.32 240.0 -356.0 -0.27 -0.4169 -0.9974 1205495 ChemDiv3_002188 CC(=O)N1CCN(CC1)c2nc(c3ccccc3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D11 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 3021968 ChemDiv3_002189 Cc1sc2NC(NC(=O)c2c1C)c3cccc(O)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D12 compound treatment 320.0 -771.0 -0.27 240.0 -356.0 -0.27 -0.3868 -1.0 1323939 ChemDiv3_002190 COc1ccc(cc1OC)C2=NN(C(C2)c3ccccc3)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D13 compound treatment 360.0 -731.0 -0.26 320.0 -276.0 -0.21 -0.3333 -0.995 1162446 ChemDiv3_002191 Brc1cc(Br)c2OC3(CCCCCC3=Cc2c1)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D14 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 3119216 ChemDiv3_002192 O=c1oc2ccccc2cc1c3nn(cc3/C=N\Cc4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D15 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 1687509 ChemDiv3_002193 O=C1C2C3C=CC(C2C(=O)N1C4CCCCC4)C53CC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D16 compound treatment 240.0 -851.0 -0.3 360.0 -236.0 -0.18 -0.3417 -0.9702 3021969 ChemDiv3_002194 CC(=O)N1CCN(CCNC=C2C(=O)CC(CC2=O)c3ccccc3)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D17 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 1716478 ChemDiv3_002195 CC1=NN(C(=O)c2ccccc2)C(O)(C1)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D18 compound treatment 280.0 -811.0 -0.29 360.0 -236.0 -0.18 -0.3317 -0.9752 3119217 ChemDiv3_002196 CCC(=O)/N=C/1\NC(=O)\C(=C\c2cn(nc2c3ccccc3)C(=O)CC)\S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D19 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 3021970 ChemDiv3_002197 NS(=O)(=O)c1ccc(cc1)n2cccc2/C=N/c3sc4CCCCc4c3C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D20 compound treatment 200.0 -891.0 -0.32 240.0 -356.0 -0.27 -0.4169 -0.9974 1437077 ChemDiv3_002198 O=C1C2C3CC(C=C3)C2C(=O)N1Cc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D21 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 1281954 ChemDiv3_002199 COc1cc2CC[N+](C)(C)C3Cc4cccc(OC)c4-c(c1O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D22 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 1714344 ChemDiv3_002200 O=C(CC(c1ccccc1)c2ccccc2)N3CCc4ccccc4C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D23 mock treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 D24 mock treatment 400.0 -691.0 -0.25 280.0 -316.0 -0.24 -0.345 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E01 compound treatment 1320.0 229.0 0.08 280.0 -316.0 -0.24 -0.1142 -0.4464 3021971 ChemDiv3_002201 CC(C)OC(=O)CSc1nc2ccccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E02 compound treatment 720.0 -371.0 -0.13 320.0 -276.0 -0.21 -0.243 -0.9738 1589754 ChemDiv3_002202 COc1cccc2c1NC3CC(C)CCC3C2(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E03 compound treatment 760.0 -331.0 -0.12 600.0 3.87 0.0 -0.081 -0.689 3119218 ChemDiv3_002203 COc1cc(ccc1O)c2nc3ccccn3c2/N=C/c4sccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E04 compound treatment 240.0 -851.0 -0.3 840.0 244.0 0.19 -0.0811 -0.2284 1535223 ChemDiv3_002204 Brc1cccc(CN2CCN(Cc3cccc(Br)c3)CC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E05 compound treatment 880.0 -211.0 -0.07 880.0 284.0 0.22 0.1011 0.4387 1399010 ChemDiv3_002205 Cc1cc(C)cc(c1)N2C(=O)CC(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E06 compound treatment 720.0 -371.0 -0.13 680.0 83.9 0.06 -0.0476 -0.3247 3021972 ChemDiv3_002206 CC1CCN(CC1)C(=O)CN(c2ccc(Cl)c(c2)C(F)(F)F)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E07 compound treatment 320.0 -771.0 -0.27 240.0 -356.0 -0.27 -0.3868 -1.0 1189059 ChemDiv3_002207 COc1cccc(NC(=O)c2ccc(o2)c3cccc(Cl)c3C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E08 compound treatment 1360.0 269.0 0.1 240.0 -356.0 -0.27 -0.1259 -0.4349 1646198 ChemDiv3_002208 Brc1ccc2oc(=O)c(cc2c1)C(=O)Oc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E09 compound treatment 280.0 -811.0 -0.29 1080.0 484.0 0.37 0.0592 0.1259 1318523 ChemDiv3_002209 O=C(COc1ccc(cc1)C2N(Cc3ccccc3)CCN2Cc4ccccc4)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E10 compound treatment 440.0 -651.0 -0.23 680.0 83.9 0.06 -0.1178 -0.4913 1328238 ChemDiv3_002210 CS(=O)(=O)N(CC(=O)Nc1cccc(Cl)c1)c2ccccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E11 compound treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 1707569 ChemDiv3_002211 Oc1ccc(CC2NC(=S)N(CC=C)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E12 compound treatment 520.0 -571.0 -0.2 320.0 -276.0 -0.21 -0.2932 -0.9997 1283056 ChemDiv3_002212 O=C(Cc1ccccc1)Nc2ccc(NC(=O)c3cccs3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E13 compound treatment 5600.0 4510.0 1.6 240.0 -356.0 -0.27 0.9377 0.5779 1392332 ChemDiv3_002213 CCOC(=O)c1cnc2c(ccc3ccccc32)c1NCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E14 compound treatment 1920.0 829.0 0.29 360.0 -236.0 -0.18 0.0797 0.2308 1615395 ChemDiv3_002214 OC(CNC1CCCCC1)CN2c3ccccc3Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E15 compound treatment 1400.0 309.0 0.11 520.0 -76.1 -0.06 0.0361 0.291 1627368 ChemDiv3_002215 CCN(CC)c1nc2ccccc2c(N)c1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E16 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 1196972 ChemDiv3_002216 Cc1cccc(c1)c2nc3n(ncc3c(=O)n2c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E17 compound treatment 2480.0 1390.0 0.49 3240.0 2640.0 2.03 1.7836 0.8539 3119219 ChemDiv3_002217 Cc1ccc(SCC(=O)N2CCc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E18 compound treatment 400.0 -691.0 -0.25 1080.0 484.0 0.37 0.0893 0.2006 1517561 ChemDiv3_002218 CN(C)c1ccc(cc1)C2N(C(=O)C)c3ccccc3NC4=C2C(=O)CCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E19 compound treatment 2480.0 1390.0 0.49 3080.0 2480.0 1.91 1.6968 0.8615 1410787 ChemDiv3_002219 CC(NC(=O)c1ccc(cc1)C2(CC3CC4CC(C3)C2)C4)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E20 compound treatment 640.0 -451.0 -0.16 2040.0 1440.0 1.11 0.6706 0.5988 3022027 ChemDiv3_002220 CC(C)C1=NN2C(=NC(=O)/C(=C\c3ccccc3)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E21 compound treatment 2680.0 1590.0 0.56 1040.0 444.0 0.34 0.6395 0.971 3022028 ChemDiv3_002221 CCOc1ccc2ccccc2c1C=C3C(=O)N(C)C(=S)N(C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E22 compound treatment 800.0 -291.0 -0.1 1080.0 484.0 0.37 0.1896 0.4918 3022029 ChemDiv3_002222 COc1ccc2c(C)nc(N/C(=N/S(=O)(=O)c3ccc(C)cc3)/N)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E23 mock treatment 640.0 -451.0 -0.16 440.0 -156.0 -0.12 -0.1979 -0.9898 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 E24 mock treatment 360.0 -731.0 -0.26 400.0 -196.0 -0.15 -0.2899 -0.9665 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F01 compound treatment 4200.0 3110.0 1.1 1520.0 924.0 0.71 1.2813 0.9772 1265045 ChemDiv3_002223 CC(C)C(NC(=O)c1ccc(CN2CCN(CC2)c3ccccc3)cc1)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F02 compound treatment 440.0 -651.0 -0.23 2120.0 1520.0 1.17 0.6639 0.5567 1158625 ChemDiv3_002224 CSc1ccccc1N2C(=O)CC(Sc3ccccc3C(=O)O)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F03 compound treatment 480.0 -611.0 -0.22 4040.0 3440.0 2.64 1.7162 0.6469 3022030 ChemDiv3_002225 COc1ccc(cc1Br)C(=O)NC(=S)Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F04 compound treatment 1520.0 429.0 0.15 1400.0 804.0 0.62 0.5439 0.8558 1652806 ChemDiv3_002226 CCN(CC)c1ccc(NS(=O)(=O)c2ccc(C)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F05 compound treatment 1040.0 -51.3 -0.02 720.0 124.0 0.1 0.0544 0.5617 1567261 ChemDiv3_002227 CCCCC(N1C(=O)c2ccccc2C1=O)C(=O)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F06 compound treatment 11320.0 10200.0 3.63 720.0 124.0 0.1 2.6331 0.7254 1434565 ChemDiv3_002228 CCN(CC)C(=O)Cn1cnc2sc(C(=O)N3CCN(CC3)c4ccc(F)cc4)c(C)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F07 compound treatment 840.0 -251.0 -0.09 2480.0 1880.0 1.45 0.9597 0.6623 1364533 ChemDiv3_002229 CCCC(=O)N1C(C2=C(CCCC2=O)Nc3ccccc13)c4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F08 compound treatment 3280.0 2190.0 0.78 1320.0 724.0 0.56 0.942 0.9866 3022031 ChemDiv3_002230 FC(F)(F)c1ccc(NC(=O)c2cnc(N3CCN(CC3)c4ccccn4)c5ccccc25)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F09 compound treatment 2520.0 1430.0 0.51 1640.0 1040.0 0.8 0.9251 0.9756 3119220 ChemDiv3_002231 Cc1cccc(c1)c2nc3sc4CCCCc4c3c(=O)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F10 compound treatment 2640.0 1550.0 0.55 1720.0 1120.0 0.86 0.9986 0.9762 1563308 ChemDiv3_002232 CC(=O)N1CCN(CC(O)COc2ccc(C)cc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F11 compound treatment 2120.0 1030.0 0.36 400.0 -196.0 -0.15 0.1516 0.384 3119221 ChemDiv3_002233 CCc1ccc(NC(=S)NC(=O)c2cccs2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F12 compound treatment 1560.0 469.0 0.17 2040.0 1440.0 1.11 0.9014 0.8042 1611026 ChemDiv3_002234 Cn1c(SCC(=O)NC(C)(C)C)nc2n(C)c(=O)n(C)c(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F13 compound treatment 5200.0 4110.0 1.46 600.0 3.87 0.0 1.0328 0.7085 3119222 ChemDiv3_002235 Cc1cc(C)c(OCC(=O)Nc2cc(ccc2C)c3nc4ncccc4o3)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F14 compound treatment 2480.0 1390.0 0.49 880.0 284.0 0.22 0.5025 0.9327 3119223 ChemDiv3_002236 O/N=C/c1cn(nc1c2cc3c(ccc4ccccc43)oc2=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F15 compound treatment 1240.0 149.0 0.05 1560.0 964.0 0.74 0.5606 0.7556 1487132 ChemDiv3_002237 COc1ccc(CCNC(=O)C2CC2(c3ccc(C)cc3)c4ccc(C)cc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F16 compound treatment 5080.0 3990.0 1.41 6520.0 5920.0 4.55 4.2164 0.8853 3119224 ChemDiv3_002238 Fc1ccc(/C=C\2/C(=N)N3N=C(SC3=NC2=O)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F17 compound treatment 1400.0 309.0 0.11 2360.0 1760.0 1.35 1.035 0.7618 1544507 ChemDiv3_002239 CC1=NN(C(=O)CCc2ccccc2)C(O)(C1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F18 compound treatment 2120.0 1030.0 0.36 600.0 3.87 0.0 0.2602 0.7128 1669701 ChemDiv3_002240 CC(=O)OCCn1c(=O)c2ccccc2c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F19 compound treatment 2800.0 1710.0 0.61 2600.0 2000.0 1.54 1.5164 0.9171 1368563 ChemDiv3_002241 C(NCC1COc2ccccc2O1)C3COc4ccccc4O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F20 compound treatment 2080.0 989.0 0.35 1760.0 1160.0 0.89 0.8798 0.9166 1013523 ChemDiv3_002242 OCCN1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F21 compound treatment 1520.0 429.0 0.15 760.0 164.0 0.13 0.1965 0.9956 1161064 ChemDiv3_002243 C[N+]1(C)C2CCC1CC(C2)OC(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F22 compound treatment 2160.0 1070.0 0.38 1240.0 644.0 0.49 0.6176 0.9914 1523557 ChemDiv3_002244 C=CCN(CC=C)C(=O)c1cc(nc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F23 mock treatment 1520.0 429.0 0.15 1920.0 1320.0 1.02 0.8262 0.804 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 F24 mock treatment 1560.0 469.0 0.17 800.0 204.0 0.16 0.2283 0.9995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G01 compound treatment 1080.0 -11.3 0.0 4040.0 3440.0 2.64 1.8667 0.706 1293446 ChemDiv3_002245 CC(C(Cc1ccc(C)cc1)C(=O)O)C(=O)Nc2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G02 compound treatment 400.0 -691.0 -0.25 360.0 -236.0 -0.18 -0.3016 -0.9889 3022032 ChemDiv3_002246 CC1=CCC2CC1C(OC2(C)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G03 compound treatment 1800.0 709.0 0.25 1520.0 924.0 0.71 0.6793 0.9027 3119356 ChemDiv3_002247 CC(=O)/N=C/1\NC(=O)\C(=C\c2cccc(Oc3ccccc3)c2)\S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G04 compound treatment 800.0 -291.0 -0.1 920.0 324.0 0.25 0.1028 0.3816 1516568 ChemDiv3_002248 COc1ccc(CN2CCN(Cc3ccccc3C)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G05 compound treatment 2280.0 1190.0 0.42 560.0 -36.1 -0.03 0.2786 0.6592 1531272 ChemDiv3_002249 Cc1cc(Br)ccc1N2C(=O)CC(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G06 compound treatment 4080.0 2990.0 1.06 800.0 204.0 0.16 0.8604 0.8028 3119357 ChemDiv3_002250 COc1cc[n+](OC(=O)N2CCCCC2)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G07 compound treatment 1800.0 709.0 0.25 480.0 -116.0 -0.09 0.1147 0.4301 1356975 ChemDiv3_002251 Clc1ccc(CC(=O)Nc2cccc(c2)c3nc4ccccc4o3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G08 compound treatment 1120.0 28.8 0.01 960.0 364.0 0.28 0.2047 0.7324 3119358 ChemDiv3_002252 CCCOC(=O)c1cc2ccccc2oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G09 compound treatment 2040.0 949.0 0.34 600.0 3.87 0.0 0.2401 0.7133 1339458 ChemDiv3_002253 COc1cc(NC(=O)COc2cc(C)c(Cl)c(C)c2)ccc1NC(=O)c3cc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G10 compound treatment 560.0 -531.0 -0.19 2720.0 2120.0 1.63 1.0197 0.6212 3022033 ChemDiv3_002254 CC(Cc1ccccc1)N/C=C/2\C(=NN(C2=S)c3ccccc3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G11 compound treatment 1200.0 109.0 0.04 1920.0 1320.0 1.02 0.746 0.7334 3119359 ChemDiv3_002255 CCCc1nnc2SCC(=Nn12)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G12 compound treatment 840.0 -251.0 -0.09 360.0 -236.0 -0.18 -0.1912 -0.9465 1382239 ChemDiv3_002256 Cc1cccc(c1)C(=O)Nc2ccc(NC(=O)c3cccs3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G13 compound treatment 320.0 -771.0 -0.27 520.0 -76.1 -0.06 -0.2348 -0.8392 1237291 ChemDiv3_002257 CCOC(=O)c1cnc2c(ccc3ccccc32)c1NCC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G14 compound treatment 480.0 -611.0 -0.22 360.0 -236.0 -0.18 -0.2815 -0.996 1277435 ChemDiv3_002258 Cc1ccc(NCC(O)CN2c3ccccc3Sc4ccccc24)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G15 compound treatment 400.0 -691.0 -0.25 440.0 -156.0 -0.12 -0.2582 -0.9458 1281377 ChemDiv3_002259 CCN(CC)CCN1C(Nc2ccccc2C1=O)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G16 compound treatment 1800.0 709.0 0.25 920.0 324.0 0.25 0.3536 1.0 3119360 ChemDiv3_002260 CCn1cc(c2ccc3ccccc3n2)c(=S)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G17 compound treatment 1120.0 28.8 0.01 640.0 43.9 0.03 0.031 0.8817 3022034 ChemDiv3_002261 Clc1ccc(SCC(=O)N2CCc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G18 compound treatment 1440.0 349.0 0.12 440.0 -156.0 -0.12 0.0027 0.0158 1146503 ChemDiv3_002262 CC(=O)N1C(C2=C(CCCC2=O)Nc3ccccc13)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G19 compound treatment 920.0 -171.0 -0.06 1160.0 564.0 0.43 0.2631 0.602 3022035 ChemDiv3_002263 Oc1ccc(/C=C\2/C(=O)NC(=S)N(CC=C)C2=O)cc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G20 compound treatment 11040.0 9950.0 3.53 6960.0 6360.0 4.89 5.9503 0.9873 3119361 ChemDiv3_002264 CCCC1=NN2C(=NC(=O)/C(=C\c3ccc(OCCOc4ccccc4)cc3)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G21 compound treatment 760.0 -331.0 -0.12 480.0 -116.0 -0.09 -0.1461 -0.9907 3022036 ChemDiv3_002265 COc1ccc(C=C2C(=O)N(C)C(=S)N(C)C2=O)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G22 compound treatment 4120.0 3030.0 1.07 680.0 83.9 0.06 0.8053 0.7481 1651487 ChemDiv3_002266 O=C(Nc1ccc(cc1)S(=O)(=O)Nc2nccs2)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G23 mock treatment 3040.0 1950.0 0.69 560.0 -36.1 -0.03 0.4692 0.6782 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 G24 mock treatment 1560.0 469.0 0.17 360.0 -236.0 -0.18 -0.0106 -0.0431 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H01 compound treatment 2680.0 1590.0 0.56 920.0 324.0 0.25 0.5743 0.9324 1245559 ChemDiv3_002267 CC(C)c1ccc(cc1)N(CC(=O)N2CCN(Cc3ccccc3)CC2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H02 compound treatment 2080.0 989.0 0.35 760.0 164.0 0.13 0.337 0.9043 1264207 ChemDiv3_002268 Cc1ccc(NC(=O)c2sc3nc4CCCCc4cc3c2N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H03 compound treatment 5320.0 4230.0 1.5 480.0 -116.0 -0.09 0.9977 0.6639 3119362 ChemDiv3_002269 CCOc1ccc(/N=C\2/NC(=O)S/C2=C\c3ccc(OC)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H04 compound treatment 560.0 -531.0 -0.19 640.0 43.9 0.03 -0.1094 -0.5717 1690321 ChemDiv3_002270 COc1ccc(Cc2c(O)nc(N)nc2O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H05 compound treatment 520.0 -571.0 -0.2 680.0 83.9 0.06 -0.0978 -0.4598 1362118 ChemDiv3_002271 CCCCC(N1C(=O)c2ccccc2C1=O)C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H06 compound treatment 720.0 -371.0 -0.13 360.0 -236.0 -0.18 -0.2213 -0.9877 1501766 ChemDiv3_002272 CCCCN(CC)C(=O)c1sc2ncnc(N3CCN(CC3)c4ccc(OC)cc4)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H07 compound treatment 1080.0 -11.3 0.0 600.0 3.87 0.0 -7.0E-4 -0.1448 1173112 ChemDiv3_002273 CC1CC(Nc2ccccc2)c3ccccc3N1C(=O)c4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H08 compound treatment 1840.0 749.0 0.27 280.0 -316.0 -0.24 0.0162 0.045 3119363 ChemDiv3_002274 COC(=O)c1nnc(Nc2ccc(Oc3ccccc3)cc2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H09 compound treatment 560.0 -531.0 -0.19 480.0 -116.0 -0.09 -0.1963 -0.9416 3022037 ChemDiv3_002275 C=CCSc1nc2CCCc2cc1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H10 compound treatment 360.0 -731.0 -0.26 520.0 -76.1 -0.06 -0.2248 -0.8452 3119364 ChemDiv3_002276 Cc1c(/N=C/2\SC(CC(=O)O)C(=O)N2/N=C/c3ccccc3O)c(=O)n(c4ccccc4)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H11 compound treatment 600.0 -491.0 -0.17 2600.0 2000.0 1.54 0.9646 0.623 1170987 ChemDiv3_002277 CCC(C)c1ccc(NC(=S)NC(=O)c2ccco2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H12 compound treatment 640.0 -451.0 -0.16 440.0 -156.0 -0.12 -0.1979 -0.9898 1736821 ChemDiv3_002278 COC(=O)Cn1c(Cl)nc2n(C)c(=O)n(C)c(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H13 compound treatment 5000.0 3910.0 1.39 440.0 -156.0 -0.12 0.8957 0.6436 3119365 ChemDiv3_002279 COc1ccc(CC(=O)N2CCC(C2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H14 compound treatment 5920.0 4830.0 1.71 720.0 124.0 0.1 1.2785 0.7452 3119366 ChemDiv3_002280 COc1ccc(cc1)c2nn(cc2C(=O)OCC(C)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H15 compound treatment 680.0 -411.0 -0.15 720.0 124.0 0.1 -0.0359 -0.2062 1268167 ChemDiv3_002281 COc1ccc-2c(CCc3c(C(=O)O)c4cc(Br)ccc4nc32)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H16 compound treatment 2920.0 1830.0 0.65 640.0 43.9 0.03 0.4825 0.7428 3119367 ChemDiv3_002282 COc1ccccc1OCCOc2ccc(cc2)c3nc4sc5CCCCc5c4c(=O)[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H17 compound treatment 400.0 -691.0 -0.25 440.0 -156.0 -0.12 -0.2582 -0.9458 1631822 ChemDiv3_002283 CCC1=NN(C(=O)C(C)C)C(O)(C1)c2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H18 compound treatment 360.0 -731.0 -0.26 480.0 -116.0 -0.09 -0.2465 -0.8985 3119368 ChemDiv3_002284 CC(=O)Oc1ccc(cc1)C(=O)Nc2ccccc2NC(=O)c3ccc(OC(=O)C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H19 compound treatment 1880.0 789.0 0.28 3720.0 3120.0 2.4 1.8937 0.7843 1277012 ChemDiv3_002285 O=C(NCC1OCCc2ccccc12)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H20 compound treatment 1080.0 -11.3 0.0 2760.0 2160.0 1.66 1.1719 0.7054 1299115 ChemDiv3_002286 O=C(CCN1C(=O)C2C3CC(C=C3)C2C1=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H21 compound treatment 800.0 -291.0 -0.1 480.0 -116.0 -0.09 -0.1361 -0.9973 1594929 ChemDiv3_002287 CCOc1ccc(cc1)C(=O)OC2CC3CCC(C2)N3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H22 compound treatment 2360.0 1270.0 0.45 3320.0 2720.0 2.09 1.7969 0.8401 1235484 ChemDiv3_002288 CCOc1ccc2N3C(=O)N(c4ccc(Cl)c(Cl)c4)C(C)(CC3(C)C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H23 mock treatment 1600.0 509.0 0.18 360.0 -236.0 -0.18 -6.0E-4 -0.0022 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 H24 mock treatment 880.0 -211.0 -0.07 880.0 284.0 0.22 0.1011 0.4387 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I01 compound treatment 320.0 -771.0 -0.27 840.0 244.0 0.19 -0.0611 -0.1842 3119369 ChemDiv3_002289 CCN1C(=O)/C(=C\c2ccc(cc2)C(C)C)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I02 compound treatment 360.0 -731.0 -0.26 840.0 244.0 0.19 -0.051 -0.1595 3022038 ChemDiv3_002290 O=C(Nc1ccccc1)OCCCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I03 compound treatment 800.0 -291.0 -0.1 400.0 -196.0 -0.15 -0.1795 -0.9831 3119514 ChemDiv3_002291 Fc1ccc(cc1)N2C(=N)S/C(=C\c3ccccc3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I04 compound treatment 3520.0 2430.0 0.86 520.0 -76.1 -0.06 0.5679 0.6576 1334372 ChemDiv3_002292 COc1ccc(CNCc2ccc(F)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I05 compound treatment 720.0 -371.0 -0.13 280.0 -316.0 -0.24 -0.2647 -0.9588 1278234 ChemDiv3_002293 CC(=O)Nc1ccc2nc(SCc3c(C)cc(C)cc3C)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I06 compound treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 1736428 ChemDiv3_002294 O=C(CN1C(=O)c2ccccc2C1=O)N(Cc3ccccc3)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I07 compound treatment 280.0 -811.0 -0.29 360.0 -236.0 -0.18 -0.3317 -0.9752 1654589 ChemDiv3_002295 O=C(NC(=S)Nc1cccc(NC(=O)c2ccccc2)c1)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I08 compound treatment 200.0 -891.0 -0.32 240.0 -356.0 -0.27 -0.4169 -0.9974 3119515 ChemDiv3_002296 CC1CCN(CC1)S(=O)(=O)c2cc(Br)ccc2Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I09 compound treatment 800.0 -291.0 -0.1 240.0 -356.0 -0.27 -0.2664 -0.9114 3022039 ChemDiv3_002297 CCCOc1ccc(Br)cc1/C=C/2\NC(=S)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I10 compound treatment 240.0 -851.0 -0.3 760.0 164.0 0.13 -0.1246 -0.3808 3022093 ChemDiv3_002298 CCN1C(=O)C(=Cc2cn(Cc3c(F)cccc3Cl)c4ccccc24)C(=O)N(CC)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I11 compound treatment 960.0 -131.0 -0.05 280.0 -316.0 -0.24 -0.2045 -0.8277 3022094 ChemDiv3_002299 O=c1[nH]c(nc2ccccc12)/C(=C/C=C/c3ccccc3)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I12 compound treatment 3920.0 2830.0 1.0 1040.0 444.0 0.34 0.9505 0.8969 1340508 ChemDiv3_002300 CCCOc1ccc(cc1)C(=O)Nc2ccc(NC(=O)c3cccs3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I13 compound treatment 440.0 -651.0 -0.23 320.0 -276.0 -0.21 -0.3133 -0.9991 1247533 ChemDiv3_002301 Brc1ccccc1OCC(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I14 compound treatment 360.0 -731.0 -0.26 440.0 -156.0 -0.12 -0.2682 -0.9385 1388737 ChemDiv3_002302 CC(C)c1cc(C(C)C)c(c(c1)C(C)C)S(=O)(=O)N2CC3C4CC(C=C4)C3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I15 compound treatment 680.0 -411.0 -0.15 360.0 -236.0 -0.18 -0.2313 -0.9942 1214196 ChemDiv3_002303 CC(C)CCOC(=O)c1cc2cc(Br)ccc2oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I16 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 3022095 ChemDiv3_002304 Brc1cc(Br)c2ncc(cc2c1)c3ccc4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I17 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 3119516 ChemDiv3_002305 N/C(=N\C(=O)c1ccccc1NC(=O)c2ccccc2)/Nc3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I18 compound treatment 360.0 -731.0 -0.26 1680.0 1080.0 0.83 0.405 0.4646 1174671 ChemDiv3_002306 CC(=O)N1C(C2=C(CCCC2=O)Nc3ccccc13)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I19 compound treatment 360.0 -731.0 -0.26 440.0 -156.0 -0.12 -0.2682 -0.9385 1639511 ChemDiv3_002307 OC(=O)CN1C(=O)c2cc(Cl)c(Cl)cc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I20 compound treatment 360.0 -731.0 -0.26 360.0 -236.0 -0.18 -0.3116 -0.9846 1138942 ChemDiv3_002308 COc1ccc(OC(=O)N2CCOCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I21 compound treatment 680.0 -411.0 -0.15 480.0 -116.0 -0.09 -0.1662 -0.9721 3119517 ChemDiv3_002309 CCOc1cc(C=C2C(=O)NC(=S)NC2=O)cc(Br)c1OCc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I22 compound treatment 400.0 -691.0 -0.25 320.0 -276.0 -0.21 -0.3233 -0.9974 3119518 ChemDiv3_002310 CC(=O)NS(=O)(=O)c1ccc(cc1)N2C(=O)CC(Sc3nccc(C)n3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I23 mock treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 I24 mock treatment 280.0 -811.0 -0.29 4000.0 3400.0 2.61 1.6443 0.6255 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J01 compound treatment 480.0 -611.0 -0.22 640.0 43.9 0.03 -0.1295 -0.5902 1214355 ChemDiv3_002311 O=C(NC1CC2CCC1C2)c3ccc(CN4CCOCC4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J02 compound treatment 560.0 -531.0 -0.19 1160.0 564.0 0.43 0.1728 0.3661 3119519 ChemDiv3_002312 CC/1=NN(C(=O)\C1=C/Nc2ccc(O)cc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J03 compound treatment 440.0 -651.0 -0.23 640.0 43.9 0.03 -0.1395 -0.5977 3022096 ChemDiv3_002313 OC(=O)/C=C/C(=O)N(Cc1ccccc1)Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J04 compound treatment 320.0 -771.0 -0.27 480.0 -116.0 -0.09 -0.2565 -0.8914 1515659 ChemDiv3_002314 CCCOc1ccc(cc1)C2(CCCC2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J05 compound treatment 1080.0 -11.3 0.0 360.0 -236.0 -0.18 -0.131 -0.7225 3022097 ChemDiv3_002315 S=C(NCc1cccs1)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J06 compound treatment 400.0 -691.0 -0.25 240.0 -356.0 -0.27 -0.3667 -0.9985 1272557 ChemDiv3_002316 CCc1ccc(Nc2ncnc3sc(C)cc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J07 compound treatment 280.0 -811.0 -0.29 360.0 -236.0 -0.18 -0.3317 -0.9752 1185170 ChemDiv3_002317 CCn1c(SCC(=O)c2ccccc2)nc3sc4CCCc4c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J08 compound treatment 280.0 -811.0 -0.29 280.0 -316.0 -0.24 -0.3751 -0.9964 3119520 ChemDiv3_002318 CCCc1n(CC(O)COCC2CCC=CC2)c3ccccc3[n+]1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J09 compound treatment 200.0 -891.0 -0.32 280.0 -316.0 -0.24 -0.3952 -0.9915 1518359 ChemDiv3_002319 CCN(CC)S(=O)(=O)c1ccc(NC(=O)c2ccccc2Cl)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J10 compound treatment 400.0 -691.0 -0.25 320.0 -276.0 -0.21 -0.3233 -0.9974 3022098 ChemDiv3_002320 O=C/1Nc2ccccc2\C1=C/3\SC(=NC3=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J11 compound treatment 480.0 -611.0 -0.22 360.0 -236.0 -0.18 -0.2815 -0.996 3119521 ChemDiv3_002321 CC(C)c1ccc(CN(C(=O)C)c2ccc3oc(nc3c2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J12 compound treatment 440.0 -651.0 -0.23 400.0 -196.0 -0.15 -0.2698 -0.9785 1416925 ChemDiv3_002322 COC(=O)CC1(C(=O)c2ccccc2C1=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J13 compound treatment 5440.0 4350.0 1.54 800.0 204.0 0.16 1.2015 0.7749 1252389 ChemDiv3_002323 CC(=O)Oc1c(Cc2ccccc2)c(=O)oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J14 compound treatment 360.0 -731.0 -0.26 320.0 -276.0 -0.21 -0.3333 -0.995 1282252 ChemDiv3_002324 CN(C)C(=O)Cn1nc(c2ccc(C)cc2)c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J15 compound treatment 280.0 -811.0 -0.29 2040.0 1440.0 1.11 0.5803 0.5067 3119522 ChemDiv3_002325 CC(C)C(=O)N1N=C(CC1(O)C(F)(F)F)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J16 compound treatment 280.0 -811.0 -0.29 480.0 -116.0 -0.09 -0.2665 -0.8847 1724879 ChemDiv3_002326 CC(C)n1nnc2c(=O)oc3ccccc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J17 compound treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 3119523 ChemDiv3_002327 CN1/C(=C/c2cccc[n+]2C)/C=Cc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J18 compound treatment 280.0 -811.0 -0.29 440.0 -156.0 -0.12 -0.2883 -0.9246 1399051 ChemDiv3_002328 O=C(Nc1ccc(cc1)c2nc3ccccc3[nH]2)c4ccc(cc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J19 compound treatment 280.0 -811.0 -0.29 400.0 -196.0 -0.15 -0.31 -0.9543 3022099 ChemDiv3_002329 C/C=C/C(=O)NCC1OCCc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J20 compound treatment 200.0 -891.0 -0.32 280.0 -316.0 -0.24 -0.3952 -0.9915 3119524 ChemDiv3_002330 C/C(=N\N1C(=O)c2ccccc2NC31CCCCC3)/c4ccccc4O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J21 compound treatment 440.0 -651.0 -0.23 360.0 -236.0 -0.18 -0.2915 -0.9928 3022100 ChemDiv3_002331 Fc1ccc(cc1)C2C3C(ON2c4ccc(Cl)cc4)C(=O)N(Cc5ccccc5)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J22 compound treatment 480.0 -611.0 -0.22 160.0 -436.0 -0.33 -0.3901 -0.9779 1474997 ChemDiv3_002332 Clc1cccc(c1)n2c(=O)n(Cc3ccccc3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J23 mock treatment 160.0 -931.0 -0.33 840.0 244.0 0.19 -0.1012 -0.2665 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 J24 mock treatment 680.0 -411.0 -0.15 280.0 -316.0 -0.24 -0.2748 -0.9703 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K01 compound treatment 600.0 -491.0 -0.17 1800.0 1200.0 0.92 0.5303 0.5638 3022101 ChemDiv3_002333 CN1C(=O)/C(=C\c2ccccc2C(F)(F)F)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K02 compound treatment 63560.0 62500.0 22.16 162000.0 161000.0 123.91 103.2894 0.8205 3119525 ChemDiv3_002334 CC/1=NOC(=O)\C1=C\c2ccc(o2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K03 compound treatment 1240.0 149.0 0.05 1960.0 1360.0 1.05 0.7777 0.7418 3119526 ChemDiv3_002335 Cc1ccsc1/C=C\2/SC(=N)N(C2=O)c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K04 compound treatment 800.0 -291.0 -0.1 960.0 364.0 0.28 0.1245 0.4179 3022102 ChemDiv3_002336 COc1ccccc1CCNCc2ccccc2C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K05 compound treatment 360.0 -731.0 -0.26 920.0 324.0 0.25 -0.0076 -0.0212 1231691 ChemDiv3_002337 CCC(=O)Nc1ccc2nc(SCc3ccc(F)c4ccccc34)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K06 compound treatment 2040.0 949.0 0.34 960.0 364.0 0.28 0.4355 0.9957 1284330 ChemDiv3_002338 Cn1ccnc1SCC(=O)Nc2ccc(cc2)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K07 compound treatment 920.0 -171.0 -0.06 360.0 -236.0 -0.18 -0.1711 -0.8951 1135846 ChemDiv3_002339 CCOc1cccc(c1)C(=O)Nc2cc3nn(nc3cc2C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K08 compound treatment 880.0 -211.0 -0.07 440.0 -156.0 -0.12 -0.1377 -0.9744 3022103 ChemDiv3_002340 CC(C)c1cc(C(C)C)c(c(c1)C(C)C)S(=O)(=O)NCCCN2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K09 compound treatment 560.0 -531.0 -0.19 480.0 -116.0 -0.09 -0.1963 -0.9416 1281351 ChemDiv3_002341 CSc1cccc(NC(=O)CSc2nc3ccccc3o2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K10 compound treatment 6280.0 5190.0 1.84 520.0 -76.1 -0.06 1.2602 0.6843 3119527 ChemDiv3_002342 CC(C)c1ccc(/C=c/2\sc3nc4cc(C)c(C)cc4n3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K11 compound treatment 680.0 -411.0 -0.15 440.0 -156.0 -0.12 -0.1879 -0.9952 1434381 ChemDiv3_002343 Cc1cc(C)cc(Oc2coc3cc(O)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K12 compound treatment 600.0 -491.0 -0.17 1000.0 404.0 0.31 0.096 0.27 1361794 ChemDiv3_002344 Clc1ccc2nc(nc(c3ccccc3)c2c1)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K13 compound treatment 1760.0 669.0 0.24 880.0 284.0 0.22 0.3219 0.9991 1502142 ChemDiv3_002345 CCC(C)NC(=O)COc1ccc(cc1)C(C)(C)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K14 compound treatment 640.0 -451.0 -0.16 520.0 -76.1 -0.06 -0.1545 -0.9067 1335752 ChemDiv3_002346 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccccc2)C3CCC(CC3O)C=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K15 compound treatment 960.0 -131.0 -0.05 240.0 -356.0 -0.27 -0.2263 -0.8158 1524452 ChemDiv3_002347 CC1CC(Nc2ccccc2C)c3cccc(C)c3N1C(=O)CN4C(=O)c5ccccc5C4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K16 compound treatment 480.0 -611.0 -0.22 440.0 -156.0 -0.12 -0.2381 -0.9609 3022104 ChemDiv3_002348 Cc1ccc2nc(ccc2c1)c3cnc4ccc(C)cc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K17 compound treatment 440.0 -651.0 -0.23 480.0 -116.0 -0.09 -0.2264 -0.9143 3022105 ChemDiv3_002349 N/C(=N\C(=O)c1ccc(Cl)c(Cl)c1)/N=c/2\[nH]c(=O)c3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K18 compound treatment 520.0 -571.0 -0.2 4360.0 3760.0 2.89 1.9 0.6559 1650441 ChemDiv3_002350 Cc1ccc(Nc2nc(Nc3ccc(C)cc3)nc(n2)N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K19 compound treatment 360.0 -731.0 -0.26 720.0 124.0 0.1 -0.1162 -0.4205 1320117 ChemDiv3_002351 OC(=O)CCN1C(=O)c2cc(Cl)c(Cl)cc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K20 compound treatment 1200.0 109.0 0.04 600.0 3.87 0.0 0.0294 0.7593 3119669 ChemDiv3_002352 Cc1ccc(NC2=NC(=O)CC(S2)C(=O)Nc3ccc(Cl)cc3)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K21 compound treatment 7160.0 6070.0 2.15 2320.0 1720.0 1.32 2.4581 0.9727 3119670 ChemDiv3_002353 CCOc1cc(/C=C/2\SC(=S)NC2=O)cc(Cl)c1OC(=O)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K22 compound treatment 800.0 -291.0 -0.1 600.0 3.87 0.0 -0.071 -0.6865 1476989 ChemDiv3_002354 Cc1ccc(NCC(=O)n2c3CCCCc3c4ccccc24)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K23 mock treatment 1560.0 469.0 0.17 520.0 -76.1 -0.06 0.0763 0.4326 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 K24 mock treatment 1000.0 -91.3 -0.03 2000.0 1400.0 1.08 0.7392 0.6856 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L01 compound treatment 880.0 -211.0 -0.07 480.0 -116.0 -0.09 -0.116 -0.9963 3119671 ChemDiv3_002355 CCOC(=O)C1=CN(C=C(C1c2cccc(OC)c2)C(=O)OCC)c3ccc(OCC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L02 compound treatment 1320.0 229.0 0.08 2160.0 1560.0 1.2 0.9063 0.7532 3022106 ChemDiv3_002356 CC/1=NN(C(=O)\C1=C/Nc2cccc(N)c2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L03 compound treatment 560.0 -531.0 -0.19 560.0 -36.1 -0.03 -0.1529 -0.8025 1437422 ChemDiv3_002357 Cc1cccc(Oc2coc3cc(OCC=C)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L04 compound treatment 360.0 -731.0 -0.26 2360.0 1760.0 1.35 0.7741 0.5614 1446427 ChemDiv3_002358 CCOC(=O)c1sc2nc(C)nc(N(C)Cc3ccccc3)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L05 compound treatment 840.0 -251.0 -0.09 720.0 124.0 0.1 0.0042 0.0324 1719093 ChemDiv3_002359 COc1ccc(NC(=S)NC2CC(C)(C)NC(C)(C)C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L06 compound treatment 560.0 -531.0 -0.19 320.0 -276.0 -0.21 -0.2832 -0.9983 1608447 ChemDiv3_002360 COC(=O)CNC(=O)c1cn(c2ccc(C)c(C)c2)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L07 compound treatment 2200.0 1110.0 0.39 400.0 -196.0 -0.15 0.1717 0.4076 1471198 ChemDiv3_002361 CC1(CN(Cc2ccccc2)CC3(C)CN(Cc4ccccc4)C1)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L08 compound treatment 1160.0 68.8 0.02 320.0 -276.0 -0.21 -0.1327 -0.6217 3119672 ChemDiv3_002362 Cc1ccc2nc(C)nc(c3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L09 compound treatment 400.0 -691.0 -0.25 360.0 -236.0 -0.18 -0.3016 -0.9889 3022107 ChemDiv3_002363 CCN(CC)c1ccc(/N=C/c2ccc(O)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L10 compound treatment 720.0 -371.0 -0.13 440.0 -156.0 -0.12 -0.1779 -0.9989 1436006 ChemDiv3_002364 CCOc1ccc2nc(SCCC(=O)Nc3ccccc3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L11 compound treatment 1120.0 28.8 0.01 480.0 -116.0 -0.09 -0.0558 -0.6222 1304871 ChemDiv3_002365 Cc1ccccc1C(=O)NC(=S)Nc2ccc(cc2)c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L12 compound treatment 480.0 -611.0 -0.22 480.0 -116.0 -0.09 -0.2164 -0.9229 3022108 ChemDiv3_002366 Cc1ccc(cc1)c2nn(cc2/C=N/O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L13 compound treatment 960.0 -131.0 -0.05 440.0 -156.0 -0.12 -0.1177 -0.9152 3119673 ChemDiv3_002367 C[n+]1cc(ccc1/C=N/O)C(=O)NCC[N+](C)(C)Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L14 compound treatment 7600.0 6510.0 2.31 400.0 -196.0 -0.15 1.5262 0.6596 1433089 ChemDiv3_002368 CN(C)S(=O)(=O)c1cc(ccc1C)c2nnc(Nc3ccc(O)cc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L15 compound treatment 360.0 -731.0 -0.26 240.0 -356.0 -0.27 -0.3768 -0.9997 3119674 ChemDiv3_002369 CCCCC1=NN(C(=O)c2ccccc2)C(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L16 compound treatment 1240.0 149.0 0.05 400.0 -196.0 -0.15 -0.0692 -0.4335 1233382 ChemDiv3_002370 CCCCn1nnc2c(=O)oc3ccccc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L17 compound treatment 2040.0 949.0 0.34 400.0 -196.0 -0.15 0.1315 0.3567 1251619 ChemDiv3_002371 Oc1nc2ccccn2c(=O)c1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L18 compound treatment 1120.0 28.8 0.01 720.0 124.0 0.1 0.0745 0.7785 1494865 ChemDiv3_002372 O=c1n(Cc2cccnc2)c(=O)c3ccccc3c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L19 compound treatment 1040.0 -51.3 -0.02 280.0 -316.0 -0.24 -0.1845 -0.758 1414725 ChemDiv3_002373 CC(NCc1ccccc1)C2COc3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L20 compound treatment 720.0 -371.0 -0.13 1480.0 884.0 0.68 0.3867 0.5594 1401815 ChemDiv3_002374 CCSc1nc2ccccc2c(=O)n1c3cccc(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L21 compound treatment 1160.0 68.8 0.02 280.0 -316.0 -0.24 -0.1544 -0.6329 3022109 ChemDiv3_002375 O=C1C2ON(C(C2C(=O)N1c3ccccc3)c4ccco4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L22 compound treatment 800.0 -291.0 -0.1 520.0 -76.1 -0.06 -0.1144 -0.9636 3022159 ChemDiv3_002376 COc1ccc2nc(N/C(=N/C(=O)N3c4ccccc4Sc5ccccc35)/N)nc(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L23 mock treatment 3680.0 2590.0 0.92 240.0 -356.0 -0.27 0.456 0.4759 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 L24 mock treatment 1000.0 -91.3 -0.03 240.0 -356.0 -0.27 -0.2162 -0.7853 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M01 compound treatment 920.0 -171.0 -0.06 1960.0 1360.0 1.05 0.6974 0.665 1276155 ChemDiv3_002377 CCc1ccccc1NC(=O)CCN2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M02 compound treatment 400.0 -691.0 -0.25 2320.0 1720.0 1.32 0.7624 0.5664 3022160 ChemDiv3_002378 CCN1C(=O)/C(=C/c2c(C)c(C#N)c3nc4ccccc4n3c2O)/N(CC)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M03 compound treatment 440.0 -651.0 -0.23 520.0 -76.1 -0.06 -0.2047 -0.8589 1545799 ChemDiv3_002379 Cn1c2C(=O)CCCc2c3cc(Oc4ccccc4)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M04 compound treatment 320.0 -771.0 -0.27 1080.0 484.0 0.37 0.0692 0.15 3022161 ChemDiv3_002380 COc1cc(CNCc2cccc(c2)C(F)(F)F)cc(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M05 compound treatment 1000.0 -91.3 -0.03 480.0 -116.0 -0.09 -0.0859 -0.906 1396765 ChemDiv3_002381 Clc1ccc(CC(=O)Nc2ccccn2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M06 compound treatment 840.0 -251.0 -0.09 560.0 -36.1 -0.03 -0.0826 -0.8853 1526311 ChemDiv3_002382 COc1ccc(OC)c(c1)C2C(=C(C)NC3=C2C(=O)CCC3)C(=O)Nc4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M07 compound treatment 1200.0 109.0 0.04 3240.0 2640.0 2.03 1.4625 0.7204 1280857 ChemDiv3_002383 CCc1nnc(NC(=O)COc2cc(C)c(Cl)c(C)c2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M08 compound treatment 280.0 -811.0 -0.29 1080.0 484.0 0.37 0.0592 0.1259 1263380 ChemDiv3_002384 Cc1ccccc1c2nc3cc(NC(=O)c4cccc(F)c4)ccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M09 compound treatment 520.0 -571.0 -0.2 280.0 -316.0 -0.24 -0.3149 -0.996 1589617 ChemDiv3_002385 CSc1cccc(NC(=O)CSc2nc3ccccc3[nH]2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M10 compound treatment 4760.0 3670.0 1.3 1160.0 564.0 0.43 1.2264 0.8941 3119675 ChemDiv3_002386 CC(Nc1nc(Nc2ccc(F)cc2)nc(SCC(=O)Nc3ccc(F)cc3)n1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M11 compound treatment 360.0 -731.0 -0.26 680.0 83.9 0.06 -0.1379 -0.5159 1511994 ChemDiv3_002387 CC(=O)Oc1ccc2c(=O)c(Oc3cc(C)cc(C)c3)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M12 compound treatment 440.0 -651.0 -0.23 1320.0 724.0 0.56 0.2296 0.3815 1565326 ChemDiv3_002388 CCOC(=O)c1c(O)nc2ccc(Cl)cc2c1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M13 compound treatment 1080.0 -11.3 0.0 840.0 244.0 0.19 0.1296 0.6919 1561823 ChemDiv3_002389 Nc1c2CCN(Cc3ccccc3)c2nc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M14 compound treatment 1160.0 68.8 0.02 1200.0 604.0 0.46 0.3451 0.7433 3022162 ChemDiv3_002390 CC(C)N/C(=N\S(=O)(=O)c1cccs1)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M15 compound treatment 480.0 -611.0 -0.22 400.0 -196.0 -0.15 -0.2598 -0.9841 1441054 ChemDiv3_002391 CC(N1C(=O)c2ccccc2C1=O)C(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M16 compound treatment 440.0 -651.0 -0.23 1240.0 644.0 0.49 0.1862 0.3412 1497947 ChemDiv3_002392 COc1cc(cc(OC)c1OC)c2nc(Nc3ccc(C)c(F)c3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M17 compound treatment 1760.0 669.0 0.24 2320.0 1720.0 1.32 1.1036 0.8208 1419232 ChemDiv3_002393 COc1cc(OC)c(cc1OC)c2nc(c3cccs3)c([nH]2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M18 compound treatment 560.0 -531.0 -0.19 560.0 -36.1 -0.03 -0.1529 -0.8025 3119676 ChemDiv3_002394 CC(N1C(=O)c2ccccc2C1=O)C(=O)/N=C(/NCc3ccc(Cl)cc3)\Nc4nc(C)cc(C)n4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M19 compound treatment 520.0 -571.0 -0.2 1480.0 884.0 0.68 0.3365 0.4752 3022163 ChemDiv3_002395 Cc1cc(/C=C/2\C(=O)NC(=S)N(C2=O)c3ccccc3F)c(C)n1c4ccc(Cl)c(c4)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M20 compound treatment 800.0 -291.0 -0.1 1320.0 724.0 0.56 0.3199 0.5659 3119677 ChemDiv3_002396 Cc1ccc(cc1)S(=O)(=O)N(C(=N)Nc2nc(C)cc(C)n2)c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M21 compound treatment 2840.0 1750.0 0.62 880.0 284.0 0.22 0.5928 0.9015 3022164 ChemDiv3_002397 CC1(C)Cc2c(CO1)sc3nc(S)n(CC=C)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M22 compound treatment 1120.0 28.8 0.01 480.0 -116.0 -0.09 -0.0558 -0.6222 3119678 ChemDiv3_002398 Cc1cc(C)nc(N/C(=N/C(=O)Cc2ccccc2)/N3CCC(CC3)C(=O)N)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M23 mock treatment 1440.0 349.0 0.12 760.0 164.0 0.13 0.1764 1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 M24 mock treatment 1240.0 149.0 0.05 1080.0 484.0 0.37 0.3 0.7995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N01 compound treatment 1520.0 429.0 0.15 1880.0 1280.0 0.99 0.8045 0.8067 1640856 ChemDiv3_002399 O=S(=O)(NC1CC1)c2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N02 compound treatment 800.0 -291.0 -0.1 1560.0 964.0 0.74 0.4502 0.6025 3119679 ChemDiv3_002400 O=C/1SC(=C\C1=C/Nc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N03 compound treatment 1560.0 469.0 0.17 560.0 -36.1 -0.03 0.098 0.5811 1605466 ChemDiv3_002401 CCCOC(=O)COc1ccc2c(=O)c(coc2c1)c3ccccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N04 compound treatment 640.0 -451.0 -0.16 1520.0 924.0 0.71 0.3883 0.5341 1160786 ChemDiv3_002402 C1CCc2c(C1)sc3ncnc(Nc4ccccc4)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N05 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 3119680 ChemDiv3_002403 Cc1ccc(NC(=S)NCC2CCCO2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N06 compound treatment 160.0 -931.0 -0.33 320.0 -276.0 -0.21 -0.3835 -0.977 1548315 ChemDiv3_002404 OC(=O)CNC(=O)Cn1cnc2sc3CCCCc3c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N07 compound treatment 240.0 -851.0 -0.3 440.0 -156.0 -0.12 -0.2983 -0.9181 3022165 ChemDiv3_002405 CN1C(=O)C(O)(C/C(=N/O)/C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N08 compound treatment 240.0 -851.0 -0.3 680.0 83.9 0.06 -0.168 -0.5441 1534538 ChemDiv3_002406 Cc1ccc2nc(NCCC(=O)O)nc(c3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N09 compound treatment 2440.0 1350.0 0.48 4280.0 3680.0 2.83 2.3381 0.8152 3022166 ChemDiv3_002407 Cc1cc(C)n(/N=C/c2ccccc2O)c(=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N10 compound treatment 600.0 -491.0 -0.17 920.0 324.0 0.25 0.0526 0.1732 1701080 ChemDiv3_002408 CCCOC(=O)C(C)Oc1ccc2c(=O)c(coc2c1)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N11 compound treatment 560.0 -531.0 -0.19 760.0 164.0 0.13 -0.0443 -0.1955 1143106 ChemDiv3_002409 Oc1ccc(NC(=S)NC(=O)c2ccccc2)cc1c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N12 compound treatment 1000.0 -91.3 -0.03 600.0 3.87 0.0 -0.0208 -0.6395 3119681 ChemDiv3_002410 COc1ccc(cc1)c2nn(cc2/C=N/O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N13 compound treatment 440.0 -651.0 -0.23 320.0 -276.0 -0.21 -0.3133 -0.9991 3119839 ChemDiv3_002411 CCOC(=O)c1ccc(/C=N/O)[n+](Cc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N14 compound treatment 1040.0 -51.3 -0.02 680.0 83.9 0.06 0.0327 0.4884 1525956 ChemDiv3_002412 COc1nnc(c2ccc(C)c(c2)S(=O)(=O)N(C)C)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N15 compound treatment 880.0 -211.0 -0.07 520.0 -76.1 -0.06 -0.0943 -0.9924 3119840 ChemDiv3_002413 CC1=NN(C(=O)c2ccccc2)C(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N16 compound treatment 1640.0 549.0 0.19 760.0 164.0 0.13 0.2266 0.9777 1151489 ChemDiv3_002414 Nc1c(NC2CCN(Cc3ccccc3)CC2)c4ccccc4oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N17 compound treatment 1000.0 -91.3 -0.03 3320.0 2720.0 2.09 1.4558 0.6961 1129246 ChemDiv3_002415 CC(C)C(=O)Nc1cccc(c1)c2nc3ncccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N18 compound treatment 1120.0 28.8 0.01 920.0 324.0 0.25 0.183 0.7355 3119841 ChemDiv3_002416 COc1cc(/C=C\2/C(=O)NC(=S)N(CC=C)C2=O)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N19 compound treatment 8280.0 7190.0 2.55 600.0 3.87 0.0 1.8054 0.7079 1662903 ChemDiv3_002417 Brc1ccc(cc1)C(=O)NCC2(CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N20 compound treatment 3680.0 2590.0 0.92 800.0 204.0 0.16 0.76 0.8159 1235375 ChemDiv3_002418 CCOC(=O)c1c2CCCc2c(=S)sc1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N21 compound treatment 259160.0 258000.0 91.55 59000.0 58400.0 44.84 96.4399 0.9461 3119842 ChemDiv3_002419 Oc1ccc2ccccc2c1/C=N/S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N22 compound treatment 4800.0 3710.0 1.32 1640.0 1040.0 0.8 1.497 0.9717 1505560 ChemDiv3_002420 O=C(N1CCCc2ccccc12)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N23 mock treatment 1240.0 149.0 0.05 2080.0 1480.0 1.14 0.8428 0.7391 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 N24 mock treatment 1280.0 189.0 0.07 520.0 -76.1 -0.06 0.006 0.0677 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O01 compound treatment 360.0 -731.0 -0.26 320.0 -276.0 -0.21 -0.3333 -0.995 1293078 ChemDiv3_002421 COC(=O)c1c(oc2c1cc(NS(=O)(=O)c3ccc(C)cc3)c4ccccc24)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O02 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 3119843 ChemDiv3_002422 Cn1c2ccc(Br)cc2c3nnc(SCC(=O)NC4=NC(=O)CS4)nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O03 compound treatment 360.0 -731.0 -0.26 280.0 -316.0 -0.24 -0.355 -0.9994 2083303 ChemDiv3_002423 Clc1cccc(Cl)c1N2C(=O)Cc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O04 compound treatment 200.0 -891.0 -0.32 400.0 -196.0 -0.15 -0.33 -0.9424 1629745 ChemDiv3_002424 O=C(CN1C(=C(N2CCOCC2)c3ccccc3S1(=O)=O)C(=O)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O05 compound treatment 200.0 -891.0 -0.32 320.0 -276.0 -0.21 -0.3735 -0.9811 1526005 ChemDiv3_002425 Cc1ccc2nsnc2c1NC(=O)Cc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O06 compound treatment 280.0 -811.0 -0.29 240.0 -356.0 -0.27 -0.3968 -0.9997 1529777 ChemDiv3_002426 CC1=C(C(C2=C(CC(C)(C)CC2=O)N1)c3ccc(C)cc3)C(=O)Nc4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O07 compound treatment 280.0 -811.0 -0.29 320.0 -276.0 -0.21 -0.3534 -0.9887 1225607 ChemDiv3_002427 Cc1ccc2nsnc2c1NC(=O)COc3ccc(Cl)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O08 compound treatment 360.0 -731.0 -0.26 240.0 -356.0 -0.27 -0.3768 -0.9997 1350277 ChemDiv3_002428 Oc1cc(NC(=O)c2ccccc2)ccc1c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O09 compound treatment 400.0 -691.0 -0.25 280.0 -316.0 -0.24 -0.345 -1.0 1230226 ChemDiv3_002429 CSc1ccccc1NC(=O)CSc2nc3cc(C)ccc3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O10 compound treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 3022167 ChemDiv3_002430 CC/N=C/1\S/C(=C\c2ccc(o2)c3cccc(c3)C(=O)O)/C(=O)N1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O11 compound treatment 360.0 -731.0 -0.26 360.0 -236.0 -0.18 -0.3116 -0.9846 1057726 ChemDiv3_002431 Cc1cc(=O)oc2c(CN3CCCCC3)c(O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O12 compound treatment 240.0 -851.0 -0.3 400.0 -196.0 -0.15 -0.32 -0.9483 3022168 ChemDiv3_002432 C/C(=N\N)/c1c(c2ccccc2)c3cc(C)ccc3[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O13 compound treatment 320.0 -771.0 -0.27 320.0 -276.0 -0.21 -0.3434 -0.992 3119844 ChemDiv3_002433 CN(C)c1cc(/N=C/2\CCCN2c3ccccc3)c4ccccc4n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O14 compound treatment 360.0 -731.0 -0.26 520.0 -76.1 -0.06 -0.2248 -0.8452 1039999 ChemDiv3_002434 Cc1nc(N)nc(O)c1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O15 compound treatment 840.0 -251.0 -0.09 920.0 324.0 0.25 0.1128 0.427 3119845 ChemDiv3_002435 CCC(CC)C(=O)N1c2ccccc2Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O16 compound treatment 2240.0 1150.0 0.41 2200.0 1600.0 1.23 1.1588 0.8935 3022169 ChemDiv3_002436 Cc1ccc(C)n1c2ccc(Oc3ccc(Br)cc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O17 compound treatment 7600.0 6510.0 2.31 8080.0 7480.0 5.75 5.6954 0.9198 3119846 ChemDiv3_002437 Cc1cc(C)cc(c1)N2C(=O)/C(=C\c3ccc(cc3)N4CCCCC4)/C(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O18 compound treatment 2280.0 1190.0 0.42 2080.0 1480.0 1.14 1.1037 0.9086 1241829 ChemDiv3_002438 Nc1c(sc2nc3CCCCCc3cc12)C(=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O19 compound treatment 1040.0 -51.3 -0.02 1200.0 604.0 0.46 0.315 0.6789 3022170 ChemDiv3_002439 CCOC(=O)C1=CN(C=C(C1c2cccs2)C(=O)OCC)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O20 compound treatment 720.0 -371.0 -0.13 520.0 -76.1 -0.06 -0.1345 -0.9331 1582713 ChemDiv3_002440 COC(=O)c1cc(=O)n2c3ccccc3nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O21 compound treatment 4280.0 3190.0 1.13 1400.0 804.0 0.62 1.2363 0.9594 1694119 ChemDiv3_002441 CSc1nc(N2CCCCC2)c3CCCCc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O22 compound treatment 520.0 -571.0 -0.2 1000.0 404.0 0.31 0.076 0.205 3119847 ChemDiv3_002442 N/C(=N\C(=O)Nc1ccc(F)cc1)/N=c/2\[nH]c(=O)c3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O23 mock treatment 440.0 -651.0 -0.23 360.0 -236.0 -0.18 -0.2915 -0.9928 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 O24 mock treatment 360.0 -731.0 -0.26 320.0 -276.0 -0.21 -0.3333 -0.995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P01 compound treatment 320.0 -771.0 -0.27 200.0 -396.0 -0.3 -0.4085 -0.9986 1505657 ChemDiv3_002443 CCc1ccccc1N(CC(=O)N2CCC(Cc3ccccc3)CC2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P02 compound treatment 280.0 -811.0 -0.29 280.0 -316.0 -0.24 -0.3751 -0.9964 3119848 ChemDiv3_002444 CN(C)/C=C\1/C=C(OC1=S)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P03 compound treatment 280.0 -811.0 -0.29 600.0 3.87 0.0 -0.2014 -0.6998 3119849 ChemDiv3_002445 C/C(=C\c1ccccc1)/C=C/2\SC(=S)N(CCC(=O)NC3CCCCC3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P04 compound treatment 240.0 -851.0 -0.3 160.0 -436.0 -0.33 -0.4503 -0.9987 1639497 ChemDiv3_002446 Cc1c(sc2ncn(Cc3ccccc3F)c(=O)c12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P05 compound treatment 280.0 -811.0 -0.29 200.0 -396.0 -0.3 -0.4185 -0.9996 1580858 ChemDiv3_002447 Clc1ccc(NC(=S)NCCN2CCOCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P06 compound treatment 200.0 -891.0 -0.32 120.0 -476.0 -0.37 -0.482 -0.9974 3022171 ChemDiv3_002448 CCn1c(C(=O)O)c(CC(=O)Nc2ccccc2F)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P07 compound treatment 160.0 -931.0 -0.33 280.0 -316.0 -0.24 -0.4052 -0.9885 3119850 ChemDiv3_002449 COc1ccc(cc1)C2C3C(=O)c4ccccc4C3=NC5=C2C(=O)CCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P08 compound treatment 320.0 -771.0 -0.27 280.0 -316.0 -0.24 -0.3651 -0.9982 1741530 ChemDiv3_002450 CC(Nc1nc(c2ccccc2)c3cc(Br)ccc3n1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P09 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 3022172 ChemDiv3_002451 COc1ccc(/C=N/n2c(C)cc(C)cc2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P10 compound treatment 240.0 -851.0 -0.3 280.0 -316.0 -0.24 -0.3851 -0.9941 1589009 ChemDiv3_002452 CC1CN(Cc2c(O)ccc3c4ccccc4c(=O)oc23)CC(C)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P11 compound treatment 240.0 -851.0 -0.3 240.0 -356.0 -0.27 -0.4069 -0.9988 1642564 ChemDiv3_002453 Fc1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P12 compound treatment 280.0 -811.0 -0.29 1040.0 444.0 0.34 0.0375 0.084 3119851 ChemDiv3_002454 Fc1ccc(cc1)c2nn(cc2/C=N\Cc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P13 compound treatment 360.0 -731.0 -0.26 320.0 -276.0 -0.21 -0.3333 -0.995 3022173 ChemDiv3_002455 OC(=O)CCC(=O)N1N=C(CC1c2ccccc2F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P14 compound treatment 400.0 -691.0 -0.25 560.0 -36.1 -0.03 -0.193 -0.7821 1129324 ChemDiv3_002456 CCn1c(C)nc2cc(ccc12)S(=O)(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P15 compound treatment 1000.0 -91.3 -0.03 1200.0 604.0 0.46 0.3049 0.6561 3119852 ChemDiv3_002457 CC1=NN(c2nc3ccccc3s2)C(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P16 compound treatment 7760.0 6670.0 2.37 6480.0 5880.0 4.52 4.8669 0.9545 1463659 ChemDiv3_002458 O=c1oc2ccccc2c3n(CCN4CCCC4)cnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P17 compound treatment 1220600.0 1220000.0 432.62 1268680.0 1270000.0 973.53 994.2962 0.9333 3119853 ChemDiv3_002459 COC(=O)/C(=C/C=C/c1ccccc1)/NC(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P18 compound treatment 10720.0 9630.0 3.42 9160.0 8560.0 6.57 7.0643 0.9535 3022283 ChemDiv3_002460 CCOC(=O)c1ccc(cc1)n2c(C)cc(/C=N/O)c2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P19 compound treatment 2680.0 1590.0 0.56 1520.0 924.0 0.71 0.9001 0.9935 1416964 ChemDiv3_002461 CC(OC(=O)C1=C(C)NC(=O)NC1c2cccc(Br)c2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P20 compound treatment 600.0 -491.0 -0.17 520.0 -76.1 -0.06 -0.1646 -0.8952 1631242 ChemDiv3_002462 O=c1[nH]cnc2c1sc3nc(N4CCOCC4)c5CCCCc5c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P21 compound treatment 440.0 -651.0 -0.23 320.0 -276.0 -0.21 -0.3133 -0.9991 1661864 ChemDiv3_002463 CC1(C)CC(=O)C(C2c3ccccc3Oc4ccccc24)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P22 compound treatment 480.0 -611.0 -0.22 280.0 -316.0 -0.24 -0.3249 -0.9984 3119995 ChemDiv3_002464 Cc1cccc(N/C(=N\S(=O)(=O)c2ccc(Cl)cc2)/Nc3nc(C)cc(C)n3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P23 mock treatment 480.0 -611.0 -0.22 280.0 -316.0 -0.24 -0.3249 -0.9984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2007 P24 mock treatment 280.0 -811.0 -0.29 360.0 -236.0 -0.18 -0.3317 -0.9752 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A01 compound treatment 320.0 -930.0 -0.33 360.0 -516.0 -0.4 -0.5135 -0.9959 3022284 ChemDiv3_002465 COc1ccc(cc1)C2CC(=O)C=C(C2)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A02 compound treatment 240.0 -1010.0 -0.36 200.0 -676.0 -0.52 -0.6204 -0.9836 3022285 ChemDiv3_002466 Cc1ccc2C(CC(=O)Oc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A03 compound treatment 120.0 -1130.0 -0.4 320.0 -556.0 -0.43 -0.5854 -0.9995 3119996 ChemDiv3_002467 Cc1cc2nc(SCc3ccc(F)cc3)[nH]c2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A04 compound treatment 320.0 -930.0 -0.33 4520.0 3640.0 2.8 1.7448 0.6194 3119997 ChemDiv3_002468 C(Cn/1c(cs\c1=N/c2ccccc2)c3ccccc3)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A05 compound treatment 400.0 -850.0 -0.3 1200.0 324.0 0.25 -0.0374 -0.0957 3022286 ChemDiv3_002469 COc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)S(=O)(=O)Nc3cnc4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A06 compound treatment 360.0 -890.0 -0.32 2080.0 1200.0 0.92 0.4303 0.4406 3119998 ChemDiv3_002470 CC(C)(C)N(Cc1ccccc1)C(=O)CCCN2C(=O)/C(=C/c3cccs3)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A07 compound treatment 280.0 -970.0 -0.34 1240.0 364.0 0.28 -0.0458 -0.1033 3119999 ChemDiv3_002471 O=C(N/C(=C/c1ccccc1)/C(=O)N2CCCCCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A08 compound treatment 360.0 -890.0 -0.32 4040.0 3160.0 2.43 1.4943 0.6101 3022287 ChemDiv3_002472 Cc1cc(/C=C/2\NC(=O)NC2=O)c(C)n1c3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A09 compound treatment 440.0 -810.0 -0.29 4800.0 3920.0 3.01 1.9269 0.6368 3120000 ChemDiv3_002473 Cc1ccc(CSc2ncnc3sc4CCCc4c23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A10 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 3022288 ChemDiv3_002474 CN(C1CCC(CC1O)C2OCCO2)C(=S)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A11 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 3120001 ChemDiv3_002475 Cn1c(SC/C=C/c2ccccc2)nc3sc4CCCCc4c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A12 compound treatment 160.0 -1090.0 -0.39 360.0 -516.0 -0.4 -0.5536 -0.9999 1445905 ChemDiv3_002476 O=C(NC(=S)c1c(cc2ccccn12)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A13 compound treatment 360.0 -890.0 -0.32 280.0 -596.0 -0.46 -0.5469 -0.9836 3022338 ChemDiv3_002477 CCN1C=C(C(C(=C1)C(=O)OC)c2cc3OCOc3cc2Br)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A14 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 1530239 ChemDiv3_002478 CCCc1c(N)c2c3CCCCCc3sc2nc1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A15 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 3022339 ChemDiv3_002479 Cc1ccc(cc1)C2=CC(=O)C=CC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A16 compound treatment 240.0 -1010.0 -0.36 640.0 -236.0 -0.18 -0.3815 -0.9502 1619080 ChemDiv3_002480 Clc1ccc(cc1)n2ncnc2c3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A17 compound treatment 840.0 -410.0 -0.15 1400.0 524.0 0.4 0.1815 0.4245 1730891 ChemDiv3_002481 O=C(NC(=S)Nc1ccc(cc1)N2CCCCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A18 compound treatment 240.0 -1010.0 -0.36 280.0 -596.0 -0.46 -0.577 -0.9927 3120002 ChemDiv3_002482 CCn1ncc(/C=N/O)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A19 compound treatment 320.0 -930.0 -0.33 360.0 -516.0 -0.4 -0.5135 -0.9959 3120003 ChemDiv3_002483 COC(=O)C/1=C(C)NC(=O)\C1=C/c2cccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A20 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 3022340 ChemDiv3_002484 Cc1cc(C)nc(SCC(=O)c2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A21 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 3120004 ChemDiv3_002485 COC(=O)C/1=C(C)N(Cc2ccc(OC)cc2)C(=O)\C1=C/c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A22 compound treatment 200.0 -1050.0 -0.37 360.0 -516.0 -0.4 -0.5436 -0.9995 1588114 ChemDiv3_002486 COc1ccc(CNCc2ccc(C)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A23 mock treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 A24 mock treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B01 compound treatment 440.0 -810.0 -0.29 400.0 -476.0 -0.37 -0.4617 -0.9929 1211077 ChemDiv3_002487 NS(=O)(=O)c1ccc(NC(=O)CN2C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B02 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 3022341 ChemDiv3_002488 COc1cc(OC)cc(c1)C(=O)/N=C(\N)/Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B03 compound treatment 200.0 -1050.0 -0.37 800.0 -76.1 -0.06 -0.3047 -0.8082 1865468 ChemDiv3_002489 Clc1cccc(c1)C(=O)Nc2cccc(c2)c3cn4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B04 compound treatment 200.0 -1050.0 -0.37 320.0 -556.0 -0.43 -0.5653 -0.9977 1442941 ChemDiv3_002490 CCn1cc(C(=O)NN)c(=O)c2cc(F)c(cc12)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B05 compound treatment 240.0 -1010.0 -0.36 280.0 -596.0 -0.46 -0.577 -0.9927 1645148 ChemDiv3_002491 Cc1ccc(cc1S(=O)(=O)N2CCCCC2)c3nnc(Nc4ccccc4)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B06 compound treatment 360.0 -890.0 -0.32 640.0 -236.0 -0.18 -0.3514 -0.9653 1255255 ChemDiv3_002492 CCOC(=O)C1=C(C)NC(=C(C#N)C1c2ccccc2)SCC(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B07 compound treatment 280.0 -970.0 -0.34 1360.0 484.0 0.37 0.0194 0.0382 1611146 ChemDiv3_002493 Cc1ccc(NS(=O)(=O)CC2(CCC3CC2=O)C3(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B08 compound treatment 200.0 -1050.0 -0.37 360.0 -516.0 -0.4 -0.5436 -0.9995 3120005 ChemDiv3_002494 CSc1nc2sc3CC(CCc3c2c4nncn14)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B09 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 1227402 ChemDiv3_002495 CCOc1ccc(cc1)c2nc3n(nc(C)c3c4cc(OC)c(OC)cc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B10 compound treatment 240.0 -1010.0 -0.36 200.0 -676.0 -0.52 -0.6204 -0.9836 3120006 ChemDiv3_002496 O=P(CCNCc1cccnc1)(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B11 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 1162676 ChemDiv3_002497 Cc1[nH]c(=S)[nH]c(=O)c1Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B12 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 1594508 ChemDiv3_002498 NS(=O)(=O)c1ccc(NC(=O)CC2SC(=O)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B13 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 3120007 ChemDiv3_002499 COc1ccc2ccc(OC)c(/C=C/3\NC(=S)N(C)C3=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B14 compound treatment 360.0 -890.0 -0.32 600.0 -276.0 -0.21 -0.3731 -0.9812 3022342 ChemDiv3_002500 COc1ccccc1/C=C/2\C(=NOC2=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B15 compound treatment 320.0 -930.0 -0.33 480.0 -396.0 -0.3 -0.4483 -0.9992 1365037 ChemDiv3_002501 Cn1c(=O)n(C)c2ncn(CC(=O)NCc3ccco3)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B16 compound treatment 400.0 -850.0 -0.3 1160.0 284.0 0.22 -0.0591 -0.1589 3022343 ChemDiv3_002502 COc1ccc2ccccc2c1C=C3C(=O)OC4(CCCC4)OC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B17 compound treatment 280.0 -970.0 -0.34 880.0 3.87 0.0 -0.2412 -0.701 3120008 ChemDiv3_002503 CN(C)c1ccc(/C=C(/NC(=O)c2cccc(C)c2)\C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B18 compound treatment 320.0 -930.0 -0.33 1520.0 644.0 0.49 0.1162 0.1956 1183856 ChemDiv3_002504 COC(=O)COc1ccc2c(C)c(C)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B19 compound treatment 240.0 -1010.0 -0.36 200.0 -676.0 -0.52 -0.6204 -0.9836 1686688 ChemDiv3_002505 Cc1[nH]c2cc(C)ccc2c1C(=O)CSc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B20 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 1707473 ChemDiv3_002506 CCc1cc2c3CCCCc3c(=O)oc2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B21 compound treatment 280.0 -970.0 -0.34 200.0 -676.0 -0.52 -0.6104 -0.9801 1310201 ChemDiv3_002507 CCCCN(CC)c1ncnc2c1sc3nc(N4CCOCC4)c5COC(C)(C)Cc5c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B22 compound treatment 240.0 -1010.0 -0.36 280.0 -596.0 -0.46 -0.577 -0.9927 3022344 ChemDiv3_002508 Clc1ccc(/C=N/CC2COc3ccccc3O2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B23 mock treatment 3120.0 1870.0 0.66 880.0 3.87 0.0 0.4712 0.7103 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 B24 mock treatment 320.0 -930.0 -0.33 240.0 -636.0 -0.49 -0.5786 -0.9818 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C01 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 3120009 ChemDiv3_002509 CCNC(=S)N1CCN(CCNC=C2C(=O)CC(CC2=O)c3ccccc3)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C02 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 1331130 ChemDiv3_002510 COc1cc2CCN(C(C)c2cc1OC)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C03 compound treatment 200.0 -1050.0 -0.37 320.0 -556.0 -0.43 -0.5653 -0.9977 3022345 ChemDiv3_002511 COc1cc(/C=c/2\sc3nc4cc(C)c(C)cc4n3c2=O)c(Br)cc1OCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C04 compound treatment 280.0 -970.0 -0.34 600.0 -276.0 -0.21 -0.3932 -0.9729 3120010 ChemDiv3_002512 CCOC(=O)c1s/c(=N\c2ccccc2)/n(Cc3ccccc3)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C05 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 1700810 ChemDiv3_002513 Brc1ccc2c3CN(COc3ccc2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C06 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 3120011 ChemDiv3_002514 CC(=O)Oc1cc(c2cccc(c2)C(F)(F)F)c3oc(=O)sc3c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C07 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 3120152 ChemDiv3_002515 COc1ccc(/C=C(/NC(=O)c2ccccc2)\C(=O)N3CC(C)OC(C)C3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C08 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 1521895 ChemDiv3_002516 CCOC(=O)c1sc(NC(=S)NC(=O)c2cc3ccccc3o2)nc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C09 compound treatment 480.0 -770.0 -0.27 240.0 -636.0 -0.49 -0.5385 -0.9623 3120153 ChemDiv3_002517 COC(=O)c1ccc(cc1)n2c(C)cc(C(=O)CSc3ncnc4sc5CCCc5c34)c2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C10 compound treatment 200.0 -1050.0 -0.37 120.0 -756.0 -0.58 -0.6739 -0.977 1371781 ChemDiv3_002518 CC(=C)CNc1nc(c(s1)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C11 compound treatment 160.0 -1090.0 -0.39 400.0 -476.0 -0.37 -0.5319 -0.9996 1255378 ChemDiv3_002519 Cc1ccc(C)c(c1)C(=O)CSc2nc(O)c3c(C)cc(C)nc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C12 compound treatment 200.0 -1050.0 -0.37 320.0 -556.0 -0.43 -0.5653 -0.9977 3022380 ChemDiv3_002520 CC(C)CSc1nnc2sc3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C13 compound treatment 280.0 -970.0 -0.34 560.0 -316.0 -0.24 -0.4149 -0.9854 3022381 ChemDiv3_002521 c1ccc(cc1)c2nnc(o2)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C14 compound treatment 360.0 -890.0 -0.32 200.0 -676.0 -0.52 -0.5903 -0.9716 1304656 ChemDiv3_002522 CCCCn1cnc2sc3CCCCCc3c2c1=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C15 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 3022382 ChemDiv3_002523 Oc1ccccc1C2=Nc3ccccc3N=C(C2)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C16 compound treatment 200.0 -1050.0 -0.37 320.0 -556.0 -0.43 -0.5653 -0.9977 3120154 ChemDiv3_002524 Clc1ccc(cc1)c2ncnn2c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C17 compound treatment 1480.0 230.0 0.08 280.0 -596.0 -0.46 -0.2659 -0.572 1362206 ChemDiv3_002525 COc1cccc(c1)C(=O)CCN2CCC(C2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C18 compound treatment 240.0 -1010.0 -0.36 4520.0 3640.0 2.8 1.7248 0.6115 3022383 ChemDiv3_002526 COC(=O)c1sc(=S)n(C)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C19 compound treatment 400.0 -850.0 -0.3 280.0 -596.0 -0.46 -0.5368 -0.9795 3022384 ChemDiv3_002527 COC(=O)C/1=C(C)N(C)C(=O)\C1=C/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C20 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 3120155 ChemDiv3_002528 O=C(CSc1nsc(SCC(=O)c2ccccc2)n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C21 compound treatment 280.0 -970.0 -0.34 320.0 -556.0 -0.43 -0.5452 -0.9943 3120156 ChemDiv3_002529 COC(=O)C/1=C(C)N(C(=O)\C1=C/c2cccc(OC)c2O)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C22 compound treatment 200.0 -1050.0 -0.37 280.0 -596.0 -0.46 -0.587 -0.9948 1130726 ChemDiv3_002530 Cc1cccc(NC(=O)CN2c3cccc4cccc(c34)S2(=O)=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C23 mock treatment 360.0 -890.0 -0.32 320.0 -556.0 -0.43 -0.5252 -0.989 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 C24 mock treatment 5440.0 4190.0 1.49 320.0 -556.0 -0.43 0.7491 0.4844 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D01 compound treatment 200.0 -1050.0 -0.37 200.0 -676.0 -0.52 -0.6304 -0.9868 1299227 ChemDiv3_002531 Cc1cc(C)nc(NS(=O)(=O)c2ccc(Br)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D02 compound treatment 200.0 -1050.0 -0.37 360.0 -516.0 -0.4 -0.5436 -0.9995 1787887 ChemDiv3_002532 COc1ccc(CC(=O)N2c3ccccc3CCc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D03 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 1865477 ChemDiv3_002533 CCCC(=O)Nc1ccc(cc1)c2cn3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D04 compound treatment 200.0 -1050.0 -0.37 320.0 -556.0 -0.43 -0.5653 -0.9977 3120157 ChemDiv3_002534 O=C(CSC(=S)N1CCSCC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D05 compound treatment 840.0 -410.0 -0.15 280.0 -596.0 -0.46 -0.4265 -0.8881 1175376 ChemDiv3_002535 CNC(=O)COc1ccc(Nc2nnc(c3ccc(C)cc3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D06 compound treatment 320.0 -930.0 -0.33 360.0 -516.0 -0.4 -0.5135 -0.9959 3022385 ChemDiv3_002536 COc1ccc(/N=C/c2cc(\C=N\c3ccc(OC)cc3)c(s2)S(=O)(=O)C(C)(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D07 compound treatment 280.0 -970.0 -0.34 560.0 -316.0 -0.24 -0.4149 -0.9854 1534598 ChemDiv3_002537 CCCCn1c2ncnc(N)c2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D08 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 3022386 ChemDiv3_002538 CCCCn1c(S)nc2sc3CCCCc3c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D09 compound treatment 160.0 -1090.0 -0.39 280.0 -596.0 -0.46 -0.597 -0.9965 1494476 ChemDiv3_002539 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)C(=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D10 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 1479378 ChemDiv3_002540 CC1C=C(C)CC(C1C(=O)O)C(=O)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D11 compound treatment 240.0 -1010.0 -0.36 480.0 -396.0 -0.3 -0.4684 -0.9967 3120158 ChemDiv3_002541 Cc1cc(=O)[nH]c(SCC2COC3(CCCCC3)O2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D12 compound treatment 200.0 -1050.0 -0.37 160.0 -716.0 -0.55 -0.6521 -0.982 1258764 ChemDiv3_002542 Oc1ccc(cc1)C(=O)OCCN2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D13 compound treatment 440.0 -810.0 -0.29 200.0 -676.0 -0.52 -0.5702 -0.9611 1556785 ChemDiv3_002543 O=C(N(Cc1ccccc1)c2ccccn2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D14 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 3120159 ChemDiv3_002544 CC1=C(C(NC(=S)N1)c2cccs2)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D15 compound treatment 2840.0 1590.0 0.56 280.0 -596.0 -0.46 0.0752 0.1036 1223419 ChemDiv3_002545 Cn1c(=O)n(C)c2ncn(CC(=O)Nc3ccncc3)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D16 compound treatment 400.0 -850.0 -0.3 240.0 -636.0 -0.49 -0.5585 -0.9731 3120160 ChemDiv3_002546 COC(=O)c1cccc(c1)c2ccc(C=C3C(=O)OC(OC3=O)c4ccccc4)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D17 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 3022387 ChemDiv3_002547 CCOC(=O)c1[nH]c2ccc(OC)cc2c1/N=C(\C)/N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D18 compound treatment 680.0 -570.0 -0.2 280.0 -596.0 -0.46 -0.4666 -0.9326 1572990 ChemDiv3_002548 Cc1c(Cc2ccccc2)c(=O)oc3cc(OCc4ccc(cc4)C(=O)O)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D19 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 1725504 ChemDiv3_002549 Cc1[nH]c2cc(C)ccc2c1C(=O)CNc3nncs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D20 compound treatment 1960.0 710.0 0.25 320.0 -556.0 -0.43 -0.1238 -0.2497 1194891 ChemDiv3_002550 CCc1cc2c3CCCCc3c(=O)oc2cc1OCC(=O)OC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D21 compound treatment 2800.0 1550.0 0.55 240.0 -636.0 -0.49 0.0435 0.0591 3120161 ChemDiv3_002551 Cc1ccc2c(C)nc(NC3=NC(CC(=O)N3)C(=O)Nc4ccc(Cl)c(Cl)c4)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D22 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 3022388 ChemDiv3_002552 CN(C)c1ccc(/C=N/CC2COc3ccccc3O2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D23 mock treatment 280.0 -970.0 -0.34 320.0 -556.0 -0.43 -0.5452 -0.9943 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 D24 mock treatment 440.0 -810.0 -0.29 520.0 -356.0 -0.27 -0.3965 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E01 compound treatment 1640.0 390.0 0.14 6440.0 5560.0 4.27 3.1182 0.7296 3120162 ChemDiv3_002553 CCc1ccc(NC=C2C(=O)NC(=S)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E02 compound treatment 1440.0 190.0 0.07 520.0 -356.0 -0.27 -0.1457 -0.5173 3022389 ChemDiv3_002554 Cc1cc(=O)oc(C)c1C(=O)Nc2ccccc2C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E03 compound treatment 200.0 -1050.0 -0.37 1320.0 444.0 0.34 -0.0224 -0.0444 3120163 ChemDiv3_002555 CCOc1cc(/C=C\2/C(=O)N(C(=S)N(C2=O)c3ccc(C)c(C)c3)c4ccccc4)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E04 compound treatment 800.0 -450.0 -0.16 1400.0 524.0 0.4 0.1715 0.3964 3022390 ChemDiv3_002556 CC(C)n/1c(cs\c1=N/c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E05 compound treatment 560.0 -690.0 -0.24 440.0 -436.0 -0.33 -0.4098 -0.9881 3120164 ChemDiv3_002557 CN(C)c1ccc2c3c(ccc(N(C)C)c13)[C@@](O)(O[C@]2(O)C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E06 compound treatment 960.0 -290.0 -0.1 1480.0 604.0 0.46 0.2551 0.5371 1542419 ChemDiv3_002558 CCc1ccc(cc1)S(=O)(=O)N2CCSC2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E07 compound treatment 2040.0 790.0 0.28 3800.0 2920.0 2.24 1.7854 0.7893 3120165 ChemDiv3_002559 COc1ccc(/C=C(/NC(=O)c2ccccc2)\C(=O)N3CC4(C)CC3CC(C)(C)C4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E08 compound treatment 680.0 -570.0 -0.2 240.0 -636.0 -0.49 -0.4883 -0.9238 1526755 ChemDiv3_002560 O=C(NC(=S)Nc1ccc(cc1)c2nc3ccccc3o2)c4cc5ccccc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E09 compound treatment 800.0 -450.0 -0.16 280.0 -596.0 -0.46 -0.4365 -0.9005 1316885 ChemDiv3_002561 CC(C)c1ccc(cc1)c2csc3ncnc(Oc4cccc(NC(=O)C)c4)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E10 compound treatment 400.0 -850.0 -0.3 320.0 -556.0 -0.43 -0.5151 -0.9855 3022391 ChemDiv3_002562 CC(C)(C)N1CCN(C1=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E11 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 3120166 ChemDiv3_002563 CCOc1cc(/C=C/c2ccccc2OC)cc(=O)c3c(C)oc(C)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E12 compound treatment 280.0 -970.0 -0.34 4200.0 3320.0 2.55 1.5611 0.6063 1320812 ChemDiv3_002564 Cc1ccc(cc1)S(=O)(=O)NC(=O)Oc2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E13 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 3120167 ChemDiv3_002565 N=C/1N2N=C(SC2=NC(=O)\C1=C/c3ccco3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E14 compound treatment 520.0 -730.0 -0.26 800.0 -76.1 -0.06 -0.2244 -0.8454 1465230 ChemDiv3_002566 COc1ccc(cc1)c2oc3ncn(CC(C)C)c(=N)c3c2c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E15 compound treatment 2480.0 1230.0 0.44 840.0 -36.1 -0.03 0.2889 0.6608 3022392 ChemDiv3_002567 Cc1ccc(O)c(c1)C2=Nc3ccccc3N=C(C2)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E16 compound treatment 5640.0 4390.0 1.56 280.0 -596.0 -0.46 0.7776 0.479 3120168 ChemDiv3_002568 COc1ccc(cc1)n2ncnc2c3ccc(Cl)cc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E17 compound treatment 760.0 -490.0 -0.17 520.0 -356.0 -0.27 -0.3162 -0.9761 3022431 ChemDiv3_002569 O=C1CC(CN1Cc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E18 compound treatment 1760.0 510.0 0.18 1800.0 924.0 0.71 0.6295 0.8599 3117887 ChemDiv3_002570 COC(=O)c1sc(=S)n(c1C)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E19 compound treatment 5680.0 4430.0 1.57 3960.0 3080.0 2.37 2.7853 0.9802 1664411 ChemDiv3_002571 OC(=O)CN(CCc1ccccc1)S(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E20 compound treatment 1960.0 710.0 0.25 800.0 -76.1 -0.06 0.1368 0.529 1431891 ChemDiv3_002572 Nc1c(sc2nc3CCCc3cc12)C(=O)Nc4ccc5ccccc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E21 compound treatment 5240.0 3990.0 1.42 320.0 -556.0 -0.43 0.699 0.4728 3117888 ChemDiv3_002573 OC(=O)COc1ccc(/C=C/2\SC(=O)N(Cc3ccc(F)cc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E22 compound treatment 1720.0 470.0 0.17 1120.0 244.0 0.19 0.2503 0.9983 3022432 ChemDiv3_002574 CCN1C(=O)S/C(=C\c2ccc3OCOc3c2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E23 mock treatment 1920.0 670.0 0.24 5040.0 4160.0 3.2 2.4285 0.7576 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 E24 mock treatment 400.0 -850.0 -0.3 2280.0 1400.0 1.08 0.5489 0.4904 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F01 compound treatment 2200.0 950.0 0.34 800.0 -76.1 -0.06 0.197 0.5759 1533782 ChemDiv3_002575 CCOC(=O)C1CCCN(C1)C(=O)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F02 compound treatment 640.0 -610.0 -0.22 1400.0 524.0 0.4 0.1314 0.2877 3022433 ChemDiv3_002576 Cc1ccc(cc1)N2C(=C)c3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F03 compound treatment 1000.0 -250.0 -0.09 6560.0 5680.0 4.36 3.0228 0.6926 1865482 ChemDiv3_002577 COc1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F04 compound treatment 1440.0 190.0 0.07 1200.0 324.0 0.25 0.2235 0.8675 3022434 ChemDiv3_002578 CC[n+]1oc(C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F05 compound treatment 5520.0 4270.0 1.51 2320.0 1440.0 1.11 1.8549 0.9882 3117889 ChemDiv3_002579 Cc1ccccc1/C=N/n2c(C)cc(C)c(C#N)c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F06 compound treatment 2560.0 1310.0 0.46 2000.0 1120.0 0.86 0.9387 0.9579 3022435 ChemDiv3_002580 O=C1NC/C(=N/c2ccccc2)/C(=O)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F07 compound treatment 2600.0 1350.0 0.48 920.0 43.9 0.03 0.3625 0.755 1539111 ChemDiv3_002581 Cc1ccc(cc1C)n2c(N)c(C#N)c3nc4ccccc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F08 compound treatment 280.0 -970.0 -0.34 6920.0 6040.0 4.64 3.0377 0.6529 1362970 ChemDiv3_002582 CCCCn1c(SCC)nc2sc3CCCCc3c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F09 compound treatment 1880.0 630.0 0.22 6440.0 5560.0 4.27 3.1784 0.7431 3117890 ChemDiv3_002583 CC1=CCC2C(C1)C(=O)N(C2=O)c3cccc(c3)C(=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F10 compound treatment 1960.0 710.0 0.25 1560.0 684.0 0.53 0.5493 0.9434 1378678 ChemDiv3_002584 OC(=O)C1C(C2CC1C=C2)C(=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F11 compound treatment 4440.0 3190.0 1.13 1040.0 164.0 0.13 0.8891 0.7809 1291546 ChemDiv3_002585 CC(C)COC(=O)CCn1[nH]c(=O)c2ccccc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F12 compound treatment 3240.0 1990.0 0.71 1240.0 364.0 0.28 0.6967 0.9177 1293113 ChemDiv3_002586 CCOC(=O)c1sc(NC(=O)CC)nc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F13 compound treatment 4120.0 2870.0 1.02 960.0 83.9 0.06 0.7655 0.7503 1488462 ChemDiv3_002587 CC(NC(=O)c1cccc(c1)C(=O)NC(C)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F14 compound treatment 1640.0 390.0 0.14 1200.0 324.0 0.25 0.2736 0.9617 1671651 ChemDiv3_002588 CCOC(=O)C1(O)N(C)C(=O)Nc2ccccc21 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F15 compound treatment 3320.0 2070.0 0.73 560.0 -316.0 -0.24 0.3476 0.4495 1629502 ChemDiv3_002589 CCOc1cc(cc(OCC)c1OCC)C(=O)Nc2cc(Cl)ccc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F16 compound treatment 2520.0 1270.0 0.45 800.0 -76.1 -0.06 0.2772 0.6103 3022436 ChemDiv3_002590 CCc1cc(=O)oc2c(C)c(OC)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F17 compound treatment 2760.0 1510.0 0.54 640.0 -236.0 -0.18 0.2506 0.4431 1227508 ChemDiv3_002591 COc1ccc2[nH]c3c(OC)ncnc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F18 compound treatment 3440.0 2190.0 0.78 600.0 -276.0 -0.21 0.3994 0.496 1648918 ChemDiv3_002592 CCc1cc(=O)oc2c(C)c(O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F19 compound treatment 3240.0 1990.0 0.71 400.0 -476.0 -0.37 0.2407 0.3028 1501783 ChemDiv3_002593 COc1ccc2n(C)c(C)c(C(=O)CNc3nc(C)cs3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F20 compound treatment 520.0 -730.0 -0.26 1440.0 564.0 0.43 0.123 0.2438 1246346 ChemDiv3_002594 COc1ccc(OCc2nc3ccccc3[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F21 compound treatment 2360.0 1110.0 0.39 3440.0 2560.0 1.97 1.6703 0.8321 3022437 ChemDiv3_002595 CCNC(=O)N1c2ccc(CC)cc2C(=CC1(C)C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F22 compound treatment 2640.0 1390.0 0.49 3080.0 2200.0 1.69 1.5451 0.8767 1589501 ChemDiv3_002596 COc1ccc(cc1)C(=O)NCC2OCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F23 mock treatment 3400.0 2150.0 0.76 960.0 83.9 0.06 0.5848 0.7641 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 F24 mock treatment 1240.0 -10.0 0.0 1040.0 164.0 0.13 0.0865 0.6869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G01 compound treatment 3440.0 2190.0 0.78 400.0 -476.0 -0.37 0.2909 0.3388 3022438 ChemDiv3_002597 N/C=C\1/C(=O)N(N=C1C(F)(F)F)c2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G02 compound treatment 5680.0 4430.0 1.57 280.0 -596.0 -0.46 0.7876 0.4812 1506877 ChemDiv3_002598 COC(=O)CN1C(C2=C(CC(C)(C)CC2=O)Nc3ccccc13)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G03 compound treatment 1720.0 470.0 0.17 440.0 -436.0 -0.33 -0.1189 -0.3178 3022439 ChemDiv3_002599 CCOC(=O)C1=C(N=C2SCC(=O)N2C1c3ccc(OCC)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G04 compound treatment 320.0 -930.0 -0.33 1240.0 364.0 0.28 -0.0358 -0.0827 3117891 ChemDiv3_002600 COc1ccc(cc1)c2cs/c(=N\c3ccc(Br)cc3)/n2CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G05 compound treatment 600.0 -650.0 -0.23 760.0 -116.0 -0.09 -0.2261 -0.9145 3117892 ChemDiv3_002601 COc1ccc(/C=C/C(=O)NC(=O)c2ccccc2OCC(=O)c3ccc(Br)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G06 compound treatment 1680.0 430.0 0.15 720.0 -156.0 -0.12 0.0231 0.1191 3022440 ChemDiv3_002602 COc1ccc(Br)cc1C2SCCN2S(=O)(=O)c3ccc(Cl)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G07 compound treatment 1240.0 -10.0 0.0 520.0 -356.0 -0.27 -0.1958 -0.7162 3117893 ChemDiv3_002603 CN(C)c1ccc(/C=C/2\SC(=O)N(Cc3ccccc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G08 compound treatment 1440.0 190.0 0.07 880.0 3.87 0.0 0.0498 0.7376 1606088 ChemDiv3_002604 O=C(NC(=S)Nc1ccc(NC(=O)c2ccco2)cc1)c3cc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G09 compound treatment 1000.0 -250.0 -0.09 480.0 -396.0 -0.3 -0.2778 -0.8768 1241306 ChemDiv3_002605 Cc1nc(NCCc2ccccc2)c3c4CCCCc4sc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G10 compound treatment 800.0 -450.0 -0.16 920.0 43.9 0.03 -0.0891 -0.5459 3022441 ChemDiv3_002606 Clc1cccc(c1)C(=O)SC2=NCCS2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G11 compound treatment 440.0 -810.0 -0.29 560.0 -316.0 -0.24 -0.3748 -0.9965 1517676 ChemDiv3_002607 CCOc1ccc(cc1)c2cc(OC)c3c(C)oc(C)c3c(=O)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G12 compound treatment 840.0 -410.0 -0.15 1400.0 524.0 0.4 0.1815 0.4245 1056016 ChemDiv3_002608 O=C1C2CCCCC2=NN1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G13 compound treatment 840.0 -410.0 -0.15 920.0 43.9 0.03 -0.079 -0.5294 3117894 ChemDiv3_002609 CN(C)c1ccc(/C=C\2/C(=N)N3N=C(COc4ccccc4)SC3=NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G14 compound treatment 1080.0 -170.0 -0.06 1080.0 204.0 0.16 0.068 0.4056 1386956 ChemDiv3_002610 COc1ccc(cc1)c2oc3ncn(Cc4ccccc4)c(=N)c3c2c5ccc(OC)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G15 compound treatment 1600.0 350.0 0.12 440.0 -436.0 -0.33 -0.149 -0.4171 3022442 ChemDiv3_002611 Cc1cc(C)c2c(=O)cc(oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G16 compound treatment 1160.0 -90.0 -0.03 960.0 83.9 0.06 0.023 0.3194 1642217 ChemDiv3_002612 COc1cc(cc(OC)c1OC)c2ncnn2c3sc4CCCCCc4c3C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G17 compound treatment 720.0 -530.0 -0.19 720.0 -156.0 -0.12 -0.2177 -0.9764 3117895 ChemDiv3_002613 COc1ccccc1/C=C/C(=O)N2CCCC(C2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G18 compound treatment 360.0 -890.0 -0.32 1440.0 564.0 0.43 0.0829 0.1546 3022476 ChemDiv3_002614 CCOC(=O)C1=C(C)N2CCN=C2S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G19 compound treatment 440.0 -810.0 -0.29 720.0 -156.0 -0.12 -0.2879 -0.9248 1293580 ChemDiv3_002615 CC(C)c1ccc(NC(=O)CN(CCc2ccccc2)S(=O)(=O)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G20 compound treatment 1880.0 630.0 0.22 360.0 -516.0 -0.4 -0.1222 -0.2685 1308860 ChemDiv3_002616 O=c1oc2ccccc2cc1c3csc(n3)C(=C4CCCC4)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G21 compound treatment 800.0 -450.0 -0.16 440.0 -436.0 -0.33 -0.3496 -0.9426 3117896 ChemDiv3_002617 CCOc1cc(/C=C/2\SC(=O)N(Cc3ccc(F)cc3)C2=O)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G22 compound treatment 4880.0 3630.0 1.29 1920.0 1040.0 0.8 1.4772 0.974 1189641 ChemDiv3_002618 CC1=C(C(C2=C(CC(CC2=O)c3ccccc3)N1)c4cccc(O)c4)C(=O)OCc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G23 mock treatment 2080.0 830.0 0.29 2440.0 1560.0 1.2 1.0572 0.8552 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 G24 mock treatment 1280.0 30.0 0.01 680.0 -196.0 -0.15 -0.0989 -0.6555 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H01 compound treatment 560.0 -690.0 -0.24 1040.0 164.0 0.13 -0.0841 -0.3057 1179631 ChemDiv3_002619 CCC(CC)NC(=O)C1c2ccccc2Oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H02 compound treatment 440.0 -810.0 -0.29 1160.0 284.0 0.22 -0.0491 -0.1361 3117897 ChemDiv3_002620 CC1CCN(CC1)C(=S)SCC(=O)n2c3CCCCc3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H03 compound treatment 440.0 -810.0 -0.29 600.0 -276.0 -0.21 -0.3531 -0.9888 1787952 ChemDiv3_002621 OC(CN1CCN(CC1)C=O)Cn2c3ccccc3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H04 compound treatment 640.0 -610.0 -0.22 600.0 -276.0 -0.21 -0.3029 -0.9999 3117898 ChemDiv3_002622 OC1(CC(=NO1)/C=C/c2ccccc2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H05 compound treatment 1560.0 310.0 0.11 640.0 -236.0 -0.18 -0.0504 -0.2378 1693003 ChemDiv3_002623 O=C(CCCC(=O)N1CCc2ccccc12)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H06 compound treatment 2360.0 1110.0 0.39 1320.0 444.0 0.34 0.5194 0.9974 1498872 ChemDiv3_002624 CCn1cc(C(=O)NN)c(=O)c2cc(F)c(NN)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H07 compound treatment 320.0 -930.0 -0.33 720.0 -156.0 -0.12 -0.318 -0.9061 1431137 ChemDiv3_002625 COC(=O)CN(Cc1ccccc1)S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H08 compound treatment 520.0 -730.0 -0.26 1360.0 484.0 0.37 0.0796 0.1757 1193183 ChemDiv3_002626 CCCCn1c(NN)nc2sc3CCCCc3c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H09 compound treatment 440.0 -810.0 -0.29 1600.0 724.0 0.56 0.1898 0.3033 3118048 ChemDiv3_002627 CN(C)CCC(=O)N1c2ccccc2Sc3ccc(cc13)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H10 compound treatment 600.0 -650.0 -0.23 600.0 -276.0 -0.21 -0.3129 -0.9991 1429742 ChemDiv3_002628 COC(CN1C(=O)C2C3CC(C=C3)C2C1=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H11 compound treatment 480.0 -770.0 -0.27 5880.0 5000.0 3.84 2.5232 0.6552 1351226 ChemDiv3_002629 COC(=O)c1ccc(cc1)N(Cc2ccccc2)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H12 compound treatment 560.0 -690.0 -0.24 640.0 -236.0 -0.18 -0.3013 -0.9891 3022477 ChemDiv3_002630 CC1(C)CC(=O)C=C(C1)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H13 compound treatment 4440.0 3190.0 1.13 320.0 -556.0 -0.43 0.4983 0.412 1715519 ChemDiv3_002631 CCc1cccc(C)c1NC(=O)c2ccc(cc2)C(=O)Nc3c(C)cccc3CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H14 compound treatment 2920.0 1670.0 0.59 440.0 -436.0 -0.33 0.1822 0.2677 3022478 ChemDiv3_002632 CSc1ccc(C=C2C(=O)OC3(CCCCC3)OC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H15 compound treatment 680.0 -570.0 -0.2 960.0 83.9 0.06 -0.0975 -0.4592 1124952 ChemDiv3_002633 Fc1ccc(NC(=O)C2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H16 compound treatment 720.0 -530.0 -0.19 720.0 -156.0 -0.12 -0.2177 -0.9764 1549958 ChemDiv3_002634 CCc1cc(=O)oc2c(C)c(OCC(=O)N)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H17 compound treatment 1040.0 -210.0 -0.07 520.0 -356.0 -0.27 -0.246 -0.8681 1176369 ChemDiv3_002635 CN(C)c1ncnc2c3cc(C)ccc3[nH]c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H18 compound treatment 1920.0 670.0 0.24 560.0 -316.0 -0.24 -0.0035 -0.0104 1448053 ChemDiv3_002636 CCCc1cc(=O)oc2cc(OC(C(=O)OCC)c3ccccc3)c(Cl)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H19 compound treatment 480.0 -770.0 -0.27 680.0 -196.0 -0.15 -0.2996 -0.9606 1482032 ChemDiv3_002637 O=C(CCN1C(=O)C2C3CC(C=C3)C2C1=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H20 compound treatment 560.0 -690.0 -0.24 1280.0 404.0 0.31 0.0462 0.1169 1430536 ChemDiv3_002638 COCn1c(COc2ccc3ccccc3c2)nc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H21 compound treatment 360.0 -890.0 -0.32 4360.0 3480.0 2.67 1.668 0.6193 3118049 ChemDiv3_002639 NC(=N)Nc1nc(c2ccccc2)c3ccccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H22 compound treatment 1000.0 -250.0 -0.09 880.0 3.87 0.0 -0.0606 -0.683 3118050 ChemDiv3_002640 COc1ccc(/C=N\CC2(CCCC2)c3ccccc3)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H23 mock treatment 560.0 -690.0 -0.24 680.0 -196.0 -0.15 -0.2796 -0.9728 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 H24 mock treatment 360.0 -890.0 -0.32 2360.0 1480.0 1.14 0.5823 0.4926 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I01 compound treatment 280.0 -970.0 -0.34 3320.0 2440.0 1.88 1.0834 0.5679 1577750 ChemDiv3_002641 CC(=C1C(=O)c2ccccc2C1=O)N3CCC(CC3)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I02 compound treatment 240.0 -1010.0 -0.36 2400.0 1520.0 1.17 0.5739 0.469 1416256 ChemDiv3_002642 Oc1ccc(cc1)c2nc3cc4ccccc4cc3nc2c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I03 compound treatment 3160.0 1910.0 0.68 2240.0 1360.0 1.05 1.2195 0.9778 3021773 ChemDiv3_002643 Cc1ccc(cc1C)N2NC(=O)/C(=C/C=C/c3ccco3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I04 compound treatment 920.0 -330.0 -0.12 400.0 -476.0 -0.37 -0.3412 -0.8891 3118051 ChemDiv3_002644 Oc1ccc(/N=c/2\scc(c3ccccc3)n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I05 compound treatment 360.0 -890.0 -0.32 960.0 83.9 0.06 -0.1777 -0.5515 1235164 ChemDiv3_002645 CC(C)CC(N1C(=O)c2ccccc2C1=O)C(=O)Nc3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I06 compound treatment 4000.0 2750.0 0.98 880.0 3.87 0.0 0.6919 0.7093 1162646 ChemDiv3_002646 Cc1ccc(cc1)C(OCC(C)(C)C[N+](C)(C)C)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I07 compound treatment 280.0 -970.0 -0.34 320.0 -556.0 -0.43 -0.5452 -0.9943 3118052 ChemDiv3_002647 CCN(CC)C(=O)n1cnc2cc(C)c(C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I08 compound treatment 200.0 -1050.0 -0.37 400.0 -476.0 -0.37 -0.5219 -1.0 1361112 ChemDiv3_002648 Cc1c(oc2ccccc12)C(=O)NC(=S)Nc3ccc(Br)cn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I09 compound treatment 400.0 -850.0 -0.3 640.0 -236.0 -0.18 -0.3414 -0.9704 1612002 ChemDiv3_002649 Cc1cc(=O)oc2cc(Oc3nc(C)nc4sc5CCCc5c34)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I10 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 1546280 ChemDiv3_002650 CCCCC1C(=O)NC(=S)NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I11 compound treatment 320.0 -930.0 -0.33 360.0 -516.0 -0.4 -0.5135 -0.9959 3021827 ChemDiv3_002651 CSc1ccc(cc1)c2cc(=O)c3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I12 compound treatment 760.0 -490.0 -0.17 240.0 -636.0 -0.49 -0.4682 -0.9033 1198111 ChemDiv3_002652 CC(=O)Oc1ccc(OC(=O)C)c(c1)S(=O)(=O)c2ccc(C)c(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I13 compound treatment 800.0 -450.0 -0.16 560.0 -316.0 -0.24 -0.2845 -0.9793 1525224 ChemDiv3_002653 OC(COc1ccccc1CC=C)Cn2c3ccccc3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I14 compound treatment 760.0 -490.0 -0.17 320.0 -556.0 -0.43 -0.4248 -0.9215 3118053 ChemDiv3_002654 COc1ccc(cc1)c2oc3ncn(CCO)c(=N)c3c2c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I15 compound treatment 360.0 -890.0 -0.32 440.0 -436.0 -0.33 -0.46 -0.9996 1531068 ChemDiv3_002655 COc1ccccc1C2C(=C(C)NC3=C2C(=O)CCC3)C(=O)Nc4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I16 compound treatment 1320.0 70.0 0.02 320.0 -556.0 -0.43 -0.2843 -0.6649 1597347 ChemDiv3_002656 CC(C)C1CC(C)(OC1=O)c2csc(Nc3ccc(C)cc3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I17 compound treatment 200.0 -1050.0 -0.37 400.0 -476.0 -0.37 -0.5219 -1.0 1510595 ChemDiv3_002657 S=c1n(CN2CCCCC2)cnn1CN3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I18 compound treatment 560.0 -690.0 -0.24 920.0 43.9 0.03 -0.1493 -0.6041 1725386 ChemDiv3_002658 CCNc1nc(NCC)nc(Oc2ccc(O)nn2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I19 compound treatment 520.0 -730.0 -0.26 280.0 -596.0 -0.46 -0.5067 -0.9636 3118054 ChemDiv3_002659 COC(=O)C/1=C(C)N(Cc2ccccc2)C(=O)\C1=C/c3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I20 compound treatment 3520.0 2270.0 0.81 240.0 -636.0 -0.49 0.2241 0.2379 1378167 ChemDiv3_002660 Cc1ccc(cc1)C(=O)CSc2nc(C)cc(C)c2C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I21 compound treatment 160.0 -1090.0 -0.39 840.0 -36.1 -0.03 -0.293 -0.7559 1016528 ChemDiv3_002661 C=CCN1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I22 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 3118055 ChemDiv3_002662 Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)/C=C/c3ccccc3)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I23 mock treatment 2600.0 1350.0 0.48 760.0 -116.0 -0.09 0.2756 0.5658 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 I24 mock treatment 280.0 -970.0 -0.34 360.0 -516.0 -0.4 -0.5235 -0.9975 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J01 compound treatment 240.0 -1010.0 -0.36 240.0 -636.0 -0.49 -0.5987 -0.9884 1742467 ChemDiv3_002663 Cc1cc(NC(=O)COc2ccccc2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J02 compound treatment 360.0 -890.0 -0.32 640.0 -236.0 -0.18 -0.3514 -0.9653 1321408 ChemDiv3_002664 CC(=CC(=O)CC(O)(c1ccccc1)c2ccccc2)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J03 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 1866882 ChemDiv3_002665 OC(CN1CCN(CC1)c2cccc(Cl)c2)Cn3c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J04 compound treatment 1160.0 -90.0 -0.03 400.0 -476.0 -0.37 -0.281 -0.766 3118056 ChemDiv3_002666 CC(C)(C)C1=NOC(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J05 compound treatment 200.0 -1050.0 -0.37 200.0 -676.0 -0.52 -0.6304 -0.9868 3118057 ChemDiv3_002667 C=CC[C@H]1Cc2ccccc2[C@H](CC=C)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J06 compound treatment 720.0 -530.0 -0.19 280.0 -596.0 -0.46 -0.4566 -0.9228 3118058 ChemDiv3_002668 CCOP1(=S)Oc2cc(Cl)ccc2C(O1)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J07 compound treatment 360.0 -890.0 -0.32 280.0 -596.0 -0.46 -0.5469 -0.9836 1177751 ChemDiv3_002669 COC(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J08 compound treatment 320.0 -930.0 -0.33 400.0 -476.0 -0.37 -0.4918 -0.9987 1503507 ChemDiv3_002670 CC1=NN(C(C1)C2=C(C)CCCC2(C)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J09 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 1550037 ChemDiv3_002671 O=C(NC1CCCCC1)N2c3ccccc3CCc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J10 compound treatment 240.0 -1010.0 -0.36 240.0 -636.0 -0.49 -0.5987 -0.9884 1126817 ChemDiv3_002672 CC(=O)N1N=C(C)CC1c2ccc(OCc3ccccc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J11 compound treatment 320.0 -930.0 -0.33 240.0 -636.0 -0.49 -0.5786 -0.9818 3118059 ChemDiv3_002673 Oc1ccc(NC(=O)CCCN2C(=O)/C(=C\c3cccs3)/SC2=S)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J12 compound treatment 240.0 -1010.0 -0.36 280.0 -596.0 -0.46 -0.577 -0.9927 3021891 ChemDiv3_002674 C/N=C\1/S/C(=C\c2ccc(cc2)N3Cc4ccccc4C3)/C(=O)N1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J13 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 1637905 ChemDiv3_002675 O=C1SCCC1NS(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J14 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 3021893 ChemDiv3_002676 Brc1ccc(C=C2C(=O)OC3(CCCC3)OC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J15 compound treatment 280.0 -970.0 -0.34 1400.0 524.0 0.4 0.0411 0.0776 1259786 ChemDiv3_002677 CC1CCCCN1C(=O)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J16 compound treatment 280.0 -970.0 -0.34 520.0 -356.0 -0.27 -0.4366 -0.9935 1345434 ChemDiv3_002678 CCCc1cc(=O)oc2c(C)c(OC(C)C(=O)O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J17 compound treatment 200.0 -1050.0 -0.37 1080.0 204.0 0.16 -0.1527 -0.378 1213781 ChemDiv3_002679 CCN(CC)c1ncnc2c3cc(C)ccc3[nH]c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J18 compound treatment 240.0 -1010.0 -0.36 720.0 -156.0 -0.12 -0.3381 -0.8949 1271531 ChemDiv3_002680 CCc1cc(=O)oc2cc(C)cc(OCC(=O)C(C)(C)C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J19 compound treatment 400.0 -850.0 -0.3 640.0 -236.0 -0.18 -0.3414 -0.9704 1605551 ChemDiv3_002681 C1C(Nc2ncnn2C1c3ccco3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J20 compound treatment 1320.0 70.0 0.02 360.0 -516.0 -0.4 -0.2626 -0.6615 1265661 ChemDiv3_002682 CSc1nc2-c3ccccc3CC4(CCCCC4)c2c(=O)n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J21 compound treatment 360.0 -890.0 -0.32 200.0 -676.0 -0.52 -0.5903 -0.9716 1627093 ChemDiv3_002683 CCc1ccc2nc(Nc3nc(=O)c4ccccc4[nH]3)nc(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J22 compound treatment 920.0 -330.0 -0.12 640.0 -236.0 -0.18 -0.211 -0.9776 3021946 ChemDiv3_002684 CC(C)(C)c1ccc(OCNC(=S)NC(=O)c2cncc(Br)c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J23 mock treatment 400.0 -850.0 -0.3 1000.0 124.0 0.1 -0.146 -0.4617 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 J24 mock treatment 200.0 -1050.0 -0.37 280.0 -596.0 -0.46 -0.587 -0.9948 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K01 compound treatment 1120.0 -130.0 -0.05 1120.0 244.0 0.19 0.0998 0.5175 1520253 ChemDiv3_002685 CC(=C1C(=O)c2ccccc2C1=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K02 compound treatment 2440.0 1190.0 0.42 760.0 -116.0 -0.09 0.2355 0.5457 1222073 ChemDiv3_002686 CC1CCC(CC1)C(=O)Nc2ccc(Oc3cccc(C)c3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K03 compound treatment 280.0 -970.0 -0.34 320.0 -556.0 -0.43 -0.5452 -0.9943 1782006 ChemDiv3_002687 C=CCN1C(=O)/C(=C\2/C(=O)Nc3ccccc23)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K04 compound treatment 840.0 -410.0 -0.15 1360.0 484.0 0.37 0.1598 0.4006 3118193 ChemDiv3_002688 CN(C)CCCn/1c(cs\c1=N/c2ccccc2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K05 compound treatment 280.0 -970.0 -0.34 480.0 -396.0 -0.3 -0.4584 -0.9981 3021950 ChemDiv3_002689 CCCc1cc(=O)[nH]c(SC)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K06 compound treatment 280.0 -970.0 -0.34 960.0 83.9 0.06 -0.1978 -0.565 1655049 ChemDiv3_002690 COc1ccc(cc1)C(C(=O)OCCN(C)C)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K07 compound treatment 600.0 -650.0 -0.23 1080.0 204.0 0.16 -0.0524 -0.1879 1734313 ChemDiv3_002691 CCOC(=O)c1c(NC(=O)CSc2cc(C)c3ccccc3n2)sc4CCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K08 compound treatment 440.0 -810.0 -0.29 560.0 -316.0 -0.24 -0.3748 -0.9965 3118194 ChemDiv3_002692 Cc1c(oc2ccccc12)C(=O)NC(=S)Nc3ccc(cc3)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K09 compound treatment 520.0 -730.0 -0.26 1920.0 1040.0 0.8 0.3836 0.4554 1227980 ChemDiv3_002693 CCOC(=O)c1cc(Oc2nc(C)nc3sc4CCCCc4c23)cc(c1)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K10 compound treatment 320.0 -930.0 -0.33 480.0 -396.0 -0.3 -0.4483 -0.9992 1073790 ChemDiv3_002694 CN1C(SC(=S)N(C)C1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K11 compound treatment 480.0 -770.0 -0.27 1320.0 444.0 0.34 0.0478 0.1095 3118195 ChemDiv3_002695 O=C(Nc1ncnc2sc3CCCc3c12)/C=C/c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K12 compound treatment 2240.0 990.0 0.35 920.0 43.9 0.03 0.2722 0.7714 1473300 ChemDiv3_002696 CC(=O)Oc1ccc(OC(=O)C)c(c1)S(=O)(=O)c2ccc(Cl)c(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K13 compound treatment 320.0 -930.0 -0.33 600.0 -276.0 -0.21 -0.3832 -0.9771 1258026 ChemDiv3_002697 Cc1cc(C)n(CC(O)CN2C(=O)NC(C)(C)C2=O)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K14 compound treatment 520.0 -730.0 -0.26 640.0 -236.0 -0.18 -0.3113 -0.9848 1715933 ChemDiv3_002698 C(c1nc2c3c4CCCCc4sc3ncn2n1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K15 compound treatment 1720.0 470.0 0.17 1120.0 244.0 0.19 0.2503 0.9983 1852555 ChemDiv3_002699 CC1=C(C(C2=C(CC(CC2=O)c3ccccc3)N1)c4ccc(F)cc4)C(=O)Nc5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K16 compound treatment 560.0 -690.0 -0.24 640.0 -236.0 -0.18 -0.3013 -0.9891 3118196 ChemDiv3_002700 CC(C)CCOCC1Cc2c(C)nn(C(=S)N)c2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K17 compound treatment 640.0 -610.0 -0.22 680.0 -196.0 -0.15 -0.2595 -0.9843 3022012 ChemDiv3_002701 COC(=O)C1=C(C)N/C(=C/c2ccc(Br)cc2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K18 compound treatment 920.0 -330.0 -0.12 480.0 -396.0 -0.3 -0.2978 -0.9139 3118197 ChemDiv3_002702 COc1ccc(cc1)C2=NN3COc4ccccc4C3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K19 compound treatment 320.0 -930.0 -0.33 640.0 -236.0 -0.18 -0.3615 -0.9602 3022016 ChemDiv3_002703 COC(=O)C1=C(C)N(/C(=C/c2cccs2)/C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K20 compound treatment 2280.0 1030.0 0.37 920.0 43.9 0.03 0.2822 0.769 1243002 ChemDiv3_002704 CCCSc1nc(C)c(cc1C#N)c2csc(n2)C(=C3CCCC3)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K21 compound treatment 1080.0 -170.0 -0.06 640.0 -236.0 -0.18 -0.1708 -0.8942 1275176 ChemDiv3_002705 O=C1C2C(C(C=CC2c3ccccc3)c4ccccc4)C(=O)N1C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K22 compound treatment 520.0 -730.0 -0.26 1160.0 284.0 0.22 -0.029 -0.0857 3022022 ChemDiv3_002706 NS(=O)(=O)c1ccc(CNC(=O)/C=C/c2ccc3OCOc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K23 mock treatment 520.0 -730.0 -0.26 1040.0 164.0 0.13 -0.0942 -0.327 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 K24 mock treatment 1840.0 590.0 0.21 800.0 -76.1 -0.06 0.1067 0.4909 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L01 compound treatment 880.0 -370.0 -0.13 320.0 -556.0 -0.43 -0.3947 -0.8837 3022024 ChemDiv3_002707 COc1ccc2[n+]([O-])c3CCCc3[n+]([O-])c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L02 compound treatment 520.0 -730.0 -0.26 720.0 -156.0 -0.12 -0.2679 -0.9387 1922669 ChemDiv3_002708 O/N=C\1/CC(O)(Oc2ccccc12)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L03 compound treatment 1960.0 710.0 0.25 760.0 -116.0 -0.09 0.1151 0.4306 3118198 ChemDiv3_002709 Clc1ccc(C(=O)CN2C3=NCCN3c4ccccc24)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L04 compound treatment 360.0 -890.0 -0.32 600.0 -276.0 -0.21 -0.3731 -0.9812 3118199 ChemDiv3_002710 Cc1c(n2cc(C(=O)O)c(=O)c3c(F)c(F)c(F)c(F)c23)c(=O)n(c4ccccc4)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L05 compound treatment 960.0 -290.0 -0.1 800.0 -76.1 -0.06 -0.1141 -0.9641 1356358 ChemDiv3_002711 Cc1ccc(cc1C)c2nnc(N3CCCCC3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L06 compound treatment 360.0 -890.0 -0.32 560.0 -316.0 -0.24 -0.3949 -0.9916 3022079 ChemDiv3_002712 COc1ccc(NC(=C(C#N)C#N)C(F)(F)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L07 compound treatment 480.0 -770.0 -0.27 880.0 3.87 0.0 -0.191 -0.6994 3118200 ChemDiv3_002713 COC(=O)Cn1c(CCS(=O)(=O)c2ccc(Cl)cc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L08 compound treatment 320.0 -930.0 -0.33 560.0 -316.0 -0.24 -0.4049 -0.9886 1315595 ChemDiv3_002714 CN(C)CCCN1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L09 compound treatment 920.0 -330.0 -0.12 5200.0 4320.0 3.32 2.2645 0.6817 3022082 ChemDiv3_002715 OCC1c2ccccc2-c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L10 compound treatment 560.0 -690.0 -0.24 640.0 -236.0 -0.18 -0.3013 -0.9891 3022084 ChemDiv3_002716 CC(C)C1NC(=NC2=C1CCCC2)S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L11 compound treatment 1160.0 -90.0 -0.03 720.0 -156.0 -0.12 -0.1073 -0.8653 3118201 ChemDiv3_002717 CC(N1C(=O)/C(=C/c2ccc(Cl)cc2)/SC1=S)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L12 compound treatment 640.0 -610.0 -0.22 680.0 -196.0 -0.15 -0.2595 -0.9843 1693076 ChemDiv3_002718 Cc1cccc(c1)n2c(N)cc(=O)[nH]c2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L13 compound treatment 720.0 -530.0 -0.19 640.0 -236.0 -0.18 -0.2611 -0.9998 1697919 ChemDiv3_002719 O=C(N1CCc2ccccc12)c3cccc(c3)C(=O)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L14 compound treatment 480.0 -770.0 -0.27 440.0 -436.0 -0.33 -0.4299 -0.9949 3118202 ChemDiv3_002720 NC1=NC(=O)CC(S1)C(=O)Nc2cccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L15 compound treatment 320.0 -930.0 -0.33 600.0 -276.0 -0.21 -0.3832 -0.9771 1548630 ChemDiv3_002721 O=C(Nc1cccnc1)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L16 compound treatment 600.0 -650.0 -0.23 1760.0 884.0 0.68 0.3168 0.442 1634226 ChemDiv3_002722 CCCCc1cc(=O)oc2cc(OCC(=O)N)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L17 compound treatment 360.0 -890.0 -0.32 920.0 43.9 0.03 -0.1994 -0.6281 3022089 ChemDiv3_002723 COc1ccc(/C=N/n2cnc3c4cc(F)ccc4[nH]c3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L18 compound treatment 880.0 -370.0 -0.13 480.0 -396.0 -0.3 -0.3079 -0.9294 1718796 ChemDiv3_002724 COc1ccc2c(c1)c(=O)oc3cc(O)ccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L19 compound treatment 360.0 -890.0 -0.32 520.0 -356.0 -0.27 -0.4166 -0.9974 1232639 ChemDiv3_002725 COc1ccc(CC(=O)NCC2COc3ccccc3O2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L20 compound treatment 520.0 -730.0 -0.26 520.0 -356.0 -0.27 -0.3764 -0.9996 1182221 ChemDiv3_002726 CC(C[N+](C)(C)C)OC(=O)C1(CCCC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L21 compound treatment 2080.0 830.0 0.29 440.0 -436.0 -0.33 -0.0286 -0.064 1251764 ChemDiv3_002727 COc1ccc(Nc2nc3ccccc3c(=O)s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L22 compound treatment 360.0 -890.0 -0.32 4640.0 3760.0 2.89 1.82 0.6261 1678958 ChemDiv3_002728 Nc1cc(N)nc(SCCC(=O)O)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L23 mock treatment 4400.0 3150.0 1.12 1160.0 284.0 0.22 0.9443 0.8294 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 L24 mock treatment 640.0 -610.0 -0.22 920.0 43.9 0.03 -0.1292 -0.5899 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M01 compound treatment 160.0 -1090.0 -0.39 320.0 -556.0 -0.43 -0.5753 -0.9988 3022148 ChemDiv3_002729 CCOC(=O)Cc1c(C)[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M02 compound treatment 240.0 -1010.0 -0.36 360.0 -516.0 -0.4 -0.5335 -0.9987 1694723 ChemDiv3_002730 CN(C(=O)c1ccccc1)c2ccc(OCC(=O)NC3CCS(=O)(=O)C3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M03 compound treatment 960.0 -290.0 -0.1 560.0 -316.0 -0.24 -0.2444 -0.927 3022151 ChemDiv3_002731 CCOC(=O)c1ccc(CSc2nnc(C)[nH]2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M04 compound treatment 360.0 -890.0 -0.32 3960.0 3080.0 2.37 1.4509 0.6074 3118336 ChemDiv3_002732 Cc1cs/c(=N\c2c(C)cc(C)cc2C)/n1Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M05 compound treatment 320.0 -930.0 -0.33 360.0 -516.0 -0.4 -0.5135 -0.9959 1606325 ChemDiv3_002733 CC(C)CN(CC(C)C)Cc1c(O)ccc2c3ccccc3c(=O)oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M06 compound treatment 360.0 -890.0 -0.32 320.0 -556.0 -0.43 -0.5252 -0.989 3118337 ChemDiv3_002734 COc1ccc(/C=C\2/C(=O)c3ccc(cc3C2=O)C(=O)O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M07 compound treatment 400.0 -850.0 -0.3 2040.0 1160.0 0.89 0.4186 0.4439 2083900 ChemDiv3_002735 c1nnc2c3c(csc3ncn12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M08 compound treatment 3440.0 2190.0 0.78 3080.0 2200.0 1.69 1.7457 0.9377 3118338 ChemDiv3_002736 Cc1ccc(cc1)S(=O)(=O)/N=C(\N2CCOCC2)/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M09 compound treatment 1520.0 270.0 0.1 5680.0 4800.0 3.69 2.6756 0.7252 1710664 ChemDiv3_002737 Fc1ccc(cc1)C(=O)N2CCCCC(Sc3nnc4sc5ccccc5n34)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M10 compound treatment 400.0 -850.0 -0.3 680.0 -196.0 -0.15 -0.3197 -0.9485 1699392 ChemDiv3_002738 CCOc1ccc(cc1)C(=O)SC2=NCCS2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M11 compound treatment 200.0 -1050.0 -0.37 760.0 -116.0 -0.09 -0.3264 -0.8523 1284546 ChemDiv3_002739 O=C(Nc1ncnc2oc(c(c3ccccc3)c12)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M12 compound treatment 440.0 -810.0 -0.29 800.0 -76.1 -0.06 -0.2445 -0.8339 3022508 ChemDiv3_002740 CCN(CC)/C=N/c1sc2CCCCCc2c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M13 compound treatment 560.0 -690.0 -0.24 320.0 -556.0 -0.43 -0.475 -0.9651 1622887 ChemDiv3_002741 Cc1ccc(cc1)N(CC(O)Cn2c3ccccc3c4ccccc24)S(=O)(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M14 compound treatment 600.0 -650.0 -0.23 3200.0 2320.0 1.78 1.0985 0.6106 3022512 ChemDiv3_002742 Clc1ccc(c2ncnn2c3ccccc3)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M15 compound treatment 280.0 -970.0 -0.34 800.0 -76.1 -0.06 -0.2846 -0.8155 3118339 ChemDiv3_002743 CC1=C(C(C2=C(CCCC2=O)N1)c3ccccc3)C(=O)Nc4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M16 compound treatment 3960.0 2710.0 0.96 5920.0 5040.0 3.87 3.4179 0.8567 1137028 ChemDiv3_002744 COc1ccccc1Nc2nc(cs2)C3(C)CCC(=O)O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M17 compound treatment 360.0 -890.0 -0.32 960.0 83.9 0.06 -0.1777 -0.5515 3118340 ChemDiv3_002745 COC(=O)C/1=C(C)N(CC(C)C)C(=O)\C1=C/c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M18 compound treatment 1480.0 230.0 0.08 800.0 -76.1 -0.06 0.0164 0.1631 3022519 ChemDiv3_002746 CC(=O)N1C(CC(=Nc2ccccc12)c3ccc(C)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M19 compound treatment 520.0 -730.0 -0.26 840.0 -36.1 -0.03 -0.2027 -0.7784 1581924 ChemDiv3_002747 CNC(=O)CN(Cc1ccccc1)S(=O)(=O)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M20 compound treatment 2600.0 1350.0 0.48 960.0 83.9 0.06 0.3842 0.795 1383371 ChemDiv3_002748 O=C(Cc1ccccc1)NCCc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M21 compound treatment 600.0 -650.0 -0.23 2040.0 1160.0 0.89 0.4688 0.508 3118341 ChemDiv3_002749 O=C1C2C(C(C=CC2c3ccccc3)c4ccccc4)C(=O)N1c5nccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M22 compound treatment 400.0 -850.0 -0.3 920.0 43.9 0.03 -0.1894 -0.6242 1556611 ChemDiv3_002750 CC(Oc1ccccc1)C(=O)NC2CCSC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M23 mock treatment 240.0 -1010.0 -0.36 2360.0 1480.0 1.14 0.5522 0.4624 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 M24 mock treatment 1360.0 110.0 0.04 1600.0 724.0 0.56 0.4206 0.7549 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N01 compound treatment 1560.0 310.0 0.11 720.0 -156.0 -0.12 -0.007 -0.043 3022523 ChemDiv3_002751 COC(=O)c1c(O)[n+]([O-])c2cc(Cl)c(Cl)cc2[n+]1[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N02 compound treatment 920.0 -330.0 -0.12 920.0 43.9 0.03 -0.059 -0.484 1922259 ChemDiv3_002752 OC(CC(=O)c1ccccc1)(c2ccccc2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N03 compound treatment 880.0 -370.0 -0.13 280.0 -596.0 -0.46 -0.4164 -0.8746 1390281 ChemDiv3_002753 Cc1cccc(Nc2nnc(c3ccc(C)c(c3)S(=O)(=O)NCCO)c4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N04 compound treatment 1600.0 350.0 0.12 440.0 -436.0 -0.33 -0.149 -0.4171 1601095 ChemDiv3_002754 CC(SC(=S)N1CCCC1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N05 compound treatment 320.0 -930.0 -0.33 800.0 -76.1 -0.06 -0.2746 -0.8196 3021727 ChemDiv3_002755 O=C/1/C(=C/c2ccccn2)/CN(Cc3ccccc3)C\C1=C\c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N06 compound treatment 400.0 -850.0 -0.3 880.0 3.87 0.0 -0.2111 -0.7001 3118342 ChemDiv3_002756 COC(=O)C(F)(F)Sc1c(C)[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N07 compound treatment 1840.0 590.0 0.21 1480.0 604.0 0.46 0.4758 0.9354 3021729 ChemDiv3_002757 Cc1ccc(SCC(=O)Nc2nncs2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N08 compound treatment 560.0 -690.0 -0.24 1040.0 164.0 0.13 -0.0841 -0.3057 1320903 ChemDiv3_002758 C(Oc1c2CCCCc2nc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N09 compound treatment 440.0 -810.0 -0.29 2800.0 1920.0 1.48 0.8412 0.5591 2080577 ChemDiv3_002759 Cc1[nH]c(=O)[nH]c(=O)c1/C=C/C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N10 compound treatment 920.0 -330.0 -0.12 320.0 -556.0 -0.43 -0.3847 -0.8689 3021733 ChemDiv3_002760 Oc1cccc(NC(=O)CN2C(=O)S/C(=C\C=C\c3ccccc3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N11 compound treatment 480.0 -770.0 -0.27 240.0 -636.0 -0.49 -0.5385 -0.9623 3118344 ChemDiv3_002761 O=C(COc1ccccc1)NC(=S)Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N12 compound treatment 3240.0 1990.0 0.71 920.0 43.9 0.03 0.523 0.74 3021735 ChemDiv3_002762 O=C/1ON=C(\C1=C\c2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N13 compound treatment 1280.0 30.0 0.01 320.0 -556.0 -0.43 -0.2944 -0.6893 1207240 ChemDiv3_002763 COC(=O)c1cc(NC(=O)c2cccc(Cl)c2)cc(c1)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N14 compound treatment 280.0 -970.0 -0.34 560.0 -316.0 -0.24 -0.4149 -0.9854 3118345 ChemDiv3_002764 Cc1cc(C)c2nc(NC3=NC(CC(=O)N3)c4ccccc4)nc(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N15 compound treatment 1320.0 70.0 0.02 680.0 -196.0 -0.15 -0.0889 -0.5826 3021737 ChemDiv3_002765 CC1CCCCN1C(=O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N16 compound treatment 680.0 -570.0 -0.2 400.0 -476.0 -0.37 -0.4015 -0.961 1353095 ChemDiv3_002766 CCCCc1cc(=O)oc2cc(OCC(=O)c3ccc(F)cc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N17 compound treatment 240.0 -1010.0 -0.36 440.0 -436.0 -0.33 -0.4901 -0.9994 3021779 ChemDiv3_002767 COc1ccc(/C=N/n2cnc3c4cc(OC)ccc4[nH]c3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N18 compound treatment 280.0 -970.0 -0.34 2360.0 1480.0 1.14 0.5622 0.4724 1231038 ChemDiv3_002768 CC(=CCOc1cc(C)cc2oc(=O)cc(c3ccccc3)c12)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N19 compound treatment 1040.0 -210.0 -0.07 1360.0 484.0 0.37 0.21 0.5543 3021783 ChemDiv3_002769 CCOC(=O)c1ccc(Oc2cc(C)nc(SC)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N20 compound treatment 1040.0 -210.0 -0.07 640.0 -236.0 -0.18 -0.1809 -0.9228 3118346 ChemDiv3_002770 COC(=O)C/1=C(C)N(C2CCCCC2)C(=O)\C1=C/c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N21 compound treatment 3040.0 1790.0 0.63 560.0 -316.0 -0.24 0.2774 0.4081 1457554 ChemDiv3_002771 CC1CC(N(C(=O)c2ccc(Cl)cc2)c3ccccc3)c4ccccc4N1C(=O)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N22 compound treatment 360.0 -890.0 -0.32 1000.0 124.0 0.1 -0.156 -0.4731 1383040 ChemDiv3_002772 CC1(C)CC(=O)C2=C(C1)OC(C(=C2N)C#N)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N23 mock treatment 1960.0 710.0 0.25 920.0 43.9 0.03 0.2019 0.7946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 N24 mock treatment 360.0 -890.0 -0.32 800.0 -76.1 -0.06 -0.2646 -0.824 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O01 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 3118347 ChemDiv3_002773 COc1ccc(/C=C/2\CCc3ccccc3C2=O)cc1CN4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O02 compound treatment 1080.0 -170.0 -0.06 240.0 -636.0 -0.49 -0.388 -0.7884 1056982 ChemDiv3_002774 C=CCn1c(=O)c2ccccc2[nH]c1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O03 compound treatment 160.0 -1090.0 -0.39 240.0 -636.0 -0.49 -0.6187 -0.9933 3021791 ChemDiv3_002775 COc1ccc(N/C=C/C(=O)c2ccc3OCOc3c2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O04 compound treatment 240.0 -1010.0 -0.36 200.0 -676.0 -0.52 -0.6204 -0.9836 3118348 ChemDiv3_002776 O=c1[nH]c(SCc2nnc(Nc3ccccc3)s2)nc4sc5CCCc5c14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O05 compound treatment 200.0 -1050.0 -0.37 240.0 -636.0 -0.49 -0.6087 -0.9911 3021793 ChemDiv3_002777 CN(C)C(=O)/C(=C\c1ccccc1)/NC(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O06 compound treatment 520.0 -730.0 -0.26 120.0 -756.0 -0.58 -0.5936 -0.9338 3021837 ChemDiv3_002778 COc1ccc(cc1)N2C(=O)/C(=C\c3ccc(cc3)C(C)C)/C(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O07 compound treatment 240.0 -1010.0 -0.36 360.0 -516.0 -0.4 -0.5335 -0.9987 3118349 ChemDiv3_002779 Cc1nc(SCC(=O)Nc2ccc(cc2)c3ccccc3)c4c5CCCc5sc4n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O08 compound treatment 320.0 -930.0 -0.33 1120.0 244.0 0.19 -0.1009 -0.266 3118350 ChemDiv3_002780 CN(C1CC(CCC1O)C=C)C(=S)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O09 compound treatment 200.0 -1050.0 -0.37 320.0 -556.0 -0.43 -0.5653 -0.9977 3021841 ChemDiv3_002781 COC(=O)c1c(C)[nH]c(C(=O)CSc2nnc3cc(C)c4ccccc4n23)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O10 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 3021843 ChemDiv3_002782 CSc1nnc2nc(C)cc(C)n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O11 compound treatment 280.0 -970.0 -0.34 2520.0 1640.0 1.26 0.6491 0.4962 1724528 ChemDiv3_002783 COc1ccc(cc1)c2cc(O)c3c(C)oc(C)c3c(=O)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O12 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 3021847 ChemDiv3_002784 N#Cc1c(/N=C/N2CCCC2)sc3CCCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O13 compound treatment 360.0 -890.0 -0.32 240.0 -636.0 -0.49 -0.5686 -0.9777 1183146 ChemDiv3_002785 COc1ccccc1N(CC(O)CN2CCOCC2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O14 compound treatment 320.0 -930.0 -0.33 360.0 -516.0 -0.4 -0.5135 -0.9959 3118480 ChemDiv3_002786 CCc1ccc(cc1)c2ncnn2c3cccc(Cl)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O15 compound treatment 320.0 -930.0 -0.33 200.0 -676.0 -0.52 -0.6003 -0.9761 1452275 ChemDiv3_002787 CC1=C(C(C2=C(CC(C)(C)CC2=O)N1)c3ccsc3)C(=O)Nc4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O16 compound treatment 240.0 -1010.0 -0.36 240.0 -636.0 -0.49 -0.5987 -0.9884 1482352 ChemDiv3_002788 Cc1ccccc1n2c(SCCc3ccccc3)nc4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O17 compound treatment 320.0 -930.0 -0.33 160.0 -716.0 -0.55 -0.622 -0.9702 3118481 ChemDiv3_002789 COC(=O)C1=C(C)N/C(=C/c2cccc3ccccc23)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O18 compound treatment 360.0 -890.0 -0.32 280.0 -596.0 -0.46 -0.5469 -0.9836 1554516 ChemDiv3_002790 Nc1c(sc2nc3CCCCc3cc12)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O19 compound treatment 280.0 -970.0 -0.34 400.0 -476.0 -0.37 -0.5018 -0.9995 3021899 ChemDiv3_002791 COC(=O)C/1=C(C)N(C(=O)\C1=C/c2ccco2)c3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O20 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 3118482 ChemDiv3_002792 CC(C)N1CCN(Cc2ccccc2C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O21 compound treatment 280.0 -970.0 -0.34 280.0 -596.0 -0.46 -0.5669 -0.9901 3021901 ChemDiv3_002793 COc1ccc(/C=N/CC2OCCc3ccccc23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O22 compound treatment 400.0 -850.0 -0.3 240.0 -636.0 -0.49 -0.5585 -0.9731 1628838 ChemDiv3_002794 O=C(CN1C(=O)c2ccccc2C1=O)Nc3ccccc3C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O23 mock treatment 320.0 -930.0 -0.33 240.0 -636.0 -0.49 -0.5786 -0.9818 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 O24 mock treatment 320.0 -930.0 -0.33 200.0 -676.0 -0.52 -0.6003 -0.9761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P01 compound treatment 240.0 -1010.0 -0.36 160.0 -716.0 -0.55 -0.6421 -0.9785 3021904 ChemDiv3_002795 CC(=O)ON(Cc1c(C)no[n+]1[O-])Cc2c(C)no[n+]2[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P02 compound treatment 280.0 -970.0 -0.34 240.0 -636.0 -0.49 -0.5886 -0.9853 3118483 ChemDiv3_002796 COc1ccc2C(=O)CC(O)(Oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P03 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 1283255 ChemDiv3_002797 Cc1ccc(cc1S(=O)(=O)NC(C)(C)C)c2nnc(Nc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P04 compound treatment 240.0 -1010.0 -0.36 280.0 -596.0 -0.46 -0.577 -0.9927 1048670 ChemDiv3_002798 CC(SC(=S)N1CCOCC1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P05 compound treatment 240.0 -1010.0 -0.36 320.0 -556.0 -0.43 -0.5553 -0.9962 1197963 ChemDiv3_002799 C=CCn1c(SCC(=O)NCCc2ccccc2)nc3sc4CCCCc4c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P06 compound treatment 360.0 -890.0 -0.32 280.0 -596.0 -0.46 -0.5469 -0.9836 3118484 ChemDiv3_002800 Cc1cc[n+](CC2OCc3ccccc3CO2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P07 compound treatment 160.0 -1090.0 -0.39 280.0 -596.0 -0.46 -0.597 -0.9965 1171875 ChemDiv3_002801 CCc1nn(c2ccccc2)c3nc(c4ccccc4O)c5cc(OC)c(OC)cc5c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P08 compound treatment 240.0 -1010.0 -0.36 240.0 -636.0 -0.49 -0.5987 -0.9884 1487683 ChemDiv3_002802 O=C(CC1CCCCCCCCCCC1)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P09 compound treatment 200.0 -1050.0 -0.37 280.0 -596.0 -0.46 -0.587 -0.9948 1780370 ChemDiv3_002803 OC(=O)CCn1cc(I)c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P10 compound treatment 280.0 -970.0 -0.34 320.0 -556.0 -0.43 -0.5452 -0.9943 1734593 ChemDiv3_002804 Oc1cccc(NC(=O)CC2SC(=O)N(CN3CCOCC3)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P11 compound treatment 200.0 -1050.0 -0.37 120.0 -756.0 -0.58 -0.6739 -0.977 1328370 ChemDiv3_002805 CCSc1nc2sc-3c(CCc4ccccc34)c2c(=O)n1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P12 compound treatment 720.0 -530.0 -0.19 200.0 -676.0 -0.52 -0.5 -0.9056 3021746 ChemDiv3_002806 CN(C)c1ccc(/C=C/2\C(=NOC2=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P13 compound treatment 2520.0 1270.0 0.45 240.0 -636.0 -0.49 -0.0268 -0.0403 1517507 ChemDiv3_002807 COC(=O)c1ccccc1NC(=O)c2cc(OC)cc(OC)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P14 compound treatment 240.0 -1010.0 -0.36 240.0 -636.0 -0.49 -0.5987 -0.9884 3118485 ChemDiv3_002808 CCN(CC)C(=O)Oc1c(Br)cc(Br)c2ccc(C)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P15 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 1715468 ChemDiv3_002809 CN(C)c1ccc(cc1)c2nc3c(n2C)c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P16 compound treatment 240.0 -1010.0 -0.36 200.0 -676.0 -0.52 -0.6204 -0.9836 1216146 ChemDiv3_002810 Cc1c(Cc2ccccc2)c(=O)oc3cc(OC4CCCCC4=O)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P17 compound treatment 440.0 -810.0 -0.29 280.0 -596.0 -0.46 -0.5268 -0.9749 1162913 ChemDiv3_002811 CCOCc1cnc(C)nc1NCC(=O)c2c(C)[nH]c3cc(C)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P18 compound treatment 320.0 -930.0 -0.33 320.0 -556.0 -0.43 -0.5352 -0.9919 3118486 ChemDiv3_002812 Cc1cc(OCc2cccc(c2)C(F)(F)F)c3c4CCCc4c(=O)oc3c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P19 compound treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 1641373 ChemDiv3_002813 Cn1nnc2c(sc3nc(N4CCOCC4)c5CCCCc5c32)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P20 compound treatment 2680.0 1430.0 0.51 400.0 -476.0 -0.37 0.1002 0.1603 1204217 ChemDiv3_002814 COC1(COc2ccccc2O1)C(=O)NN 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P21 compound treatment 2520.0 1270.0 0.45 3920.0 3040.0 2.34 1.971 0.8282 1515951 ChemDiv3_002815 Cc1ccc2N(C(=O)c3ccncc3)C(C)(C)c4ssc(=S)c4-c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P22 compound treatment 2280.0 1030.0 0.37 2000.0 1120.0 0.86 0.8685 0.9269 3118487 ChemDiv3_002816 Clc1ccc2nc(cc(c3ccccc3)c2c1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P23 mock treatment 2560.0 1310.0 0.46 880.0 3.87 0.0 0.3307 0.7116 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2008 P24 mock treatment 320.0 -930.0 -0.33 280.0 -596.0 -0.46 -0.5569 -0.9871 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A01 compound treatment 9960.0 8150.0 2.89 280.0 -501.0 -0.38 1.7722 0.6076 3021807 ChemDiv3_002817 CC(=O)Nc1nc(NC(=O)C)n(n1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A02 compound treatment 7040.0 5230.0 1.86 480.0 -301.0 -0.23 1.1483 0.6142 3118488 ChemDiv3_002818 Fc1cccc(c1)N2C(=O)NC(=O)/C(=C\c3cn(CC#N)c4ccccc34)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A03 compound treatment 2480.0 670.0 0.24 800.0 18.6 0.01 0.1781 0.7482 3021809 ChemDiv3_002819 COc1cccc(/C=N/n2cnc3sc4CCCCc4c3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A04 compound treatment 7440.0 5630.0 2.0 3440.0 2660.0 2.04 2.8555 0.9999 3118489 ChemDiv3_002820 CCCOC(=O)c1cc(ccc1Cl)c2ccc(/C=C\3/C(=C(C#N)C(=O)N(CCO)C3=O)C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A05 compound treatment 320.0 -1490.0 -0.53 360.0 -421.0 -0.32 -0.6025 -0.9723 1538576 ChemDiv3_002821 CCc1ccc(NC(=O)C(C)N2C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A06 compound treatment 320.0 -1490.0 -0.53 360.0 -421.0 -0.32 -0.6025 -0.9723 1182782 ChemDiv3_002822 CC[N+]1(CCC2CC1)CC2C(=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A07 compound treatment 360.0 -1450.0 -0.51 200.0 -581.0 -0.45 -0.6794 -0.9975 1424746 ChemDiv3_002823 CCOC(=O)N1CCN(CC(O)COCc2ccc(Cl)cc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A08 compound treatment 280.0 -1530.0 -0.54 4280.0 3500.0 2.69 1.5154 0.553 3118490 ChemDiv3_002824 CN(C)/C=N/c1ncc2c3ccccc3[nH]c2c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A09 compound treatment 280.0 -1530.0 -0.54 280.0 -501.0 -0.38 -0.656 -0.9858 1484360 ChemDiv3_002825 CCCS(=O)(=O)N1CCN(Cc2ccco2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A10 compound treatment 240.0 -1570.0 -0.56 200.0 -581.0 -0.45 -0.7095 -0.994 3118491 ChemDiv3_002826 N/C(=C(\C=C\1/Nc2ccccc2C1=O)/C#N)/NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A11 compound treatment 320.0 -1490.0 -0.53 320.0 -461.0 -0.35 -0.6242 -0.9811 3021864 ChemDiv3_002827 CN1C(=O)N(C)C(=O)C(=Cc2cn(CC(=O)NCc3ccco3)c4ccccc24)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A12 compound treatment 200.0 -1610.0 -0.57 280.0 -501.0 -0.38 -0.6761 -0.9816 1374824 ChemDiv3_002828 Nc1c(C#N)c2CCCn2c1C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A13 compound treatment 280.0 -1530.0 -0.54 5040.0 4260.0 3.27 1.928 0.5818 1492318 ChemDiv3_002829 CC(C)C(N1C(=O)c2ccccc2C1=O)C(=O)Nc3nc(c(C)s3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A14 compound treatment 160.0 -1650.0 -0.59 440.0 -341.0 -0.26 -0.5992 -0.9344 1193090 ChemDiv3_002830 CC1(C)CC(=O)c2cc(C#N)c(SCc3ccccc3)nc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A15 compound treatment 600.0 -1210.0 -0.43 200.0 -581.0 -0.45 -0.6192 -0.9998 1464685 ChemDiv3_002831 Cc1ccc(CNC(=O)CN(Cc2ccccc2)S(=O)(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A16 compound treatment 240.0 -1570.0 -0.56 2680.0 1900.0 1.46 0.6368 0.4081 3118492 ChemDiv3_002832 CCOc1ccc(CSc2nnc(CC)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A17 compound treatment 160.0 -1650.0 -0.59 440.0 -341.0 -0.26 -0.5992 -0.9344 1729504 ChemDiv3_002833 CCCC(=O)Nn1cnc2-c3ccccc3CC4(CCCC4)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A18 compound treatment 240.0 -1570.0 -0.56 560.0 -221.0 -0.17 -0.514 -0.8827 3021919 ChemDiv3_002834 CN(C)c1ccc(/C=C/C=C\2/C(=O)NC(=O)N(C2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A19 compound treatment 240.0 -1570.0 -0.56 440.0 -341.0 -0.26 -0.5792 -0.9409 3118493 ChemDiv3_002835 Cc1ccc(/N=C\c2cc3ccccc3nc2O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A20 compound treatment 3840.0 2030.0 0.72 6160.0 5380.0 4.13 3.429 0.8181 3118617 ChemDiv3_002836 CC1CN(Cc2c(O)ccc3c(=O)c(Oc4cc(C)cc(C)c4)c(oc23)C(F)(F)F)CC(C)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A21 compound treatment 920.0 -890.0 -0.32 320.0 -461.0 -0.35 -0.4737 -0.9984 3021923 ChemDiv3_002837 COc1ccc(/C=C\2/C(=N)N3N=C(Cc4ccccc4)SC3=NC2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A22 compound treatment 320.0 -1490.0 -0.53 880.0 98.6 0.08 -0.3202 -0.5998 3118618 ChemDiv3_002838 COc1ccc2nc(N3CCCCC3)c(/C=C/4\SC(=S)NC4=O)cc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A23 mock treatment 320.0 -1490.0 -0.53 560.0 -221.0 -0.17 -0.494 -0.8896 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 A24 mock treatment 280.0 -1530.0 -0.54 5160.0 4380.0 3.36 1.9932 0.5854 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B01 compound treatment 360.0 -1450.0 -0.51 200.0 -581.0 -0.45 -0.6794 -0.9975 3021926 ChemDiv3_002839 CCN1C(=O)/C(=C/C=C\2/CCCN2C)/N(C1=S)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B02 compound treatment 240.0 -1570.0 -0.56 320.0 -461.0 -0.35 -0.6443 -0.9761 1353210 ChemDiv3_002840 CC(C)(SC(=S)N1CCCCCC1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B03 compound treatment 480.0 -1330.0 -0.47 1840.0 1060.0 0.81 0.241 0.2565 1173431 ChemDiv3_002841 O=C(N(Cc1ccccc1)Cc2ccccc2)c3cc4ccccc4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B04 compound treatment 400.0 -1410.0 -0.5 280.0 -501.0 -0.38 -0.6259 -0.9916 3118619 ChemDiv3_002842 Cc1nc(SCC(=O)O)c2oc3ccccc3c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B05 compound treatment 360.0 -1450.0 -0.51 480.0 -301.0 -0.23 -0.5274 -0.935 1513490 ChemDiv3_002843 COc1ccc(cc1OC)C(=O)NC(=S)Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B06 compound treatment 360.0 -1450.0 -0.51 320.0 -461.0 -0.35 -0.6142 -0.9834 3022740 ChemDiv3_002844 FC(F)(F)c1cccc(/N=C\2/NC(=O)/C(=C\3/C(=O)Nc4ccccc34)/S2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B07 compound treatment 400.0 -1410.0 -0.5 280.0 -501.0 -0.38 -0.6259 -0.9916 3022741 ChemDiv3_002845 CCCSc1nc(=O)cc(C)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B08 compound treatment 240.0 -1570.0 -0.56 320.0 -461.0 -0.35 -0.6443 -0.9761 1155824 ChemDiv3_002846 CC1CN(CC(C)O1)c2nc(nc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B09 compound treatment 240.0 -1570.0 -0.56 320.0 -461.0 -0.35 -0.6443 -0.9761 1210251 ChemDiv3_002847 COc1ccc(cc1OC)C2SCC(=O)N2CCCN(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B10 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3022742 ChemDiv3_002848 Cc1ccc(cc1)S(=O)(=O)N2Cc3ccccc3C[C@H]2C(=O)Nc4cccc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B11 compound treatment 320.0 -1490.0 -0.53 280.0 -501.0 -0.38 -0.646 -0.9879 1728781 ChemDiv3_002849 Cc1ccc(cc1)n2c(NN)nc3sc4CCCCc4c3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B12 compound treatment 400.0 -1410.0 -0.5 240.0 -541.0 -0.42 -0.6476 -0.9958 3118620 ChemDiv3_002850 CN(C)C(=O)Oc1cccnc1C[N+](C)(C)COC(=O)C2CC3CC4CC3CC2C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B13 compound treatment 200.0 -1610.0 -0.57 5640.0 4860.0 3.73 2.2337 0.5919 1660469 ChemDiv3_002851 COc1ccccc1NC(=O)c2ccc3C(=O)N(CC4CCCO4)C(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B14 compound treatment 400.0 -1410.0 -0.5 440.0 -341.0 -0.26 -0.539 -0.9545 1602268 ChemDiv3_002852 O=S(=O)(c1nc(Cc2ccccc2)oc1N3CCOCC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B15 compound treatment 280.0 -1530.0 -0.54 320.0 -461.0 -0.35 -0.6343 -0.9786 3022743 ChemDiv3_002853 CN(C)c1ccc(/C=C/2\C(=C(C#N)C(=O)NC2=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B16 compound treatment 320.0 -1490.0 -0.53 560.0 -221.0 -0.17 -0.494 -0.8896 1569371 ChemDiv3_002854 Clc1ccc(CS(=O)(=O)CCSc2nc3CCCCc3cc2C#N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B17 compound treatment 480.0 -1330.0 -0.47 280.0 -501.0 -0.38 -0.6058 -0.9949 1481179 ChemDiv3_002855 C=CCNc1oc(nc1C#N)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B18 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 3118621 ChemDiv3_002856 CCS(=O)CCSc1nc(cc(c1C#N)c2ccccc2)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B19 compound treatment 320.0 -1490.0 -0.53 320.0 -461.0 -0.35 -0.6242 -0.9811 1278163 ChemDiv3_002857 CCN(CC)S(=O)(=O)c1ccc(cc1)c2cn3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B20 compound treatment 560.0 -1250.0 -0.44 480.0 -301.0 -0.23 -0.4772 -0.954 3118622 ChemDiv3_002858 Nc1c(sc2nc(cc(c3ccccc3)c12)c4cccs4)S(=O)Cc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B21 compound treatment 640.0 -1170.0 -0.42 320.0 -461.0 -0.35 -0.544 -0.9969 3022744 ChemDiv3_002859 Brc1ccc(cc1)C(=O)NCC(=O)NC2=NCCS2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B22 compound treatment 760.0 -1050.0 -0.37 600.0 -181.0 -0.14 -0.3619 -0.91 3118623 ChemDiv3_002860 Cc1cc(C)nc(SCCS(=O)Cc2ccc(Cl)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B23 mock treatment 3280.0 1470.0 0.52 680.0 -101.0 -0.08 0.3137 0.5949 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 B24 mock treatment 280.0 -1530.0 -0.54 4360.0 3580.0 2.75 1.5589 0.5567 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C01 compound treatment 200.0 -1610.0 -0.57 640.0 -141.0 -0.11 -0.4806 -0.8267 3118624 ChemDiv3_002861 CC1(C)C2CCC1(C)c3nc(SCC(=O)Nc4cccc(c4)C(F)(F)F)nnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C02 compound treatment 240.0 -1570.0 -0.56 760.0 -21.4 -0.02 -0.4055 -0.7277 3022745 ChemDiv3_002862 CN(C)c1ccc(/C=C/C=C2C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C03 compound treatment 280.0 -1530.0 -0.54 200.0 -581.0 -0.45 -0.6994 -0.9953 3022746 ChemDiv3_002863 Cc1ccc(/C=N/n2cnc3sc4CCCCc4c3c2=O)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C04 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3118625 ChemDiv3_002864 CCOC(=O)C/C(=N/c1ncn(c1C(=O)c2ccccc2)c3ccc(OC)cc3)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C05 compound treatment 240.0 -1570.0 -0.56 320.0 -461.0 -0.35 -0.6443 -0.9761 3022747 ChemDiv3_002865 N=c1[cH-][n+](CC2(CC3CC4CC(C3)C2)C4)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C06 compound treatment 520.0 -1290.0 -0.46 280.0 -501.0 -0.38 -0.5958 -0.9963 3118626 ChemDiv3_002866 O=C(OC1CN2CCC1CC2)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C07 compound treatment 6320.0 4510.0 1.6 280.0 -501.0 -0.38 0.8591 0.5221 3118627 ChemDiv3_002867 Cc1sc2nc(SC/C=C/c3ccccc3)nc(N)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C08 compound treatment 400.0 -1410.0 -0.5 200.0 -581.0 -0.45 -0.6693 -0.9984 3022748 ChemDiv3_002868 NC(=S)CN1CCCC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C09 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 1579280 ChemDiv3_002869 O=C1NC(Nc2sc3CCCCc3c12)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C10 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3022749 ChemDiv3_002870 N/C(=C(\C=C\1/Nc2ccccc2C1=O)/C#N)/N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C11 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3118628 ChemDiv3_002871 CN1C(=O)N(C)C(=O)C(=Cc2cn(CC(=O)N3CCCC3)c4ccccc24)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C12 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3022750 ChemDiv3_002872 CCOC(=O)c1c(/N=C/N(C)C)c(C#N)c2CCCn12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C13 compound treatment 240.0 -1570.0 -0.56 360.0 -421.0 -0.32 -0.6226 -0.9666 1221349 ChemDiv3_002873 CCN1CCN(CC1)c2nc(nc3ccccc23)c4ccc(cc4)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C14 compound treatment 480.0 -1330.0 -0.47 280.0 -501.0 -0.38 -0.6058 -0.9949 1161473 ChemDiv3_002874 CC1(C)CC(=O)c2cc3c(N)c(sc3nc2C1)C(=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C15 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 1250012 ChemDiv3_002875 CCOc1ccc(NC(=O)CN(Cc2ccccc2)S(=O)(=O)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C16 compound treatment 240.0 -1570.0 -0.56 280.0 -501.0 -0.38 -0.666 -0.9837 3022751 ChemDiv3_002876 CCc1nnc(SCC(=O)O)n1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C17 compound treatment 280.0 -1530.0 -0.54 280.0 -501.0 -0.38 -0.656 -0.9858 1283511 ChemDiv3_002877 COc1ccccc1NC(=O)CC(c2ccccc2)c3ccc(C)cc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C18 compound treatment 240.0 -1570.0 -0.56 320.0 -461.0 -0.35 -0.6443 -0.9761 3022752 ChemDiv3_002878 CN1C(=O)S/C(=C\c2cc(Cl)c(OCC(=O)O)c(Cl)c2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C19 compound treatment 240.0 -1570.0 -0.56 280.0 -501.0 -0.38 -0.666 -0.9837 3118629 ChemDiv3_002879 CC/1=NN(C(=O)\C1=C/c2cc3ccccc3nc2O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C20 compound treatment 320.0 -1490.0 -0.53 280.0 -501.0 -0.38 -0.646 -0.9879 1430355 ChemDiv3_002880 COc1ccccc1c2coc3cc(OCc4ccc(C)cc4)ccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C21 compound treatment 240.0 -1570.0 -0.56 440.0 -341.0 -0.26 -0.5792 -0.9409 1530511 ChemDiv3_002881 Cc1ccc(o1)C(O)c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C22 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 3022753 ChemDiv3_002882 CCOC(=O)c1c(C)[nH]c(/C(=N\O)/C)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C23 mock treatment 480.0 -1330.0 -0.47 280.0 -501.0 -0.38 -0.6058 -0.9949 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 C24 mock treatment 240.0 -1570.0 -0.56 400.0 -381.0 -0.29 -0.6009 -0.9549 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D01 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 3118630 ChemDiv3_002883 CCn1/c(=C/C=C/2\SC(=S)N(CC=C)C2=O)/c3cccc4cccc1c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D02 compound treatment 360.0 -1450.0 -0.51 320.0 -461.0 -0.35 -0.6142 -0.9834 1561724 ChemDiv3_002884 OC(=O)CCSC(=S)N1CCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D03 compound treatment 520.0 -1290.0 -0.46 240.0 -541.0 -0.42 -0.6175 -0.9988 1649229 ChemDiv3_002885 COc1ccc2oc(=N)c(cc2c1)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D04 compound treatment 280.0 -1530.0 -0.54 280.0 -501.0 -0.38 -0.656 -0.9858 3118631 ChemDiv3_002886 C(/N=C/c1c2ccccc2cc3ccccc13)c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D05 compound treatment 440.0 -1370.0 -0.49 320.0 -461.0 -0.35 -0.5941 -0.9879 3118632 ChemDiv3_002887 COC(=O)C1=CN(C=C(C1c2ccc(F)cc2)C(=O)OC)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D06 compound treatment 21600.0 19800.0 7.02 5800.0 5020.0 3.85 7.6886 0.9601 3022754 ChemDiv3_002888 Cc1ccc(/C=C\2/SC(=O)NC2=S)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D07 compound treatment 2680.0 870.0 0.31 280.0 -501.0 -0.38 -0.054 -0.1094 3022755 ChemDiv3_002889 COc1ccccc1OCCSc2nnnn2C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D08 compound treatment 3000.0 1190.0 0.42 400.0 -381.0 -0.29 0.0914 0.178 1631453 ChemDiv3_002890 C=CCN(CC=C)c1nc(nc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D09 compound treatment 360.0 -1450.0 -0.51 320.0 -461.0 -0.35 -0.6142 -0.9834 1641006 ChemDiv3_002891 COc1ccc(CC(CC(=O)O)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D10 compound treatment 280.0 -1530.0 -0.54 320.0 -461.0 -0.35 -0.6343 -0.9786 3118633 ChemDiv3_002892 Fc1ccccc1Cn2cc(/C=C\3/NC(=O)NC3=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D11 compound treatment 200.0 -1610.0 -0.57 400.0 -381.0 -0.29 -0.6109 -0.9518 1703384 ChemDiv3_002893 COc1ccc(OCCn2c(nc3ccccc3c2=O)c4ccc(Cl)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D12 compound treatment 280.0 -1530.0 -0.54 320.0 -461.0 -0.35 -0.6343 -0.9786 3022756 ChemDiv3_002894 CN(C)Cc1ccc(C)cc1OC(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D13 compound treatment 360.0 -1450.0 -0.51 440.0 -341.0 -0.26 -0.5491 -0.9511 3022757 ChemDiv3_002895 COc1ccc(cc1)c2noc(n2)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D14 compound treatment 360.0 -1450.0 -0.51 240.0 -541.0 -0.42 -0.6576 -0.9944 3118634 ChemDiv3_002896 O=C(NCSC1=NCCS1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D15 compound treatment 280.0 -1530.0 -0.54 280.0 -501.0 -0.38 -0.656 -0.9858 3118770 ChemDiv3_002897 COC(=O)c1ccccc1c2ccc(/C=C\3/C(=C(C#N)C(=O)N(C)C3=O)C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D16 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 1455196 ChemDiv3_002898 CC(C)(C)c1ccc(cc1)S(=O)(=O)CCSc2nc3CCCCc3cc2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D17 compound treatment 360.0 -1450.0 -0.51 240.0 -541.0 -0.42 -0.6576 -0.9944 3118771 ChemDiv3_002899 CN(C)CCCN1C(C(=C(O)C1=O)C(=O)c2ccc(Br)cc2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D18 compound treatment 400.0 -1410.0 -0.5 320.0 -461.0 -0.35 -0.6042 -0.9857 1280705 ChemDiv3_002900 COc1ccc(cc1)c2cc(c(C#N)c(n2)S(=O)Cc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D19 compound treatment 240.0 -1570.0 -0.56 200.0 -581.0 -0.45 -0.7095 -0.994 3118772 ChemDiv3_002901 CC(C)Oc1ccc(cc1)c2nn(cc2/C=C(\C#N)/S(=O)(=O)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D20 compound treatment 360.0 -1450.0 -0.51 240.0 -541.0 -0.42 -0.6576 -0.9944 3022758 ChemDiv3_002902 Cc1cc(C)c(C#N)c(SC2CCCCC2=O)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D21 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3118773 ChemDiv3_002903 CCOC(=O)c1ccc(NC(=O)CNC(=O)C2(CC3CC4CC(C3)C2)C4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D22 compound treatment 160.0 -1650.0 -0.59 240.0 -541.0 -0.42 -0.7078 -0.9859 3022759 ChemDiv3_002904 O=S(CCSc1nc2ccccc2s1)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D23 mock treatment 400.0 -1410.0 -0.5 160.0 -621.0 -0.48 -0.691 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 D24 mock treatment 4040.0 2230.0 0.79 280.0 -501.0 -0.38 0.2872 0.3264 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E01 compound treatment 2200.0 390.0 0.14 520.0 -261.0 -0.2 -0.0441 -0.1809 1223104 ChemDiv3_002905 CC(C)(C)c1ccc(Oc2ccc(NC(=O)CCCC(=O)O)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E02 compound treatment 1000.0 -810.0 -0.29 400.0 -381.0 -0.29 -0.4102 -1.0 1544828 ChemDiv3_002906 CCCCC(C(=O)N)C1=NC(C)(C)Cc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E03 compound treatment 1400.0 -410.0 -0.15 920.0 139.0 0.11 -0.0276 -0.1533 3022760 ChemDiv3_002907 Cc1[nH]c2ccccc2c1/C=N/n3cnc4sc5CCCCc5c4c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E04 compound treatment 400.0 -1410.0 -0.5 800.0 18.6 0.01 -0.3436 -0.6867 1386791 ChemDiv3_002908 CCOC(=O)c1sc(C)c2c(=O)n(Cc3ccccc3)c(C)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E05 compound treatment 1080.0 -730.0 -0.26 1400.0 619.0 0.47 0.1527 0.2823 3118774 ChemDiv3_002909 Cc1sc2nc(SCC(=O)c3ccc(O)c(O)c3)[nH]c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E06 compound treatment 5280.0 3470.0 1.23 4840.0 4060.0 3.12 3.0737 0.9175 1921600 ChemDiv3_002910 Oc1ccccc1N/C=C\2/C(=O)CNC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E07 compound treatment 2440.0 630.0 0.22 640.0 -141.0 -0.11 0.0813 0.327 1551909 ChemDiv3_002911 Cn1c(=O)[nH]c(=O)c2n(Cc3ccc(F)cc3)cnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E08 compound treatment 640.0 -1170.0 -0.42 1040.0 259.0 0.2 -0.1531 -0.3328 3118775 ChemDiv3_002912 COc1ccc(/N=C\2/CCc3ccccc3N2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E09 compound treatment 2920.0 1110.0 0.39 1760.0 979.0 0.75 0.8097 0.9546 3022761 ChemDiv3_002913 NC(=O)Cn1cc(/C=C\2/C(=O)NC(=O)N(C3CCCCC3)C2=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E10 compound treatment 1600.0 -210.0 -0.07 480.0 -301.0 -0.23 -0.2163 -0.8898 3118776 ChemDiv3_002914 CC(=O)N1/C(=C\NCc2ccccc2)/C(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E11 compound treatment 600.0 -1210.0 -0.43 960.0 179.0 0.14 -0.2066 -0.4585 1288465 ChemDiv3_002915 CCCC(=O)Nc1ccc(cc1)c2nc3cc(ccc3o2)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E12 compound treatment 1960.0 150.0 0.05 360.0 -421.0 -0.32 -0.1911 -0.583 1138540 ChemDiv3_002916 Cc1ccc(c(C)c1)S(=O)(=O)N2C=Cc3ccccc3C2c4c[nH]c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E13 compound treatment 1520.0 -290.0 -0.1 600.0 -181.0 -0.14 -0.1712 -0.9889 3118777 ChemDiv3_002917 CCc1ccc(/N=C/2\NC(=N)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E14 compound treatment 3280.0 1470.0 0.52 400.0 -381.0 -0.29 0.1617 0.2703 1308638 ChemDiv3_002918 Cc1cccc(NC(=O)CSc2nc3CCCCc3c(c4ccco4)c2C#N)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E15 compound treatment 1880.0 70.0 0.02 840.0 58.6 0.04 0.0494 0.9608 1250243 ChemDiv3_002919 COc1ccc(cc1OC)S(=O)(=O)N(CCc2ccccc2)CC(=O)Nc3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E16 compound treatment 440.0 -1370.0 -0.49 8880.0 8100.0 6.22 4.0527 0.6499 3118778 ChemDiv3_002920 COC(=O)c1ccc(CSc2nncn2N)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E17 compound treatment 5800.0 3990.0 1.42 920.0 139.0 0.11 1.0761 0.7581 1661835 ChemDiv3_002921 Nn1c(Cc2ccccc2)nc3sc4CCCCc4c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E18 compound treatment 4000.0 2190.0 0.78 360.0 -421.0 -0.32 0.3206 0.3809 3022812 ChemDiv3_002922 CN1C(=O)S/C(=C\c2ccc(o2)c3ccc(C(=O)O)c(Cl)c3)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E19 compound treatment 1880.0 70.0 0.02 840.0 58.6 0.04 0.0494 0.9608 3022813 ChemDiv3_002923 CC(=O)N/1C(=S)NC(=O)\C1=C\c2cc3cccc(C)c3nc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E20 compound treatment 2840.0 1030.0 0.37 880.0 98.6 0.08 0.3119 0.8358 3022814 ChemDiv3_002924 COC(=O)C1=C(Nc2cccc(c2)C(F)(F)F)SCC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E21 compound treatment 880.0 -930.0 -0.33 760.0 -21.4 -0.02 -0.2449 -0.7414 3022815 ChemDiv3_002925 CC(C)CC1=NN2C(=NC(=O)/C(=C\c3cccs3)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E22 compound treatment 3160.0 1350.0 0.48 880.0 98.6 0.08 0.3921 0.8088 3022816 ChemDiv3_002926 CCN1C(=O)/C(=C/2\C=Cc3ccccc3N2CC)/OC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E23 mock treatment 680.0 -1130.0 -0.4 1040.0 259.0 0.2 -0.1431 -0.3199 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 E24 mock treatment 6920.0 5110.0 1.81 2320.0 1540.0 1.18 2.117 0.9785 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F01 compound treatment 2920.0 1110.0 0.39 920.0 139.0 0.11 0.3537 0.8671 3118779 ChemDiv3_002927 CCN1/C(=C\C=C\2/N(C)C(=S)N(C)C2=O)/Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F02 compound treatment 720.0 -1090.0 -0.39 520.0 -261.0 -0.2 -0.4153 -0.9534 3022817 ChemDiv3_002928 Oc1ccccc1C2=NNC(O)(C2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F03 compound treatment 1160.0 -650.0 -0.23 680.0 -101.0 -0.08 -0.2181 -0.8962 3118780 ChemDiv3_002929 NC(=O)c/1cc2ccccc2o\c1=N/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F04 compound treatment 5600.0 3790.0 1.34 9200.0 8420.0 6.46 5.5208 0.8363 1710580 ChemDiv3_002930 OC(=O)c1c(oc2ccc(OCc3ccc(Cl)cc3)cc12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F05 compound treatment 440.0 -1370.0 -0.49 600.0 -181.0 -0.14 -0.4421 -0.8746 3022818 ChemDiv3_002931 COC(=O)C(N1C=C(C(C(=C1)C(=O)OC)c2ccc(F)cc2)C(=O)OC)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F06 compound treatment 3960.0 2150.0 0.76 600.0 -181.0 -0.14 0.4408 0.5686 3118781 ChemDiv3_002932 CC/1=NN(C(=O)\C1=C\c2ccc(o2)c3ccc4C(=O)NC(=O)c4c3)c5ccc(Br)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F07 compound treatment 800.0 -1010.0 -0.36 1360.0 579.0 0.44 0.0607 0.1064 3022819 ChemDiv3_002933 CCOc1ccc(OCCSc2nnnn2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F08 compound treatment 1240.0 -570.0 -0.2 760.0 -21.4 -0.02 -0.1546 -0.7621 3118782 ChemDiv3_002934 CCc1ccc(OCCCC(=O)Oc2ccc3c(c2)oc(=O)c4ccccc43)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F09 compound treatment 1400.0 -410.0 -0.15 800.0 18.6 0.01 -0.0928 -0.6347 1717369 ChemDiv3_002935 Cc1ccc(cc1)N2C(=O)CC(Cc3ccccc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F10 compound treatment 1240.0 -570.0 -0.2 7920.0 7140.0 5.48 3.7323 0.6806 3118783 ChemDiv3_002936 COc1ccc(/C=C\2/NC(=O)NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F11 compound treatment 400.0 -1410.0 -0.5 7160.0 6380.0 4.9 3.109 0.6316 3118784 ChemDiv3_002937 Cc1ccc(cc1)N2C3=C(C(C4=C2CC(C)(C)CC4=O)c5cnn(C)c5)C(=O)CC(C)(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F12 compound treatment 3760.0 1950.0 0.69 3160.0 2380.0 1.83 1.7804 0.9117 3022820 ChemDiv3_002938 CN(C)c1ccc(cc1)C2OCC3(CO2)SC4=NCN(C)CN4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F13 compound treatment 1880.0 70.0 0.02 1120.0 339.0 0.26 0.2014 0.7711 3118785 ChemDiv3_002939 COc1ccc(cc1)c2noc(n2)c3ccc(Cl)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F14 compound treatment 1480.0 -330.0 -0.12 11080.0 10300.0 7.91 5.5079 0.6966 1273850 ChemDiv3_002940 Fc1cnc(Nc2cccc(Br)c2)nc1Nc3cccc(Br)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F15 compound treatment 520.0 -1290.0 -0.46 1120.0 339.0 0.26 -0.1398 -0.2656 3118786 ChemDiv3_002941 COc1cc(/C=C(/NC(=O)c2ccccc2)\C(=O)O)ccc1OCC(=C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F16 compound treatment 2360.0 550.0 0.2 1000.0 219.0 0.17 0.2566 0.9972 1650847 ChemDiv3_002942 Nc1c(sc2nc3CCCCc3cc12)S(=O)(=O)Cc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F17 compound treatment 640.0 -1170.0 -0.42 7160.0 6380.0 4.9 3.1692 0.6449 3118787 ChemDiv3_002943 OC(=O)CN1C(=O)/C(=C\2/C(=O)N(CC=C)c3ccc(Br)cc23)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F18 compound treatment 3560.0 1750.0 0.62 1080.0 299.0 0.23 0.6011 0.9083 1236421 ChemDiv3_002944 CCCCS(=O)CSc1nc(cc(c1C#N)c2ccccc2)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F19 compound treatment 960.0 -850.0 -0.3 760.0 -21.4 -0.02 -0.2248 -0.7446 1355414 ChemDiv3_002945 Cc1ccc2nc(cn2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F20 compound treatment 7720.0 5910.0 2.1 3800.0 3020.0 2.32 3.1211 0.9988 3118788 ChemDiv3_002946 OC(CSc1nc(cc(c1C#N)c2ccccc2)c3ccccc3)CS(=O)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F21 compound treatment 1280.0 -530.0 -0.19 2520.0 1740.0 1.33 0.8109 0.6016 1183876 ChemDiv3_002947 COC(=O)C(C)NC(=O)C1(CC2(C)CC3(C)CC(C)(C2)C1)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F22 compound treatment 1400.0 -410.0 -0.15 1920.0 1140.0 0.87 0.5152 0.5815 3118789 ChemDiv3_002948 CC(C)(C)c1ccc(cc1)S(=O)(=O)CCSc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F23 mock treatment 1480.0 -330.0 -0.12 6200.0 5420.0 4.16 2.8587 0.6869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 F24 mock treatment 1560.0 -250.0 -0.09 880.0 98.6 0.08 -0.0092 -0.0789 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G01 compound treatment 1000.0 -810.0 -0.29 1880.0 1100.0 0.84 0.3932 0.4413 1222574 ChemDiv3_002949 CCSc1nc2-c3ccccc3CC4(CCCC4)c2c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G02 compound treatment 1600.0 -210.0 -0.07 320.0 -461.0 -0.35 -0.3032 -0.8375 3118790 ChemDiv3_002950 CC1(C)Cc2ccccc2CN1C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G03 compound treatment 6560.0 4750.0 1.69 440.0 -341.0 -0.26 1.0062 0.59 3022821 ChemDiv3_002951 COCc1cc(C)nc(N)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G04 compound treatment 1760.0 -50.0 -0.02 360.0 -421.0 -0.32 -0.2413 -0.7448 1491781 ChemDiv3_002952 COc1ccc(cc1)c2c3CCCc3nc4c(C#N)c(C)n(c5ccccc5)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G05 compound treatment 1400.0 -410.0 -0.15 1760.0 979.0 0.75 0.4284 0.5598 3022822 ChemDiv3_002953 Clc1ccc(cc1)[n+]2[cH-]c(=N)on2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G06 compound treatment 480.0 -1330.0 -0.47 440.0 -341.0 -0.26 -0.519 -0.9615 1921290 ChemDiv3_002954 O=C/1CNC(=O)\C1=C/Nc2ccc(cc2)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G07 compound treatment 600.0 -1210.0 -0.43 920.0 139.0 0.11 -0.2283 -0.5162 1518514 ChemDiv3_002955 COc1ccc(cc1)C(=O)CSc2nc3n(C)c(=O)n(C)c(=O)c3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G08 compound treatment 1120.0 -690.0 -0.24 560.0 -221.0 -0.17 -0.2933 -0.9841 3022823 ChemDiv3_002956 NC(=O)/C(=C/1\CCc2ccccc2N1)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G09 compound treatment 520.0 -1290.0 -0.46 1160.0 379.0 0.29 -0.1181 -0.2178 3118928 ChemDiv3_002957 Cc1cc(ccc1/C=C\2/C(=O)NC(=O)N(C3CCCCC3)C2=O)N4Cc5ccccc5C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G10 compound treatment 480.0 -1330.0 -0.47 920.0 139.0 0.11 -0.2584 -0.5343 3022824 ChemDiv3_002958 O=C1/C(=C/N2CCCCC2)/Nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G11 compound treatment 960.0 -850.0 -0.3 480.0 -301.0 -0.23 -0.3768 -0.9915 3118929 ChemDiv3_002959 CCOC(=O)c1ccc(cc1)c2ccc(/C=c\3/sc4nc5c(C)c(C)ccc5n4c3=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G12 compound treatment 1120.0 -690.0 -0.24 680.0 -101.0 -0.08 -0.2281 -0.8882 1387158 ChemDiv3_002960 CN1CCN(CC1)C(=O)c2cc3c(ccc4ccccc43)oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G13 compound treatment 1840.0 30.0 0.01 880.0 98.6 0.08 0.061 0.7987 1788002 ChemDiv3_002961 Cc1cc(C(=O)OCC(=O)N2c3ccccc3Sc4ccccc24)c5ccccc5n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G14 compound treatment 480.0 -1330.0 -0.47 7800.0 7020.0 5.39 3.4765 0.6427 1462003 ChemDiv3_002962 Cc1cccc(NC(=O)CSC2=C(C#N)C(C3=C(CCCC3=O)N2)c4ccco4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G15 compound treatment 720.0 -1090.0 -0.39 600.0 -181.0 -0.14 -0.3719 -0.9049 3022825 ChemDiv3_002963 COC(=O)C1=C(C)N(/C(=C/c2ccco2)/C1=O)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G16 compound treatment 440.0 -1370.0 -0.49 440.0 -341.0 -0.26 -0.529 -0.958 1443214 ChemDiv3_002964 COc1ccc(cc1)c2cc(C(=O)N)c3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G17 compound treatment 680.0 -1130.0 -0.4 760.0 -21.4 -0.02 -0.2951 -0.7355 3118930 ChemDiv3_002965 COc1ccc(cc1)C2=Nc3ccccc3N=C(C2)c4ccc5ccccc5c4O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G18 compound treatment 600.0 -1210.0 -0.43 440.0 -341.0 -0.26 -0.4889 -0.972 3022826 ChemDiv3_002966 COC(=O)C/1=C(C)N(Cc2cccnc2)C(=O)\C1=C/c3ccccc3C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G19 compound treatment 480.0 -1330.0 -0.47 360.0 -421.0 -0.32 -0.5624 -0.9831 1271973 ChemDiv3_002967 CCc1ccc(CN2CCN(Cc3ccc(CC)cc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G20 compound treatment 1560.0 -250.0 -0.09 920.0 139.0 0.11 0.0125 0.0904 3118931 ChemDiv3_002968 COC(=O)C1=C(Nc2ccccc2)S/C(=C\c3ccc(O)cc3)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G21 compound treatment 680.0 -1130.0 -0.4 1200.0 419.0 0.32 -0.0562 -0.1094 3022827 ChemDiv3_002969 CC1=NN2C(=NC(=O)/C(=C\c3cn(CCOc4c(C)cccc4C)c5ccccc35)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G22 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 1923007 ChemDiv3_002970 CCN1/C(=C/C(=S)CC)/Sc2ccc(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G23 mock treatment 600.0 -1210.0 -0.43 440.0 -341.0 -0.26 -0.4889 -0.972 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 G24 mock treatment 400.0 -1410.0 -0.5 1040.0 259.0 0.2 -0.2133 -0.3964 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H01 compound treatment 400.0 -1410.0 -0.5 880.0 98.6 0.08 -0.3002 -0.5934 3118932 ChemDiv3_002971 CCN1C(=O)/C(=C/C=C\2/Sc3cc(NC(=O)C)ccc3N2CC)/N(C1=S)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H02 compound treatment 1280.0 -530.0 -0.19 480.0 -301.0 -0.23 -0.2966 -0.9947 3022829 ChemDiv3_002972 OC1(CC(=NO1)c2ccc(F)cc2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H03 compound treatment 1760.0 -50.0 -0.02 720.0 -61.4 -0.05 -0.0459 -0.9108 1421390 ChemDiv3_002973 CCOc1ccc(cc1)S(=O)(=O)n2cnc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H04 compound treatment 1920.0 110.0 0.04 760.0 -21.4 -0.02 0.016 0.3769 1922573 ChemDiv3_002974 CCc1cc2c(=O)c(c3nc4ccccc4s3)c(oc2cc1O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H05 compound treatment 1520.0 -290.0 -0.1 1040.0 259.0 0.2 0.0676 0.3025 1453753 ChemDiv3_002975 Clc1ccc(cc1)C2CC(=O)Nc3ncnn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H06 compound treatment 920.0 -890.0 -0.32 600.0 -181.0 -0.14 -0.3217 -0.9324 3118933 ChemDiv3_002976 Nc1nnnn1/N=C\C=C\c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H07 compound treatment 640.0 -1170.0 -0.42 600.0 -181.0 -0.14 -0.392 -0.8953 1013278 ChemDiv3_002977 OC(=O)CSc1nc2ccc(Br)cc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H08 compound treatment 720.0 -1090.0 -0.39 600.0 -181.0 -0.14 -0.3719 -0.9049 1282681 ChemDiv3_002978 COc1ccc2c(=O)c(Oc3cc(C)ccc3C)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H09 compound treatment 9520.0 7710.0 2.74 2640.0 1860.0 1.43 2.9429 0.954 1608087 ChemDiv3_002979 COc1ccc(cc1)N2C(=O)CC(Cc3ccccc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H10 compound treatment 880.0 -930.0 -0.33 640.0 -141.0 -0.11 -0.3101 -0.8927 3118934 ChemDiv3_002980 Cc1ccc(NC(=O)Cn2cc(/C=C\3/NC(=O)NC3=O)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H11 compound treatment 5520.0 3710.0 1.32 1600.0 819.0 0.63 1.375 0.9428 1375560 ChemDiv3_002981 Fc1cccc(c1)C2Nc3ccccc3C(=O)N2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H12 compound treatment 640.0 -1170.0 -0.42 320.0 -461.0 -0.35 -0.544 -0.9969 3118935 ChemDiv3_002982 OCC1(CO)SC(=NC1=O)Nc2ccc(cc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H13 compound treatment 2320.0 510.0 0.18 360.0 -421.0 -0.32 -0.1008 -0.2721 3022830 ChemDiv3_002983 CCOc1cc(/C=C/2\C(=NOC2=O)C)ccc1OC(=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H14 compound treatment 520.0 -1290.0 -0.46 880.0 98.6 0.08 -0.2701 -0.5823 3118936 ChemDiv3_002984 Cc1cc(C)c(C#N)c(SCCS(=O)(=O)Cc2ccc(Cl)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H15 compound treatment 5560.0 3750.0 1.33 2200.0 1420.0 1.09 1.7107 0.9951 3022831 ChemDiv3_002985 CCCn/1c(cs\c1=N/c2ccccc2)c3ccc(cc3)S(=O)(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H16 compound treatment 3640.0 1830.0 0.65 720.0 -61.4 -0.05 0.4257 0.654 1522547 ChemDiv3_002986 CC(C)(C)c1ccc(cc1)S(=O)c2sc3nc4CCCCc4cc3c2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H17 compound treatment 7040.0 5230.0 1.86 400.0 -381.0 -0.29 1.1048 0.5882 3118937 ChemDiv3_002987 Brc1ccc(/C=C(\C(=O)NCc2cccnc2)/S(=O)(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H18 compound treatment 20320.0 18500.0 6.57 2360.0 1580.0 1.21 5.5001 0.8237 3022832 ChemDiv3_002988 COc1ccc(cc1)c2cc(c(C#N)c(SCS(=O)Cc3ccccc3)n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H19 compound treatment 600.0 -1210.0 -0.43 560.0 -221.0 -0.17 -0.4237 -0.9178 1156911 ChemDiv3_002989 Cc1ccc(cc1)c2cn3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H20 compound treatment 480.0 -1330.0 -0.47 1200.0 419.0 0.32 -0.1064 -0.1864 1343150 ChemDiv3_002990 COc1ccc(cc1)c2cc(c(C#N)c(SC3CCCCC3O)n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H21 compound treatment 800.0 -1010.0 -0.36 1200.0 419.0 0.32 -0.0261 -0.0543 3022833 ChemDiv3_002991 CC1(CC2(C)CC3(C)C1)CC(C2)(C3)C(=O)NC4=NCCS4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H22 compound treatment 2240.0 430.0 0.15 800.0 18.6 0.01 0.1179 0.7698 3118938 ChemDiv3_002992 O=S(=O)(CCSc1nc2ccccc2s1)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H23 mock treatment 960.0 -850.0 -0.3 680.0 -101.0 -0.08 -0.2683 -0.8615 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 H24 mock treatment 520.0 -1290.0 -0.46 440.0 -341.0 -0.26 -0.5089 -0.965 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I01 compound treatment 240.0 -1570.0 -0.56 2080.0 1300.0 1.0 0.3111 0.2724 3022834 ChemDiv3_002993 OC(=O)Cn1cc(Br)c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I02 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3118939 ChemDiv3_002994 CCN(CC)c1ccc(C=C2C(=O)c3ccccc3C2=O)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I03 compound treatment 1360.0 -450.0 -0.16 280.0 -501.0 -0.38 -0.3851 -0.924 1923199 ChemDiv3_002995 CC1(C)CC(=O)C(=C(N)NC(=O)c2ccccc2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I04 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 3022835 ChemDiv3_002996 COc1ccc(cc1)n2cnc3nc(C)c(C(=O)/C=C/N(C)C)c(c4ccccc4)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I05 compound treatment 360.0 -1450.0 -0.51 320.0 -461.0 -0.35 -0.6142 -0.9834 3118940 ChemDiv3_002997 Cc1nnc(SCC(=O)c2c[nH]c3ccccc23)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I06 compound treatment 160.0 -1650.0 -0.59 280.0 -501.0 -0.38 -0.6861 -0.9793 1921203 ChemDiv3_002998 CCOc1ccc(N/C=C\2/C(=O)CNC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I07 compound treatment 280.0 -1530.0 -0.54 320.0 -461.0 -0.35 -0.6343 -0.9786 1430050 ChemDiv3_002999 NNc1ncnc2c3ccccc3oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I08 compound treatment 3720.0 1910.0 0.68 240.0 -541.0 -0.42 0.1852 0.233 3118941 ChemDiv3_003000 COc1ccc(/N=C/2\CCCN2CC(=O)N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I09 compound treatment 400.0 -1410.0 -0.5 800.0 18.6 0.01 -0.3436 -0.6867 1183787 ChemDiv3_003001 CCSc1nc2ccccc2n1CC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I10 compound treatment 240.0 -1570.0 -0.56 360.0 -421.0 -0.32 -0.6226 -0.9666 3022885 ChemDiv3_003002 CC(=O)N1/C(=C\Nc2ccccc2)/C(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I11 compound treatment 400.0 -1410.0 -0.5 280.0 -501.0 -0.38 -0.6259 -0.9916 1236436 ChemDiv3_003003 OC1(CC(=O)c2ccc3ccccc3c2)C(=O)Nc4ccccc41 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I12 compound treatment 3800.0 1990.0 0.71 360.0 -421.0 -0.32 0.2704 0.3482 1699598 ChemDiv3_003004 CCOC(=O)N1CCN(CC1)C(=O)c2cc3c(ccc4ccccc43)oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I13 compound treatment 360.0 -1450.0 -0.51 320.0 -461.0 -0.35 -0.6142 -0.9834 3022886 ChemDiv3_003005 Cn1c(n[nH]c1=S)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I14 compound treatment 360.0 -1450.0 -0.51 400.0 -381.0 -0.29 -0.5708 -0.9643 3022887 ChemDiv3_003006 NC(=O)c1ccc(N/C=C(\C#N)/c2nc(cs2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I15 compound treatment 1320.0 -490.0 -0.17 760.0 -21.4 -0.02 -0.1345 -0.7706 3022888 ChemDiv3_003007 COC(=O)C/1=C(C)N(Cc2ccc(C)cc2)C(=O)\C1=C/c3ccccc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I16 compound treatment 440.0 -1370.0 -0.49 200.0 -581.0 -0.45 -0.6593 -0.9991 1457003 ChemDiv3_003008 COc1ccc(cc1)S(=O)(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I17 compound treatment 680.0 -1130.0 -0.4 480.0 -301.0 -0.23 -0.4471 -0.9659 1093189 ChemDiv3_003009 CC(=O)NC1CC(C)(C)NC(C)(C)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I18 compound treatment 480.0 -1330.0 -0.47 920.0 139.0 0.11 -0.2584 -0.5343 3022889 ChemDiv3_003010 COC(=O)C1=C(C)N/C(=C/c2ccc(CNS(=O)(=O)c3ccccc3)o2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I19 compound treatment 1640.0 -170.0 -0.06 280.0 -501.0 -0.38 -0.3148 -0.808 3118942 ChemDiv3_003011 O=c/1n2CN(CN=c2s\c1=C/c3ccccn3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I20 compound treatment 240.0 -1570.0 -0.56 280.0 -501.0 -0.38 -0.666 -0.9837 3118943 ChemDiv3_003012 CN(C)c1ccc2C(=O)N(NC(=O)C)C(=O)c3cccc1c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I21 compound treatment 880.0 -930.0 -0.33 800.0 18.6 0.01 -0.2232 -0.6759 1912727 ChemDiv3_003013 COCc1cc(C)nc(Cl)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I22 compound treatment 400.0 -1410.0 -0.5 440.0 -341.0 -0.26 -0.539 -0.9545 3022890 ChemDiv3_003014 COc1ccc(/C=C/2\OC(=S)N(C)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I23 mock treatment 280.0 -1530.0 -0.54 400.0 -381.0 -0.29 -0.5909 -0.9581 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 I24 mock treatment 800.0 -1010.0 -0.36 520.0 -261.0 -0.2 -0.3953 -0.9625 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J01 compound treatment 280.0 -1530.0 -0.54 1760.0 979.0 0.75 0.1474 0.1591 3118944 ChemDiv3_003015 CCN1C(=O)/C(=C/C=C/2\N(C)c3c(ccc4cccnc34)C2(C)C)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J02 compound treatment 720.0 -1090.0 -0.39 280.0 -501.0 -0.38 -0.5456 -1.0 3022891 ChemDiv3_003016 COc1ccc2oc(=O)c3SC(Cc3c2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J03 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 1614526 ChemDiv3_003017 CC(C)OC(=O)c1cc2cc(Br)ccc2oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J04 compound treatment 5240.0 3430.0 1.22 600.0 -181.0 -0.14 0.7619 0.6221 1247339 ChemDiv3_003018 CCN(CC)Cc1c(O)ccc2cc(c3nc4ccccc4s3)c(=O)oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J05 compound treatment 320.0 -1490.0 -0.53 320.0 -461.0 -0.35 -0.6242 -0.9811 1534522 ChemDiv3_003019 OCCn1c(SC2CCCCC2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J06 compound treatment 600.0 -1210.0 -0.43 320.0 -461.0 -0.35 -0.554 -0.9955 3119080 ChemDiv3_003020 Cc1c(/C=N/n2cnnc2)c(O)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J07 compound treatment 280.0 -1530.0 -0.54 360.0 -421.0 -0.32 -0.6126 -0.9694 3119081 ChemDiv3_003021 Cc1c(/C=N/c2ccc(N3CCOCC3)c(Cl)c2)c(O)n4c5ccccc5nc4c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J08 compound treatment 2000.0 190.0 0.07 400.0 -381.0 -0.29 -0.1594 -0.5305 1151347 ChemDiv3_003022 CCOC(=O)c1cnc2c(Cl)c(Cl)ccc2c1N(C)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J09 compound treatment 440.0 -1370.0 -0.49 280.0 -501.0 -0.38 -0.6159 -0.9933 1313461 ChemDiv3_003023 COc1ccc(cc1OC)C2(CCCC2)C(=O)Nc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J10 compound treatment 280.0 -1530.0 -0.54 440.0 -341.0 -0.26 -0.5691 -0.9442 3022892 ChemDiv3_003024 COc1cc2CC(C)(C)N/C(=N\c3ccc(Br)cc3)/c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J11 compound treatment 320.0 -1490.0 -0.53 640.0 -141.0 -0.11 -0.4505 -0.8349 3119082 ChemDiv3_003025 O=c1n(Cc2ccccn2)c(=O)c3ccccc3c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J12 compound treatment 360.0 -1450.0 -0.51 360.0 -421.0 -0.32 -0.5925 -0.975 3022893 ChemDiv3_003026 OCC1(CO)SC(=NC1=O)Nc2cccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J13 compound treatment 1240.0 -570.0 -0.2 1680.0 899.0 0.69 0.3448 0.4797 3119083 ChemDiv3_003027 CC/1=C(C#N)C(=NC(=O)\C1=C/c2ccc(o2)c3ccccc3)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J14 compound treatment 360.0 -1450.0 -0.51 360.0 -421.0 -0.32 -0.5925 -0.975 1708679 ChemDiv3_003028 Cc1cc(C)c2c(N)c(sc2n1)S(=O)c3ccc(cc3)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J15 compound treatment 280.0 -1530.0 -0.54 320.0 -461.0 -0.35 -0.6343 -0.9786 1425945 ChemDiv3_003029 COc1ccc(cc1)C2N(CCN3CCOCC3)C(=O)C(=C2C(=O)c4ccccc4)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J16 compound treatment 320.0 -1490.0 -0.53 400.0 -381.0 -0.29 -0.5808 -0.9612 3119084 ChemDiv3_003030 CCS(=O)(=O)CCSc1nc(cc(c1C#N)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J17 compound treatment 280.0 -1530.0 -0.54 360.0 -421.0 -0.32 -0.6126 -0.9694 3119085 ChemDiv3_003031 O=C(NCc1cccnc1)/C(=C\c2cccc(Oc3ccccc3)c2)/S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J18 compound treatment 320.0 -1490.0 -0.53 640.0 -141.0 -0.11 -0.4505 -0.8349 3022894 ChemDiv3_003032 COc1ccc(cc1)c2cc(c(C#N)c(SCCS(=O)Cc3ccccc3)n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J19 compound treatment 360.0 -1450.0 -0.51 240.0 -541.0 -0.42 -0.6576 -0.9944 3119086 ChemDiv3_003033 C(c1ccco1)n/2c(cs\c2=N/c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J20 compound treatment 840.0 -970.0 -0.34 560.0 -221.0 -0.17 -0.3635 -0.9472 1409898 ChemDiv3_003034 COc1ccc(cc1)c2cc(c(C#N)c(SC3CCCCC3=O)n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J21 compound treatment 360.0 -1450.0 -0.51 280.0 -501.0 -0.38 -0.6359 -0.9898 3022895 ChemDiv3_003035 O=C1CCCN1CC(CN2CCOCC2)Sc3nnnn3c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J22 compound treatment 240.0 -1570.0 -0.56 5640.0 4860.0 3.73 2.2437 0.5949 1275651 ChemDiv3_003036 COc1cc(cc(OC)c1OC)C(=O)n2nc(c3cccnc3)n(CC=C)c2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J23 mock treatment 200.0 -1610.0 -0.57 320.0 -461.0 -0.35 -0.6543 -0.9736 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 J24 mock treatment 1000.0 -810.0 -0.29 760.0 -21.4 -0.02 -0.2148 -0.7464 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K01 compound treatment 640.0 -1170.0 -0.42 1280.0 499.0 0.38 -0.0228 -0.0404 3022896 ChemDiv3_003037 O=c1[nH]cc(/N=C/c2ccncc2)c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K02 compound treatment 7480.0 5670.0 2.01 600.0 -181.0 -0.14 1.3238 0.6566 3119087 ChemDiv3_003038 CCN1C(=O)/C(=C/c2ccc(o2)c3ccc(Br)cc3)/N(CC)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K03 compound treatment 440.0 -1370.0 -0.49 480.0 -301.0 -0.23 -0.5073 -0.9424 1358081 ChemDiv3_003039 CCSc1nc2ccccc2c(=O)n1C3CCOC(C)(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K04 compound treatment 320.0 -1490.0 -0.53 4360.0 3580.0 2.75 1.5689 0.5608 1594272 ChemDiv3_003040 Cc1c(C#N)c2nc3CCCCc3c(c4ccccc4)c2n1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K05 compound treatment 720.0 -1090.0 -0.39 360.0 -421.0 -0.32 -0.5022 -0.9961 3022897 ChemDiv3_003041 CC(Oc1ccc(C=C2C(=O)c3ccccc3C2=O)cc1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K06 compound treatment 440.0 -1370.0 -0.49 440.0 -341.0 -0.26 -0.529 -0.958 3119088 ChemDiv3_003042 CC(Cc1ccccc1)N/C=C\2/CC(=O)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K07 compound treatment 720.0 -1090.0 -0.39 920.0 139.0 0.11 -0.1982 -0.4942 1628644 ChemDiv3_003043 CCOC(=O)C1(CCN(CC1)C(=O)c2c(C)oc3ccc(OC)cc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K08 compound treatment 2440.0 630.0 0.22 480.0 -301.0 -0.23 -0.0056 -0.0174 1662593 ChemDiv3_003044 NC(=O)CN1CCCCCC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K09 compound treatment 1080.0 -730.0 -0.26 400.0 -381.0 -0.29 -0.3902 -0.9981 3119089 ChemDiv3_003045 CCN1C(=O)NC(=O)/C(=C\c2cn(CC(=O)N3CCCC3)c4ccccc24)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K10 compound treatment 640.0 -1170.0 -0.42 640.0 -141.0 -0.11 -0.3703 -0.863 1363537 ChemDiv3_003046 Cc1ccc2nc(C)n3c4ccccc4c(NC=O)c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K11 compound treatment 520.0 -1290.0 -0.46 520.0 -261.0 -0.2 -0.4655 -0.9316 3022898 ChemDiv3_003047 COC(=O)c1ccc(cc1)C(=O)Nc2ccc3[nH]c(nc3c2)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K12 compound treatment 680.0 -1130.0 -0.4 1280.0 499.0 0.38 -0.0128 -0.0231 3119090 ChemDiv3_003048 NC(=S)C(=C1CCCC1)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K13 compound treatment 1080.0 -730.0 -0.26 320.0 -461.0 -0.35 -0.4336 -0.9881 1509060 ChemDiv3_003049 O=c1[nH]cnc2n(ncc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K14 compound treatment 2080.0 270.0 0.1 3400.0 2620.0 2.01 1.4892 0.74 1733288 ChemDiv3_003050 CC1(CN2CC3(C)CN(C1)C2c4ccc(O)cc4O)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K15 compound treatment 880.0 -930.0 -0.33 440.0 -341.0 -0.26 -0.4186 -0.9935 3119091 ChemDiv3_003051 COC(=O)C/1=C(C)N(C)C(=O)\C1=C/c2cc(C)n(c2C)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K16 compound treatment 1120.0 -690.0 -0.24 880.0 98.6 0.08 -0.1196 -0.4667 3022899 ChemDiv3_003052 Cc1ccc(cc1)C2=C/C(=C\c3ccccc3C)/C(=O)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K17 compound treatment 800.0 -1010.0 -0.36 400.0 -381.0 -0.29 -0.4604 -0.995 1528158 ChemDiv3_003053 COc1ccc(cc1)n2c(C)nc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K18 compound treatment 480.0 -1330.0 -0.47 200.0 -581.0 -0.45 -0.6493 -0.9996 1492398 ChemDiv3_003054 O=c1oc2ccccc2cc1c3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K19 compound treatment 440.0 -1370.0 -0.49 720.0 -61.4 -0.05 -0.377 -0.7721 3022900 ChemDiv3_003055 CC(C)Oc1ccc2c(cc(=O)oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K20 compound treatment 640.0 -1170.0 -0.42 560.0 -221.0 -0.17 -0.4137 -0.9224 3119092 ChemDiv3_003056 CCSc1ccsc1C2C(=C(N)N(C3=C2C(=O)CC(C)(C)C3)c4cccnc4)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K21 compound treatment 880.0 -930.0 -0.33 400.0 -381.0 -0.29 -0.4403 -0.9982 1582251 ChemDiv3_003057 O=C(CN1c2cccc3cccc(c23)S1(=O)=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K22 compound treatment 6800.0 4990.0 1.77 760.0 -21.4 -0.02 1.2401 0.7005 3022901 ChemDiv3_003058 CN1C(=O)/C(=C\c2ccc(Cl)cc2Cl)/OC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K23 mock treatment 7200.0 5390.0 1.91 640.0 -141.0 -0.11 1.2753 0.6659 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 K24 mock treatment 2200.0 390.0 0.14 1240.0 459.0 0.35 0.3468 0.9167 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L01 compound treatment 440.0 -1370.0 -0.49 560.0 -221.0 -0.17 -0.4639 -0.9009 3022902 ChemDiv3_003059 CCN1C(=O)/C(=C/N(C)c2ccccc2)/OC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L02 compound treatment 440.0 -1370.0 -0.49 880.0 98.6 0.08 -0.2901 -0.5899 3119093 ChemDiv3_003060 FC(F)(F)C1Cc2c(S1)c(=O)oc3ccc4ccccc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L03 compound treatment 360.0 -1450.0 -0.51 440.0 -341.0 -0.26 -0.5491 -0.9511 1682835 ChemDiv3_003061 Cc1ccccc1CN2C(=O)C(O)(CC(=O)c3ccc4CCCCc4c3)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L04 compound treatment 400.0 -1410.0 -0.5 560.0 -221.0 -0.17 -0.4739 -0.897 1213120 ChemDiv3_003062 OC(=O)CCc1oc2cc(O)ccc2c(=O)c1c3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L05 compound treatment 520.0 -1290.0 -0.46 480.0 -301.0 -0.23 -0.4872 -0.9501 3022903 ChemDiv3_003063 CSc1nc2ccccc2n1CCO 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L06 compound treatment 560.0 -1250.0 -0.44 3800.0 3020.0 2.32 1.3251 0.5616 3119094 ChemDiv3_003064 CCc1c(C)nc2ncnn2c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L07 compound treatment 9200.0 7390.0 2.62 360.0 -421.0 -0.32 1.625 0.6152 3119095 ChemDiv3_003065 CCCCc1ccc(/N=C/c2c(C)c(C#N)c3nc4ccccc4n3c2O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L08 compound treatment 11560.0 9750.0 3.46 440.0 -341.0 -0.26 2.2604 0.6517 1574439 ChemDiv3_003066 CCOC(=O)c1cnc2c(C)cc(C)cc2c1Nc3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L09 compound treatment 520.0 -1290.0 -0.46 600.0 -181.0 -0.14 -0.4221 -0.8824 1292966 ChemDiv3_003067 CC1(C)CC(=O)C(=C(C1)NCc2ccccc2)C(=S)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L10 compound treatment 520.0 -1290.0 -0.46 2080.0 1300.0 1.0 0.3814 0.3476 1711945 ChemDiv3_003068 COc1cc(CN(C)C)c(O)c(CN(C)C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L11 compound treatment 440.0 -1370.0 -0.49 400.0 -381.0 -0.29 -0.5507 -0.9706 1592604 ChemDiv3_003069 Clc1ccc(CN2C(=O)c3ccc(cc3C2=O)c4nc5ccccc5c(=O)o4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L12 compound treatment 400.0 -1410.0 -0.5 360.0 -421.0 -0.32 -0.5825 -0.9778 1628631 ChemDiv3_003070 Nc1c(sc2nc3CCCc3cc12)C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L13 compound treatment 440.0 -1370.0 -0.49 360.0 -421.0 -0.32 -0.5724 -0.9805 3119096 ChemDiv3_003071 CN(C)c1ccc(/N=C\2/C(=C(C#N)C(=O)N(C)C2=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L14 compound treatment 520.0 -1290.0 -0.46 2120.0 1340.0 1.03 0.4031 0.3583 3119225 ChemDiv3_003072 Cc1cc(C)c2c(N)c(sc2n1)S(=O)Cc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L15 compound treatment 520.0 -1290.0 -0.46 360.0 -421.0 -0.32 -0.5524 -0.9856 1171680 ChemDiv3_003073 OC1=C(C(N(CCCn2ccnc2)C1=O)c3cccc(Br)c3)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L16 compound treatment 9280.0 7470.0 2.65 320.0 -461.0 -0.35 1.6233 0.6072 1601690 ChemDiv3_003074 CCCCS(=O)c1nc(cc(c1C#N)c2ccccc2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L17 compound treatment 2160.0 350.0 0.12 280.0 -501.0 -0.38 -0.1844 -0.4559 3119226 ChemDiv3_003075 OC(=O)CN1C(=O)/C(=c\2/sc3nc4ccccc4n3c2=O)/c5cc(Br)ccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L18 compound treatment 320.0 -1490.0 -0.53 440.0 -341.0 -0.26 -0.5591 -0.9476 3022904 ChemDiv3_003076 CCCCS(=O)CSc1nc(cc(c1C#N)c2ccccc2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L19 compound treatment 280.0 -1530.0 -0.54 360.0 -421.0 -0.32 -0.6126 -0.9694 1492207 ChemDiv3_003077 CN(CCO)S(=O)(=O)c1ccc-2c(c1)C(=NO)c3cc(ccc32)S(=O)(=O)N(C)CCO 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L20 compound treatment 440.0 -1370.0 -0.49 600.0 -181.0 -0.14 -0.4421 -0.8746 3022905 ChemDiv3_003078 CS(=O)C1CCCCC1(O)CSc2nc(cc(c2C#N)c3ccccc3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L21 compound treatment 960.0 -850.0 -0.3 5600.0 4820.0 3.7 2.4026 0.6473 3119227 ChemDiv3_003079 COC(=O)/C=c/1\sc2=NCCn2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L22 compound treatment 720.0 -1090.0 -0.39 720.0 -61.4 -0.05 -0.3068 -0.7875 1138814 ChemDiv3_003080 CC(=O)Nc1nc(NC(=O)C)nc(n1)c2ccccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L23 mock treatment 920.0 -890.0 -0.32 880.0 98.6 0.08 -0.1697 -0.5228 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 L24 mock treatment 1000.0 -810.0 -0.29 560.0 -221.0 -0.17 -0.3234 -0.9686 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M01 compound treatment 240.0 -1570.0 -0.56 4320.0 3540.0 2.72 1.5271 0.5507 1484138 ChemDiv3_003081 CC[N+]1(CC)Cc2c(C1)c(C(=C)C)c3ccccc3c2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M02 compound treatment 440.0 -1370.0 -0.49 560.0 -221.0 -0.17 -0.4639 -0.9009 3119228 ChemDiv3_003082 CC/1=NOC(=O)\C1=C\c2ccc(cc2)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M03 compound treatment 360.0 -1450.0 -0.51 400.0 -381.0 -0.29 -0.5708 -0.9643 1526199 ChemDiv3_003083 CCSc1nc2-c3ccccc3CC4(CCCC4)c2c(=O)n1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M04 compound treatment 400.0 -1410.0 -0.5 400.0 -381.0 -0.29 -0.5608 -0.9675 1671329 ChemDiv3_003084 CC[N+]1(Cc2ccccc2)C3=C(CN(C)CC3)c4ccccc41 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M05 compound treatment 1120.0 -690.0 -0.24 280.0 -501.0 -0.38 -0.4453 -0.9761 1542244 ChemDiv3_003085 CCCOc1ccc(cc1)c2nc(N(CC)CC)c3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M06 compound treatment 320.0 -1490.0 -0.53 280.0 -501.0 -0.38 -0.646 -0.9879 3022952 ChemDiv3_003086 Oc1ccc(/C=C\2/C(=O)CNC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M07 compound treatment 440.0 -1370.0 -0.49 240.0 -541.0 -0.42 -0.6376 -0.997 1350361 ChemDiv3_003087 Fc1ccc(Nc2ncnc3c4ccccc4oc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M08 compound treatment 1200.0 -610.0 -0.22 920.0 139.0 0.11 -0.0778 -0.3226 1709021 ChemDiv3_003088 COc1cccc2oc(c(Br)c12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M09 compound treatment 280.0 -1530.0 -0.54 480.0 -301.0 -0.23 -0.5474 -0.9278 3022953 ChemDiv3_003089 Fc1ccccc1N2C(=O)NC(=O)/C(=C\c3cn(CC(=O)N4CCCC4)c5ccccc35)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M10 compound treatment 400.0 -1410.0 -0.5 360.0 -421.0 -0.32 -0.5825 -0.9778 3022954 ChemDiv3_003090 CCOC(=O)/C(=C\1/CCCN1)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M11 compound treatment 240.0 -1570.0 -0.56 400.0 -381.0 -0.29 -0.6009 -0.9549 1509599 ChemDiv3_003091 CCc1nnc(NC(=O)C(CC(C)C)N2C(=O)c3ccccc3C2=O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M12 compound treatment 2440.0 630.0 0.22 280.0 -501.0 -0.38 -0.1142 -0.2565 1712524 ChemDiv3_003092 CC1=C(C(C(=C(N1)SCC(=O)N)C#N)c2ccco2)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M13 compound treatment 880.0 -930.0 -0.33 480.0 -301.0 -0.23 -0.3969 -0.985 3119229 ChemDiv3_003093 CCN(CC)CC#Cc1cccc(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M14 compound treatment 2040.0 230.0 0.08 600.0 -181.0 -0.14 -0.0408 -0.2527 1297646 ChemDiv3_003094 CC1(CN2CC3(C)CN(C1)C2C4CCCCC4)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M15 compound treatment 400.0 -1410.0 -0.5 1120.0 339.0 0.26 -0.1699 -0.3014 3119230 ChemDiv3_003095 CCC1(CC)Cc2ccccc2-c3nc(oc(=O)c31)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M16 compound treatment 2400.0 590.0 0.21 400.0 -381.0 -0.29 -0.0591 -0.1641 3119231 ChemDiv3_003096 CCc1ccc(cc1)n2c(C)cc(/C=C/3\SC(=S)N(CC=C)C3=O)c2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M17 compound treatment 280.0 -1530.0 -0.54 5360.0 4580.0 3.52 2.1017 0.5909 1403000 ChemDiv3_003097 O=c1n(c(CNc2ccccc2)nc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M18 compound treatment 400.0 -1410.0 -0.5 680.0 -101.0 -0.08 -0.4088 -0.8075 1363942 ChemDiv3_003098 Nc1cccc(Nc2ncnc3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M19 compound treatment 760.0 -1050.0 -0.37 360.0 -421.0 -0.32 -0.4922 -0.9975 3022955 ChemDiv3_003099 CN(C)c1ccc(cc1)c2nc(cc(=O)o2)c3cccc(I)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M20 compound treatment 2160.0 350.0 0.12 400.0 -381.0 -0.29 -0.1193 -0.375 3119232 ChemDiv3_003100 Cc1cc(C2C(=C(N)N(C3=C2C(=O)CC(C3)c4ccccc4)c5ccccc5Cl)C#N)c(C)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M21 compound treatment 440.0 -1370.0 -0.49 680.0 -101.0 -0.08 -0.3987 -0.8101 1607622 ChemDiv3_003101 CC(C)OC(=O)c1ccc(NC(=O)CSc2nc3cccnc3[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M22 compound treatment 520.0 -1290.0 -0.46 440.0 -341.0 -0.26 -0.5089 -0.965 1914743 ChemDiv3_003102 CCCN1C(=O)/C(=C/C=C\2/Oc3ccccc3N2CCC(=O)O)/N(CCO)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M23 mock treatment 360.0 -1450.0 -0.51 560.0 -221.0 -0.17 -0.4839 -0.8933 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 M24 mock treatment 960.0 -850.0 -0.3 3960.0 3180.0 2.44 1.5123 0.6151 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N01 compound treatment 1640.0 -170.0 -0.06 560.0 -221.0 -0.17 -0.1628 -0.9028 3022956 ChemDiv3_003103 OCC[n+]1ccc(/C=C/c2c[nH]c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N02 compound treatment 320.0 -1490.0 -0.53 880.0 98.6 0.08 -0.3202 -0.5998 3119233 ChemDiv3_003104 COC(=O)C1SC2(CC1(O)c3c(OC)c4ccoc4c(OC)c3O2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N03 compound treatment 400.0 -1410.0 -0.5 480.0 -301.0 -0.23 -0.5173 -0.9387 3022957 ChemDiv3_003105 Cc1ccccc1CN2C(=O)C(O)(CC(=O)/C=C\c3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N04 compound treatment 240.0 -1570.0 -0.56 280.0 -501.0 -0.38 -0.666 -0.9837 1613163 ChemDiv3_003106 COC(=O)c1c(C)oc2ccc(OCc3ccc(Br)cc3)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N05 compound treatment 440.0 -1370.0 -0.49 1600.0 819.0 0.63 0.1007 0.1268 1321741 ChemDiv3_003107 CCCn1c(SCC(=O)N2c3ccccc3Sc4ccccc24)nc5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N06 compound treatment 2320.0 510.0 0.18 280.0 -501.0 -0.38 -0.1443 -0.3392 1696278 ChemDiv3_003108 Cc1ccc2nc(c(CN3CCCC3)c(O)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N07 compound treatment 320.0 -1490.0 -0.53 520.0 -261.0 -0.2 -0.5157 -0.9121 1343499 ChemDiv3_003109 CCCN1C(Nc2ccccc2C1=O)c3ccc(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N08 compound treatment 3440.0 1630.0 0.58 360.0 -421.0 -0.32 0.1801 0.2718 1737251 ChemDiv3_003110 CCOC(=O)C1=C(Nc2ncnn2C1c3ccc(OCc4ccccc4)cc3)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N09 compound treatment 320.0 -1490.0 -0.53 3120.0 2340.0 1.8 0.8958 0.4786 1201402 ChemDiv3_003111 CN(C)CCc1cc2OCOc2c3c1ccc4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N10 compound treatment 320.0 -1490.0 -0.53 1080.0 299.0 0.23 -0.2117 -0.3674 1739556 ChemDiv3_003112 Oc1ccccc1CN2CCCN(Cc3ccccc3O)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N11 compound treatment 320.0 -1490.0 -0.53 1080.0 299.0 0.23 -0.2117 -0.3674 1119081 ChemDiv3_003113 Clc1ccc(CC(=O)Nc2cccc(c2)c3nc4cc5ccccc5cc4[nH]3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N12 compound treatment 440.0 -1370.0 -0.49 200.0 -581.0 -0.45 -0.6593 -0.9991 1853335 ChemDiv3_003114 CCN(CC)C(=O)c1sc2nc3CCCCCc3cc2c1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N13 compound treatment 480.0 -1330.0 -0.47 480.0 -301.0 -0.23 -0.4973 -0.9462 3119234 ChemDiv3_003115 CC/1=NOC(=O)\C1=C/c2ccc(O)c(O)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N14 compound treatment 560.0 -1250.0 -0.44 320.0 -461.0 -0.35 -0.564 -0.9938 3022958 ChemDiv3_003116 Cc1cc(C)c(C#N)c(SCSCc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N15 compound treatment 400.0 -1410.0 -0.5 560.0 -221.0 -0.17 -0.4739 -0.897 1503378 ChemDiv3_003117 OC1=C(C(N(CCCN2CCOCC2)C1=O)c3cccs3)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N16 compound treatment 560.0 -1250.0 -0.44 280.0 -501.0 -0.38 -0.5858 -0.9975 3119235 ChemDiv3_003118 Cc1ccc(cc1)c2cc(c(C#N)c(SCS(=O)Cc3ccccc3)n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N17 compound treatment 2120.0 310.0 0.11 320.0 -461.0 -0.35 -0.1727 -0.4657 1283724 ChemDiv3_003119 Cc1ccc(OCC(=O)n2c(SCc3ccc(F)cc3)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N18 compound treatment 2680.0 870.0 0.31 320.0 -461.0 -0.35 -0.0323 -0.0687 3119236 ChemDiv3_003120 O=S(CSc1nc(cc(c1C#N)c2ccccc2)c3cccs3)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N19 compound treatment 10360.0 8550.0 3.03 4080.0 3300.0 2.53 3.9354 0.996 1526293 ChemDiv3_003121 O=C(Nc1nccs1)C2(CC3CC4C2)CC(C3)(C4)C(=O)Nc5nccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N20 compound treatment 400.0 -1410.0 -0.5 480.0 -301.0 -0.23 -0.5173 -0.9387 1056485 ChemDiv3_003122 O=C1CCCCC1Sc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N21 compound treatment 10680.0 8870.0 3.15 320.0 -461.0 -0.35 1.9745 0.6236 3022959 ChemDiv3_003123 FC(F)(F)c1cc(nn1C(=S)N2CCOCC2)c3ccc4ccccc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N22 compound treatment 400.0 -1410.0 -0.5 400.0 -381.0 -0.29 -0.5608 -0.9675 1160068 ChemDiv3_003124 CCN(CC)C(=O)Sc1cccc2cccnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N23 mock treatment 5080.0 3270.0 1.16 600.0 -181.0 -0.14 0.7218 0.6178 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 N24 mock treatment 1560.0 -250.0 -0.09 3400.0 2620.0 2.01 1.3588 0.6753 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O01 compound treatment 400.0 -1410.0 -0.5 280.0 -501.0 -0.38 -0.6259 -0.9916 3022960 ChemDiv3_003125 CC1(C)OC(=O)C(=Cc2ccccc2F)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O02 compound treatment 240.0 -1570.0 -0.56 360.0 -421.0 -0.32 -0.6226 -0.9666 3119237 ChemDiv3_003126 Clc1cc(Cl)cc(c1)N2NC(=O)/C(=C\3/Nc4ccccc4C3=O)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O03 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 3022961 ChemDiv3_003127 COC(=O)CN1C=C(C(C(=C1)C(=O)OC)c2ccc(Cl)cc2)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O04 compound treatment 360.0 -1450.0 -0.51 200.0 -581.0 -0.45 -0.6794 -0.9975 1192351 ChemDiv3_003128 CC[N+]1(CCC2CC1)CC2C(O)(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O05 compound treatment 400.0 -1410.0 -0.5 400.0 -381.0 -0.29 -0.5608 -0.9675 3119238 ChemDiv3_003129 CCCOc1ccc(cc1)c2nc(OCC)c3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O06 compound treatment 320.0 -1490.0 -0.53 280.0 -501.0 -0.38 -0.646 -0.9879 3022962 ChemDiv3_003130 Cc1ccc(NC2=CC(=O)NC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O07 compound treatment 440.0 -1370.0 -0.49 280.0 -501.0 -0.38 -0.6159 -0.9933 1516607 ChemDiv3_003131 CCS(=O)(=O)N1CCN(CC2CCC=CC2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O08 compound treatment 200.0 -1610.0 -0.57 200.0 -581.0 -0.45 -0.7195 -0.9926 3022963 ChemDiv3_003132 COc1ccc(N/C(=C(/C=C/2\Nc3ccccc3C2=O)\C#N)/N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O09 compound treatment 320.0 -1490.0 -0.53 280.0 -501.0 -0.38 -0.646 -0.9879 3119370 ChemDiv3_003133 COc1ccc(OCCn2cc(C=C3C(=O)N(C)C(=O)N(C)C3=O)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O10 compound treatment 200.0 -1610.0 -0.57 1640.0 859.0 0.66 0.0622 0.0713 3022964 ChemDiv3_003134 CN(C)/C=N/c1c(C#N)c(C)n(c1C(=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O11 compound treatment 440.0 -1370.0 -0.49 240.0 -541.0 -0.42 -0.6376 -0.997 1338630 ChemDiv3_003135 CC(C)(c1ccccc1)c2ccc(OCC(=O)NC3CCCC3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O12 compound treatment 320.0 -1490.0 -0.53 200.0 -581.0 -0.45 -0.6894 -0.9965 1623139 ChemDiv3_003136 O=C1N(CCSc2nc(cc(c3ccco3)c2C#N)c4ccccc4)C(=O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O13 compound treatment 240.0 -1570.0 -0.56 160.0 -621.0 -0.48 -0.7312 -0.997 3022965 ChemDiv3_003137 Cc1cccc(C#CCN2CCCCC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O14 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 1073936 ChemDiv3_003138 Nn1cnnc1SCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O15 compound treatment 280.0 -1530.0 -0.54 160.0 -621.0 -0.48 -0.7211 -0.9979 1709316 ChemDiv3_003139 CC1(C)Cc2ccccc2-c3nc(c4ccccc4)n(CCO)c(=O)c31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O16 compound treatment 240.0 -1570.0 -0.56 200.0 -581.0 -0.45 -0.7095 -0.994 3022966 ChemDiv3_003140 CN1C(=O)C(=CC2CC(=NN(C2=O)c3ccccc3)C)C(=O)N(C)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O17 compound treatment 320.0 -1490.0 -0.53 320.0 -461.0 -0.35 -0.6242 -0.9811 1457475 ChemDiv3_003141 CCOC(=S)SCc1nc2ccccc2c(=O)n1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O18 compound treatment 400.0 -1410.0 -0.5 280.0 -501.0 -0.38 -0.6259 -0.9916 1557182 ChemDiv3_003142 C1CCCN(CC1)c2nc(nc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O19 compound treatment 480.0 -1330.0 -0.47 440.0 -341.0 -0.26 -0.519 -0.9615 3022967 ChemDiv3_003143 Ic1cccc(c1)c2nc(cc(=O)o2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O20 compound treatment 440.0 -1370.0 -0.49 200.0 -581.0 -0.45 -0.6593 -0.9991 3119371 ChemDiv3_003144 CCSc1sc(CC)cc1C2C(=C(C)NC3=C2C(=O)CCC3)C(=O)Nc4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O21 compound treatment 400.0 -1410.0 -0.5 240.0 -541.0 -0.42 -0.6476 -0.9958 3119372 ChemDiv3_003145 COc1cc(Br)cc(/C=N/N(CCO)C2=NS(=O)(=O)c3ccccc23)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O22 compound treatment 400.0 -1410.0 -0.5 200.0 -581.0 -0.45 -0.6693 -0.9984 3022968 ChemDiv3_003146 CCn1c(=S)ccc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O23 mock treatment 440.0 -1370.0 -0.49 320.0 -461.0 -0.35 -0.5941 -0.9879 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 O24 mock treatment 400.0 -1410.0 -0.5 280.0 -501.0 -0.38 -0.6259 -0.9916 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P01 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 1125247 ChemDiv3_003147 OC(=O)c1cc2cccc(CC=C)c2oc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P02 compound treatment 520.0 -1290.0 -0.46 200.0 -581.0 -0.45 -0.6392 -0.9999 1617401 ChemDiv3_003148 COc1ccc2n(Cc3ccccc3)c(C)c(C(=O)N4CCCC4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P03 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 1563489 ChemDiv3_003149 Fc1cccc(c1)C(=O)Nc2ccc(cc2)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P04 compound treatment 320.0 -1490.0 -0.53 520.0 -261.0 -0.2 -0.5157 -0.9121 1184530 ChemDiv3_003150 Cc1ccccc1COc2ccc3oc(c(C(=O)O)c3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P05 compound treatment 200.0 -1610.0 -0.57 320.0 -461.0 -0.35 -0.6543 -0.9736 3022969 ChemDiv3_003151 CCC(C)Sc1nc(=O)c2ccccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P06 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 1012560 ChemDiv3_003152 OCCNc1ncnc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P07 compound treatment 320.0 -1490.0 -0.53 240.0 -541.0 -0.42 -0.6677 -0.9929 1510943 ChemDiv3_003153 CCCCN1CNC(=S)NC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P08 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 1188027 ChemDiv3_003154 CCOc1ccc2c3CCCc3c(=O)oc2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P09 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3119373 ChemDiv3_003155 COc1cccc(NC2=Nc3cccc4cccc2c34)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P10 compound treatment 280.0 -1530.0 -0.54 360.0 -421.0 -0.32 -0.6126 -0.9694 1058532 ChemDiv3_003156 OC1CCCN(Cc2ccccc2)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P11 compound treatment 200.0 -1610.0 -0.57 280.0 -501.0 -0.38 -0.6761 -0.9816 1124382 ChemDiv3_003157 COc1cccc(c1)c2nc3cc(OC)c(OC)cc3c(=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P12 compound treatment 200.0 -1610.0 -0.57 280.0 -501.0 -0.38 -0.6761 -0.9816 3022970 ChemDiv3_003158 Clc1ccc(CN2C(=O)N/C(=C\c3ccccc3Cl)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P13 compound treatment 280.0 -1530.0 -0.54 360.0 -421.0 -0.32 -0.6126 -0.9694 3119374 ChemDiv3_003159 CC/1=C(C#N)C(=O)N(CCc2ccccc2)C(=O)\C1=C/c3ccc(o3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P14 compound treatment 360.0 -1450.0 -0.51 320.0 -461.0 -0.35 -0.6142 -0.9834 1353343 ChemDiv3_003160 Clc1ccc(CS(=O)c2nc3CCCCc3cc2C#N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P15 compound treatment 240.0 -1570.0 -0.56 240.0 -541.0 -0.42 -0.6877 -0.9896 3119375 ChemDiv3_003161 Cc1ccc(cc1)c2nc(C#N)c(NCCCn3ccnc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P16 compound treatment 320.0 -1490.0 -0.53 560.0 -221.0 -0.17 -0.494 -0.8896 1505579 ChemDiv3_003162 CCS(=O)CCSc1nc(cc(c1C#N)c2ccccc2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P17 compound treatment 280.0 -1530.0 -0.54 280.0 -501.0 -0.38 -0.656 -0.9858 1293590 ChemDiv3_003163 COc1ccc(cc1OC)C2N(C(=O)C(=C2C(=O)c3ccc(F)cc3)O)c4nnc(C)s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P18 compound treatment 240.0 -1570.0 -0.56 280.0 -501.0 -0.38 -0.666 -0.9837 3119376 ChemDiv3_003164 CCCCS(=O)c1sc2nc(cc(c3ccccc3)c2c1N)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P19 compound treatment 200.0 -1610.0 -0.57 400.0 -381.0 -0.29 -0.6109 -0.9518 1334571 ChemDiv3_003165 COC(=O)C(NC(=O)c1ccc(cc1)S(=O)(=O)N2CCOCC2)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P20 compound treatment 280.0 -1530.0 -0.54 240.0 -541.0 -0.42 -0.6777 -0.9913 3119377 ChemDiv3_003166 CCS(=O)(=O)CCSc1nc(C)cc(C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P21 compound treatment 240.0 -1570.0 -0.56 320.0 -461.0 -0.35 -0.6443 -0.9761 3023071 ChemDiv3_003167 FC(F)(F)c1cc(nn1C(=S)N2CCCCCC2)c3ccc4ccccc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P22 compound treatment 320.0 -1490.0 -0.53 320.0 -461.0 -0.35 -0.6242 -0.9811 3119378 ChemDiv3_003168 N=C/1N2C(=CSC2=NC(=O)\C1=C/c3cccs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P23 mock treatment 3240.0 1430.0 0.51 1040.0 259.0 0.2 0.4991 0.9162 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2009 P24 mock treatment 9840.0 8030.0 2.85 1160.0 379.0 0.29 2.2198 0.7752 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A01 compound treatment 320.0 -1890.0 -0.67 3240.0 2380.0 1.83 0.8215 0.4214 1286976 ChemDiv3_003169 COc1ccc(cc1)n2c(NN)nc3sc4CCCc4c3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A02 compound treatment 200.0 -2010.0 -0.71 560.0 -295.0 -0.23 -0.6635 -0.8883 1560637 ChemDiv3_003170 COC(=O)c1c(C)oc2ccc(cc12)N(C(=O)C)S(=O)(=O)c3ccc4ccccc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A03 compound treatment 440.0 -1770.0 -0.63 5600.0 4740.0 3.64 2.1327 0.577 3119379 ChemDiv3_003171 CCN(CC)S(=O)(=O)c1ccc(cc1)c2cs/c(=N\c3ccc(C)cc3)/n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A04 compound treatment 280.0 -1930.0 -0.68 360.0 -495.0 -0.38 -0.752 -0.9617 1585858 ChemDiv3_003172 CC1(CC2(C)CC3(C)C1)CC(C2)(C3)C(=O)NC(=S)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A05 compound treatment 320.0 -1890.0 -0.67 4240.0 3380.0 2.6 1.3643 0.5084 1866874 ChemDiv3_003173 CN(CC(O)Cn1c2ccccc2c3ccccc13)S(=O)(=O)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A06 compound treatment 320.0 -1890.0 -0.67 1320.0 465.0 0.36 -0.2208 -0.2912 1618410 ChemDiv3_003174 CC1(C)Cc2c(CO1)sc3nc(NN)n(Cc4ccccc4)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A07 compound treatment 440.0 -1770.0 -0.63 360.0 -495.0 -0.38 -0.7119 -0.9713 1669656 ChemDiv3_003175 C(NC1CCCc2c1[nH]c3ccc(cc23)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A08 compound treatment 280.0 -1930.0 -0.68 200.0 -655.0 -0.5 -0.8389 -0.9886 3023072 ChemDiv3_003176 Cc1cc(NC2CCCCC2)nc(NCc3ccccc3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A09 compound treatment 440.0 -1770.0 -0.63 200.0 -655.0 -0.5 -0.7987 -0.9941 1313123 ChemDiv3_003177 Clc1ccccc1C(=O)Nc2ccc(cc2)c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A10 compound treatment 320.0 -1890.0 -0.67 1680.0 825.0 0.63 -0.0254 -0.0276 1391391 ChemDiv3_003178 O=C(CN1C(=O)c2ccccc2C1=O)N(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A11 compound treatment 800.0 -1410.0 -0.5 240.0 -615.0 -0.47 -0.6867 -0.9996 1356650 ChemDiv3_003179 Fc1ccccc1Nc2nc(NCc3ccccc3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A12 compound treatment 280.0 -1930.0 -0.68 240.0 -615.0 -0.47 -0.8171 -0.9837 3119380 ChemDiv3_003180 COc1ccc(/C=C/2\SC(=S)N(CC3CCCO3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A13 compound treatment 240.0 -1970.0 -0.7 440.0 -415.0 -0.32 -0.7186 -0.937 1433370 ChemDiv3_003181 Cc1ccc(cc1)C(=O)Nc2cccc(c2)c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A14 compound treatment 3200.0 994.0 0.35 360.0 -495.0 -0.38 -0.0195 -0.0377 1026172 ChemDiv3_003182 NC(=N)Nc1nc2ccccc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A15 compound treatment 4480.0 2270.0 0.81 200.0 -655.0 -0.5 0.2147 0.2258 3119381 ChemDiv3_003183 CC(=O)Nc1c(O)[nH]c2ccc(C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A16 compound treatment 760.0 -1450.0 -0.51 280.0 -575.0 -0.44 -0.675 -0.9972 1236383 ChemDiv3_003184 Fc1ccccc1C(=O)n2c3CCCCc3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A17 compound treatment 360.0 -1850.0 -0.65 360.0 -495.0 -0.38 -0.7319 -0.9665 3023073 ChemDiv3_003185 CCSc1nc2ccccc2n1C(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A18 compound treatment 320.0 -1890.0 -0.67 760.0 -95.2 -0.07 -0.5248 -0.7797 3119528 ChemDiv3_003186 CCC(N1C(=O)c2ccccc2C1=O)C(=O)N3c4ccccc4Sc5ccc(cc35)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A19 compound treatment 280.0 -1930.0 -0.68 240.0 -615.0 -0.47 -0.8171 -0.9837 1545724 ChemDiv3_003187 COc1ccc(cc1)C2N(CCN2C(=O)c3ccc(C)cc3)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A20 compound treatment 9840.0 7630.0 2.71 360.0 -495.0 -0.38 1.6461 0.6019 3119529 ChemDiv3_003188 Cc1cc(C)c(C#N)c(SCc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A21 compound treatment 8320.0 6110.0 2.17 760.0 -95.2 -0.07 1.4819 0.6829 1360295 ChemDiv3_003189 CCCC(=O)Oc1ccc(cc1)N(C(=O)CCC)S(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A22 compound treatment 520.0 -1690.0 -0.6 600.0 -255.0 -0.2 -0.5615 -0.8921 1447802 ChemDiv3_003190 Fc1ccc(cc1)C(=O)N2c3ccccc3C=Cc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A23 mock treatment 480.0 -1730.0 -0.61 280.0 -575.0 -0.44 -0.7453 -0.9871 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 A24 mock treatment 560.0 -1650.0 -0.58 320.0 -535.0 -0.41 -0.7035 -0.9852 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B01 compound treatment 2040.0 -166.0 -0.06 360.0 -495.0 -0.38 -0.3105 -0.8072 3119530 ChemDiv3_003191 CC1C=CCC2C1C(=O)N(C2=O)c3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B02 compound treatment 3720.0 1510.0 0.54 4080.0 3220.0 2.48 2.1303 0.8409 3119531 ChemDiv3_003192 Nc1nc(SC/C=C/c2ccccc2)nc3sc4CCCCc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B03 compound treatment 360.0 -1850.0 -0.65 4560.0 3700.0 2.84 1.5481 0.5304 1464526 ChemDiv3_003193 CCOC(=O)c1c(NC(=O)c2ccco2)sc3C(=O)CCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B04 compound treatment 400.0 -1810.0 -0.64 640.0 -215.0 -0.17 -0.5699 -0.8612 3119532 ChemDiv3_003194 CCOC(=O)c1c(C)oc-2c1/C(=C/NCCC3=CCCCC3)/C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B05 compound treatment 280.0 -1930.0 -0.68 2960.0 2100.0 1.62 0.6594 0.3759 3119533 ChemDiv3_003195 OC(=O)CCN1C(=O)/C(=C/c2ccccn2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B06 compound treatment 320.0 -1890.0 -0.67 600.0 -255.0 -0.2 -0.6117 -0.8773 3119534 ChemDiv3_003196 CCOC(=O)C1=CC(=C2C(=O)NC(=O)NC2=O)c3ccccc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B07 compound treatment 240.0 -1970.0 -0.7 680.0 -175.0 -0.13 -0.5883 -0.8282 3023099 ChemDiv3_003197 FC(F)(F)c1ccccc1NC(=O)CN2C(=O)/C(=C/c3ccccc3Cl)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B08 compound treatment 280.0 -1930.0 -0.68 320.0 -535.0 -0.41 -0.7737 -0.9704 1219353 ChemDiv3_003198 O=C(CSC1=C(C#N)C(CC(=O)N1)c2ccccc2)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B09 compound treatment 240.0 -1970.0 -0.7 720.0 -135.0 -0.1 -0.5666 -0.8035 3023100 ChemDiv3_003199 CN(Cc1ccccc1)C(=S)NC(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B10 compound treatment 280.0 -1930.0 -0.68 360.0 -495.0 -0.38 -0.752 -0.9617 3119535 ChemDiv3_003200 Cc1[nH]c2ccccc2c1C(Nc3cccc(c3)C(F)(F)F)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B11 compound treatment 360.0 -1850.0 -0.65 280.0 -575.0 -0.44 -0.7754 -0.9816 1069911 ChemDiv3_003201 Cc1ccc(cc1)S(=O)(=O)N2CN3CN(CN(C2)C3)S(=O)(=O)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B12 compound treatment 320.0 -1890.0 -0.67 280.0 -575.0 -0.44 -0.7854 -0.9796 1300854 ChemDiv3_003202 CN(Cc1ccccc1)S(=O)(=O)c2ccc(cc2)C(=O)Nc3ccc4sc(C)nc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B13 compound treatment 560.0 -1650.0 -0.58 200.0 -655.0 -0.5 -0.7686 -0.9972 1562840 ChemDiv3_003203 CC(C)Cc1ccc(cc1)C(C)C(=O)NC(C)Cc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B14 compound treatment 320.0 -1890.0 -0.67 320.0 -535.0 -0.41 -0.7637 -0.9726 3119536 ChemDiv3_003204 CCOC(=O)C1=CC(=C2C(=O)N(CC)C(=S)N(CC)C2=O)c3ccccc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B15 compound treatment 400.0 -1810.0 -0.64 280.0 -575.0 -0.44 -0.7653 -0.9835 1519780 ChemDiv3_003205 NS(=O)(=O)c1ccc(NC(=O)C2CCCNC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B16 compound treatment 320.0 -1890.0 -0.67 320.0 -535.0 -0.41 -0.7637 -0.9726 1286586 ChemDiv3_003206 CCOC(=O)c1c(oc2ccc(OCc3ccc(cc3)C(=O)OC)cc12)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B17 compound treatment 1160.0 -1050.0 -0.37 1040.0 185.0 0.14 -0.1621 -0.408 1529438 ChemDiv3_003207 CCc1ccc(cc1)n2nc3ccc(NC(=O)c4ccccc4Br)cc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B18 compound treatment 1400.0 -806.0 -0.29 560.0 -295.0 -0.23 -0.3625 -0.9934 3119537 ChemDiv3_003208 CCc1nnc2c3c(c(C)sc3ncn12)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B19 compound treatment 320.0 -1890.0 -0.67 320.0 -535.0 -0.41 -0.7637 -0.9726 3119538 ChemDiv3_003209 CC1=CCC2(C(C1)c3ccc(Br)cc3)C(=O)OC(C)(C)OC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B20 compound treatment 560.0 -1650.0 -0.58 520.0 -335.0 -0.26 -0.5949 -0.9322 3023101 ChemDiv3_003210 C1CCc2c(C1)c(nc3ccc4ccccc4c23)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B21 compound treatment 4000.0 1790.0 0.64 480.0 -375.0 -0.29 0.2463 0.3526 3119539 ChemDiv3_003211 Clc1ccc(OCCn2c(NC(=S)Nc3ccccc3)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B22 compound treatment 4080.0 1870.0 0.66 4520.0 3660.0 2.81 2.4595 0.8507 3023102 ChemDiv3_003212 CCOC(=O)N1CCN(CC1)C(=O)/C(=C/c2ccccc2Cl)/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B23 mock treatment 3840.0 1630.0 0.58 5720.0 4860.0 3.73 3.0507 0.8072 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 B24 mock treatment 6400.0 4190.0 1.49 5400.0 4540.0 3.49 3.5192 0.9278 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C01 compound treatment 800.0 -1410.0 -0.5 360.0 -495.0 -0.38 -0.6216 -0.991 3119540 ChemDiv3_003213 CCC1(CN(CC2(CC)CN(C1)S(=O)(=O)c3ccccc3)S(=O)(=O)c4ccccc4)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C02 compound treatment 3880.0 1670.0 0.59 680.0 -175.0 -0.13 0.3248 0.5334 1175485 ChemDiv3_003214 CCOC(=O)c1c(oc2ccc(NS(=O)(=O)c3ccc(CC)cc3)cc12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C03 compound treatment 320.0 -1890.0 -0.67 400.0 -455.0 -0.35 -0.7202 -0.9541 3023103 ChemDiv3_003215 CCOc1ccc(/N=c/2\scc(c3ccc(Cl)s3)n2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C04 compound treatment 2760.0 554.0 0.2 2280.0 1420.0 1.09 0.9124 0.821 3023104 ChemDiv3_003216 O=C1c2ccccc2C(=Cc3cccs3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C05 compound treatment 480.0 -1730.0 -0.61 6520.0 5660.0 4.35 2.6422 0.6016 3119541 ChemDiv3_003217 CC1=C(C(NC(=O)N1)c2ccc(C)cc2)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C06 compound treatment 280.0 -1930.0 -0.68 440.0 -415.0 -0.32 -0.7086 -0.9397 1374480 ChemDiv3_003218 CCNC(=S)Nc1sc2COC(C)(C)Cc2c1C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C07 compound treatment 200.0 -2010.0 -0.71 240.0 -615.0 -0.47 -0.8372 -0.9802 1491281 ChemDiv3_003219 CCNC(=O)C1CCCc2c1[nH]c3ccc(Cl)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C08 compound treatment 200.0 -2010.0 -0.71 280.0 -575.0 -0.44 -0.8155 -0.9736 3023105 ChemDiv3_003220 Cc1cc(OCC=C)nc(n1)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C09 compound treatment 240.0 -1970.0 -0.7 280.0 -575.0 -0.44 -0.8055 -0.9757 1399234 ChemDiv3_003221 CCc1ccc2oc(nc2c1)c3ccc(NC(=O)c4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C10 compound treatment 280.0 -1930.0 -0.68 280.0 -575.0 -0.44 -0.7954 -0.9777 1371725 ChemDiv3_003222 O=P(CN(CC1CCCO1)Cc2cccs2)(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C11 compound treatment 280.0 -1930.0 -0.68 280.0 -575.0 -0.44 -0.7954 -0.9777 3023106 ChemDiv3_003223 CCOC(=O)c1cnn(c1N)c2ncnc3sc4CCCCc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C12 compound treatment 760.0 -1450.0 -0.51 880.0 24.8 0.02 -0.3493 -0.6804 3119542 ChemDiv3_003224 O=C/1N(CC2CCCO2)C(=S)S\C1=C/C3CCC=CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C13 compound treatment 360.0 -1850.0 -0.65 280.0 -575.0 -0.44 -0.7754 -0.9816 1425019 ChemDiv3_003225 COc1ccc(cc1)C(=O)Nc2cccc(c2)c3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C14 compound treatment 280.0 -1930.0 -0.68 320.0 -535.0 -0.41 -0.7737 -0.9704 3119543 ChemDiv3_003226 CC1CC(C)(C)N(C(=O)c2ccccc2F)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C15 compound treatment 280.0 -1930.0 -0.68 280.0 -575.0 -0.44 -0.7954 -0.9777 3023107 ChemDiv3_003227 CCOC(=O)c1cccc2/C(=N\O)/c3ccccc3-c21 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C16 compound treatment 200.0 -2010.0 -0.71 240.0 -615.0 -0.47 -0.8372 -0.9802 3119544 ChemDiv3_003228 CCOC(=O)C1=CS/C(=C\2/C(=S)C(C)(C)N(C(=O)CC(C)C)c3ccc(OCC)cc23)/S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C17 compound treatment 1640.0 -566.0 -0.2 320.0 -535.0 -0.41 -0.4326 -0.9458 1029312 ChemDiv3_003229 OC(=O)c1ccc(cc1)S(=O)(=O)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C18 compound treatment 400.0 -1810.0 -0.64 320.0 -535.0 -0.41 -0.7436 -0.9769 3119545 ChemDiv3_003230 Cc1ccc(cc1)C(=O)N2CCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C19 compound treatment 2840.0 634.0 0.22 320.0 -535.0 -0.41 -0.1316 -0.2809 3119546 ChemDiv3_003231 CC(C)CCSc1nc(N)c2c3C(C)CCCc3sc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C20 compound treatment 3360.0 1150.0 0.41 240.0 -615.0 -0.47 -0.0445 -0.0713 3023108 ChemDiv3_003232 CSc1nc(cc(c2cccs2)c1C#N)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C21 compound treatment 320.0 -1890.0 -0.67 400.0 -455.0 -0.35 -0.7202 -0.9541 3023109 ChemDiv3_003233 Cc1ccc(cc1)S(=O)(=O)N=C2C=CC(=O)C=C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C22 compound treatment 2160.0 -46.3 -0.02 760.0 -95.2 -0.07 -0.0633 -0.8449 1523680 ChemDiv3_003234 CN1C2CCC1C=C(C2)N(C(=O)c3ccc(Cl)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C23 mock treatment 6840.0 4630.0 1.64 360.0 -495.0 -0.38 0.8935 0.5296 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 C24 mock treatment 5480.0 3270.0 1.16 280.0 -575.0 -0.44 0.509 0.4096 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D01 compound treatment 360.0 -1850.0 -0.65 720.0 -135.0 -0.1 -0.5365 -0.8091 1419514 ChemDiv3_003235 Brc1ccc(cc1)C(=O)COC(=O)C(Cc2ccccc2)N3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D02 compound treatment 4480.0 2270.0 0.81 5680.0 4820.0 3.7 3.1896 0.8414 1537888 ChemDiv3_003236 CCCn1c(N)nc2n(C)c(=O)n(C)c(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D03 compound treatment 440.0 -1770.0 -0.63 720.0 -135.0 -0.1 -0.5164 -0.8131 3119547 ChemDiv3_003237 CCOC(=O)N1CCC(=C(C#N)C(=O)Nc2cc(OC)ccc2OC)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D04 compound treatment 480.0 -1730.0 -0.61 3240.0 2380.0 1.83 0.8616 0.4463 3119682 ChemDiv3_003238 CCOC(=O)c1c(C)oc-2c1/C(=C/NCCc3c[nH]c4ccccc34)/C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D05 compound treatment 600.0 -1610.0 -0.57 440.0 -415.0 -0.32 -0.6283 -0.9623 1526203 ChemDiv3_003239 Cc1cccc(Oc2coc3cc(OC(=O)c4ccc(F)cc4)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D06 compound treatment 280.0 -1930.0 -0.68 160.0 -695.0 -0.53 -0.8606 -0.9925 1546958 ChemDiv3_003240 CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCCc4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D07 compound treatment 320.0 -1890.0 -0.67 280.0 -575.0 -0.44 -0.7854 -0.9796 3023138 ChemDiv3_003241 CCOC(=O)C1=C(NC(=O)c2ccco2)Oc3ccc4ccccc4c3C1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D08 compound treatment 400.0 -1810.0 -0.64 240.0 -615.0 -0.47 -0.787 -0.9887 1685642 ChemDiv3_003242 Cc1ccccc1NC(=O)CSC2=C(C#N)C(C3=C(CCCC3=O)N2)c4ccccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D09 compound treatment 360.0 -1850.0 -0.65 360.0 -495.0 -0.38 -0.7319 -0.9665 3023139 ChemDiv3_003243 S=C(NCCCN1CCOCC1)N(Cc2ccccc2)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D10 compound treatment 280.0 -1930.0 -0.68 280.0 -575.0 -0.44 -0.7954 -0.9777 3119683 ChemDiv3_003244 Cc1[nH]c2ccccc2c1C(Nc3ccccc3C(F)(F)F)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D11 compound treatment 240.0 -1970.0 -0.7 360.0 -495.0 -0.38 -0.762 -0.9593 1631606 ChemDiv3_003245 CCOc1ccc(cc1)C(=O)n2cnc3cc(C)c(C)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D12 compound treatment 440.0 -1770.0 -0.63 320.0 -535.0 -0.41 -0.7336 -0.9791 1137693 ChemDiv3_003246 CCN1C(=O)c2cccc3c(NC(=O)c4ccc(cc4)S(=O)(=O)N5CCCCC5C)ccc1c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D13 compound treatment 1040.0 -1170.0 -0.41 280.0 -575.0 -0.44 -0.6048 -0.9995 1575379 ChemDiv3_003247 O=C(CCCN1C(=O)c2ccccc2C1=O)n3ccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D14 compound treatment 280.0 -1930.0 -0.68 320.0 -535.0 -0.41 -0.7737 -0.9704 1720106 ChemDiv3_003248 Cc1nn(C(=O)C2CCCN2S(=O)(=O)c3ccccc3)c(C)c1Sc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D15 compound treatment 240.0 -1970.0 -0.7 360.0 -495.0 -0.38 -0.762 -0.9593 3119684 ChemDiv3_003249 CC(Cc1c[nH]c2ccccc12)N(Cc3ccccc3)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D16 compound treatment 240.0 -1970.0 -0.7 240.0 -615.0 -0.47 -0.8272 -0.982 3023140 ChemDiv3_003250 Brc1ccc(cc1)N2Cc3ccccc3C2=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D17 compound treatment 240.0 -1970.0 -0.7 320.0 -535.0 -0.41 -0.7837 -0.9681 3119685 ChemDiv3_003251 CC1(C)CC(=O)C(=CNn2cnc3ccccc3c2=O)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D18 compound treatment 320.0 -1890.0 -0.67 200.0 -655.0 -0.5 -0.8288 -0.9901 3023141 ChemDiv3_003252 Cc1ccc(SCc2cn3cccnc3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D19 compound treatment 320.0 -1890.0 -0.67 400.0 -455.0 -0.35 -0.7202 -0.9541 3023142 ChemDiv3_003253 CC(NC=C1C(=O)OC(C)(C)OC1=O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D20 compound treatment 440.0 -1770.0 -0.63 360.0 -495.0 -0.38 -0.7119 -0.9713 1469730 ChemDiv3_003254 O=C1CC(c2ccccc2)c3c(N1)ccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D21 compound treatment 320.0 -1890.0 -0.67 480.0 -375.0 -0.29 -0.6768 -0.9291 3119686 ChemDiv3_003255 Clc1ccc(Cn2c(NC(=S)Nc3ccccc3)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D22 compound treatment 1040.0 -1170.0 -0.41 360.0 -495.0 -0.38 -0.5614 -0.9991 3023143 ChemDiv3_003256 COc1ccc(NC(=O)CN(c2ccc(C)cc2)S(=O)(=O)c3ccc(OC)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D23 mock treatment 5400.0 3190.0 1.13 2680.0 1820.0 1.4 1.7918 0.9945 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 D24 mock treatment 4320.0 2110.0 0.75 560.0 -295.0 -0.23 0.37 0.4723 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E01 compound treatment 6120.0 3910.0 1.39 2480.0 1620.0 1.25 1.8638 0.9986 1562483 ChemDiv3_003257 CCSc1nc2sc3CCCc3c2c(=O)n1CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E02 compound treatment 15720.0 13500.0 4.79 174000.0 173000.0 132.93 97.3831 0.7321 3119687 ChemDiv3_003258 OC(=O)c1cccc(c1)S(=O)(=O)/N=C\2/C=C(NS(=O)(=O)c3ccccc3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E03 compound treatment 1800.0 -406.0 -0.14 3600.0 2740.0 2.11 1.3881 0.6572 3023144 ChemDiv3_003259 COC(=O)CSc1nc(C)c(Br)c(O)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E04 compound treatment 6880.0 4670.0 1.66 920.0 64.8 0.05 1.2076 0.728 1316178 ChemDiv3_003260 CC1(C)CC(=O)C2=C(C1)C(Nc3ccc4ccccc4c23)c5cccnc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E05 compound treatment 600.0 -1610.0 -0.57 240.0 -615.0 -0.47 -0.7369 -0.9956 1294879 ChemDiv3_003261 COc1ccc(cc1OC)C2NC(=O)NC(=C2C(=O)c3ccccc3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E06 compound treatment 360.0 -1850.0 -0.65 320.0 -535.0 -0.41 -0.7536 -0.9748 3119688 ChemDiv3_003262 C(CC1OCCCO1)Sc2nnc(o2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E07 compound treatment 560.0 -1650.0 -0.58 560.0 -295.0 -0.23 -0.5732 -0.915 1321422 ChemDiv3_003263 Cc1ccc2n(C)c3C(CCCc3c2c1)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E08 compound treatment 6600.0 4390.0 1.56 1000.0 145.0 0.11 1.1808 0.7556 1409750 ChemDiv3_003264 O=C1CC(c2csc(n2)c3ccccc3)C4(CCCCC4)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E09 compound treatment 5920.0 3710.0 1.32 360.0 -495.0 -0.38 0.6628 0.4833 1852910 ChemDiv3_003265 CN(C)N1C(=C(C#N)C(C2=C1CCCC2=O)c3ccccc3)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E10 compound treatment 760.0 -1450.0 -0.51 400.0 -455.0 -0.35 -0.6099 -0.9825 3119689 ChemDiv3_003266 O=c1c(/C=N/CCc2ccccc2)c(NCCc3ccccc3)nc4ccccn14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E11 compound treatment 640.0 -1570.0 -0.56 1520.0 665.0 0.51 -0.032 -0.0424 3023145 ChemDiv3_003267 CCc1cc2c(SCC(=O)c3ccc(Br)cc3)ncnc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E12 compound treatment 280.0 -1930.0 -0.68 1480.0 625.0 0.48 -0.144 -0.1725 1550911 ChemDiv3_003268 Cc1ccc(NC(NC(=O)c2cccs2)C(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E13 compound treatment 600.0 -1610.0 -0.57 1880.0 1020.0 0.79 0.1534 0.1579 1203438 ChemDiv3_003269 Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc3OCCOc3c2)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E14 compound treatment 1360.0 -846.0 -0.3 800.0 -55.2 -0.04 -0.2422 -0.799 3119690 ChemDiv3_003270 CC1(C)CC(C)(c2ccccc2)c3ccccc3N1C(=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E15 compound treatment 3200.0 994.0 0.35 2360.0 1500.0 1.16 1.0662 0.8827 3119691 ChemDiv3_003271 CCOc1ccc(cc1C)C(=O)C2=C(O)C(=O)N(CCN(CC)CC)C2c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E16 compound treatment 5880.0 3670.0 1.3 1520.0 665.0 0.51 1.2824 0.9163 3023146 ChemDiv3_003272 N/C(=N\C(=O)Nc1ccc(Cl)c(Cl)c1)/Nc2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E17 compound treatment 800.0 -1410.0 -0.5 1240.0 385.0 0.3 -0.1438 -0.2481 3119692 ChemDiv3_003273 COc1ccc(cc1)C2(CNC(=O)C(c3ccccc3)c4ccccc4)CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E18 compound treatment 520.0 -1690.0 -0.6 320.0 -535.0 -0.41 -0.7135 -0.9832 3023147 ChemDiv3_003274 Cc1c(C)c2ccccc2n1C(=O)CSc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E19 compound treatment 1000.0 -1210.0 -0.43 1320.0 465.0 0.36 -0.0502 -0.0902 3119693 ChemDiv3_003275 Brc1ccc(CN2C(=O)N/C(=C/c3c[nH]c4ccc(Br)cc34)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E20 compound treatment 920.0 -1290.0 -0.46 1160.0 305.0 0.23 -0.1572 -0.3065 3023148 ChemDiv3_003276 NC(=N)NS(=O)(=O)c1ccc(/N=C/c2cccs2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E21 compound treatment 3280.0 1070.0 0.38 720.0 -135.0 -0.1 0.196 0.4964 1153257 ChemDiv3_003277 CCCc1oc2c(cc(NS(=O)(=O)c3ccc(CC)cc3)c4ccccc24)c1C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E22 compound treatment 5160.0 2950.0 1.05 920.0 64.8 0.05 0.7761 0.7399 1596083 ChemDiv3_003278 OCCNc1ccc2ccccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E23 mock treatment 2280.0 73.8 0.03 640.0 -215.0 -0.17 -0.0983 -0.5878 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 E24 mock treatment 360.0 -1850.0 -0.65 480.0 -375.0 -0.29 -0.6668 -0.9319 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F01 compound treatment 6520.0 4310.0 1.53 2480.0 1620.0 1.25 1.9641 0.9949 1378106 ChemDiv3_003279 Cc1cccc(Oc2ccc(cc2)N3C(=O)C4C5CC(C=C5)C4(C)C3=O)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F02 compound treatment 1800.0 -406.0 -0.14 4000.0 3140.0 2.41 1.6053 0.6637 1397787 ChemDiv3_003280 COc1ccc(cc1)c2nc(c(SC)[nH]2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F03 compound treatment 5800.0 3590.0 1.27 800.0 -55.2 -0.04 0.8715 0.6832 3119694 ChemDiv3_003281 OC(=O)c1cccc(c1)c2ccc(/C=c\3/sc4nc5ccccc5n4c3=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F04 compound treatment 10560.0 8350.0 2.96 1120.0 265.0 0.2 2.2392 0.7538 3023149 ChemDiv3_003282 CCOC(=O)c1c(C)oc-2c1/C(=C/NC(C)c3ccccc3)/C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F05 compound treatment 2480.0 274.0 0.1 800.0 -55.2 -0.04 0.0387 0.3654 1703292 ChemDiv3_003283 Cc1cccc(Oc2coc3cc(OC(=O)c4cccnc4)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F06 compound treatment 1520.0 -686.0 -0.24 600.0 -255.0 -0.2 -0.3107 -0.9942 1582822 ChemDiv3_003284 Fc1ccccc1c2nc(C#N)c(NCC3CCCO3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F07 compound treatment 1200.0 -1010.0 -0.36 1760.0 905.0 0.69 0.2388 0.3057 1065799 ChemDiv3_003285 S=C(Nc1ccccc1)N(Cc2ccccc2)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F08 compound treatment 720.0 -1490.0 -0.53 5320.0 4460.0 3.43 2.051 0.5914 3023184 ChemDiv3_003286 CN(C)S(=O)(=O)c1ccc(cc1)C(=O)/N=c/2\sc3cc(ccc3n2C)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F09 compound treatment 6480.0 4270.0 1.52 2680.0 1820.0 1.4 2.0627 0.9992 3119695 ChemDiv3_003287 CC1=CCC2C(C1)C(=O)N(C2=O)c3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F10 compound treatment 3280.0 1070.0 0.38 5720.0 4860.0 3.73 2.9103 0.7752 3023185 ChemDiv3_003288 CCc1ccc(NC(=O)CC(NCc2ccccc2)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F11 compound treatment 3680.0 1470.0 0.52 680.0 -175.0 -0.13 0.2746 0.5087 3119854 ChemDiv3_003289 C(c1ccccc1)n2c-3c(CCOc4ccccc34)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F12 compound treatment 1960.0 -246.0 -0.09 1040.0 185.0 0.14 0.0386 0.2314 1658105 ChemDiv3_003290 CC1CCCN(C1)S(=O)(=O)c2ccc(cc2)C(=O)Nc3ccccc3c4nc5ccccc5[nH]4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F13 compound treatment 680.0 -1530.0 -0.54 3880.0 3020.0 2.32 1.2592 0.5281 1261842 ChemDiv3_003291 COc1ccc(cc1)C(=O)O[C@H](C2CC3CCN2CC3C=C)c4ccnc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F14 compound treatment 6000.0 3790.0 1.35 2960.0 2100.0 1.62 2.0943 0.9959 1569329 ChemDiv3_003292 COc1ccc(cc1)S(=O)(=O)N2CCCC2C(=O)n3nc(C)cc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F15 compound treatment 2400.0 194.0 0.07 2280.0 1420.0 1.09 0.8221 0.7501 3119855 ChemDiv3_003293 Brc1ccc(NC(=O)C2CC(=O)N(/C(=N/c3ccccc3)/S2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F16 compound treatment 3800.0 1590.0 0.57 1320.0 465.0 0.36 0.6521 0.9754 1411088 ChemDiv3_003294 CCN1C(=O)C(C2CC1(C)Oc3ccccc23)C(=O)N(Cc4ccccc4)Cc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F17 compound treatment 2440.0 234.0 0.08 2000.0 1140.0 0.88 0.6801 0.7704 3023186 ChemDiv3_003295 CNC=C1C(=O)c2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F18 compound treatment 1360.0 -846.0 -0.3 1560.0 705.0 0.54 0.1703 0.2753 1692589 ChemDiv3_003296 C(Sc1nc2ccccc2s1)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F19 compound treatment 8240.0 6030.0 2.14 1160.0 305.0 0.23 1.679 0.7798 3023187 ChemDiv3_003297 COc1ccc(cc1)c2noc(n2)c3cccc(F)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F20 compound treatment 2200.0 -6.25 0.0 2000.0 1140.0 0.88 0.6199 0.7053 1402907 ChemDiv3_003298 ON1C(Nc2ccccc2C1=O)c3cccc(O)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F21 compound treatment 2240.0 33.8 0.01 840.0 -15.2 -0.01 2.0E-4 0.0137 1260345 ChemDiv3_003299 Cn1c(=O)n(CCOc2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F22 compound treatment 4920.0 2710.0 0.96 3600.0 2740.0 2.11 2.1708 0.937 3119856 ChemDiv3_003300 CCOc1ccc(cc1)S(=O)(=O)N(CC(=O)NC2CC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F23 mock treatment 1120.0 -1090.0 -0.39 2560.0 1700.0 1.31 0.653 0.4786 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 F24 mock treatment 5560.0 3350.0 1.19 360.0 -495.0 -0.38 0.5725 0.4583 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G01 compound treatment 9400.0 7190.0 2.55 640.0 -215.0 -0.17 1.6877 0.66 3119857 ChemDiv3_003301 O=S(=O)(N1CCCC1)c2ccc(cc2)c3cs/c(=N\c4ccccc4)/n3CCc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G02 compound treatment 9240.0 7030.0 2.5 560.0 -295.0 -0.23 1.6041 0.6403 3023188 ChemDiv3_003302 CC1(C)Cc2c(ccc3ccccc23)C(=N1)NCCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G03 compound treatment 520.0 -1690.0 -0.6 3240.0 2380.0 1.83 0.8716 0.4525 3119858 ChemDiv3_003303 CN(C)c1nc(SCCOC(=O)COc2ccc(Cl)cc2Cl)nc(n1)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G04 compound treatment 680.0 -1530.0 -0.54 1880.0 1020.0 0.79 0.1735 0.1816 1481926 ChemDiv3_003304 O=CNC1c2ccccc2Oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G05 compound treatment 400.0 -1810.0 -0.64 280.0 -575.0 -0.44 -0.7653 -0.9835 1448737 ChemDiv3_003305 OC(=O)CCN1C(C(=C(O)C1=O)C(=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G06 compound treatment 1080.0 -1130.0 -0.4 1440.0 585.0 0.45 0.035 0.0582 1566191 ChemDiv3_003306 CCC1C(NC(CC1(O)c2ccc(F)cc2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G07 compound treatment 280.0 -1930.0 -0.68 1440.0 585.0 0.45 -0.1657 -0.2027 1652661 ChemDiv3_003307 CCN1CCn2c3C1CCCc3c4cc(Cl)ccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G08 compound treatment 360.0 -1850.0 -0.65 1240.0 385.0 0.3 -0.2542 -0.3538 1433683 ChemDiv3_003308 CC1(C)CC(=O)c2c(coc2C1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G09 compound treatment 760.0 -1450.0 -0.51 1960.0 1100.0 0.85 0.237 0.2391 1852959 ChemDiv3_003309 CCc1ccc(cc1)C2C(=C(N)N(N3CCOCC3)C4=C2C(=O)CC(C)(C)C4)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G10 compound treatment 640.0 -1570.0 -0.56 4720.0 3860.0 2.97 1.7052 0.5649 3119859 ChemDiv3_003310 CC(C)CN1C(=O)/C(=C/C=C/c2ccccc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G11 compound treatment 1200.0 -1010.0 -0.36 480.0 -375.0 -0.29 -0.4561 -0.9943 3023189 ChemDiv3_003311 Nc1nnnn1/N=C/c2ccc(o2)c3ccc4C(=O)OCc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G12 compound treatment 1280.0 -926.0 -0.33 320.0 -535.0 -0.41 -0.5229 -0.9939 1159102 ChemDiv3_003312 CCOc1ccc(NC(NC(=O)c2cccs2)C(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G13 compound treatment 400.0 -1810.0 -0.64 840.0 -15.2 -0.01 -0.4613 -0.7198 3023190 ChemDiv3_003313 CN(CC(=O)Nc1ccc(cc1)S(=O)(=O)N)S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G14 compound treatment 6000.0 3790.0 1.35 720.0 -135.0 -0.1 0.8783 0.6507 3119860 ChemDiv3_003314 Cc1nc(N/C(=N/C(=O)c2ccccc2)/N)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G15 compound treatment 1360.0 -846.0 -0.3 360.0 -495.0 -0.38 -0.4811 -0.9932 1346700 ChemDiv3_003315 Cc1ccc(cc1)C(O)(C(=O)NN2CCOCC2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G16 compound treatment 760.0 -1450.0 -0.51 520.0 -335.0 -0.26 -0.5447 -0.9491 3023191 ChemDiv3_003316 Cc1cc(C)n(n1)C(=O)Nc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G17 compound treatment 920.0 -1290.0 -0.46 760.0 -95.2 -0.07 -0.3743 -0.81 1424365 ChemDiv3_003317 CC(C)c1ccc(cc1)S(=O)(=O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G18 compound treatment 1040.0 -1170.0 -0.41 280.0 -575.0 -0.44 -0.6048 -0.9995 1360094 ChemDiv3_003318 COC(=O)c1ccccc1NC(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G19 compound treatment 7800.0 5590.0 1.98 440.0 -415.0 -0.32 1.1778 0.586 3119861 ChemDiv3_003319 COC(=O)c1ccc(/C=C\2/NC(=O)N(Cc3ccc(Br)cc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G20 compound treatment 1480.0 -726.0 -0.26 6480.0 5620.0 4.32 2.8713 0.6637 3023192 ChemDiv3_003320 Fc1ccc(NC(=S)N2CCc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G21 compound treatment 2560.0 354.0 0.13 920.0 64.8 0.05 0.1239 0.918 1104701 ChemDiv3_003321 Cc1ccc(cc1)S(=O)(=O)N=C2C=CC(=NS(=O)(=O)c3ccc(C)cc3)C=C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G22 compound treatment 4160.0 1950.0 0.69 280.0 -575.0 -0.44 0.1778 0.2164 1056920 ChemDiv3_003322 Cc1ccc(Oc2nc(Cl)nc(Oc3ccc(C)cc3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G23 mock treatment 1320.0 -886.0 -0.31 2640.0 1780.0 1.37 0.7466 0.5311 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 G24 mock treatment 320.0 -1890.0 -0.67 2200.0 1340.0 1.03 0.2569 0.2088 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H01 compound treatment 5280.0 3070.0 1.09 600.0 -255.0 -0.2 0.6325 0.5709 1634360 ChemDiv3_003323 COC(=O)c1cc(nc2ccccc12)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H02 compound treatment 2160.0 -46.3 -0.02 1400.0 545.0 0.42 0.2842 0.6788 3119862 ChemDiv3_003324 CN1C(=O)NC(C(C(=O)c2cccs2)C1(O)C(F)(F)F)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H03 compound treatment 7800.0 5590.0 1.98 1120.0 265.0 0.2 1.5469 0.7755 3119863 ChemDiv3_003325 Cc1ccc(cc1)C(=O)N2N=C3N(C2N4CCCCC4)S(=O)(=O)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H04 compound treatment 720.0 -1490.0 -0.53 560.0 -295.0 -0.23 -0.5331 -0.9289 1358055 ChemDiv3_003326 CCOC(=O)c1c(C)oc2c1c3CN(COc3c4ccccc24)C5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H05 compound treatment 760.0 -1450.0 -0.51 520.0 -335.0 -0.26 -0.5447 -0.9491 1274629 ChemDiv3_003327 COc1ccc(Nc2ncnc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H06 compound treatment 1320.0 -886.0 -0.31 600.0 -255.0 -0.2 -0.3608 -0.9741 1496041 ChemDiv3_003328 CCSC1=C(C#N)C(C2=C(CCCC2=O)N1)c3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H07 compound treatment 1080.0 -1130.0 -0.4 680.0 -175.0 -0.13 -0.3776 -0.8957 3023235 ChemDiv3_003329 S=C(NC1CCCCC1)N(Cc2ccccc2)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H08 compound treatment 760.0 -1450.0 -0.51 840.0 -15.2 -0.01 -0.371 -0.723 3119864 ChemDiv3_003330 Cn1/c(=N\C(=O)c2cc(nc3ccccc23)c4ccccc4)/sc5cc(ccc15)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H09 compound treatment 680.0 -1530.0 -0.54 760.0 -95.2 -0.07 -0.4345 -0.7953 1302654 ChemDiv3_003331 CC(NC(=O)CSc1nc(N)cc(=O)[nH]1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H10 compound treatment 1240.0 -966.0 -0.34 640.0 -215.0 -0.17 -0.3592 -0.944 3119865 ChemDiv3_003332 Cc1ccc(NC(=O)CC(NCCc2ccccc2)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H11 compound treatment 3800.0 1590.0 0.57 1080.0 225.0 0.17 0.5218 0.8828 1349929 ChemDiv3_003333 OCC(=O)c1c[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H12 compound treatment 1040.0 -1170.0 -0.41 440.0 -415.0 -0.32 -0.5179 -0.9917 1430458 ChemDiv3_003334 CCCCN(CC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccccc2c3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H13 compound treatment 10320.0 8110.0 2.88 520.0 -335.0 -0.26 1.8533 0.6413 1534077 ChemDiv3_003335 O=C1CCC(=O)N1CCc2c[nH]c3ccc(OCc4ccccc4)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H14 compound treatment 1080.0 -1130.0 -0.4 1080.0 225.0 0.17 -0.1605 -0.3687 1226556 ChemDiv3_003336 OC(=O)CSc1nnc(c2ccc3OCOc3c2)n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H15 compound treatment 9560.0 7350.0 2.61 720.0 -135.0 -0.1 1.7713 0.6784 3119866 ChemDiv3_003337 COc1ccccc1NC(=O)C2CC(=O)N(C)/C(=N/c3ccccc3)/S2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H16 compound treatment 10160.0 7950.0 2.82 640.0 -215.0 -0.17 1.8783 0.6646 1518221 ChemDiv3_003338 O=S1(=O)CC2C(C1)N(C(=S)N2c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H17 compound treatment 600.0 -1610.0 -0.57 1360.0 505.0 0.39 -0.1289 -0.187 3119867 ChemDiv3_003339 Oc1ccccc1NC=C2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H18 compound treatment 720.0 -1490.0 -0.53 400.0 -455.0 -0.35 -0.6199 -0.98 3023236 ChemDiv3_003340 CCOC(=S)SCc1cn2cccnc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H19 compound treatment 1160.0 -1050.0 -0.37 520.0 -335.0 -0.26 -0.4444 -0.984 3119868 ChemDiv3_003341 NC(=O)C1CCN(CC1)C(=O)c2cccc(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H20 compound treatment 1400.0 -806.0 -0.29 1760.0 905.0 0.69 0.289 0.3846 3120012 ChemDiv3_003342 O=C1c2ccccc2-c3c1c4ccccc4nc3c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H21 compound treatment 1480.0 -726.0 -0.26 760.0 -95.2 -0.07 -0.2338 -0.8732 3120013 ChemDiv3_003343 Cc1cc(/C=C\2/NC(=O)N(Cc3ccc(Br)cc3)C2=O)c(C)n1c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H22 compound treatment 840.0 -1370.0 -0.48 4240.0 3380.0 2.6 1.4948 0.5655 3023237 ChemDiv3_003344 Clc1ccccc1/C=C(/C(=O)NCc2ccccn2)\c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H23 mock treatment 760.0 -1450.0 -0.51 480.0 -375.0 -0.29 -0.5664 -0.9627 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 H24 mock treatment 2480.0 274.0 0.1 4800.0 3940.0 3.03 2.2102 0.7294 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I01 compound treatment 1680.0 -526.0 -0.19 1480.0 625.0 0.48 0.2072 0.4025 3120014 ChemDiv3_003345 COc1cc(/N=c/2\scc(c3ccc(cc3)S(=O)(=O)N4CCCC4)n2C)c(OC)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I02 compound treatment 320.0 -1890.0 -0.67 840.0 -15.2 -0.01 -0.4814 -0.7193 3023238 ChemDiv3_003346 COc1cc2CC(C)(C)N=C(NCCC(=O)O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I03 compound treatment 13720.0 11500.0 4.08 1160.0 305.0 0.23 3.0536 0.7464 3023239 ChemDiv3_003347 COc1cc(C)nc(OCCNS(=O)(=O)c2cc(C)ccc2C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I04 compound treatment 3560.0 1350.0 0.48 800.0 -55.2 -0.04 0.3096 0.6422 1482999 ChemDiv3_003348 Cc1ccc(OC(=O)C2c3ccccc3Oc4ccccc24)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I05 compound treatment 680.0 -1530.0 -0.54 440.0 -415.0 -0.32 -0.6082 -0.9681 3120015 ChemDiv3_003349 CCC(=O)c1ccc(OC(=O)c2cn(nc2c3ccccc3)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I06 compound treatment 440.0 -1770.0 -0.63 320.0 -535.0 -0.41 -0.7336 -0.9791 1537398 ChemDiv3_003350 CCC1C(NC(C(CC)C1=NO)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I07 compound treatment 6560.0 4350.0 1.54 920.0 64.8 0.05 1.1273 0.7295 3120016 ChemDiv3_003351 Cn1c2-c3cnn(c3CC(C)(C)c2c4ccccc14)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I08 compound treatment 1080.0 -1130.0 -0.4 920.0 64.8 0.05 -0.2473 -0.6143 1580288 ChemDiv3_003352 Cc1cc(C)cc(OCCn2c(nc3ccccc3c2=O)c4ccc(Cl)cc4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I09 compound treatment 440.0 -1770.0 -0.63 480.0 -375.0 -0.29 -0.6467 -0.9378 1853000 ChemDiv3_003353 NC1=C(C#N)C(C2=C(CC(CC2=O)c3ccccc3)N1N4CCOCC4)c5ccccc5Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I10 compound treatment 600.0 -1610.0 -0.57 440.0 -415.0 -0.32 -0.6283 -0.9623 3120017 ChemDiv3_003354 COc1ccc(CCN2C(=O)/C(=C/C3CCC=CC3)/SC2=S)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I11 compound treatment 9360.0 7150.0 2.54 1720.0 865.0 0.66 2.2639 0.8631 3120018 ChemDiv3_003355 COc1cc(/C=C/2\C(=O)N(N=C2C(F)(F)F)c3ccc(cc3)S(=O)(=O)N)ccc1OCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I12 compound treatment 8400.0 6190.0 2.2 3920.0 3060.0 2.35 3.2174 0.9994 1472706 ChemDiv3_003356 CC(=O)Nc1ccc(NC(NC(=O)c2cccs2)C(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I13 compound treatment 520.0 -1690.0 -0.6 560.0 -295.0 -0.23 -0.5832 -0.9117 1582486 ChemDiv3_003357 COc1ccc2[nH]c3nc(=S)[nH]nc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I14 compound treatment 4600.0 2390.0 0.85 600.0 -255.0 -0.2 0.4619 0.5301 3120019 ChemDiv3_003358 CCC(=O)/N=C(\N)/Nc1nc(C)c2ccccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I15 compound treatment 1040.0 -1170.0 -0.41 440.0 -415.0 -0.32 -0.5179 -0.9917 3023240 ChemDiv3_003359 CC(C)(C)C(=O)/C=C/1\Nc2ccccc2OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I16 compound treatment 560.0 -1650.0 -0.58 1040.0 185.0 0.14 -0.3126 -0.5202 3120020 ChemDiv3_003360 Cc1ccc2NC(C)(C)c3ss/c(=N/c4ccc(cc4)S(=O)(=O)N)/c3-c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I17 compound treatment 1880.0 -326.0 -0.12 360.0 -495.0 -0.38 -0.3506 -0.8824 1374353 ChemDiv3_003361 CN(C)C1OC2=C(C=C1C)C(=O)c3cccc4cccc2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I18 compound treatment 720.0 -1490.0 -0.53 320.0 -535.0 -0.41 -0.6633 -0.9924 1323310 ChemDiv3_003362 C1Cc2ccccc2CN1c3nc(Nc4ccccc4)nc(Nc5ccccc5)n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I19 compound treatment 440.0 -1770.0 -0.63 560.0 -295.0 -0.23 -0.6033 -0.9054 3120021 ChemDiv3_003363 CC(C)(C)c1ccc(/C=C\2/NC(=O)N(Cc3ccc(Br)cc3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I20 compound treatment 720.0 -1490.0 -0.53 2320.0 1460.0 1.12 0.4224 0.3401 3023241 ChemDiv3_003364 FC(F)(F)c1cccc(CC(=O)Nc2ccccc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I21 compound treatment 59000.0 56800.0 20.15 5400.0 4540.0 3.49 16.7135 0.8174 3120022 ChemDiv3_003365 Fc1ccc(cc1)S(=O)(=O)/N=C/2\C=C(NS(=O)(=O)c3ccccc3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I22 compound treatment 1840.0 -366.0 -0.13 520.0 -335.0 -0.26 -0.2738 -0.9499 3023242 ChemDiv3_003366 C=CCN1C(=O)/C(=C\c2ccc(OCc3ccccc3C#N)cc2)/C(=O)NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I23 mock treatment 680.0 -1530.0 -0.54 440.0 -415.0 -0.32 -0.6082 -0.9681 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 I24 mock treatment 3680.0 1470.0 0.52 720.0 -135.0 -0.1 0.2963 0.5559 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J01 compound treatment 280.0 -1930.0 -0.68 6640.0 5780.0 4.44 2.6572 0.5913 3120023 ChemDiv3_003367 CCCCC(=O)/C=C/1\Nc2ccccc2NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J02 compound treatment 5520.0 3310.0 1.18 1000.0 145.0 0.11 0.9099 0.7705 3120024 ChemDiv3_003368 CCOC(=O)N1CCN(CC1)C(=O)CCN2C(=O)/C(=C/C=C/c3ccccc3)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J03 compound treatment 5840.0 3630.0 1.29 1240.0 385.0 0.3 1.1204 0.8472 1324615 ChemDiv3_003369 Clc1ccc(cc1)C2SCC(=O)N2Nc3nc(Nc4ccccc4)nc(n3)N5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J04 compound treatment 560.0 -1650.0 -0.58 320.0 -535.0 -0.41 -0.7035 -0.9852 1715130 ChemDiv3_003370 Clc1cc2CN(CCC3=CCCCC3)COc2c4ncccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J05 compound treatment 3720.0 1510.0 0.54 520.0 -335.0 -0.26 0.1978 0.3321 1591815 ChemDiv3_003371 COC(=O)c1ccc(Nc2cc(C)nc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J06 compound treatment 360.0 -1850.0 -0.65 280.0 -575.0 -0.44 -0.7754 -0.9816 1445792 ChemDiv3_003372 Fc1ccc(NC(=O)CSC2=C(C#N)C3(CCCCC3)C(C#N)C(=O)N2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J07 compound treatment 480.0 -1730.0 -0.61 400.0 -455.0 -0.35 -0.6801 -0.9646 3022562 ChemDiv3_003373 S=C(NC1CCCCC1)N(CC2CCC=CC2)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J08 compound treatment 1200.0 -1010.0 -0.36 320.0 -535.0 -0.41 -0.5429 -0.9975 3120025 ChemDiv3_003374 COc1cccc(OC)c1C(=O)/N=c/2\sc3cc(ccc3n2C)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J09 compound treatment 560.0 -1650.0 -0.58 280.0 -575.0 -0.44 -0.7252 -0.9905 3022578 ChemDiv3_003375 COc1ccc(cc1)C2=[N+]([O-])C(C)(C)C(=N2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J10 compound treatment 6800.0 4590.0 1.63 440.0 -415.0 -0.32 0.9269 0.5582 3120026 ChemDiv3_003376 CN(C)C(CC(=O)Nc1ccccc1C)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J11 compound treatment 800.0 -1410.0 -0.5 280.0 -575.0 -0.44 -0.665 -0.9981 3120027 ChemDiv3_003377 COC(=O)C1O[N+](=C(C1c2c[nH]c3ccccc23)C(=O)OC)[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J12 compound treatment 1480.0 -726.0 -0.26 440.0 -415.0 -0.32 -0.4076 -0.9944 1251370 ChemDiv3_003378 CN(Cc1ccccc1)S(=O)(=O)c2ccc(cc2)C(=O)Nc3ccc(cc3)c4nc5ccccc5[nH]4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J13 compound treatment 360.0 -1850.0 -0.65 360.0 -495.0 -0.38 -0.7319 -0.9665 3120028 ChemDiv3_003379 CN1CCc2cc(ccc12)/C(=C/c3ccccc3)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J14 compound treatment 440.0 -1770.0 -0.63 1160.0 305.0 0.23 -0.2776 -0.415 3022585 ChemDiv3_003380 OC(=O)CSc1nnc(c2sc3ccccc3c2Cl)n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J15 compound treatment 4760.0 2550.0 0.91 520.0 -335.0 -0.26 0.4586 0.487 3120029 ChemDiv3_003381 Clc1ccc(NC(=S)N2CCSC2c3ccc(Br)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J16 compound treatment 520.0 -1690.0 -0.6 800.0 -55.2 -0.04 -0.4529 -0.7553 1628252 ChemDiv3_003382 Cn1c(=O)n(C)c2nc(SCC(=O)c3ccccc3)n(CCCc4ccccc4)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J17 compound treatment 10920.0 8710.0 3.09 400.0 -455.0 -0.35 1.9387 0.6232 3022590 ChemDiv3_003383 CC1(C)CC(=O)C(=CNc2cccc(NC3=C(C#N)C(=O)CC(C)(C)C3)c2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J18 compound treatment 1600.0 -606.0 -0.22 600.0 -255.0 -0.2 -0.2906 -0.9989 3120030 ChemDiv3_003384 CCN(CC)C(=S)SCc1cn2cccnc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J19 compound treatment 840.0 -1370.0 -0.48 480.0 -375.0 -0.29 -0.5464 -0.9691 1198374 ChemDiv3_003385 COc1cccc(c1)C(=O)NC2CC(C)(C)NC(C)(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J20 compound treatment 4800.0 2590.0 0.92 640.0 -215.0 -0.17 0.5338 0.571 3120031 ChemDiv3_003386 Cc1ccc(CN(CC(=O)NC2CC2)S(=O)(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J21 compound treatment 2240.0 33.8 0.01 8880.0 8020.0 6.16 4.3648 0.7085 3022623 ChemDiv3_003387 CCOC(=O)c1ccc(cc1)N2N=C(/C(=C/C=C/c3ccco3)/C2=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J22 compound treatment 1240.0 -966.0 -0.34 560.0 -295.0 -0.23 -0.4026 -0.9798 3120032 ChemDiv3_003388 CNC(=O)CN(c1cccc(C)c1C)S(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J23 mock treatment 2960.0 754.0 0.27 280.0 -575.0 -0.44 -0.1232 -0.2386 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 J24 mock treatment 1600.0 -606.0 -0.22 1160.0 305.0 0.23 0.0134 0.0422 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K01 compound treatment 1480.0 -726.0 -0.26 960.0 105.0 0.08 -0.1253 -0.4641 3120169 ChemDiv3_003389 CCOc1ccc(/N=c/2\scc(c3ccc(cc3)S(=O)(=O)N(CC)CC)n2CCCO)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K02 compound treatment 6440.0 4230.0 1.5 2600.0 1740.0 1.34 2.0092 0.9984 1658725 ChemDiv3_003390 C1C2CC3CC1CC(C2)(C3)c4cc5ccccc5[nH]4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K03 compound treatment 600.0 -1610.0 -0.57 1120.0 265.0 0.2 -0.2592 -0.4284 1415577 ChemDiv3_003391 CCCOc1ccc(CNC(=S)NCc2ccc(OC(C)C)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K04 compound treatment 720.0 -1490.0 -0.53 440.0 -415.0 -0.32 -0.5982 -0.9709 1601172 ChemDiv3_003392 Clc1ccc(OC(=O)C2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K05 compound treatment 440.0 -1770.0 -0.63 480.0 -375.0 -0.29 -0.6467 -0.9378 3120170 ChemDiv3_003393 O=C(Oc1cccc2cccnc12)c3cn(nc3c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K06 compound treatment 560.0 -1650.0 -0.58 840.0 -15.2 -0.01 -0.4212 -0.7211 1273524 ChemDiv3_003394 CC(=O)OC1C(OC(=O)C)N(C(=O)C)C(=O)N1C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K07 compound treatment 3120.0 914.0 0.32 7840.0 6980.0 5.36 4.021 0.7485 1721819 ChemDiv3_003395 CCOC(=O)c1sc(C)c2C(=O)NC(C)(Nc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K08 compound treatment 3400.0 1190.0 0.42 680.0 -175.0 -0.13 0.2044 0.4599 3022632 ChemDiv3_003396 CCOC(=O)Cn1cc(F)c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K09 compound treatment 1240.0 -966.0 -0.34 560.0 -295.0 -0.23 -0.4026 -0.9798 1853144 ChemDiv3_003397 CC1(C)CC(=O)C2=C(C1)N(C(=C(C#N)C2c3ccsc3)N)c4nc[nH]n4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K10 compound treatment 1400.0 -806.0 -0.29 1560.0 705.0 0.54 0.1804 0.2947 3120171 ChemDiv3_003398 C=CCN1C(=O)/C(=c/2\sc3nc(nn3c2=O)c4ccccc4)/c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K11 compound treatment 840.0 -1370.0 -0.48 520.0 -335.0 -0.26 -0.5247 -0.9561 1685244 ChemDiv3_003399 CC(C)c1ccc(C)cc1OCC(=O)Nc2cc(ccc2C)c3nc4ncccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K12 compound treatment 1720.0 -486.0 -0.17 5240.0 4380.0 3.37 2.2584 0.67 3120172 ChemDiv3_003400 FC(F)(F)c1cccc(NC(NC(=O)c2cccs2)C(=O)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K13 compound treatment 600.0 -1610.0 -0.57 760.0 -95.2 -0.07 -0.4546 -0.7913 3022674 ChemDiv3_003401 CN(C)c1cccc2c(/C=N/O)ccc(N(C)C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K14 compound treatment 920.0 -1290.0 -0.46 840.0 -15.2 -0.01 -0.3309 -0.7249 1204566 ChemDiv3_003402 COc1cccc(c1)C(=O)N2C(C)CC(Nc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K15 compound treatment 920.0 -1290.0 -0.46 760.0 -95.2 -0.07 -0.3743 -0.81 3120173 ChemDiv3_003403 O=S1(=O)CCC(C1)/N=C/c2cn(nc2c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K16 compound treatment 2440.0 234.0 0.08 3680.0 2820.0 2.17 1.5921 0.7336 3022677 ChemDiv3_003404 Cc1cc(C)nc(N/C(=N\C(=O)Nc2cccc(Cl)c2)/Nc3ccccc3C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K17 compound treatment 2600.0 394.0 0.14 840.0 -15.2 -0.01 0.0905 0.6459 1257823 ChemDiv3_003405 Cc1ccc(cc1)S(=O)(=O)N2CCN(C2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K18 compound treatment 1440.0 -766.0 -0.27 1000.0 145.0 0.11 -0.1136 -0.3868 3022679 ChemDiv3_003406 Cc1nnc(Sc2nc(Nc3ccccc3)nc(Nc4ccccc4)n2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K19 compound treatment 1120.0 -1090.0 -0.39 840.0 -15.2 -0.01 -0.2807 -0.7281 3120174 ChemDiv3_003407 CCOC(=O)CN1C(=O)S/C(=C/c2ccc3n(C)c(=O)n(C)c3c2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K20 compound treatment 1600.0 -606.0 -0.22 680.0 -175.0 -0.13 -0.2472 -0.9744 3022681 ChemDiv3_003408 COc1ccccc1/C=C/c2ccccc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K21 compound treatment 1400.0 -806.0 -0.29 7240.0 6380.0 4.9 3.2638 0.6647 1498680 ChemDiv3_003409 CC1(C)CC(=O)c2c(C1)oc3ccc(NS(=O)(=O)c4ccc5ccccc5c4)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K22 compound treatment 480.0 -1730.0 -0.61 920.0 64.8 0.05 -0.3978 -0.6475 1249568 ChemDiv3_003410 CCOC(=O)c1ccc2C(=O)N(C3CCCCC3)C(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K23 mock treatment 680.0 -1530.0 -0.54 2120.0 1260.0 0.97 0.3038 0.2732 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 K24 mock treatment 600.0 -1610.0 -0.57 1800.0 945.0 0.73 0.11 0.1192 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L01 compound treatment 2080.0 -126.0 -0.04 1120.0 265.0 0.2 0.1121 0.5384 3120175 ChemDiv3_003411 FC(F)(F)c1cc(nc(SCC2COc3ccccc3O2)c1C#N)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L02 compound treatment 640.0 -1570.0 -0.56 520.0 -335.0 -0.26 -0.5748 -0.9388 1425939 ChemDiv3_003412 CCOC(=O)c1c(C)oc2c1c(C(N3CCOCC3)c4ccc(OC)cc4)c(O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L03 compound treatment 2840.0 634.0 0.22 280.0 -575.0 -0.44 -0.1533 -0.3093 3022724 ChemDiv3_003413 COc1cccc(c1)C(=O)NC(=S)Nc2ccc(O)c(c2)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L04 compound treatment 1280.0 -926.0 -0.33 320.0 -535.0 -0.41 -0.5229 -0.9939 1551789 ChemDiv3_003414 CCOC(=O)c1c(C)oc2c1c(CN3CCN(CC3)c4ccccc4F)c(O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L05 compound treatment 3640.0 1430.0 0.51 400.0 -455.0 -0.35 0.1126 0.1824 1695085 ChemDiv3_003415 Cc1cc(C)cc(Oc2coc3c(CN4CCCCCC4)c(O)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L06 compound treatment 320.0 -1890.0 -0.67 440.0 -415.0 -0.32 -0.6985 -0.9425 1264677 ChemDiv3_003416 CC1(C)CC(=O)c2cc(C#N)c(SCSc3nc4CC(C)(C)CC(=O)c4cc3C#N)nc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L07 compound treatment 360.0 -1850.0 -0.65 440.0 -415.0 -0.32 -0.6885 -0.9452 3022730 ChemDiv3_003417 CNC(=S)N(Cc1ccccc1)Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L08 compound treatment 640.0 -1570.0 -0.56 480.0 -375.0 -0.29 -0.5965 -0.9532 1376336 ChemDiv3_003418 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc4NC(=O)c5cccc3c45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L09 compound treatment 640.0 -1570.0 -0.56 440.0 -415.0 -0.32 -0.6183 -0.9652 3022732 ChemDiv3_003419 CC1(C)N(O)C([N+](=C1c2ccccc2)[O-])c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L10 compound treatment 1280.0 -926.0 -0.33 680.0 -175.0 -0.13 -0.3274 -0.9223 1170952 ChemDiv3_003420 CC1CCCCN1S(=O)(=O)c2ccc(cc2)C(=O)Nc3nc4ccc5ccccc5c4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L11 compound treatment 1240.0 -966.0 -0.34 360.0 -495.0 -0.38 -0.5112 -0.9987 1148202 ChemDiv3_003421 OC(=O)C(c1c(O)c2ccccc2oc1=O)c3c(O)c4ccccc4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L12 compound treatment 880.0 -1330.0 -0.47 600.0 -255.0 -0.2 -0.4712 -0.9246 1446893 ChemDiv3_003422 CC1CCCCN1S(=O)(=O)c2ccc(cc2)C(=O)Nc3cccc(c3)c4nc5ccccc5[nH]4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L13 compound treatment 1040.0 -1170.0 -0.41 360.0 -495.0 -0.38 -0.5614 -0.9991 1283305 ChemDiv3_003423 CC(Cc1c[nH]c2ccccc12)NC(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L14 compound treatment 10880.0 8670.0 3.08 3320.0 2460.0 1.89 3.5138 0.9727 1042488 ChemDiv3_003424 Nc1cc(=O)[nH]c(=O)n1Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L15 compound treatment 1760.0 -446.0 -0.16 480.0 -375.0 -0.29 -0.3156 -0.9603 3022737 ChemDiv3_003425 O=C1CCCN1CN2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L16 compound treatment 1240.0 -966.0 -0.34 520.0 -335.0 -0.26 -0.4243 -0.99 3120176 ChemDiv3_003426 O=C(CSc1nnc2ccccn12)Nc3ccc4ccccc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L17 compound treatment 960.0 -1250.0 -0.44 4240.0 3380.0 2.6 1.5249 0.5785 1376805 ChemDiv3_003427 CC1(C)CC(=O)c2c(N)n(nc2C1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L18 compound treatment 5560.0 3350.0 1.19 920.0 64.8 0.05 0.8765 0.736 1683693 ChemDiv3_003428 N1C(=CC(c2cccs2)n3ncnc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L19 compound treatment 2520.0 314.0 0.11 320.0 -535.0 -0.41 -0.2118 -0.4976 1148459 ChemDiv3_003429 CCn1c2ccccc2c3cc(NC(=O)C(C)C)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L20 compound treatment 920.0 -1290.0 -0.46 400.0 -455.0 -0.35 -0.5697 -0.9913 3120177 ChemDiv3_003430 Brc1ccc(cc1)S(=O)(=O)N(CCc2ccccc2)CC(=O)NC3CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L21 compound treatment 1680.0 -526.0 -0.19 1120.0 265.0 0.2 0.0118 0.0426 3022799 ChemDiv3_003431 COc1ccc(cc1)c2c(C)oc3cc(OC)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L22 compound treatment 400.0 -1810.0 -0.64 400.0 -455.0 -0.35 -0.7002 -0.9593 3120178 ChemDiv3_003432 Cc1cccc(N(CC(=O)Nc2ccccc2)S(=O)(=O)C)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L23 mock treatment 2600.0 394.0 0.14 400.0 -455.0 -0.35 -0.1483 -0.3941 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 L24 mock treatment 800.0 -1410.0 -0.5 520.0 -335.0 -0.26 -0.5347 -0.9526 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M01 compound treatment 4400.0 2190.0 0.78 320.0 -535.0 -0.41 0.2598 0.2952 3022801 ChemDiv3_003433 CCn/1c(cs\c1=N/c2ccc(C)cc2)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M02 compound treatment 440.0 -1770.0 -0.63 400.0 -455.0 -0.35 -0.6901 -0.962 1692578 ChemDiv3_003434 C1C2CC3CC1CC(C2)(C3)c4csc(n4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M03 compound treatment 760.0 -1450.0 -0.51 840.0 -15.2 -0.01 -0.371 -0.723 1182241 ChemDiv3_003435 COc1ccc(cc1)N(C(=O)c2ccccc2)S(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M04 compound treatment 480.0 -1730.0 -0.61 2920.0 2060.0 1.59 0.6879 0.4048 1022728 ChemDiv3_003436 Cc1ccc(cc1)S(=O)(=O)NC2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M05 compound treatment 10520.0 8310.0 2.95 880.0 24.8 0.02 2.0989 0.7117 3120179 ChemDiv3_003437 CC1(CC(=Nc2ccccc2N1)c3cccs3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M06 compound treatment 1120.0 -1090.0 -0.39 560.0 -295.0 -0.23 -0.4327 -0.968 1002478 ChemDiv3_003438 Clc1ccc(Nc2ncnc3n(ncc23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M07 compound treatment 800.0 -1410.0 -0.5 440.0 -415.0 -0.32 -0.5781 -0.9766 1660145 ChemDiv3_003439 CCOC(=O)c1sc(C)c2C(=O)NC(Nc12)c3ccc(cc3)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M08 compound treatment 1080.0 -1130.0 -0.4 1960.0 1100.0 0.85 0.3173 0.3384 1199493 ChemDiv3_003440 Cc1nc2sccn2c1c3csc(Nc4ccc(cc4)C(=O)O)n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M09 compound treatment 1240.0 -966.0 -0.34 2760.0 1900.0 1.46 0.7917 0.5271 1703311 ChemDiv3_003441 Cc1ccc(NC(=O)CSc2nc3sc4CCCCc4c3c(=O)n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M10 compound treatment 760.0 -1450.0 -0.51 3440.0 2580.0 1.98 1.0404 0.5076 3022808 ChemDiv3_003442 Oc1ccc(/C=C/2\SC(=S)N(CC3CCCO3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M11 compound treatment 640.0 -1570.0 -0.56 560.0 -295.0 -0.23 -0.5531 -0.9218 1271724 ChemDiv3_003443 Cc1cc(C)c2oc(nc2c1)c3cc(NC(=O)COc4ccccc4C)ccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M12 compound treatment 400.0 -1810.0 -0.64 3640.0 2780.0 2.14 1.0587 0.4743 3022874 ChemDiv3_003444 Cc1ccc(cc1)c2nn(cc2/C=C/3\SC(=S)N(CCCC(=O)O)C3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M13 compound treatment 320.0 -1890.0 -0.67 520.0 -335.0 -0.26 -0.6551 -0.9138 1216346 ChemDiv3_003445 CN(C)c1ccc2COC(=O)c3ccc(N(C)C)c1c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M14 compound treatment 7840.0 5630.0 2.0 680.0 -175.0 -0.13 1.3181 0.658 1120750 ChemDiv3_003446 COc1ccc2N(C(=O)C)C(C)(C)c3ssc(=S)c3-c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M15 compound treatment 600.0 -1610.0 -0.57 560.0 -295.0 -0.23 -0.5632 -0.9184 3117899 ChemDiv3_003447 Oc1ccc(cc1)C2NC(=O)NC(O)(C2C(=O)c3ccccc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M16 compound treatment 600.0 -1610.0 -0.57 1800.0 945.0 0.73 0.11 0.1192 3022878 ChemDiv3_003448 Cc1cc(C)nc(NC(=N)NO)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M17 compound treatment 920.0 -1290.0 -0.46 5840.0 4980.0 3.83 2.3834 0.6184 1151303 ChemDiv3_003449 Cc1ccc(cc1)C(=O)N2CCN(C2)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M18 compound treatment 640.0 -1570.0 -0.56 1840.0 985.0 0.76 0.1417 0.1511 1358369 ChemDiv3_003450 C(Oc1cccc2ccccc12)c3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M19 compound treatment 960.0 -1250.0 -0.44 560.0 -295.0 -0.23 -0.4729 -0.9518 3117900 ChemDiv3_003451 CCOC(=O)CN1C(=O)S/C(=C/c2cc(C)n(c2C)c3cc(C)ccn3)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M20 compound treatment 1120.0 -1090.0 -0.39 1080.0 225.0 0.17 -0.1504 -0.3563 1153417 ChemDiv3_003452 Cc1cc(c2cccs2)c3c(N)c(sc3n1)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M21 compound treatment 720.0 -1490.0 -0.53 600.0 -255.0 -0.2 -0.5113 -0.9091 1524326 ChemDiv3_003453 CC(NS(=O)(=O)c1ccc(cc1)C(C)(C)C)C2C3CC4CC(C3)CC2C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M22 compound treatment 3600.0 1390.0 0.49 680.0 -175.0 -0.13 0.2545 0.4967 1630427 ChemDiv3_003454 CC(C)OC(=O)c1cccc(NC(=O)c2ccc(Br)cc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M23 mock treatment 1040.0 -1170.0 -0.41 800.0 -55.2 -0.04 -0.3225 -0.7754 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 M24 mock treatment 1120.0 -1090.0 -0.39 400.0 -455.0 -0.35 -0.5196 -0.9988 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N01 compound treatment 1680.0 -526.0 -0.19 440.0 -415.0 -0.32 -0.3574 -0.9675 1576679 ChemDiv3_003455 C(Sc1nnc(c2ccccc2)c(n1)c3ccccc3)C4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N02 compound treatment 560.0 -1650.0 -0.58 440.0 -415.0 -0.32 -0.6383 -0.9594 3117901 ChemDiv3_003456 CCOC(=O)c1c(C)oc-2c1/C(=C/Nc3cccc(C)n3)/C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N03 compound treatment 2480.0 274.0 0.1 400.0 -455.0 -0.35 -0.1784 -0.492 1365406 ChemDiv3_003457 Cc1cc(C)cc(Oc2coc3cc(OC(=O)C4CCCCC4)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N04 compound treatment 8960.0 6750.0 2.4 960.0 105.0 0.08 1.751 0.7304 3117902 ChemDiv3_003458 Clc1ccc(cc1)c2nc(/C=N/c3ccccc3)c4ccccn24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N05 compound treatment 600.0 -1610.0 -0.57 400.0 -455.0 -0.35 -0.65 -0.9724 3117903 ChemDiv3_003459 CCOC(=O)N1CCN(CC1)C(=O)CCCN2C(=O)/C(=C\c3cccs3)/SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N06 compound treatment 1360.0 -846.0 -0.3 720.0 -135.0 -0.1 -0.2857 -0.8993 3117904 ChemDiv3_003460 COC(=O)C1C(C(=C(NC1=O)SCC(=O)NCc2ccccc2)C#N)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N07 compound treatment 360.0 -1850.0 -0.65 240.0 -615.0 -0.47 -0.7971 -0.9871 3022943 ChemDiv3_003461 CC(N(Cc1ccccc1)C(=S)Nc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N08 compound treatment 6280.0 4070.0 1.45 560.0 -295.0 -0.23 0.8616 0.589 1661674 ChemDiv3_003462 Clc1ccccc1C(=O)Oc2c(CN3CCOCC3)cc(Cl)c4cccnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N09 compound treatment 600.0 -1610.0 -0.57 320.0 -535.0 -0.41 -0.6934 -0.9871 1593593 ChemDiv3_003463 CCC1=NC(N(O)C1(C)C)c2ccccc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N10 compound treatment 560.0 -1650.0 -0.58 1040.0 185.0 0.14 -0.3126 -0.5202 1174273 ChemDiv3_003464 CN(Cc1ccccc1)S(=O)(=O)c2ccc(cc2)C(=O)Nc3nc4ccc5ccccc5c4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N11 compound treatment 4800.0 2590.0 0.92 320.0 -535.0 -0.41 0.3601 0.3574 1124946 ChemDiv3_003465 CCC(=O)c1cn(c2ccccc12)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N12 compound treatment 560.0 -1650.0 -0.58 800.0 -55.2 -0.04 -0.4429 -0.7564 1374319 ChemDiv3_003466 CC(NC(=O)c1ccc(cc1)C(C)(C)C)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N13 compound treatment 320.0 -1890.0 -0.67 400.0 -455.0 -0.35 -0.7202 -0.9541 1187438 ChemDiv3_003467 COc1ccc(OC)c(NC(=O)C2CCCNC2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N14 compound treatment 520.0 -1690.0 -0.6 400.0 -455.0 -0.35 -0.6701 -0.9672 1589905 ChemDiv3_003468 CC1=C(C(c2ccc(O)cc2)c3c(N1)[nH]c(=O)[nH]c3=O)C(=O)OCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N15 compound treatment 1760.0 -446.0 -0.16 520.0 -335.0 -0.26 -0.2939 -0.9728 1548201 ChemDiv3_003469 CC(Cn1nnc2ccccc12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N16 compound treatment 3720.0 1510.0 0.54 640.0 -215.0 -0.17 0.2629 0.4679 1198691 ChemDiv3_003470 CCOC(=O)c1c(NC(=O)CSc2nnc3ccccn23)scc1c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N17 compound treatment 4360.0 2150.0 0.76 1040.0 185.0 0.14 0.6406 0.8243 3117905 ChemDiv3_003471 CC1(C)CC(=O)C(=C2Nc3ccc(cc3N2)C(=O)c4ccccc4)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N18 compound treatment 880.0 -1330.0 -0.47 400.0 -455.0 -0.35 -0.5798 -0.9893 1540618 ChemDiv3_003472 CCOC(=O)N1CCN(CC1)C(=O)CSCC(=O)Nc2nc(cs2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N19 compound treatment 480.0 -1730.0 -0.61 280.0 -575.0 -0.44 -0.7453 -0.9871 1143371 ChemDiv3_003473 CCn1c2ccccc2c3cc(NC(=O)COc4ccc(OC)cc4)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N20 compound treatment 5640.0 3430.0 1.22 440.0 -415.0 -0.32 0.636 0.5051 1639873 ChemDiv3_003474 Cc1ccc(cc1)S(=O)(=O)N(CC(=O)NC2CC2)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N21 compound treatment 1120.0 -1090.0 -0.39 520.0 -335.0 -0.26 -0.4544 -0.9807 1383609 ChemDiv3_003475 CCC(CC)NCc1oc2ccc(Cl)cc2c1c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N22 compound treatment 520.0 -1690.0 -0.6 360.0 -495.0 -0.38 -0.6918 -0.9761 3023230 ChemDiv3_003476 Cc1cccc(N(CC(=O)N)S(=O)(=O)C)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N23 mock treatment 5120.0 2910.0 1.03 480.0 -375.0 -0.29 0.5272 0.4914 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 N24 mock treatment 960.0 -1250.0 -0.44 720.0 -135.0 -0.1 -0.386 -0.85 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O01 compound treatment 320.0 -1890.0 -0.67 200.0 -655.0 -0.5 -0.8288 -0.9901 3117906 ChemDiv3_003477 CCOc1ccc(/N=c/2\scc(c3ccc(cc3)S(=O)(=O)N4CCCC4)n2CC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O02 compound treatment 240.0 -1970.0 -0.7 360.0 -495.0 -0.38 -0.762 -0.9593 3023233 ChemDiv3_003478 Nc1nc(cs1)C2(CC3CC4C2)CC(C3)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O03 compound treatment 320.0 -1890.0 -0.67 320.0 -535.0 -0.41 -0.7637 -0.9726 1118743 ChemDiv3_003479 Cc1ccc(cc1)N(C(=O)c2ccccc2C)S(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O04 compound treatment 320.0 -1890.0 -0.67 280.0 -575.0 -0.44 -0.7854 -0.9796 1346452 ChemDiv3_003480 COC(=O)CSc1nc2sc3CCCc3c2c(=O)n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O05 compound treatment 520.0 -1690.0 -0.6 320.0 -535.0 -0.41 -0.7135 -0.9832 3023234 ChemDiv3_003481 CC[n+]1c(/C=C/2\Sc3ccccc3N2CCO)sc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O06 compound treatment 1560.0 -646.0 -0.23 360.0 -495.0 -0.38 -0.4309 -0.9707 3022550 ChemDiv3_003482 Cc1cccc(/N=C/C=C2OC(C)(C)C(C)(C)O2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O07 compound treatment 440.0 -1770.0 -0.63 400.0 -455.0 -0.35 -0.6901 -0.962 1137751 ChemDiv3_003483 O=C(Nc1ccc(cc1)c2nc3ncccc3o2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O08 compound treatment 240.0 -1970.0 -0.7 280.0 -575.0 -0.44 -0.8055 -0.9757 3117907 ChemDiv3_003484 CCc1cc2c(=O)n(c(SCC(=O)c3ccccc3)nc2s1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O09 compound treatment 360.0 -1850.0 -0.65 320.0 -535.0 -0.41 -0.7536 -0.9748 3117908 ChemDiv3_003485 CCc1cc2c(=O)n(CC=C)c(SCC(=O)c3ccc(C)cc3)nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O10 compound treatment 400.0 -1810.0 -0.64 320.0 -535.0 -0.41 -0.7436 -0.9769 1672847 ChemDiv3_003486 Cc1ccccc1NC(NC(=O)c2ccco2)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O11 compound treatment 360.0 -1850.0 -0.65 200.0 -655.0 -0.5 -0.8188 -0.9915 1634367 ChemDiv3_003487 O=C(Nc1cccc(c1)c2nc3ccccc3o2)c4cccc(OCc5ccccc5)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O12 compound treatment 640.0 -1570.0 -0.56 1040.0 185.0 0.14 -0.2925 -0.5102 3022557 ChemDiv3_003488 COc1ccc(cc1)c2nn(cc2C=C3C(=O)CC(C)(C)CC3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O13 compound treatment 1640.0 -566.0 -0.2 360.0 -495.0 -0.38 -0.4108 -0.9555 3117909 ChemDiv3_003489 COc1ccc2NC(=O)/C(=N/O)/c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O14 compound treatment 400.0 -1810.0 -0.64 320.0 -535.0 -0.41 -0.7436 -0.9769 1437035 ChemDiv3_003490 CC1CC(Nc2ccccc2C)c3cccc(C)c3N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O15 compound treatment 360.0 -1850.0 -0.65 440.0 -415.0 -0.32 -0.6885 -0.9452 3022560 ChemDiv3_003491 CCCNc1nc2ccccn2c(=O)c1/C=C/3\SC(=S)NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O16 compound treatment 320.0 -1890.0 -0.67 240.0 -615.0 -0.47 -0.8071 -0.9855 3118060 ChemDiv3_003492 Nc1nnc(SCC(=O)N2c3ccccc3Sc4ccc(cc24)C(F)(F)F)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O17 compound treatment 1560.0 -646.0 -0.23 280.0 -575.0 -0.44 -0.4743 -0.9534 1398200 ChemDiv3_003493 CS(=O)(=O)N1CCN(C1)C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O18 compound treatment 1840.0 -366.0 -0.13 440.0 -415.0 -0.32 -0.3173 -0.9217 3118061 ChemDiv3_003494 NC1=C(C#N)C(c2c(nn(c2O1)c3ccccc3)c4ccccc4)c5ccc(Cl)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O19 compound treatment 240.0 -1970.0 -0.7 280.0 -575.0 -0.44 -0.8055 -0.9757 3022592 ChemDiv3_003495 COC(=O)CSc1sc(=S)sc1SCC[n+]2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O20 compound treatment 920.0 -1290.0 -0.46 520.0 -335.0 -0.26 -0.5046 -0.9633 3022594 ChemDiv3_003496 C/C(=N\n1c(C)cc(C)c(C#N)c1=O)/C=C/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O21 compound treatment 240.0 -1970.0 -0.7 320.0 -535.0 -0.41 -0.7837 -0.9681 1248779 ChemDiv3_003497 CC(NS(=O)(=O)c1c(C)cc(C)cc1C)C2C3CC4CC(C3)CC2C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O22 compound treatment 320.0 -1890.0 -0.67 320.0 -535.0 -0.41 -0.7637 -0.9726 1259680 ChemDiv3_003498 CC(C)C1CCC(C)CC1OC(=O)CN2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O23 mock treatment 400.0 -1810.0 -0.64 280.0 -575.0 -0.44 -0.7653 -0.9835 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 O24 mock treatment 360.0 -1850.0 -0.65 240.0 -615.0 -0.47 -0.7971 -0.9871 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P01 compound treatment 280.0 -1930.0 -0.68 240.0 -615.0 -0.47 -0.8171 -0.9837 1241332 ChemDiv3_003499 Brc1cccc(OCc2cccc(c2)C(=O)NN3CCOCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P02 compound treatment 240.0 -1970.0 -0.7 320.0 -535.0 -0.41 -0.7837 -0.9681 3118062 ChemDiv3_003500 CCOC(=O)c1c(C)oc-2c1/C(=C/NC3CCCC3)/C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P03 compound treatment 360.0 -1850.0 -0.65 360.0 -495.0 -0.38 -0.7319 -0.9665 1385678 ChemDiv3_003501 CCC(CC)c1nc(Nc2ccccc2)c3ccccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P04 compound treatment 280.0 -1930.0 -0.68 240.0 -615.0 -0.47 -0.8171 -0.9837 3118063 ChemDiv3_003502 CCOC(=O)C(C)Sc1nnc(CNC(=O)C2(CC3CC4CC(C3)C2)C4)n1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P05 compound treatment 400.0 -1810.0 -0.64 240.0 -615.0 -0.47 -0.787 -0.9887 3022600 ChemDiv3_003503 CCN(CCO)C(=O)CCN1C(=O)/C(=C/c2ccc(OC)c(OC)c2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P06 compound treatment 240.0 -1970.0 -0.7 240.0 -615.0 -0.47 -0.8272 -0.982 1357646 ChemDiv3_003504 CCOc1ccc(NC(=O)CSC2=C(C#N)C(C3=C(CC(C)(C)CC3=O)N2)c4cccs4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P07 compound treatment 1920.0 -286.0 -0.1 240.0 -615.0 -0.47 -0.4058 -0.8399 1315615 ChemDiv3_003505 Cc1ccc(NC(=S)N(CCc2ccccc2)Cc3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P08 compound treatment 240.0 -1970.0 -0.7 200.0 -655.0 -0.5 -0.8489 -0.9871 3118064 ChemDiv3_003506 CN1CCN(CC1)/N=C/c2nc(c3ccccc3)n4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P09 compound treatment 360.0 -1850.0 -0.65 240.0 -615.0 -0.47 -0.7971 -0.9871 3118065 ChemDiv3_003507 Fc1ccccc1CN2C(=O)S/C(=C\c3ccc4OCOc4c3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P10 compound treatment 240.0 -1970.0 -0.7 240.0 -615.0 -0.47 -0.8272 -0.982 1727777 ChemDiv3_003508 CCCCN(C)S(=O)(=O)c1ccc(cc1)C(=O)Nc2nc3ccc4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P11 compound treatment 320.0 -1890.0 -0.67 240.0 -615.0 -0.47 -0.8071 -0.9855 1646615 ChemDiv3_003509 Clc1ccc(cc1)C(=O)OCc2cccc(COC(=O)c3ccc(Cl)cc3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P12 compound treatment 320.0 -1890.0 -0.67 280.0 -575.0 -0.44 -0.7854 -0.9796 1266949 ChemDiv3_003510 CC(NC(=O)CC1(CC2CC3CC(C2)C1)C3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P13 compound treatment 360.0 -1850.0 -0.65 360.0 -495.0 -0.38 -0.7319 -0.9665 1141185 ChemDiv3_003511 Cc1ccc2[nH]cc(CCNC(=O)c3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P14 compound treatment 280.0 -1930.0 -0.68 200.0 -655.0 -0.5 -0.8389 -0.9886 1623182 ChemDiv3_003512 Cn1c(nc2ccccc12)c3cc4ccc(O)c(CN5CCCC5)c4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P15 compound treatment 360.0 -1850.0 -0.65 200.0 -655.0 -0.5 -0.8188 -0.9915 3022639 ChemDiv3_003513 CC(C)c1nccn1CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P16 compound treatment 240.0 -1970.0 -0.7 360.0 -495.0 -0.38 -0.762 -0.9593 1601523 ChemDiv3_003514 O=c1n(c2ccccc2)c(=S)[nH]c3scc(c4cccs4)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P17 compound treatment 360.0 -1850.0 -0.65 520.0 -335.0 -0.26 -0.6451 -0.9167 3118066 ChemDiv3_003515 CC1(C)CC(=O)C(=CN2CCOCC2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P18 compound treatment 280.0 -1930.0 -0.68 280.0 -575.0 -0.44 -0.7954 -0.9777 3022643 ChemDiv3_003516 Cc1cs/c(=N\C(=S)Nc2ccccc2)/n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P19 compound treatment 360.0 -1850.0 -0.65 360.0 -495.0 -0.38 -0.7319 -0.9665 3118067 ChemDiv3_003517 CC(=O)Nc1ccccc1NC(=O)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P20 compound treatment 1360.0 -846.0 -0.3 280.0 -575.0 -0.44 -0.5245 -0.9823 1615664 ChemDiv3_003518 Brc1ccc(CN(CC(=O)Nc2ccccc2)S(=O)(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P21 compound treatment 360.0 -1850.0 -0.65 320.0 -535.0 -0.41 -0.7536 -0.9748 1741961 ChemDiv3_003519 CCOC(=O)c1c(CSc2ccc(C)cc2)n(C)c3cc(Br)c(O)c(CN(C)C)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P22 compound treatment 280.0 -1930.0 -0.68 280.0 -575.0 -0.44 -0.7954 -0.9777 1152994 ChemDiv3_003520 COc1ccccc1N(CC(=O)NCC2CCCO2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P23 mock treatment 200.0 -2010.0 -0.71 240.0 -615.0 -0.47 -0.8372 -0.9802 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2010 P24 mock treatment 280.0 -1930.0 -0.68 360.0 -495.0 -0.38 -0.752 -0.9617 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A01 compound treatment 440.0 -679.0 -0.24 600.0 -80.0 -0.06 -0.2137 -0.8599 3022646 ChemDiv3_003521 CCN(CC)C(=O)c1ccc(cc1)N(Cc2ccccc2Cl)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A02 compound treatment 240.0 -879.0 -0.31 200.0 -480.0 -0.37 -0.481 -0.9965 3118068 ChemDiv3_003522 Fc1nc(F)c(F)c(NCCOC(=O)c2ccccc2)c1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A03 compound treatment 320.0 -799.0 -0.28 200.0 -480.0 -0.37 -0.4609 -0.9916 1531239 ChemDiv3_003523 S=C(NCc1ccccc1)N2CCN(CC2)c3nc(c4ccccc4)c5CCCCc5c3C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A04 compound treatment 480.0 -639.0 -0.23 2440.0 1760.0 1.35 0.7952 0.5804 1218136 ChemDiv3_003524 C=CC[N+]1(CC#Cc2ccccc2)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A05 compound treatment 680.0 -439.0 -0.16 280.0 -400.0 -0.31 -0.3272 -0.9504 1599397 ChemDiv3_003525 COc1ccc(cc1)N2CCN(CC2)C(=S)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A06 compound treatment 2760.0 1640.0 0.58 240.0 -440.0 -0.34 0.1728 0.2568 3118069 ChemDiv3_003526 C[N+](C)(CCN1C(=O)C2C(C(C=CC2c3ccccc3)c4ccccc4)C1=O)CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A07 compound treatment 640.0 -479.0 -0.17 280.0 -400.0 -0.31 -0.3372 -0.961 3022686 ChemDiv3_003527 O=S(=O)(Nc1ccc(CSc2ccccc2)cc1)c3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A08 compound treatment 960.0 -159.0 -0.06 320.0 -360.0 -0.28 -0.2353 -0.8341 1787354 ChemDiv3_003528 CS(=O)(=O)N(CC(=O)N1CCc2ccccc2C1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A09 compound treatment 240.0 -879.0 -0.31 360.0 -320.0 -0.25 -0.3941 -0.993 3118070 ChemDiv3_003529 COc1ccc(/N=C/2\C(=O)N3c4c2cc(C)cc4C(=CC3(C)C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A10 compound treatment 240.0 -879.0 -0.31 6440.0 5760.0 4.42 2.9064 0.6556 3022689 ChemDiv3_003530 CCOC(=O)c1cc(C)sc1/N=C/C2C(=O)NC(=S)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A11 compound treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 1683008 ChemDiv3_003531 CC(C)c1ccc(cc1)C2=C(O)C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A12 compound treatment 200.0 -919.0 -0.33 240.0 -440.0 -0.34 -0.4693 -0.9998 1674919 ChemDiv3_003532 O=C(Nc1ccccc1Sc2ncnc3sc4CCCCc4c23)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A13 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 1258553 ChemDiv3_003533 CCc1ccc(Oc2coc3cc(OC(=O)C(C)C)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A14 compound treatment 320.0 -799.0 -0.28 240.0 -440.0 -0.34 -0.4392 -0.9962 1515482 ChemDiv3_003534 ON(C1CC(=O)N(C1=O)c2ccc(cc2)N3CCOCC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A15 compound treatment 240.0 -879.0 -0.31 280.0 -400.0 -0.31 -0.4376 -1.0 1334348 ChemDiv3_003535 O=C(Oc1cccc(Nc2ncnc3ccccc23)c1)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A16 compound treatment 240.0 -879.0 -0.31 280.0 -400.0 -0.31 -0.4376 -1.0 3118071 ChemDiv3_003536 O=C/1N(C2CCCCC2)C(=S)S\C1=C/c3c(NCC4CCCO4)nc5ccccn5c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A17 compound treatment 360.0 -759.0 -0.27 240.0 -440.0 -0.34 -0.4292 -0.9937 3022693 ChemDiv3_003537 CN1C(=O)NC(C2=C1CC(C)(C)CC2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A18 compound treatment 480.0 -639.0 -0.23 360.0 -320.0 -0.25 -0.3339 -0.9992 1298375 ChemDiv3_003538 CC(=O)N1CCN(CC1)C2C(NS(=O)(=O)c3ccc(Cl)cc3)c4cccc5cccc2c45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A19 compound treatment 440.0 -679.0 -0.24 320.0 -360.0 -0.28 -0.3657 -0.9976 1788606 ChemDiv3_003539 Clc1ccc(CNC(=O)C2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A20 compound treatment 320.0 -799.0 -0.28 240.0 -440.0 -0.34 -0.4392 -0.9962 1872134 ChemDiv3_003540 Cc1ccc(Oc2cc(C#N)c3ccccc3n2)c(c1)n4nc5ccccc5n4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A21 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 3022649 ChemDiv3_003541 CC(C)C(=O)N1N=C2CCCCC2C1(O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A22 compound treatment 240.0 -879.0 -0.31 280.0 -400.0 -0.31 -0.4376 -1.0 1372518 ChemDiv3_003542 CN(C)c1c2CCCc2c(C#N)c3nc4ccccc4n13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A23 mock treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 A24 mock treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B01 compound treatment 920.0 -199.0 -0.07 1880.0 1200.0 0.92 0.6016 0.6511 1153643 ChemDiv3_003543 CC(C)c1cc(O)n2c3ccccc3nc2c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B02 compound treatment 280.0 -839.0 -0.3 240.0 -440.0 -0.34 -0.4493 -0.998 1581286 ChemDiv3_003544 Oc1ccc2c(=O)c(coc2c1CN(CC=C)CC=C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B03 compound treatment 280.0 -839.0 -0.3 240.0 -440.0 -0.34 -0.4493 -0.998 1464911 ChemDiv3_003545 CC(C)Nc1ccc(Nc2ccnc3cc4ccccc4cc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B04 compound treatment 200.0 -919.0 -0.33 280.0 -400.0 -0.31 -0.4476 -0.9996 3118203 ChemDiv3_003546 COC(=O)c1cccc(/N=C/2\NC(=N)c3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B05 compound treatment 960.0 -159.0 -0.06 280.0 -400.0 -0.31 -0.257 -0.8231 1377576 ChemDiv3_003547 COc1cc(NC(=O)COc2ccc(F)cc2)nc(OC)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B06 compound treatment 520.0 -599.0 -0.21 320.0 -360.0 -0.28 -0.3456 -0.9915 3118204 ChemDiv3_003548 c1csc(c1)c2nc(no2)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B07 compound treatment 3520.0 2400.0 0.85 520.0 -160.0 -0.12 0.5155 0.5989 3118205 ChemDiv3_003549 CC(/N=C/1\CCCc2ccccc2N1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B08 compound treatment 440.0 -679.0 -0.24 240.0 -440.0 -0.34 -0.4091 -0.9862 1556957 ChemDiv3_003550 CC(C)CCNc1ncnc2c3cc4COC(C)(C)Cc4nc3sc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B09 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3022697 ChemDiv3_003551 OC(=O)c1ccc(COc2ccccc2/C=C/3\NC(=O)N(Cc4ccccc4)C3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B10 compound treatment 200.0 -919.0 -0.33 360.0 -320.0 -0.25 -0.4042 -0.9903 3118206 ChemDiv3_003552 Clc1cccc(c1)N/2CCC\C2=N/c3ccc(Br)cc3C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B11 compound treatment 240.0 -879.0 -0.31 240.0 -440.0 -0.34 -0.4593 -0.9992 3022699 ChemDiv3_003553 FC(F)(F)C(NC(=O)OCc1ccccc1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B12 compound treatment 280.0 -839.0 -0.3 240.0 -440.0 -0.34 -0.4493 -0.998 3118207 ChemDiv3_003554 COc1cccc(c1)c2nc3cccc4cccc([nH]2)c43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B13 compound treatment 320.0 -799.0 -0.28 360.0 -320.0 -0.25 -0.3741 -0.9975 1719480 ChemDiv3_003555 S=C(N1CCCC1)c2cn(CCOc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B14 compound treatment 680.0 -439.0 -0.16 400.0 -280.0 -0.21 -0.2621 -0.9874 1867694 ChemDiv3_003556 OC(COc1ccc(NC(=O)c2ccccc2)cc1)Cn3c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B15 compound treatment 240.0 -879.0 -0.31 160.0 -520.0 -0.4 -0.5027 -0.9925 3118208 ChemDiv3_003557 Fc1ccc(cc1)C2CC(=O)C(=CNCCN3CCNCC3)C(=O)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B16 compound treatment 320.0 -799.0 -0.28 320.0 -360.0 -0.28 -0.3958 -0.9999 3022706 ChemDiv3_003558 O=C1CC(CC(=O)C1=CNc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B17 compound treatment 280.0 -839.0 -0.3 240.0 -440.0 -0.34 -0.4493 -0.998 3118209 ChemDiv3_003559 CC1(C)CC(=O)c2cc(C(=O)N3CC[N+](C)(C)CC3)c(=O)n(c4ccc(Cl)cc4)c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B18 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3022709 ChemDiv3_003560 CC1CCc2sc3ncnc(n4nc(C)cc4C)c3c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B19 compound treatment 240.0 -879.0 -0.31 440.0 -240.0 -0.18 -0.3507 -0.9685 3023520 ChemDiv3_003561 C=CCN1C(=O)NC(=O)/C(=C\c2cn(Cc3ccccc3)c4ccccc24)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B20 compound treatment 240.0 -879.0 -0.31 240.0 -440.0 -0.34 -0.4593 -0.9992 3023521 ChemDiv3_003562 COc1cccc(c1)C(=O)CN2C3=NCCCN3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B21 compound treatment 320.0 -799.0 -0.28 240.0 -440.0 -0.34 -0.4392 -0.9962 1225293 ChemDiv3_003563 CCOC(=O)c1cnc2ccc(cc2c1N3CC4(C)CC3CC(C)(C)C4)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B22 compound treatment 320.0 -799.0 -0.28 320.0 -360.0 -0.28 -0.3958 -0.9999 3023522 ChemDiv3_003564 Clc1snc(C(=O)Nc2ccc(I)cc2)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B23 mock treatment 3720.0 2600.0 0.92 240.0 -440.0 -0.34 0.4136 0.4209 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 B24 mock treatment 360.0 -759.0 -0.27 360.0 -320.0 -0.25 -0.364 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C01 compound treatment 280.0 -839.0 -0.3 240.0 -440.0 -0.34 -0.4493 -0.998 3023523 ChemDiv3_003565 COc1ccccc1N(CC(=O)NC2CC3CCC2C3)S(=O)(=O)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C02 compound treatment 320.0 -799.0 -0.28 200.0 -480.0 -0.37 -0.4609 -0.9916 1788093 ChemDiv3_003566 CC(CS(=O)(=O)c1ccc(C)cc1S(=O)(=O)CC(C)N2CCOCC2)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C03 compound treatment 240.0 -879.0 -0.31 320.0 -360.0 -0.28 -0.4159 -0.9982 1737011 ChemDiv3_003567 CC(C)c1nc(N2CCN(CC2)C(=S)NC3CCCCC3)c(C#N)c4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C04 compound treatment 680.0 -439.0 -0.16 600.0 -80.0 -0.06 -0.1535 -0.9173 3023524 ChemDiv3_003568 C[N+](C)(CC=C)CC#Cc1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C05 compound treatment 280.0 -839.0 -0.3 3680.0 3000.0 2.3 1.4182 0.6107 3118210 ChemDiv3_003569 COc1ccccc1N(CC(=O)Nc2ccccc2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C06 compound treatment 200.0 -919.0 -0.33 320.0 -360.0 -0.28 -0.4259 -0.9966 1699766 ChemDiv3_003570 C(C1OCc2ccccc2CO1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C07 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 3118211 ChemDiv3_003571 CS(=O)(=O)N(Cc1ccccc1Cl)c2ccc(cc2)C(=O)Nc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C08 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3118212 ChemDiv3_003572 Cc1ccc(cc1)S(=O)(=O)N(CC(=O)N2CCCCCC2)c3ccc(C)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C09 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 1301544 ChemDiv3_003573 Cc1onc(c1C(=O)NC(C)(C)CO)c2c(Cl)cccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C10 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 3118213 ChemDiv3_003574 CCOC(=O)c1cc(CC)sc1/N=C/C2C(=O)NC(=S)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C11 compound treatment 160.0 -959.0 -0.34 320.0 -360.0 -0.28 -0.4359 -0.9947 1870864 ChemDiv3_003575 CC(C)c1ccc(cc1)C2C3=C(NC4=C2C(=O)CCC4)c5ccccc5C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C12 compound treatment 320.0 -799.0 -0.28 320.0 -360.0 -0.28 -0.3958 -0.9999 1314792 ChemDiv3_003576 Cc1cc(=O)oc2cc(OCC(=O)NCc3cccnc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C13 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 1372263 ChemDiv3_003577 CCc1ccc(Oc2coc3cc(OC(=O)c4ccco4)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C14 compound treatment 240.0 -879.0 -0.31 160.0 -520.0 -0.4 -0.5027 -0.9925 3023525 ChemDiv3_003578 CC/N=C/1\SC(CC(=O)Nc2cccc(c2)C(=O)O)C(=O)N1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C15 compound treatment 240.0 -879.0 -0.31 360.0 -320.0 -0.25 -0.3941 -0.993 3118214 ChemDiv3_003579 Cc1cccc(c1)c2nc(NCCCN3CCOCC3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C16 compound treatment 400.0 -719.0 -0.25 400.0 -280.0 -0.21 -0.3323 -0.9964 3023526 ChemDiv3_003580 CC(C)(C)c1ccc(/C=C/C(=O)Nc2cccnc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C17 compound treatment 240.0 -879.0 -0.31 280.0 -400.0 -0.31 -0.4376 -1.0 1440542 ChemDiv3_003581 CCN1C(=O)NC(C2=C1CCCC2=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C18 compound treatment 360.0 -759.0 -0.27 1000.0 320.0 0.25 -0.0166 -0.0456 1435850 ChemDiv3_003582 Cc1cc(C)cc(OC2CCCCC2NS(=O)(=O)c3ccc(Cl)cc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C19 compound treatment 320.0 -799.0 -0.28 3920.0 3240.0 2.49 1.5585 0.6225 1879422 ChemDiv3_003583 Cc1onc(c1C(=O)n2nnc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C20 compound treatment 200.0 -919.0 -0.33 320.0 -360.0 -0.28 -0.4259 -0.9966 1610175 ChemDiv3_003584 Oc1cc2ccccc2cc1C(=O)OCC(=O)c3ccc(OCc4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C21 compound treatment 240.0 -879.0 -0.31 320.0 -360.0 -0.28 -0.4159 -0.9982 3023527 ChemDiv3_003585 CCC1=NN(C(=O)COc2ccc(Cl)c(C)c2)C(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C22 compound treatment 360.0 -759.0 -0.27 240.0 -440.0 -0.34 -0.4292 -0.9937 1145589 ChemDiv3_003586 N#Cc1c2CCCc2c(NCCN3CCCCC3)n4c5ccccc5nc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C23 mock treatment 2280.0 1160.0 0.41 280.0 -400.0 -0.31 0.0741 0.1443 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 C24 mock treatment 1280.0 161.0 0.06 280.0 -400.0 -0.31 -0.1767 -0.5657 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D01 compound treatment 3000.0 1880.0 0.67 400.0 -280.0 -0.21 0.3199 0.4563 3023528 ChemDiv3_003587 CC(=O)NC1C(=O)SC1(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D02 compound treatment 240.0 -879.0 -0.31 280.0 -400.0 -0.31 -0.4376 -1.0 1694459 ChemDiv3_003588 CC(C)OC(=O)C(C)Oc1ccc2c(=O)c(coc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D03 compound treatment 360.0 -759.0 -0.27 360.0 -320.0 -0.25 -0.364 -0.999 3023529 ChemDiv3_003589 Oc1ccccc1/C=C/2\SC(=NC2=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D04 compound treatment 400.0 -719.0 -0.25 400.0 -280.0 -0.21 -0.3323 -0.9964 1245012 ChemDiv3_003590 Cc1cccc(Oc2coc3cc(OC(=O)c4cccs4)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D05 compound treatment 320.0 -799.0 -0.28 4320.0 3640.0 2.79 1.7756 0.6322 3023530 ChemDiv3_003591 Cc1ccc(C#N)c(SCc2nnc(o2)c3ccc(Cl)cc3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D06 compound treatment 240.0 -879.0 -0.31 400.0 -280.0 -0.21 -0.3724 -0.9835 1788087 ChemDiv3_003592 COc1cc2c(cc1NC(=O)Cc3ccccc3)oc4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D07 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 1917902 ChemDiv3_003593 OC(=O)CC/N=C\1/CCCc2ccccc2N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D08 compound treatment 320.0 -799.0 -0.28 760.0 80.0 0.06 -0.1569 -0.5413 1538253 ChemDiv3_003594 CC(C)(C)Nc1ncnc2c3cc4COC(C)(C)Cc4nc3sc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D09 compound treatment 360.0 -759.0 -0.27 240.0 -440.0 -0.34 -0.4292 -0.9937 3023531 ChemDiv3_003595 Cc1ccccc1N2C(=O)NC(=O)/C(=C\c3cn(CC(=O)N4CCOCC4)c5ccccc35)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D10 compound treatment 520.0 -599.0 -0.21 240.0 -440.0 -0.34 -0.3891 -0.975 3118215 ChemDiv3_003596 Cc1sc2c(c1C)c(=O)n(c3ccccc3)c4nnc(SCC=C)n42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D11 compound treatment 320.0 -799.0 -0.28 360.0 -320.0 -0.25 -0.3741 -0.9975 3023532 ChemDiv3_003597 FC(F)(F)C(NC(=O)OC1CCCC1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D12 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 3118216 ChemDiv3_003598 Clc1ccc(/C=C/c2nc3cccc4cccc([nH]2)c43)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D13 compound treatment 400.0 -719.0 -0.25 600.0 -80.0 -0.06 -0.2237 -0.853 1699463 ChemDiv3_003599 S=C(NCCc1c[nH]c2ccccc12)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D14 compound treatment 280.0 -839.0 -0.3 360.0 -320.0 -0.25 -0.3841 -0.9955 3023533 ChemDiv3_003600 CCOC(=O)C1=C(O)CCN(C)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D15 compound treatment 320.0 -799.0 -0.28 360.0 -320.0 -0.25 -0.3741 -0.9975 3118217 ChemDiv3_003601 Fc1ccc(cc1)C2CC(=O)C(=CNCCN3CCN(CC3)C(=S)Nc4ccccc4)C(=O)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D16 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3023534 ChemDiv3_003602 COC(=O)N(C)CC1Cc2ccccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D17 compound treatment 280.0 -839.0 -0.3 560.0 -120.0 -0.09 -0.2755 -0.8846 3118351 ChemDiv3_003603 CC1(C)CC(=O)c2cc(C(=O)NCCC3=CCCCC3)c(=O)n(c4ccccc4)c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D18 compound treatment 240.0 -879.0 -0.31 240.0 -440.0 -0.34 -0.4593 -0.9992 1642387 ChemDiv3_003604 CCCCc1c(C)c(C#N)c2nc3ccccc3n2c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D19 compound treatment 320.0 -799.0 -0.28 400.0 -280.0 -0.21 -0.3524 -0.9907 3118352 ChemDiv3_003605 CC(C)(C)N1C(=O)NC(=O)/C(=C\c2cn(Cc3ccccc3)c4ccccc24)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D20 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 3023535 ChemDiv3_003606 Clc1ccc(Cn2c(NC(=O)C3CCCCC3)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D21 compound treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 1181214 ChemDiv3_003607 CCOC(=O)c1cnc2c(ccc3ccccc32)c1NC4CC(C)(C)NC(C)(C)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D22 compound treatment 320.0 -799.0 -0.28 360.0 -320.0 -0.25 -0.3741 -0.9975 3023536 ChemDiv3_003608 Cc1ccc(NCc2ccc(Cl)nc2)c(NCc3ccc(Cl)nc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D23 mock treatment 440.0 -679.0 -0.24 280.0 -400.0 -0.31 -0.3874 -0.9928 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 D24 mock treatment 920.0 -199.0 -0.07 200.0 -480.0 -0.37 -0.3104 -0.8274 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E01 compound treatment 600.0 -519.0 -0.18 480.0 -200.0 -0.15 -0.2387 -0.9959 3118353 ChemDiv3_003609 CS(=O)(=O)N(CC(=O)NCc1ccccc1)c2cc(ccc2Cl)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E02 compound treatment 1280.0 161.0 0.06 3720.0 3040.0 2.33 1.6907 0.7242 3023537 ChemDiv3_003610 C=CCN1C(=O)/C(=C/c2c(nc3ccccn3c2=O)N4CCCCC4)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E03 compound treatment 640.0 -479.0 -0.17 960.0 280.0 0.21 0.0319 0.1165 3118354 ChemDiv3_003611 CCCCc1nc2sc3c(Cl)ncnc3c2c4CC(C)(C)OCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E04 compound treatment 1160.0 41.3 0.01 880.0 200.0 0.15 0.1189 0.771 1442521 ChemDiv3_003612 C=CC[N+]1(CC#Cc2ccccc2)CCOCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E05 compound treatment 1080.0 -38.8 -0.01 9240.0 8560.0 6.57 4.6372 0.7056 1231207 ChemDiv3_003613 COc1ccccc1N(CC(=O)N2CCN(CC2)c3ccccc3OC)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E06 compound treatment 680.0 -439.0 -0.16 400.0 -280.0 -0.21 -0.2621 -0.9874 1028555 ChemDiv3_003614 O=C1CCN(Cc2ccccc2)C(=O)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E07 compound treatment 3280.0 2160.0 0.77 5080.0 4400.0 3.38 2.9307 0.8461 3118355 ChemDiv3_003615 CN1C(=O)/C(=C/c2c(nc3c(C)cccn3c2=O)N4CCCC4)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E08 compound treatment 1120.0 1.25 0.0 760.0 80.0 0.06 0.0437 0.7122 1863421 ChemDiv3_003616 O=C(NCCc1ccccc1)c2cc3c(ccc4ccccc34)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E09 compound treatment 560.0 -559.0 -0.2 720.0 40.0 0.03 -0.1184 -0.5905 3023538 ChemDiv3_003617 Cc1cc2nc(NC3=NC(O)C=C(CSc4nc5ccccc5[nH]4)N3)nc(C)c2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E10 compound treatment 280.0 -839.0 -0.3 720.0 40.0 0.03 -0.1887 -0.6308 3118356 ChemDiv3_003618 CCOC(=O)c1c(/N=C/C2C(=O)NC(=S)NC2=O)scc1c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E11 compound treatment 1280.0 161.0 0.06 800.0 120.0 0.09 0.1056 0.9737 1870801 ChemDiv3_003619 Cc1ccc(cc1Cl)n2c(=O)oc3ccc(Cl)cc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E12 compound treatment 4200.0 3080.0 1.09 4120.0 3440.0 2.64 2.6403 0.9238 3118357 ChemDiv3_003620 CC(Oc1ccc(Cl)cc1Cl)C(=O)NC2=NN(C(=O)C2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E13 compound treatment 720.0 -399.0 -0.14 880.0 200.0 0.15 0.0085 0.0409 1610886 ChemDiv3_003621 CCc1ccc(Oc2coc3cc(OC(=O)c4cccs4)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E14 compound treatment 600.0 -519.0 -0.18 400.0 -280.0 -0.21 -0.2821 -0.997 3023539 ChemDiv3_003622 Cc1ccc(NC(=O)CC2Sc3ccc(cc3NC2=O)C(F)(F)F)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E15 compound treatment 1240.0 121.0 0.04 560.0 -120.0 -0.09 -0.0347 -0.3416 3118358 ChemDiv3_003623 COc1cc(/C=N\c2ccc(O)cc2)ccc1OC(=O)CC3SC(=O)NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E16 compound treatment 2160.0 1040.0 0.37 920.0 240.0 0.18 0.3915 0.9484 3118359 ChemDiv3_003624 O=C(NC(Nc1sc2CCCCc2c1C#N)C(=O)c3cccs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E17 compound treatment 1040.0 -78.8 -0.03 400.0 -280.0 -0.21 -0.1718 -0.7923 1490011 ChemDiv3_003625 Cc1ccc(CCP(=O)(O)CCC(=O)O)cn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E18 compound treatment 3000.0 1880.0 0.67 320.0 -360.0 -0.28 0.2765 0.3827 3023540 ChemDiv3_003626 OC(=O)c1c(F)c(F)cc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E19 compound treatment 1360.0 241.0 0.09 960.0 280.0 0.21 0.2125 0.9185 1413652 ChemDiv3_003627 Cc1onc(c1C(=O)NCc2ccc3OCOc3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E20 compound treatment 5760.0 4640.0 1.65 2960.0 2280.0 1.75 2.4019 0.9995 3023541 ChemDiv3_003628 N#Cc1cc2N(Cc3ccccc3)CCN(Cc4ccccc4)c2cc1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E21 compound treatment 4240.0 3120.0 1.11 4120.0 3440.0 2.64 2.6504 0.9255 3118360 ChemDiv3_003629 Clc1ccc(cc1)C(=O)/C=C/N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E22 compound treatment 960.0 -159.0 -0.06 1240.0 560.0 0.43 0.2642 0.6093 1455387 ChemDiv3_003630 CCc1c(C)c(C#N)c2nc3ccccc3n2c1Nc4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E23 mock treatment 2800.0 1680.0 0.6 2480.0 1800.0 1.38 1.3989 0.9294 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 E24 mock treatment 360.0 -759.0 -0.27 1120.0 440.0 0.34 0.0485 0.1124 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F01 compound treatment 440.0 -679.0 -0.24 1600.0 920.0 0.71 0.3292 0.4411 1286483 ChemDiv3_003631 O=c1n(CN2CCCCC2)nc3-c4ccccc4-c5cccc1c53 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F02 compound treatment 560.0 -559.0 -0.2 9320.0 8640.0 6.63 4.5501 0.6857 1204240 ChemDiv3_003632 CC1CN(Cc2c(O)ccc3c(=O)c(coc23)c4ccccc4)CC(C)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F03 compound treatment 2720.0 1600.0 0.57 1840.0 1160.0 0.89 1.0314 0.9764 3023542 ChemDiv3_003633 CCC1(C)NN(C(=S)N1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F04 compound treatment 960.0 -159.0 -0.06 760.0 80.0 0.06 0.0036 0.0433 3118361 ChemDiv3_003634 C1C(Nc2nnnn2C1c3cccs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F05 compound treatment 680.0 -439.0 -0.16 3240.0 2560.0 1.97 1.2797 0.6491 3118362 ChemDiv3_003635 NC(=O)C1CCN(CC1)C(=O)/C(=C/c2ccco2)/NC(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F06 compound treatment 2800.0 1680.0 0.6 3800.0 3120.0 2.4 2.1155 0.857 1239837 ChemDiv3_003636 O=C(CCc1ccccc1)NCc2ccccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F07 compound treatment 600.0 -519.0 -0.18 960.0 280.0 0.21 0.0219 0.0773 3023543 ChemDiv3_003637 C(/N=C/1\CCCCN1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F08 compound treatment 1040.0 -78.8 -0.03 2800.0 2120.0 1.63 1.1311 0.6949 3118363 ChemDiv3_003638 CC1C(NC(C(C)C1=O)c2ccccc2C)c3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F09 compound treatment 320.0 -799.0 -0.28 5200.0 4520.0 3.47 2.2534 0.6472 3118364 ChemDiv3_003639 C=CCN1C(=O)S/C(=C\c2cn(CC(=O)N3CCOCC3)c4ccccc24)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F10 compound treatment 2880.0 1760.0 0.62 2800.0 2120.0 1.63 1.5927 0.9136 3023595 ChemDiv3_003640 CC(C)CSc1nc2sc3COC(C)(C)Cc3c2c(=O)n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F11 compound treatment 3760.0 2640.0 0.94 680.0 0.0 0.0 0.6625 0.7071 3023596 ChemDiv3_003641 Cc1cccnc1NC(=O)NC(C)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F12 compound treatment 1080.0 -38.8 -0.01 800.0 120.0 0.09 0.0554 0.595 3023597 ChemDiv3_003642 C=CCn1c(=O)n(CC=C)c2cccc3cccc1c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F13 compound treatment 7600.0 6480.0 2.3 1040.0 360.0 0.28 1.8212 0.7864 1391530 ChemDiv3_003643 COc1ccc(NC(=S)NCCc2c[nH]c3ccccc23)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F14 compound treatment 2600.0 1480.0 0.53 7320.0 6640.0 5.1 3.9761 0.7759 3023598 ChemDiv3_003644 CC(=O)NS(=O)(=O)c1ccc(cc1)c2ccc(/C=C/3\C(=C(C#N)C(=O)N(CCCO)C3=O)C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F15 compound treatment 3400.0 2280.0 0.81 2120.0 1440.0 1.11 1.354 0.9882 3023599 ChemDiv3_003645 Cc1cccc(NC(=S)N(CCCNC2=CC(=O)CC(C)(C)C2)C3CCCCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F16 compound treatment 1000.0 -119.0 -0.04 1240.0 560.0 0.43 0.2742 0.6348 1521665 ChemDiv3_003646 Cc1ccc(OCCN2CCN(CC2)c3cc(C)c(C#N)c4nc5ccccc5n34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F17 compound treatment 1240.0 121.0 0.04 1360.0 680.0 0.52 0.3996 0.7628 3023600 ChemDiv3_003647 CCN(CC)CC#CCN1c2ccccc2Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F18 compound treatment 1120.0 1.25 0.0 1600.0 920.0 0.71 0.4997 0.7076 1373357 ChemDiv3_003648 CCCCc1c(C)c(C#N)c2nc3ccccc3n2c1NCCN4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F19 compound treatment 400.0 -719.0 -0.25 520.0 -160.0 -0.12 -0.2672 -0.9439 3023601 ChemDiv3_003649 CCOC(=O)c1cc(c2ccccc2)n(n1)c3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F20 compound treatment 1520.0 401.0 0.14 3800.0 3120.0 2.4 1.7944 0.7478 3118365 ChemDiv3_003650 O=C(Nc1nc2ccccc2n1CCN3CCOCC3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F21 compound treatment 760.0 -359.0 -0.13 2640.0 1960.0 1.5 0.974 0.645 3023602 ChemDiv3_003651 CCOC(=O)c1cnc2c(ccc3ccccc32)c1NCCOC(=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F22 compound treatment 4440.0 3320.0 1.18 2480.0 1800.0 1.38 1.8103 0.9968 1866848 ChemDiv3_003652 CCOC(=O)CN(C1SC(=O)N(Cc2cccc(c2)C(=O)O)C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F23 mock treatment 1000.0 -119.0 -0.04 880.0 200.0 0.15 0.0788 0.4948 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 F24 mock treatment 1840.0 721.0 0.26 1080.0 400.0 0.31 0.3981 0.9959 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G01 compound treatment 520.0 -599.0 -0.21 1760.0 1080.0 0.83 0.4361 0.5095 3118366 ChemDiv3_003653 COC(=O)C1=CN(C=C(C1c2ccc(F)cc2)C(=O)OC)c3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G02 compound treatment 1760.0 641.0 0.23 360.0 -320.0 -0.25 -0.0129 -0.0384 3023603 ChemDiv3_003654 CCNc1nc2ccccn2c(=O)c1/C=C/3\SC(=S)N(CC=C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G03 compound treatment 1560.0 441.0 0.16 760.0 80.0 0.06 0.1541 0.9165 3118367 ChemDiv3_003655 CCCc1nc2sc3c(Cl)ncnc3c2c4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G04 compound treatment 1480.0 361.0 0.13 280.0 -400.0 -0.31 -0.1265 -0.3802 3023604 ChemDiv3_003656 COCN(C#N)c1nc(nc(n1)N(C)C)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G05 compound treatment 1240.0 121.0 0.04 1080.0 400.0 0.31 0.2476 0.7984 3118368 ChemDiv3_003657 COc1ccc(cc1)S(=O)(=O)N(CC(=O)N)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G06 compound treatment 1160.0 41.3 0.01 1280.0 600.0 0.46 0.3361 0.7292 3023605 ChemDiv3_003658 COc1ccc(NC(=O)CSc2nc(cc(=O)[nH]2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G07 compound treatment 600.0 -519.0 -0.18 1120.0 440.0 0.34 0.1087 0.2827 3118494 ChemDiv3_003659 CN(C)c1nc2ccccn2c(=O)c1/C=C/3\SC(=S)N(C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G08 compound treatment 440.0 -679.0 -0.24 440.0 -240.0 -0.18 -0.3005 -0.9913 3023606 ChemDiv3_003660 O=C1N=C(SC1=C2CCCC2)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G09 compound treatment 880.0 -239.0 -0.08 1840.0 1160.0 0.89 0.5698 0.637 3118495 ChemDiv3_003661 NC(=N)/N=c\1/[nH]c(=O)c2ccccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G10 compound treatment 360.0 -759.0 -0.27 1480.0 800.0 0.61 0.244 0.3638 3023607 ChemDiv3_003662 CCOC(=O)c1cc(C)sc1/N=C/C2C(=O)CCCC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G11 compound treatment 1000.0 -119.0 -0.04 600.0 -80.0 -0.06 -0.0732 -0.9831 3118496 ChemDiv3_003663 CCc1ccc(cc1)C2CC(=NN2C(=O)CCCC(=O)O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G12 compound treatment 2360.0 1240.0 0.44 1440.0 760.0 0.58 0.7239 0.9904 1155587 ChemDiv3_003664 COC1(OC(=O)c2ccccc21)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G13 compound treatment 600.0 -519.0 -0.18 2440.0 1760.0 1.35 0.8253 0.6052 1357257 ChemDiv3_003665 CCc1ccc(Oc2coc3cc(OC(=O)C4CCCCC4)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G14 compound treatment 920.0 -199.0 -0.07 1960.0 1280.0 0.98 0.645 0.6547 1610546 ChemDiv3_003666 OC(=O)c1cccnc1SC2CC(=O)N(Cc3ccccc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G15 compound treatment 1240.0 121.0 0.04 640.0 -40.0 -0.03 0.0087 0.1646 1448429 ChemDiv3_003667 CCOC(=O)Nc1nc2ccc(OC)cc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G16 compound treatment 440.0 -679.0 -0.24 1200.0 520.0 0.4 0.112 0.2403 1873982 ChemDiv3_003668 CC(C)OC(=O)C1=C(C)NC(=O)NC1c2cn(nc2c3ccc(OC(C)C)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G17 compound treatment 320.0 -799.0 -0.28 7240.0 6560.0 5.04 3.3608 0.6663 1605638 ChemDiv3_003669 CN(CP(=O)(O)CN1CCCCC1)C=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G18 compound treatment 680.0 -439.0 -0.16 720.0 40.0 0.03 -0.0883 -0.5569 1298680 ChemDiv3_003670 CCN1C2C(C(=NC2Nc3ccccc13)OC)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G19 compound treatment 560.0 -559.0 -0.2 600.0 -80.0 -0.06 -0.1836 -0.8847 3023608 ChemDiv3_003671 CC(C)(C)C(=O)NC1CCSC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G20 compound treatment 680.0 -439.0 -0.16 800.0 120.0 0.09 -0.0449 -0.2483 3023609 ChemDiv3_003672 CN/1C(=O)CS\C1=N\c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G21 compound treatment 2520.0 1400.0 0.5 1600.0 920.0 0.71 0.8509 0.9852 3118497 ChemDiv3_003673 CCCCC1=NN(C(=O)C2CC2)C(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G22 compound treatment 840.0 -279.0 -0.1 520.0 -160.0 -0.12 -0.1568 -0.9942 1600165 ChemDiv3_003674 CCc1c(C)c(C#N)c2nc3ccccc3n2c1N4CCN(CCO)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G23 mock treatment 1440.0 321.0 0.11 280.0 -400.0 -0.31 -0.1366 -0.4169 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 G24 mock treatment 360.0 -759.0 -0.27 360.0 -320.0 -0.25 -0.364 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H01 compound treatment 840.0 -279.0 -0.1 880.0 200.0 0.15 0.0386 0.2116 3118498 ChemDiv3_003675 CC(C)(C)C1=CC(=O)c2c(O)c(ccc2C1=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H02 compound treatment 880.0 -239.0 -0.08 1640.0 960.0 0.74 0.4613 0.6218 1535282 ChemDiv3_003676 CC(C)COC(=O)C(C)Oc1ccc2c(=O)c(coc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H03 compound treatment 600.0 -519.0 -0.18 800.0 120.0 0.09 -0.065 -0.3158 1658754 ChemDiv3_003677 Cc1ccc(cc1)N2CCN(C2c3cccs3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H04 compound treatment 680.0 -439.0 -0.16 680.0 0.0 0.0 -0.1101 -0.7071 1871037 ChemDiv3_003678 CCc1ccc(cc1)N2C(=O)CC(Sc3ccccn3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H05 compound treatment 2600.0 1480.0 0.53 560.0 -120.0 -0.09 0.3064 0.5744 3118499 ChemDiv3_003679 Brc1ccc(NC(=O)CC2OCCN(Cc3ccccc3)C2=O)c(Br)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H06 compound treatment 480.0 -639.0 -0.23 600.0 -80.0 -0.06 -0.2037 -0.8675 1785758 ChemDiv3_003680 COC(=O)c1cn(C(=O)CCc2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H07 compound treatment 2600.0 1480.0 0.53 1000.0 320.0 0.25 0.5453 0.94 1468921 ChemDiv3_003681 Cc1cc(C)c2c(N)c(sc2n1)C(=O)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H08 compound treatment 680.0 -439.0 -0.16 2120.0 1440.0 1.11 0.6717 0.6016 3118500 ChemDiv3_003682 O=C(Nc1c2CCCc2nc3CCCCc13)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H09 compound treatment 440.0 -679.0 -0.24 680.0 0.0 0.0 -0.1703 -0.7071 3118501 ChemDiv3_003683 Cc1ccc(CN2C(=O)N/C(=C\c3cn(CC(=O)N4CCOCC4)c5ccccc35)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H10 compound treatment 1920.0 801.0 0.28 1160.0 480.0 0.37 0.4616 0.9918 3023610 ChemDiv3_003684 CSc1nc2sc3CCCc3c2c(=O)n1CC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H11 compound treatment 480.0 -639.0 -0.23 560.0 -120.0 -0.09 -0.2254 -0.9214 3023611 ChemDiv3_003685 Cc1ccc(C)c(OC(=O)NC(C)(C(F)(F)F)C(F)(F)F)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H12 compound treatment 3680.0 2560.0 0.91 800.0 120.0 0.09 0.7076 0.7748 3118502 ChemDiv3_003686 O=c1n(Cc2ccccc2)c3cccc4cccc(n1Cc5ccccc5)c43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H13 compound treatment 640.0 -479.0 -0.17 6520.0 5840.0 4.48 3.0502 0.6798 1457236 ChemDiv3_003687 CCOC(=O)c1ccc(NC(=S)NN2CCN(C)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H14 compound treatment 600.0 -519.0 -0.18 8800.0 8120.0 6.23 4.2779 0.6859 1170967 ChemDiv3_003688 CCOC1(NC(=O)c2ccccc2)C(=CC(=O)C=C1C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H15 compound treatment 520.0 -599.0 -0.21 640.0 -40.0 -0.03 -0.1719 -0.801 1870851 ChemDiv3_003689 Cc1ccc(NC(=O)CSc2nnc(C3CC3)n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H16 compound treatment 320.0 -799.0 -0.28 9680.0 9000.0 6.91 4.6854 0.6775 1633513 ChemDiv3_003690 CCc1c(C)c(C#N)c2nc3ccccc3n2c1N4CCN(Cc5cc(Cl)ccc5OC)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H17 compound treatment 1520.0 401.0 0.14 880.0 200.0 0.15 0.2092 0.9993 1255680 ChemDiv3_003691 CC(C)(C)NC(=O)c1cccc(NC(=O)CCC(=O)O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H18 compound treatment 440.0 -679.0 -0.24 880.0 200.0 0.15 -0.0617 -0.216 3023612 ChemDiv3_003692 Cc1cc(o[n+]1C)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H19 compound treatment 1440.0 321.0 0.11 480.0 -200.0 -0.15 -0.028 -0.1464 3118503 ChemDiv3_003693 CCCOc1ccc(/C=C/C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ncccn3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H20 compound treatment 800.0 -319.0 -0.11 8720.0 8040.0 6.17 4.2846 0.694 3023613 ChemDiv3_003694 CCOc1cccc(OCC)c2c(C)[o+]c(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H21 compound treatment 760.0 -359.0 -0.13 720.0 40.0 0.03 -0.0683 -0.5215 3118504 ChemDiv3_003695 CCOC(=O)c1cnc2c(ccc3ccccc32)c1NCCOC(=O)c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H22 compound treatment 560.0 -559.0 -0.2 760.0 80.0 0.06 -0.0967 -0.4661 3023614 ChemDiv3_003696 CCCCS(=O)(=O)N=C1NCN(CN1)C2CCN(Cc3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H23 mock treatment 360.0 -759.0 -0.27 560.0 -120.0 -0.09 -0.2555 -0.898 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 H24 mock treatment 1120.0 1.25 0.0 640.0 -40.0 -0.03 -0.0214 -0.6968 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I01 compound treatment 320.0 -799.0 -0.28 320.0 -360.0 -0.28 -0.3958 -0.9999 3118505 ChemDiv3_003697 COC(=O)C1=CN(C=C(C1c2cccc(O)c2)C(=O)OC)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I02 compound treatment 680.0 -439.0 -0.16 720.0 40.0 0.03 -0.0883 -0.5569 3023615 ChemDiv3_003698 CNc1nc2ccccn2c(=O)c1/C=C/3\SC(=S)N(C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I03 compound treatment 320.0 -799.0 -0.28 360.0 -320.0 -0.25 -0.3741 -0.9975 1485518 ChemDiv3_003699 CCCc1nc2sc3c(ncnc3c2c4CCCCc14)N5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I04 compound treatment 4320.0 3200.0 1.14 320.0 -360.0 -0.28 0.6076 0.5198 1560479 ChemDiv3_003700 CN(C)C(=S)N(C#N)c1nc(nc(n1)N(C)C)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I05 compound treatment 320.0 -799.0 -0.28 560.0 -120.0 -0.09 -0.2655 -0.8911 3118506 ChemDiv3_003701 CCOc1ccc(cc1)N(C(C)C(=O)NCc2ccc(C)cc2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I06 compound treatment 360.0 -759.0 -0.27 480.0 -200.0 -0.15 -0.2989 -0.9646 3118507 ChemDiv3_003702 COc1cccc(OCCSc2nc(cc(=O)[nH]2)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I07 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 3023616 ChemDiv3_003703 C=CCN1C(=O)/C(=C/c2c(Sc3ccccc3)nc4ccccn4c2=O)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I08 compound treatment 2040.0 921.0 0.33 360.0 -320.0 -0.25 0.0574 0.1403 3118508 ChemDiv3_003704 CCOc1ccc(cc1)c2n[nH]c(=S)n2C3CCCC=C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I09 compound treatment 440.0 -679.0 -0.24 400.0 -280.0 -0.21 -0.3223 -0.9984 3023617 ChemDiv3_003705 CSc1nc(c2ccccc2)c3cc(Cl)ccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I10 compound treatment 280.0 -839.0 -0.3 400.0 -280.0 -0.21 -0.3624 -0.9873 3118509 ChemDiv3_003706 CCOC(=O)c1c(CC(C)C)csc1/N=C/C2C(=O)CCCC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I11 compound treatment 200.0 -919.0 -0.33 520.0 -160.0 -0.12 -0.3173 -0.911 1633966 ChemDiv3_003707 CCCOc1ccc(cc1)C(=O)Nc2ccc(NC(=O)c3ccco3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I12 compound treatment 440.0 -679.0 -0.24 280.0 -400.0 -0.31 -0.3874 -0.9928 1787094 ChemDiv3_003708 CCOC(=O)C(C1CCCCC1)C(=O)Nc2cccc(C)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I13 compound treatment 760.0 -359.0 -0.13 520.0 -160.0 -0.12 -0.1768 -0.9998 1440221 ChemDiv3_003709 CCc1ccc(Oc2coc3cc(OC(C)C(=O)OC(C)C)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I14 compound treatment 200.0 -919.0 -0.33 520.0 -160.0 -0.12 -0.3173 -0.911 3023618 ChemDiv3_003710 CCSc1nc(nc2CCCCc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I15 compound treatment 440.0 -679.0 -0.24 720.0 40.0 0.03 -0.1485 -0.612 1433865 ChemDiv3_003711 Clc1ccc(cc1)c2nc(C#N)c(NCCc3ccccc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I16 compound treatment 400.0 -719.0 -0.25 480.0 -200.0 -0.15 -0.2889 -0.9705 3118635 ChemDiv3_003712 O=C1NC(=O)C(=Cc2cn(CCOc3ccc4OCOc4c3)c5ccccc25)C(=O)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I17 compound treatment 560.0 -559.0 -0.2 440.0 -240.0 -0.18 -0.2704 -0.9993 1334972 ChemDiv3_003713 NS(=O)(=O)c1ccc2NC(C3CC=CC3c2c1)C4CCC=CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I18 compound treatment 320.0 -799.0 -0.28 520.0 -160.0 -0.12 -0.2872 -0.93 3118636 ChemDiv3_003714 COC(=O)C1=C(C)N(/C(=C/c2ccc(OC)cc2)/C1=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I19 compound treatment 160.0 -959.0 -0.34 400.0 -280.0 -0.21 -0.3925 -0.9755 3023619 ChemDiv3_003715 Cc1cc(Cl)ccc1OCCCC(=O)NC2CCSC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I20 compound treatment 480.0 -639.0 -0.23 1920.0 1240.0 0.95 0.5129 0.5242 1863329 ChemDiv3_003716 COc1ccc(CCCc2nnc(SCC(=O)NN)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I21 compound treatment 280.0 -839.0 -0.3 1040.0 360.0 0.28 -0.015 -0.0369 3023620 ChemDiv3_003717 OC1(CC(=NN1C(=O)C2CC2)C3CCCCC3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I22 compound treatment 360.0 -759.0 -0.27 960.0 280.0 0.21 -0.0383 -0.1113 1139133 ChemDiv3_003718 CCOC(=O)CCc1c(C)c(C#N)c2nc3ccccc3n2c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I23 mock treatment 400.0 -719.0 -0.25 240.0 -440.0 -0.34 -0.4192 -0.9904 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 I24 mock treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J01 compound treatment 1000.0 -119.0 -0.04 5360.0 4680.0 3.59 2.5108 0.6988 1498091 ChemDiv3_003719 OC(=O)c1ccc(Nc2ncnc3n(Cc4ccccc4)ncc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J02 compound treatment 400.0 -719.0 -0.25 400.0 -280.0 -0.21 -0.3323 -0.9964 1326070 ChemDiv3_003720 O=C(COc1ccc2c(=O)c(coc2c1)c3ccccc3)OC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J03 compound treatment 840.0 -279.0 -0.1 520.0 -160.0 -0.12 -0.1568 -0.9942 3023670 ChemDiv3_003721 Clc1ccc(cc1)c2nc3SCCCn3c(=O)c2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J04 compound treatment 280.0 -839.0 -0.3 360.0 -320.0 -0.25 -0.3841 -0.9955 1870982 ChemDiv3_003722 Cc1nc(=S)sn1c2nc(Nc3ccc(C)cc3)nc(Nc4ccc(C)cc4)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J05 compound treatment 360.0 -759.0 -0.27 640.0 -40.0 -0.03 -0.212 -0.7827 1743126 ChemDiv3_003723 Cc1ccc(C)n1c2sc3CCCCc3c2C(=O)Nc4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J06 compound treatment 120.0 -999.0 -0.35 4760.0 4080.0 3.13 1.9643 0.6232 1262325 ChemDiv3_003724 CCOc1ccc(Nc2nc(nc(n2)N3CCCCC3)N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J07 compound treatment 400.0 -719.0 -0.25 280.0 -400.0 -0.31 -0.3974 -0.9957 3023671 ChemDiv3_003725 Cc1cc(C)c2c(n1)sc3c(=O)n(Cc4ccccc4Cl)nnc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J08 compound treatment 3040.0 1920.0 0.68 320.0 -360.0 -0.28 0.2865 0.3896 1740377 ChemDiv3_003726 CCCCC(CC)C(=O)Nc1c2CCCc2nc3CCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J09 compound treatment 520.0 -599.0 -0.21 280.0 -400.0 -0.31 -0.3673 -0.9838 3023672 ChemDiv3_003727 Cc1cc(/C=C\2/SC(=O)N(C2=O)c3ccccc3)c(C)n1c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J10 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 1371047 ChemDiv3_003728 CC1CCc2c(C1)sc3nc(NN)n(C)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J11 compound treatment 360.0 -759.0 -0.27 360.0 -320.0 -0.25 -0.364 -0.999 3023673 ChemDiv3_003729 CC(NC(=O)Nc1ncccn1)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J12 compound treatment 360.0 -759.0 -0.27 360.0 -320.0 -0.25 -0.364 -0.999 3118637 ChemDiv3_003730 CC1=CC(c2ccc(Cl)cc2)n3nc(NC(=O)CCCC(=O)O)nc3N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J13 compound treatment 200.0 -919.0 -0.33 360.0 -320.0 -0.25 -0.4042 -0.9903 1870817 ChemDiv3_003731 O=c1cc(CSc2nc3ccccc3o2)[nH]c(=S)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J14 compound treatment 640.0 -479.0 -0.17 360.0 -320.0 -0.25 -0.2938 -0.9837 1613843 ChemDiv3_003732 CC1(C)CC2(CCCN(C2)C(=S)Nc3ccccc3)CCO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J15 compound treatment 320.0 -799.0 -0.28 3600.0 2920.0 2.24 1.3848 0.6129 1495361 ChemDiv3_003733 NC(=O)c1cc2C(=O)CCCc2n(c3ccccc3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J16 compound treatment 320.0 -799.0 -0.28 480.0 -200.0 -0.15 -0.3089 -0.9586 1259661 ChemDiv3_003734 CCCc1cc(NCCc2ccccc2)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J17 compound treatment 360.0 -759.0 -0.27 2560.0 1880.0 1.44 0.8302 0.5655 1705780 ChemDiv3_003735 CC(C)C(=O)Nc1cccc(c1)c2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J18 compound treatment 240.0 -879.0 -0.31 320.0 -360.0 -0.28 -0.4159 -0.9982 3023674 ChemDiv3_003736 CC[n+]1oc(cc1C)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J19 compound treatment 440.0 -679.0 -0.24 520.0 -160.0 -0.12 -0.2571 -0.9512 3118638 ChemDiv3_003737 COc1ccc(OCCCC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nccs3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J20 compound treatment 880.0 -239.0 -0.08 1240.0 560.0 0.43 0.2441 0.5571 3023675 ChemDiv3_003738 CCOc1cccc(OCC)c2c(C)[n+](C)c(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J21 compound treatment 360.0 -759.0 -0.27 1400.0 720.0 0.55 0.2005 0.3262 1594999 ChemDiv3_003739 C=CCOc1ccc2c3CCCc3c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J22 compound treatment 440.0 -679.0 -0.24 360.0 -320.0 -0.25 -0.344 -0.9999 3118639 ChemDiv3_003740 Cc1ccc(cc1)S(=O)(=O)N=C2NCN(CN2)C3CCN(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J23 mock treatment 240.0 -879.0 -0.31 360.0 -320.0 -0.25 -0.3941 -0.993 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 J24 mock treatment 1000.0 -119.0 -0.04 360.0 -320.0 -0.25 -0.2035 -0.8164 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K01 compound treatment 280.0 -839.0 -0.3 6720.0 6040.0 4.64 3.0685 0.6604 1440044 ChemDiv3_003741 Nc1cc(=O)nc(SCC(=O)Nc2ccc(Cl)cn2)n1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K02 compound treatment 2120.0 1000.0 0.36 1040.0 360.0 0.28 0.4466 0.9923 1668322 ChemDiv3_003742 Cc1cc(C(=S)N2CCOCC2)c(C)n1c3cccc(C)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K03 compound treatment 520.0 -599.0 -0.21 1920.0 1240.0 0.95 0.523 0.5362 3023676 ChemDiv3_003743 CCOc1ccc(cc1)N(C(C)C(=O)N(C)Cc2ccccc2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K04 compound treatment 480.0 -639.0 -0.23 8000.0 7320.0 5.62 3.8135 0.678 1685444 ChemDiv3_003744 O=C(NCC1COc2ccccc2O1)c3cc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K05 compound treatment 640.0 -479.0 -0.17 1000.0 320.0 0.25 0.0536 0.1795 3118640 ChemDiv3_003745 CCOC(=O)N1CCN(CC1)C(=O)CN(c2cc(ccc2Cl)C(F)(F)F)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K06 compound treatment 360.0 -759.0 -0.27 6320.0 5640.0 4.33 2.8714 0.6619 3023677 ChemDiv3_003746 COc1cccc(NC(=O)CSc2nc(N)cc(=O)[nH]2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K07 compound treatment 520.0 -599.0 -0.21 800.0 120.0 0.09 -0.085 -0.3673 3118641 ChemDiv3_003747 CN1C(=O)/C(=C/c2c(Sc3ccccc3)nc4ccc(C)cn4c2=O)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K08 compound treatment 440.0 -679.0 -0.24 560.0 -120.0 -0.09 -0.2354 -0.9131 3023678 ChemDiv3_003748 CC1CC2(CC(C)(C)C1)NN(C(=S)N2)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K09 compound treatment 2960.0 1840.0 0.65 520.0 -160.0 -0.12 0.375 0.5642 1788362 ChemDiv3_003749 O=C(Sc1ccccn1)N2c3ccccc3Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K10 compound treatment 1320.0 201.0 0.07 520.0 -160.0 -0.12 -0.0364 -0.256 3023679 ChemDiv3_003750 CCOC(=O)c1c(/N=C/C2C(=O)CCCC2=O)scc1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K11 compound treatment 440.0 -679.0 -0.24 1520.0 840.0 0.64 0.2857 0.4151 3118642 ChemDiv3_003751 OC(=O)c1ccccc1C(=O)n2c(COc3ccc(Cl)cc3Cl)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K12 compound treatment 680.0 -439.0 -0.16 680.0 0.0 0.0 -0.1101 -0.7071 3023680 ChemDiv3_003752 Cc1nn(c(C)c1Sc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K13 compound treatment 1000.0 -119.0 -0.04 1320.0 640.0 0.49 0.3176 0.6441 1193366 ChemDiv3_003753 CCc1ccc(Oc2coc3cc(OC(C)C(=O)OCC(C)C)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K14 compound treatment 1240.0 121.0 0.04 6240.0 5560.0 4.27 3.0487 0.7142 3118643 ChemDiv3_003754 NNC(=O)CSc1nc(nc2CCCCc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K15 compound treatment 640.0 -479.0 -0.17 1240.0 560.0 0.43 0.1839 0.3979 3023681 ChemDiv3_003755 O=c1[nH]c(SC/C=C/c2ccccc2)nc3sc4CCCc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K16 compound treatment 600.0 -519.0 -0.18 9720.0 9040.0 6.94 4.7773 0.6881 3118644 ChemDiv3_003756 COc1ccccc1OCCSc2nc(c([nH]2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K17 compound treatment 440.0 -679.0 -0.24 1000.0 320.0 0.25 0.0035 0.01 3023682 ChemDiv3_003757 CC1(C)C(OC(=O)C2(CCCCC2)C1=O)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K18 compound treatment 2120.0 1000.0 0.36 4840.0 4160.0 3.19 2.5095 0.7809 3118645 ChemDiv3_003758 COC(=O)C1=C(C)N/C(=C/c2ccccc2OC)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K19 compound treatment 5280.0 4160.0 1.48 920.0 240.0 0.18 1.1741 0.7892 3118646 ChemDiv3_003759 Cc1cc2ncn(C(=O)CCCOc3ccccc3)c2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K20 compound treatment 560.0 -559.0 -0.2 800.0 120.0 0.09 -0.075 -0.3432 1319748 ChemDiv3_003760 COc1ccc(CCCc2nnc(S)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K21 compound treatment 240.0 -879.0 -0.31 720.0 40.0 0.03 -0.1987 -0.6344 3118647 ChemDiv3_003761 COc1ccc(CC(=O)N2N=C(CC2(O)C(C)(C)C)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K22 compound treatment 720.0 -399.0 -0.14 2120.0 1440.0 1.11 0.6817 0.6116 1425470 ChemDiv3_003762 CC(=O)Nc1ccc(Nc2c3CCCCc3c(C#N)c4nc5ccccc5n24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K23 mock treatment 560.0 -559.0 -0.2 1320.0 640.0 0.49 0.2073 0.3912 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 K24 mock treatment 2120.0 1000.0 0.36 1000.0 320.0 0.25 0.4249 0.9838 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L01 compound treatment 680.0 -439.0 -0.16 1720.0 1040.0 0.8 0.4545 0.5587 3118648 ChemDiv3_003763 CCOc1ccc(N/C=C/C2=[O+]C(C)(C)C(C)(C)O2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L02 compound treatment 560.0 -559.0 -0.2 320.0 -360.0 -0.28 -0.3356 -0.9867 1148259 ChemDiv3_003764 CCOC(=O)c1cnc2ccc(C)cc2c1Nc3ccc(cc3)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L03 compound treatment 920.0 -199.0 -0.07 480.0 -200.0 -0.15 -0.1584 -0.9377 1668601 ChemDiv3_003765 CCOc1ccc(cc1)N2C(=O)c3ccccc3NC2(CC)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L04 compound treatment 1320.0 201.0 0.07 760.0 80.0 0.06 0.0939 0.9972 1871007 ChemDiv3_003766 CC1CC(C)(C)N(C(=O)CSc2nc(C)cc(C)n2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L05 compound treatment 440.0 -679.0 -0.24 520.0 -160.0 -0.12 -0.2571 -0.9512 3118649 ChemDiv3_003767 Cc1ccc(cc1)N2C(=O)C(/C=N/Cc3ccc(cc3)C(=O)O)C(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L06 compound treatment 400.0 -719.0 -0.25 440.0 -240.0 -0.18 -0.3106 -0.9873 1409959 ChemDiv3_003768 CCOc1nc(NC(C)(C)CO)nc(OCC)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L07 compound treatment 520.0 -599.0 -0.21 1000.0 320.0 0.25 0.0235 0.0724 3023683 ChemDiv3_003769 O=c1c(cc2[nH]c3ccccc3c2n1c4ccccc4)[n+]5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L08 compound treatment 1000.0 -119.0 -0.04 2480.0 1800.0 1.38 0.9474 0.6852 1287509 ChemDiv3_003770 CCCn1c2CCCc2c(=N)c3CCCc31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L09 compound treatment 6360.0 5240.0 1.86 1400.0 720.0 0.55 1.7056 0.8793 3118791 ChemDiv3_003771 Cc1ccc(/N=C/2\NC(=O)\C(=C/c3ccc4n(C)c(=O)n(C)c4c3)\S2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L10 compound treatment 480.0 -639.0 -0.23 9200.0 8520.0 6.54 4.4649 0.6822 3023684 ChemDiv3_003772 CCOC(=O)c1sc(nc1C)N2N=C(C)/C(=C\c3ccco3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L11 compound treatment 920.0 -199.0 -0.07 520.0 -160.0 -0.12 -0.1367 -0.9653 1686077 ChemDiv3_003773 CCOc1cc(ccc1OCc2ccccc2F)C(=S)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L12 compound treatment 1600.0 481.0 0.17 640.0 -40.0 -0.03 0.099 0.5708 3023685 ChemDiv3_003774 O=C(Nc1nc2nc(cc(c3ccccc3)n2n1)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L13 compound treatment 520.0 -599.0 -0.21 680.0 0.0 0.0 -0.1502 -0.7071 3118792 ChemDiv3_003775 COc1cc(NC=C2C(=O)c3ccccc3C2=O)cc(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L14 compound treatment 360.0 -759.0 -0.27 3960.0 3280.0 2.52 1.5903 0.6279 3118793 ChemDiv3_003776 COc1ccc(/C=C/C(=O)NCC2(CCOCC2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L15 compound treatment 640.0 -479.0 -0.17 2960.0 2280.0 1.75 1.1176 0.6355 3023686 ChemDiv3_003777 COc1ccc(cc1)n2c3CC(C)(C)CC(=O)c3cc(C(=O)N)c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L16 compound treatment 1040.0 -78.8 -0.03 920.0 240.0 0.18 0.1105 0.5931 1339113 ChemDiv3_003778 CCCc1cc(n2cnc3ccccc23)n4c5ccccc5nc4c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L17 compound treatment 720.0 -399.0 -0.14 920.0 240.0 0.18 0.0303 0.1303 1197106 ChemDiv3_003779 COc1cc2nc(COc3ccccc3)oc(=O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L18 compound treatment 3760.0 2640.0 0.94 600.0 -80.0 -0.06 0.6191 0.6593 1224201 ChemDiv3_003780 CC1CN(CC(C)O1)C(=S)SCC(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L19 compound treatment 1080.0 -38.8 -0.01 1080.0 400.0 0.31 0.2074 0.6748 3023687 ChemDiv3_003781 CCCc1nnc2c3c4CCCCc4sc3ncn12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L20 compound treatment 520.0 -599.0 -0.21 920.0 240.0 0.18 -0.0199 -0.0708 3118794 ChemDiv3_003782 CCOc1ccc/c(=N\C2CCCCC2)/c3c(C)n(C)c(C)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L21 compound treatment 240.0 -879.0 -0.31 600.0 -80.0 -0.06 -0.2639 -0.8305 1403487 ChemDiv3_003783 COC(=O)Oc1ccc2c(=O)c(coc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L22 compound treatment 400.0 -719.0 -0.25 1000.0 320.0 0.25 -0.0066 -0.0186 3118795 ChemDiv3_003784 NC(=NS(=O)(=O)c1ccc(NC(=O)c2ccco2)cc1)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L23 mock treatment 1120.0 1.25 0.0 1120.0 440.0 0.34 0.2392 0.708 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 L24 mock treatment 2280.0 1160.0 0.41 1080.0 400.0 0.31 0.5084 0.9895 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M01 compound treatment 960.0 -159.0 -0.06 1000.0 320.0 0.25 0.1339 0.5312 1167509 ChemDiv3_003785 CCCc1nc(NCc2ccccc2)c(C#N)c3CCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M02 compound treatment 8040.0 6920.0 2.46 1320.0 640.0 0.49 2.0836 0.8321 3023688 ChemDiv3_003786 CC(=O)NS(=O)(=O)c1ccc(cc1)c2ccc(/C=C\3/C(=O)NN(C3=O)c4cccc(Cl)c4)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M03 compound treatment 5440.0 4320.0 1.53 6200.0 5520.0 4.24 4.0805 0.9055 3118796 ChemDiv3_003787 CCOc1ccc(cc1)S(=O)(=O)N(CC(=O)NCc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M04 compound treatment 2760.0 1640.0 0.58 1400.0 720.0 0.55 0.8026 0.9997 1306758 ChemDiv3_003788 CC(NC(=O)COc1ccccc1)C2COc3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M05 compound treatment 600.0 -519.0 -0.18 440.0 -240.0 -0.18 -0.2604 -1.0 1714591 ChemDiv3_003789 COc1ccccc1N(CC(=O)NCc2ccco2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M06 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 1642367 ChemDiv3_003790 Cc1ccc(cc1)N2CCN(C2c3ccncc3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M07 compound treatment 880.0 -239.0 -0.08 880.0 200.0 0.15 0.0487 0.2776 3118797 ChemDiv3_003791 C=CCNc1nc2ccccn2c(=O)c1/C=C/3\SC(=S)N(Cc4ccc5OCOc5c4)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M08 compound treatment 280.0 -839.0 -0.3 400.0 -280.0 -0.21 -0.3624 -0.9873 1732117 ChemDiv3_003792 CCC(=O)NC(=S)Nc1cc(ccc1OC)c2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M09 compound treatment 520.0 -599.0 -0.21 3360.0 2680.0 2.06 1.3047 0.6308 1788364 ChemDiv3_003793 Cc1nnc(SC(=O)N2c3ccccc3Sc4ccccc24)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M10 compound treatment 680.0 -439.0 -0.16 3360.0 2680.0 2.06 1.3448 0.6518 3118798 ChemDiv3_003794 CCOC(=O)c1c(C)c(C)sc1/N=C/C2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M11 compound treatment 400.0 -719.0 -0.25 720.0 40.0 0.03 -0.1586 -0.6175 1693706 ChemDiv3_003795 OC(=O)c1cccc(c1)N2C(SCC2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M12 compound treatment 480.0 -639.0 -0.23 520.0 -160.0 -0.12 -0.2471 -0.9586 3118799 ChemDiv3_003796 COc1ccc(NC(=O)CC2S/C(=N\c3ccccc3)/N(C2=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M13 compound treatment 520.0 -599.0 -0.21 880.0 200.0 0.15 -0.0416 -0.1588 1234541 ChemDiv3_003797 CC1CCc2[nH]c3ccc(cc3c2C1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M14 compound treatment 1080.0 -38.8 -0.01 360.0 -320.0 -0.25 -0.1834 -0.7455 1255457 ChemDiv3_003798 CN(C(=O)Oc1cccc2cccnc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M15 compound treatment 1680.0 561.0 0.2 960.0 280.0 0.21 0.2928 0.9993 3023739 ChemDiv3_003799 CCOC(=O)c1c(C)c(C)sc1N2C(=O)C3ON(C(C3C2=O)c4ccccc4)c5ccccc5C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M16 compound treatment 400.0 -719.0 -0.25 1040.0 360.0 0.28 0.0151 0.0403 3023740 ChemDiv3_003800 CN1C(=O)N(C)C(=O)C(=Cc2cn(Cc3noc(n3)c4ccc(C)cc4)c5ccccc25)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M17 compound treatment 520.0 -599.0 -0.21 5520.0 4840.0 3.72 2.4772 0.6656 3023741 ChemDiv3_003801 O=C(Nc1ccc(cc1)S(=O)(=O)Nc2nccs2)c3cc(nc4ccccc34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M18 compound treatment 400.0 -719.0 -0.25 1000.0 320.0 0.25 -0.0066 -0.0186 3023742 ChemDiv3_003802 COC(=O)C1=C(C)N/C(=C/c2cccs2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M19 compound treatment 600.0 -519.0 -0.18 1240.0 560.0 0.43 0.1739 0.3718 3023743 ChemDiv3_003803 CC1=NN(C(=O)COc2cc(C)cc(C)c2)C(O)(C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M20 compound treatment 960.0 -159.0 -0.06 1000.0 320.0 0.25 0.1339 0.5312 3118800 ChemDiv3_003804 Sc1nnc(COc2ccc3CCCCc3c2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M21 compound treatment 720.0 -399.0 -0.14 2000.0 1320.0 1.01 0.6166 0.6026 3118801 ChemDiv3_003805 COc1ccc(cc1)C2=NN(C(=O)c3ccccc3O)C(O)(C2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M22 compound treatment 280.0 -839.0 -0.3 880.0 200.0 0.15 -0.1018 -0.3041 1363934 ChemDiv3_003806 Cc1nccn1c2c3CCCCc3c(C#N)c4nc5ccccc5n24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M23 mock treatment 400.0 -719.0 -0.25 2920.0 2240.0 1.72 1.0357 0.5958 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 M24 mock treatment 840.0 -279.0 -0.1 5680.0 5000.0 3.84 2.6444 0.6887 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N01 compound treatment 760.0 -359.0 -0.13 960.0 280.0 0.21 0.062 0.2482 3023744 ChemDiv3_003807 CCOC(=O)c1c(NC(=O)C)no[n+]1[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N02 compound treatment 400.0 -719.0 -0.25 520.0 -160.0 -0.12 -0.2672 -0.9439 1330639 ChemDiv3_003808 CC(C)OC(=O)COc1cc2oc(=O)c3CCCc3c2cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N03 compound treatment 520.0 -599.0 -0.21 600.0 -80.0 -0.06 -0.1936 -0.8757 3118802 ChemDiv3_003809 NC(=O)COc1ccc(/C=c\2/sc3nc4ccccc4n3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N04 compound treatment 320.0 -799.0 -0.28 720.0 40.0 0.03 -0.1786 -0.6268 3023745 ChemDiv3_003810 Cc1c(oc2ccc3c(C)cc(=O)oc3c12)/C(=N/O)/c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N05 compound treatment 560.0 -559.0 -0.2 2400.0 1720.0 1.32 0.7936 0.5943 3118803 ChemDiv3_003811 CCn1c(=N)n(CCOc2ccc(C)cc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N06 compound treatment 240.0 -879.0 -0.31 320.0 -360.0 -0.28 -0.4159 -0.9982 3118804 ChemDiv3_003812 Cc1[nH]nc2OC(=C(C#N)C(c12)c3cc(COc4ccccc4Cl)c(C)cc3C)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N07 compound treatment 600.0 -519.0 -0.18 360.0 -320.0 -0.25 -0.3038 -0.9899 1788734 ChemDiv3_003813 Clc1ccc2[nH]c3C(CCCc3c2c1)C(=O)N4CCN(CC4)C(=O)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N08 compound treatment 360.0 -759.0 -0.27 1000.0 320.0 0.25 -0.0166 -0.0456 1583570 ChemDiv3_003814 CCCCN1CCc2c1nc3ccc(Br)cc3c2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N09 compound treatment 320.0 -799.0 -0.28 840.0 160.0 0.12 -0.1135 -0.3675 3118805 ChemDiv3_003815 CCOC(=O)Cn1cc(/C=C/2\C(=O)NC(=O)N(C2=O)c3ccc(F)cc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N10 compound treatment 360.0 -759.0 -0.27 760.0 80.0 0.06 -0.1469 -0.5321 3023746 ChemDiv3_003816 CC1SC(=S)N(C1=O)c2ccc(cc2)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N11 compound treatment 640.0 -479.0 -0.17 400.0 -280.0 -0.21 -0.2721 -0.9932 3023747 ChemDiv3_003817 S=C(N1CCCC1)c2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N12 compound treatment 440.0 -679.0 -0.24 920.0 240.0 0.18 -0.04 -0.1318 3118806 ChemDiv3_003818 C1N2CN3CN1CC(C2)(C3)/N=C\c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N13 compound treatment 320.0 -799.0 -0.28 400.0 -280.0 -0.21 -0.3524 -0.9907 3118807 ChemDiv3_003819 COc1cc(N/C(=C\2/C(=NN(C2=O)c3nc4ccccc4s3)C)/C)cc(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N14 compound treatment 2680.0 1560.0 0.55 880.0 200.0 0.15 0.5002 0.8703 1134380 ChemDiv3_003820 CCCCN(C)c1ncnc2c3cc4COC(C)(C)Cc4nc3sc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N15 compound treatment 1440.0 321.0 0.11 520.0 -160.0 -0.12 -0.0063 -0.0374 3118808 ChemDiv3_003821 Cc1ccc(cc1)n2c3CCCC(=O)c3cc(C(=O)NC4CCSC4=O)c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N16 compound treatment 3400.0 2280.0 0.81 520.0 -160.0 -0.12 0.4854 0.593 1534750 ChemDiv3_003822 CCN(CC)CCNc1c2CCCCc2c(C#N)c3nc4ccccc4n13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N17 compound treatment 320.0 -799.0 -0.28 480.0 -200.0 -0.15 -0.3089 -0.9586 1570102 ChemDiv3_003823 COc1ccc(CC(=O)Nc2cccc(c2)c3nnc(o3)c4ccco4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N18 compound treatment 400.0 -719.0 -0.25 8520.0 7840.0 6.02 4.0757 0.6765 3118809 ChemDiv3_003824 CCc1nnc(NC(=O)c2ccc(cc2)N3C(=O)C4C5CC(C=C5)C4C3=O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N19 compound treatment 360.0 -759.0 -0.27 800.0 120.0 0.09 -0.1252 -0.44 1492524 ChemDiv3_003825 O=c1oc(nc2sc3CCCCc3c12)c4cc5ccccc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N20 compound treatment 440.0 -679.0 -0.24 840.0 160.0 0.12 -0.0834 -0.3085 3118810 ChemDiv3_003826 CC(CCC(=O)O)C1CC[C@H]2C3CCC4CC(=O)CCC4(C)[C@H]3CC(=O)C12C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N21 compound treatment 760.0 -359.0 -0.13 760.0 80.0 0.06 -0.0466 -0.3295 1224438 ChemDiv3_003827 CC(C)COC(=O)C(C)Oc1ccc2c3CCCc3c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N22 compound treatment 2920.0 1800.0 0.64 800.0 120.0 0.09 0.517 0.8008 3118945 ChemDiv3_003828 CCCCS(=O)(=O)N=C1NCN(Cc2ccco2)CN1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N23 mock treatment 2440.0 1320.0 0.47 960.0 280.0 0.21 0.4834 0.9375 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 N24 mock treatment 2880.0 1760.0 0.62 760.0 80.0 0.06 0.4852 0.7729 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O01 compound treatment 240.0 -879.0 -0.31 320.0 -360.0 -0.28 -0.4159 -0.9982 1741234 ChemDiv3_003829 CCCc1nc(NC2CCCCC2)c(C#N)c3CCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O02 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3118946 ChemDiv3_003830 Cc1c(/C=N/c2cccc(NC(=O)c3ccccc3)c2)c(O)n4c5ccccc5nc4c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O03 compound treatment 240.0 -879.0 -0.31 480.0 -200.0 -0.15 -0.329 -0.9468 3023748 ChemDiv3_003831 COc1ccccc1N(CC(=O)N(C)Cc2ccccc2)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O04 compound treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 3118947 ChemDiv3_003832 COc1ccccc1CC(=O)NCC2OCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O05 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 1275170 ChemDiv3_003833 CCOc1ccc(cc1)S(=O)(=O)N(CC(=O)N2CCC(C)CC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O06 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3023749 ChemDiv3_003834 Brc1ccc(cc1)C2=CC(=O)C=CC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O07 compound treatment 440.0 -679.0 -0.24 280.0 -400.0 -0.31 -0.3874 -0.9928 1119910 ChemDiv3_003835 COc1ccc2c(C)c(CC(C)O)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O08 compound treatment 720.0 -399.0 -0.14 280.0 -400.0 -0.31 -0.3172 -0.9381 3118948 ChemDiv3_003836 CCOC(=O)c1c(/N=C/C2C(=O)NC(=S)NC2=O)sc3CCCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O09 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 1870831 ChemDiv3_003837 CCOC(=O)Oc1ccc2N(C(=O)OCC)C(C)(C)C=C(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O10 compound treatment 280.0 -839.0 -0.3 360.0 -320.0 -0.25 -0.3841 -0.9955 3118949 ChemDiv3_003838 CCOC(=O)c1cc(CC)sc1/N=C/C2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O11 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 1259659 ChemDiv3_003839 Cc1ccc2nc(C)cc(NC3CCCCC3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O12 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 1450973 ChemDiv3_003840 CCOc1ccccc1N2C(=O)CC(N(O)c3ccccc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O13 compound treatment 360.0 -759.0 -0.27 400.0 -280.0 -0.21 -0.3423 -0.9938 1696898 ChemDiv3_003841 COC(=O)c1ccc2nc(C)cc(O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O14 compound treatment 1000.0 -119.0 -0.04 240.0 -440.0 -0.34 -0.2686 -0.7892 1458066 ChemDiv3_003842 CCN(CC)C(=O)Oc1ccnc2cc(Cl)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O15 compound treatment 320.0 -799.0 -0.28 280.0 -400.0 -0.31 -0.4175 -0.9992 1562065 ChemDiv3_003843 CCOC(=O)C1=C(Nc2nnnn2C1c3ccc(Br)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O16 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 3023750 ChemDiv3_003844 CNC(=O)CN1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O17 compound treatment 240.0 -879.0 -0.31 400.0 -280.0 -0.21 -0.3724 -0.9835 3118950 ChemDiv3_003845 COC(=O)C(CC(C)C)NC(=O)c1cc(nc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O18 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 1303884 ChemDiv3_003846 Nc1ncn(n1)C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O19 compound treatment 240.0 -879.0 -0.31 560.0 -120.0 -0.09 -0.2856 -0.8785 3118951 ChemDiv3_003847 OC1(C2CCCCC2=NN1C(=O)c3ccccc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O20 compound treatment 360.0 -759.0 -0.27 440.0 -240.0 -0.18 -0.3206 -0.9829 1381604 ChemDiv3_003848 Cc1cc(N2CCCC2)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O21 compound treatment 240.0 -879.0 -0.31 240.0 -440.0 -0.34 -0.4593 -0.9992 3118952 ChemDiv3_003849 OC1(CC(=NN1C(=O)C2CC2)c3ccc(Cl)cc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O22 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 1172393 ChemDiv3_003850 COc1ccc(CN2CCN(CC2)c3ncnc4scc(c5ccc(Cl)cc5)c34)cc1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O23 mock treatment 440.0 -679.0 -0.24 240.0 -440.0 -0.34 -0.4091 -0.9862 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 O24 mock treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P01 compound treatment 160.0 -959.0 -0.34 200.0 -480.0 -0.37 -0.5011 -0.9992 1604660 ChemDiv3_003851 CCC(Sc1nnnn1c2ccccc2)C(=O)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P02 compound treatment 400.0 -719.0 -0.25 360.0 -320.0 -0.25 -0.354 -0.9998 3118953 ChemDiv3_003852 FC(F)(F)c1cccc(/N=C/2\NC(=N)c3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P03 compound treatment 200.0 -919.0 -0.33 200.0 -480.0 -0.37 -0.491 -0.9981 1143801 ChemDiv3_003853 OC1(CC(=O)c2ccc(Br)cc2)C(=O)N(Cc3ccccc3)c4ccccc41 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P04 compound treatment 240.0 -879.0 -0.31 200.0 -480.0 -0.37 -0.481 -0.9965 1397253 ChemDiv3_003854 COc1ccc(cc1)C(=O)NCc2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P05 compound treatment 240.0 -879.0 -0.31 280.0 -400.0 -0.31 -0.4376 -1.0 3118954 ChemDiv3_003855 CCOC(=O)N1CCN(CC1)C(=O)CN(Cc2cccc(C)c2)S(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P06 compound treatment 320.0 -799.0 -0.28 240.0 -440.0 -0.34 -0.4392 -0.9962 1737242 ChemDiv3_003856 CC1(C)Cc2nc3sc4c(NN)ncnc4c3cc2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P07 compound treatment 280.0 -839.0 -0.3 320.0 -360.0 -0.28 -0.4058 -0.9993 3118955 ChemDiv3_003857 CS(=O)(=O)N(Cc1ccccc1)c2ccc(cc2)C(=O)NCCSc3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P08 compound treatment 360.0 -759.0 -0.27 280.0 -400.0 -0.31 -0.4075 -0.9978 1681828 ChemDiv3_003858 CCOc1ccc(cc1)N2CCc3c2nc4ccc(Br)cc4c3N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P09 compound treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 3023751 ChemDiv3_003859 Cc1cc(C=C2C(=O)OC(C)(C)OC2=O)c(C)n1c3ccc(I)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P10 compound treatment 5240.0 4120.0 1.46 200.0 -480.0 -0.37 0.7732 0.5128 3023752 ChemDiv3_003860 Clc1ccc(cc1)c2nc3cccc4cccc([nH]2)c43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P11 compound treatment 360.0 -759.0 -0.27 360.0 -320.0 -0.25 -0.364 -0.999 1334154 ChemDiv3_003861 Clc1ccc(Cn2cc(C(=S)N3CCCC3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P12 compound treatment 2440.0 1320.0 0.47 240.0 -440.0 -0.34 0.0926 0.1602 1027643 ChemDiv3_003862 OC(=O)CSC(=S)N1CCOCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P13 compound treatment 4480.0 3360.0 1.19 240.0 -440.0 -0.34 0.6043 0.4876 3118956 ChemDiv3_003863 O=C1CC(CC(=O)C1=CNCCN2CCNCC2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P14 compound treatment 920.0 -199.0 -0.07 240.0 -440.0 -0.34 -0.2887 -0.8367 1538427 ChemDiv3_003864 CC1(C)Cc2nc3sc4c(NCC5CCCO5)ncnc4c3cc2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P15 compound treatment 2560.0 1440.0 0.51 280.0 -400.0 -0.31 0.1444 0.2421 1219327 ChemDiv3_003865 O=C(Nc1ccccc1)c2cc3C(=O)CCCc3n(c4ccccc4)c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P16 compound treatment 680.0 -439.0 -0.16 280.0 -400.0 -0.31 -0.3272 -0.9504 1621677 ChemDiv3_003866 Cc1ccc(OCCN2CCN(CC2)c3ncnc4scc(c5ccccc5)c34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P17 compound treatment 640.0 -479.0 -0.17 200.0 -480.0 -0.37 -0.3807 -0.9382 3118957 ChemDiv3_003867 O=C1NC(=O)/C(=C/c2c[nH]c3ccccc23)/C(=O)N1C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P18 compound treatment 280.0 -839.0 -0.3 240.0 -440.0 -0.34 -0.4493 -0.998 3023753 ChemDiv3_003868 CCc1nnc(NC(=O)C(C)N2C(=O)C3C4CC(C=C4)C3C2=O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P19 compound treatment 1880.0 761.0 0.27 280.0 -400.0 -0.31 -0.0262 -0.064 3118958 ChemDiv3_003869 CCC(C)OC(=O)CSc1ncnc2sc3CC(C)CCc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P20 compound treatment 560.0 -559.0 -0.2 240.0 -440.0 -0.34 -0.379 -0.9677 3023754 ChemDiv3_003870 Cc1cc2NC(=CC(=Nc2cc1C)c3cccs3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P21 compound treatment 280.0 -839.0 -0.3 480.0 -200.0 -0.15 -0.319 -0.9526 1262711 ChemDiv3_003871 CCC(C)OC(=O)C(C)Oc1ccc2c3CCCc3c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P22 compound treatment 360.0 -759.0 -0.27 320.0 -360.0 -0.28 -0.3858 -0.9999 1606981 ChemDiv3_003872 OC1(CC(=O)c2ccccc2)C(=O)N(CC=C)c3ccccc31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P23 mock treatment 280.0 -839.0 -0.3 280.0 -400.0 -0.31 -0.4275 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2011 P24 mock treatment 1320.0 201.0 0.07 240.0 -440.0 -0.34 -0.1884 -0.5456 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A01 compound treatment 600.0 -275.0 -0.1 320.0 -240.0 -0.18 -0.1993 -0.9558 1871572 ChemDiv3_004225 O=C(CSC(=S)N1CCCCC1)N2c3ccccc3CCc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A02 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 3120044 ChemDiv3_004226 CCOc1ccc2cc(C3CC(=NN3S(=O)(=O)c4ccccc4)c5ccco5)c(Cl)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A03 compound treatment 360.0 -515.0 -0.18 320.0 -240.0 -0.18 -0.2595 -1.0 1572427 ChemDiv3_004227 Cc1nn2c(c1C(=S)Nc3ccccc3)n(C)c4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A04 compound treatment 1080.0 205.0 0.07 280.0 -280.0 -0.21 -0.1006 -0.4432 1416443 ChemDiv3_004228 OC1CCC(CC1)n2c(nc(=S)c3CCCCc32)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A05 compound treatment 920.0 45.0 0.02 600.0 40.0 0.03 0.033 0.9535 1490702 ChemDiv3_004229 CS(=O)(=O)c1ccc2nc(NC(=O)Oc3ccccc3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A06 compound treatment 240.0 -635.0 -0.23 5880.0 5320.0 4.08 2.7287 0.6671 3023292 ChemDiv3_004230 Cc1[nH]c2ccccc2c1C(Nc3ccccn3)c4ccc(cc4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A07 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 3120045 ChemDiv3_004231 Cn1c(=N)n(CCOc2ccccc2Cl)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A08 compound treatment 1080.0 205.0 0.07 280.0 -280.0 -0.21 -0.1006 -0.4432 1873167 ChemDiv3_004232 CC(Nc1cc(C)c(C#N)c2nc3ccccc3n12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A09 compound treatment 440.0 -435.0 -0.15 280.0 -280.0 -0.21 -0.2611 -0.9868 3023296 ChemDiv3_004233 CCn1c2/C(=N/O)/CCCc2c3cc(ccc13)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A10 compound treatment 1080.0 205.0 0.07 320.0 -240.0 -0.18 -0.0789 -0.3981 1873230 ChemDiv3_004234 COc1ccc(CCNc2c(CC=C)c(C)c(C#N)c3nc4ccccc4n23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A11 compound treatment 280.0 -595.0 -0.21 200.0 -360.0 -0.28 -0.3447 -0.9911 3023348 ChemDiv3_004235 O/N=C/1\C(=O)N(CN2CCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A12 compound treatment 480.0 -395.0 -0.14 160.0 -400.0 -0.31 -0.3162 -0.9368 1286346 ChemDiv3_004236 COc1ccc(cc1)c2nn(cc2C(=O)N(C)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A13 compound treatment 280.0 -595.0 -0.21 440.0 -120.0 -0.09 -0.2144 -0.9309 1242885 ChemDiv3_004237 O=C(N1CCCCC1)N2c3ccccc3Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A14 compound treatment 280.0 -595.0 -0.21 720.0 160.0 0.12 -0.0624 -0.2555 1191358 ChemDiv3_004238 CCOC(=O)Nc1cc(C(=O)OCC)c(C)nc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A15 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 1469246 ChemDiv3_004239 CC1(C)CC2(CCO1)OC(=O)CC2C(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A16 compound treatment 240.0 -635.0 -0.23 4200.0 3640.0 2.79 1.8167 0.648 1401727 ChemDiv3_004240 CNS(=O)(=O)c1ccc2[nH]c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A17 compound treatment 280.0 -595.0 -0.21 480.0 -80.0 -0.06 -0.1927 -0.8765 1494565 ChemDiv3_004241 COc1ccc(cc1)C(C2=C(O)CC(C)(C)CC2=O)c3c(C)[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A18 compound treatment 160.0 -715.0 -0.25 280.0 -280.0 -0.21 -0.3314 -0.9966 1028707 ChemDiv3_004242 C(N1CCN(Cc2c[nH]c3ccccc23)CC1)c4c[nH]c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A19 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 1584523 ChemDiv3_004243 COc1ccc(cc1OC)c2n[nH]c(=S)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A20 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 1669366 ChemDiv3_004244 COc1ccc(cc1)c2nc3ccccc3n2CCOc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A21 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 3023360 ChemDiv3_004245 Cc1ccc(NC(=O)CC(NCC2CCCO2)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A22 compound treatment 280.0 -595.0 -0.21 480.0 -80.0 -0.06 -0.1927 -0.8765 1639148 ChemDiv3_004246 Brc1ccc(NC(=O)CCNS(=O)(=O)c2ccccc2)c(c1)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A23 mock treatment 160.0 -715.0 -0.25 360.0 -200.0 -0.15 -0.2879 -0.9711 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 A24 mock treatment 400.0 -475.0 -0.17 240.0 -320.0 -0.25 -0.2929 -0.9831 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B01 compound treatment 160.0 -715.0 -0.25 280.0 -280.0 -0.21 -0.3314 -0.9966 1208457 ChemDiv3_004247 Cc1ccc(cc1C)C(=O)COC(=O)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B02 compound treatment 320.0 -555.0 -0.2 160.0 -400.0 -0.31 -0.3564 -0.9769 3023400 ChemDiv3_004248 Cc1ccc(cc1)C(=O)/C=C/2\NC(=NC2=O)NS(=O)(=O)c3ccc(N)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B03 compound treatment 320.0 -555.0 -0.2 240.0 -320.0 -0.25 -0.3129 -0.994 3120180 ChemDiv3_004249 CC(NC(=O)c1cc2c(=O)n3cccc(C)c3nc2n(CC4CCCO4)c1=N)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B04 compound treatment 240.0 -635.0 -0.23 360.0 -200.0 -0.15 -0.2679 -0.9825 3120181 ChemDiv3_004250 CCC1CCc2nc3sc(C(=O)Nc4cc(Cl)ccc4OC)c(N)c3cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B05 compound treatment 600.0 -275.0 -0.1 280.0 -280.0 -0.21 -0.221 -0.9361 3023403 ChemDiv3_004251 CCCn1c(=N)c(cc2c(=O)n3cc(C)ccc3nc12)C(=O)NC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B06 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3120182 ChemDiv3_004252 Cn1cc(C2Nc3sc4CCCCc4c3C(=N2)O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B07 compound treatment 360.0 -515.0 -0.18 360.0 -200.0 -0.15 -0.2378 -0.9963 3023406 ChemDiv3_004253 CCN/1C(=O)C(S\C1=N\c2ccc(cc2)C(=O)OC)C(O)c3cc(OC)ccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B08 compound treatment 360.0 -515.0 -0.18 240.0 -320.0 -0.25 -0.3029 -0.9894 3120183 ChemDiv3_004254 COc1cc(/C=C/2\NC(=S)N(C)C2=O)ccc1OCc3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B09 compound treatment 520.0 -355.0 -0.13 320.0 -240.0 -0.18 -0.2193 -0.9828 1671194 ChemDiv3_004255 Cc1cccc(c1)C(=O)Nc2nc3CC(C)(C)CC(=O)c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B10 compound treatment 240.0 -635.0 -0.23 200.0 -360.0 -0.28 -0.3547 -0.9948 3120184 ChemDiv3_004256 OC(=O)CCc1nc2cc(ccc2[nH]1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B11 compound treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 3120185 ChemDiv3_004257 FC(F)(F)c1cc(nc(n1)S(=O)(=O)Cc2cccc(Cl)c2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B12 compound treatment 440.0 -435.0 -0.15 240.0 -320.0 -0.25 -0.2828 -0.9749 1719820 ChemDiv3_004258 CC1(C)C2CCC1(C)c3c2c(nn3c4ccccc4)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B13 compound treatment 400.0 -475.0 -0.17 200.0 -360.0 -0.28 -0.3146 -0.9718 3120186 ChemDiv3_004259 C=CCN1C2=NC(=O)CN2c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B14 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 1317554 ChemDiv3_004260 CC(C)(C)Nc1nc2nonc2nc1NC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B15 compound treatment 560.0 -315.0 -0.11 240.0 -320.0 -0.25 -0.2527 -0.9364 3120187 ChemDiv3_004261 CCCn1c(SCCCc2ccccc2)nc3n(C)c(=O)[nH]c(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B16 compound treatment 360.0 -515.0 -0.18 680.0 120.0 0.09 -0.064 -0.313 3120188 ChemDiv3_004262 COC(=O)c1ccc(cc1)[C@@H]2Nc3c(C)cccc3[C@@H]4C=CC[C@@H]42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B17 compound treatment 400.0 -475.0 -0.17 320.0 -240.0 -0.18 -0.2494 -0.999 1361311 ChemDiv3_004263 CCOC(=O)c1cc2c(C)n(c(C)c2cc(C(=O)OCC)c1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B18 compound treatment 200.0 -675.0 -0.24 240.0 -320.0 -0.25 -0.343 -0.9999 3120189 ChemDiv3_004264 OC(=O)c1ccc(CSc2nnc(COc3ccc(Cl)cc3Cl)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B19 compound treatment 560.0 -315.0 -0.11 280.0 -280.0 -0.21 -0.231 -0.9535 1150810 ChemDiv3_004265 COc1ccc(OCC(O)CNC(=O)c2ccccc2C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B20 compound treatment 360.0 -515.0 -0.18 640.0 80.0 0.06 -0.0858 -0.4449 3120190 ChemDiv3_004266 S=C(Nc1ccc2nsnc2c1)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B21 compound treatment 200.0 -675.0 -0.24 1280.0 720.0 0.55 0.2215 0.3678 3120191 ChemDiv3_004267 NC(=O)c1c(NCCO)nc(cc1C(F)(F)F)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B22 compound treatment 320.0 -555.0 -0.2 19400.0 18800.0 14.46 10.0882 0.6974 3023474 ChemDiv3_004268 OC(=O)c1ccc(cc1)N2N=C(/C(=C/c3ccc(OC(=O)c4cccs4)cc3)/C2=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B23 mock treatment 200.0 -675.0 -0.24 6360.0 5800.0 4.45 2.9793 0.6681 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 B24 mock treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C01 compound treatment 280.0 -595.0 -0.21 440.0 -120.0 -0.09 -0.2144 -0.9309 3023414 ChemDiv3_004269 Cc1cc(O)nc(NC(=N)Nc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C02 compound treatment 160.0 -715.0 -0.25 240.0 -320.0 -0.25 -0.3531 -0.9999 3120192 ChemDiv3_004270 Cc1ccc(cc1)C2=NN(C(C2)c3ccc4nccnc4c3)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C03 compound treatment 320.0 -555.0 -0.2 360.0 -200.0 -0.15 -0.2478 -0.9924 3023419 ChemDiv3_004271 COc1ccc(C=C2C(=O)OC(C)(OC2=O)C(C)(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C04 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 1343660 ChemDiv3_004272 NS(=O)(=O)c1ccc(CCn2c(nc(=S)c3CCCCc32)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C05 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 1645275 ChemDiv3_004273 CCOC(=O)c1cnc2c(C)c(Cl)ccc2c1Nc3cc(C)ccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C06 compound treatment 160.0 -715.0 -0.25 360.0 -200.0 -0.15 -0.2879 -0.9711 3120193 ChemDiv3_004274 COc1cccc(c1)C(Nc2ccccn2)c3c(C)[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C07 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 1260066 ChemDiv3_004275 N=c1n(CCOc2ccccc2)c3ccccc3n1Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C08 compound treatment 2320.0 1450.0 0.51 400.0 -160.0 -0.12 0.2756 0.5229 1873175 ChemDiv3_004276 CCc1c(C)c(C#N)c2nc3ccccc3n2c1NCCC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C09 compound treatment 520.0 -355.0 -0.13 240.0 -320.0 -0.25 -0.2628 -0.9518 3120194 ChemDiv3_004277 N#CCCN1CCn2c3ccc(cc3c4cccc1c24)C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C10 compound treatment 240.0 -635.0 -0.23 240.0 -320.0 -0.25 -0.333 -0.9991 3120195 ChemDiv3_004278 CC1CCN(CC1)c2ncnc3n(Cc4ccc(Cl)cc4)ncc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C11 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 3023477 ChemDiv3_004279 COc1cc(ccc1O)c2nc3c([nH]2)c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C12 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 3120196 ChemDiv3_004280 COc1ccc(cc1OC)c2nn(cc2C(=O)Oc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C13 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 1388153 ChemDiv3_004281 Cc1ccc(NC(=O)N2c3ccccc3Sc4ccccc24)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C14 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 3120197 ChemDiv3_004282 COC(=O)c1ccc(O)c(/C=N/N(CCO)C2=NS(=O)(=O)c3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C15 compound treatment 560.0 -315.0 -0.11 280.0 -280.0 -0.21 -0.231 -0.9535 1407736 ChemDiv3_004283 COC(=O)c1c(C)c(C)sc1NC(=O)CC2Nc3cc(C)c(C)cc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C16 compound treatment 13240.0 12400.0 4.39 3000.0 2440.0 1.87 4.4263 0.928 3023484 ChemDiv3_004284 CC/1=NN(C(=O)\C1=C/C=C\c2ccccc2)c3ccc(cc3)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C17 compound treatment 280.0 -595.0 -0.21 360.0 -200.0 -0.15 -0.2578 -0.9878 1706298 ChemDiv3_004285 CCOC(=O)c1c(C)oc2c1c3CN(CCc4ccccc4)COc3c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C18 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 1247453 ChemDiv3_004286 CCOC(=O)c1ccc(NCc2ccc(cc2)N(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C19 compound treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 1444763 ChemDiv3_004287 CCOC(=O)c1c(C)n(c2ccc(C)cc2)c3ccc(OCC(O)CNCC4CCCO4)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C20 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3024350 ChemDiv3_004288 Nc1ccc(cc1)c2nc3ccccc3n2CCCOc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C21 compound treatment 320.0 -555.0 -0.2 360.0 -200.0 -0.15 -0.2478 -0.9924 3024351 ChemDiv3_004289 Cc1cc(C)cc(NC(=O)CC(NCc2cccnc2)C(=O)O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C22 compound treatment 360.0 -515.0 -0.18 560.0 0.0 0.0 -0.1292 -0.7071 1315276 ChemDiv3_004290 CC(C)(C)SCC(O)Cn1c2ccc(Cl)cc2c3cc(Cl)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C23 mock treatment 240.0 -635.0 -0.23 360.0 -200.0 -0.15 -0.2679 -0.9825 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 C24 mock treatment 600.0 -275.0 -0.1 240.0 -320.0 -0.25 -0.2427 -0.9182 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D01 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3024352 ChemDiv3_004291 OC(=O)c1ccc(cc1)c2nnc(o2)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D02 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 3024353 ChemDiv3_004292 OC1=C(C(=O)c2ccc(F)cc2)C3(OC1=O)C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D03 compound treatment 240.0 -635.0 -0.23 240.0 -320.0 -0.25 -0.333 -0.9991 3024354 ChemDiv3_004293 COC(=O)c1cc2c(=O)n3cccc(C)c3nc2n(CC=C)c1=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D04 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 3024355 ChemDiv3_004294 CN1CCc2nc(SCc3cccc(Cl)c3)c(C#N)cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D05 compound treatment 400.0 -475.0 -0.17 280.0 -280.0 -0.21 -0.2712 -0.9927 3120198 ChemDiv3_004295 CCCn1c(=N)c(cc2c(=O)n3ccccc3nc12)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D06 compound treatment 360.0 -515.0 -0.18 240.0 -320.0 -0.25 -0.3029 -0.9894 3024356 ChemDiv3_004296 CCc1ccc(Nc2cc(=O)oc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D07 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3120199 ChemDiv3_004297 O=S(=O)(Nc1ccccc1)c2ccc3oc4ccc(cc4c3c2)S(=O)(=O)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D08 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 3024357 ChemDiv3_004298 CC(Sc1nc2ccc(Br)cc2[nH]1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D09 compound treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 3117747 ChemDiv3_004299 O=C(Nc1ccc(cc1)S(=O)(=O)NCCc2ccccc2)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D10 compound treatment 200.0 -675.0 -0.24 280.0 -280.0 -0.21 -0.3213 -0.9986 3024358 ChemDiv3_004300 COC(=O)c1ccccc1NC(=O)CSc2nnc(CSc3nc(C)cc(C)n3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D11 compound treatment 320.0 -555.0 -0.2 240.0 -320.0 -0.25 -0.3129 -0.994 3117748 ChemDiv3_004301 COc1ccc(OC)c2c(cc(nc12)C(F)(F)F)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D12 compound treatment 320.0 -555.0 -0.2 400.0 -160.0 -0.12 -0.2261 -0.9742 3024359 ChemDiv3_004302 CCOC(=O)CC1=NN=C(N)SC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D13 compound treatment 200.0 -675.0 -0.24 440.0 -120.0 -0.09 -0.2345 -0.9139 3117749 ChemDiv3_004303 CN(C)CCCn1c(=N)n(CC(O)C(C)(C)C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D14 compound treatment 280.0 -595.0 -0.21 200.0 -360.0 -0.28 -0.3447 -0.9911 1785039 ChemDiv3_004304 CCOC(=O)/C=C/1\CC(=O)Nc2cc(C)c(C)cc2N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D15 compound treatment 360.0 -515.0 -0.18 280.0 -280.0 -0.21 -0.2812 -0.9967 3117750 ChemDiv3_004305 Fc1ccc(cc1)C(=O)N2CCCCC(Sc3ncnc4sc5CCCc5c34)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D16 compound treatment 440.0 -435.0 -0.15 400.0 -160.0 -0.12 -0.196 -0.9936 3117751 ChemDiv3_004306 COc1cc(/C=C\2/C(=O)ON=C2c3ccccc3)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D17 compound treatment 400.0 -475.0 -0.17 320.0 -240.0 -0.18 -0.2494 -0.999 1307290 ChemDiv3_004307 Oc1c(ccc2cccnc12)C(N3CCCCC3)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D18 compound treatment 360.0 -515.0 -0.18 320.0 -240.0 -0.18 -0.2595 -1.0 3117752 ChemDiv3_004308 Cn1c(=O)n(C)c2cc(/C=C\3/NC(=O)NC3=O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D19 compound treatment 240.0 -635.0 -0.23 560.0 0.0 0.0 -0.1593 -0.7071 1180264 ChemDiv3_004309 OC(CN1C(=O)c2ccccc2S1(=O)=O)Cn3c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D20 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3024361 ChemDiv3_004310 CCN(CC)C(=S)Nc1ccc2nsnc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D21 compound treatment 360.0 -515.0 -0.18 320.0 -240.0 -0.18 -0.2595 -1.0 1118442 ChemDiv3_004311 Fc1cn(C2CCCO2)c(=O)n(Cc3ccc(Cl)cc3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D22 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3117753 ChemDiv3_004312 Cc1ccc(cc1)C2=NCN(C(=S)N2)c3ccc(cc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D23 mock treatment 440.0 -435.0 -0.15 200.0 -360.0 -0.28 -0.3045 -0.9621 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 D24 mock treatment 320.0 -555.0 -0.2 600.0 40.0 0.03 -0.1175 -0.5897 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E01 compound treatment 1720.0 845.0 0.3 1360.0 800.0 0.61 0.6462 0.9456 3117754 ChemDiv3_004313 COCc1cc(=O)[nH]c(N/C(=N/C(=O)c2ccc(C)cc2)/Nc3cccc(Cl)c3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E02 compound treatment 480.0 -395.0 -0.14 1560.0 1000.0 0.77 0.4438 0.5687 3024362 ChemDiv3_004314 CCS(=O)(=O)N1N=C(CC1c2cc3cc4OCCOc4cc3nc2Cl)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E03 compound treatment 1600.0 725.0 0.26 320.0 -240.0 -0.18 0.0516 0.163 1488515 ChemDiv3_004315 Cc1c(N)c2c3CCCCc3sc2nc1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E04 compound treatment 1080.0 205.0 0.07 400.0 -160.0 -0.12 -0.0354 -0.2482 3117755 ChemDiv3_004316 Cc1ccc(cc1)S(=O)(=O)NC2C(Sc3ccccn3)c4cccc5cccc2c45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E05 compound treatment 4400.0 3530.0 1.25 680.0 120.0 0.09 0.9494 0.7571 1192256 ChemDiv3_004317 CCn1cc(C(=O)O)c(=O)c2cc(F)c(F)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E06 compound treatment 1240.0 365.0 0.13 320.0 -240.0 -0.18 -0.0387 -0.172 3024363 ChemDiv3_004318 CCOC(=S)SCc1cn2ccc(C)cc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E07 compound treatment 680.0 -195.0 -0.07 920.0 360.0 0.28 0.1465 0.5143 3117756 ChemDiv3_004319 CCC(C)c1ccc(NC(=O)C2CN(C(=O)C2)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E08 compound treatment 280.0 -595.0 -0.21 640.0 80.0 0.06 -0.1058 -0.4814 3024364 ChemDiv3_004320 Cc1c(Cc2ccc(Cl)cc2)c(=O)n3c4ccccc4[nH]c3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E09 compound treatment 2840.0 1970.0 0.7 800.0 240.0 0.18 0.6232 0.8643 3117757 ChemDiv3_004321 Cc1cc(C)c2c(n1)sc3c(SCc4ccccc4)nc(C)nc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E10 compound treatment 640.0 -235.0 -0.08 360.0 -200.0 -0.15 -0.1675 -0.9588 3117758 ChemDiv3_004322 Cc1ccc(s1)S(=O)(=O)N2CCC(CC2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E11 compound treatment 640.0 -235.0 -0.08 2280.0 1720.0 1.32 0.8748 0.6611 1202603 ChemDiv3_004323 O=C(Nc1cccc2CCCCc12)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E12 compound treatment 280.0 -595.0 -0.21 2080.0 1520.0 1.17 0.6759 0.57 3117759 ChemDiv3_004324 COC(=O)c1cn(nc1c2cccnc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E13 compound treatment 920.0 45.0 0.02 1160.0 600.0 0.46 0.337 0.7312 3117760 ChemDiv3_004325 Cc1ccccc1n2c(S)nc3nc4CCCCc4cc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E14 compound treatment 4440.0 3570.0 1.26 3440.0 2880.0 2.21 2.4577 0.9649 3024365 ChemDiv3_004326 O=C(OCCNC1=NS(=O)(=O)c2ccccc12)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E15 compound treatment 2560.0 1690.0 0.6 2200.0 1640.0 1.26 1.313 0.942 1253252 ChemDiv3_004327 COc1ccc(cc1)C2C3C(ON2c4ccccc4)C(=O)NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E16 compound treatment 560.0 -315.0 -0.11 600.0 40.0 0.03 -0.0573 -0.4945 3024366 ChemDiv3_004328 CCCCC1(C)OC(=O)C(=Cc2ccc(OCC)c(OC)c2)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E17 compound treatment 720.0 -155.0 -0.05 1000.0 440.0 0.34 0.2 0.5843 1304057 ChemDiv3_004329 CCCCN1COc2c(C1)cc(Cl)c3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E18 compound treatment 1080.0 205.0 0.07 5080.0 4520.0 3.47 2.5051 0.7218 1268625 ChemDiv3_004330 CC(C)Oc1ccc(NP(=O)(C)Oc2cc(C)cc(C)c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E19 compound treatment 880.0 5.0 0.0 2680.0 2120.0 1.63 1.1521 0.7079 1125399 ChemDiv3_004331 O=C1CC(=O)N(N1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E20 compound treatment 920.0 45.0 0.02 680.0 120.0 0.09 0.0764 0.8175 1655164 ChemDiv3_004332 COC(=O)c1ccc(cc1)N2C(=O)C3ON(C(C3C2=O)c4ccc(F)cc4)c5ccccc5C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E21 compound treatment 1480.0 605.0 0.21 600.0 40.0 0.03 0.1735 0.8001 3024367 ChemDiv3_004333 Cc1c(Cl)cccc1NC(=O)CC(NCc2ccccn2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E22 compound treatment 4680.0 3810.0 1.35 760.0 200.0 0.15 1.063 0.7825 3117761 ChemDiv3_004334 CN(C)c1ccc(cc1)C2CC(=NN2S(=O)(=O)C)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E23 mock treatment 1760.0 885.0 0.31 640.0 80.0 0.06 0.2654 0.8297 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 E24 mock treatment 320.0 -555.0 -0.2 1320.0 760.0 0.58 0.2734 0.4439 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F01 compound treatment 560.0 -315.0 -0.11 520.0 -40.0 -0.03 -0.1007 -0.8692 3024368 ChemDiv3_004335 Cc1cc(/C=N/n2cnnc2)c(C)n1c3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F02 compound treatment 3360.0 2490.0 0.88 1000.0 440.0 0.34 0.8622 0.9133 3117762 ChemDiv3_004336 CN(C)C(=N)c1nn[nH]c1SCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F03 compound treatment 720.0 -155.0 -0.05 1480.0 920.0 0.71 0.4605 0.6501 1558689 ChemDiv3_004337 C=CCn1c(=N)c(C#N)cc2c(=O)n3ccccc3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F04 compound treatment 640.0 -235.0 -0.08 920.0 360.0 0.28 0.1365 0.4728 3117763 ChemDiv3_004338 Cc1cc(nc2sc(C(=O)c3cccc(Cl)c3)c(N)c12)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F05 compound treatment 1080.0 205.0 0.07 920.0 360.0 0.28 0.2469 0.8638 3117764 ChemDiv3_004339 CCCn1c(=N)c(cc2c(=O)n3ccccc3nc12)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F06 compound treatment 1720.0 845.0 0.3 480.0 -80.0 -0.06 0.1685 0.5508 3024369 ChemDiv3_004340 Cc1cc(C)cc(Nc2cc(=O)oc3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F07 compound treatment 3880.0 3010.0 1.07 920.0 360.0 0.28 0.9492 0.8619 3024370 ChemDiv3_004341 CNS(=O)(=O)c1ccc2oc3ccc(cc3c2c1)S(=O)(=O)NC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F08 compound treatment 800.0 -75.0 -0.03 1200.0 640.0 0.49 0.3286 0.6678 3117765 ChemDiv3_004342 CCCOc1ccc(OCCSc2nc(=O)cc(N)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F09 compound treatment 3080.0 2210.0 0.78 6760.0 6200.0 4.76 3.9188 0.8124 3117766 ChemDiv3_004343 Cc1ccc(NC(=N)Nc2nc(cc(n2)C(F)(F)F)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F10 compound treatment 3400.0 2530.0 0.9 1160.0 600.0 0.46 0.9591 0.9522 3024371 ChemDiv3_004344 Cc1cc(C)nc(SCc2nnc(SC/C=C/c3ccccc3)o2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F11 compound treatment 2280.0 1410.0 0.5 1520.0 960.0 0.74 0.8736 0.9819 3117767 ChemDiv3_004345 CCOc1ccc(NC(=N)Nc2nc(cc(n2)C(F)(F)F)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F12 compound treatment 1880.0 1010.0 0.36 760.0 200.0 0.15 0.3607 0.9291 3024372 ChemDiv3_004346 CCOC(=O)Cc1csc(n1)/C(=N/O)/C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F13 compound treatment 400.0 -475.0 -0.17 1000.0 440.0 0.34 0.1197 0.3171 3117768 ChemDiv3_004347 COC(=O)c1c(F)c(F)c(Oc2ccc(Cl)cc2)c(F)c1N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F14 compound treatment 1040.0 165.0 0.06 600.0 40.0 0.03 0.0631 0.9547 1296118 ChemDiv3_004348 CC(Nc1nc2nonc2nc1NC(C)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F15 compound treatment 920.0 45.0 0.02 4840.0 4280.0 3.29 2.3347 0.7105 3024373 ChemDiv3_004349 Clc1ccccc1C(=O)Oc2ccccc2/C=C\3/N=C4CCCCCN4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F16 compound treatment 3920.0 3050.0 1.08 1440.0 880.0 0.68 1.2415 0.9745 3117910 ChemDiv3_004350 O=C/1ON=C(\C1=C/c2ccc3OCOc3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F17 compound treatment 3440.0 2570.0 0.91 920.0 360.0 0.28 0.8388 0.8821 1675128 ChemDiv3_004351 CC1=C(C(c2ccncc2)n3ncnc3N1)C(=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F18 compound treatment 17120.0 16200.0 5.76 8840.0 8280.0 6.36 8.5698 0.9988 3117911 ChemDiv3_004352 COc1cc(/C=C/2\C(=NOC2=O)C)cc(Cl)c1OCc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F19 compound treatment 520.0 -355.0 -0.13 2640.0 2080.0 1.6 1.0401 0.6493 3117912 ChemDiv3_004353 CC(C)CNS(=O)(=O)c1ccccc1C(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F20 compound treatment 760.0 -115.0 -0.04 840.0 280.0 0.21 0.1232 0.5629 3024374 ChemDiv3_004354 S=C(NCCC1=CCCCC1)Nc2ccc3nsnc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F21 compound treatment 1560.0 685.0 0.24 800.0 240.0 0.18 0.3021 0.9907 1516017 ChemDiv3_004355 Clc1ccc(CN2C(=O)c3ccccc3S2(=O)=O)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F22 compound treatment 1000.0 125.0 0.04 2080.0 1520.0 1.17 0.8565 0.7334 3024375 ChemDiv3_004356 C(Sc1nnc(o1)c2cccnc2)/C=C/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F23 mock treatment 5000.0 4130.0 1.46 5360.0 4800.0 3.69 3.6405 0.9182 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 F24 mock treatment 760.0 -115.0 -0.04 1760.0 1200.0 0.92 0.6226 0.6751 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G01 compound treatment 560.0 -315.0 -0.11 1080.0 520.0 0.4 0.2033 0.4903 1561444 ChemDiv3_004357 COC(=O)C1=C(C)NC2=C(C1c3ccc(OC)cc3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G02 compound treatment 760.0 -115.0 -0.04 640.0 80.0 0.06 0.0146 0.1978 3024376 ChemDiv3_004358 Cc1ccc2cc(C3CC(=NN3S(=O)(=O)C)c4ccco4)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G03 compound treatment 1240.0 365.0 0.13 520.0 -40.0 -0.03 0.0698 0.5248 3117913 ChemDiv3_004359 COc1ccccc1NC(=O)C(NC(=O)c2ccccc2NC(=O)c3ccccc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G04 compound treatment 360.0 -515.0 -0.18 1160.0 600.0 0.46 0.1965 0.3966 1365443 ChemDiv3_004360 Cc1ccc(cc1)S(=O)(=O)NCC(O)Cn2c3ccccc3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G05 compound treatment 1200.0 325.0 0.12 600.0 40.0 0.03 0.1032 0.8653 1229059 ChemDiv3_004361 CCOC(=O)c1cn(CC)c2cc(F)c(F)cc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G06 compound treatment 760.0 -115.0 -0.04 1200.0 640.0 0.49 0.3186 0.6462 3117914 ChemDiv3_004362 CC(=O)N1CN(Cc2ccccc2)Cc3c4CCCCc4sc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G07 compound treatment 600.0 -275.0 -0.1 840.0 280.0 0.21 0.083 0.3517 3024377 ChemDiv3_004363 Clc1ccc(Sc2c(nc3ncccn23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G08 compound treatment 800.0 -75.0 -0.03 720.0 160.0 0.12 0.068 0.5414 3117915 ChemDiv3_004364 CCCc1cc(N2CCN(CC2)c3ccccc3)n4c5ccccc5nc4c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G09 compound treatment 920.0 45.0 0.02 520.0 -40.0 -0.03 -0.0104 -0.3013 3024378 ChemDiv3_004365 COc1ccc(NC(=O)CSc2nc(O)cc(=O)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G10 compound treatment 560.0 -315.0 -0.11 520.0 -40.0 -0.03 -0.1007 -0.8692 3024435 ChemDiv3_004366 Clc1ccc(Cn2cccc2/C=C\3/C(=N)N4C=CSC4=NC3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G11 compound treatment 1160.0 285.0 0.1 360.0 -200.0 -0.15 -0.0371 -0.2017 1393315 ChemDiv3_004367 COc1ccc(NC(=O)N2c3ccccc3Sc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G12 compound treatment 760.0 -115.0 -0.04 400.0 -160.0 -0.12 -0.1157 -0.8939 3024436 ChemDiv3_004368 N(=c/1\oc2ccccc2cc1c3nc4ccccc4[nH]3)\c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G13 compound treatment 240.0 -635.0 -0.23 360.0 -200.0 -0.15 -0.2679 -0.9825 3024437 ChemDiv3_004369 CCC1(C)Cc2nc3nc(SCC(=O)c4ccccc4)n(Cc5ccccc5)c(=O)c3cc2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G14 compound treatment 720.0 -155.0 -0.05 2360.0 1800.0 1.38 0.9383 0.6784 3024438 ChemDiv3_004370 Cc1cc(C(=O)OCCN2CCN(CC2)C3=NS(=O)(=O)c4ccccc34)c5ccccc5n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G15 compound treatment 840.0 -35.0 -0.01 480.0 -80.0 -0.06 -0.0522 -0.8332 1264788 ChemDiv3_004371 COc1ccc(cc1)C2C3C(ON2c4ccc(Cl)cc4)C(=O)N(C(C)C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G16 compound treatment 480.0 -395.0 -0.14 680.0 120.0 0.09 -0.0339 -0.2024 3117916 ChemDiv3_004372 CCCCC1(C)OC(=O)C(=Cc2ccc(F)cc2)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G17 compound treatment 880.0 5.0 0.0 320.0 -240.0 -0.18 -0.129 -0.7003 1307836 ChemDiv3_004373 CCCCN1COc2ccc3c4C(=O)c5ccccc5C(=O)c4oc3c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G18 compound treatment 520.0 -355.0 -0.13 400.0 -160.0 -0.12 -0.1759 -0.9999 1527245 ChemDiv3_004374 CP(=O)(Nc1ccc(Cl)cc1)Oc2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G19 compound treatment 1160.0 285.0 0.1 840.0 280.0 0.21 0.2235 0.9408 1557708 ChemDiv3_004375 CCN(CC)CCNc1nc2n(C)c(=O)n(C)c(=O)c2n1C(C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G20 compound treatment 1600.0 725.0 0.26 1960.0 1400.0 1.07 0.9419 0.8523 1285083 ChemDiv3_004376 NS(=O)(=O)c1ccc(NC(=O)CCCC(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G21 compound treatment 440.0 -435.0 -0.15 400.0 -160.0 -0.12 -0.196 -0.9936 3117917 ChemDiv3_004377 Cc1ccc(NC(=O)CC(NCCN2CCOCC2)C(=O)O)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G22 compound treatment 1000.0 125.0 0.04 400.0 -160.0 -0.12 -0.0555 -0.425 1782201 ChemDiv3_004378 N#CSCc1nc2ccccc2c3nc4ccccc4n13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G23 mock treatment 480.0 -395.0 -0.14 520.0 -40.0 -0.03 -0.1208 -0.8421 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 G24 mock treatment 680.0 -195.0 -0.07 1000.0 440.0 0.34 0.1899 0.5509 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H01 compound treatment 680.0 -195.0 -0.07 600.0 40.0 0.03 -0.0272 -0.3594 3117918 ChemDiv3_004379 CCOC(=O)C1=C(C)N=C(NC1c2ccc(OCC)cc2)SCc3ccc(cc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H02 compound treatment 1440.0 565.0 0.2 320.0 -240.0 -0.18 0.0114 0.042 3024439 ChemDiv3_004380 CCOC(=O)/C(=C\1/C=CN(C)C=N1)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H03 compound treatment 760.0 -115.0 -0.04 600.0 40.0 0.03 -0.0071 -0.1397 3117919 ChemDiv3_004381 Cc1ccc2nc3n(Cc4cccnc4)c(=N)c(cc3c(=O)n2c1)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H04 compound treatment 360.0 -515.0 -0.18 560.0 0.0 0.0 -0.1292 -0.7071 3024440 ChemDiv3_004382 NC(=O)COc1cccc(/C=C/2\CC/C(=C/c3cccc(OCC(=O)N)c3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H05 compound treatment 480.0 -395.0 -0.14 360.0 -200.0 -0.15 -0.2077 -0.999 3117920 ChemDiv3_004383 N=c1c(C#N)cc2c(=O)n3ccccc3nc2n1C4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H06 compound treatment 520.0 -355.0 -0.13 560.0 0.0 0.0 -0.089 -0.7071 1915671 ChemDiv3_004384 N1C(=CC(c2ccccc2)n3c1nc4ccccc34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H07 compound treatment 1320.0 445.0 0.16 760.0 200.0 0.15 0.2202 0.9999 3024441 ChemDiv3_004385 CC1(C)OC(=O)C=C(O1)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H08 compound treatment 520.0 -355.0 -0.13 7160.0 6600.0 5.07 3.4938 0.6893 1820724 ChemDiv3_004386 Nc1cc(N)nc(SCC(=O)N2c3ccccc3Sc4ccccc24)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H09 compound treatment 1560.0 685.0 0.24 480.0 -80.0 -0.06 0.1284 0.5123 3117921 ChemDiv3_004387 CN(C)c1ccc(NC(=N)Nc2nc(cc(n2)C(F)(F)F)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H10 compound treatment 360.0 -515.0 -0.18 520.0 -40.0 -0.03 -0.1509 -0.8145 3024442 ChemDiv3_004388 Cc1cc(C)nc(SCc2nnc(SCC(=O)NCc3ccccc3)o2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H11 compound treatment 480.0 -395.0 -0.14 520.0 -40.0 -0.03 -0.1208 -0.8421 3117922 ChemDiv3_004389 Cc1ccccc1NC2=NC(=NC3(CCCCC3)N2)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H12 compound treatment 440.0 -435.0 -0.15 560.0 0.0 0.0 -0.1091 -0.7071 1869886 ChemDiv3_004390 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(=O)CCN2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H13 compound treatment 520.0 -355.0 -0.13 520.0 -40.0 -0.03 -0.1108 -0.8545 3117923 ChemDiv3_004391 Cc1onc(c1C(=O)NC(=S)NC2CCSC2=O)c3c(F)cccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H14 compound treatment 440.0 -435.0 -0.15 720.0 160.0 0.12 -0.0223 -0.1129 1513000 ChemDiv3_004392 O=c1nc(Nc2ccc3ccccc3c2)nc([nH]1)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H15 compound treatment 1440.0 565.0 0.2 840.0 280.0 0.21 0.2937 0.9994 1396416 ChemDiv3_004393 Cc1cc(NC(=O)CSc2ccc(C)cc2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H16 compound treatment 1400.0 525.0 0.19 440.0 -120.0 -0.09 0.0665 0.3203 3117924 ChemDiv3_004394 Cc1cc(Cl)ccc1NS(=O)(=O)c2ccc3N[C@@H]([C@@H]4CC=C[C@@H]4c3c2)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H17 compound treatment 2280.0 1410.0 0.5 680.0 120.0 0.09 0.4176 0.8239 3024443 ChemDiv3_004395 CC/1=CC(=O)C=C\C1=N\C(=N/S(=O)(=O)c2ccc(C)cc2)\c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H18 compound treatment 2080.0 1210.0 0.43 1720.0 1160.0 0.89 0.932 0.9435 3117925 ChemDiv3_004396 CCOc1cc(/C=C/2\C(=NOC2=O)C)cc(Cl)c1OCc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H19 compound treatment 440.0 -435.0 -0.15 440.0 -120.0 -0.09 -0.1743 -0.9696 3024444 ChemDiv3_004397 O=C(N1CCCC1)c2ccccc2S(=O)(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H20 compound treatment 520.0 -355.0 -0.13 1040.0 480.0 0.37 0.1715 0.4404 3117926 ChemDiv3_004398 C=CCn1cc(/C=C\2/NC(=O)N(C2=O)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H21 compound treatment 680.0 -195.0 -0.07 440.0 -120.0 -0.09 -0.1141 -0.99 3024445 ChemDiv3_004399 CCOc1ccc(cc1)C2=NCCNC3=C2C(N(C3=O)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H22 compound treatment 5480.0 4610.0 1.63 1160.0 600.0 0.46 1.4808 0.8725 1672517 ChemDiv3_004400 O=C(Cc1c[nH]c2ccccc12)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H23 mock treatment 440.0 -435.0 -0.15 920.0 360.0 0.28 0.0863 0.2727 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 H24 mock treatment 520.0 -355.0 -0.13 1400.0 840.0 0.64 0.367 0.5585 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I01 compound treatment 240.0 -635.0 -0.23 3600.0 3040.0 2.33 1.491 0.6359 3117927 ChemDiv3_004401 CCC1(CN2CC3(CC)CN(C1)C(=O)c4ccccc4C2=O)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I02 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 3024446 ChemDiv3_004402 FC(F)(F)C1(NC(=O)N2CCCN=C2S1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I03 compound treatment 360.0 -515.0 -0.18 400.0 -160.0 -0.12 -0.216 -0.9813 3117928 ChemDiv3_004403 Cc1csc(/C=C/2\CCc3c(cnc4ccc5ccccc5c34)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I04 compound treatment 280.0 -595.0 -0.21 360.0 -200.0 -0.15 -0.2578 -0.9878 3024447 ChemDiv3_004404 Cc1cc2nnc(SCc3ccc(Cl)cc3)n2c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I05 compound treatment 320.0 -555.0 -0.2 4360.0 3800.0 2.92 1.9236 0.6579 1803276 ChemDiv3_004405 CCC(Sc1nc2CCCCCc2cc1C#N)C(=O)Nc3cc(C)on3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I06 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 3118072 ChemDiv3_004406 CC(=O)Nc1sc2CCCCc2c1CN3CCN(CC3)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I07 compound treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 3024448 ChemDiv3_004407 FC(F)(F)c1cc(nc2c(cnn12)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I08 compound treatment 520.0 -355.0 -0.13 520.0 -40.0 -0.03 -0.1108 -0.8545 3118073 ChemDiv3_004408 CCCc1cc(NC(C)c2ccccc2)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I09 compound treatment 280.0 -595.0 -0.21 1160.0 600.0 0.46 0.1765 0.3483 3024449 ChemDiv3_004409 Cc1cc(C)c(c(C)c1)S(=O)(=O)/N=C/2\SCCN2S(=O)(=O)c3c(C)cc(C)cc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I10 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3118074 ChemDiv3_004410 CCCc1nn(c(O)c1/C(=N/c2ccc(cc2)C(=O)OCC)/C)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I11 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 1190406 ChemDiv3_004411 CC(C)CNC(=O)N1c2ccccc2Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I12 compound treatment 480.0 -395.0 -0.14 240.0 -320.0 -0.25 -0.2728 -0.9646 3118075 ChemDiv3_004412 COc1cc(=O)n(C)c2cc(ccc12)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I13 compound treatment 360.0 -515.0 -0.18 240.0 -320.0 -0.25 -0.3029 -0.9894 3024450 ChemDiv3_004413 CSc1nc(C)cc(OCCO)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I14 compound treatment 440.0 -435.0 -0.15 480.0 -80.0 -0.06 -0.1525 -0.9185 3118076 ChemDiv3_004414 Clc1cc(/C=C\2/C(=N)N3C=CSC3=NC2=O)ccc1OCCOc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I15 compound treatment 4120.0 3250.0 1.15 320.0 -240.0 -0.18 0.6837 0.5865 1567868 ChemDiv3_004415 Cc1ccc2[nH]c(SCc3nc4cccc(C)n4c3Br)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I16 compound treatment 400.0 -475.0 -0.17 280.0 -280.0 -0.21 -0.2712 -0.9927 3118077 ChemDiv3_004416 CCOC(=O)N1C(=O)c2ccccc2NC1(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I17 compound treatment 440.0 -435.0 -0.15 320.0 -240.0 -0.18 -0.2394 -0.9961 1709676 ChemDiv3_004417 O=C1N(CN2CCc3ccccc3C2)c4cccc5cccc1c45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I18 compound treatment 560.0 -315.0 -0.11 320.0 -240.0 -0.18 -0.2093 -0.9713 3024451 ChemDiv3_004418 Cc1onc(c1C(=O)OC(c2ccccc2)C(F)(F)F)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I19 compound treatment 280.0 -595.0 -0.21 360.0 -200.0 -0.15 -0.2578 -0.9878 3118078 ChemDiv3_004419 Cc1ccc2sc(nc2c1)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I20 compound treatment 280.0 -595.0 -0.21 680.0 120.0 0.09 -0.0841 -0.3652 3024452 ChemDiv3_004420 CCCCn1c2ccccc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I21 compound treatment 200.0 -675.0 -0.24 240.0 -320.0 -0.25 -0.343 -0.9999 1873833 ChemDiv3_004421 Cc1cccc(NC2=C(C(=O)c3ccccc3C2=O)n4nnc5ccccc45)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I22 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3024453 ChemDiv3_004422 COc1nc(c2ccccc2Cl)c3cc(Br)ccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I23 mock treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 I24 mock treatment 200.0 -675.0 -0.24 320.0 -240.0 -0.18 -0.2996 -0.9916 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J01 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3118079 ChemDiv3_004423 CN(C)c1ccc(cc1)C2NC(=S)NC(=C2C(=O)Nc3cc(C)ccc3C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J02 compound treatment 240.0 -635.0 -0.23 240.0 -320.0 -0.25 -0.333 -0.9991 3024454 ChemDiv3_004424 C[N+]1(CCn2ccc3ccccc23)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J03 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3118080 ChemDiv3_004425 N=c1c(cc2c(=O)n3ccccc3nc2n1Cc4cccnc4)C(=O)NC5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J04 compound treatment 400.0 -475.0 -0.17 320.0 -240.0 -0.18 -0.2494 -0.999 3118081 ChemDiv3_004426 CCOC(=O)C1=C(OC(=C(C#N)C1c2cccnc2)N)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J05 compound treatment 320.0 -555.0 -0.2 360.0 -200.0 -0.15 -0.2478 -0.9924 3024455 ChemDiv3_004427 COC(=O)C/1=C(C)N(C(C)C)C(=O)\C1=C/c2ccc(cc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J06 compound treatment 160.0 -715.0 -0.25 400.0 -160.0 -0.12 -0.2662 -0.9446 1162906 ChemDiv3_004428 COc1cc2c(cc1NC(=O)c3ccccc3)oc4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J07 compound treatment 200.0 -675.0 -0.24 1520.0 960.0 0.74 0.3518 0.454 3024456 ChemDiv3_004429 COc1ccc(cc1)C2=CC(=O)OC3(CCCCC3)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J08 compound treatment 360.0 -515.0 -0.18 320.0 -240.0 -0.18 -0.2595 -1.0 3118082 ChemDiv3_004430 COc1ccccc1n2c(C)nc(=O)c(c2C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J09 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3024457 ChemDiv3_004431 Cc1cccc(c1)N2C(=NC(=NC32CCCCC3)N)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J10 compound treatment 440.0 -435.0 -0.15 360.0 -200.0 -0.15 -0.2177 -1.0 1868948 ChemDiv3_004432 CCSc1nc2OC(=C(C#N)C(C(C)C)c2c(=O)[nH]1)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J11 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 3118083 ChemDiv3_004433 CCOC(=O)c1cccc(NC2=NC(=NC3(CCCCC3)N2)N)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J12 compound treatment 200.0 -675.0 -0.24 400.0 -160.0 -0.12 -0.2562 -0.9519 3024458 ChemDiv3_004434 CC(=O)OC(C(=O)Nc1nc2ccccc2s1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J13 compound treatment 320.0 -555.0 -0.2 360.0 -200.0 -0.15 -0.2478 -0.9924 3118084 ChemDiv3_004435 Cc1nn(c2ccccc2)c3sc(cc13)C(=O)NC(=S)NC4CCSC4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J14 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3024459 ChemDiv3_004436 CCOC(=O)CC1(C)NNC(=S)NN1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J15 compound treatment 320.0 -555.0 -0.2 360.0 -200.0 -0.15 -0.2478 -0.9924 1554274 ChemDiv3_004437 COc1ccc(cc1)C2=NN(C(C2)c3cccc(OC)c3OC)C(=O)CSCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J16 compound treatment 320.0 -555.0 -0.2 440.0 -120.0 -0.09 -0.2044 -0.9401 3024460 ChemDiv3_004438 COc1cccc([C@H]2Nc3ccc(cc3[C@H]4C=CC[C@H]42)S(=O)(=O)Nc5ccc(C)c(C)c5)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J17 compound treatment 320.0 -555.0 -0.2 360.0 -200.0 -0.15 -0.2478 -0.9924 1189392 ChemDiv3_004439 COc1ccc(cc1OC)C(O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J18 compound treatment 520.0 -355.0 -0.13 360.0 -200.0 -0.15 -0.1976 -0.9952 3118085 ChemDiv3_004440 Cc1ccc(cc1)c2ccc(CCC(=O)O)n2c3cc(C)cc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J19 compound treatment 200.0 -675.0 -0.24 280.0 -280.0 -0.21 -0.3213 -0.9986 3024461 ChemDiv3_004441 CCn1cnc2cc(NS(=O)(=O)c3ccc(C)cc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J20 compound treatment 200.0 -675.0 -0.24 520.0 -40.0 -0.03 -0.191 -0.7913 1913074 ChemDiv3_004442 CC(C)C/C(=N\O)/c1cn(C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J21 compound treatment 640.0 -235.0 -0.08 920.0 360.0 0.28 0.1365 0.4728 3118086 ChemDiv3_004443 OC1=C(C(OC1=O)c2ccc(Cl)cc2)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J22 compound treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 1565919 ChemDiv3_004444 Cc1oc2c(C)c3oc(=O)c4CCCCc4c3cc2c1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J23 mock treatment 720.0 -155.0 -0.05 480.0 -80.0 -0.06 -0.0823 -0.9985 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 J24 mock treatment 3160.0 2290.0 0.81 4120.0 3560.0 2.73 2.5058 0.879 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K01 compound treatment 3280.0 2410.0 0.85 360.0 -200.0 -0.15 0.4947 0.5707 3024519 ChemDiv3_004445 CCNc1nc(NC(C)C)nc(Oc2ccc(/C=N/O)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K02 compound treatment 440.0 -435.0 -0.15 360.0 -200.0 -0.15 -0.2177 -1.0 3024520 ChemDiv3_004446 COc1ccc2N3C(=NC(NC3=O)(c4ccccc4)C(F)(F)F)Sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K03 compound treatment 720.0 -155.0 -0.05 400.0 -160.0 -0.12 -0.1257 -0.9343 3024521 ChemDiv3_004447 COC(=O)CCC(=O)C1=C(CC(C)(C)CC1=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K04 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 3024522 ChemDiv3_004448 Cc1nn(c(O)c1Sc2ccc(Cl)cc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K05 compound treatment 360.0 -515.0 -0.18 320.0 -240.0 -0.18 -0.2595 -1.0 1868645 ChemDiv3_004449 CCc1ccc(cc1)c2csc(Nc3ccc(cc3)S(=O)(=O)Nc4cc(OC)nc(OC)n4)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K06 compound treatment 520.0 -355.0 -0.13 720.0 160.0 0.12 -0.0022 -0.0125 3024523 ChemDiv3_004450 Cc1sc(NC(=O)c2ccco2)c(C(N3CCCC3)c4cccnc4)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K07 compound treatment 360.0 -515.0 -0.18 3000.0 2440.0 1.87 1.1954 0.6351 3118087 ChemDiv3_004451 COC(=O)C1=CN(CCc2ccc(F)cc2)C=C(C1c3ccccc3C(F)(F)F)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K08 compound treatment 640.0 -235.0 -0.08 640.0 80.0 0.06 -0.0155 -0.1499 1873196 ChemDiv3_004452 CC(C)c1cc(NC2CCCCC2)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K09 compound treatment 800.0 -75.0 -0.03 440.0 -120.0 -0.09 -0.084 -0.8755 3118088 ChemDiv3_004453 CC1=CCC(COC(=O)Nc2ccccc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K10 compound treatment 5720.0 4850.0 1.72 1560.0 1000.0 0.77 1.7582 0.934 1871904 ChemDiv3_004454 COC(=O)CSc1c(c2ccccc2)c3cc(Cl)ccc3[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K11 compound treatment 680.0 -195.0 -0.07 280.0 -280.0 -0.21 -0.2009 -0.8897 1712836 ChemDiv3_004455 CCC(C)NC(=O)N1c2ccccc2Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K12 compound treatment 2240.0 1370.0 0.48 1040.0 480.0 0.37 0.603 0.9909 1183223 ChemDiv3_004456 O=C(CNC(=O)C1CCCCC1)Nc2nc(CC3(CC4CC5CC(C4)C3)C5)cs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K13 compound treatment 440.0 -435.0 -0.15 400.0 -160.0 -0.12 -0.196 -0.9936 3024524 ChemDiv3_004457 CC(C)Oc1ccc(CNCCC(c2ccco2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K14 compound treatment 520.0 -355.0 -0.13 680.0 120.0 0.09 -0.0239 -0.1532 3118089 ChemDiv3_004458 Cc1ccc(COc2ccc(/C=C\3/C(=N)N4C=CSC4=NC3=O)cc2Br)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K15 compound treatment 400.0 -475.0 -0.17 5240.0 4680.0 3.59 2.4214 0.6732 1204806 ChemDiv3_004459 Cc1nn(c2ccccc2)c3sc(cc13)C(=O)OCN4C(=O)c5ccccc5C4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K16 compound treatment 1080.0 205.0 0.07 560.0 0.0 0.0 0.0514 0.7071 3118090 ChemDiv3_004460 NC1=C(C#N)C(C2=C(CCC2)N1c3ccc(cc3)S(=O)(=O)N)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K17 compound treatment 400.0 -475.0 -0.17 3400.0 2840.0 2.18 1.4226 0.6505 1453567 ChemDiv3_004461 CCSc1nc2NC(=C(C(c3ccncc3)c2c(=O)[nH]1)C(=O)OC)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K18 compound treatment 880.0 5.0 0.0 400.0 -160.0 -0.12 -0.0856 -0.6968 1234228 ChemDiv3_004462 CC1CN(CC(C)O1)C(=O)NC(C)(C)c2cccc(c2)C(=C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K19 compound treatment 440.0 -435.0 -0.15 400.0 -160.0 -0.12 -0.196 -0.9936 1601073 ChemDiv3_004463 CCc1ccc(cc1)S(=O)(=O)Nc2ccc3oc(=O)sc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K20 compound treatment 680.0 -195.0 -0.07 1160.0 600.0 0.46 0.2768 0.5943 1200402 ChemDiv3_004464 CCOC(=O)Cc1c(c2ccccc2)c3cc(Cl)ccc3[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K21 compound treatment 480.0 -395.0 -0.14 400.0 -160.0 -0.12 -0.1859 -0.9978 1869882 ChemDiv3_004465 CCOc1ccc2n(CO)c(=S)n(CO)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K22 compound treatment 2040.0 1170.0 0.41 280.0 -280.0 -0.21 0.1402 0.301 3024525 ChemDiv3_004466 Cc1cccc(OCC(=O)OC2CN3CCC2CC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K23 mock treatment 5200.0 4330.0 1.53 440.0 -120.0 -0.09 1.0198 0.6635 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 K24 mock treatment 440.0 -435.0 -0.15 1040.0 480.0 0.37 0.1515 0.3791 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L01 compound treatment 440.0 -435.0 -0.15 640.0 80.0 0.06 -0.0657 -0.3955 1875198 ChemDiv3_004467 CCOC(=O)c1cc2c(=O)n3cc(C)ccc3nc2n(Cc4ccco4)c1=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L02 compound treatment 480.0 -395.0 -0.14 440.0 -120.0 -0.09 -0.1642 -0.9793 3024526 ChemDiv3_004468 CC(N)Cc1c[nH]c2ccc(C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L03 compound treatment 400.0 -475.0 -0.17 520.0 -40.0 -0.03 -0.1409 -0.8224 3118218 ChemDiv3_004469 CN1CCN(CC1)C(=O)c2cc3c(=O)n4cccc(C)c4nc3n(Cc5cccnc5)c2=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L04 compound treatment 440.0 -435.0 -0.15 560.0 0.0 0.0 -0.1091 -0.7071 3118219 ChemDiv3_004470 CN1CCc2nc(SCC(=O)Nc3ccccc3OC(F)(F)F)c(C#N)cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L05 compound treatment 600.0 -275.0 -0.1 720.0 160.0 0.12 0.0179 0.114 3024527 ChemDiv3_004471 COC(=O)C/1=C(C)N(C(C)c2ccccc2)C(=O)\C1=C/c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L06 compound treatment 440.0 -435.0 -0.15 360.0 -200.0 -0.15 -0.2177 -1.0 1604904 ChemDiv3_004472 COC(=O)c1cn(C(=O)c2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L07 compound treatment 440.0 -435.0 -0.15 320.0 -240.0 -0.18 -0.2394 -0.9961 1406130 ChemDiv3_004473 COc1ccc(cc1)C2=CC(=O)N(C(O2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L08 compound treatment 1240.0 365.0 0.13 2040.0 1480.0 1.14 0.895 0.7826 1691728 ChemDiv3_004474 C(c1nc2ccc3nsnc3c2[nH]1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L09 compound treatment 640.0 -235.0 -0.08 360.0 -200.0 -0.15 -0.1675 -0.9588 3118220 ChemDiv3_004475 COc1ccccc1N2C(=NC(=NC32CCCCC3)N)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L10 compound treatment 680.0 -195.0 -0.07 640.0 80.0 0.06 -0.0055 -0.0593 3024528 ChemDiv3_004476 CN(C)c1nc(c2ccccc2)[n+](C)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L11 compound treatment 640.0 -235.0 -0.08 360.0 -200.0 -0.15 -0.1675 -0.9588 3118221 ChemDiv3_004477 COc1cccc(NC2=NC3(CCCC3)NC(=N2)N)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L12 compound treatment 360.0 -515.0 -0.18 2000.0 1440.0 1.11 0.6525 0.5824 3024529 ChemDiv3_004478 COC(=O)CSc1nnc2sc3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L13 compound treatment 240.0 -635.0 -0.23 360.0 -200.0 -0.15 -0.2679 -0.9825 1151035 ChemDiv3_004479 COc1ccc(CCNC(=O)CSc2nc(C)cc(C)n2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L14 compound treatment 280.0 -595.0 -0.21 960.0 400.0 0.31 0.0679 0.1822 3024530 ChemDiv3_004480 COC(=O)c1ccc2nsnc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L15 compound treatment 440.0 -435.0 -0.15 5760.0 5200.0 3.99 2.7137 0.6793 3118222 ChemDiv3_004481 COc1ccc(cc1)C2CC(=NN2C(=O)CSc3nc4ccccc4s3)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L16 compound treatment 480.0 -395.0 -0.14 440.0 -120.0 -0.09 -0.1642 -0.9793 3024531 ChemDiv3_004482 CCOC(=O)[C@@H]1Nc2ccc(cc2[C@@H]3C=CC[C@@H]31)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L17 compound treatment 440.0 -435.0 -0.15 560.0 0.0 0.0 -0.1091 -0.7071 3118223 ChemDiv3_004483 Cc1c(c2ccccc2)c3cc(C)cc4CCCn1c43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L18 compound treatment 480.0 -395.0 -0.14 640.0 80.0 0.06 -0.0557 -0.3638 3024532 ChemDiv3_004484 OC(=O)CCc1ccc(c2cccs2)n1c3ccccc3C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L19 compound treatment 520.0 -355.0 -0.13 600.0 40.0 0.03 -0.0673 -0.5195 3118224 ChemDiv3_004485 CCCCn1c(=N)n(CC(O)COc2ccc(OC)cc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L20 compound treatment 320.0 -555.0 -0.2 4920.0 4360.0 3.35 2.2276 0.6644 3024533 ChemDiv3_004486 C(Sc1nc2ccccc2n1Cc3ccccn3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L21 compound treatment 1560.0 685.0 0.24 480.0 -80.0 -0.06 0.1284 0.5123 3118225 ChemDiv3_004487 Brc1ccc(cc1)C(=O)/C=C\2/NCCNC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L22 compound treatment 360.0 -515.0 -0.18 360.0 -200.0 -0.15 -0.2378 -0.9963 1635205 ChemDiv3_004488 CCCc1cc(=O)oc2cc3occ(c4ccccc4)c3cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L23 mock treatment 560.0 -315.0 -0.11 440.0 -120.0 -0.09 -0.1442 -0.9954 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 L24 mock treatment 480.0 -395.0 -0.14 440.0 -120.0 -0.09 -0.1642 -0.9793 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M01 compound treatment 280.0 -595.0 -0.21 360.0 -200.0 -0.15 -0.2578 -0.9878 3024534 ChemDiv3_004489 COc1nc(Oc2ccc(/C=N/O)cc2)nc(n1)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M02 compound treatment 640.0 -235.0 -0.08 760.0 200.0 0.15 0.0496 0.284 3118226 ChemDiv3_004490 O=C(Oc1nsnc1N2CCCCC2)N(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M03 compound treatment 1400.0 525.0 0.19 320.0 -240.0 -0.18 0.0014 0.0054 3024535 ChemDiv3_004491 CCOC(=O)Nc1nc2ccc(C)cc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M04 compound treatment 1600.0 725.0 0.26 280.0 -280.0 -0.21 0.0299 0.0891 3118227 ChemDiv3_004492 Cc1nn(c(O)c1Sc2ccc(C)cc2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M05 compound treatment 960.0 85.0 0.03 2360.0 1800.0 1.38 0.9985 0.7224 1868767 ChemDiv3_004493 COc1ccc(cc1C)c2csc(Nc3ccc(cc3)S(=O)(=O)Nc4cc(C)on4)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M06 compound treatment 2400.0 1530.0 0.54 440.0 -120.0 -0.09 0.3174 0.5784 3024536 ChemDiv3_004494 O=C1CC(SC(=N1)N(c2ccccc2)c3ccccc3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M07 compound treatment 440.0 -435.0 -0.15 680.0 120.0 0.09 -0.044 -0.2447 3118228 ChemDiv3_004495 COC(=O)C1=CN(Cc2cccs2)C=C(C1c3cccc(OC)c3)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M08 compound treatment 240.0 -635.0 -0.23 560.0 0.0 0.0 -0.1593 -0.7071 3024537 ChemDiv3_004496 CC(C)CCNc1cc(C(C)C)c(C#N)c2nc3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M09 compound treatment 320.0 -555.0 -0.2 440.0 -120.0 -0.09 -0.2044 -0.9401 3118229 ChemDiv3_004497 COC(=O)c1cc(c(Cl)cc1Cl)S(=O)(=O)/C=C/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M10 compound treatment 3280.0 2410.0 0.85 320.0 -240.0 -0.18 0.473 0.5419 3024538 ChemDiv3_004498 CCOC(=O)Cc1cc(O)n(n1)c2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M11 compound treatment 320.0 -555.0 -0.2 680.0 120.0 0.09 -0.0741 -0.3408 1623227 ChemDiv3_004499 O=C(NCc1ccccc1)N2c3ccccc3Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M12 compound treatment 320.0 -555.0 -0.2 2600.0 2040.0 1.57 0.9682 0.6134 1497208 ChemDiv3_004500 O=C(CNC(=O)COc1ccccc1)Nc2nc(CC3(CC4CC5CC(C4)C3)C5)cs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M13 compound treatment 520.0 -355.0 -0.13 360.0 -200.0 -0.15 -0.1976 -0.9952 1480171 ChemDiv3_004501 C=CCSc1nc2-c3ccccc3CC4(CCCCC4)c2c(=O)n1Cc5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M14 compound treatment 880.0 5.0 0.0 360.0 -200.0 -0.15 -0.1073 -0.6989 3024539 ChemDiv3_004502 CN(C)c1ccc(cc1)n2cccc2/C=N/n3cnnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M15 compound treatment 240.0 -635.0 -0.23 1080.0 520.0 0.4 0.123 0.2683 1730629 ChemDiv3_004503 O=C(OCn1nnc2ccccc2c1=O)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M16 compound treatment 640.0 -235.0 -0.08 360.0 -200.0 -0.15 -0.1675 -0.9588 3118230 ChemDiv3_004504 FC(F)(F)C(NCc1ccccc1Cl)(NC(=O)c2ccccc2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M17 compound treatment 600.0 -275.0 -0.1 480.0 -80.0 -0.06 -0.1124 -0.9751 1482041 ChemDiv3_004505 CCc1ccc(cc1)C2C3=C(CCCC3=O)Nc4c2c(=O)n(C)c(=O)n4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M18 compound treatment 3080.0 2210.0 0.78 2040.0 1480.0 1.14 1.3565 0.9834 1232456 ChemDiv3_004506 COc1ccccc1OCc2nc3ccccc3n2CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M19 compound treatment 640.0 -235.0 -0.08 880.0 320.0 0.25 0.1148 0.4424 3024540 ChemDiv3_004507 CC1=NN2C(=NNC2(C)c3ccccc3)NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M20 compound treatment 920.0 45.0 0.02 640.0 80.0 0.06 0.0547 0.8622 3118231 ChemDiv3_004508 Clc1ccc2[nH]c(=O)c(c(c3ccccc3)c2c1)[n+]4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M21 compound treatment 320.0 -555.0 -0.2 4120.0 3560.0 2.73 1.7934 0.6545 3118232 ChemDiv3_004509 Cc1cccc(C)c1NC2OC(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M22 compound treatment 840.0 -35.0 -0.01 280.0 -280.0 -0.21 -0.1608 -0.7467 3024541 ChemDiv3_004510 COC(=O)c1ccccc1Oc2c(F)c(F)nc(N3CCOCC3)c2F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M23 mock treatment 1200.0 325.0 0.12 800.0 240.0 0.18 0.2118 0.9745 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 M24 mock treatment 760.0 -115.0 -0.04 320.0 -240.0 -0.18 -0.1591 -0.8432 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N01 compound treatment 1560.0 685.0 0.24 400.0 -160.0 -0.12 0.085 0.3121 3118233 ChemDiv3_004511 Cc1cccn2c(=O)c3cc(C(=O)NCC=C)c(=N)n(CC4CCCO4)c3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N02 compound treatment 1320.0 445.0 0.16 440.0 -120.0 -0.09 0.0465 0.2543 3118234 ChemDiv3_004512 CCC1CCc2nc3sc(C(=O)Nc4ccccc4C(F)(F)F)c(N)c3cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N03 compound treatment 360.0 -515.0 -0.18 2040.0 1480.0 1.14 0.6742 0.5859 1874938 ChemDiv3_004513 N=c1c(cc2c(=O)n3ccccc3nc2n1CCCN4CCOCC4)C(=O)NCC5CCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N04 compound treatment 560.0 -315.0 -0.11 640.0 80.0 0.06 -0.0356 -0.2791 3118235 ChemDiv3_004514 CCN(CC)c1ccc(NC(=O)c2cc(=O)c3ccccc3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N05 compound treatment 800.0 -75.0 -0.03 240.0 -320.0 -0.25 -0.1925 -0.7791 3118369 ChemDiv3_004515 COc1cc(/C=C\2/S\C(=N\c3ccccc3)\N(CCc4ccccc4)C2=O)ccc1OCC(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N06 compound treatment 520.0 -355.0 -0.13 880.0 320.0 0.25 0.0847 0.3067 3024542 ChemDiv3_004516 CN1CCN(CC1)C(=S)c2cn(Cc3ccc(F)cc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N07 compound treatment 4240.0 3370.0 1.19 440.0 -120.0 -0.09 0.7789 0.6506 3118370 ChemDiv3_004517 CC(Oc1ccc(Cl)cc1Cl)C(=O)Nc2nc3CC(C)(C)CC(=O)c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N08 compound treatment 400.0 -475.0 -0.17 360.0 -200.0 -0.15 -0.2277 -0.9989 3024543 ChemDiv3_004518 CCOC(=O)Cn1c(=N)n(Cc2ccc(Cl)c(Cl)c2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N09 compound treatment 480.0 -395.0 -0.14 440.0 -120.0 -0.09 -0.1642 -0.9793 3024544 ChemDiv3_004519 CC1(C)N=C(N)N=C(N)N1c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N10 compound treatment 360.0 -515.0 -0.18 440.0 -120.0 -0.09 -0.1943 -0.9498 3118371 ChemDiv3_004520 Clc1ccc(cc1)N2CN=C(NC2=S)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N11 compound treatment 800.0 -75.0 -0.03 1040.0 480.0 0.37 0.2418 0.6544 3118372 ChemDiv3_004521 Cn1cc(C=C2C(=O)OC3(CCCCC3)OC2=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N12 compound treatment 520.0 -355.0 -0.13 360.0 -200.0 -0.15 -0.1976 -0.9952 3024545 ChemDiv3_004522 Cc1nc2-c3ccccc3C(=O)c2c(c1C#N)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N13 compound treatment 360.0 -515.0 -0.18 440.0 -120.0 -0.09 -0.1943 -0.9498 3024607 ChemDiv3_004523 CC1Oc2ccccc2C=C1/C=C/C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N14 compound treatment 480.0 -395.0 -0.14 720.0 160.0 0.12 -0.0122 -0.0656 1284692 ChemDiv3_004524 OC(=O)c1ccc(OC2CSC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N15 compound treatment 400.0 -475.0 -0.17 560.0 0.0 0.0 -0.1192 -0.7071 1312878 ChemDiv3_004525 COc1cccc(C2CC(=NN2C(=O)CSC3CCCCC3)c4cccs4)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N16 compound treatment 360.0 -515.0 -0.18 520.0 -40.0 -0.03 -0.1509 -0.8145 3024608 ChemDiv3_004526 O=C(Oc1ccc2oc(=O)sc2c1)/C=C/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N17 compound treatment 360.0 -515.0 -0.18 440.0 -120.0 -0.09 -0.1943 -0.9498 3024609 ChemDiv3_004527 Cc1cc(C)nc(SCCS(=O)(=O)c2ccc(cc2)C(C)(C)C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N18 compound treatment 400.0 -475.0 -0.17 600.0 40.0 0.03 -0.0974 -0.5689 3024610 ChemDiv3_004528 CC(C)(C)c1cc(n2ncnc2n1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N19 compound treatment 2400.0 1530.0 0.54 440.0 -120.0 -0.09 0.3174 0.5784 3024611 ChemDiv3_004529 O=C1N=C2Nc3cc4ccccc4cc3NC=C2N1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N20 compound treatment 680.0 -195.0 -0.07 400.0 -160.0 -0.12 -0.1358 -0.9631 3024612 ChemDiv3_004530 COC(=O)CSc1nnnn1c2ccc(cc2)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N21 compound treatment 200.0 -675.0 -0.24 440.0 -120.0 -0.09 -0.2345 -0.9139 3118373 ChemDiv3_004531 CCOc1ccc(cc1)C(=O)/C=C\2/NCCNC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N22 compound treatment 280.0 -595.0 -0.21 400.0 -160.0 -0.12 -0.2361 -0.9668 1434883 ChemDiv3_004532 Fc1ccc(cc1)c2coc3cc4oc(=O)ccc4cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N23 mock treatment 640.0 -235.0 -0.08 400.0 -160.0 -0.12 -0.1458 -0.9822 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 N24 mock treatment 320.0 -555.0 -0.2 400.0 -160.0 -0.12 -0.2261 -0.9742 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O01 compound treatment 320.0 -555.0 -0.2 240.0 -320.0 -0.25 -0.3129 -0.994 3118374 ChemDiv3_004533 CCNc1nc(OC)nc(Oc2ccc(/C=N/O)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O02 compound treatment 200.0 -675.0 -0.24 320.0 -240.0 -0.18 -0.2996 -0.9916 3024613 ChemDiv3_004534 CCOc1ccccc1NC2=NC(=O)CS2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O03 compound treatment 240.0 -635.0 -0.23 240.0 -320.0 -0.25 -0.333 -0.9991 3118375 ChemDiv3_004535 COc1ccc(/C=C/C(=O)Nc2nc3ccc(cc3s2)S(=O)(=O)C)cc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O04 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 3024614 ChemDiv3_004536 Cc1ccc(cc1)n2cc(c3ccccc3)c4c(O)ncnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O05 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 1788936 ChemDiv3_004537 COc1ccc(OCCn2c(NC(=O)c3ccccc3Cl)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O06 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 1873162 ChemDiv3_004538 CCC(C)Nc1cc(C)c(C#N)c2nc3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O07 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 3118376 ChemDiv3_004539 CCOC(=O)c1sc(C)c2c(=O)[nH]c(nc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O08 compound treatment 240.0 -635.0 -0.23 200.0 -360.0 -0.28 -0.3547 -0.9948 3118377 ChemDiv3_004540 CC(C)c1cc(NC(C)c2ccccc2)n3c4ccccc4nc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O09 compound treatment 320.0 -555.0 -0.2 440.0 -120.0 -0.09 -0.2044 -0.9401 3024615 ChemDiv3_004541 COC(=O)c1ccc(CN2C(=O)/C(=N\O)/c3ccccc23)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O10 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 3118378 ChemDiv3_004542 COC(=O)c1ccc(cc1)C2N(C(=O)C(C)C)c3ccccc3NC4=C2C(=O)CC(C)(C)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O11 compound treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 1579211 ChemDiv3_004543 OCCNC(=O)N1c2ccccc2Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O12 compound treatment 360.0 -515.0 -0.18 240.0 -320.0 -0.25 -0.3029 -0.9894 3024616 ChemDiv3_004544 CCOC(=O)c1cc(c2nnc(o2)c3cccc(C)c3)c(C)nc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O13 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 3118379 ChemDiv3_004545 COC(=O)CCc1c(C)[nH]c(=S)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O14 compound treatment 320.0 -555.0 -0.2 240.0 -320.0 -0.25 -0.3129 -0.994 3118380 ChemDiv3_004546 OC(=O)COc1ccccc1C=C2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O15 compound treatment 320.0 -555.0 -0.2 200.0 -360.0 -0.28 -0.3346 -0.9862 1605579 ChemDiv3_004547 Cc1nn(c2ccccc2)c3sc(cc13)C(=O)N(Cc4ccccc4)Cc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O16 compound treatment 360.0 -515.0 -0.18 280.0 -280.0 -0.21 -0.2812 -0.9967 3118381 ChemDiv3_004548 COC(NC(=O)Nc1nc2ccccc2s1)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O17 compound treatment 360.0 -515.0 -0.18 240.0 -320.0 -0.25 -0.3029 -0.9894 3118382 ChemDiv3_004549 S(c1nnc([nH]1)c2ccccc2)c3ncnc4n(ncc34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O18 compound treatment 120.0 -755.0 -0.27 360.0 -200.0 -0.15 -0.298 -0.9651 1189918 ChemDiv3_004550 CCCc1nc2ccccc2n1CC(=O)N(COCC)c3c(C)cccc3CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O19 compound treatment 240.0 -635.0 -0.23 240.0 -320.0 -0.25 -0.333 -0.9991 1251160 ChemDiv3_004551 COc1ccc(cc1)C(=O)N2CCc3cc(OC)c(OC)cc3C2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O20 compound treatment 280.0 -595.0 -0.21 320.0 -240.0 -0.18 -0.2795 -0.9977 1160379 ChemDiv3_004552 Cc1ccc(NC(=O)CNS(=O)(=O)c2ccccc2)c(c1)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O21 compound treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 3118383 ChemDiv3_004553 Cc1ccc(cc1C)c2csc(NC3OC(=O)c4ccccc34)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O22 compound treatment 280.0 -595.0 -0.21 360.0 -200.0 -0.15 -0.2578 -0.9878 3118384 ChemDiv3_004554 CCOC(=O)c1ccccc1Oc2c(F)c(F)nc(NCCO)c2F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O23 mock treatment 240.0 -635.0 -0.23 280.0 -280.0 -0.21 -0.3113 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 O24 mock treatment 800.0 -75.0 -0.03 240.0 -320.0 -0.25 -0.1925 -0.7791 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P01 compound treatment 360.0 -515.0 -0.18 240.0 -320.0 -0.25 -0.3029 -0.9894 3118385 ChemDiv3_004555 Cc1ccc2nc3n(CC4CCCO4)c(=N)c(cc3c(=O)n2c1)C(=O)NCCN5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P02 compound treatment 280.0 -595.0 -0.21 1600.0 1040.0 0.8 0.4153 0.5029 3024617 ChemDiv3_004556 CCC1CCc2nc3sc(C(=O)NC(C)c4ccccc4)c(N)c3cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P03 compound treatment 320.0 -555.0 -0.2 280.0 -280.0 -0.21 -0.2912 -0.999 3024618 ChemDiv3_004557 CCCn1c(=N)c(cc2c(=O)n3ccccc3nc12)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P04 compound treatment 320.0 -555.0 -0.2 240.0 -320.0 -0.25 -0.3129 -0.994 3118386 ChemDiv3_004558 COc1ccc(OC)c(c1)C(=O)CC2(O)C(=O)Nc3ccccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P05 compound treatment 240.0 -635.0 -0.23 400.0 -160.0 -0.12 -0.2461 -0.9593 3118387 ChemDiv3_004559 CN/1C(=O)/C(=C\c2cccc(OCC(=O)O)c2)/S\C1=N\c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P06 compound treatment 280.0 -595.0 -0.21 200.0 -360.0 -0.28 -0.3447 -0.9911 3024619 ChemDiv3_004560 CN1C(=O)/C(=C/c2ccccc2OCc3ccc(cc3)C(=O)O)/NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P07 compound treatment 200.0 -675.0 -0.24 200.0 -360.0 -0.28 -0.3647 -0.9974 3118388 ChemDiv3_004561 CC(C)C(=O)Nc1cccc(c1)C(=O)NC2CCSC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P08 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 3024620 ChemDiv3_004562 OCCn1c(=N)n(CCOc2ccc(Cl)cc2Cl)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P09 compound treatment 280.0 -595.0 -0.21 160.0 -400.0 -0.31 -0.3664 -0.9833 3118389 ChemDiv3_004563 Cc1ccc(NC2=NC(=NC(C)(C)N2)N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P10 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 1137559 ChemDiv3_004564 Clc1sc(nc1S(=O)(=O)c2ccccc2)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P11 compound treatment 280.0 -595.0 -0.21 200.0 -360.0 -0.28 -0.3447 -0.9911 3024621 ChemDiv3_004565 O=C(N1CCN(CC1)C2=NS(=O)(=O)c3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P12 compound treatment 280.0 -595.0 -0.21 200.0 -360.0 -0.28 -0.3447 -0.9911 3118390 ChemDiv3_004566 Clc1ccccc1/C=N/c2c(nc3ccccn23)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P13 compound treatment 320.0 -555.0 -0.2 240.0 -320.0 -0.25 -0.3129 -0.994 3024622 ChemDiv3_004567 COc1cc2cc(cc(c3ccc(C)cc3)c2cc1OC)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P14 compound treatment 280.0 -595.0 -0.21 680.0 120.0 0.09 -0.0841 -0.3652 3118391 ChemDiv3_004568 CC(C)c1ccc(cc1)[C@@H]2Nc3ccc(cc3[C@@H]4C=CC[C@@H]42)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P15 compound treatment 280.0 -595.0 -0.21 360.0 -200.0 -0.15 -0.2578 -0.9878 1588117 ChemDiv3_004569 COc1cccc(C2CC(=NN2C(=O)CSc3nncn3C)c4cccs4)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P16 compound treatment 240.0 -635.0 -0.23 320.0 -240.0 -0.18 -0.2896 -0.995 1691077 ChemDiv3_004570 Cc1ccc(cc1)C(=O)Oc2ccc3oc(=O)sc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P17 compound treatment 200.0 -675.0 -0.24 280.0 -280.0 -0.21 -0.3213 -0.9986 1636095 ChemDiv3_004571 CCC[N+]1(C)CCC2C(C1)c3ccccc3N2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P18 compound treatment 120.0 -755.0 -0.27 240.0 -320.0 -0.25 -0.3631 -0.9991 3024623 ChemDiv3_004572 C=CCN(CC=C)C(=S)Nc1ccc2nsnc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P19 compound treatment 240.0 -635.0 -0.23 200.0 -360.0 -0.28 -0.3547 -0.9948 3118392 ChemDiv3_004573 Cc1cn(C/C=C\c2ccccc2)c(=O)n(C/C=C/c3ccccc3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P20 compound treatment 320.0 -555.0 -0.2 320.0 -240.0 -0.18 -0.2695 -0.9995 1171466 ChemDiv3_004574 CN1C(=O)C2ON(C(C2C1=O)c3ccc(C)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P21 compound treatment 240.0 -635.0 -0.23 360.0 -200.0 -0.15 -0.2679 -0.9825 3118510 ChemDiv3_004575 CCOc1ccc(cc1)C(=O)/C=C(\O)/C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P22 compound treatment 280.0 -595.0 -0.21 280.0 -280.0 -0.21 -0.3013 -1.0 1689473 ChemDiv3_004576 COc1ccc(cc1F)c2coc3c(C)c4oc(=O)c5CCCCc5c4cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P23 mock treatment 200.0 -675.0 -0.24 240.0 -320.0 -0.25 -0.343 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2013 P24 mock treatment 280.0 -595.0 -0.21 240.0 -320.0 -0.25 -0.323 -0.9971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A01 compound treatment 360.0 -918.0 -0.33 400.0 -284.0 -0.22 -0.3842 -0.9809 1460156 ChemDiv3_004577 Cc1c(Cc2ccccc2)c(=O)oc3cc4oc5CCCCc5c4cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A02 compound treatment 400.0 -878.0 -0.31 360.0 -324.0 -0.25 -0.3959 -0.9938 3118511 ChemDiv3_004578 CCNc1nc(OCCO)nc(n1)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A03 compound treatment 320.0 -958.0 -0.34 520.0 -164.0 -0.13 -0.3291 -0.9086 1870447 ChemDiv3_004579 CCCc1cc(=O)oc2c(C)c3oc(C)c(C)c3cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A04 compound treatment 400.0 -878.0 -0.31 960.0 276.0 0.21 -0.0702 -0.1862 3118512 ChemDiv3_004580 Cc1cc(NCCNc2ccccc2)c3ccc4ccccc4c3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A05 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3024624 ChemDiv3_004581 Fc1nc(Nc2ccccc2)c3Oc4ccccc4Oc3c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A06 compound treatment 480.0 -798.0 -0.28 240.0 -444.0 -0.34 -0.4409 -0.9957 3118513 ChemDiv3_004582 C[n+]1ccc(/C=C\c2ccco2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A07 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3118514 ChemDiv3_004583 Fc1c(F)c2Oc3cc(Cl)c(Cl)cc3Oc2c(F)c1C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A08 compound treatment 720.0 -558.0 -0.2 240.0 -444.0 -0.34 -0.3807 -0.9665 3024625 ChemDiv3_004584 CCc1ccc(cc1)C2Nc3sc4CN(C)CCc4c3C(=N2)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A09 compound treatment 560.0 -718.0 -0.25 280.0 -404.0 -0.31 -0.3992 -0.9952 1316234 ChemDiv3_004585 CN(C)c1ccc(cc1)C2C=C(Nc3ncnn23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A10 compound treatment 240.0 -1040.0 -0.37 200.0 -484.0 -0.37 -0.5229 -1.0 1745023 ChemDiv3_004586 COc1ccc(cc1)C(=O)CSc2nnc(c3ccco3)c(n2)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A11 compound treatment 360.0 -918.0 -0.33 320.0 -364.0 -0.28 -0.4276 -0.9971 1655325 ChemDiv3_004587 OC(=O)c1cc(NC(=O)CSc2ccccn2)cc(c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A12 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 3024626 ChemDiv3_004588 CCC(Sc1nc(c([nH]1)c2ccccc2)c3ccccc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A13 compound treatment 400.0 -878.0 -0.31 680.0 -3.75 0.0 -0.2222 -0.7136 3118515 ChemDiv3_004589 CCC(Sc1nnc2c3ccccc3n(CC=C)c2n1)C(=O)Nc4nc5CCCCc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A14 compound treatment 360.0 -918.0 -0.33 160.0 -524.0 -0.4 -0.5145 -0.9945 3024627 ChemDiv3_004590 CCSc1nnc(NC(=O)CCC(=O)OC2CCC(C)C(C)C2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A15 compound treatment 280.0 -998.0 -0.35 160.0 -524.0 -0.4 -0.5345 -0.998 3118516 ChemDiv3_004591 COC(=O)c1ccccc1NC(=O)COC(=O)c2cc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A16 compound treatment 240.0 -1040.0 -0.37 240.0 -444.0 -0.34 -0.5011 -0.9993 3118517 ChemDiv3_004592 Cc1nc(C)c(o1)C(=O)/C=C\2/Nc3cc(Cl)ccc3OC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A17 compound treatment 360.0 -918.0 -0.33 280.0 -404.0 -0.31 -0.4493 -0.9997 3024628 ChemDiv3_004593 O=C(COc1ccc(cc1)c2nnc(N3CCCCC3)c4ccccc24)N5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A18 compound treatment 200.0 -1080.0 -0.38 400.0 -284.0 -0.22 -0.4243 -0.9645 1446068 ChemDiv3_004594 CC1(C)C2CCC1(C)C(C2)OCC[N+]3(C)CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A19 compound treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 3118518 ChemDiv3_004595 CN(C1=NC(=O)/C(=C/C(=C/c2ccccc2)/C)/S1)c3ccc(O)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A20 compound treatment 200.0 -1080.0 -0.38 520.0 -164.0 -0.13 -0.3592 -0.8926 1566657 ChemDiv3_004596 CN(C)CCNC(=O)c1ccccn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A21 compound treatment 240.0 -1040.0 -0.37 240.0 -444.0 -0.34 -0.5011 -0.9993 3024629 ChemDiv3_004597 Cc1cccc[n+]1C/C=C\c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A22 compound treatment 160.0 -1120.0 -0.4 320.0 -364.0 -0.28 -0.4778 -0.9853 1268592 ChemDiv3_004598 O=C(Nc1ccccc1)N2c3ccccc3CCc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A23 mock treatment 200.0 -1080.0 -0.38 320.0 -364.0 -0.28 -0.4677 -0.9881 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 A24 mock treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B01 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3118519 ChemDiv3_004599 CCCC1(CN2CC3(CCC)CN(C1)C2C(O)C(O)C(O)CO)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B02 compound treatment 320.0 -958.0 -0.34 680.0 -3.75 0.0 -0.2422 -0.7131 3024630 ChemDiv3_004600 O=C(/C=C/c1ccco1)N2CCN(CC2)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B03 compound treatment 240.0 -1040.0 -0.37 360.0 -324.0 -0.25 -0.436 -0.9817 1681379 ChemDiv3_004601 CCCN1CCc2c(C#N)c(NC(=S)NC(=O)c3ccccc3)sc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B04 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3024754 ChemDiv3_004602 CCOc1ccc(cc1)C2=CC(c3cccc(OC)c3)c4ccccc4O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B05 compound treatment 440.0 -838.0 -0.3 240.0 -444.0 -0.34 -0.451 -0.9977 1128626 ChemDiv3_004603 CCOC(=O)c1ccc2[nH]c3C(CCCc3c2c1)NC=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B06 compound treatment 4240.0 2960.0 1.05 160.0 -524.0 -0.4 0.4588 0.4077 1152940 ChemDiv3_004604 CC(C)OC(=O)Cn1cnc2ccc(Br)cc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B07 compound treatment 240.0 -1040.0 -0.37 1120.0 436.0 0.33 -0.0234 -0.0471 1774881 ChemDiv3_004605 CCOC(=O)/C(=C\1/NC(=O)Nc2ccccc12)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B08 compound treatment 320.0 -958.0 -0.34 320.0 -364.0 -0.28 -0.4376 -0.9953 3118521 ChemDiv3_004606 COc1ccccc1N2CCN(CC2)C3CCN(Cc4cc(OC)c(OC)c(OC)c4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B09 compound treatment 5120.0 3840.0 1.36 1040.0 356.0 0.27 1.1573 0.8324 1248651 ChemDiv3_004607 Cc1oc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2c1C(=O)NN 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B10 compound treatment 480.0 -798.0 -0.28 320.0 -364.0 -0.28 -0.3975 -1.0 3118522 ChemDiv3_004608 CCN1C(=O)C(=Cc2cccn2c3ccc(O)cc3)C(=O)N(CC)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B11 compound treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 1683239 ChemDiv3_004609 CC(=O)N(c1ccc2oc3CCCCc3c2c1)S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B12 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3118523 ChemDiv3_004610 CC1(C)CC2(CC(C)(OC2=O)C(=O)CSc3nc4ccccc4s3)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B13 compound treatment 600.0 -678.0 -0.24 240.0 -444.0 -0.34 -0.4108 -0.9854 1235086 ChemDiv3_004611 Clc1ccc(CCN2C(CC(=O)Nc3ccccc3)C(=O)N(Cc4ccccc4)C2=S)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B14 compound treatment 240.0 -1040.0 -0.37 360.0 -324.0 -0.25 -0.436 -0.9817 3024755 ChemDiv3_004612 COc1ccc(/C=C/2\SC(=N)NC2=O)cc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B15 compound treatment 2080.0 803.0 0.28 240.0 -444.0 -0.34 -0.0396 -0.0892 1578381 ChemDiv3_004613 COc1ccc(CN2C(CC(=O)Nc3ccccc3)C(=O)N(C2=S)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B16 compound treatment 280.0 -998.0 -0.35 400.0 -284.0 -0.22 -0.4043 -0.9728 3024756 ChemDiv3_004614 COc1cccc(/C=C\2/NC(=O)N(Cc3ccc(F)cc3)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B17 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3118524 ChemDiv3_004615 N/C(=N\C(=O)/C=C/c1ccccc1)/Nc2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B18 compound treatment 400.0 -878.0 -0.31 360.0 -324.0 -0.25 -0.3959 -0.9938 3024757 ChemDiv3_004616 CCSc1nc2sc3COC(Cc3c2c(=O)n1c4ccc(OC)cc4)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B19 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 3118525 ChemDiv3_004617 N/C(=N\C(=O)c1cccc(Cl)c1)/Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B20 compound treatment 600.0 -678.0 -0.24 560.0 -124.0 -0.1 -0.2371 -0.9175 3118526 ChemDiv3_004618 O=C(Nc1nnc(s1)C2CCCCC2)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B21 compound treatment 240.0 -1040.0 -0.37 1200.0 516.0 0.4 0.02 0.037 1556779 ChemDiv3_004619 CC(N1C(=O)c2ccccc2C1=O)C(=O)OCC(=O)n3c4CCCCc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B22 compound treatment 280.0 -998.0 -0.35 320.0 -364.0 -0.28 -0.4477 -0.9931 3118527 ChemDiv3_004620 CCOc1ccc(cc1)c2nc3s/c(=C\C4=Cc5ccccc5OC4)/c(=O)n3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B23 mock treatment 280.0 -998.0 -0.35 360.0 -324.0 -0.25 -0.426 -0.9851 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 B24 mock treatment 440.0 -838.0 -0.3 240.0 -444.0 -0.34 -0.451 -0.9977 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C01 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 1870380 ChemDiv3_004621 CCc1cc(=O)oc2c(C)c3occ(c4ccc(Cl)cc4)c3cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C02 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 3118528 ChemDiv3_004622 CCCOc1ccc(Oc2nc(nc(n2)N(C)C)N(C)C)nn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C03 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3024758 ChemDiv3_004623 COC(=O)N1N=C(CC(C)C)CC1(O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C04 compound treatment 2080.0 803.0 0.28 200.0 -484.0 -0.37 -0.0613 -0.131 3118529 ChemDiv3_004624 CC(C)(C)C1=CC(=Nc2ccccc2N)C=C(C1O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C05 compound treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 3118650 ChemDiv3_004625 O=C1c2ccccc2-c3n[nH]c(=O)c4ccc(N5CCOCC5)c1c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C06 compound treatment 400.0 -878.0 -0.31 360.0 -324.0 -0.25 -0.3959 -0.9938 3024759 ChemDiv3_004626 C[n+]1ccc(/C=C/c2ccccc2F)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C07 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3118651 ChemDiv3_004627 Fc1nc(N2CCOCC2)c(F)c(NC(=O)CCC(=O)N3CCOCC3)c1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C08 compound treatment 320.0 -958.0 -0.34 360.0 -324.0 -0.25 -0.4159 -0.9882 3024760 ChemDiv3_004628 COc1ccc(/C=C/2\SC(=NC2=O)N(C)c3ccc(Cl)cc3)c(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C09 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3118652 ChemDiv3_004629 Cn1c(nc2cccc3cccc1c32)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C10 compound treatment 200.0 -1080.0 -0.38 240.0 -444.0 -0.34 -0.5112 -0.9984 3118653 ChemDiv3_004630 Cc1cc2/C(=c\3/sc4=NCN(Cn4c3=O)c5cccc(Br)c5)/C(=O)Nc2c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C11 compound treatment 280.0 -998.0 -0.35 320.0 -364.0 -0.28 -0.4477 -0.9931 1849841 ChemDiv3_004631 COc1cccc(NC(=O)CSc2nnc(N)s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C12 compound treatment 320.0 -958.0 -0.34 280.0 -404.0 -0.31 -0.4594 -0.999 3118654 ChemDiv3_004632 COc1ccc(cc1)c2c(c3ccc(OC)cc3)c4c(O)ncnc4n2Cc5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C13 compound treatment 320.0 -958.0 -0.34 440.0 -244.0 -0.19 -0.3725 -0.9605 3024761 ChemDiv3_004633 Oc1ccc(=O)n(CN2CCC(Cc3ccccc3)CC2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C14 compound treatment 520.0 -758.0 -0.27 240.0 -444.0 -0.34 -0.4309 -0.9931 1873344 ChemDiv3_004634 Cc1cccc(NC(=O)CSc2nc3CC(C)(C)CC(=O)c3cc2C#N)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C15 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3118655 ChemDiv3_004635 Clc1cccc(NC(=O)COC(=O)CCc2c[nH]c(=O)[nH]2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C16 compound treatment 280.0 -998.0 -0.35 400.0 -284.0 -0.22 -0.4043 -0.9728 3118656 ChemDiv3_004636 CC(C)CC(=O)/C=C\1/Nc2cc(Cl)ccc2OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C17 compound treatment 280.0 -998.0 -0.35 360.0 -324.0 -0.25 -0.426 -0.9851 3024762 ChemDiv3_004637 Clc1ccc(cc1)c2nn(CC(=O)Nc3cccc4ccccc34)c(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C18 compound treatment 320.0 -958.0 -0.34 1240.0 556.0 0.43 0.0618 0.1132 1281710 ChemDiv3_004638 CC1(C)C2CCC1(C)C(C2)OCC[N+]3(C)CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C19 compound treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 1406364 ChemDiv3_004639 O=c1sc2C3C(COc4ccccc34)CSc2n1c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C20 compound treatment 240.0 -1040.0 -0.37 440.0 -244.0 -0.19 -0.3926 -0.9508 3118657 ChemDiv3_004640 Clc1ccccc1C(=O)Nc2c3CCCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C21 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 1056705 ChemDiv3_004641 CCOC(=O)C[n+]1ccccc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C22 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3118658 ChemDiv3_004642 Clc1ccc2Sc3ccccc3N(C(=O)CCN4CCOCC4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C23 mock treatment 3320.0 2040.0 0.72 320.0 -364.0 -0.28 0.3149 0.4055 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 C24 mock treatment 4120.0 2840.0 1.01 240.0 -444.0 -0.34 0.4721 0.4436 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D01 compound treatment 360.0 -918.0 -0.33 320.0 -364.0 -0.28 -0.4276 -0.9971 3024797 ChemDiv3_004643 CCC1(CN2CC3(CC)CN(C1)C2c4ccc(cc4)C(C)C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D02 compound treatment 200.0 -1080.0 -0.38 280.0 -404.0 -0.31 -0.4895 -0.9946 3118659 ChemDiv3_004644 O=C(N1CCN=C1c2ccccc2)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D03 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3118660 ChemDiv3_004645 Cc1ccccc1n2c(SCC(=O)O)nc3sc4COC(C)(C)Cc4c3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D04 compound treatment 480.0 -798.0 -0.28 280.0 -404.0 -0.31 -0.4192 -0.999 1163303 ChemDiv3_004646 CC(=O)Nc1ccc(cc1)n2c(C)nc(=O)c(c2C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D05 compound treatment 560.0 -718.0 -0.25 400.0 -284.0 -0.22 -0.334 -0.997 3118661 ChemDiv3_004647 CCn1c2/C(=N/O)/CCCc2c3cc(Br)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D06 compound treatment 360.0 -918.0 -0.33 320.0 -364.0 -0.28 -0.4276 -0.9971 1215655 ChemDiv3_004648 CC(C)COC(=O)Cn1cnc2ccc(Br)cc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D07 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3118662 ChemDiv3_004649 NC(=O)CCNCc1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D08 compound treatment 520.0 -758.0 -0.27 240.0 -444.0 -0.34 -0.4309 -0.9931 3024798 ChemDiv3_004650 CC1CCCN(C1)C2CCN(Cc3ccccc3Cl)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D09 compound treatment 480.0 -798.0 -0.28 280.0 -404.0 -0.31 -0.4192 -0.999 1184645 ChemDiv3_004651 Cc1cc(C)c(cc1C)S(=O)(=O)Nc2cc3c4C(=O)CCCc4oc3c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D10 compound treatment 280.0 -998.0 -0.35 400.0 -284.0 -0.22 -0.4043 -0.9728 3024799 ChemDiv3_004652 Oc1ccc(Br)cc1/C=N/c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D11 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3118663 ChemDiv3_004653 COc1ccc(NS(=O)(=O)c2ccc3SC(=O)c4cccc2c34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D12 compound treatment 400.0 -878.0 -0.31 280.0 -404.0 -0.31 -0.4393 -1.0 3118664 ChemDiv3_004654 CC(CC1CC(C)(C)OC1=O)C(=O)Nc2nncs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D13 compound treatment 400.0 -878.0 -0.31 280.0 -404.0 -0.31 -0.4393 -1.0 1338252 ChemDiv3_004655 CCN1C(=O)C(CC(=O)Nc2ccc(F)cc2)N(CCc3ccccc3)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D14 compound treatment 360.0 -918.0 -0.33 320.0 -364.0 -0.28 -0.4276 -0.9971 3118665 ChemDiv3_004656 CCSC1=N/C(=C\c2ccc(cc2)C(C)C)/C(=O)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D15 compound treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 3024800 ChemDiv3_004657 NC(=O)C1CCN(CC1)C(=S)Nc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D16 compound treatment 360.0 -918.0 -0.33 360.0 -324.0 -0.25 -0.4059 -0.9911 1485635 ChemDiv3_004658 CCn1c2ccccc2c3cc(NC(=O)c4ccccc4C)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D17 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 1155119 ChemDiv3_004659 Clc1ccc(NC(=O)Nc2nc(cs2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D18 compound treatment 400.0 -878.0 -0.31 320.0 -364.0 -0.28 -0.4176 -0.9985 3118666 ChemDiv3_004660 CCOC(=O)c1c(NC(=O)c2ccccc2)sc3COC(Cc13)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D19 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 1236887 ChemDiv3_004661 CC(=O)NC(=S)Nc1nc2ccccc2n1C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D20 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3118667 ChemDiv3_004662 CC(C)c1nnc(NC(=O)/C=C/c2ccc3OCOc3c2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D21 compound treatment 3560.0 2280.0 0.81 360.0 -324.0 -0.25 0.3968 0.4685 1788359 ChemDiv3_004663 COc1ccc(cc1)C(=O)OCC(=O)n2c(C)c(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D22 compound treatment 360.0 -918.0 -0.33 360.0 -324.0 -0.25 -0.4059 -0.9911 3118668 ChemDiv3_004664 Cc1nn2c(=O)/c(=C/c3ccccc3)/sc2nc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D23 mock treatment 400.0 -878.0 -0.31 240.0 -444.0 -0.34 -0.461 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 D24 mock treatment 280.0 -998.0 -0.35 320.0 -364.0 -0.28 -0.4477 -0.9931 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E01 compound treatment 1920.0 643.0 0.23 1320.0 636.0 0.49 0.5066 0.9398 1865983 ChemDiv3_004665 COc1ccc(cc1)c2cc(=O)oc3cc4occ(c5cccc(OC)c5)c4cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E02 compound treatment 1120.0 -158.0 -0.06 1520.0 836.0 0.64 0.4145 0.6431 1539024 ChemDiv3_004666 O=C(NC1(CC2CC3CC(C2)C1)C3)c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E03 compound treatment 2280.0 1000.0 0.36 640.0 -43.8 -0.03 0.2277 0.6375 3118669 ChemDiv3_004667 CCOc1ccc(/N=C/2\C(=O)N(CN3CCCCC3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E04 compound treatment 2200.0 923.0 0.33 1040.0 356.0 0.27 0.4248 0.996 3024801 ChemDiv3_004668 CCNc1nc(NCC)nc(SCCOc2ccc(Br)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E05 compound treatment 5160.0 3880.0 1.38 360.0 -324.0 -0.25 0.7981 0.5703 3118670 ChemDiv3_004669 OC(=O)CNc1c(F)c(F)nc(F)c1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E06 compound treatment 920.0 -358.0 -0.13 280.0 -404.0 -0.31 -0.3089 -0.9222 3024802 ChemDiv3_004670 C[n+]1ccc(/C=C/c2ccccc2O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E07 compound treatment 2160.0 883.0 0.31 2400.0 1720.0 1.32 1.1531 0.8514 3118671 ChemDiv3_004671 Fc1nc(N2CCCCC2)c(F)c(N3C(=O)CCC3=O)c1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E08 compound treatment 3080.0 1800.0 0.64 1680.0 996.0 0.76 0.993 0.996 3118672 ChemDiv3_004672 Oc1ccc(/N=C\2/SC(CC(=O)Nc3ccccc3)C(=O)N2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E09 compound treatment 280.0 -998.0 -0.35 2840.0 2160.0 1.66 0.9203 0.5437 3024803 ChemDiv3_004673 CC1(C)CC(=O)/C(=C/c2ccccc2)/C(C)(C)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E10 compound treatment 1400.0 123.0 0.04 1280.0 596.0 0.46 0.3544 0.7708 3118673 ChemDiv3_004674 COc1cc(cc(OC)c1OC)N2CN=c3s/c(=C\C=C\c4ccccc4)/c(=O)n3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E11 compound treatment 1040.0 -238.0 -0.08 7840.0 7160.0 5.49 3.8253 0.6962 3024804 ChemDiv3_004675 CCCc1cc(O)nc(SCC(=O)NCCc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E12 compound treatment 1160.0 -118.0 -0.04 2400.0 1720.0 1.32 0.9022 0.6844 1364723 ChemDiv3_004676 Cc1ccc(OCC(=O)NC2CC(C)(C)NC(C)(C)C2)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E13 compound treatment 4120.0 2840.0 1.01 440.0 -244.0 -0.19 0.5807 0.5662 3118674 ChemDiv3_004677 Cc1ccc(cc1)c2nnc(o2)c3cc(C(=O)NN)c(C)nc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E14 compound treatment 2880.0 1600.0 0.57 1600.0 916.0 0.7 0.8994 0.9944 3024845 ChemDiv3_004678 CC1(C)OC(=O)C(=CNc2ccccc2)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E15 compound treatment 1200.0 -77.5 -0.03 2080.0 1400.0 1.07 0.7385 0.6887 3118811 ChemDiv3_004679 COC(=O)c1ccc(NC(=O)CSc2nc(=O)cc(N)n2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E16 compound treatment 6600.0 5320.0 1.89 1160.0 476.0 0.37 1.5936 0.8286 3024846 ChemDiv3_004680 O/N=C/1\NC(=O)\C(=C/c2ccc(O)cc2)\S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E17 compound treatment 5960.0 4680.0 1.66 600.0 -83.8 -0.06 1.1291 0.6792 3118812 ChemDiv3_004681 FC(F)(F)c1cccc(NC(=O)Cn2nc(c3ccccc3)c4ccccc4c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E18 compound treatment 1480.0 203.0 0.07 320.0 -364.0 -0.28 -0.1467 -0.5087 1283219 ChemDiv3_004682 CC1(C)C2CCC1(C)C(C2)NC(=O)CC[N+](C)(C)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E19 compound treatment 1440.0 163.0 0.06 1000.0 316.0 0.24 0.2124 0.8513 3118813 ChemDiv3_004683 Brc1ccc(cc1)N2C(=O)C3Sc4[nH]c(=O)sc4C(/C=C/c5ccccc5)C3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E20 compound treatment 1720.0 443.0 0.16 960.0 276.0 0.21 0.261 0.989 3024848 ChemDiv3_004684 CN1CCCNC1c2ccc(o2)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E21 compound treatment 1320.0 42.5 0.02 720.0 36.3 0.03 0.0303 0.9586 3118814 ChemDiv3_004685 CCOC(=O)C[N+](C)(C)Cc1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E22 compound treatment 880.0 -398.0 -0.14 320.0 -364.0 -0.28 -0.2972 -0.9499 1279489 ChemDiv3_004686 CCn1c(nc2ccccc12)c3nonc3N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E23 mock treatment 5560.0 4280.0 1.52 1680.0 996.0 0.76 1.6151 0.9496 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 E24 mock treatment 360.0 -918.0 -0.33 880.0 196.0 0.15 -0.1236 -0.3447 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F01 compound treatment 1320.0 42.5 0.02 1840.0 1160.0 0.89 0.6383 0.719 3118815 ChemDiv3_004687 CCC1(CC)Cc2ccccc2-c3[nH]c4nnc(S)n4c(=O)c31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F02 compound treatment 3320.0 2040.0 0.72 720.0 36.3 0.03 0.532 0.7337 3024849 ChemDiv3_004688 COc1ccc(/C=C/C(=O)N2CCN=C2c3ccccc3)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F03 compound treatment 2600.0 1320.0 0.47 1200.0 516.0 0.4 0.612 0.9965 3118816 ChemDiv3_004689 COc1ccccc1n2c(=O)c3c4CCCc4sc3n5c(S)nnc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F04 compound treatment 4600.0 3320.0 1.18 1680.0 996.0 0.76 1.3742 0.9781 1684840 ChemDiv3_004690 Cc1cc(=O)oc2cc(OCC(=O)N)c(Cl)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F05 compound treatment 1200.0 -77.5 -0.03 1200.0 516.0 0.4 0.2608 0.6565 1206179 ChemDiv3_004691 CC(C)c1ccc2[nH]c3C(O)CCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F06 compound treatment 1760.0 483.0 0.17 840.0 156.0 0.12 0.2059 0.9849 3118817 ChemDiv3_004692 COc1cc(/C=C/C(=O)N2CCC(C)CC2)ccc1OCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F07 compound treatment 1360.0 82.5 0.03 5400.0 4720.0 3.62 2.581 0.7128 3024850 ChemDiv3_004693 O=C(C[n+]1ccccc1)Nc2c3CCCc3nc4CCCCc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F08 compound treatment 1320.0 42.5 0.02 2520.0 1840.0 1.41 1.0075 0.7146 1604185 ChemDiv3_004694 COc1cccc(OC)c1C(=O)N2CCN(CC2)C(=O)COc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F09 compound treatment 1400.0 123.0 0.04 5040.0 4360.0 3.34 2.3956 0.7162 3118818 ChemDiv3_004695 Cc1cc(ccc1Cl)S(=O)(=O)Nc2ccc3oc4CCC(Cc4c3c2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F10 compound treatment 1720.0 443.0 0.16 6000.0 5320.0 4.08 2.997 0.7338 1142903 ChemDiv3_004696 NS(=O)(=O)c1ccc(NC(=O)c2ccccc2C(=O)N3CCCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F11 compound treatment 760.0 -518.0 -0.18 5200.0 4520.0 3.47 2.3219 0.6687 1284552 ChemDiv3_004697 CCOC(=O)c1c(oc2ccc(cc12)N(C(=O)C)S(=O)(=O)c3ccc(OC)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F12 compound treatment 4120.0 2840.0 1.01 3520.0 2840.0 2.18 2.2527 0.9388 3024851 ChemDiv3_004698 CC(CC1CC(C)OC1=O)C(=O)NC(=S)Nc2nncs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F13 compound treatment 4080.0 2800.0 0.99 1200.0 516.0 0.4 0.9832 0.9187 1398812 ChemDiv3_004699 COC(=O)CN1C(CC(=O)Nc2ccc(F)cc2)C(=O)N(C1=S)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F14 compound treatment 3960.0 2680.0 0.95 1040.0 356.0 0.27 0.8663 0.8749 3024852 ChemDiv3_004700 CCOC(=O)COc1ccccc1/C=C/2\N=C(SCC)SC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F15 compound treatment 9640.0 8360.0 2.97 4040.0 3360.0 2.58 3.9196 0.9975 1332272 ChemDiv3_004701 CCNC(=O)CC1N(NC(=O)c2ccccc2)C(=S)N(CC)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F16 compound treatment 7320.0 6040.0 2.14 2560.0 1880.0 1.44 2.5343 0.9813 3118819 ChemDiv3_004702 CCn1c2ccccc2c3cc(NC(=O)Oc4ccccc4)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F17 compound treatment 3760.0 2480.0 0.88 3440.0 2760.0 2.12 2.119 0.9245 1303305 ChemDiv3_004703 COc1ccc2nc(SC(=O)c3ccccc3)nc(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F18 compound treatment 8280.0 7000.0 2.48 840.0 156.0 0.12 1.8414 0.7404 3118820 ChemDiv3_004704 CC(C)C1Cc2c(CO1)sc3nc(SCc4ccc(Cl)c(Cl)c4)nc(N)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F19 compound treatment 2240.0 963.0 0.34 1120.0 436.0 0.33 0.4783 1.0 3024853 ChemDiv3_004705 CCc1ccc2NC(=O)N(C(=C)c2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F20 compound treatment 1080.0 -198.0 -0.07 2000.0 1320.0 1.01 0.665 0.6565 3118821 ChemDiv3_004706 COCc1nnc(NC(=O)/C=C/c2ccc3OCOc3c2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F21 compound treatment 2480.0 1200.0 0.43 1240.0 556.0 0.43 0.6036 1.0 1870814 ChemDiv3_004707 Fc1ccc(Nc2nc(Nc3ccc(F)cc3)nc(n2)N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F22 compound treatment 5160.0 3880.0 1.38 3560.0 2880.0 2.21 2.5353 0.9742 3118822 ChemDiv3_004708 O=c1/c(=C/c2cccs2)/sc3nc(=O)c(Cc4ccccc4)nn13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F23 mock treatment 2120.0 843.0 0.3 440.0 -244.0 -0.19 0.079 0.2241 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 F24 mock treatment 1000.0 -278.0 -0.1 800.0 116.0 0.09 -0.0065 -0.0489 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G01 compound treatment 800.0 -478.0 -0.17 3320.0 2640.0 2.02 1.3113 0.6457 1867727 ChemDiv3_004709 CCCCc1cc(=O)oc2cc3oc4CCCCc4c3cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G02 compound treatment 840.0 -438.0 -0.16 1800.0 1120.0 0.86 0.4962 0.5698 3118823 ChemDiv3_004710 Cc1ccccc1OCc2nnc3c4cnn(Cc5ccccc5)c4ncn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G03 compound treatment 360.0 -918.0 -0.33 360.0 -324.0 -0.25 -0.4059 -0.9911 3118824 ChemDiv3_004711 CC1CCN(CN2C(=O)/C(=N\c3ccccc3C)/c4ccccc24)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G04 compound treatment 360.0 -918.0 -0.33 400.0 -284.0 -0.22 -0.3842 -0.9809 3024855 ChemDiv3_004712 CCNc1nc(OCC=C)nc(n1)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G05 compound treatment 1440.0 163.0 0.06 800.0 116.0 0.09 0.1039 0.9776 3118825 ChemDiv3_004713 Fc1nc(OCC=C)c2Oc3cc(Br)c(Br)cc3Oc2c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G06 compound treatment 360.0 -918.0 -0.33 560.0 -124.0 -0.1 -0.2973 -0.8769 3024856 ChemDiv3_004714 Oc1ccccc1/C=C/c2cc[n+](CC=C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G07 compound treatment 1760.0 483.0 0.17 1400.0 716.0 0.55 0.5099 0.8853 3118826 ChemDiv3_004715 COc1ccccc1/C=C/C(=O)Nc2nc(N)n(n2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G08 compound treatment 920.0 -358.0 -0.13 360.0 -324.0 -0.25 -0.2654 -0.9512 3024857 ChemDiv3_004716 Oc1ccc(/N=C\2/SCC(=O)N2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G09 compound treatment 400.0 -878.0 -0.31 1080.0 396.0 0.3 -0.005 -0.0115 3118827 ChemDiv3_004717 CC1(C)NC(C)(C)C(=C1)C(=O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G10 compound treatment 1240.0 -37.5 -0.01 400.0 -284.0 -0.22 -0.1634 -0.7489 3024858 ChemDiv3_004718 Cc1cc(C)cc(c1)N2C(SCC2=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G11 compound treatment 1280.0 2.5 0.0 720.0 36.3 0.03 0.0203 0.7293 3118828 ChemDiv3_004719 COc1ccc(cc1NC(=S)NC(=O)Cc2ccc(Cl)cc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G12 compound treatment 2160.0 883.0 0.31 440.0 -244.0 -0.19 0.089 0.2441 3024899 ChemDiv3_004720 COc1cccc(/C=C/2\CC(C)C/C(=C\c3ccccc3OC)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G13 compound treatment 1080.0 -198.0 -0.07 1760.0 1080.0 0.83 0.5347 0.6448 3118829 ChemDiv3_004721 CCCc1n(CC(O)COc2ccccc2C)c3ccccc3[n+]1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G14 compound treatment 3800.0 2520.0 0.89 1000.0 316.0 0.24 0.8044 0.8676 3024900 ChemDiv3_004722 CC(C)n1nc(O)c2C(SCC(=O)Nc21)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G15 compound treatment 1080.0 -198.0 -0.07 360.0 -324.0 -0.25 -0.2253 -0.8724 3118830 ChemDiv3_004723 CN(/C(=N/S(=O)(=O)c1ccc(C)cc1)/c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G16 compound treatment 560.0 -718.0 -0.25 2640.0 1960.0 1.5 0.882 0.579 3024901 ChemDiv3_004724 CCOC(=O)CN1C(=O)S/C(=C\c2ccc(cc2)C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G17 compound treatment 5880.0 4600.0 1.63 400.0 -284.0 -0.22 1.0005 0.6074 3118831 ChemDiv3_004725 CCN(CC)S(=O)(=O)c1cc(ccc1C)c2nn(C)c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G18 compound treatment 1080.0 -198.0 -0.07 280.0 -404.0 -0.31 -0.2687 -0.8456 3024902 ChemDiv3_004726 COC(=O)COc1ccc(Oc2nc(SC)nc(n2)N(C)C)nn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G19 compound treatment 720.0 -558.0 -0.2 320.0 -364.0 -0.28 -0.3373 -0.9857 1436626 ChemDiv3_004727 COc1cc2CCN(Cc2cc1OC)C(=S)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G20 compound treatment 520.0 -758.0 -0.27 960.0 276.0 0.21 -0.04 -0.117 3118832 ChemDiv3_004728 CN(C)c1ccc(/C=C\2/S/C(=N/O)/NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G21 compound treatment 800.0 -478.0 -0.17 600.0 -83.8 -0.06 -0.1652 -0.912 3024903 ChemDiv3_004729 CCCOc1ccc(=O)n(C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G22 compound treatment 760.0 -518.0 -0.18 520.0 -164.0 -0.13 -0.2187 -0.9829 3024904 ChemDiv3_004730 COC(=O)Cn1c2ccc(Cl)cc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G23 mock treatment 880.0 -398.0 -0.14 320.0 -364.0 -0.28 -0.2972 -0.9499 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 G24 mock treatment 1560.0 283.0 0.1 1200.0 516.0 0.4 0.3511 0.8589 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H01 compound treatment 1040.0 -238.0 -0.08 3240.0 2560.0 1.96 1.3281 0.6761 3118833 ChemDiv3_004731 CC1(C)Cc2ccccc2-c3c1c(=O)n(Cc4ccccc4)c5nnc(S)n35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H02 compound treatment 520.0 -758.0 -0.27 480.0 -204.0 -0.16 -0.3006 -0.9668 1871178 ChemDiv3_004732 O=C(Oc1cccc2cccnc12)N3c4ccccc4Sc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H03 compound treatment 520.0 -758.0 -0.27 600.0 -83.8 -0.06 -0.2355 -0.8522 3024905 ChemDiv3_004733 CC(C)C1Cc2c(CO1)sc3nc(SCC(=O)Nc4ccccc4)nc(N)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H04 compound treatment 880.0 -398.0 -0.14 880.0 196.0 0.15 0.0068 0.0331 1556837 ChemDiv3_004734 CC(C)C(N1C(=O)c2ccccc2C1=O)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4ncccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H05 compound treatment 800.0 -478.0 -0.17 520.0 -164.0 -0.13 -0.2087 -0.9892 3024907 ChemDiv3_004735 Cc1ccc2[nH]c3/C(=N\CC=C)/CCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H06 compound treatment 600.0 -678.0 -0.24 3480.0 2800.0 2.15 1.348 0.624 1227251 ChemDiv3_004736 COc1cc(cc(OC)c1OC)C(=O)OCC(=O)Nc2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H07 compound treatment 960.0 -318.0 -0.11 1080.0 396.0 0.3 0.1355 0.4176 3118962 ChemDiv3_004737 COc1ccc(/C=C/C(=O)Nc2c3CCCc3nc4CCCCc24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H08 compound treatment 3040.0 1760.0 0.63 720.0 36.3 0.03 0.4618 0.7378 3024908 ChemDiv3_004738 CCCOC(=O)CSc1nc(N)c(C#N)c(c1C#N)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H09 compound treatment 1240.0 -37.5 -0.01 680.0 -3.75 0.0 -0.0114 -0.8407 1320144 ChemDiv3_004739 Cc1cc(ccc1Cl)S(=O)(=O)Nc2cc(Br)c3oc4CCCC(=O)c4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H10 compound treatment 6040.0 4760.0 1.69 800.0 116.0 0.09 1.2577 0.7434 1303471 ChemDiv3_004740 O=C1N(CNc2ccccc2)CCN1CNc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H11 compound treatment 1000.0 -278.0 -0.1 1440.0 756.0 0.58 0.3409 0.5789 1244728 ChemDiv3_004741 Cc1ccc(C)c(c1)S(=O)(=O)Nc2ccc3oc4CCC(Cc4c3c2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H12 compound treatment 3800.0 2520.0 0.89 800.0 116.0 0.09 0.6959 0.7738 3118963 ChemDiv3_004742 CCOc1ccc(Nc2nc(cs2)C3(C)CC4(CC(C)(C)OC4=O)C(=O)O3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H13 compound treatment 720.0 -558.0 -0.2 680.0 -3.75 0.0 -0.1419 -0.7173 3024909 ChemDiv3_004743 CCN/1C(=O)CC(S\C1=N/c2ccccc2)C(=O)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H14 compound treatment 1680.0 403.0 0.14 880.0 196.0 0.15 0.2075 0.9996 3024910 ChemDiv3_004744 CCSC1=N/C(=C\c2cc(Br)c(OC(=O)C)c(OC)c2)/C(=O)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H15 compound treatment 7440.0 6160.0 2.19 480.0 -204.0 -0.16 1.4352 0.6548 1580209 ChemDiv3_004745 COC(=O)CN1C(CC(=O)Nc2ccc(OC)cc2)C(=O)N(Cc3ccccc3)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H16 compound treatment 600.0 -678.0 -0.24 600.0 -83.8 -0.06 -0.2154 -0.8658 3024911 ChemDiv3_004746 O=C(NCc1ccc2OCOc2c1)Oc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H17 compound treatment 3360.0 2080.0 0.74 400.0 -284.0 -0.22 0.3683 0.4782 3118964 ChemDiv3_004747 N(c1ccccc1)c2nc(Nc3ccccc3)nc(Sc4nc5ccccc5[nH]4)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H18 compound treatment 560.0 -718.0 -0.25 400.0 -284.0 -0.22 -0.334 -0.997 3118965 ChemDiv3_004748 CSc1nc2sc3COC(C)(C)Cc3c2c(=O)n1c4cccc(Br)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H19 compound treatment 480.0 -798.0 -0.28 560.0 -124.0 -0.1 -0.2672 -0.8954 1787885 ChemDiv3_004749 O=C(N1c2ccccc2Sc3ccccc13)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H20 compound treatment 920.0 -358.0 -0.13 680.0 -3.75 0.0 -0.0917 -0.723 3118966 ChemDiv3_004750 COCc1nnc(NC(=O)/C=C/c2cc(OC)c(OC)c(OC)c2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H21 compound treatment 1280.0 2.5 0.0 920.0 236.0 0.18 0.1289 0.7106 3024912 ChemDiv3_004751 N/C(=N/C=C1C(=O)NC(=O)NC1=O)/Nc2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H22 compound treatment 9280.0 8000.0 2.84 520.0 -164.0 -0.13 1.9185 0.6751 3118967 ChemDiv3_004752 Cc1nn2c(=O)/c(=C/C=C/c3ccccc3)/sc2nc1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H23 mock treatment 2720.0 1440.0 0.51 1840.0 1160.0 0.89 0.9895 0.9658 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 H24 mock treatment 640.0 -638.0 -0.23 440.0 -244.0 -0.19 -0.2922 -0.9956 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I01 compound treatment 240.0 -1040.0 -0.37 400.0 -284.0 -0.22 -0.4143 -0.9687 1277008 ChemDiv3_004753 O=c1oc2cc3occ(c4ccccc4)c3cc2c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I02 compound treatment 280.0 -998.0 -0.35 240.0 -444.0 -0.34 -0.4911 -0.9998 3118968 ChemDiv3_004754 Cc1ccc(cc1)c2nnc3c4cnn(c5ccccc5)c4ncn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I03 compound treatment 3320.0 2040.0 0.72 520.0 -164.0 -0.13 0.4235 0.5758 3024913 ChemDiv3_004755 N/C(=N/O)/CC(=O)Nc1cccc(c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I04 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3118969 ChemDiv3_004756 Cc1c(NC(=O)Nc2ccc(C)cc2)sc(=S)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I05 compound treatment 440.0 -838.0 -0.3 280.0 -404.0 -0.31 -0.4293 -0.9998 3024914 ChemDiv3_004757 Brc1cnc(nc1N2CCOCC2)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I06 compound treatment 320.0 -958.0 -0.34 520.0 -164.0 -0.13 -0.3291 -0.9086 3118970 ChemDiv3_004758 OC(=O)CC(NCc1ccccc1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I07 compound treatment 1480.0 203.0 0.07 1520.0 836.0 0.64 0.5048 0.7814 3118971 ChemDiv3_004759 OC(=O)CCC(=O)Nc1nc2NC(=O)CC(c3ccccc3)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I08 compound treatment 360.0 -918.0 -0.33 320.0 -364.0 -0.28 -0.4276 -0.9971 3024915 ChemDiv3_004760 COc1cc(/C=C/2\SC(=NC2=O)N(C)c3ccc(O)cc3)ccc1OCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I09 compound treatment 560.0 -718.0 -0.25 600.0 -83.8 -0.06 -0.2254 -0.8588 1474160 ChemDiv3_004761 Clc1cccc(NC(=O)Nc2ccc3c(c2)oc4ccccc43)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I10 compound treatment 360.0 -918.0 -0.33 280.0 -404.0 -0.31 -0.4493 -0.9997 3118972 ChemDiv3_004762 COc1ccc(cc1OC)C2NC(=S)NC(=C2)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I11 compound treatment 400.0 -878.0 -0.31 400.0 -284.0 -0.22 -0.3742 -0.9848 3118973 ChemDiv3_004763 NC(=O)c1ccccc1OCC(=O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I12 compound treatment 360.0 -918.0 -0.33 280.0 -404.0 -0.31 -0.4493 -0.9997 1870736 ChemDiv3_004764 COc1ccc2[nH]c3C(NCCc3c2c1)C4CCC(=CC4)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I13 compound treatment 240.0 -1040.0 -0.37 240.0 -444.0 -0.34 -0.5011 -0.9993 1866294 ChemDiv3_004765 OC(COc1ccc(Br)cc1)Cn2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I14 compound treatment 280.0 -998.0 -0.35 680.0 -3.75 0.0 -0.2523 -0.7128 3118974 ChemDiv3_004766 COc1ccc(CNCC(C)NCc2ccc(OC)c(OC)c2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I15 compound treatment 360.0 -918.0 -0.33 440.0 -244.0 -0.19 -0.3625 -0.9655 3024962 ChemDiv3_004767 Cc1ccc(cc1S(=O)(=O)NCc2cccnc2)c3nnc(S)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I16 compound treatment 320.0 -958.0 -0.34 680.0 -3.75 0.0 -0.2422 -0.7131 3118975 ChemDiv3_004768 CN1C(=O)S/C(=C/c2ccccc2OCc3ccc(cc3)C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I17 compound treatment 400.0 -878.0 -0.31 2120.0 1440.0 1.1 0.5596 0.4884 3024963 ChemDiv3_004769 Cc1ccc(cc1S(=O)(=O)N2CCOCC2)c3nn(C)c(=O)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I18 compound treatment 240.0 -1040.0 -0.37 360.0 -324.0 -0.25 -0.436 -0.9817 3118976 ChemDiv3_004770 CC(CC(=O)O)CC(=O)Nc1ccccc1C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I19 compound treatment 360.0 -918.0 -0.33 560.0 -124.0 -0.1 -0.2973 -0.8769 1470431 ChemDiv3_004771 CCOc1ccc(cc1)C(=O)N2CCc3cc(OC)c(OC)cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I20 compound treatment 240.0 -1040.0 -0.37 2320.0 1640.0 1.26 0.628 0.4798 3024964 ChemDiv3_004772 CC(CN1CCCCC1)OC(=O)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I21 compound treatment 720.0 -558.0 -0.2 360.0 -324.0 -0.25 -0.3156 -0.9936 3118977 ChemDiv3_004773 CCSc1nc(SCC)c2c3CCCCc3[nH]c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I22 compound treatment 400.0 -878.0 -0.31 240.0 -444.0 -0.34 -0.461 -0.999 3024965 ChemDiv3_004774 CC(C)n1c2ccc(Cl)cc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I23 mock treatment 560.0 -718.0 -0.25 400.0 -284.0 -0.22 -0.334 -0.997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 I24 mock treatment 440.0 -838.0 -0.3 240.0 -444.0 -0.34 -0.451 -0.9977 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J01 compound treatment 640.0 -638.0 -0.23 320.0 -364.0 -0.28 -0.3574 -0.9945 1370693 ChemDiv3_004775 OC(=O)CCNC(=O)c1cccnc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J02 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3118978 ChemDiv3_004776 CC1=CC(C)(C)N(C(=O)/C=C/c2ccccc2)c3ccc(C)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J03 compound treatment 360.0 -918.0 -0.33 3400.0 2720.0 2.09 1.2444 0.5896 1327411 ChemDiv3_004777 Fc1ccc(Nc2cccc3nonc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J04 compound treatment 240.0 -1040.0 -0.37 360.0 -324.0 -0.25 -0.436 -0.9817 1573339 ChemDiv3_004778 COc1ccccc1c2coc3cc(OCC(=O)OCC(C)C)ccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J05 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 1494509 ChemDiv3_004779 Cc1ccc2[nH]c3C(CCCc3c2c1)NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J06 compound treatment 800.0 -478.0 -0.17 360.0 -324.0 -0.25 -0.2955 -0.9825 3118979 ChemDiv3_004780 Cc1cccc(NC(=O)COC(=O)/C=C/c2ccc(F)cc2)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J07 compound treatment 440.0 -838.0 -0.3 360.0 -324.0 -0.25 -0.3858 -0.9961 3119110 ChemDiv3_004781 NC(=O)CN1C(=O)C2(C(=C(N)OC3=C2C(=O)CCC3)C#N)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J08 compound treatment 1560.0 283.0 0.1 440.0 -244.0 -0.19 -0.0615 -0.2895 3024966 ChemDiv3_004782 CC(C)c1ccc(/C=C/C(=O)NC(=S)Nc2ccc(cc2)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J09 compound treatment 1920.0 643.0 0.23 200.0 -484.0 -0.37 -0.1014 -0.2328 3119111 ChemDiv3_004783 CCc1ccc(cc1)S(=O)(=O)/N=C\2/C=C(Nc3ccccc3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J10 compound treatment 560.0 -718.0 -0.25 240.0 -444.0 -0.34 -0.4209 -0.9897 3024967 ChemDiv3_004784 Cc1ccc(cc1)S(=O)(=O)c2cc3c(=O)n4ccccc4nc3n(Cc5ccccc5)c2=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J11 compound treatment 240.0 -1040.0 -0.37 600.0 -83.8 -0.06 -0.3057 -0.8182 1676345 ChemDiv3_004785 CC(C)c1ccc(cc1)S(=O)(=O)Nc2cc3c4CCCCc4oc3c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J12 compound treatment 320.0 -958.0 -0.34 320.0 -364.0 -0.28 -0.4376 -0.9953 3119112 ChemDiv3_004786 Cc1ccc(cc1)C2=NNC(=O)C(C2)P(=O)(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J13 compound treatment 240.0 -1040.0 -0.37 400.0 -284.0 -0.22 -0.4143 -0.9687 1618837 ChemDiv3_004787 OC(C1CCN(CC1)C(=S)Nc2ccccc2)(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J14 compound treatment 4080.0 2800.0 0.99 1360.0 676.0 0.52 1.0701 0.9541 3024968 ChemDiv3_004788 CC/1=NOC(=O)\C1=C/C=C\c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J15 compound treatment 440.0 -838.0 -0.3 360.0 -324.0 -0.25 -0.3858 -0.9961 3119113 ChemDiv3_004789 Fc1ccc(CCN2C(CC(=O)Nc3ccc(F)cc3)C(=O)N(C2=S)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J16 compound treatment 200.0 -1080.0 -0.38 280.0 -404.0 -0.31 -0.4895 -0.9946 1548968 ChemDiv3_004790 CCn1c2ccccc2c3cc(NC(=O)CCC4CCCCC4)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J17 compound treatment 360.0 -918.0 -0.33 360.0 -324.0 -0.25 -0.4059 -0.9911 3024969 ChemDiv3_004791 COc1ccccc1C(=O)n2nc(C)cc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J18 compound treatment 360.0 -918.0 -0.33 280.0 -404.0 -0.31 -0.4493 -0.9997 3119114 ChemDiv3_004792 Cc1cccc(c1)n2c(=O)c3c4CCCCc4sc3n5c(S)nnc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J19 compound treatment 5240.0 3960.0 1.41 400.0 -284.0 -0.22 0.8399 0.5905 3024970 ChemDiv3_004793 CC1(C)CC(C)(c2ccc(Cl)cc2)c3ccccc3N1C(=O)c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J20 compound treatment 1040.0 -238.0 -0.08 1160.0 476.0 0.37 0.199 0.5303 3119115 ChemDiv3_004794 O=c1/c(=C/c2ccccc2)/sc3nc(nn13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J21 compound treatment 3640.0 2360.0 0.84 320.0 -364.0 -0.28 0.3952 0.4473 3024971 ChemDiv3_004795 Cc1ccc(/N=C(\N)/Nc2nc(=O)cc(C)[nH]2)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J22 compound treatment 520.0 -758.0 -0.27 240.0 -444.0 -0.34 -0.4309 -0.9931 3119116 ChemDiv3_004796 CCCN1C(=O)/C(=c/2\sc3nc(=O)c(nn3c2=O)c4ccccc4)/c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J23 mock treatment 240.0 -1040.0 -0.37 200.0 -484.0 -0.37 -0.5229 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 J24 mock treatment 6680.0 5400.0 1.92 240.0 -444.0 -0.34 1.1143 0.5724 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K01 compound treatment 1880.0 603.0 0.21 760.0 76.3 0.06 0.1925 0.8688 1870397 ChemDiv3_004797 COc1ccc(cc1)c2coc3c(C)c4oc(=O)c5cc(OC)ccc5c4cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K02 compound treatment 440.0 -838.0 -0.3 6240.0 5560.0 4.27 2.8062 0.6563 3119117 ChemDiv3_004798 COc1ccc(cc1)c2nc3c4cnn(c5cccc(C)c5)c4ncn3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K03 compound treatment 600.0 -678.0 -0.24 520.0 -164.0 -0.13 -0.2588 -0.9543 1862416 ChemDiv3_004799 CCCCC(=O)Nc1ccc2oc(nc2c1)c3ccc(O)c(Br)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K04 compound treatment 1440.0 163.0 0.06 720.0 36.3 0.03 0.0604 0.9442 3024972 ChemDiv3_004800 CCSc1nc2sc3CCCCc3c2c4nnc(S)n14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K05 compound treatment 1760.0 483.0 0.17 600.0 -83.8 -0.06 0.0756 0.4133 3119118 ChemDiv3_004801 Oc1ccccc1Oc2c(F)c(F)nc(N3CCCC3)c2F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K06 compound treatment 560.0 -718.0 -0.25 360.0 -324.0 -0.25 -0.3557 -0.9999 3024973 ChemDiv3_004802 Cc1ccccc1OCCn2cc(/C(=N/O)/N)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K07 compound treatment 1400.0 123.0 0.04 320.0 -364.0 -0.28 -0.1667 -0.59 3119119 ChemDiv3_004803 O=C1CCC(=O)N1c2nc3NC(=O)CC(c4ccccc4)n3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K08 compound treatment 920.0 -358.0 -0.13 3120.0 2440.0 1.87 1.2329 0.6577 3024974 ChemDiv3_004804 CC1(C)Cc2nc3sc4c(=O)n(CC(=O)c5ccc(Cl)cc5)cnc4c3cc2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K09 compound treatment 600.0 -678.0 -0.24 720.0 36.3 0.03 -0.1503 -0.6211 1204823 ChemDiv3_004805 COc1ccc(CNC(=O)NC(C)(C)c2cccc(c2)C(=C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K10 compound treatment 560.0 -718.0 -0.25 440.0 -244.0 -0.19 -0.3123 -0.9886 3119120 ChemDiv3_004806 CCCC(=O)Nc1ccc(cc1)c2nc3cc4ccccc4cc3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K11 compound treatment 640.0 -638.0 -0.23 240.0 -444.0 -0.34 -0.4008 -0.9802 3024127 ChemDiv3_004807 CCOc1nc(NCC=C)nc(Nc2ccc(cc2)c3nc4ccccc4o3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K12 compound treatment 1480.0 203.0 0.07 880.0 196.0 0.15 0.1573 0.9426 1545881 ChemDiv3_004808 Cn1ccnc1SCC(=O)Nc2cccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K13 compound treatment 440.0 -838.0 -0.3 440.0 -244.0 -0.19 -0.3424 -0.9752 1325413 ChemDiv3_004809 C=CCNC(=S)N1CCN(CC1)C(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K14 compound treatment 1160.0 -118.0 -0.04 1160.0 476.0 0.37 0.2291 0.6225 3119121 ChemDiv3_004810 CC(CNCc1ccc2OCOc2c1)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K15 compound treatment 640.0 -638.0 -0.23 840.0 156.0 0.12 -0.0751 -0.2933 3119122 ChemDiv3_004811 CCOc1ccc(cc1)c2nnc(N3CCCCC3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K16 compound treatment 1600.0 323.0 0.11 600.0 -83.8 -0.06 0.0354 0.27 3024128 ChemDiv3_004812 CC(C)N1C(=O)S/C(=C/c2cc(Br)c(OCC(=O)O)c(Br)c2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K17 compound treatment 2600.0 1320.0 0.47 600.0 -83.8 -0.06 0.2863 0.6045 3119123 ChemDiv3_004813 CCNS(=O)(=O)c1cc(ccc1C)c2nn(C)c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K18 compound treatment 760.0 -518.0 -0.18 360.0 -324.0 -0.25 -0.3056 -0.9889 3024129 ChemDiv3_004814 CC(CC(=O)O)CC(=O)Nc1cccc(c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K19 compound treatment 960.0 -318.0 -0.11 4320.0 3640.0 2.79 1.8943 0.678 3119124 ChemDiv3_004815 O=C1CS/C(=N\c2ccccc2)/N1S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K20 compound treatment 960.0 -318.0 -0.11 880.0 196.0 0.15 0.0269 0.143 3024130 ChemDiv3_004816 CN(CCOC(=O)C1c2ccccc2Oc3ccccc13)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K21 compound treatment 800.0 -478.0 -0.17 400.0 -284.0 -0.22 -0.2738 -0.9923 1215426 ChemDiv3_004817 CC(C)CCNc1nnnc2c1sc3nc(N4CCOCC4)c5CCCCc5c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K22 compound treatment 960.0 -318.0 -0.11 600.0 -83.8 -0.06 -0.1251 -0.9646 3119125 ChemDiv3_004818 Cc1nn(C(=O)CNC(=O)c2ccccc2)c(C)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K23 mock treatment 920.0 -358.0 -0.13 520.0 -164.0 -0.13 -0.1786 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 K24 mock treatment 1000.0 -278.0 -0.1 640.0 -43.8 -0.03 -0.0934 -0.8976 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L01 compound treatment 920.0 -358.0 -0.13 960.0 276.0 0.21 0.0603 0.244 1529468 ChemDiv3_004819 CC(C)Oc1ccc(cc1)C(=O)NC(CC(=O)O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L02 compound treatment 5680.0 4400.0 1.56 720.0 36.3 0.03 1.124 0.7196 1439481 ChemDiv3_004820 CCOc1ccc(cc1)C2=C(CN3CCOCC3)C(c4ccccc4)c5ccccc5O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L03 compound treatment 960.0 -318.0 -0.11 3520.0 2840.0 2.18 1.46 0.6696 1562687 ChemDiv3_004821 CC(C)COc1ccc(cc1)C(CC(=O)O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L04 compound treatment 720.0 -558.0 -0.2 360.0 -324.0 -0.25 -0.3156 -0.9936 3119126 ChemDiv3_004822 FC(F)(F)c1oc2cc(OC(=O)c3ccco3)ccc2c(=O)c1c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L05 compound treatment 680.0 -598.0 -0.21 480.0 -204.0 -0.16 -0.2605 -0.9888 3119127 ChemDiv3_004823 Cc1ccc2n3CCN(C/C(=N/O)/c4ccc(Br)cc4)C5CCCc(c53)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L06 compound treatment 400.0 -878.0 -0.31 360.0 -324.0 -0.25 -0.3959 -0.9938 1360838 ChemDiv3_004824 CC(C)c1cc(C(C)C)c(c(c1)C(C)C)S(=O)(=O)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L07 compound treatment 640.0 -638.0 -0.23 560.0 -124.0 -0.1 -0.2271 -0.9258 3119128 ChemDiv3_004825 CC/1=NN(C(=O)\C1=C\Nc2ccc(cc2)S(=O)(=O)NC(=N)N)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L08 compound treatment 2800.0 1520.0 0.54 480.0 -204.0 -0.16 0.2713 0.4825 3024131 ChemDiv3_004826 Cc1[nH]c2ccccc2c1/C=C/3\SC(=O)N(C3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L09 compound treatment 680.0 -598.0 -0.21 520.0 -164.0 -0.13 -0.2388 -0.9689 3119129 ChemDiv3_004827 Cc1ccc(NC2=C/C(=N/S(=O)(=O)c3ccc(F)cc3)/c4ccccc4C2=O)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L10 compound treatment 440.0 -838.0 -0.3 240.0 -444.0 -0.34 -0.451 -0.9977 3024132 ChemDiv3_004828 N=c1c(cc2c(=O)n3ccccc3nc2n1Cc4ccco4)S(=O)(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L11 compound treatment 600.0 -678.0 -0.24 1440.0 756.0 0.58 0.2406 0.3829 1694361 ChemDiv3_004829 CCC(C)(C)C1CCc2oc3ccc(NS(=O)(=O)c4cccs4)cc3c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L12 compound treatment 7800.0 6520.0 2.31 2400.0 1720.0 1.32 2.5678 0.9644 1919128 ChemDiv3_004830 O=C1NN=C(CC1c2c[nH]c3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L13 compound treatment 960.0 -318.0 -0.11 640.0 -43.8 -0.03 -0.1034 -0.8797 3119254 ChemDiv3_004831 COc1ccc(cc1)C2SCCN2C(=S)Nc3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L14 compound treatment 360.0 -918.0 -0.33 480.0 -204.0 -0.16 -0.3408 -0.9436 3024133 ChemDiv3_004832 COC(=O)C/1=C(C)N(C(=O)\C1=C/c2cccs2)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L15 compound treatment 800.0 -478.0 -0.17 320.0 -364.0 -0.28 -0.3172 -0.9713 1223261 ChemDiv3_004833 CCOc1ccc(NC(=O)CC2N(CCc3ccccc3)C(=S)N(C)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L16 compound treatment 1040.0 -238.0 -0.08 600.0 -83.8 -0.06 -0.105 -0.9911 3024134 ChemDiv3_004834 COc1cc2c(cc1NC(=O)CC(C)(C)C)oc3ccccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L17 compound treatment 640.0 -638.0 -0.23 1920.0 1240.0 0.95 0.5112 0.5239 1674175 ChemDiv3_004835 O=C(Cn1c2ccccc2c3ccccc13)Sc4nc5ccccc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L18 compound treatment 1360.0 82.5 0.03 680.0 -3.75 0.0 0.0187 0.6345 3024135 ChemDiv3_004836 COCc1nnc(NS(=O)(=O)c2ccc(OC)cc2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L19 compound treatment 3120.0 1840.0 0.65 2760.0 2080.0 1.59 1.5893 0.9225 3024136 ChemDiv3_004837 Cc1cc(C)n(n1)C(=O)c2ccncc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L20 compound treatment 560.0 -718.0 -0.25 6040.0 5360.0 4.11 2.7277 0.6621 3119255 ChemDiv3_004838 CCN(CC)c1ccc(/C=c/2\sc3ncnn3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L21 compound treatment 1800.0 523.0 0.19 1240.0 556.0 0.43 0.433 0.9302 3119256 ChemDiv3_004839 Cc1ccc(cc1)c2nnc(SC3CC(=O)N(C3=O)c4ccccc4)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L22 compound treatment 640.0 -638.0 -0.23 600.0 -83.8 -0.06 -0.2054 -0.8735 1250836 ChemDiv3_004840 CC(Sc1ccccn1)C(=O)Nc2ccc(cc2)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L23 mock treatment 1200.0 -77.5 -0.03 1200.0 516.0 0.4 0.2608 0.6565 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 L24 mock treatment 1560.0 283.0 0.1 960.0 276.0 0.21 0.2208 0.9414 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M01 compound treatment 360.0 -918.0 -0.33 1240.0 556.0 0.43 0.0718 0.1338 1870017 ChemDiv3_004841 COc1ccc2c(c1)c(=O)oc3c(C)c4occ(C)c4cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M02 compound treatment 5120.0 3840.0 1.36 1400.0 716.0 0.55 1.3527 0.9203 3024137 ChemDiv3_004842 Cc1cccc(c1)n2ncc3c4nc(COc5c(C)cccc5C)nn4cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M03 compound treatment 360.0 -918.0 -0.33 640.0 -43.8 -0.03 -0.2539 -0.776 3119257 ChemDiv3_004843 COc1ccc(Oc2c(F)c(F)nc(F)c2Cl)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M04 compound treatment 1280.0 2.5 0.0 280.0 -404.0 -0.31 -0.2186 -0.7051 1696007 ChemDiv3_004844 CC(C)CCOc1ccc(cc1)C(=O)C(CN2CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M05 compound treatment 440.0 -838.0 -0.3 440.0 -244.0 -0.19 -0.3424 -0.9752 3024138 ChemDiv3_004845 O=C1c2ccccc2-c3n[nH]c(=O)c4ccc(NC5CCCCC5)c1c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M06 compound treatment 880.0 -398.0 -0.14 920.0 236.0 0.18 0.0285 0.1242 3119258 ChemDiv3_004846 N/C(=N\O)/c1cn(CCOc2ccccc2Cl)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M07 compound treatment 400.0 -878.0 -0.31 2000.0 1320.0 1.01 0.4944 0.4676 3024190 ChemDiv3_004847 O=C(Nc1nc2NC(=O)CC(c3ccccc3)n2n1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M08 compound treatment 400.0 -878.0 -0.31 1040.0 356.0 0.27 -0.0267 -0.0645 3119259 ChemDiv3_004848 Cc1ccc(cc1)S(=O)(=O)/N=C(\NC2CCCCC2)/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M09 compound treatment 960.0 -318.0 -0.11 320.0 -364.0 -0.28 -0.2771 -0.9203 1477219 ChemDiv3_004849 CC(=C)c1cccc(c1)C(C)(C)NC(=O)NCCc2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M10 compound treatment 6880.0 5600.0 1.99 320.0 -364.0 -0.28 1.2079 0.6018 1248399 ChemDiv3_004850 CCC(C)c1ccc(O)c(NC(=O)c2cccnc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M11 compound treatment 440.0 -838.0 -0.3 400.0 -284.0 -0.22 -0.3641 -0.9884 3119260 ChemDiv3_004851 C=CCNc1nc(Nc2ccc(cc2)c3nc4ccccc4o3)nc(n1)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M12 compound treatment 480.0 -798.0 -0.28 320.0 -364.0 -0.28 -0.3975 -1.0 3024191 ChemDiv3_004852 CS(=O)(=O)CCC(N1C(=O)c2ccccc2C1=O)C(=O)n3nnc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M13 compound treatment 320.0 -958.0 -0.34 360.0 -324.0 -0.25 -0.4159 -0.9882 3119261 ChemDiv3_004853 CCC(=O)Nc1ccccc1C(=O)OCC(=O)Nc2ccc(cc2)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M14 compound treatment 760.0 -518.0 -0.18 440.0 -244.0 -0.19 -0.2621 -1.0 1631121 ChemDiv3_004854 O=C(NCCC1=CCCCC1)c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M15 compound treatment 720.0 -558.0 -0.2 1320.0 636.0 0.49 0.2055 0.3901 3119262 ChemDiv3_004855 CCOc1ccc(cc1)c2nnc(Nc3ccc(OC)cc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M16 compound treatment 360.0 -918.0 -0.33 400.0 -284.0 -0.22 -0.3842 -0.9809 3119263 ChemDiv3_004856 COC(=O)CN1C(=O)S/C(=C/c2ccc(o2)c3ccc(cc3)C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M17 compound treatment 1240.0 -37.5 -0.01 480.0 -204.0 -0.16 -0.12 -0.7645 3024192 ChemDiv3_004857 Cc1ccc(OCC(=O)Nc2cc(ccc2N3CCOCC3)c4nn(C)c(=O)c5ccccc45)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M18 compound treatment 400.0 -878.0 -0.31 560.0 -124.0 -0.1 -0.2873 -0.8827 3119264 ChemDiv3_004858 CC(C)NC(=O)/C(=N\O)/c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M19 compound treatment 2200.0 923.0 0.33 1040.0 356.0 0.27 0.4248 0.996 3119265 ChemDiv3_004859 COC(=O)/C=C/1\S/C(=N\S(=O)(=O)c2ccccc2)/N(C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M20 compound treatment 320.0 -958.0 -0.34 1200.0 516.0 0.4 0.0401 0.0768 1222873 ChemDiv3_004860 O=C(Nc1nc2ccccc2s1)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M21 compound treatment 280.0 -998.0 -0.35 320.0 -364.0 -0.28 -0.4477 -0.9931 3119266 ChemDiv3_004861 C=CCSc1ncnc2c1sc3nc(N4CCOCC4)c5CCCCc5c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M22 compound treatment 400.0 -878.0 -0.31 720.0 36.3 0.03 -0.2004 -0.6413 1867990 ChemDiv3_004862 CC1CC(c2ccccc2)c3cc(C)ccc3N1C(=O)c4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M23 mock treatment 560.0 -718.0 -0.25 1280.0 596.0 0.46 0.1437 0.2744 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 M24 mock treatment 1000.0 -278.0 -0.1 3360.0 2680.0 2.05 1.3832 0.6725 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N01 compound treatment 440.0 -838.0 -0.3 480.0 -204.0 -0.16 -0.3207 -0.9551 3024156 ChemDiv3_004863 CCOc1ccc(cc1)C(N)CC(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N02 compound treatment 440.0 -838.0 -0.3 360.0 -324.0 -0.25 -0.3858 -0.9961 1357341 ChemDiv3_004864 CCOc1ccc(cc1)C2=C(CN(C)C)C(c3ccc(F)cc3)c4ccccc4O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N03 compound treatment 720.0 -558.0 -0.2 400.0 -284.0 -0.22 -0.2939 -0.9988 1466560 ChemDiv3_004865 CC[N+]1(CC)Cc2cc3ccccc3cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N04 compound treatment 760.0 -518.0 -0.18 960.0 276.0 0.21 0.0202 0.0718 3024160 ChemDiv3_004866 CCOc1ccc(/C=C/C(=O)Nc2nc(c(C)s2)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N05 compound treatment 680.0 -598.0 -0.21 960.0 276.0 0.21 1.0E-4 3.0E-4 3024162 ChemDiv3_004867 CCOC(=O)/C=C/1\CCCCCN1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N06 compound treatment 360.0 -918.0 -0.33 880.0 196.0 0.15 -0.1236 -0.3447 3119267 ChemDiv3_004868 CCCC1(CC(CSC(=N)N)OC1=O)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N07 compound treatment 5240.0 3960.0 1.41 760.0 76.3 0.06 1.0354 0.7359 3119268 ChemDiv3_004869 Cc1ccc(c(C)c1)S(=O)(=O)/N=C/2\C=CC(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N08 compound treatment 1120.0 -158.0 -0.06 840.0 156.0 0.12 0.0453 0.3424 3024166 ChemDiv3_004870 CCc1ccc(cc1)N2C(=O)/C(=C/c3cccn3C(C)(C)C)/C(=O)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N09 compound treatment 840.0 -438.0 -0.16 280.0 -404.0 -0.31 -0.3289 -0.9489 1207988 ChemDiv3_004871 CC(C)c1ccc(cc1)S(=O)(=O)Nc2cc(SCC(=O)O)c(O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N10 compound treatment 480.0 -798.0 -0.28 400.0 -284.0 -0.22 -0.3541 -0.9917 1875255 ChemDiv3_004872 CCn1c(=N)c(cc2c(=O)n3ccccc3nc12)S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N11 compound treatment 320.0 -958.0 -0.34 360.0 -324.0 -0.25 -0.4159 -0.9882 1240844 ChemDiv3_004873 Clc1ccc(NC(=O)CSC2CC(=O)N(C2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N12 compound treatment 560.0 -718.0 -0.25 360.0 -324.0 -0.25 -0.3557 -0.9999 3119269 ChemDiv3_004874 CCSC1=N/C(=C\c2cc3OCOc3cc2Br)/C(=O)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N13 compound treatment 520.0 -758.0 -0.27 320.0 -364.0 -0.28 -0.3875 -0.9998 3119270 ChemDiv3_004875 CCOC(=O)c1ccc(/N=C/2\SC(CC(=O)N2Cc3cccs3)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N14 compound treatment 440.0 -838.0 -0.3 800.0 116.0 0.09 -0.147 -0.4738 3024171 ChemDiv3_004876 FC(F)(F)c1ccc(/C=C\2/NC(=O)N(C2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N15 compound treatment 320.0 -958.0 -0.34 480.0 -204.0 -0.16 -0.3508 -0.9381 1264989 ChemDiv3_004877 CN1C(=O)C(CC(=O)Nc2ccc(F)cc2)N(Cc3ccccc3)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N16 compound treatment 1080.0 -198.0 -0.07 640.0 -43.8 -0.03 -0.0733 -0.9433 3024216 ChemDiv3_004878 CC(C)C1Cc2c(CO1)sc3[nH]c(=S)n(Cc4ccccc4)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N17 compound treatment 880.0 -398.0 -0.14 400.0 -284.0 -0.22 -0.2537 -0.9778 3119271 ChemDiv3_004879 COC(=O)/C=C/1\SC(=NC1=O)NC(=O)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N18 compound treatment 520.0 -758.0 -0.27 440.0 -244.0 -0.19 -0.3223 -0.9844 3119272 ChemDiv3_004880 CC1CCN(CC1)S(=O)(=O)c2ccc(NC(=O)c3c(C)onc3c4ccccc4Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N19 compound treatment 760.0 -518.0 -0.18 640.0 -43.8 -0.03 -0.1536 -0.8228 1733561 ChemDiv3_004881 COc1cc(OC)cc(c1)C(=O)n2nc(C)cc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N20 compound treatment 960.0 -318.0 -0.11 560.0 -124.0 -0.1 -0.1468 -0.9964 3024219 ChemDiv3_004882 Cc1ccc(/C=c/2\sc3ncnn3c2=O)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N21 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3119398 ChemDiv3_004883 CCSc1nc(C)c2cc(OC)ccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N22 compound treatment 800.0 -478.0 -0.17 520.0 -164.0 -0.13 -0.2087 -0.9892 3024221 ChemDiv3_004884 CC(Sc1nc(=O)cc(N)n1CC=C)C(=O)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N23 mock treatment 480.0 -798.0 -0.28 760.0 76.3 0.06 -0.1587 -0.5492 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 N24 mock treatment 800.0 -478.0 -0.17 1040.0 356.0 0.27 0.0736 0.2288 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O01 compound treatment 240.0 -1040.0 -0.37 400.0 -284.0 -0.22 -0.4143 -0.9687 3119399 ChemDiv3_004885 CCc1cc(=O)oc2cc(C)c3c(coc3c12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O02 compound treatment 360.0 -918.0 -0.33 320.0 -364.0 -0.28 -0.4276 -0.9971 3119400 ChemDiv3_004886 Cc1cc(NCCN2CCCCC2)c3ccc4ccccc4c3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O03 compound treatment 200.0 -1080.0 -0.38 280.0 -404.0 -0.31 -0.4895 -0.9946 3024223 ChemDiv3_004887 Fc1nc(N2CCOCC2)c(F)c(Oc3ccc4C(=O)CCC(c5ccccc5)c4c3)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O04 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 3119401 ChemDiv3_004888 C[n+]1ccc(/C=C/c2ccc3OCOc3c2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O05 compound treatment 200.0 -1080.0 -0.38 200.0 -484.0 -0.37 -0.5329 -0.9999 3119402 ChemDiv3_004889 Fc1nc(N2CCOCC2)c3Oc4ccccc4Oc3c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O06 compound treatment 160.0 -1120.0 -0.4 1680.0 996.0 0.76 0.2605 0.3024 3024226 ChemDiv3_004890 CN1CCc2c(C1)sc3NC(/C=C/c4ccco4)N=C(O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O07 compound treatment 280.0 -998.0 -0.35 360.0 -324.0 -0.25 -0.426 -0.9851 3119403 ChemDiv3_004891 O=C1CC(c2ccccc2)n3nc(NS(=O)(=O)c4ccccc4)nc3N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O08 compound treatment 280.0 -998.0 -0.35 320.0 -364.0 -0.28 -0.4477 -0.9931 3119404 ChemDiv3_004892 CC(=O)Nc1ccc(NC(=O)[C@@H]2CCCC[C@@H]2C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O09 compound treatment 360.0 -918.0 -0.33 400.0 -284.0 -0.22 -0.3842 -0.9809 1275727 ChemDiv3_004893 CC(=C)c1cccc(c1)C(C)(C)NC(=O)NC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O10 compound treatment 320.0 -958.0 -0.34 360.0 -324.0 -0.25 -0.4159 -0.9882 3024270 ChemDiv3_004894 CC1Cc2cc(/C=C/3\N=C(OC3=O)c4ccccc4F)ccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O11 compound treatment 280.0 -998.0 -0.35 240.0 -444.0 -0.34 -0.4911 -0.9998 3119405 ChemDiv3_004895 COc1ccc(CCNc2nc(Nc3ccc(Cl)cc3)nc(OC)n2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O12 compound treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 1378371 ChemDiv3_004896 OC(=O)Cn1c(=O)oc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O13 compound treatment 320.0 -958.0 -0.34 200.0 -484.0 -0.37 -0.5028 -0.999 3119406 ChemDiv3_004897 CCOC(=O)c1ccc(NC(=O)CSC2=NC(=O)C(CC)C(=O)N2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O14 compound treatment 360.0 -918.0 -0.33 1400.0 716.0 0.55 0.1587 0.2483 3024272 ChemDiv3_004898 CCS(=O)(=O)c1ccc2OC(=O)/C(=C\C(=O)c3oc(C)nc3C)/Nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O15 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 3119407 ChemDiv3_004899 CCOc1ccc(cc1)c2n[nH]c(=S)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O16 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3119408 ChemDiv3_004900 CC(C)N1C(=O)S/C(=C/c2ccccc2OCc3ccc(cc3)C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O17 compound treatment 360.0 -918.0 -0.33 360.0 -324.0 -0.25 -0.4059 -0.9911 3024275 ChemDiv3_004901 CN(C1=NC(=O)/C(=C\c2ccccc2Cl)/S1)c3ccc(O)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O18 compound treatment 280.0 -998.0 -0.35 320.0 -364.0 -0.28 -0.4477 -0.9931 3024277 ChemDiv3_004902 CCNC(=O)/C(=N\O)/c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O19 compound treatment 360.0 -918.0 -0.33 360.0 -324.0 -0.25 -0.4059 -0.9911 3119409 ChemDiv3_004903 CC1N(CCc2c1[nH]c3ccccc23)C(=S)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O20 compound treatment 360.0 -918.0 -0.33 200.0 -484.0 -0.37 -0.4928 -0.9978 3119410 ChemDiv3_004904 O=C(C1c2ccccc2Oc3ccccc13)N4CCC(C4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O21 compound treatment 320.0 -958.0 -0.34 320.0 -364.0 -0.28 -0.4376 -0.9953 3024279 ChemDiv3_004905 Cc1nc(SCCOc2ccccc2)sc1C(=O)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O22 compound treatment 280.0 -998.0 -0.35 200.0 -484.0 -0.37 -0.5128 -0.9997 3119411 ChemDiv3_004906 C1N(N2CN(N1C2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O23 mock treatment 240.0 -1040.0 -0.37 200.0 -484.0 -0.37 -0.5229 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 O24 mock treatment 440.0 -838.0 -0.3 320.0 -364.0 -0.28 -0.4075 -0.9995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P01 compound treatment 200.0 -1080.0 -0.38 280.0 -404.0 -0.31 -0.4895 -0.9946 1204591 ChemDiv3_004907 NC(=O)c1ccc(cc1)c2nnc(o2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P02 compound treatment 320.0 -958.0 -0.34 240.0 -444.0 -0.34 -0.4811 -1.0 3119412 ChemDiv3_004908 CCC(O)C1=C(Oc2ccccc2C1c3ccccc3C)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P03 compound treatment 240.0 -1040.0 -0.37 600.0 -83.8 -0.06 -0.3057 -0.8182 1620080 ChemDiv3_004909 CC[N+](C)(CC)Cc1cc2ccccc2c3COCc31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P04 compound treatment 360.0 -918.0 -0.33 240.0 -444.0 -0.34 -0.471 -0.9997 3119413 ChemDiv3_004910 Clc1ccc(cc1)c2csc3nc[nH]c(=S)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P05 compound treatment 360.0 -918.0 -0.33 280.0 -404.0 -0.31 -0.4493 -0.9997 3119414 ChemDiv3_004911 CCCCC1(CC)C(=O)NC(=O)N=C1Nc2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P06 compound treatment 400.0 -878.0 -0.31 360.0 -324.0 -0.25 -0.3959 -0.9938 3119415 ChemDiv3_004912 CCC1CCCCN1S(=O)(=O)c2ccc(NC(=O)COc3ccc(OC)cc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P07 compound treatment 5480.0 4200.0 1.49 6080.0 5400.0 4.14 3.9836 0.9048 3024336 ChemDiv3_004913 CCc1ccc(cc1)S(=O)(=O)/N=C/2\C=CC(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P08 compound treatment 320.0 -958.0 -0.34 400.0 -284.0 -0.22 -0.3942 -0.9769 3119416 ChemDiv3_004914 COC(=O)CN1C(=O)S/C(=C/c2cn(CC=C)c3ccccc23)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P09 compound treatment 240.0 -1040.0 -0.37 240.0 -444.0 -0.34 -0.5011 -0.9993 1330391 ChemDiv3_004915 O=C(N(c1ccc2oc3CCCCc3c2c1)S(=O)(=O)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P10 compound treatment 240.0 -1040.0 -0.37 160.0 -524.0 -0.4 -0.5446 -0.999 3119417 ChemDiv3_004916 N=c1c(cc2c(=O)n3ccccc3nc2n1C4CCCC4)S(=O)(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P11 compound treatment 280.0 -998.0 -0.35 240.0 -444.0 -0.34 -0.4911 -0.9998 1651800 ChemDiv3_004917 CC(=O)N(CCc1ccccc1)C2CC(=O)N(C2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P12 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3024341 ChemDiv3_004918 CCSC1=N/C(=C\c2ccc(Br)s2)/C(=O)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P13 compound treatment 200.0 -1080.0 -0.38 160.0 -524.0 -0.4 -0.5546 -0.9997 3119418 ChemDiv3_004919 CNC(=O)CC1N(NC(=O)c2cccc(F)c2)C(=S)N(C1=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P14 compound treatment 400.0 -878.0 -0.31 160.0 -524.0 -0.4 -0.5044 -0.992 3024342 ChemDiv3_004920 COc1cccc(/C=C\2/NC(=O)N(C2=O)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P15 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 1153500 ChemDiv3_004921 CC1CC(Nc2ccccc2)c3ccccc3N1C(=O)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P16 compound treatment 320.0 -958.0 -0.34 280.0 -404.0 -0.31 -0.4594 -0.999 3024345 ChemDiv3_004922 CCOC(=O)c1c(NC(=S)Nc2ccc(OC)cc2)sc3COC(Cc13)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P17 compound treatment 280.0 -998.0 -0.35 280.0 -404.0 -0.31 -0.4694 -0.9978 3119419 ChemDiv3_004923 COC(=O)/C=C/1\SC(=NC1=O)NC(=O)c2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P18 compound treatment 320.0 -958.0 -0.34 280.0 -404.0 -0.31 -0.4594 -0.999 3119420 ChemDiv3_004924 CC(C)c1nnc(NC(=O)C2c3ccccc3Oc4ccccc24)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P19 compound treatment 200.0 -1080.0 -0.38 280.0 -404.0 -0.31 -0.4895 -0.9946 3024347 ChemDiv3_004925 CC1=CC(C)(C)N(C(=O)Nc2ccc(C)cc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P20 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 3119421 ChemDiv3_004926 CCc1ccc(/C=c/2\sc3nc(nn3c2=O)C4COc5ccccc5O4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P21 compound treatment 240.0 -1040.0 -0.37 280.0 -404.0 -0.31 -0.4794 -0.9964 1871084 ChemDiv3_004927 CC(N1C(=O)c2ccccc2C1=O)C(=O)N3CCN(CC3)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P22 compound treatment 200.0 -1080.0 -0.38 280.0 -404.0 -0.31 -0.4895 -0.9946 3119422 ChemDiv3_004928 CCc1ccc(NC2SC(=O)N(C2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P23 mock treatment 320.0 -958.0 -0.34 320.0 -364.0 -0.28 -0.4376 -0.9953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2014 P24 mock treatment 240.0 -1040.0 -0.37 320.0 -364.0 -0.28 -0.4577 -0.9907 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A01 compound treatment 280.0 -324.0 -0.11 400.0 -348.0 -0.27 -0.2702 -0.9288 3119423 ChemDiv3_004929 COc1cc(cc(OC)c1OC)C(=O)/C=C/Nc2ccc(cc2)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A02 compound treatment 240.0 -364.0 -0.13 3600.0 2850.0 2.19 1.4569 0.6643 3024419 ChemDiv3_004930 OC(=O)c1ccc(NC(=O)CCCN2C(=O)S/C(=C\C=C\c3ccccc3)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A03 compound treatment 280.0 -324.0 -0.11 360.0 -388.0 -0.3 -0.2919 -0.9141 3119424 ChemDiv3_004931 Cc1ccc(cc1C)n2nc(C(=O)O)c(C)c(C#N)c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A04 compound treatment 240.0 -364.0 -0.13 280.0 -468.0 -0.36 -0.3454 -0.9045 3119563 ChemDiv3_004932 CC1(C)C2CCC1(C)C(C2)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A05 compound treatment 600.0 -3.75 0.0 280.0 -468.0 -0.36 -0.2551 -0.7097 3024422 ChemDiv3_004933 COc1ccc2-c3nc(/N=C/c4ccc(C)cc4)sc3CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A06 compound treatment 320.0 -284.0 -0.1 360.0 -388.0 -0.3 -0.2819 -0.8962 3119564 ChemDiv3_004934 COc1ccc(cc1)C2NC(C(C)C(O)(Cc3ccccc3)C2C)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A07 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 3024425 ChemDiv3_004935 CC1(C)COC(=N1)Nc2cccc(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A08 compound treatment 280.0 -324.0 -0.11 320.0 -428.0 -0.33 -0.3136 -0.9008 1195009 ChemDiv3_004936 COc1ccc(cc1)c2cc(=O)c3cc(OC(=O)c4ccc(OC)c(OC)c4)ccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A09 compound treatment 320.0 -284.0 -0.1 360.0 -388.0 -0.3 -0.2819 -0.8962 3024428 ChemDiv3_004937 CC(C)(C)C(=O)NC(=S)Nc1ccc2C(=O)OCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A10 compound treatment 280.0 -324.0 -0.11 360.0 -388.0 -0.3 -0.2919 -0.9141 3119565 ChemDiv3_004938 CCOC(=O)c1cnc2c(cccc2c1N3CCN(C)CC3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A11 compound treatment 280.0 -324.0 -0.11 800.0 51.9 0.04 -0.0531 -0.4365 3024430 ChemDiv3_004939 CCOc1ccc(/C=C/2\N(CC(=O)OC)C(=S)N(C)C2=O)c(OCC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A12 compound treatment 360.0 -244.0 -0.09 3200.0 2450.0 1.88 1.2699 0.6739 3119566 ChemDiv3_004940 COC(=O)c1sc(c(C(=O)OC)c1C)S(=O)(=O)NC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A13 compound treatment 1880.0 1280.0 0.45 320.0 -428.0 -0.33 0.0877 0.1568 3024433 ChemDiv3_004941 COC(=O)c1cc2c(=O)n3ccccc3nc2n(C(C)C)c1=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A14 compound treatment 280.0 -324.0 -0.11 1120.0 372.0 0.29 0.1207 0.3921 3119567 ChemDiv3_004942 COc1cc(/C=C/C(=O)\C=C\c2ccc(cc2)N(C)C)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A15 compound treatment 320.0 -284.0 -0.1 3000.0 2250.0 1.73 1.1513 0.6648 1280049 ChemDiv3_004943 CC1(C)CC(=O)C(C(=S)Nc2ccccc2)C(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A16 compound treatment 480.0 -124.0 -0.04 280.0 -468.0 -0.36 -0.2852 -0.7876 3119568 ChemDiv3_004944 S=C1NCN(Cc2ccccc2)CN1CC3CCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A17 compound treatment 200.0 -404.0 -0.14 160.0 -588.0 -0.45 -0.4206 -0.8878 1874490 ChemDiv3_004945 CCC1(C)CC(CCN2C(=O)c3ccccc3C2=O)(CCO1)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A18 compound treatment 400.0 -204.0 -0.07 1640.0 892.0 0.68 0.433 0.629 3119569 ChemDiv3_004946 Cc1sc2ncnc(Oc3cccc(c3)C(F)(F)F)c2c1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A19 compound treatment 200.0 -404.0 -0.14 280.0 -468.0 -0.36 -0.3554 -0.9186 1524496 ChemDiv3_004947 NC(=O)NC(=O)CC1Nc2ccccc2NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A20 compound treatment 360.0 -244.0 -0.09 200.0 -548.0 -0.42 -0.3587 -0.835 1242544 ChemDiv3_004948 OC(=O)c1ccc(Nc2nccc(Nc3ccccc3C(=O)O)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A21 compound treatment 880.0 276.0 0.1 320.0 -428.0 -0.33 -0.1631 -0.4756 3024507 ChemDiv3_004949 CN(C)c1ccc(/C=C\2/N(C(=O)C)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A22 compound treatment 320.0 -284.0 -0.1 1320.0 572.0 0.44 0.2393 0.5312 3119570 ChemDiv3_004950 C=CCNC(=N)SCc1nc2ccccc2c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A23 mock treatment 200.0 -404.0 -0.14 360.0 -388.0 -0.3 -0.312 -0.9436 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 A24 mock treatment 440.0 -164.0 -0.06 320.0 -428.0 -0.33 -0.2735 -0.8194 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B01 compound treatment 400.0 -204.0 -0.07 400.0 -348.0 -0.27 -0.2401 -0.8672 3119571 ChemDiv3_004951 CCOC(=O)C1CCN(CC1)C(=C2C(=O)c3ccccc3C2=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B02 compound treatment 280.0 -324.0 -0.11 2000.0 1250.0 0.96 0.5984 0.6182 3024512 ChemDiv3_004952 CCc1ccc(/C=C/2\N(C)C(=S)N(C3CCCCC3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B03 compound treatment 280.0 -324.0 -0.11 680.0 -68.1 -0.05 -0.1182 -0.9366 1481254 ChemDiv3_004953 CCOc1ccc2C(=CC(C)(C)[N+](C)(C)c2c1)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B04 compound treatment 160.0 -444.0 -0.16 320.0 -428.0 -0.33 -0.3437 -0.9432 1385231 ChemDiv3_004954 Cc1nn(S(=O)c2ccc3ccccc3c2)c(C)c1Sc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B05 compound treatment 280.0 -324.0 -0.11 320.0 -428.0 -0.33 -0.3136 -0.9008 1871664 ChemDiv3_004955 Clc1nc(nc(n1)N2CCCc3ccccc23)N4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B06 compound treatment 320.0 -284.0 -0.1 240.0 -508.0 -0.39 -0.347 -0.8613 3119572 ChemDiv3_004956 COc1ccc(NC(=O)CSc2nc(O)cc(=O)n2c3ccccc3OC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B07 compound treatment 320.0 -284.0 -0.1 320.0 -428.0 -0.33 -0.3036 -0.8832 3024517 ChemDiv3_004957 CCOC(=O)C1=C(C)N=C2C(C1c3ccc(Br)cc3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B08 compound treatment 360.0 -244.0 -0.09 360.0 -388.0 -0.3 -0.2719 -0.8762 3119573 ChemDiv3_004958 CCc1ccc2N(C)C(=O)C(NC(=O)C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B09 compound treatment 280.0 -324.0 -0.11 1200.0 452.0 0.35 0.1641 0.449 3119574 ChemDiv3_004959 COC(=O)C/1=C(C)N(C(=O)\C1=C/c2cc(C)n(c2C)c3ccc(F)cc3)c4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B10 compound treatment 360.0 -244.0 -0.09 360.0 -388.0 -0.3 -0.2719 -0.8762 3024588 ChemDiv3_004960 CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)OCCN2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B11 compound treatment 440.0 -164.0 -0.06 5200.0 4450.0 3.42 2.3757 0.695 3024591 ChemDiv3_004961 Fc1cc(/C=C\2/NC(=O)NC2=O)ccc1N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B12 compound treatment 320.0 -284.0 -0.1 560.0 -188.0 -0.14 -0.1733 -0.9844 3119575 ChemDiv3_004962 CN1C(=O)c2ccc(cc2C1=O)c3nc4ccc(Cl)cc4c(=O)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B13 compound treatment 520.0 -83.8 -0.03 280.0 -468.0 -0.36 -0.2751 -0.763 3024594 ChemDiv3_004963 CCOc1cc2OCOc2cc1/C=C\3/NC(=O)N(Cc4ccccc4)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B14 compound treatment 400.0 -204.0 -0.07 480.0 -268.0 -0.21 -0.1967 -0.9014 3119576 ChemDiv3_004964 CCOc1cc2OCOc2cc1/C=C(\C#N)/c3ccc(cc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B15 compound treatment 3440.0 2840.0 1.01 400.0 -348.0 -0.27 0.5225 0.5019 1217444 ChemDiv3_004965 COc1ccc(NCN2C(=O)CCC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B16 compound treatment 680.0 76.3 0.03 320.0 -428.0 -0.33 -0.2133 -0.6467 3119577 ChemDiv3_004966 CCOC(=O)c1nc(NCc2ccccc2)c3ccccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B17 compound treatment 720.0 116.0 0.04 240.0 -508.0 -0.39 -0.2467 -0.6289 1165861 ChemDiv3_004967 Fc1ccc(NC(=O)Nc2ccc3COC(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B18 compound treatment 240.0 -364.0 -0.13 280.0 -468.0 -0.36 -0.3454 -0.9045 3024598 ChemDiv3_004968 CC(C)(C)C(=O)C(=C1Nc2ccccc2N1)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B19 compound treatment 280.0 -324.0 -0.11 400.0 -348.0 -0.27 -0.2702 -0.9288 3024601 ChemDiv3_004969 CC(C)Cn1c(S)nc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B20 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 3119578 ChemDiv3_004970 OC(=O)CCc1ccc(c2ccccc2)n1c3cccc(O)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B21 compound treatment 360.0 -244.0 -0.09 360.0 -388.0 -0.3 -0.2719 -0.8762 3119579 ChemDiv3_004971 Clc1cccc(Cc2cn3cc(nc3s2)c4ccccc4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B22 compound treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 3024603 ChemDiv3_004972 NC(=O)CSc1ccc2ccccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B23 mock treatment 280.0 -324.0 -0.11 720.0 -28.1 -0.02 -0.0965 -0.8257 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 B24 mock treatment 520.0 -83.8 -0.03 280.0 -468.0 -0.36 -0.2751 -0.763 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C01 compound treatment 2120.0 1520.0 0.54 320.0 -428.0 -0.33 0.1479 0.2347 3119580 ChemDiv3_004973 COc1cc(cc(OC)c1OC)C(=O)/C=C/Nc2ccccc2C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C02 compound treatment 720.0 116.0 0.04 280.0 -468.0 -0.36 -0.225 -0.6219 3024606 ChemDiv3_004974 Cc1ccc(NC(=O)/C=C\2/SC(=O)N(CN3CCCCC3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C03 compound treatment 680.0 76.3 0.03 320.0 -428.0 -0.33 -0.2133 -0.6467 1251629 ChemDiv3_004975 COc1ccc(cc1)c2cc3nc(C)cc(C)n3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C04 compound treatment 320.0 -284.0 -0.1 320.0 -428.0 -0.33 -0.3036 -0.8832 3024954 ChemDiv3_004976 CC(NC(CC(=C)C)c1ccco1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C05 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 3119581 ChemDiv3_004977 O=C(Nc1ccccc1)C2CCN(CC2)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C06 compound treatment 280.0 -324.0 -0.11 360.0 -388.0 -0.3 -0.2919 -0.9141 1157212 ChemDiv3_004978 COc1ccccc1NC(=O)CN2c3cccc4cccc(c34)S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C07 compound treatment 920.0 316.0 0.11 240.0 -508.0 -0.39 -0.1965 -0.4841 3119582 ChemDiv3_004979 Cc1cc(C)nc(NC(=O)CSC(=S)N2CCOCC2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C08 compound treatment 360.0 -244.0 -0.09 240.0 -508.0 -0.39 -0.337 -0.8434 3119583 ChemDiv3_004980 COc1ccc(cc1)c2c/c(=N\C(CC(C)C)C(=O)O)/c3cc(C)ccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C09 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3024959 ChemDiv3_004981 O=C(COn1c(=O)n(COC(=O)c2ccccc2)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C10 compound treatment 240.0 -364.0 -0.13 2200.0 1450.0 1.11 0.6969 0.6211 1641003 ChemDiv3_004982 CCOC(=O)c1cnc2ccc(Cl)cc2c1Nc3ccc(cc3)S(=O)(=O)Nc4ncccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C11 compound treatment 1720.0 1120.0 0.4 360.0 -388.0 -0.3 0.0693 0.1398 3024961 ChemDiv3_004983 COC(=O)CN/1C(=S)N(C)C(=O)\C1=C\c2ccc(o2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C12 compound treatment 840.0 236.0 0.08 240.0 -508.0 -0.39 -0.2166 -0.5428 3119584 ChemDiv3_004984 COC(=O)c1sc(c(C(=O)OC)c1C)S(=O)(=O)N2CCN(CC2)c3ccccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C13 compound treatment 3120.0 2520.0 0.89 440.0 -308.0 -0.24 0.4639 0.5024 3024114 ChemDiv3_004985 CCNC(=O)c1cc2c(=O)n3ccccc3nc2n(C(C)C)c1=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C14 compound treatment 2080.0 1480.0 0.52 3240.0 2490.0 1.91 1.723 0.8687 3119715 ChemDiv3_004986 CN(C)c1ccc(/C=C/C(=O)\C=C\c2ccc3OCOc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C15 compound treatment 4560.0 3960.0 1.4 320.0 -428.0 -0.33 0.76 0.5272 3024117 ChemDiv3_004987 CN(C)c1nc(nc(n1)N(CC=C)C#N)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C16 compound treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 3119716 ChemDiv3_004988 S=C1NCN(Cc2ccccc2)CN1Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C17 compound treatment 200.0 -404.0 -0.14 240.0 -508.0 -0.39 -0.3771 -0.9075 1723905 ChemDiv3_004989 COc1ccc(CN(CCC(c2ccco2)c3ccccc3)C(=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C18 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3024121 ChemDiv3_004990 CC(C)C1N(CCCN1S(=O)(=O)c2ccc(C)cc2)/C(=N/S(=O)(=O)c3ccc(C)cc3)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C19 compound treatment 360.0 -244.0 -0.09 240.0 -508.0 -0.39 -0.337 -0.8434 3119717 ChemDiv3_004991 O=S(=O)(C1c2ccccc2Oc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C20 compound treatment 240.0 -364.0 -0.13 240.0 -508.0 -0.39 -0.3671 -0.8934 1300285 ChemDiv3_004992 CC(Sc1cc(C)c2ccccc2n1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C21 compound treatment 480.0 -124.0 -0.04 280.0 -468.0 -0.36 -0.2852 -0.7876 3119718 ChemDiv3_004993 Clc1cccc(N/C=C/2\C(=O)Nc3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C22 compound treatment 360.0 -244.0 -0.09 640.0 -108.0 -0.08 -0.1199 -0.9998 3119719 ChemDiv3_004994 COC(=O)Cc1nn(c(O)c1/C=N/c2ccc(C)cc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C23 mock treatment 400.0 -204.0 -0.07 240.0 -508.0 -0.39 -0.327 -0.8241 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 C24 mock treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D01 compound treatment 3520.0 2920.0 1.03 280.0 -468.0 -0.36 0.4774 0.4359 3024125 ChemDiv3_004995 CC(=C1C(=O)c2ccccc2C1=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D02 compound treatment 400.0 -204.0 -0.07 240.0 -508.0 -0.39 -0.327 -0.8241 3024172 ChemDiv3_004996 CN/1C(=S)N(C2CCCCC2)C(=O)\C1=C\c3cc(C)n(c3C)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D03 compound treatment 280.0 -324.0 -0.11 880.0 132.0 0.1 -0.0096 -0.0629 1532710 ChemDiv3_004997 Cc1ccnc(SCC(=O)N2CCc3ccccc3C2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D04 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3024176 ChemDiv3_004998 Cc1nn(C(=O)c2cc3CCCCc3s2)c(C)c1Sc4ccc(Br)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D05 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 1871526 ChemDiv3_004999 Nc1nc(CSC(=S)N2CCCCC2)nc(Nc3ccccc3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D06 compound treatment 320.0 -284.0 -0.1 320.0 -428.0 -0.33 -0.3036 -0.8832 3119720 ChemDiv3_005000 CCOc1ccccc1n2c(SCC(=O)c3ccc4OCCOc4c3)nc(O)cc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D07 compound treatment 200.0 -404.0 -0.14 360.0 -388.0 -0.3 -0.312 -0.9436 3024181 ChemDiv3_005001 Clc1cccc(c1)C2C3C(=O)c4ccccc4C3=NC5=C2C(=O)CCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D08 compound treatment 320.0 -284.0 -0.1 200.0 -548.0 -0.42 -0.3687 -0.8522 3119721 ChemDiv3_005002 COC(=O)Nc1c(C)nc2n(C)c3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D09 compound treatment 400.0 -204.0 -0.07 240.0 -508.0 -0.39 -0.327 -0.8241 3119722 ChemDiv3_005003 CC/1=NN(C(=O)\C1=C\c2ccc3n(C)c(=O)n(C)c3c2)c4ccc(C)c(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D10 compound treatment 240.0 -364.0 -0.13 440.0 -308.0 -0.24 -0.2585 -0.9594 3024186 ChemDiv3_005004 Clc1ccccc1C(=O)NCCCn2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D11 compound treatment 360.0 -244.0 -0.09 280.0 -468.0 -0.36 -0.3153 -0.8529 3119723 ChemDiv3_005005 Cc1cc(/C=C\2/NC(=O)N(Cc3ccccc3F)C2=O)c(C)n1c4ccc(cc4)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D12 compound treatment 400.0 -204.0 -0.07 320.0 -428.0 -0.33 -0.2835 -0.8425 1402147 ChemDiv3_005006 Cc1c(C)c2ccccc2n1CCc3ccc(C)nc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D13 compound treatment 6000.0 5400.0 1.91 320.0 -428.0 -0.33 1.1212 0.5772 3024189 ChemDiv3_005007 CN1C(=O)/C(=C/c2ccc(Cl)cc2)/N(C)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D14 compound treatment 720.0 116.0 0.04 360.0 -388.0 -0.3 -0.1815 -0.6035 3024228 ChemDiv3_005008 Cc1nc2ncnn2c(O)c1NS(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D15 compound treatment 360.0 -244.0 -0.09 640.0 -108.0 -0.08 -0.1199 -0.9998 3119724 ChemDiv3_005009 COc1ccc(cc1)N(C2CC(=O)N(C2=O)c3ccc(OC)cc3)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D16 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 3024235 ChemDiv3_005010 CCOC(=O)c1nc(Nc2cccc(C)c2C)c3ccccc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D17 compound treatment 200.0 -404.0 -0.14 400.0 -348.0 -0.27 -0.2903 -0.9572 1305881 ChemDiv3_005011 COc1ccc(NC(=O)Nc2ccc3COC(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D18 compound treatment 360.0 -244.0 -0.09 400.0 -348.0 -0.27 -0.2501 -0.8904 3119725 ChemDiv3_005012 CCc1ccc(Oc2c(oc3c(CN4CCCCC4)c(O)ccc3c2=O)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D19 compound treatment 320.0 -284.0 -0.1 200.0 -548.0 -0.42 -0.3687 -0.8522 3024238 ChemDiv3_005013 CCn1c(S)nc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D20 compound treatment 1400.0 796.0 0.28 360.0 -388.0 -0.3 -0.011 -0.0267 1388420 ChemDiv3_005014 COC(=O)c1ccc(cc1)C2Nc3cccc4cccc(N2)c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D21 compound treatment 160.0 -444.0 -0.16 280.0 -468.0 -0.36 -0.3655 -0.9314 1523877 ChemDiv3_005015 CC(C)c1nc2ccccc2n1C(=O)c3ccccc3C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D22 compound treatment 320.0 -284.0 -0.1 360.0 -388.0 -0.3 -0.2819 -0.8962 3024241 ChemDiv3_005016 Cc1noc(C)c1CSc2ccc3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D23 mock treatment 360.0 -244.0 -0.09 2440.0 1690.0 1.3 0.8573 0.6586 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 D24 mock treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E01 compound treatment 1800.0 1200.0 0.42 7640.0 6890.0 5.29 4.0414 0.7614 3119726 ChemDiv3_005017 CCc1ccc(cc1)C(=O)/C=C/Nc2ccc(C)cc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E02 compound treatment 400.0 -204.0 -0.07 5360.0 4610.0 3.54 2.4525 0.6925 3024284 ChemDiv3_005018 COc1ccc(/C=C\2/SC(=O)N(CC(=O)NCCO)C2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E03 compound treatment 760.0 156.0 0.06 720.0 -28.1 -0.02 0.0239 0.402 3119727 ChemDiv3_005019 Cc1cc(c2ccccc2)n3ncc(c4ccccc4)c3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E04 compound treatment 1600.0 996.0 0.35 1000.0 252.0 0.19 0.3866 0.9597 3024286 ChemDiv3_005020 CC(=O)N1c2c(ccc3ccccc23)C(=CC1(C)C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E05 compound treatment 520.0 -83.8 -0.03 720.0 -28.1 -0.02 -0.0363 -0.9878 3119728 ChemDiv3_005021 O=C(NCc1ccccc1)C2CCN(CC2)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E06 compound treatment 680.0 76.3 0.03 920.0 172.0 0.13 0.1124 0.8347 3119729 ChemDiv3_005022 COC(=O)c1ccc(Oc2nc(Nc3cccc(C)c3C)nc(n2)N4CCC(C)CC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E07 compound treatment 520.0 -83.8 -0.03 680.0 -68.1 -0.05 -0.058 -0.9641 3024291 ChemDiv3_005023 COc1ccc(NCC(=O)n2c3ccccc3c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E08 compound treatment 480.0 -124.0 -0.04 880.0 132.0 0.1 0.0405 0.3674 3119730 ChemDiv3_005024 CCC(/N=c/1\cc(oc2ccc(C)cc12)c3ccc(OC)cc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E09 compound treatment 640.0 36.3 0.01 680.0 -68.1 -0.05 -0.0279 -0.5179 3024295 ChemDiv3_005025 CCN1C(=O)/C(=N/O)/N(CC)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E10 compound treatment 480.0 -124.0 -0.04 640.0 -108.0 -0.08 -0.0898 -0.9556 1702577 ChemDiv3_005026 CCOC(=O)c1cnc2c(C)cc(C)cc2c1Nc3ccc(cc3)S(=O)(=O)Nc4ncccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E11 compound treatment 560.0 -43.8 -0.02 520.0 -228.0 -0.18 -0.1348 -0.7668 3024297 ChemDiv3_005027 COC(=O)CN/1C(=S)N(C(=O)\C1=C\c2ccc(o2)c3ccc(Cl)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E12 compound treatment 680.0 76.3 0.03 1680.0 932.0 0.72 0.525 0.7333 3024299 ChemDiv3_005028 Clc1ccccc1CSc2nc(=O)cc[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E13 compound treatment 720.0 116.0 0.04 6720.0 5970.0 4.58 3.271 0.7134 3119731 ChemDiv3_005029 CC(C)n1c(=N)c(cc2c(=O)n3cccc(C)c3nc12)C(=O)NCCN4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E14 compound treatment 560.0 -43.8 -0.02 320.0 -428.0 -0.33 -0.2434 -0.7397 3119732 ChemDiv3_005030 COc1ccc(/C=C/2\CCc3ccccc3C2=O)cc1COc4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E15 compound treatment 960.0 356.0 0.13 760.0 11.9 0.01 0.0958 0.7561 3024306 ChemDiv3_005031 CC(C)CCSc1nc(N)c2c(C)c(C)sc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E16 compound treatment 2000.0 1400.0 0.5 1120.0 372.0 0.29 0.5521 0.9657 3119733 ChemDiv3_005032 Cc1cccc(c1)N2CN(Cc3ccco3)CNC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E17 compound treatment 2120.0 1520.0 0.54 1280.0 532.0 0.41 0.6691 0.9908 3024308 ChemDiv3_005033 Cc1ccc(cc1)C(CC(=O)O)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E18 compound treatment 880.0 276.0 0.1 360.0 -388.0 -0.3 -0.1414 -0.4508 3119734 ChemDiv3_005034 Cc1nnc(s1)N2C(=N)S/C(=C\c3ccccc3Cl)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E19 compound treatment 520.0 -83.8 -0.03 960.0 212.0 0.16 0.094 0.5685 3024312 ChemDiv3_005035 Clc1ccc(N/C=C/2\Nc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E20 compound treatment 880.0 276.0 0.1 1960.0 1210.0 0.93 0.7272 0.7773 3119735 ChemDiv3_005036 Cc1cc(OCC[N+]2(C)CCCCC2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E21 compound treatment 4360.0 3760.0 1.33 680.0 -68.1 -0.05 0.9052 0.6788 3024315 ChemDiv3_005037 CC(C)N/C=C/1\C(=O)Nc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E22 compound treatment 760.0 156.0 0.06 1480.0 732.0 0.56 0.4365 0.7731 3119736 ChemDiv3_005038 COC(=O)CC/1=NN(C(=O)\C1=C\Nc2ccc(C)cc2)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E23 mock treatment 2760.0 2160.0 0.76 8120.0 7370.0 5.66 4.5428 0.7954 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 E24 mock treatment 920.0 316.0 0.11 1120.0 372.0 0.29 0.2812 0.9167 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F01 compound treatment 880.0 276.0 0.1 1320.0 572.0 0.44 0.3797 0.8442 3025240 ChemDiv3_005039 Sc1nnc(c2ccncc2)n1C3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F02 compound treatment 840.0 236.0 0.08 7320.0 6570.0 5.05 3.6269 0.7188 3025241 ChemDiv3_005040 CCc1ccc(/C=C/2\NC(=S)N(C3CCCCC3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F03 compound treatment 800.0 196.0 0.07 880.0 132.0 0.1 0.1208 0.9833 1185203 ChemDiv3_005041 COc1ccc(CC(=O)N2c3ccccc3Sc4ccccc24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F04 compound treatment 2320.0 1720.0 0.61 8680.0 7930.0 6.09 4.7364 0.7739 3025242 ChemDiv3_005042 Cc1nn(CO)c(C)c1Sc2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F05 compound treatment 600.0 -3.75 0.0 1200.0 452.0 0.35 0.2444 0.7044 3025243 ChemDiv3_005043 CCN(CC)C(=S)SCc1nc(N)nc(Nc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F06 compound treatment 800.0 196.0 0.07 1400.0 652.0 0.5 0.4031 0.7978 3025244 ChemDiv3_005044 Cc1oc2cc(Br)c(O)c(Br)c2c1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F07 compound treatment 1000.0 396.0 0.14 520.0 -228.0 -0.18 -0.0245 -0.1089 1429843 ChemDiv3_005045 COc1ccc(cc1)C(=O)OC2=C(C(=O)c3ccccc3C2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F08 compound treatment 760.0 156.0 0.06 920.0 172.0 0.13 0.1325 0.9258 3119737 ChemDiv3_005046 COc1ccc(cc1)n2nc3ccc(NC(=O)CSc4ccc(Cl)cc4)cc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F09 compound treatment 4480.0 3880.0 1.38 1120.0 372.0 0.29 1.1742 0.8361 3025245 ChemDiv3_005047 Cn1nc(c2ccc(N3CCCCC3)c(NC(=O)c4ccccc4)c2)c5ccccc5c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F10 compound treatment 880.0 276.0 0.1 1160.0 412.0 0.32 0.2929 0.8847 3119738 ChemDiv3_005048 CCOC(=O)C1C(C2CCOC2=O)c3c(OC1=O)ccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F11 compound treatment 1920.0 1320.0 0.47 2480.0 1730.0 1.33 1.2703 0.9015 3025246 ChemDiv3_005049 Clc1cccc(c1)N2C(=O)N/C(=C/c3ccccc3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F12 compound treatment 880.0 276.0 0.1 2040.0 1290.0 0.99 0.7706 0.7732 1483558 ChemDiv3_005050 Brc1cccc2C(CC=C)NCCc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F13 compound treatment 1080.0 476.0 0.17 4000.0 3250.0 2.5 1.8848 0.7532 1345308 ChemDiv3_005051 CCOC(=O)c1sc(NN)nc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F14 compound treatment 2240.0 1640.0 0.58 640.0 -108.0 -0.08 0.3517 0.5999 3119883 ChemDiv3_005052 FC(F)(F)c1cc(nc(SCC(=O)N2CCCCC2)c1C#N)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F15 compound treatment 920.0 316.0 0.11 680.0 -68.1 -0.05 0.0423 0.342 3025247 ChemDiv3_005053 Clc1ccccc1NC(=O)c2cc(nc3ccccc23)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F16 compound treatment 880.0 276.0 0.1 800.0 51.9 0.04 0.0974 0.9212 3119884 ChemDiv3_005054 COc1ccc(/C=C/2\Oc3cc(OC(=O)c4ccc(F)cc4)ccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F17 compound treatment 4680.0 4080.0 1.45 3760.0 3010.0 2.31 2.6575 0.9745 1705934 ChemDiv3_005055 O=C(Nc1ccccc1)N2CCN3C(=O)c4ccccc4C23c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F18 compound treatment 1000.0 396.0 0.14 1240.0 492.0 0.38 0.3664 0.9094 3025248 ChemDiv3_005056 CCc1ccc(Oc2c(oc3c(CN(C)C)c(O)ccc3c2=O)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F19 compound treatment 1000.0 396.0 0.14 1640.0 892.0 0.68 0.5835 0.8349 1681490 ChemDiv3_005057 CCOc1ccc2[nH]c(SCC(=O)Nc3ccccc3)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F20 compound treatment 840.0 236.0 0.08 1840.0 1090.0 0.84 0.652 0.7739 3119885 ChemDiv3_005058 COc1ccc(cc1)c2c3C(=O)CC(C)(C)Cc3nc4sc(C(=O)N5CCCCCC5)c(N)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F21 compound treatment 760.0 156.0 0.06 1320.0 572.0 0.44 0.3496 0.7901 1693546 ChemDiv3_005059 Cc1cc(C)c(c(C)c1)S(=O)(=O)N2CCN(Cc3ccc4OCOc4c3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F22 compound treatment 360.0 -244.0 -0.09 2760.0 2010.0 1.54 1.031 0.6665 3025249 ChemDiv3_005060 Cc1ccc(NC(=O)CSc2nnc3ccccn23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F23 mock treatment 1520.0 916.0 0.33 1360.0 612.0 0.47 0.562 0.9838 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 F24 mock treatment 1200.0 596.0 0.21 920.0 172.0 0.13 0.2429 0.9742 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G01 compound treatment 840.0 236.0 0.08 1480.0 732.0 0.56 0.4566 0.8037 3119886 ChemDiv3_005061 O/C(=C\1/CCC/C(=C\c2ccccc2)/C1=O)/C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G02 compound treatment 1000.0 396.0 0.14 840.0 91.9 0.07 0.1493 0.9491 1563591 ChemDiv3_005062 S=C1NC2(CCS1)Oc3ccccc3C4CC(=NN42)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G03 compound treatment 1760.0 1160.0 0.41 5720.0 4970.0 3.82 2.9891 0.7786 3025250 ChemDiv3_005063 CCOC(=O)c1cnc2c(C#N)c(C)nn2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G04 compound treatment 960.0 356.0 0.13 600.0 -148.0 -0.11 0.0089 0.0526 3119887 ChemDiv3_005064 CC(=C)CC(Nc1ccccc1F)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G05 compound treatment 1000.0 396.0 0.14 1000.0 252.0 0.19 0.2361 0.9877 3025251 ChemDiv3_005065 CCOc1ccc(NC(=O)C2CCN(CC2)C(=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G06 compound treatment 1000.0 396.0 0.14 920.0 172.0 0.13 0.1927 0.9995 3119888 ChemDiv3_005066 FC(F)(F)c1cccc(CN2c3cccc4cccc(c34)S2(=O)=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G07 compound treatment 320.0 -284.0 -0.1 480.0 -268.0 -0.21 -0.2167 -0.9458 3025252 ChemDiv3_005067 Cc1ccc(cc1)c2csc(n2)N3C(=O)CN=C3SCc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G08 compound treatment 1080.0 476.0 0.17 2680.0 1930.0 1.48 1.1682 0.7826 3119889 ChemDiv3_005068 COc1ccc(/N=c/2\cc(oc3ccc(O)cc23)c4ccc(OC)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G09 compound treatment 640.0 36.3 0.01 920.0 172.0 0.13 0.1024 0.7724 3119890 ChemDiv3_005069 CN/1C(=O)/C(=C/c2cccs2)/S\C1=N\c3ccc(cc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G10 compound treatment 5120.0 4520.0 1.6 1760.0 1010.0 0.78 1.6822 0.9448 1551423 ChemDiv3_005070 CCN(CC)CC(O)COc1ccc(cc1C(C)(C)CC)C(C)(C)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G11 compound treatment 600.0 -3.75 0.0 600.0 -148.0 -0.11 -0.0814 -0.7153 3119891 ChemDiv3_005071 CCN1C(=O)/C(=C/c2ccco2)/NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G12 compound treatment 360.0 -244.0 -0.09 400.0 -348.0 -0.27 -0.2501 -0.8904 1281346 ChemDiv3_005072 COc1ccc(NC(=O)c2cc[nH]n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G13 compound treatment 400.0 -204.0 -0.07 480.0 -268.0 -0.21 -0.1967 -0.9014 3119892 ChemDiv3_005073 CC(=O)N1N=C(OC1c2cccnc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G14 compound treatment 400.0 -204.0 -0.07 1080.0 332.0 0.25 0.129 0.4873 3025253 ChemDiv3_005074 COC(=O)C1Cc2c([nH]c3ccccc23)C(C)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G15 compound treatment 1120.0 516.0 0.18 920.0 172.0 0.13 0.2228 0.9871 1321601 ChemDiv3_005075 CC(C)Nc1nc(NC(C)C)nc(n1)N(n2cnnc2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G16 compound treatment 400.0 -204.0 -0.07 640.0 -108.0 -0.08 -0.1098 -0.9976 3025254 ChemDiv3_005076 CC(C)CN1CN(Cc2ccco2)CNC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G17 compound treatment 1000.0 396.0 0.14 1040.0 292.0 0.22 0.2578 0.9748 3119893 ChemDiv3_005077 CC1(C)CC(CCC(=O)NC(=S)Nc2ccccc2Cl)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G18 compound treatment 1000.0 396.0 0.14 1120.0 372.0 0.29 0.3013 0.9467 3119894 ChemDiv3_005078 COC(=O)c1ccc(Oc2nc(Nc3ccccc3F)nc(n2)N4CCCCC4C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G19 compound treatment 360.0 -244.0 -0.09 480.0 -268.0 -0.21 -0.2067 -0.9258 3025255 ChemDiv3_005079 Clc1c2C(=O)/C(=C/NCc3ccccc3)/Nc2ccc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G20 compound treatment 440.0 -164.0 -0.06 960.0 212.0 0.16 0.0739 0.4281 3119895 ChemDiv3_005080 CN1CCc2c(C1=O)n(CC(O)Cn3nc(C)c(Br)c3C)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G21 compound treatment 320.0 -284.0 -0.1 1000.0 252.0 0.19 0.0655 0.3007 3025256 ChemDiv3_005081 COc1ccc(/C=C/C(=O)CC(=O)c2ccccc2O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G22 compound treatment 440.0 -164.0 -0.06 1120.0 372.0 0.29 0.1608 0.5519 3119896 ChemDiv3_005082 O=C1OC(N2CCN(CCNC=C3C(=O)CC(CC3=O)c4ccccc4)CC2)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G23 mock treatment 1720.0 1120.0 0.4 520.0 -228.0 -0.18 0.1562 0.3606 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 G24 mock treatment 680.0 76.3 0.03 640.0 -108.0 -0.08 -0.0396 -0.4533 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H01 compound treatment 400.0 -204.0 -0.07 720.0 -28.1 -0.02 -0.0664 -0.88 3025257 ChemDiv3_005083 CC1(C)CC(CC(C)(C)N1)NC(=S)Nc2ccc(cc2)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H02 compound treatment 5880.0 5280.0 1.87 760.0 11.9 0.01 1.3299 0.7105 3119897 ChemDiv3_005084 CCC1=[N+]([O-])C(C)(N(O)C1(C)C)/C(=N\O)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H03 compound treatment 720.0 116.0 0.04 640.0 -108.0 -0.08 -0.0295 -0.3187 1599271 ChemDiv3_005085 Cc1ccc(SCC(=O)n2c3ccccc3c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H04 compound treatment 480.0 -124.0 -0.04 1000.0 252.0 0.19 0.1057 0.533 3119898 ChemDiv3_005086 CCN1C(=O)/C(=C\c2cccc3C(=O)c4ccccc4-c32)/OC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H05 compound treatment 2320.0 1720.0 0.61 440.0 -308.0 -0.24 0.2632 0.403 3119899 ChemDiv3_005087 Cc1ccc(Nc2nc(N)nc(CC(=O)CSc3nc4ccccc4s3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H06 compound treatment 440.0 -164.0 -0.06 1280.0 532.0 0.41 0.2476 0.6005 3025258 ChemDiv3_005088 CCOC(=O)c1nc(N)c(=O)n(n1)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H07 compound treatment 2600.0 2000.0 0.71 960.0 212.0 0.16 0.6158 0.8474 1535790 ChemDiv3_005089 Cc1ccc(cc1)C(=O)OC2=C(C(=O)c3ccccc3C2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H08 compound treatment 600.0 -3.75 0.0 14080.0 13300.0 10.24 7.2364 0.707 3025259 ChemDiv3_005090 O=C1c2ncn(c2C(=O)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H09 compound treatment 320.0 -284.0 -0.1 1080.0 332.0 0.25 0.109 0.3978 3119900 ChemDiv3_005091 CS(=O)(=O)Nc1cc(ccc1N2CCOCC2)c3nnc(Nc4ccccc4)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H10 compound treatment 480.0 -124.0 -0.04 7680.0 6930.0 5.32 3.732 0.7012 3025260 ChemDiv3_005092 CCOC(=O)C1C(c2cc(Br)ccc2OC1=O)C3(CCCCC3)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H11 compound treatment 3040.0 2440.0 0.86 680.0 -68.1 -0.05 0.5741 0.6631 3119901 ChemDiv3_005093 CCN(CC)c1ccc(cc1)n2c(C)cc(/C=C\3/NC(=O)N(Cc4ccccc4F)C3=O)c2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H12 compound treatment 5240.0 4640.0 1.64 760.0 11.9 0.01 1.1694 0.711 1277443 ChemDiv3_005094 COc1ccc(cc1)n2c(N)c(c3nc4ccccc4s3)c5nc(C#N)c(C#N)nc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H13 compound treatment 800.0 196.0 0.07 1040.0 292.0 0.22 0.2077 0.8851 3119902 ChemDiv3_005095 CCN1C(=O)/C(=C/c2ccc(Cl)cc2)/NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H14 compound treatment 440.0 -164.0 -0.06 840.0 91.9 0.07 0.0088 0.0962 1602494 ChemDiv3_005096 O=C(CSc1nc2CCCCc2cc1C#N)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H15 compound treatment 360.0 -244.0 -0.09 880.0 132.0 0.1 0.0104 0.0784 3025261 ChemDiv3_005097 Cc1ccc(C)c(NC(CC(=O)c2ccccc2)C(=O)O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H16 compound treatment 440.0 -164.0 -0.06 600.0 -148.0 -0.11 -0.1215 -0.9514 3119903 ChemDiv3_005098 COc1ccc(/C=C/2\Oc3cc(OCc4cccc(C)c4)ccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H17 compound treatment 520.0 -83.8 -0.03 7640.0 6890.0 5.29 3.7203 0.7031 1119051 ChemDiv3_005099 CC1(C)NC(=O)N(CC(O)Cn2c3ccccc3c4ccccc24)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H18 compound treatment 600.0 -3.75 0.0 680.0 -68.1 -0.05 -0.0379 -0.7249 3025262 ChemDiv3_005100 COc1ccc(CCNC(=O)COc2ccc3c(=O)c(coc3c2)c4ccccc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H19 compound treatment 480.0 -124.0 -0.04 2120.0 1370.0 1.05 0.7137 0.677 3120046 ChemDiv3_005101 Clc1ccc(CSc2nc3ccccc3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H20 compound treatment 2480.0 1880.0 0.67 3280.0 2530.0 1.94 1.8451 0.898 3025263 ChemDiv3_005102 Cc1nc2cc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)ccc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H21 compound treatment 760.0 156.0 0.06 520.0 -228.0 -0.18 -0.0847 -0.4608 3120047 ChemDiv3_005103 CS(=O)(=O)N1CCC(CC1)C(=O)NCCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H22 compound treatment 360.0 -244.0 -0.09 840.0 91.9 0.07 -0.0113 -0.1011 3120048 ChemDiv3_005104 O=C(CSc1nnc2ccccn12)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H23 mock treatment 880.0 276.0 0.1 1000.0 252.0 0.19 0.206 0.9504 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 H24 mock treatment 440.0 -164.0 -0.06 760.0 11.9 0.01 -0.0346 -0.5892 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I01 compound treatment 1880.0 1280.0 0.45 280.0 -468.0 -0.36 0.066 0.1142 1405649 ChemDiv3_005105 COc1cccc(NC(=O)COc2ccc(cc2)N3CC(CC3=O)C(=O)NCC(C)C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I02 compound treatment 400.0 -204.0 -0.07 320.0 -428.0 -0.33 -0.2835 -0.8425 1546533 ChemDiv3_005106 Cc1ccc(cc1)N2C(=O)C3Sc4[nH]c(=O)sc4C(C3C2=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I03 compound treatment 240.0 -364.0 -0.13 1000.0 252.0 0.19 0.0455 0.1956 1209298 ChemDiv3_005107 CCOC(=O)c1cnc2c(cnn2c1C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I04 compound treatment 520.0 -83.8 -0.03 280.0 -468.0 -0.36 -0.2751 -0.763 1582005 ChemDiv3_005108 Cc1ccc(cc1)N2CC3(OC4C=C3)C(C4C(=O)O)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I05 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 3120049 ChemDiv3_005109 CCc1ccc(NC(=O)C2CCN(CC2)C(=O)c3ccccc3C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I06 compound treatment 280.0 -324.0 -0.11 800.0 51.9 0.04 -0.0531 -0.4365 3025264 ChemDiv3_005110 Brc1cccc(CN2c3cccc4cccc(c34)S2(=O)=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I07 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3120050 ChemDiv3_005111 N/C(=N\c1nc(=O)c2CCCCc2[nH]1)/Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I08 compound treatment 320.0 -284.0 -0.1 560.0 -188.0 -0.14 -0.1733 -0.9844 3120051 ChemDiv3_005112 COc1ccc(cc1)c2c/c(=N\c3ccc(C)cc3C)/c4cc(O)ccc4o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I09 compound treatment 240.0 -364.0 -0.13 640.0 -108.0 -0.08 -0.15 -0.9773 3025265 ChemDiv3_005113 CCN/1C(=O)CS\C1=N\c2cccc(c2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I10 compound treatment 280.0 -324.0 -0.11 360.0 -388.0 -0.3 -0.2919 -0.9141 1298232 ChemDiv3_005114 O=C(Oc1cccc2cccnc12)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I11 compound treatment 560.0 -43.8 -0.02 280.0 -468.0 -0.36 -0.2651 -0.737 3120052 ChemDiv3_005115 CCCCN1C(=O)S/C(=C\c2cc(C)n(C)c2C)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I12 compound treatment 440.0 -164.0 -0.06 320.0 -428.0 -0.33 -0.2735 -0.8194 1336653 ChemDiv3_005116 CCC(=O)n1ccc(n1)C(=O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I13 compound treatment 240.0 -364.0 -0.13 320.0 -428.0 -0.33 -0.3237 -0.9166 3025316 ChemDiv3_005117 CC(=O)N1N=C(OC21CCCC2)c3ccc4ccccc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I14 compound treatment 240.0 -364.0 -0.13 280.0 -468.0 -0.36 -0.3454 -0.9045 3025317 ChemDiv3_005118 Cc1ccc(cc1)C2NC(=S)NC(=C2)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I15 compound treatment 280.0 -324.0 -0.11 440.0 -308.0 -0.24 -0.2485 -0.9449 3025318 ChemDiv3_005119 COC(=O)NCCOc1nc(nc(n1)N(C)C)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I16 compound treatment 320.0 -284.0 -0.1 200.0 -548.0 -0.42 -0.3687 -0.8522 3025319 ChemDiv3_005120 CCN1CNC(=S)N(C1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I17 compound treatment 400.0 -204.0 -0.07 320.0 -428.0 -0.33 -0.2835 -0.8425 3025320 ChemDiv3_005121 CC(C)c1ccc(C)cc1OCC(=O)Nn2c(=O)[nH]c3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I18 compound treatment 160.0 -444.0 -0.16 440.0 -308.0 -0.24 -0.2786 -0.9804 3025321 ChemDiv3_005122 CCN(CC)c1ccc(cc1)c2cc(C(=O)O)c3c(ccc4ccccc43)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I19 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3025322 ChemDiv3_005123 O=C/1Nc2ccccc2\C1=C\NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I20 compound treatment 400.0 -204.0 -0.07 1120.0 372.0 0.29 0.1508 0.5119 3120053 ChemDiv3_005124 CN1CCc2c(C1=O)n(CC(O)CNCc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I21 compound treatment 240.0 -364.0 -0.13 280.0 -468.0 -0.36 -0.3454 -0.9045 3025323 ChemDiv3_005125 O=c1cc(/C=C/c2ccccc2)oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I22 compound treatment 360.0 -244.0 -0.09 360.0 -388.0 -0.3 -0.2719 -0.8762 3120054 ChemDiv3_005126 CCCNC(=O)CSc1c(c2ccccc2)c3cc(Cl)ccc3[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I23 mock treatment 280.0 -324.0 -0.11 440.0 -308.0 -0.24 -0.2485 -0.9449 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 I24 mock treatment 240.0 -364.0 -0.13 320.0 -428.0 -0.33 -0.3237 -0.9166 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J01 compound treatment 840.0 236.0 0.08 440.0 -308.0 -0.24 -0.108 -0.4304 3025324 ChemDiv3_005127 CCCCc1ccc(NC(=S)NCCCN2CCOCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J02 compound treatment 440.0 -164.0 -0.06 320.0 -428.0 -0.33 -0.2735 -0.8194 3120055 ChemDiv3_005128 CC1=[N+]([O-])C2(CCCC2)[N+](=C1c3ccccc3)[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J03 compound treatment 320.0 -284.0 -0.1 600.0 -148.0 -0.11 -0.1516 -0.9981 3120056 ChemDiv3_005129 O=C(Nc1ccccc1)C2CC(=O)NC(=N2)Nc3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J04 compound treatment 560.0 -43.8 -0.02 400.0 -348.0 -0.27 -0.2 -0.7469 3025325 ChemDiv3_005130 Cc1ccc(NS(=O)(=O)c2ccc3n(C(=O)Oc4ccccc4)c(=O)oc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J05 compound treatment 320.0 -284.0 -0.1 240.0 -508.0 -0.39 -0.347 -0.8613 3120057 ChemDiv3_005131 COc1ccc(Cl)cc1Nc2nc(N)nc(CC(=O)CSc3nc4ccccc4s3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J06 compound treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 1919405 ChemDiv3_005132 CCn1c2ccccc2c3nnc(S)nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J07 compound treatment 1240.0 636.0 0.23 720.0 -28.1 -0.02 0.1443 0.6365 3025326 ChemDiv3_005133 Fc1ccc(cc1)C2Sc3ccccc3N=C4C2C(=O)c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J08 compound treatment 400.0 -204.0 -0.07 360.0 -388.0 -0.3 -0.2618 -0.8539 3120058 ChemDiv3_005134 Cc1cccc(c1)C(=O)NCCCn2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J09 compound treatment 1080.0 476.0 0.17 320.0 -428.0 -0.33 -0.113 -0.3056 3120059 ChemDiv3_005135 CCN(CC)C(=O)COc1ccc(cc1)c2nnc(Nc3ccc(OC)c(c3)C(=O)N)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J10 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 3025327 ChemDiv3_005136 CCCC(CCC)C(=O)Nc1cc(cc(c1)C(=O)O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J11 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 1472732 ChemDiv3_005137 Cc1ccc(NC2CS(=O)(=O)C=C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J12 compound treatment 680.0 76.3 0.03 360.0 -388.0 -0.3 -0.1916 -0.6403 1452920 ChemDiv3_005138 OC(=O)CCC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J13 compound treatment 240.0 -364.0 -0.13 240.0 -508.0 -0.39 -0.3671 -0.8934 3120060 ChemDiv3_005139 CCOc1ccc(cc1)N2C(=O)/C(=C/c3ccccc3)/N(C)C2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J14 compound treatment 320.0 -284.0 -0.1 320.0 -428.0 -0.33 -0.3036 -0.8832 3025328 ChemDiv3_005140 CC(C)c1ccccc1Oc2coc3cc(OCC(=O)NC4CCCCC4)ccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J15 compound treatment 320.0 -284.0 -0.1 200.0 -548.0 -0.42 -0.3687 -0.8522 1599429 ChemDiv3_005141 COc1ccc(cc1)c2cc(C(=O)OCC(=O)c3ccccc3)c4cccc(Cl)c4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J16 compound treatment 240.0 -364.0 -0.13 360.0 -388.0 -0.3 -0.302 -0.9299 3025329 ChemDiv3_005142 COc1cc(cc(OC)c1OC)C(=O)Oc2ccc3C(=O)COc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J17 compound treatment 360.0 -244.0 -0.09 280.0 -468.0 -0.36 -0.3153 -0.8529 3120061 ChemDiv3_005143 COCn1c(nc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J18 compound treatment 320.0 -284.0 -0.1 440.0 -308.0 -0.24 -0.2385 -0.9275 1585270 ChemDiv3_005144 CCCc1cc(ccn1)c2nc(cs2)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J19 compound treatment 280.0 -324.0 -0.11 1000.0 252.0 0.19 0.0555 0.2468 3025330 ChemDiv3_005145 COc1ccc(CSc2nc3ccccc3s2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J20 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3120062 ChemDiv3_005146 Cc1nnc(SCCC(=O)Nc2cccc(c2)c3nc4ccccc4s3)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J21 compound treatment 4400.0 3800.0 1.35 2400.0 1650.0 1.27 1.849 0.9995 3025331 ChemDiv3_005147 CN/1C(=S)N(C2CCCCC2)C(=O)\C1=C\c3ccccc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J22 compound treatment 400.0 -204.0 -0.07 360.0 -388.0 -0.3 -0.2618 -0.8539 3120063 ChemDiv3_005148 O=C(CCSc1nnc2ccccn12)Nc3cccc(c3)c4nc5ccccc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J23 mock treatment 240.0 -364.0 -0.13 4040.0 3290.0 2.53 1.6958 0.6701 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 J24 mock treatment 280.0 -324.0 -0.11 4480.0 3730.0 2.87 1.9447 0.6782 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K01 compound treatment 960.0 356.0 0.13 1480.0 732.0 0.56 0.4867 0.845 3120064 ChemDiv3_005149 COc1ccc(cc1)N2CC(CC2=O)C(=O)OCC(=O)Nc3ccccc3C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K02 compound treatment 5640.0 5040.0 1.79 760.0 11.9 0.01 1.2697 0.7107 3025332 ChemDiv3_005150 Cc1ccccc1NC(CC=C)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K03 compound treatment 2200.0 1600.0 0.57 400.0 -348.0 -0.27 0.2114 0.3376 3025333 ChemDiv3_005151 CC(C)(C)c1ccc(cc1)c2cc3ncc(c(N)n3n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K04 compound treatment 760.0 156.0 0.06 680.0 -68.1 -0.05 0.0022 0.0289 1246311 ChemDiv3_005152 OC(=O)C1C2OC3(CN(CCc4ccccc4)C(=O)C13)C=C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K05 compound treatment 1240.0 636.0 0.23 840.0 91.9 0.07 0.2095 0.8858 3120065 ChemDiv3_005153 CC(C)CNC(=O)C1CCN(CC1)C(=O)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K06 compound treatment 680.0 76.3 0.03 720.0 -28.1 -0.02 0.0038 0.1111 1524928 ChemDiv3_005154 Cc1ccc(cc1)c2csc3ncnc(NCCC(=O)O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K07 compound treatment 520.0 -83.8 -0.03 1000.0 252.0 0.19 0.1157 0.5915 3120066 ChemDiv3_005155 COc1cc(OC)cc(c1)C2=NC(C)(C)CO2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K08 compound treatment 720.0 116.0 0.04 1240.0 492.0 0.38 0.2962 0.7797 1424113 ChemDiv3_005156 CC(C)Oc1ccccc1Nc2ncnc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K09 compound treatment 760.0 156.0 0.06 360.0 -388.0 -0.3 -0.1715 -0.5659 3120067 ChemDiv3_005157 Oc1ccc(/C=C/2\SC(=O)N(CC(=O)N3CCOCC3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K10 compound treatment 400.0 -204.0 -0.07 800.0 51.9 0.04 -0.023 -0.2783 3120068 ChemDiv3_005158 COc1ccc(CCN2C(=O)CC(Sc3ccccc3C(=O)O)C2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K11 compound treatment 400.0 -204.0 -0.07 440.0 -308.0 -0.24 -0.2184 -0.8829 3025334 ChemDiv3_005159 C=CCn1cc(C=C2C(=O)OC(OC2=O)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K12 compound treatment 360.0 -244.0 -0.09 2240.0 1490.0 1.15 0.7487 0.6519 1125429 ChemDiv3_005160 Clc1ccc(C(=O)n2ccc(n2)C(=O)N3CCCCC3)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K13 compound treatment 1000.0 396.0 0.14 560.0 -188.0 -0.14 -0.0027 -0.0136 3025335 ChemDiv3_005161 O=C(Nc1cccc2cccnc12)/C=C/c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K14 compound treatment 6200.0 5600.0 1.99 1200.0 452.0 0.35 1.6491 0.8183 3117769 ChemDiv3_005162 CC1C/C(=C\c2ccc(Cl)cc2)/C3=C(C1)C(NC(=S)N3)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K15 compound treatment 640.0 36.3 0.01 1080.0 332.0 0.25 0.1892 0.7419 1289908 ChemDiv3_005163 CCNc1nc(Oc2ccc(cc2)C(=O)OC)nc(SC)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K16 compound treatment 560.0 -43.8 -0.02 1080.0 332.0 0.25 0.1692 0.6628 3117770 ChemDiv3_005164 CCN1CNC(=S)N(C1)C2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K17 compound treatment 360.0 -244.0 -0.09 840.0 91.9 0.07 -0.0113 -0.1011 1050895 ChemDiv3_005165 Cc1ccc(cc1)S(=O)(=O)N2Cc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K18 compound treatment 1360.0 756.0 0.27 680.0 -68.1 -0.05 0.1527 0.5587 3117771 ChemDiv3_005166 Cc1ccc(NC(=O)CCn2nnc(n2)c3ccc(OCc4ccccc4F)cc3)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K19 compound treatment 560.0 -43.8 -0.02 520.0 -228.0 -0.18 -0.1348 -0.7668 3025336 ChemDiv3_005167 Cc1ccccc1N/C=C/2\C(=O)Nc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K20 compound treatment 400.0 -204.0 -0.07 680.0 -68.1 -0.05 -0.0881 -0.9874 3117772 ChemDiv3_005168 O=C1OC(N2CCc3ccccc3C2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K21 compound treatment 440.0 -164.0 -0.06 1360.0 612.0 0.47 0.2911 0.615 3117773 ChemDiv3_005169 Cc1ccc(cc1)c2cc(=O)c3ccc4ccccc4c3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K22 compound treatment 600.0 -3.75 0.0 1680.0 932.0 0.72 0.5049 0.7058 3025337 ChemDiv3_005170 Cc1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc(cc2)c3nc4ccc(C)cc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K23 mock treatment 1040.0 436.0 0.15 5320.0 4570.0 3.51 2.5913 0.7376 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 K24 mock treatment 760.0 156.0 0.06 1080.0 332.0 0.25 0.2193 0.8413 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L01 compound treatment 600.0 -3.75 0.0 800.0 51.9 0.04 0.0272 0.6831 3117774 ChemDiv3_005171 NS(=O)(=O)c1ccc(NC(=S)N2CCc3ccccc3C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L02 compound treatment 640.0 36.3 0.01 3640.0 2890.0 2.22 1.579 0.7112 3025338 ChemDiv3_005172 CCC1(C)[N+](=C(C)C(=[N+]1[O-])c2ccccc2)[O-] 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L03 compound treatment 400.0 -204.0 -0.07 720.0 -28.1 -0.02 -0.0664 -0.88 3117775 ChemDiv3_005173 CCOc1ccc2NC(C)(C)c3ss/c(=N\c4ccc(NC(=O)C)cc4)/c3-c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L04 compound treatment 360.0 -244.0 -0.09 960.0 212.0 0.16 0.0539 0.2924 3117776 ChemDiv3_005174 CC(C)Cn1c2ccc(Br)cc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L05 compound treatment 640.0 36.3 0.01 840.0 91.9 0.07 0.059 0.8225 1871645 ChemDiv3_005175 COc1ccc(CC(=O)N(CC=C)c2nnc(s2)c3ccc(Cl)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L06 compound treatment 560.0 -43.8 -0.02 280.0 -468.0 -0.36 -0.2651 -0.737 3117777 ChemDiv3_005176 CCc1ccc2[nH]c3nc(S)nnc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L07 compound treatment 400.0 -204.0 -0.07 520.0 -228.0 -0.18 -0.175 -0.9234 3117778 ChemDiv3_005177 CCc1ccc(cc1)N2NC(=O)/C(=C/c3ccc4n(C)c(=O)n(C)c4c3)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L08 compound treatment 480.0 -124.0 -0.04 640.0 -108.0 -0.08 -0.0898 -0.9556 3025339 ChemDiv3_005178 CC(CN1C(C)CCCC1C)OC(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L09 compound treatment 320.0 -284.0 -0.1 840.0 91.9 0.07 -0.0213 -0.1734 3117779 ChemDiv3_005179 O=C/1NC(=S)S\C1=C/c2c(NCc3ccco3)nc4ccccn4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L10 compound treatment 320.0 -284.0 -0.1 440.0 -308.0 -0.24 -0.2385 -0.9275 3025340 ChemDiv3_005180 CCC(=O)Oc1ccc(cc1)C(=O)Nc2cc(cc(c2)C(=O)O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L11 compound treatment 800.0 196.0 0.07 720.0 -28.1 -0.02 0.0339 0.4657 3117780 ChemDiv3_005181 COC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L12 compound treatment 440.0 -164.0 -0.06 720.0 -28.1 -0.02 -0.0564 -0.9093 3025341 ChemDiv3_005182 OC(=O)c1cc(/N=C\c2ccc(N3CCCC3)c(F)c2)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L13 compound treatment 2520.0 1920.0 0.68 600.0 -148.0 -0.11 0.4003 0.5807 3117781 ChemDiv3_005183 CN/1C(=S)N(C(=O)\C1=C\c2ccccc2O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L14 compound treatment 1160.0 556.0 0.2 520.0 -228.0 -0.18 0.0157 0.0594 3117782 ChemDiv3_005184 Cc1ccc(Oc2coc3cc(OCC(=O)N4CCCCC4)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L15 compound treatment 600.0 -3.75 0.0 560.0 -188.0 -0.14 -0.1031 -0.7136 3025342 ChemDiv3_005185 CCCC/1=NN(C(=O)\C1=C\c2ccc3OCOc3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L16 compound treatment 520.0 -83.8 -0.03 680.0 -68.1 -0.05 -0.058 -0.9641 1224155 ChemDiv3_005186 CC(Oc1ccc2c(=O)c(coc2c1)c3ccc(Cl)cc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L17 compound treatment 720.0 116.0 0.04 920.0 172.0 0.13 0.1225 0.8859 1151018 ChemDiv3_005187 CCCCn1c(nc2ccccc12)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L18 compound treatment 640.0 36.3 0.01 400.0 -348.0 -0.27 -0.1799 -0.6723 3117783 ChemDiv3_005188 Cc1ncc2COC(C)(C)OCc2c1OC(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L19 compound treatment 600.0 -3.75 0.0 680.0 -68.1 -0.05 -0.0379 -0.7249 3025343 ChemDiv3_005189 NC(=O)/C(=C\1/Oc2c(S1)cc(O)cc2c3ccccc3)/C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L20 compound treatment 3760.0 3160.0 1.12 5560.0 4810.0 3.69 3.4039 0.8818 3117784 ChemDiv3_005190 COc1ccc(NC(=O)CCSc2ccc3ccccc3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L21 compound treatment 760.0 156.0 0.06 640.0 -108.0 -0.08 -0.0195 -0.1955 3117785 ChemDiv3_005191 CCCN1C(=O)/C(=C/c2ccc(CC)cc2)/NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L22 compound treatment 440.0 -164.0 -0.06 1120.0 372.0 0.29 0.1608 0.5519 3025344 ChemDiv3_005192 O=C(CSc1nnc2ccc3ccccc3n12)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L23 mock treatment 320.0 -284.0 -0.1 1200.0 452.0 0.35 0.1741 0.482 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 L24 mock treatment 840.0 236.0 0.08 4760.0 4010.0 3.08 2.2371 0.7261 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M01 compound treatment 1160.0 556.0 0.2 1240.0 492.0 0.38 0.4065 0.9542 3117786 ChemDiv3_005193 OC(=O)CCc1ccc(c2ccccc2)n1NC(=O)c3ccccc3Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M02 compound treatment 480.0 -124.0 -0.04 1000.0 252.0 0.19 0.1057 0.533 3025345 ChemDiv3_005194 Cc1ccc(o1)c2cccc(c2)n3c(C)ccc3c4cccc(N)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M03 compound treatment 320.0 -284.0 -0.1 680.0 -68.1 -0.05 -0.1082 -0.9535 3117787 ChemDiv3_005195 COc1ccc(cc1)C2=C/C(=C/c3ccccc3)/C(=O)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M04 compound treatment 1000.0 396.0 0.14 280.0 -468.0 -0.36 -0.1547 -0.401 3025395 ChemDiv3_005196 CC1CC2N(C(=O)c3c2cccc3C(=O)O)c4ccc(F)cc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M05 compound treatment 360.0 -244.0 -0.09 400.0 -348.0 -0.27 -0.2501 -0.8904 3025396 ChemDiv3_005197 CCc1ccc(NC(=O)C2CCN(CC2)C(=O)c3ccc(F)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M06 compound treatment 2960.0 2360.0 0.84 640.0 -108.0 -0.08 0.5323 0.6338 1364255 ChemDiv3_005198 CCCC(=O)Oc1ccc2oc(cc(=O)c2c1)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M07 compound treatment 480.0 -124.0 -0.04 7040.0 6290.0 4.83 3.3845 0.7007 3025397 ChemDiv3_005199 CN1C(=O)/C(=C/c2cn(CC(=O)N3CCOCC3)c4ccccc24)/C(=O)NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M08 compound treatment 1000.0 396.0 0.14 480.0 -268.0 -0.21 -0.0462 -0.1852 3025398 ChemDiv3_005200 CCOC(=O)c1cnc2c(Cl)c(Cl)ccc2c1NCCOC(=O)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M09 compound treatment 440.0 -164.0 -0.06 400.0 -348.0 -0.27 -0.2301 -0.8412 3025399 ChemDiv3_005201 COc1ccccc1/C=C/2\SC(=O)N(CC(=O)N3CCOCC3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M10 compound treatment 280.0 -324.0 -0.11 1080.0 332.0 0.25 0.0989 0.354 3025400 ChemDiv3_005202 OC(=O)CCNS(=O)(=O)c1ccccc1C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M11 compound treatment 440.0 -164.0 -0.06 440.0 -308.0 -0.24 -0.2084 -0.8553 3117788 ChemDiv3_005203 COc1ccc(C=C2C(=O)OC(OC2=O)c3ccccc3)c(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M12 compound treatment 240.0 -364.0 -0.13 360.0 -388.0 -0.3 -0.302 -0.9299 3117789 ChemDiv3_005204 COc1ccc(/C=C/C(=O)C2CC2)cc1COc3cccc(C)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M13 compound treatment 520.0 -83.8 -0.03 600.0 -148.0 -0.11 -0.1014 -0.8629 3025401 ChemDiv3_005205 Nc1oc2cc3c(C(=O)OCC=C)c(N)oc3c(c4ccccc4)c2c1C(=O)OCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M14 compound treatment 560.0 -43.8 -0.02 520.0 -228.0 -0.18 -0.1348 -0.7668 3117790 ChemDiv3_005206 CC1C/C(=C\c2ccc(C)cc2)/C3=C(C1)C(NC(=S)N3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M15 compound treatment 560.0 -43.8 -0.02 560.0 -188.0 -0.14 -0.1131 -0.7786 3025402 ChemDiv3_005207 Cc1ccc(NC(=S)NC(=O)CC2CC(C)(C)OC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M16 compound treatment 1880.0 1280.0 0.45 7040.0 6290.0 4.83 3.7357 0.77 1419022 ChemDiv3_005208 S=C1NCN(CCc2ccccc2)CN1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M17 compound treatment 480.0 -124.0 -0.04 640.0 -108.0 -0.08 -0.0898 -0.9556 3117791 ChemDiv3_005209 N#Cc1nc(COc2ccccc2)oc1NCc3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M18 compound treatment 280.0 -324.0 -0.11 320.0 -428.0 -0.33 -0.3136 -0.9008 3025403 ChemDiv3_005210 Cn1nnc(n1)c2ccc(OCc3ccccc3F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M19 compound treatment 320.0 -284.0 -0.1 720.0 -28.1 -0.02 -0.0865 -0.8398 3117792 ChemDiv3_005211 O=C/1Nc2ccccc2\C1=C\NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M20 compound treatment 880.0 276.0 0.1 400.0 -348.0 -0.27 -0.1197 -0.4205 3117793 ChemDiv3_005212 Cc1noc(NS(=O)(=O)c2ccc(NC3OC(=O)c4ccccc34)cc2)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M21 compound treatment 480.0 -124.0 -0.04 680.0 -68.1 -0.05 -0.068 -0.9962 3025404 ChemDiv3_005213 O=c1cc(oc2c1ccc3ccccc32)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M22 compound treatment 760.0 156.0 0.06 920.0 172.0 0.13 0.1325 0.9258 3025405 ChemDiv3_005214 CC(=C1C(=O)c2ccccc2C1=O)N3CCc4ccccc4C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M23 mock treatment 400.0 -204.0 -0.07 600.0 -148.0 -0.11 -0.1315 -0.9761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 M24 mock treatment 360.0 -244.0 -0.09 2360.0 1610.0 1.24 0.8139 0.6561 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N01 compound treatment 400.0 -204.0 -0.07 1920.0 1170.0 0.9 0.585 0.6482 3117794 ChemDiv3_005215 NS(=O)(=O)c1ccc(NC(=S)N2CCC(Cc3ccccc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N02 compound treatment 200.0 -404.0 -0.14 640.0 -108.0 -0.08 -0.16 -0.9664 3025406 ChemDiv3_005216 C/C(=[N+](/[O-])\C\1CCC/C1=N\O)/C(=O)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N03 compound treatment 1120.0 516.0 0.18 520.0 -228.0 -0.18 0.0056 0.0223 3117795 ChemDiv3_005217 Sc1nnc(OCc2ccccc2)n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N04 compound treatment 280.0 -324.0 -0.11 440.0 -308.0 -0.24 -0.2485 -0.9449 3117796 ChemDiv3_005218 CC(C)c1ccc2[nH]c3/C(=N/O)/CCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N05 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 1457228 ChemDiv3_005219 Cn1c2N=C3C(C(c4cccc(Cl)c4)c2c(=O)n(C)c1=O)C(=O)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N06 compound treatment 400.0 -204.0 -0.07 1000.0 252.0 0.19 0.0856 0.4147 3117929 ChemDiv3_005220 CCc1ccc2n(C)c3nc(S)nnc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N07 compound treatment 5800.0 5200.0 1.84 520.0 -228.0 -0.18 1.1796 0.637 3117930 ChemDiv3_005221 COC(=O)C/1=C(C)NC(=O)\C1=C/c2cc(C)n(c2C)c3ccc(OC)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N08 compound treatment 640.0 36.3 0.01 600.0 -148.0 -0.11 -0.0713 -0.6232 3025407 ChemDiv3_005222 CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)NCCCn2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N09 compound treatment 480.0 -124.0 -0.04 240.0 -508.0 -0.39 -0.3069 -0.7817 3117931 ChemDiv3_005223 CC1=C(C(/C=C/c2ccccc2)N3C(=O)CCSC3=N1)C(=O)OCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N10 compound treatment 680.0 76.3 0.03 600.0 -148.0 -0.11 -0.0613 -0.5243 1320385 ChemDiv3_005224 OC(=O)c1ccc(cc1)C(=O)c2ccc3C(=O)N(CC4CCCO4)C(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N11 compound treatment 360.0 -244.0 -0.09 600.0 -148.0 -0.11 -0.1416 -0.9909 3025408 ChemDiv3_005225 CCCN(CCC)C(=O)c1cc2C(=O)CC(C)(C)Cc2n(c3ccc(Cl)c(Cl)c3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N12 compound treatment 720.0 116.0 0.04 640.0 -108.0 -0.08 -0.0295 -0.3187 3117932 ChemDiv3_005226 CC1(C)Cc2ccccc2C(=N1)c3cc4ccccc4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N13 compound treatment 720.0 116.0 0.04 1240.0 492.0 0.38 0.2962 0.7797 3025409 ChemDiv3_005227 CCc1ccc(/C=C/2\N(C)C(=S)N(C2=O)c3ccc(C)c(C)c3)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N14 compound treatment 680.0 76.3 0.03 1320.0 572.0 0.44 0.3296 0.7493 3117933 ChemDiv3_005228 CCCN(CCC)Cc1c(O)ccc2c(=O)c(coc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N15 compound treatment 840.0 236.0 0.08 520.0 -228.0 -0.18 -0.0646 -0.3326 3025410 ChemDiv3_005229 Oc1ccc(Br)cc1/C=N/c2sc3N4CCC(CC4)c3c2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N16 compound treatment 640.0 36.3 0.01 1520.0 772.0 0.59 0.4281 0.7223 3117934 ChemDiv3_005230 FC(F)(F)c1nnc2Sc3nc4ccccc4nc3Nn12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N17 compound treatment 360.0 -244.0 -0.09 240.0 -508.0 -0.39 -0.337 -0.8434 1245770 ChemDiv3_005231 CCc1cccc(CC)c1N(COC)C(=O)Cn2c(Cc3ccccc3)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N18 compound treatment 1760.0 1160.0 0.41 800.0 51.9 0.04 0.3182 0.7721 3025411 ChemDiv3_005232 CC(=O)Oc1c(C)[n+](C)cc2COC(C)(C)OCc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N19 compound treatment 320.0 -284.0 -0.1 760.0 11.9 0.01 -0.0647 -0.6406 3117935 ChemDiv3_005233 CCCOc1ccc(/C=C\2/SC(=O)N(CN3CCCCC3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N20 compound treatment 240.0 -364.0 -0.13 360.0 -388.0 -0.3 -0.302 -0.9299 3025412 ChemDiv3_005234 CC(C)(C)c1ccc(NC(=O)CCSc2ccc3ccccc3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N21 compound treatment 360.0 -244.0 -0.09 600.0 -148.0 -0.11 -0.1416 -0.9909 1452765 ChemDiv3_005235 O=c1nc(CC#N)sc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N22 compound treatment 1560.0 956.0 0.34 800.0 51.9 0.04 0.268 0.7847 3117936 ChemDiv3_005236 COc1cccc(NC(=O)CCSc2nnc3ccc4ccccc4n23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N23 mock treatment 240.0 -364.0 -0.13 600.0 -148.0 -0.11 -0.1717 -0.998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 N24 mock treatment 360.0 -244.0 -0.09 640.0 -108.0 -0.08 -0.1199 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O01 compound treatment 400.0 -204.0 -0.07 880.0 132.0 0.1 0.0205 0.1646 1414377 ChemDiv3_005237 Cc1ccc(cc1)c2ccc(CCC(=O)O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O02 compound treatment 200.0 -404.0 -0.14 320.0 -428.0 -0.33 -0.3337 -0.9307 3025413 ChemDiv3_005238 CC(NC1(CC(=C)C)CCCCC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O03 compound treatment 280.0 -324.0 -0.11 360.0 -388.0 -0.3 -0.2919 -0.9141 3117937 ChemDiv3_005239 COc1ccc(Br)c2Cc3sc(/N=C/c4ccc(C)cc4)nc3-c21 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O04 compound treatment 360.0 -244.0 -0.09 400.0 -348.0 -0.27 -0.2501 -0.8904 3117938 ChemDiv3_005240 OC(=O)c1cccc2C(CC=C)N(C(=O)c21)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O05 compound treatment 360.0 -244.0 -0.09 280.0 -468.0 -0.36 -0.3153 -0.8529 3025414 ChemDiv3_005241 CCC1CCC(CC1)c2nnc(o2)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O06 compound treatment 320.0 -284.0 -0.1 360.0 -388.0 -0.3 -0.2819 -0.8962 1327740 ChemDiv3_005242 COc1ccc(cc1)c2cc(=O)c3cc(OC(=O)Cc4ccccc4)ccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O07 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 3025415 ChemDiv3_005243 CN1C(=O)/C(=C/c2cc(C)n(c2C)c3ccc(cc3)C(=O)O)/C(=O)NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O08 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 3117939 ChemDiv3_005244 CCC(=O)OCCNc1nc(nc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O09 compound treatment 760.0 156.0 0.06 480.0 -268.0 -0.21 -0.1064 -0.4989 3025416 ChemDiv3_005245 CCOC(=O)C1=C(NC(=O)c2ccc(C)cc2)S/C(=C\c3cccs3)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O10 compound treatment 22680.0 22100.0 7.83 10960.0 10200.0 7.84 11.0813 1.0 3117940 ChemDiv3_005246 FC(F)(F)c1cccc(c1)S(=O)(=O)NC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O11 compound treatment 360.0 -244.0 -0.09 360.0 -388.0 -0.3 -0.2719 -0.8762 3117941 ChemDiv3_005247 CCn1cc(C=C2C(=O)OC(C)(OC2=O)C(C)(C)C)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O12 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 3025417 ChemDiv3_005248 O=C(/C=C/c1ccc2OCOc2c1)/C=C/c3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O13 compound treatment 240.0 -364.0 -0.13 360.0 -388.0 -0.3 -0.302 -0.9299 1501347 ChemDiv3_005249 CC1CC1c2ccc(CCC(=O)Nc3ncc(Cc4cccc(Cl)c4)s3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O14 compound treatment 360.0 -244.0 -0.09 320.0 -428.0 -0.33 -0.2936 -0.8637 3025418 ChemDiv3_005250 CCc1ccc(cc1)N2CN(Cc3ccccc3)CNC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O15 compound treatment 3840.0 3240.0 1.15 240.0 -508.0 -0.39 0.5359 0.442 1874484 ChemDiv3_005251 Cc1ccc(cc1)S(=O)(=O)NC2CCOC(C)(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O16 compound treatment 360.0 -244.0 -0.09 280.0 -468.0 -0.36 -0.3153 -0.8529 3025419 ChemDiv3_005252 CCCN1CNC(=S)N(C1)c2cc(C)ccc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O17 compound treatment 280.0 -324.0 -0.11 400.0 -348.0 -0.27 -0.2702 -0.9288 3117942 ChemDiv3_005253 CCOc1ccc(cc1OC)C(NC(=O)c2ccco2)NC(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O18 compound treatment 200.0 -404.0 -0.14 280.0 -468.0 -0.36 -0.3554 -0.9186 3117943 ChemDiv3_005254 CC1CCCC(C1=O)C2(O)C(=O)Nc3ccccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O19 compound treatment 320.0 -284.0 -0.1 240.0 -508.0 -0.39 -0.347 -0.8613 3025420 ChemDiv3_005255 Clc1c2C(=O)/C(=C\NC3CCCCC3)/Nc2ccc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O20 compound treatment 160.0 -444.0 -0.16 240.0 -508.0 -0.39 -0.3872 -0.9203 3117944 ChemDiv3_005256 O=C1OC(Nc2ccc(cc2)S(=O)(=O)Nc3ccccn3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O21 compound treatment 200.0 -404.0 -0.14 360.0 -388.0 -0.3 -0.312 -0.9436 3025421 ChemDiv3_005257 COC(=O)CC/1SC(=O)N\C1=N/c2ccc(O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O22 compound treatment 400.0 -204.0 -0.07 200.0 -548.0 -0.42 -0.3487 -0.8166 3117945 ChemDiv3_005258 CC(=C1C(=O)c2ccccc2C1=O)N3CCC(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O23 mock treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 O24 mock treatment 200.0 -404.0 -0.14 400.0 -348.0 -0.27 -0.2903 -0.9572 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P01 compound treatment 240.0 -364.0 -0.13 320.0 -428.0 -0.33 -0.3237 -0.9166 1382485 ChemDiv3_005259 O=C(N1N=C(CC1c2ccccc2)c3ccccc3)c4cc5ccccc5oc4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P02 compound treatment 200.0 -404.0 -0.14 280.0 -468.0 -0.36 -0.3554 -0.9186 3117946 ChemDiv3_005260 Cc1cc(ccc1Cl)/C(=N/O)/C(C)(C)NO 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P03 compound treatment 280.0 -324.0 -0.11 280.0 -468.0 -0.36 -0.3353 -0.8888 3117947 ChemDiv3_005261 CC1CCN(CC1)C(=S)SCC(=O)n2c(C)c(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P04 compound treatment 280.0 -324.0 -0.11 160.0 -588.0 -0.45 -0.4005 -0.8596 3025422 ChemDiv3_005262 COc1ccc(Nc2ccc3nnc(c4ccc(Br)cc4)n3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P05 compound treatment 240.0 -364.0 -0.13 240.0 -508.0 -0.39 -0.3671 -0.8934 3117948 ChemDiv3_005263 CC1(C)CC(=O)C2=C(C1)N=C3C(C2c4cccc(Br)c4)C(=O)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P06 compound treatment 720.0 116.0 0.04 160.0 -588.0 -0.45 -0.2901 -0.6399 3025423 ChemDiv3_005264 CCc1ccc2n(CC)c3nc4ccccc4nc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P07 compound treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 3117949 ChemDiv3_005265 COC(=O)C/1=C(C)N(CC2CCCO2)C(=O)\C1=C/c3cc(C)n(c3C)c4ccc(OC)c(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P08 compound treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 3025424 ChemDiv3_005266 CC(CN1CCCC1)OC(=O)c2cc(cc(c2)C(C)(C)C)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P09 compound treatment 400.0 -204.0 -0.07 480.0 -268.0 -0.21 -0.1967 -0.9014 3117950 ChemDiv3_005267 Cc1cc(ccc1/C=C/2\NC(=O)N(Cc3ccccc3)C2=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P10 compound treatment 640.0 36.3 0.01 480.0 -268.0 -0.21 -0.1365 -0.6616 3117951 ChemDiv3_005268 CCN1C(=O)c2ccc(cc2C1=O)C(=O)Nc3cc(cc(c3)C(=O)O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P11 compound treatment 320.0 -284.0 -0.1 400.0 -348.0 -0.27 -0.2602 -0.9109 3025425 ChemDiv3_005269 OC(=O)c1cccc(c1)n2cccc2C=C3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P12 compound treatment 440.0 -164.0 -0.06 280.0 -468.0 -0.36 -0.2952 -0.8109 3118091 ChemDiv3_005270 CCC1(CC)Cc2ccccc2C(=N1)c3cc4ccccc4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P13 compound treatment 440.0 -164.0 -0.06 360.0 -388.0 -0.3 -0.2518 -0.8293 3025426 ChemDiv3_005271 Cc1cc(I)ccc1n2nc(cc2O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P14 compound treatment 240.0 -364.0 -0.13 320.0 -428.0 -0.33 -0.3237 -0.9166 3118092 ChemDiv3_005272 COc1ccc(cc1OC)c2c(oc3c(CN4CCCC(C)C4)c(O)ccc3c2=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P15 compound treatment 1520.0 916.0 0.33 200.0 -548.0 -0.42 -0.0677 -0.1274 3025475 ChemDiv3_005273 O=C(Nc1ccc(CN2CCOCC2)cc1)/C=C/c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P16 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 3025476 ChemDiv3_005274 CCc1cccc(OCC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nccs3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P17 compound treatment 240.0 -364.0 -0.13 280.0 -468.0 -0.36 -0.3454 -0.9045 3025477 ChemDiv3_005275 C=CCn1c(=O)[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P18 compound treatment 320.0 -284.0 -0.1 280.0 -468.0 -0.36 -0.3253 -0.8716 3025478 ChemDiv3_005276 CN(CC(=O)N1CCc2ccccc2C1)S(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P19 compound treatment 360.0 -244.0 -0.09 280.0 -468.0 -0.36 -0.3153 -0.8529 3025479 ChemDiv3_005277 O=C1S/C(=C\c2cn(Cc3ccccc3)c4ccccc24)/C(=O)N1CN5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P20 compound treatment 280.0 -324.0 -0.11 440.0 -308.0 -0.24 -0.2485 -0.9449 3025480 ChemDiv3_005278 O=C(CCSc1ccc2ccccc2n1)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P21 compound treatment 240.0 -364.0 -0.13 280.0 -468.0 -0.36 -0.3454 -0.9045 3025481 ChemDiv3_005279 CCCN1C(=O)/C(=C/c2cc(C)n(c2C)c3ccc(Cl)cc3)/NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P22 compound treatment 280.0 -324.0 -0.11 240.0 -508.0 -0.39 -0.3571 -0.878 3118093 ChemDiv3_005280 O=C(CSc1nnc2scc(c3ccccc3)n12)N4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P23 mock treatment 240.0 -364.0 -0.13 320.0 -428.0 -0.33 -0.3237 -0.9166 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2015 P24 mock treatment 320.0 -284.0 -0.1 800.0 51.9 0.04 -0.043 -0.3975 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A01 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 3025482 ChemDiv3_005281 Cc1nc(CSc2nnc3scc(c4ccccc4)n23)cs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A02 compound treatment 280.0 -663.0 -0.24 600.0 -23.2 -0.02 -0.1788 -0.7586 3118094 ChemDiv3_005282 COc1cc2nc(oc(=O)c2cc1OC)c3ccc4C(=O)N(CC(C)C)C(=O)c4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A03 compound treatment 240.0 -703.0 -0.25 200.0 -423.0 -0.32 -0.406 -0.9914 1863770 ChemDiv3_005283 COc1cc(CNC2C3CC4CC(C3)CC2C4)ccc1OCc5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A04 compound treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 1692810 ChemDiv3_005284 CCN(CC)C(=O)CSc1nc2n(C)c(=O)n(C)c(=O)c2n1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A05 compound treatment 200.0 -743.0 -0.26 1200.0 577.0 0.44 0.1269 0.2462 3118095 ChemDiv3_005285 CC/N=C/1\S/C(=C\c2cn(CC(=O)Nc3cccc(C)c3)c4ccccc24)/C(=O)N1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A06 compound treatment 280.0 -663.0 -0.24 360.0 -263.0 -0.2 -0.3091 -0.9972 3025483 ChemDiv3_005286 CCCCn1c(nc2c(=O)oc3ccccc3c12)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A07 compound treatment 320.0 -623.0 -0.22 560.0 -63.2 -0.05 -0.1905 -0.8424 3025484 ChemDiv3_005287 O=C1N(CCn2c(=O)oc3ccccc23)C(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A08 compound treatment 360.0 -583.0 -0.21 240.0 -383.0 -0.29 -0.3542 -0.9851 3118096 ChemDiv3_005288 CC(C)c1ccc(cc1)C2Nc3ccccc3S(=O)(=O)N2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A09 compound treatment 200.0 -743.0 -0.26 200.0 -423.0 -0.32 -0.416 -0.9946 3118097 ChemDiv3_005289 COc1ccc(NC(=O)C2CC(=O)N(C(=O)N2NC(=O)c3ccncc3)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A10 compound treatment 240.0 -703.0 -0.25 160.0 -463.0 -0.36 -0.4277 -0.9849 3025485 ChemDiv3_005290 Cc1cc(/C=C\2/C(=N)N3C=CSC3=NC2=O)c(C)n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A11 compound treatment 200.0 -743.0 -0.26 200.0 -423.0 -0.32 -0.416 -0.9946 3118098 ChemDiv3_005291 Cc1ccc(O)c(c1)C(CC(=O)NCC2(CCOCC2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A12 compound treatment 200.0 -743.0 -0.26 360.0 -263.0 -0.2 -0.3291 -0.9914 3025486 ChemDiv3_005292 Cc1ccc2NC(C3CCOC3c2c1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A13 compound treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 1685959 ChemDiv3_005293 CCCCN(C)c1nc(CC)c2COC(C)(C)Cc2c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A14 compound treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 3025487 ChemDiv3_005294 Fc1ccccc1COc2ccc3c(=O)c(coc3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A15 compound treatment 360.0 -583.0 -0.21 200.0 -423.0 -0.32 -0.3759 -0.9761 3118099 ChemDiv3_005295 CCc1nc2sc3c(SCC=C)ncnc3c2c4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A16 compound treatment 240.0 -703.0 -0.25 280.0 -343.0 -0.26 -0.3625 -0.9996 3118100 ChemDiv3_005296 O=C(C1CCCN(C1)C(=O)c2ccccc2)N3CCC(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A17 compound treatment 200.0 -743.0 -0.26 240.0 -383.0 -0.29 -0.3943 -0.9985 3025488 ChemDiv3_005297 CCOC(=O)c1c(N)oc2c(c3ccc(CC)cc3)c4c(C(=O)OCC)c(N)oc4cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A18 compound treatment 280.0 -663.0 -0.24 320.0 -303.0 -0.23 -0.3308 -1.0 3118101 ChemDiv3_005298 CCCN1CCC(CC1)N2CCCC(C2)C(=O)N(C)CCc3ccc(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A19 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3025489 ChemDiv3_005299 CCCCc1ccc(NCc2nc(no2)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A20 compound treatment 360.0 -583.0 -0.21 400.0 -223.0 -0.17 -0.2673 -0.9957 3118102 ChemDiv3_005300 OC(=O)c1cccc(NC(=O)CCN2C(=O)c3ccccc3S2(=O)=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A21 compound treatment 160.0 -783.0 -0.28 200.0 -423.0 -0.32 -0.426 -0.9969 3025490 ChemDiv3_005301 CN1CCN(CC1)C(=O)NCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A22 compound treatment 200.0 -743.0 -0.26 280.0 -343.0 -0.26 -0.3726 -1.0 3118103 ChemDiv3_005302 CCOc1ccc2c(c1)sc3c(C)cc(=O)oc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A23 mock treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 A24 mock treatment 240.0 -703.0 -0.25 200.0 -423.0 -0.32 -0.406 -0.9914 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B01 compound treatment 640.0 -303.0 -0.11 160.0 -463.0 -0.36 -0.3273 -0.8812 3118104 ChemDiv3_005303 CCN(CC)c1ccc(/N=c\2/ccc3ccccc3n2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B02 compound treatment 200.0 -743.0 -0.26 240.0 -383.0 -0.29 -0.3943 -0.9985 3025491 ChemDiv3_005304 Cc1n[nH]c(C)c1CCCOc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B03 compound treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 3118105 ChemDiv3_005305 CC1N(C)C(=O)N(OC1=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B04 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 3025492 ChemDiv3_005306 COC(=O)c1cc(on1)c2cccc(OC)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B05 compound treatment 320.0 -623.0 -0.22 200.0 -423.0 -0.32 -0.3859 -0.9823 1346624 ChemDiv3_005307 C1CCC(CC1)c2ccc3n4CCN=C5CCCc(c54)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B06 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 1692119 ChemDiv3_005308 Cc1cccc(NC(=O)C2c3ccccc3Oc4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B07 compound treatment 280.0 -663.0 -0.24 360.0 -263.0 -0.2 -0.3091 -0.9972 3025493 ChemDiv3_005309 COC(=O)N(C)c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B08 compound treatment 280.0 -663.0 -0.24 240.0 -383.0 -0.29 -0.3742 -0.9938 3118106 ChemDiv3_005310 CC(Oc1ccc(Cl)cc1C)C(=O)N2CCN(CC2)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B09 compound treatment 200.0 -743.0 -0.26 280.0 -343.0 -0.26 -0.3726 -1.0 1341182 ChemDiv3_005311 CC1=C(C#N)C(C2=C(CC(CC2=O)c3ccccc3)N1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B10 compound treatment 200.0 -743.0 -0.26 240.0 -383.0 -0.29 -0.3943 -0.9985 3025494 ChemDiv3_005312 COc1cccc(/C=C/2\CCC/C(=C/c3cccc(OC)c3OC)/C2=O)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B11 compound treatment 280.0 -663.0 -0.24 640.0 16.8 0.01 -0.1571 -0.6674 1875367 ChemDiv3_005313 CCn1c(N)c(sc1=S)C(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B12 compound treatment 360.0 -583.0 -0.21 360.0 -263.0 -0.2 -0.289 -0.9999 3118107 ChemDiv3_005314 CCn1c(S)nnc1c2csc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B13 compound treatment 320.0 -623.0 -0.22 4840.0 4220.0 3.24 2.133 0.6573 3118108 ChemDiv3_005315 Cc1ccc(c(C)c1C)S(=O)(=O)NCCN2CCN(CC2)S(=O)(=O)c3ccc(C)c(C)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B14 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 1248039 ChemDiv3_005316 Cc1cc(NC(=O)CCC2CCCCC2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B15 compound treatment 360.0 -583.0 -0.21 240.0 -383.0 -0.29 -0.3542 -0.9851 3118109 ChemDiv3_005317 Cc1ccc(cc1CNS(=O)(=O)C)c2nn(C)c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B16 compound treatment 480.0 -463.0 -0.16 240.0 -383.0 -0.29 -0.3241 -0.962 1550315 ChemDiv3_005318 OC(=O)C1C(C2CC1C=C2)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B17 compound treatment 200.0 -743.0 -0.26 280.0 -343.0 -0.26 -0.3726 -1.0 3025495 ChemDiv3_005319 COC(=O)CCn1nc(c2ccc(Cl)cc2)c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B18 compound treatment 200.0 -743.0 -0.26 320.0 -303.0 -0.23 -0.3509 -0.9981 1302577 ChemDiv3_005320 CCCc1ccc(CC2(CC(=O)OCC)C(=O)c3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B19 compound treatment 360.0 -583.0 -0.21 400.0 -223.0 -0.17 -0.2673 -0.9957 3118110 ChemDiv3_005321 CC/1=NN(C(=S)\C1=C/Nc2nc(cs2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B20 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 1585203 ChemDiv3_005322 O=C(C1CC1)N2CCN(CC2)c3ncccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B21 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3118111 ChemDiv3_005323 O=C(CN1C(=O)c2cccc3cccc1c23)N(Cc4ccccc4)Cc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B22 compound treatment 360.0 -583.0 -0.21 400.0 -223.0 -0.17 -0.2673 -0.9957 3025496 ChemDiv3_005324 Cc1ccc(NCc2nnc(SCC(=O)c3ccccc3)n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B23 mock treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 B24 mock treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C01 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 3118112 ChemDiv3_005325 Clc1ccc(cc1)c2csc3nnc(SCC(=O)NCc4ccc5OCOc5c4)n23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C02 compound treatment 160.0 -783.0 -0.28 280.0 -343.0 -0.26 -0.3826 -0.9997 3118113 ChemDiv3_005326 COc1ccc(cc1)n2c(n[nH]c2=S)c3ccc(cc3)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C03 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 1863776 ChemDiv3_005327 CCOc1cc(CNC2(CC3CC4CC(C3)C2)C4)ccc1OCc5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C04 compound treatment 400.0 -543.0 -0.19 200.0 -423.0 -0.32 -0.3658 -0.9687 3118236 ChemDiv3_005328 CCn1c(SCc2ccc(Br)cc2)nnc1c3ccncc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C05 compound treatment 280.0 -663.0 -0.24 200.0 -423.0 -0.32 -0.3959 -0.9874 1718306 ChemDiv3_005329 CC(c1ccccc1)n2c(COc3ccccc3)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C06 compound treatment 200.0 -743.0 -0.26 280.0 -343.0 -0.26 -0.3726 -1.0 3025497 ChemDiv3_005330 FC(F)(F)c1nc2c(=O)oc3ccccc3c2n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C07 compound treatment 1480.0 538.0 0.19 320.0 -303.0 -0.23 -0.0298 -0.099 3118237 ChemDiv3_005331 O=C1N(CCCn2c(=O)oc3ccccc23)C(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C08 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 3025498 ChemDiv3_005332 COC(=O)c1ccc2NC(C3C4CCC(C4)C3c2c1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C09 compound treatment 360.0 -583.0 -0.21 200.0 -423.0 -0.32 -0.3759 -0.9761 3118238 ChemDiv3_005333 Cn1nc(SCC(=O)n2c3CCCCc3c4ccccc24)sc1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C10 compound treatment 280.0 -663.0 -0.24 160.0 -463.0 -0.36 -0.4176 -0.9798 3118239 ChemDiv3_005334 CC1=CN2C(=NC(=O)/C(=C\c3cc(C)n(Cc4ccccc4)c3C)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C11 compound treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 3025499 ChemDiv3_005335 OC(=O)CCN1C(=O)SC(CC(=O)Nc2nccs2)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C12 compound treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 3118240 ChemDiv3_005336 COc1cccc(c1)N2C(CC=C)c3cccc(C(=O)O)c3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C13 compound treatment 360.0 -583.0 -0.21 400.0 -223.0 -0.17 -0.2673 -0.9957 1674657 ChemDiv3_005337 CC1(C)Cc2c(C#N)c(NCC3CCCO3)nc(c4ccccc4)c2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C14 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3025500 ChemDiv3_005338 CCOC(=O)c1sc2ncn3c(nnc3c2c1C)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C15 compound treatment 320.0 -623.0 -0.22 480.0 -143.0 -0.11 -0.2339 -0.9482 3118241 ChemDiv3_005339 Cc1cc(Oc2ccccc2)nc(Oc3ccc(OCCOc4ccc(Br)cc4)nn3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C16 compound treatment 280.0 -663.0 -0.24 360.0 -263.0 -0.2 -0.3091 -0.9972 3025501 ChemDiv3_005340 COc1ccc(cc1)C(=O)N2CCCC(C2)C(=O)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C17 compound treatment 360.0 -583.0 -0.21 200.0 -423.0 -0.32 -0.3759 -0.9761 3118242 ChemDiv3_005341 FC(F)(F)c1cccc(Cc2cn3cc(nc3s2)c4cc5ccccc5oc4=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C18 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3025502 ChemDiv3_005342 O=C(C1CCCN(C1)S(=O)(=O)c2ccccc2)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C19 compound treatment 280.0 -663.0 -0.24 360.0 -263.0 -0.2 -0.3091 -0.9972 3118243 ChemDiv3_005343 Cc1ccc(cc1)c2noc(CN3CCN(CC3)c4ccccc4F)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C20 compound treatment 600.0 -343.0 -0.12 200.0 -423.0 -0.32 -0.3157 -0.91 3025503 ChemDiv3_005344 Cc1ccc(NC(=O)CCN2C(=O)c3ccccc3S2(=O)=O)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C21 compound treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 3118244 ChemDiv3_005345 OCCN1CCN(CC1)C(=O)NCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C22 compound treatment 360.0 -583.0 -0.21 280.0 -343.0 -0.26 -0.3324 -0.9928 3118245 ChemDiv3_005346 CCn1/c(=N\c2ccc(C)cc2)/ccc3cc(C)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C23 mock treatment 160.0 -783.0 -0.28 240.0 -383.0 -0.29 -0.4043 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 C24 mock treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D01 compound treatment 4840.0 3900.0 1.38 360.0 -263.0 -0.2 0.8348 0.5974 3025504 ChemDiv3_005347 OC(=O)c1cccc(Nc2nc(Nc3ccccc3)nc(n2)N4CCCC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D02 compound treatment 440.0 -503.0 -0.18 320.0 -303.0 -0.23 -0.2907 -0.9913 3118246 ChemDiv3_005348 CC(C)c1ccc(OCCCN2CCCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D03 compound treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 1230490 ChemDiv3_005349 Cc1ccc2n3CCN(C=O)C4CCCc(c43)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D04 compound treatment 360.0 -583.0 -0.21 280.0 -343.0 -0.26 -0.3324 -0.9928 3118247 ChemDiv3_005350 CC1CN/C(=C/C(=O)/C=C/c2ccccc2)/C(=O)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D05 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 1147135 ChemDiv3_005351 CC(C)(C)c1ccc2n3CCN(CCC#N)C4CCCc(c43)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D06 compound treatment 280.0 -663.0 -0.24 200.0 -423.0 -0.32 -0.3959 -0.9874 3025635 ChemDiv3_005352 CCc1c(C)sc(NC(=O)C2c3ccccc3Oc4ccccc24)c1C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D07 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 3118248 ChemDiv3_005353 CN(C(=O)C)c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D08 compound treatment 320.0 -623.0 -0.22 240.0 -383.0 -0.29 -0.3642 -0.99 3118249 ChemDiv3_005354 Cc1cc(Cl)ccc1OCCCC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ncccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D09 compound treatment 2600.0 1660.0 0.59 360.0 -263.0 -0.2 0.2729 0.4389 3025636 ChemDiv3_005355 OC(=O)COc1ccccc1C2Nc3ccccc3-c4nnc(SCC=C)nc4O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D10 compound treatment 600.0 -343.0 -0.12 240.0 -383.0 -0.29 -0.294 -0.9235 3118250 ChemDiv3_005356 Cc1ccc(cc1C)c2cc(n3nc(cc3n2)C(=O)Nc4ccn(Cc5ccccc5)n4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D11 compound treatment 360.0 -583.0 -0.21 640.0 16.8 0.01 -0.137 -0.6618 3025637 ChemDiv3_005357 Nc1c(sc(=S)n1CC=C)C(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D12 compound treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 3118251 ChemDiv3_005358 Cc1cc(C(=O)N2N=C(CC2(O)C(F)(F)F)C3CC3)c4ccccc4n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D13 compound treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 3025638 ChemDiv3_005359 Oc1c(CC=C)cccc1/C=N/c2cccn3cc(nc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D14 compound treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 1607969 ChemDiv3_005360 Cc1cc(NC(=O)C2CCCCC2C(=O)O)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D15 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3118252 ChemDiv3_005361 Cc1cc(C)nc(SCc2cc(ccc2C)c3nn(C)c(=O)c4ccccc34)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D16 compound treatment 200.0 -743.0 -0.26 320.0 -303.0 -0.23 -0.3509 -0.9981 3025639 ChemDiv3_005362 Cc1cc(C)n(n1)C(=O)CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D17 compound treatment 320.0 -623.0 -0.22 880.0 257.0 0.2 -0.0168 -0.0566 3118253 ChemDiv3_005363 Clc1ccc(cc1)c2nn(CCC(=O)NCCN3CCOCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D18 compound treatment 320.0 -623.0 -0.22 160.0 -463.0 -0.36 -0.4076 -0.9737 1244787 ChemDiv3_005364 Cc1cccc(N2CCN(CC2)C(=O)CCC(=O)O)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D19 compound treatment 400.0 -543.0 -0.19 400.0 -223.0 -0.17 -0.2573 -0.9983 3118254 ChemDiv3_005365 CCCc1nnc(N/C=C\2/C=C(OC2=O)c3ccccc3)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D20 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 1550669 ChemDiv3_005366 O=C(N1CCN(CC1)C(c2ccccc2)c3ccccc3)c4cc5ccccc5c(=O)o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D21 compound treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 3118255 ChemDiv3_005367 CCCC1(CNCC2(C)CNC1)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D22 compound treatment 240.0 -703.0 -0.25 400.0 -223.0 -0.17 -0.2974 -0.9833 1138350 ChemDiv3_005368 O=C(Nc1nnn[nH]1)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D23 mock treatment 240.0 -703.0 -0.25 200.0 -423.0 -0.32 -0.406 -0.9914 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 D24 mock treatment 320.0 -623.0 -0.22 520.0 -103.0 -0.08 -0.2122 -0.9044 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E01 compound treatment 520.0 -423.0 -0.15 8080.0 7460.0 5.72 3.942 0.6884 3118256 ChemDiv3_005369 Clc1ccc(cc1)c2csc3nnc(SCCC(=O)NCCc4ccccc4)n23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E02 compound treatment 920.0 -22.5 -0.01 1600.0 977.0 0.75 0.5246 0.6995 3118257 ChemDiv3_005370 Fc1ccc(cc1)n2c(n[nH]c2=S)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E03 compound treatment 360.0 -583.0 -0.21 360.0 -263.0 -0.2 -0.289 -0.9999 1863813 ChemDiv3_005371 COc1cccc(CNC(C)C2(CC3CC4CC(C3)C2)C4)c1OCc5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E04 compound treatment 320.0 -623.0 -0.22 1840.0 1220.0 0.93 0.5044 0.5255 3118258 ChemDiv3_005372 CC(C)Cn1c(SCc2ccccc2)nnc1c3ccncc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E05 compound treatment 560.0 -383.0 -0.14 600.0 -23.2 -0.02 -0.1086 -0.7932 1732699 ChemDiv3_005373 CC(C)C(=O)Nc1cccc(c1)c2cn3c(C)cccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E06 compound treatment 480.0 -463.0 -0.16 320.0 -303.0 -0.23 -0.2806 -0.9853 3025640 ChemDiv3_005374 CC1(C)Cc2c(c3ccccc3n2c4ccccc4)C(C)(C)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E07 compound treatment 920.0 -22.5 -0.01 3560.0 2940.0 2.25 1.5886 0.7046 3118259 ChemDiv3_005375 COC(=O)/C(=C/c1ccc2OCOc2c1)/NC(=O)c3ccc(cc3)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E08 compound treatment 4240.0 3300.0 1.17 360.0 -263.0 -0.2 0.6843 0.5764 3118260 ChemDiv3_005376 C=CCNC(=O)c1ccc2NC(C3C4CCC(C4)C3c2c1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E09 compound treatment 520.0 -423.0 -0.15 560.0 -63.2 -0.05 -0.1403 -0.8906 3025641 ChemDiv3_005377 NC(=O)C1CCN(CC1)C(=O)CSc2ncccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E10 compound treatment 2360.0 1420.0 0.5 600.0 -23.2 -0.02 0.343 0.6816 3118393 ChemDiv3_005378 CCOc1cc(/C=C/2\C(=N)N3C(=CSC3=NC2=O)C)ccc1OCc4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E11 compound treatment 2880.0 1940.0 0.69 680.0 56.8 0.04 0.5168 0.7504 3025677 ChemDiv3_005379 O=C1CSC(=N1)Nc2nccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E12 compound treatment 4800.0 3860.0 1.37 3000.0 2380.0 1.82 2.2579 0.9899 1523673 ChemDiv3_005380 CN1C(CC=C(C)C1c2ccccc2)c3cnc(c(C)c3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E13 compound treatment 600.0 -343.0 -0.12 520.0 -103.0 -0.08 -0.142 -0.9786 3025678 ChemDiv3_005381 CCc1nc2sc3c(NCCc4ccccc4)ncnc3c2c5CCCCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E14 compound treatment 400.0 -543.0 -0.19 840.0 217.0 0.17 -0.0184 -0.0723 3118394 ChemDiv3_005382 COc1ccc(cc1)c2c/c(=N\CCc3ccccc3)/c4cc(C)ccc4o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E15 compound treatment 720.0 -223.0 -0.08 480.0 -143.0 -0.11 -0.1336 -0.9868 1875998 ChemDiv3_005383 Cc1cc(Oc2ccc(=O)n(C)n2)nc(Oc3ccc(=O)n(C)n3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E16 compound treatment 2400.0 1460.0 0.52 640.0 16.8 0.01 0.3747 0.7245 3025679 ChemDiv3_005384 Clc1cccc(CN2CCCC(C2)C(=O)N3CCCCCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E17 compound treatment 1600.0 658.0 0.23 800.0 177.0 0.14 0.2609 0.9668 3118395 ChemDiv3_005385 Clc1ccccc1Cc2cn3cc(nc3s2)c4cc5ccccc5oc4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E18 compound treatment 880.0 -62.5 -0.02 400.0 -223.0 -0.17 -0.1369 -0.792 3118396 ChemDiv3_005386 CCn1c2ccccc2c3cc(CN4CCC(CC4)N5CCCCC5)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E19 compound treatment 1640.0 698.0 0.25 560.0 -63.2 -0.05 0.1406 0.5578 3025680 ChemDiv3_005387 O=C(NCN1C(=O)C2C3CC(C=C3)C2C1=O)Nc4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E20 compound treatment 360.0 -583.0 -0.21 2440.0 1820.0 1.39 0.8401 0.5958 3118397 ChemDiv3_005388 O=C(CCN1C(=O)c2ccccc2S1(=O)=O)Nc3ccc4CCc5cccc3c54 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E21 compound treatment 1440.0 498.0 0.18 800.0 177.0 0.14 0.2208 0.9916 3025681 ChemDiv3_005389 CN(C)S(=O)(=O)c1ccc(cc1)C(=O)NCCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E22 compound treatment 480.0 -463.0 -0.16 880.0 257.0 0.2 0.0234 0.0911 3118398 ChemDiv3_005390 Cn1/c(=N/c2ccccc2C(=O)O)/sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E23 mock treatment 1120.0 178.0 0.06 3120.0 2500.0 1.92 1.3999 0.7299 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 E24 mock treatment 200.0 -743.0 -0.26 2680.0 2060.0 1.58 0.9303 0.5811 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F01 compound treatment 2800.0 1860.0 0.66 7080.0 6460.0 4.96 3.9711 0.7941 3118399 ChemDiv3_005391 O=C(NCCN1C(=O)C2C3CC(C=C3)C2C1=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F02 compound treatment 1680.0 738.0 0.26 2320.0 1700.0 1.3 1.1061 0.8325 1301199 ChemDiv3_005392 OC(=O)c1ccc(NC(CC(=O)c2ccc(Cl)cc2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F03 compound treatment 920.0 -22.5 -0.01 480.0 -143.0 -0.11 -0.0834 -0.7564 1472870 ChemDiv3_005393 CC(C)c1ccc2[nH]c3C(=O)CCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F04 compound treatment 1240.0 298.0 0.11 400.0 -223.0 -0.17 -0.0466 -0.2313 3118400 ChemDiv3_005394 COC(=O)C1=C(C(c2ccc(cc2)C(=O)OC)n3nnnc3N1)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F05 compound treatment 1120.0 178.0 0.06 1880.0 1260.0 0.96 0.7268 0.7517 1302281 ChemDiv3_005395 Cc1ccc(NC(=S)N2CCn3c4C2CCc4c(=O)c5cc(C)ccc35)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F06 compound treatment 800.0 -143.0 -0.05 2560.0 1940.0 1.49 1.0157 0.6827 3118401 ChemDiv3_005396 COc1ccccc1N2CCN(CC2)C(=O)C3C(C4OC3C=C4)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F07 compound treatment 920.0 -22.5 -0.01 8440.0 7820.0 6.0 4.2378 0.7062 3025682 ChemDiv3_005397 C/C(=C\C(=O)Nc1ccccc1)/N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F08 compound treatment 1160.0 218.0 0.08 880.0 257.0 0.2 0.194 0.9162 1123206 ChemDiv3_005398 O=C(CCC1CCCCC1)Nc2ccc(cc2)S(=O)(=O)Nc3ncccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F09 compound treatment 1040.0 97.5 0.03 2440.0 1820.0 1.39 1.0107 0.7244 1399432 ChemDiv3_005399 Cc1cccc(OCC(=O)N2CCCc3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F10 compound treatment 3000.0 2060.0 0.73 2800.0 2180.0 1.67 1.6978 0.931 3118402 ChemDiv3_005400 Cc1ccc(cc1)n2c(S)nnc2c3nn(C)cc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F11 compound treatment 840.0 -103.0 -0.04 1360.0 737.0 0.57 0.3743 0.6603 3118403 ChemDiv3_005401 COc1ccc(cc1)n2c(N)c(sc2=S)c3nc4ccccc4n3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F12 compound treatment 4040.0 3100.0 1.1 680.0 56.8 0.04 0.8078 0.7346 3025683 ChemDiv3_005402 COc1ccc(/N=C/c2c(C)c(C#N)c3[nH]c4ccccc4n3c2=O)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F13 compound treatment 4920.0 3980.0 1.41 6920.0 6300.0 4.83 4.416 0.8769 3118404 ChemDiv3_005403 Oc1ccc2ccccc2c1/C=N/c3cccn4cc(nc34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F14 compound treatment 2520.0 1580.0 0.56 1480.0 857.0 0.66 0.8608 0.9968 1691290 ChemDiv3_005404 COc1cccc(c1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nccc(C)n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F15 compound treatment 760.0 -183.0 -0.06 680.0 56.8 0.04 -0.015 -0.1917 3025684 ChemDiv3_005405 CCN(CC)C(=O)CCn1nc(c2ccc(C)cc2)c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F16 compound treatment 760.0 -183.0 -0.06 440.0 -183.0 -0.14 -0.1452 -0.938 1623425 ChemDiv3_005406 Cc1cc(NS(=O)(=O)c2ccc(NC(=O)c3ccncc3)cc2)nc(C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F17 compound treatment 1640.0 698.0 0.25 960.0 337.0 0.26 0.3578 0.9998 3025685 ChemDiv3_005407 Clc1ccc(cc1)c2nn(CCC(=O)N3CCN(Cc4ccccc4)CC3)c(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F18 compound treatment 720.0 -223.0 -0.08 4400.0 3780.0 2.9 1.9944 0.6876 1377550 ChemDiv3_005408 CCOC(=O)c1c(NC(=O)c2cc3ccccc3c(=O)o2)sc4CCCCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F19 compound treatment 640.0 -303.0 -0.11 3760.0 3140.0 2.41 1.6269 0.6749 3025686 ChemDiv3_005409 CCOc1ccc(cc1)S(=O)(=O)/N=C(\N)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F20 compound treatment 640.0 -303.0 -0.11 600.0 -23.2 -0.02 -0.0885 -0.8134 1483573 ChemDiv3_005410 O=C(Nc1ccc2OCOc2c1)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F21 compound treatment 760.0 -183.0 -0.06 2720.0 2100.0 1.61 1.0925 0.6781 3025687 ChemDiv3_005411 C(c1ccccc1)[n+]2cccc(c2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F22 compound treatment 3200.0 2260.0 0.8 6440.0 5820.0 4.47 3.724 0.8208 3118405 ChemDiv3_005412 COc1ccc(CC(=O)Nc2ccc3c(cc(=O)oc3c2)C(F)(F)F)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F23 mock treatment 960.0 17.5 0.01 1040.0 417.0 0.32 0.2306 0.7207 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 F24 mock treatment 1040.0 97.5 0.03 5800.0 5180.0 3.97 2.8347 0.7132 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G01 compound treatment 4560.0 3620.0 1.28 840.0 217.0 0.17 1.0251 0.7922 1863502 ChemDiv3_005413 CCOc1cc(CNc2ccc(cc2)N3CCOCC3)ccc1OCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G02 compound treatment 720.0 -223.0 -0.08 320.0 -303.0 -0.23 -0.2204 -0.8967 3025688 ChemDiv3_005414 COc1ccccc1n2c(n[nH]c2=S)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G03 compound treatment 760.0 -183.0 -0.06 680.0 56.8 0.04 -0.015 -0.1917 1863847 ChemDiv3_005415 CCOc1cc(CNc2ccc(NC(=O)CC)cc2)ccc1OCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G04 compound treatment 1200.0 258.0 0.09 2440.0 1820.0 1.39 1.0508 0.7518 3025689 ChemDiv3_005416 COc1ccc(cc1)C2(CNC(=S)Nc3ccccc3)CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G05 compound treatment 680.0 -263.0 -0.09 1440.0 817.0 0.63 0.3775 0.5956 1476189 ChemDiv3_005417 CCOc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3cn4cccc(C)c4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G06 compound treatment 520.0 -423.0 -0.15 800.0 177.0 0.14 -0.01 -0.0495 3025690 ChemDiv3_005418 CC(C)CCn1c(=O)n(CC(C)C)c2[nH]c(S)nc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G07 compound treatment 760.0 -183.0 -0.06 760.0 137.0 0.11 0.0285 0.2308 3118406 ChemDiv3_005419 CNC(=O)/C(=C\c1ccc2OCOc2c1)/NC(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G08 compound treatment 400.0 -543.0 -0.19 1560.0 937.0 0.72 0.3725 0.5003 1861617 ChemDiv3_005420 O=C(Nc1ccccc1N2CCCC2)c3cccc(OCc4ccccc4)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G09 compound treatment 3720.0 2780.0 0.99 600.0 -23.2 -0.02 0.6841 0.6942 3118407 ChemDiv3_005421 Cn1c(=O)n(C)c2ncn(CC/N=C/3\CCCN3)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G10 compound treatment 1080.0 138.0 0.05 1520.0 897.0 0.69 0.5213 0.7553 3025733 ChemDiv3_005422 CCN(CC)Cn1nc2-c3ccccc3-c4cccc(c1=O)c42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G11 compound treatment 440.0 -503.0 -0.18 520.0 -103.0 -0.08 -0.1821 -0.9334 3118408 ChemDiv3_005423 FC(F)(F)c1cccc(NC(=O)CC2SC(=O)NC2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G12 compound treatment 1240.0 298.0 0.11 360.0 -263.0 -0.2 -0.0683 -0.2994 1400276 ChemDiv3_005424 COC(=O)CN(c1cccc2ccccc12)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G13 compound treatment 480.0 -463.0 -0.16 2440.0 1820.0 1.39 0.8702 0.6197 1177986 ChemDiv3_005425 CCCC(=O)N1CCN(CC1)c2nc(Cc3ccccc3)c4COC(C)(C)Cc4c2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G14 compound treatment 560.0 -383.0 -0.14 1160.0 537.0 0.41 0.1954 0.4505 3118530 ChemDiv3_005426 COc1ccc(cc1)c2c/c(=N/c3ccc(O)cc3)/c4cc(C)ccc4o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G15 compound treatment 880.0 -62.5 -0.02 1480.0 857.0 0.66 0.4494 0.6829 3025734 ChemDiv3_005427 COc1cc(C)nc(SCC(=O)N)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G16 compound treatment 1040.0 97.5 0.03 440.0 -183.0 -0.14 -0.075 -0.5178 3118531 ChemDiv3_005428 COc1ccc(CCN(C)C(=O)C2CCCN(Cc3ccc(OC)c(OC)c3)C2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G17 compound treatment 800.0 -143.0 -0.05 1320.0 697.0 0.53 0.3425 0.6374 3118532 ChemDiv3_005429 Cc1ccc2n(CC(O)CN3C(=O)CNC3=O)c4C(=O)CCCc4c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G18 compound treatment 360.0 -583.0 -0.21 400.0 -223.0 -0.17 -0.2673 -0.9957 1912397 ChemDiv3_005430 CCOC(=O)/C=C(\C)/Sc1cc(=O)oc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G19 compound treatment 480.0 -463.0 -0.16 1160.0 537.0 0.41 0.1754 0.3954 3025735 ChemDiv3_005431 CC(NC(=O)Nc1ccccn1)N2C(=O)C3C4CC(C=C4)C3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G20 compound treatment 320.0 -623.0 -0.22 640.0 16.8 0.01 -0.147 -0.6647 3118533 ChemDiv3_005432 O=C(CCN1C(=O)c2ccccc2S1(=O)=O)Nc3nc(cs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G21 compound treatment 320.0 -623.0 -0.22 1320.0 697.0 0.53 0.2221 0.3838 3025736 ChemDiv3_005433 Clc1ccc(OCC(=O)NCCC2(CC3CC4CC(C3)C2)C4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G22 compound treatment 760.0 -183.0 -0.06 520.0 -103.0 -0.08 -0.1018 -0.995 3118534 ChemDiv3_005434 CCOc1ccc(/N=c\2/ccc3ccccc3n2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G23 mock treatment 2240.0 1300.0 0.46 400.0 -223.0 -0.17 0.2043 0.4159 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 G24 mock treatment 1000.0 57.5 0.02 1720.0 1100.0 0.84 0.6098 0.724 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H01 compound treatment 4600.0 3660.0 1.3 1680.0 1060.0 0.81 1.4911 0.9744 3118535 ChemDiv3_005435 O=C(NCCN1C(=O)C2C3CC(C=C3)C2C1=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H02 compound treatment 6320.0 5380.0 1.91 1000.0 377.0 0.29 1.5534 0.8051 3025737 ChemDiv3_005436 Clc1ccc(cc1)C2C3=C(CCCC3=O)Nc4ccc5ccccc5c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H03 compound treatment 800.0 -143.0 -0.05 2000.0 1380.0 1.06 0.7116 0.6725 1915152 ChemDiv3_005437 ON(C(=O)Nc1ccccc1)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H04 compound treatment 600.0 -343.0 -0.12 760.0 137.0 0.11 -0.0117 -0.0726 1394020 ChemDiv3_005438 CCOC(=O)c1c(C)nsc1Nc2cc(C)ccc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H05 compound treatment 800.0 -143.0 -0.05 400.0 -223.0 -0.17 -0.1569 -0.8783 1417285 ChemDiv3_005439 Cc1ccc2n(CCN(Cc3ccccc3)Cc4ccccc4)c5C(=O)CCCc5c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H06 compound treatment 680.0 -263.0 -0.09 560.0 -63.2 -0.05 -0.1002 -0.9539 3118536 ChemDiv3_005440 Clc1ccc(cc1)c2csc(NC(=O)C3c4ccccc4Oc5ccccc35)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H07 compound treatment 440.0 -503.0 -0.18 440.0 -183.0 -0.14 -0.2255 -0.9931 3025738 ChemDiv3_005441 CN(C(=O)c1ccccc1)c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H08 compound treatment 560.0 -383.0 -0.14 2880.0 2260.0 1.73 1.1292 0.6497 1234713 ChemDiv3_005442 Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3ccncc3)cc2)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H09 compound treatment 1000.0 57.5 0.02 5840.0 5220.0 4.01 2.8464 0.7107 3025739 ChemDiv3_005443 Clc1ccccc1OCC(=O)N2CCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H10 compound treatment 1040.0 97.5 0.03 720.0 96.8 0.07 0.077 0.9395 1454824 ChemDiv3_005444 Cc1ccc2nc3CCC(Cc3c(C(=O)O)c2c1)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H11 compound treatment 2480.0 1540.0 0.55 920.0 297.0 0.23 0.5468 0.925 3025740 ChemDiv3_005445 COc1ccccc1/C=C/C2N3C(=O)CCSC3=NC(=C2C(=O)OCC(C)C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H12 compound treatment 1040.0 97.5 0.03 440.0 -183.0 -0.14 -0.075 -0.5178 3118537 ChemDiv3_005446 Fc1cccc(c1)C2=N/C(=C\C=C\c3ccccc3)/C(=O)N2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H13 compound treatment 960.0 17.5 0.01 560.0 -63.2 -0.05 -0.0299 -0.6117 1015846 ChemDiv3_005447 O=S(=O)(N1CCCN(CC1)S(=O)(=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H14 compound treatment 440.0 -503.0 -0.18 480.0 -143.0 -0.11 -0.2038 -0.973 1377150 ChemDiv3_005448 O=C(Nc1ccccc1)c2cc3ccccc3c(=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H15 compound treatment 600.0 -343.0 -0.12 440.0 -183.0 -0.14 -0.1854 -0.9973 3118538 ChemDiv3_005449 Cc1ccc(cc1)c2nn(CCC(=O)Nc3cccc(c3)C(F)(F)F)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H16 compound treatment 2000.0 1060.0 0.38 3880.0 3260.0 2.5 2.0332 0.8042 1382411 ChemDiv3_005450 OC(=O)CCC(=O)N1CCN(CC1)C(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H17 compound treatment 640.0 -303.0 -0.11 480.0 -143.0 -0.11 -0.1536 -0.9999 3118539 ChemDiv3_005451 CCCNC(=O)Cn1c(=O)n(C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H18 compound treatment 520.0 -423.0 -0.15 560.0 -63.2 -0.05 -0.1403 -0.8906 1714411 ChemDiv3_005452 COc1ccc(CCNC(=O)c2cc3ccccc3c(=O)o2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H19 compound treatment 480.0 -463.0 -0.16 600.0 -23.2 -0.02 -0.1286 -0.7794 3118540 ChemDiv3_005453 CN(C)/C(=N\S(=O)(=O)c1ccc(F)cc1)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H20 compound treatment 1960.0 1020.0 0.36 2320.0 1700.0 1.3 1.1763 0.8702 1880109 ChemDiv3_005454 CC1CN(C(C)CN1C(=O)C2CCCCC2)C(=O)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H21 compound treatment 680.0 -263.0 -0.09 480.0 -143.0 -0.11 -0.1436 -0.9966 3025782 ChemDiv3_005455 COc1ccc(CCNC(=O)CC(c2ccccc2)c3cccc(C)c3O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H22 compound treatment 520.0 -423.0 -0.15 480.0 -143.0 -0.11 -0.1837 -0.9884 3025741 ChemDiv3_005456 FC(F)(F)C(=O)N1C(C2=C(CC(CC2=O)c3ccco3)Nc4ccccc14)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H23 mock treatment 6680.0 5740.0 2.04 560.0 -63.2 -0.05 1.4049 0.69 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 H24 mock treatment 1320.0 378.0 0.13 880.0 257.0 0.2 0.2341 0.9823 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I01 compound treatment 1360.0 418.0 0.15 560.0 -63.2 -0.05 0.0704 0.4517 3118541 ChemDiv3_005457 Cc1ccc(CNc2ccc(N3CCOCC3)c(Cl)c2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I02 compound treatment 400.0 -543.0 -0.19 2160.0 1540.0 1.18 0.6982 0.584 3118542 ChemDiv3_005458 COCCn1c(n[nH]c1=S)c2ccc(cc2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I03 compound treatment 600.0 -343.0 -0.12 480.0 -143.0 -0.11 -0.1637 -0.9988 1863874 ChemDiv3_005459 Cn1nnc(NCc2cc(Br)ccc2OCc3ccccc3F)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I04 compound treatment 480.0 -463.0 -0.16 280.0 -343.0 -0.26 -0.3023 -0.974 1566392 ChemDiv3_005460 CCOC(=O)c1ccc(Nc2cc(C)nc(C)c2C(=O)OCC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I05 compound treatment 320.0 -623.0 -0.22 3400.0 2780.0 2.13 1.3512 0.6305 1351464 ChemDiv3_005461 Cc1cccn2cc(nc12)c3cccc(NS(=O)(=O)c4ccc(Cl)cc4)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I06 compound treatment 280.0 -663.0 -0.24 560.0 -63.2 -0.05 -0.2005 -0.8355 3118543 ChemDiv3_005462 CCOc1ccc(Br)cc1C2C(=C(N)Oc3cc(ccc23)N(C)C)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I07 compound treatment 440.0 -503.0 -0.18 320.0 -303.0 -0.23 -0.2907 -0.9913 1132528 ChemDiv3_005463 OC(=O)c1ccccc1NC(=O)c2ccc(CN3CCOCC3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I08 compound treatment 440.0 -503.0 -0.18 280.0 -343.0 -0.26 -0.3124 -0.9819 3025742 ChemDiv3_005464 CC(=O)N1N=C(CC1c2cccs2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I09 compound treatment 240.0 -703.0 -0.25 440.0 -183.0 -0.14 -0.2757 -0.9634 3118544 ChemDiv3_005465 C(Cn1c2ccccc2c3nc4ccccc4nc13)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I10 compound treatment 360.0 -583.0 -0.21 440.0 -183.0 -0.14 -0.2456 -0.9824 3025743 ChemDiv3_005466 CN1C(c2ccccc2)n3c(nc4ccccc34)-c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I11 compound treatment 360.0 -583.0 -0.21 320.0 -303.0 -0.23 -0.3107 -0.9982 1431675 ChemDiv3_005467 Clc1ccccc1C2N(Cc3ccccc3)CCN2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I12 compound treatment 280.0 -663.0 -0.24 200.0 -423.0 -0.32 -0.3959 -0.9874 3118545 ChemDiv3_005468 Brc1c(cnn(c2ccccc2)c1=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I13 compound treatment 1200.0 258.0 0.09 560.0 -63.2 -0.05 0.0303 0.2926 3025783 ChemDiv3_005469 CCc1nc(Cl)c(C#N)c2CCCCc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I14 compound treatment 360.0 -583.0 -0.21 320.0 -303.0 -0.23 -0.3107 -0.9982 1304796 ChemDiv3_005470 Cc1ccc(SC2=C(N3CCOCC3)C(=O)N(C2=O)c4cc(C)cc(C)c4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I15 compound treatment 480.0 -463.0 -0.16 440.0 -183.0 -0.14 -0.2155 -0.9971 3118546 ChemDiv3_005471 COc1ccc(/C=C(/NC(=O)c2ccco2)\C(=O)N3CCCC3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I16 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 3025784 ChemDiv3_005472 Fc1ccccc1CN2CCCC(C2)C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I17 compound treatment 240.0 -703.0 -0.25 280.0 -343.0 -0.26 -0.3625 -0.9996 3118547 ChemDiv3_005473 COc1ccc(cc1)C2NN=C3C2CCc4c3[nH]c5ccc(C)cc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I18 compound treatment 280.0 -663.0 -0.24 240.0 -383.0 -0.29 -0.3742 -0.9938 1436055 ChemDiv3_005474 Oc1c(Sc2ccccc2)c(=O)oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I19 compound treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 1124479 ChemDiv3_005475 Cc1ccc(cc1)S(=O)(=O)N2CC3CCC2C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I20 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3118548 ChemDiv3_005476 COc1ccc(CN(C(=O)CCN2C(=O)c3ccccc3S2(=O)=O)c4ccccc4O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I21 compound treatment 280.0 -663.0 -0.24 1160.0 537.0 0.41 0.1252 0.2639 3025785 ChemDiv3_005477 CC(C)c1ccc(C)cc1OCC(=O)NCCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I22 compound treatment 320.0 -623.0 -0.22 600.0 -23.2 -0.02 -0.1688 -0.7617 3118549 ChemDiv3_005478 Cn1/c(=N/c2ccccc2C(=O)O)/ccc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I23 mock treatment 360.0 -583.0 -0.21 240.0 -383.0 -0.29 -0.3542 -0.9851 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 I24 mock treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J01 compound treatment 280.0 -663.0 -0.24 320.0 -303.0 -0.23 -0.3308 -1.0 3118550 ChemDiv3_005479 O=C(NCCN1C(=O)C2C3CC(C=C3)C2C1=O)Nc4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J02 compound treatment 280.0 -663.0 -0.24 240.0 -383.0 -0.29 -0.3742 -0.9938 1252670 ChemDiv3_005480 CCOc1ccc(NC(=O)NS(=O)(=O)c2ccc(C)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J03 compound treatment 320.0 -623.0 -0.22 680.0 56.8 0.04 -0.1253 -0.5568 1661781 ChemDiv3_005481 CCc1ccc(cc1)C(=O)c2cncc(Br)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J04 compound treatment 360.0 -583.0 -0.21 280.0 -343.0 -0.26 -0.3324 -0.9928 1297371 ChemDiv3_005482 OC(=O)c1sc2ccccc2c1Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J05 compound treatment 280.0 -663.0 -0.24 400.0 -223.0 -0.17 -0.2874 -0.988 817062 ChemDiv3_005483 OC(=O)Cc1ccc(O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J06 compound treatment 280.0 -663.0 -0.24 360.0 -263.0 -0.2 -0.3091 -0.9972 3118675 ChemDiv3_005484 OC(=O)C1C(C2OC1C=C2)C(=O)Nc3nc(cs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J07 compound treatment 360.0 -583.0 -0.21 600.0 -23.2 -0.02 -0.1587 -0.7653 1661374 ChemDiv3_005485 CN(C)C1(CCCCC1)c2nnnn2CCOC(=O)Nc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J08 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 1119745 ChemDiv3_005486 CCOC(=O)c1c(NC(=O)c2ccn(CC)n2)sc3CCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J09 compound treatment 280.0 -663.0 -0.24 1320.0 697.0 0.53 0.2121 0.363 3025786 ChemDiv3_005487 Clc1ccc(/C=C/C(=O)NCCCn2ccnc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J10 compound treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 3118676 ChemDiv3_005488 CCOc1ccc(cc1)n2c(S)nnc2c3nn(C)cc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J11 compound treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 3118677 ChemDiv3_005489 CN(C)c1ccc(cc1)C2Nc3sc4CCCCc4c3C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J12 compound treatment 280.0 -663.0 -0.24 600.0 -23.2 -0.02 -0.1788 -0.7586 1628099 ChemDiv3_005490 O=C(Nc1ccc2OCOc2c1)c3ccncc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J13 compound treatment 240.0 -703.0 -0.25 400.0 -223.0 -0.17 -0.2974 -0.9833 3118678 ChemDiv3_005491 CCOC(=O)C1=C(C)N(C)C2(C)CC1c3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J14 compound treatment 200.0 -743.0 -0.26 200.0 -423.0 -0.32 -0.416 -0.9946 1258498 ChemDiv3_005492 CN(C)c1ccc(NC(=O)c2ccoc2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J15 compound treatment 360.0 -583.0 -0.21 760.0 137.0 0.11 -0.0719 -0.3101 3118679 ChemDiv3_005493 COC(=O)CCn1nc(c2ccc(C)cc2)c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J16 compound treatment 320.0 -623.0 -0.22 240.0 -383.0 -0.29 -0.3642 -0.99 1151532 ChemDiv3_005494 COc1ccc(CC(=O)N2CCc3ccccc3C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J17 compound treatment 360.0 -583.0 -0.21 520.0 -103.0 -0.08 -0.2022 -0.9134 3118680 ChemDiv3_005495 OC(=O)c1ccc(cc1)S(=O)(=O)N(CC2CCCO2)Cc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J18 compound treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 1879815 ChemDiv3_005496 CCOc1ccccc1C(=O)N2CC(C)N(CC2C)C(=O)c3ccccc3OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J19 compound treatment 320.0 -623.0 -0.22 480.0 -143.0 -0.11 -0.2339 -0.9482 3025787 ChemDiv3_005497 Cc1ccccc1S(=O)(=O)/N=C(\N)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J20 compound treatment 400.0 -543.0 -0.19 360.0 -263.0 -0.2 -0.279 -0.9997 3118681 ChemDiv3_005498 OC(=O)C1CC=CCC1C(=O)N2CCN(C/C=C/c3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J21 compound treatment 320.0 -623.0 -0.22 440.0 -183.0 -0.14 -0.2556 -0.9763 3025788 ChemDiv3_005499 COc1ccc(CCNC(=O)CC(c2ccccc2)c3cc(Br)ccc3O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J22 compound treatment 200.0 -743.0 -0.26 280.0 -343.0 -0.26 -0.3726 -1.0 1480862 ChemDiv3_005500 O=C(CCc1ccccc1)N2CCCN(CC2)C(=O)CCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J23 mock treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 J24 mock treatment 4080.0 3140.0 1.11 240.0 -383.0 -0.29 0.579 0.5029 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K01 compound treatment 1360.0 418.0 0.15 880.0 257.0 0.2 0.2441 0.9901 1863608 ChemDiv3_005501 C(Nn1cnnc1)c2cccc(OCc3ccccc3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K02 compound treatment 640.0 -303.0 -0.11 680.0 56.8 0.04 -0.0451 -0.389 3118682 ChemDiv3_005502 CC(C)Cn1c(n[nH]c1=S)c2ccncc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K03 compound treatment 480.0 -463.0 -0.16 360.0 -263.0 -0.2 -0.2589 -0.9947 3118683 ChemDiv3_005503 COc1cccc(CC2CC(=O)N(C2=O)c3ccc4c(C)cc(=O)oc4c3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K04 compound treatment 1480.0 538.0 0.19 360.0 -263.0 -0.2 -0.0081 -0.029 1788155 ChemDiv3_005504 O=C(OCc1ccccc1)N2CN(Cc3ccccc3)Cc4c2oc5ccccc5c4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K05 compound treatment 1040.0 97.5 0.03 400.0 -223.0 -0.17 -0.0967 -0.5532 1500365 ChemDiv3_005505 Cc1ccccc1C(=O)Nc2cccc(c2)c3cn4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K06 compound treatment 480.0 -463.0 -0.16 880.0 257.0 0.2 0.0234 0.0911 3025789 ChemDiv3_005506 CCc1ccc(cc1)C2C(=C(N)Oc3cc4OCOc4cc23)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K07 compound treatment 680.0 -263.0 -0.09 400.0 -223.0 -0.17 -0.187 -0.9589 1203882 ChemDiv3_005507 O=C(N1CCCCCC1)c2ccc(CN3CCc4ccccc4C3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K08 compound treatment 320.0 -623.0 -0.22 640.0 16.8 0.01 -0.147 -0.6647 3118684 ChemDiv3_005508 CC(=O)N1N=C(CC1c2cc3cc4OCOc4cc3nc2Cl)c5ccc(C)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K09 compound treatment 600.0 -343.0 -0.12 480.0 -143.0 -0.11 -0.1637 -0.9988 3025791 ChemDiv3_005509 CC(Cc1ccccc1)NC(=O)CC(c2ccccc2)c3cc(Br)ccc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K10 compound treatment 520.0 -423.0 -0.15 320.0 -303.0 -0.23 -0.2706 -0.9773 1541015 ChemDiv3_005510 N1C(c2ccncc2)n3c(nc4ccccc34)-c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K11 compound treatment 5040.0 4100.0 1.45 440.0 -183.0 -0.14 0.9284 0.6357 3118685 ChemDiv3_005511 Cc1ccc(cc1)N(CC(=O)NC(c2ccccc2)c3ccccc3)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K12 compound treatment 680.0 -263.0 -0.09 520.0 -103.0 -0.08 -0.1219 -0.9968 3118686 ChemDiv3_005512 CCC(C)OC(=O)COc1ccc2c(=O)c(c3ccc(OC)c(OC)c3)c(oc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K13 compound treatment 680.0 -263.0 -0.09 520.0 -103.0 -0.08 -0.1219 -0.9968 1344366 ChemDiv3_005513 CCc1nc(N2CCCCC2)c(C#N)c3CCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K14 compound treatment 560.0 -383.0 -0.14 360.0 -263.0 -0.2 -0.2388 -0.9812 1538233 ChemDiv3_005514 CCc1ccccc1OCC(=O)Nc2ccc(cc2)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K15 compound treatment 440.0 -503.0 -0.18 440.0 -183.0 -0.14 -0.2255 -0.9931 3118687 ChemDiv3_005515 CCc1ccc(cc1)C2=CC(=O)C=CC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K16 compound treatment 560.0 -383.0 -0.14 1720.0 1100.0 0.84 0.4994 0.5856 3118688 ChemDiv3_005516 O=C(C1CCCN(Cc2ccco2)C1)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K17 compound treatment 6400.0 5460.0 1.94 1600.0 977.0 0.75 1.8992 0.9148 3025829 ChemDiv3_005517 Cc1ccc2[nH]c3C4=NNC(C4CCc3c2c1)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K18 compound treatment 440.0 -503.0 -0.18 840.0 217.0 0.17 -0.0084 -0.0343 3118689 ChemDiv3_005518 COC(=O)C1=C(N)OC2=C(C1c3ccc(OCc4ccccc4F)cc3)C(=O)CCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K19 compound treatment 600.0 -343.0 -0.12 960.0 337.0 0.26 0.0969 0.3392 3025830 ChemDiv3_005519 Cc1ccc(cc1)S(=O)(=O)N2CC3CC2C=C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K20 compound treatment 840.0 -103.0 -0.04 2320.0 1700.0 1.3 0.8954 0.6871 3118690 ChemDiv3_005520 CC(C)CNC(=O)CCN1C(=O)c2ccccc2S1(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K21 compound treatment 800.0 -143.0 -0.05 840.0 217.0 0.17 0.0819 0.4711 1184424 ChemDiv3_005521 O=C(NCCC1(CC2CC3CC(C2)C1)C3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K22 compound treatment 720.0 -223.0 -0.08 760.0 137.0 0.11 0.0184 0.1403 3025831 ChemDiv3_005522 Cn1/c(=N\c2ccc(cc2)N3CCOCC3)/ccc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K23 mock treatment 1120.0 178.0 0.06 320.0 -303.0 -0.23 -0.1201 -0.4979 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 K24 mock treatment 1080.0 138.0 0.05 840.0 217.0 0.17 0.1522 0.8774 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L01 compound treatment 280.0 -663.0 -0.24 6280.0 5660.0 4.34 2.9046 0.6679 3118691 ChemDiv3_005523 O=C(Nc1nncs1)Nc2ccc(cc2)N3C(=O)C4C5CC(C=C5)C4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L02 compound treatment 8600.0 7660.0 2.72 440.0 -183.0 -0.14 1.8214 0.6696 3025832 ChemDiv3_005524 COC(=O)C1CCN(CC1)C(=O)Cc2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L03 compound treatment 600.0 -343.0 -0.12 840.0 217.0 0.17 0.0318 0.1542 3118692 ChemDiv3_005525 CC1ON(C(=O)NC1=O)c2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L04 compound treatment 440.0 -503.0 -0.18 520.0 -103.0 -0.08 -0.1821 -0.9334 3025833 ChemDiv3_005526 CCc1cccc(NC(=O)C2c3ccccc3Oc4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L05 compound treatment 440.0 -503.0 -0.18 2360.0 1740.0 1.33 0.8168 0.6072 3118693 ChemDiv3_005527 CC(C)COc1ccc2c(c1)c3CCCc4[n+](C)ccn2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L06 compound treatment 520.0 -423.0 -0.15 1160.0 537.0 0.41 0.1854 0.4228 3118694 ChemDiv3_005528 CCN(CC)c1ccc(NC(=O)C2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L07 compound treatment 560.0 -383.0 -0.14 1000.0 377.0 0.29 0.1086 0.3399 1478251 ChemDiv3_005529 CN(C)c1ccc(cc1)C(N2CCOCC2)c3nnnn3CCOC(=O)Nc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L08 compound treatment 240.0 -703.0 -0.25 680.0 56.8 0.04 -0.1454 -0.5747 1142691 ChemDiv3_005530 CCOC(=O)c1cc(NC(=O)C2C(C3OC2C=C3)C(=O)O)cc(c1)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L09 compound treatment 7120.0 6180.0 2.19 400.0 -223.0 -0.17 1.4284 0.6498 3118834 ChemDiv3_005531 CC(C)(C)c1ccc(/C=C/C(=O)NCCCn2ccnc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L10 compound treatment 440.0 -503.0 -0.18 680.0 56.8 0.04 -0.0952 -0.5189 3025834 ChemDiv3_005532 CCn1c(S)nnc1c2cc(C)n(C)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L11 compound treatment 560.0 -383.0 -0.14 560.0 -63.2 -0.05 -0.1303 -0.904 3025835 ChemDiv3_005533 CC1(C)Cc2c(CO1)sc3nc(CCCc4ccccc4)n(N)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L12 compound treatment 320.0 -623.0 -0.22 560.0 -63.2 -0.05 -0.1905 -0.8424 3118835 ChemDiv3_005534 Cc1ccsc1C2C(=C(N)Oc3[nH]c(nc23)c4ccccc4)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L13 compound treatment 880.0 -62.5 -0.02 400.0 -223.0 -0.17 -0.1369 -0.792 3118836 ChemDiv3_005535 COc1ccc(NC(=O)N2CCN(C/C=C/c3ccccc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L14 compound treatment 360.0 -583.0 -0.21 360.0 -263.0 -0.2 -0.289 -0.9999 1459940 ChemDiv3_005536 O=C(NCC1CCCO1)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L15 compound treatment 840.0 -103.0 -0.04 280.0 -343.0 -0.26 -0.212 -0.7971 3118837 ChemDiv3_005537 Cc1ccc(cc1)c2nn(CCC(=O)N3CCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L16 compound treatment 400.0 -543.0 -0.19 440.0 -183.0 -0.14 -0.2355 -0.9881 1569367 ChemDiv3_005538 OC(=O)C1CCCCC1C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L17 compound treatment 560.0 -383.0 -0.14 1200.0 577.0 0.44 0.2172 0.4689 3025836 ChemDiv3_005539 Fc1ccccc1c2nc(no2)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L18 compound treatment 280.0 -663.0 -0.24 400.0 -223.0 -0.17 -0.2874 -0.988 1310245 ChemDiv3_005540 OC(=O)C1C(C2CC1C=C2)C(=O)NCc3ccncc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L19 compound treatment 320.0 -623.0 -0.22 520.0 -103.0 -0.08 -0.2122 -0.9044 3118838 ChemDiv3_005541 CC(C)(C)N/C(=N\S(=O)(=O)c1ccc(Br)cc1)/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L20 compound treatment 440.0 -503.0 -0.18 520.0 -103.0 -0.08 -0.1821 -0.9334 1202411 ChemDiv3_005542 COC(=O)CN(C(=O)c1cc2ccccc2oc1=O)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L21 compound treatment 760.0 -183.0 -0.06 4920.0 4300.0 3.3 2.2868 0.6931 3025837 ChemDiv3_005543 COc1ccc(cc1OC)C2(CCCC2)C(=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L22 compound treatment 240.0 -703.0 -0.25 1000.0 377.0 0.29 0.0283 0.0742 3118839 ChemDiv3_005544 OC(=O)C1C(C2CCC1O2)C(=O)N3CCN(C/C=C/c4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L23 mock treatment 680.0 -263.0 -0.09 400.0 -223.0 -0.17 -0.187 -0.9589 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 L24 mock treatment 1880.0 938.0 0.33 600.0 -23.2 -0.02 0.2226 0.6682 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M01 compound treatment 400.0 -543.0 -0.19 2360.0 1740.0 1.33 0.8067 0.5988 1863694 ChemDiv3_005545 CCCCC(=O)Nc1ccc(NCc2ccc(C)s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M02 compound treatment 320.0 -623.0 -0.22 520.0 -103.0 -0.08 -0.2122 -0.9044 1844088 ChemDiv3_005546 COc1ccccc1n2c(n[nH]c2=S)c3ccncc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M03 compound treatment 360.0 -583.0 -0.21 320.0 -303.0 -0.23 -0.3107 -0.9982 3118840 ChemDiv3_005547 CCOC(=O)C(C)N1C(=O)S/C(=C/c2ccc(o2)c3ccccc3C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M04 compound treatment 1160.0 218.0 0.08 360.0 -263.0 -0.2 -0.0883 -0.4084 3025838 ChemDiv3_005548 CCOC(=O)Nc1oc2ccccc2c(=O)c1CN3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M05 compound treatment 1200.0 258.0 0.09 520.0 -103.0 -0.08 0.0086 0.0707 3118841 ChemDiv3_005549 CN(C)c1oc(nc1S(=O)(=O)c2ccc(C)cc2)c3ccccc3Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M06 compound treatment 440.0 -503.0 -0.18 560.0 -63.2 -0.05 -0.1604 -0.868 3118842 ChemDiv3_005550 CCN(CC)C(=O)c1ccc2NC(C3C4CCC(C4)C3c2c1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M07 compound treatment 3720.0 2780.0 0.99 5040.0 4420.0 3.39 3.0944 0.8763 3025839 ChemDiv3_005551 CC1=Nc2ccccc2N=C(O)C1Sc3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M08 compound treatment 2880.0 1940.0 0.69 2280.0 1660.0 1.27 1.3854 0.9583 1645771 ChemDiv3_005552 Cc1ccc2nc(cc(c3ccccc3)c2c1)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M09 compound treatment 440.0 -503.0 -0.18 640.0 16.8 0.01 -0.1169 -0.6543 3118843 ChemDiv3_005553 CCCN(CCC)C(=O)CC(c1ccccc1)c2cc(Br)ccc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M10 compound treatment 440.0 -503.0 -0.18 320.0 -303.0 -0.23 -0.2907 -0.9913 1210079 ChemDiv3_005554 N1C(c2ccco2)n3c(nc4ccccc34)-c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M11 compound treatment 400.0 -543.0 -0.19 680.0 56.8 0.04 -0.1053 -0.5334 3118844 ChemDiv3_005555 COc1ccc(C)cc1Cn2c(nc3ccccc23)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M12 compound treatment 320.0 -623.0 -0.22 360.0 -263.0 -0.2 -0.299 -0.999 3118845 ChemDiv3_005556 CCC(C)OC(=O)COc1ccc2c(=O)c(Oc3cc(C)ccc3C)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M13 compound treatment 320.0 -623.0 -0.22 560.0 -63.2 -0.05 -0.1905 -0.8424 1459137 ChemDiv3_005557 CCc1nc(NCCN2CCOCC2)c(C#N)c3CCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M14 compound treatment 440.0 -503.0 -0.18 400.0 -223.0 -0.17 -0.2472 -0.9998 3118846 ChemDiv3_005558 CCN(CC)C(=O)CSc1nc(O)c2c(C)cc(C)nc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M15 compound treatment 10960.0 10000.0 3.55 760.0 137.0 0.11 2.5871 0.7277 3025063 ChemDiv3_005559 CCc1ccc(cc1)c2cc(O)cc3sc(=O)oc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M16 compound treatment 1600.0 658.0 0.23 480.0 -143.0 -0.11 0.0872 0.3381 3118847 ChemDiv3_005560 O=C(C1CCCN(CC2CC3CC2C=C3)C1)N4CCC(Cc5ccccc5)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M17 compound treatment 600.0 -343.0 -0.12 400.0 -223.0 -0.17 -0.2071 -0.9858 3025066 ChemDiv3_005561 Cc1ccc2n(CCC(=O)O)c3C(=O)CCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M18 compound treatment 480.0 -463.0 -0.16 520.0 -103.0 -0.08 -0.1721 -0.9443 3025068 ChemDiv3_005562 Clc1ccc(CSc2ncccn2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M19 compound treatment 640.0 -303.0 -0.11 5440.0 4820.0 3.7 2.5389 0.6863 1194966 ChemDiv3_005563 O=C(NCc1ccccc1)N2CC3CC2C=C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M20 compound treatment 360.0 -583.0 -0.21 400.0 -223.0 -0.17 -0.2673 -0.9957 3118848 ChemDiv3_005564 COc1ccccc1C2=NC(CN2c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M21 compound treatment 360.0 -583.0 -0.21 600.0 -23.2 -0.02 -0.1587 -0.7653 1272874 ChemDiv3_005565 O=C(CCC1CCCCC1)NCCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M22 compound treatment 520.0 -423.0 -0.15 1320.0 697.0 0.53 0.2723 0.4901 3118849 ChemDiv3_005566 OC(=O)CC[n+]1ccc(cc1)c2cc[n+](CCC(=O)O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M23 mock treatment 480.0 -463.0 -0.16 640.0 16.8 0.01 -0.1069 -0.6496 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 M24 mock treatment 920.0 -22.5 -0.01 280.0 -343.0 -0.26 -0.192 -0.7282 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N01 compound treatment 480.0 -463.0 -0.16 400.0 -223.0 -0.17 -0.2372 -0.9998 3025074 ChemDiv3_005567 COC(=O)NCN1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N02 compound treatment 480.0 -463.0 -0.16 360.0 -263.0 -0.2 -0.2589 -0.9947 3118850 ChemDiv3_005568 CC1(C)CC(=O)c2sc(NS(=O)(=O)C)nc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N03 compound treatment 320.0 -623.0 -0.22 480.0 -143.0 -0.11 -0.2339 -0.9482 1577663 ChemDiv3_005569 Clc1ccc(cc1Cl)N2OCC(=O)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N04 compound treatment 280.0 -663.0 -0.24 400.0 -223.0 -0.17 -0.2874 -0.988 3118851 ChemDiv3_005570 Clc1ncccc1C(=O)N(Cc2ccccc2)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N05 compound treatment 240.0 -703.0 -0.25 360.0 -263.0 -0.2 -0.3191 -0.9946 3118852 ChemDiv3_005571 NNC(=O)c1ccc2[nH]c3/C(=N/N)/CCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N06 compound treatment 240.0 -703.0 -0.25 520.0 -103.0 -0.08 -0.2323 -0.8881 3025109 ChemDiv3_005572 Cc1cc(NC(=O)/C=C/c2ccc(F)cc2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N07 compound treatment 240.0 -703.0 -0.25 720.0 96.8 0.07 -0.1237 -0.4756 1467529 ChemDiv3_005573 Cc1ccc(NC2(CCCCC2)c3nnnn3CCOC(=O)Nc4ccc(Cl)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N08 compound treatment 960.0 17.5 0.01 720.0 96.8 0.07 0.0569 0.7635 3025111 ChemDiv3_005574 Cn1ccc(/C=C/2\CCC/C(=C/c3ccn(C)n3)/C2=O)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N09 compound treatment 280.0 -663.0 -0.24 440.0 -183.0 -0.14 -0.2656 -0.9699 1875080 ChemDiv3_005575 Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C5CCCCC5)c3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N10 compound treatment 240.0 -703.0 -0.25 560.0 -63.2 -0.05 -0.2105 -0.8293 1217360 ChemDiv3_005576 COc1ccc(cc1COc2ccccc2Cl)C(=O)NCc3cc4cc(Cl)ccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N11 compound treatment 760.0 -183.0 -0.06 840.0 217.0 0.17 0.0719 0.4026 3118853 ChemDiv3_005577 O=S(=O)(N1CCCCCC1)c2ccc3oc4ccc(cc4c3c2)S(=O)(=O)N5CCCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N12 compound treatment 760.0 -183.0 -0.06 640.0 16.8 0.01 -0.0367 -0.5556 1327882 ChemDiv3_005578 Cc1nc(C(C(C#N)C#N)c2ccccc2F)c(O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N13 compound treatment 440.0 -503.0 -0.18 320.0 -303.0 -0.23 -0.2907 -0.9913 3118854 ChemDiv3_005579 CCCC(=O)N1CCC(=N1)c2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N14 compound treatment 640.0 -303.0 -0.11 1000.0 377.0 0.29 0.1287 0.417 1390843 ChemDiv3_005580 CC(C)CN(CC(C)C)C(=O)C1c2ccccc2Oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N15 compound treatment 400.0 -543.0 -0.19 520.0 -103.0 -0.08 -0.1921 -0.9231 3118980 ChemDiv3_005581 CNC(=O)COc1ccc(NC(=O)CCn2nc(c3ccc(Cl)cc3)c4ccccc4c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N16 compound treatment 440.0 -503.0 -0.18 480.0 -143.0 -0.11 -0.2038 -0.973 1879391 ChemDiv3_005582 Brc1cccc(c1)c2cc(C(=O)NCc3cccnc3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N17 compound treatment 800.0 -143.0 -0.05 4360.0 3740.0 2.87 1.9928 0.6945 3118981 ChemDiv3_005583 COc1ccc(CC(=O)Nc2ccc(O)c(c2)c3nc4ccccc4o3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N18 compound treatment 640.0 -303.0 -0.11 480.0 -143.0 -0.11 -0.1536 -0.9999 1132559 ChemDiv3_005584 CC(C)OC(=O)c1c(NC(=O)c2ccc(Cn3nc(C)c(Cl)c3C)o2)sc4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N19 compound treatment 320.0 -623.0 -0.22 3160.0 2540.0 1.95 1.221 0.6229 3118982 ChemDiv3_005585 Oc1ccccc1c2nnc(SCc3ccccc3)n2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N20 compound treatment 680.0 -263.0 -0.09 560.0 -63.2 -0.05 -0.1002 -0.9539 1923004 ChemDiv3_005586 CCOC(=O)c1ccc2n(Cc3ccccc3)c(C)c(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N21 compound treatment 680.0 -263.0 -0.09 320.0 -303.0 -0.23 -0.2305 -0.9192 3025118 ChemDiv3_005587 CCOc1ccc(NC(=O)C2(CCOCC2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N22 compound treatment 640.0 -303.0 -0.11 840.0 217.0 0.17 0.0418 0.2111 1121345 ChemDiv3_005588 O=C(N1CCN(CC1)c2ncccn2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N23 mock treatment 280.0 -663.0 -0.24 440.0 -183.0 -0.14 -0.2656 -0.9699 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 N24 mock treatment 720.0 -223.0 -0.08 640.0 16.8 0.01 -0.0467 -0.584 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O01 compound treatment 360.0 -583.0 -0.21 280.0 -343.0 -0.26 -0.3324 -0.9928 1863698 ChemDiv3_005589 CCOc1ccc(CNc2ccc(cc2)N3CCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O02 compound treatment 280.0 -663.0 -0.24 440.0 -183.0 -0.14 -0.2656 -0.9699 1314044 ChemDiv3_005590 CCOC(=O)c1c(C)n(c2ccc(C)cc2)c3ccc(OCC(O)CN4CCN(C)CC4)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O03 compound treatment 280.0 -663.0 -0.24 240.0 -383.0 -0.29 -0.3742 -0.9938 3118983 ChemDiv3_005591 Oc1ccc(cc1)n2cccc2C=C3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O04 compound treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 3025165 ChemDiv3_005592 Cn1c(nc2c(=O)oc3ccccc3c12)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O05 compound treatment 240.0 -703.0 -0.25 400.0 -223.0 -0.17 -0.2974 -0.9833 1629009 ChemDiv3_005593 CCOC(=O)c1ccc(NC(=O)C2C3CC(C)(Oc4ccccc34)N(C)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O06 compound treatment 200.0 -743.0 -0.26 360.0 -263.0 -0.2 -0.3291 -0.9914 3025167 ChemDiv3_005594 CNC(=O)CN1C(=O)c2ccccc2S1(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O07 compound treatment 280.0 -663.0 -0.24 640.0 16.8 0.01 -0.1571 -0.6674 3118984 ChemDiv3_005595 OCCN1CNC(=Nc2nc3ccccc3o2)NC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O08 compound treatment 280.0 -663.0 -0.24 200.0 -423.0 -0.32 -0.3959 -0.9874 3118985 ChemDiv3_005596 CCOC(=O)C1C(CC(=CC1=O)c2cccs2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O09 compound treatment 400.0 -543.0 -0.19 360.0 -263.0 -0.2 -0.279 -0.9997 3025170 ChemDiv3_005597 CCCN(CCC)C(=O)CC(c1ccccc1)c2cc(C)ccc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O10 compound treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 3118986 ChemDiv3_005598 C1CC2C(O1)c3ccc4ccccc4c3NC2c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O11 compound treatment 200.0 -743.0 -0.26 240.0 -383.0 -0.29 -0.3943 -0.9985 1497180 ChemDiv3_005599 CCCCc1nc2sc3c(NCc4ccccc4)ncnc3c2c5CC(C)(C)OCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O12 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 3025173 ChemDiv3_005600 CCC(C)OC(=O)COc1ccc2c(=O)c(Oc3ccccc3Cl)coc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O13 compound treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 1391398 ChemDiv3_005601 CCc1nc(NCC(C)C)c(C#N)c2CCCCc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O14 compound treatment 320.0 -623.0 -0.22 280.0 -343.0 -0.26 -0.3425 -0.9961 3025175 ChemDiv3_005602 Cc1cc(C)c2c(O)nc(SCC(=O)Nc3ccccc3)nc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O15 compound treatment 320.0 -623.0 -0.22 600.0 -23.2 -0.02 -0.1688 -0.7617 3118987 ChemDiv3_005603 Oc1cc(c2cc(ccc2Cl)C(F)(F)F)c3oc(=O)sc3c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O16 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 3118988 ChemDiv3_005604 COc1cc(CN2CCCC(C2)C(=O)N3CCCCCC3)ccc1OCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O17 compound treatment 720.0 -223.0 -0.08 200.0 -423.0 -0.32 -0.2856 -0.854 3118989 ChemDiv3_005605 Cc1ccc(cc1)c2noc(CNc3ccc(Oc4ccccc4)cc3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O18 compound treatment 320.0 -623.0 -0.22 320.0 -303.0 -0.23 -0.3208 -0.9997 3025225 ChemDiv3_005606 OC(=O)c1ccc(CSc2nc(cc(n2)C(F)(F)F)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O19 compound treatment 240.0 -703.0 -0.25 320.0 -303.0 -0.23 -0.3408 -0.9994 1658529 ChemDiv3_005607 OC(=O)C1(CCCCC1)NS(=O)(=O)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O20 compound treatment 280.0 -663.0 -0.24 240.0 -383.0 -0.29 -0.3742 -0.9938 3025227 ChemDiv3_005608 O=C/1N(C(=S)S\C1=C/2\Nc3ccccc3C2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O21 compound treatment 320.0 -623.0 -0.22 200.0 -423.0 -0.32 -0.3859 -0.9823 3118990 ChemDiv3_005609 COc1ccc(cc1)C(=O)Nc2ccc3C(=O)N(CCC(=O)O)C(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O22 compound treatment 480.0 -463.0 -0.16 440.0 -183.0 -0.14 -0.2155 -0.9971 3025229 ChemDiv3_005610 Cn1/c(=N\c2cccc(O)c2)/ccc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O23 mock treatment 200.0 -743.0 -0.26 240.0 -383.0 -0.29 -0.3943 -0.9985 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 O24 mock treatment 400.0 -543.0 -0.19 600.0 -23.2 -0.02 -0.1487 -0.7693 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P01 compound treatment 400.0 -543.0 -0.19 280.0 -343.0 -0.26 -0.3224 -0.9881 3118991 ChemDiv3_005611 COC(=O)NC(C)N1C(=O)C2C3CC(C=C3)C2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P02 compound treatment 440.0 -503.0 -0.18 560.0 -63.2 -0.05 -0.1604 -0.868 3025231 ChemDiv3_005612 CC(C)Cn1c2ccccc2c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P03 compound treatment 240.0 -703.0 -0.25 360.0 -263.0 -0.2 -0.3191 -0.9946 1152346 ChemDiv3_005613 CC(C)c1ccc2n3CCN(CC#N)C4CCCc(c43)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P04 compound treatment 240.0 -703.0 -0.25 200.0 -423.0 -0.32 -0.406 -0.9914 3118992 ChemDiv3_005614 O=C(Nc1ccc(Oc2ccccc2)cc1)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P05 compound treatment 2840.0 1900.0 0.67 360.0 -263.0 -0.2 0.3331 0.4739 3025234 ChemDiv3_005615 CC(C)OC(=O)N(C)c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P06 compound treatment 440.0 -503.0 -0.18 240.0 -383.0 -0.29 -0.3341 -0.9712 1670317 ChemDiv3_005616 COC(=O)c1c(NC(=O)C(C)Oc2ccccc2)sc3CCc4ccccc4-c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P07 compound treatment 2160.0 1220.0 0.43 400.0 -223.0 -0.17 0.1842 0.3965 3025236 ChemDiv3_005617 FC(F)(F)c1cccc(NC(=O)C(=C2CCCCCC2)C#N)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P08 compound treatment 360.0 -583.0 -0.21 280.0 -343.0 -0.26 -0.3324 -0.9928 3118993 ChemDiv3_005618 CCN1CCc2c(C1)sc3NC(NC(=O)c23)c4ccc(COc5cccc(c5)C(F)(F)F)o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P09 compound treatment 400.0 -543.0 -0.19 320.0 -303.0 -0.23 -0.3007 -0.9955 1875125 ChemDiv3_005619 CC1CCCCN1S(=O)(=O)c2ccc(NC(=O)c3oc4ccccc4c3C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P10 compound treatment 280.0 -663.0 -0.24 280.0 -343.0 -0.26 -0.3525 -0.9984 3118994 ChemDiv3_005620 Cn1c2ccccc2c3cc(ccc13)C4Nc5ccccc5C(=O)N4O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P11 compound treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 3118995 ChemDiv3_005621 O=S(=O)(NCC1CCCO1)c2ccc3oc4ccc(cc4c3c2)S(=O)(=O)NCC5CCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P12 compound treatment 280.0 -663.0 -0.24 320.0 -303.0 -0.23 -0.3308 -1.0 1257085 ChemDiv3_005622 Cc1cc(C)n(n1)C(=S)CSc2nc(cc(c3ccco3)c2C#N)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P13 compound treatment 480.0 -463.0 -0.16 160.0 -463.0 -0.36 -0.3675 -0.9383 3118996 ChemDiv3_005623 Cc1ccc(cc1CNC(=O)CSc2nc3ccccc3s2)c4nn(C)c(=O)c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P14 compound treatment 240.0 -703.0 -0.25 440.0 -183.0 -0.14 -0.2757 -0.9634 1731321 ChemDiv3_005624 O=C(C(Sc1ccccc1)c2ccccc2)n3cnc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P15 compound treatment 240.0 -703.0 -0.25 280.0 -343.0 -0.26 -0.3625 -0.9996 3118997 ChemDiv3_005625 Clc1ccc(cc1)c2nn(CCC(=O)NCC3CCCO3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P16 compound treatment 240.0 -703.0 -0.25 240.0 -383.0 -0.29 -0.3843 -0.9966 1308799 ChemDiv3_005626 CC1CCN(CC1)C(=O)C2c3ccccc3Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P17 compound treatment 200.0 -743.0 -0.26 320.0 -303.0 -0.23 -0.3509 -0.9981 1147363 ChemDiv3_005627 C1CCN(CC1)c2nc(N3CCCCC3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P18 compound treatment 320.0 -623.0 -0.22 240.0 -383.0 -0.29 -0.3642 -0.99 1443626 ChemDiv3_005628 CCOc1ccc(cc1)c2cc(C(=O)N3CCc4ccccc4C3)c5ccccc5n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P19 compound treatment 2080.0 1140.0 0.4 280.0 -343.0 -0.26 0.099 0.2054 1859661 ChemDiv3_005629 CC(=O)Nc1ccc(NC(=O)CCSc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P20 compound treatment 280.0 -663.0 -0.24 320.0 -303.0 -0.23 -0.3308 -1.0 1880335 ChemDiv3_005630 COc1ccc(cc1OC)C(=O)N2CC(C)N(CC2C)C(=O)c3ccc(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P21 compound treatment 2640.0 1700.0 0.6 200.0 -423.0 -0.32 0.1961 0.2865 3025305 ChemDiv3_005631 COc1ccc(cc1OC)C2(CCCC2)C(=O)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P22 compound treatment 400.0 -543.0 -0.19 240.0 -383.0 -0.29 -0.3441 -0.9788 3119130 ChemDiv3_005632 Cc1cc(nn1Cc2ccc(o2)C(=O)Nc3ncc(Br)s3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P23 mock treatment 280.0 -663.0 -0.24 200.0 -423.0 -0.32 -0.3959 -0.9874 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2016 P24 mock treatment 280.0 -663.0 -0.24 360.0 -263.0 -0.2 -0.3091 -0.9972 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A01 compound treatment 440.0 -919.0 -0.33 320.0 -376.0 -0.29 -0.4347 -0.9982 1345241 ChemDiv3_005633 COc1ccc(CNC(=O)C2C(C3CCC2O3)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A02 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 3025307 ChemDiv3_005634 OCCCN1CC2(CN(CCCO)CC(C1)(C2=O)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A03 compound treatment 320.0 -1040.0 -0.37 240.0 -456.0 -0.35 -0.5082 -0.9997 3119131 ChemDiv3_005635 Clc1ccc(Cl)c(OCc2ccc(o2)C(=O)N3CCSCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A04 compound treatment 800.0 -559.0 -0.2 320.0 -376.0 -0.29 -0.3444 -0.9831 3025310 ChemDiv3_005636 Oc1cc(=O)[nH]c2c1sc3nc4CCCCCc4c(c32)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A05 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 1445484 ChemDiv3_005637 Fc1ccc(cc1)N2CCN(CC2)C(=O)CSc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A06 compound treatment 600.0 -759.0 -0.27 1160.0 464.0 0.36 0.0614 0.1376 3025311 ChemDiv3_005638 C[N+]1(CCC(=O)NCc2ccccc2)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A07 compound treatment 360.0 -999.0 -0.35 320.0 -376.0 -0.29 -0.4548 -0.9949 1882257 ChemDiv3_005639 Cc1onc(c1C(=O)N(Cc2ccccc2)Cc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A08 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3025314 ChemDiv3_005640 Cc1ccc(NC(=O)CC(O)(C(F)(F)F)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A09 compound treatment 240.0 -1120.0 -0.4 280.0 -416.0 -0.32 -0.5066 -0.9942 3119132 ChemDiv3_005641 CCCc1nc2ccccc2c3nc(N)nn13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A10 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 1574613 ChemDiv3_005642 CC1CCc2cc(F)ccc2N1C(=O)NC(C)(C)c3cccc(c3)C(=C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A11 compound treatment 240.0 -1120.0 -0.4 240.0 -456.0 -0.35 -0.5283 -0.9981 3025379 ChemDiv3_005643 CCOC(=O)Cc1nc2ccccc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A12 compound treatment 360.0 -999.0 -0.35 240.0 -456.0 -0.35 -0.4982 -1.0 3119133 ChemDiv3_005644 Cc1[nH]c2ccccc2c1Cc3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A13 compound treatment 280.0 -1080.0 -0.38 840.0 144.0 0.11 -0.1926 -0.4835 3025381 ChemDiv3_005645 Nc1ccc(Cc2nc3cc4ccccc4cc3[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A14 compound treatment 440.0 -919.0 -0.33 320.0 -376.0 -0.29 -0.4347 -0.9982 3119134 ChemDiv3_005646 COC(=O)C1Cc2ccccc2CN1S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A15 compound treatment 280.0 -1080.0 -0.38 960.0 264.0 0.2 -0.1274 -0.2943 3025383 ChemDiv3_005647 OC(=O)/C=C/C(=O)N1CCC(=CC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A16 compound treatment 280.0 -1080.0 -0.38 640.0 -56.3 -0.04 -0.3011 -0.7819 1875879 ChemDiv3_005648 COC(=O)c1c2C(=O)c3ccccc3C(=O)c2n4cc5ccccc5cc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A17 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3119135 ChemDiv3_005649 CC12C3CC(C=C3)C2C(=O)N(CCC(=O)O)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A18 compound treatment 960.0 -399.0 -0.14 360.0 -336.0 -0.26 -0.2826 -0.9599 3025387 ChemDiv3_005650 Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)C3(CCOCC3)c4ccccc4)cc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A19 compound treatment 240.0 -1120.0 -0.4 240.0 -456.0 -0.35 -0.5283 -0.9981 3119136 ChemDiv3_005651 CCOC(=O)COc1ccc(=O)n(n1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A20 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 1271566 ChemDiv3_005652 Cc1cccc(c1)N(CC(=O)N)C2SC(=O)NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A21 compound treatment 440.0 -919.0 -0.33 1080.0 384.0 0.29 -0.0221 -0.0504 3025389 ChemDiv3_005653 COC(=O)N(c1ccc(OC)cc1)P2(=S)OCCC(C)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A22 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 1070090 ChemDiv3_005654 Cc1cn2C3CC(Oc2nc1=O)C(CO)O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A23 mock treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 A24 mock treatment 320.0 -1040.0 -0.37 240.0 -456.0 -0.35 -0.5082 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B01 compound treatment 880.0 -479.0 -0.17 400.0 -296.0 -0.23 -0.2809 -0.9897 3119137 ChemDiv3_005655 CC(=O)N1c2ccccc2C(=CC1(C)C)CSc3nnc(o3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B02 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3025391 ChemDiv3_005656 NC(=O)Cn1nnc2sc3CCCCc3c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B03 compound treatment 480.0 -879.0 -0.31 360.0 -336.0 -0.26 -0.403 -0.9956 3119138 ChemDiv3_005657 CN(C1CCCCC1)C(=S)SCc2nc(N)nc(Nc3cccc(Cl)c3C)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B04 compound treatment 400.0 -959.0 -0.34 320.0 -376.0 -0.29 -0.4447 -0.9967 3025393 ChemDiv3_005658 CC(C)CCNc1ncc2C(=O)CC(Cc2n1)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B05 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 3119139 ChemDiv3_005659 OC(=O)c1ccc2NC(C3Cc4ccccc4C3c2c1)c5cccc(Cl)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B06 compound treatment 360.0 -999.0 -0.35 400.0 -296.0 -0.23 -0.4114 -0.977 3119140 ChemDiv3_005660 CC(NC(=S)NCCc1ccc(cc1)S(=O)(=O)N)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B07 compound treatment 1120.0 -239.0 -0.08 280.0 -416.0 -0.32 -0.2859 -0.8647 3119141 ChemDiv3_005661 Cc1ccc(cc1)S(=O)(=O)/N=C(/NCc2ccc(Cl)cc2)\Nc3nc(C)cc(C)n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B08 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 3119142 ChemDiv3_005662 COc1cc(OC)nc(NC(=O)CS(=O)(=O)c2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B09 compound treatment 520.0 -839.0 -0.3 560.0 -136.0 -0.1 -0.2844 -0.9016 3025462 ChemDiv3_005663 CC(=O)OC(C(=O)Nc1cccc(C)n1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B10 compound treatment 360.0 -999.0 -0.35 3880.0 3180.0 2.44 1.4778 0.5984 3119143 ChemDiv3_005664 CN(C)c1ccc(/C=c\2/sc3nnc(c4ccccc4)n3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B11 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3025465 ChemDiv3_005665 Cc1cc(C)c2nc(SCC=C)nc(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B12 compound treatment 240.0 -1120.0 -0.4 240.0 -456.0 -0.35 -0.5283 -0.9981 3119144 ChemDiv3_005666 Cc1nn(CC(O)c2ccccc2)c(C)c1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B13 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3025466 ChemDiv3_005667 O=C(Nc1ccccc1)C(=C2Nc3ccccc3N2)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B14 compound treatment 320.0 -1040.0 -0.37 400.0 -296.0 -0.23 -0.4214 -0.9731 3119145 ChemDiv3_005668 COc1ccc(cc1CNC(=O)c2ccco2)c3nn(C)c(=O)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B15 compound treatment 280.0 -1080.0 -0.38 800.0 104.0 0.08 -0.2143 -0.5482 3025468 ChemDiv3_005669 Brc1ccc2NC(=O)/C(=C\3/C(=O)N(CC=C)c4ccccc34)/c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B16 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 1428305 ChemDiv3_005670 Cn1c(nn(CN2CCC(CC2)C(=O)N)c1=S)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B17 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 3119146 ChemDiv3_005671 O=c1[nH]c2SC3C4CCC(C4)C3C(c5ccco5)c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B18 compound treatment 360.0 -999.0 -0.35 240.0 -456.0 -0.35 -0.4982 -1.0 1327349 ChemDiv3_005672 Cn1c(=S)n(CN2CCC(CC2)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B19 compound treatment 1320.0 -38.8 -0.01 320.0 -376.0 -0.29 -0.214 -0.7399 3119147 ChemDiv3_005673 Clc1ccc2oc(cc(=NCc3ccco3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B20 compound treatment 240.0 -1120.0 -0.4 280.0 -416.0 -0.32 -0.5066 -0.9942 3119148 ChemDiv3_005674 COc1cc(CN(C2CCCCC2)C(=O)/C(=C/c3cccnc3)/NC(=O)c4ccccc4)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B21 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 3025473 ChemDiv3_005675 NC(=O)c1ccccc1/N=c\2/cc(oc3ccc(Cl)cc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B22 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 1669328 ChemDiv3_005676 C[N+]1(CCOC(=O)Nc2ccccc2)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B23 mock treatment 360.0 -999.0 -0.35 440.0 -256.0 -0.2 -0.3896 -0.9615 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 B24 mock treatment 360.0 -999.0 -0.35 800.0 104.0 0.08 -0.1942 -0.5348 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C01 compound treatment 2760.0 1400.0 0.5 360.0 -336.0 -0.26 0.169 0.3016 3119149 ChemDiv3_005677 FC(F)(F)c1cc(nc2c(Br)c(nn12)C(=O)N3CCN4CCCC4C3)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C02 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 1786599 ChemDiv3_005678 COc1ccc(CCNC(=O)c2ccc(cc2)C3SCC(=O)N3Cc4ccccc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C03 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 1533618 ChemDiv3_005679 COC(=O)c1c(NC(=O)C2C(C3CCC2O3)C(=O)O)scc1c4ccc(cc4)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C04 compound treatment 240.0 -1120.0 -0.4 360.0 -336.0 -0.26 -0.4632 -0.9783 3119273 ChemDiv3_005680 CC(Sc1nc(ccc1C#N)c2cccnc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C05 compound treatment 360.0 -999.0 -0.35 200.0 -496.0 -0.38 -0.5199 -0.9993 3119274 ChemDiv3_005681 Cc1nn(C)cc1CNC(=O)c2cc(nc3ccc(Br)cc23)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C06 compound treatment 440.0 -919.0 -0.33 320.0 -376.0 -0.29 -0.4347 -0.9982 3025028 ChemDiv3_005682 C[N+]1(CCOC(=O)C2(CCCC2)c3ccccc3)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C07 compound treatment 5600.0 4240.0 1.5 440.0 -256.0 -0.2 0.9248 0.6095 1669227 ChemDiv3_005683 CCOc1ccccc1C(=O)N2c3ccccc3Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C08 compound treatment 280.0 -1080.0 -0.38 400.0 -296.0 -0.23 -0.4314 -0.9691 3119275 ChemDiv3_005684 CCOP(=Nc1nc2ccccc2n3nnnc13)(OCC)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C09 compound treatment 280.0 -1080.0 -0.38 400.0 -296.0 -0.23 -0.4314 -0.9691 3025032 ChemDiv3_005685 CCSc1nc2c(N)ncnc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C10 compound treatment 240.0 -1120.0 -0.4 400.0 -296.0 -0.23 -0.4415 -0.9651 1567167 ChemDiv3_005686 COc1ccc(cc1)S(=O)(=O)Nc2cc3oc4ccccc4c3cc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C11 compound treatment 440.0 -919.0 -0.33 200.0 -496.0 -0.38 -0.4999 -0.997 3025036 ChemDiv3_005687 Cc1ccc(cc1)N2Cc3cc(C)c(C)cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C12 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 3119276 ChemDiv3_005688 CN1CCCc2cc(/C=N/n3c(S)nnc3C(F)(F)F)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C13 compound treatment 280.0 -1080.0 -0.38 240.0 -456.0 -0.35 -0.5183 -0.999 3025038 ChemDiv3_005689 Clc1ccc2oc(nc2c1)c3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C14 compound treatment 240.0 -1120.0 -0.4 120.0 -576.0 -0.44 -0.5935 -0.9985 1582370 ChemDiv3_005690 O=S(=O)(Nc1ccccc1)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C15 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3025041 ChemDiv3_005691 OC(=O)CCSC1CC(=O)N(C1=O)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C16 compound treatment 280.0 -1080.0 -0.38 240.0 -456.0 -0.35 -0.5183 -0.999 3119277 ChemDiv3_005692 O=c1oc2ccc(NS(=O)(=O)c3cccc4ccccc34)cc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C17 compound treatment 280.0 -1080.0 -0.38 640.0 -56.3 -0.04 -0.3011 -0.7819 3025042 ChemDiv3_005693 C[N+]1(Cc2ccccc2C1)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C18 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 1403217 ChemDiv3_005694 Brc1ccc2n(CC=C)c3nc4ccccc4nc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C19 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 3119278 ChemDiv3_005695 CCCN1C(=O)C(O)(C2CC(=O)CC(C)(C)O2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C20 compound treatment 320.0 -1040.0 -0.37 400.0 -296.0 -0.23 -0.4214 -0.9731 1197673 ChemDiv3_005696 Cc1ccc(NC2SC(=O)NC2=O)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C21 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 1696774 ChemDiv3_005697 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2cc(OC)ccc2OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C22 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3442336 ChemDiv3_005698 Cc1cn(C2CCC(CO)O2)c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C23 mock treatment 240.0 -1120.0 -0.4 280.0 -416.0 -0.32 -0.5066 -0.9942 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 C24 mock treatment 3400.0 2040.0 0.72 240.0 -456.0 -0.35 0.2644 0.3286 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D01 compound treatment 2160.0 801.0 0.28 280.0 -416.0 -0.32 -0.025 -0.0584 3119279 ChemDiv3_005699 COc1ccc(NC(=N)Nc2nc(=O)cc(CSc3nc4ccccc4s3)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D02 compound treatment 6120.0 4760.0 1.69 240.0 -456.0 -0.35 0.9466 0.5488 3025080 ChemDiv3_005700 CC(C)(C)c1cc(c2Oc3cc(C#N)c(C#N)cc3Oc2c1)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D03 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 3119280 ChemDiv3_005701 Cc1ccc(Nc2nc(=O)cc(CSc3nc4ccccc4s3)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D04 compound treatment 240.0 -1120.0 -0.4 240.0 -456.0 -0.35 -0.5283 -0.9981 3025082 ChemDiv3_005702 Clc1ccccc1C2CC(=O)c3cnn(c4nc5ccccc5s4)c3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D05 compound treatment 360.0 -999.0 -0.35 320.0 -376.0 -0.29 -0.4548 -0.9949 3119281 ChemDiv3_005703 C/N=C/1\SC(CC(=O)Nc2cccc(c2)C(=O)O)C(=O)N1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D06 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3119282 ChemDiv3_005704 CC(NC(=S)N1CCc2ccccc2C1)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D07 compound treatment 440.0 -919.0 -0.33 320.0 -376.0 -0.29 -0.4347 -0.9982 1192680 ChemDiv3_005705 CC(C)C(=O)N1C2=C(C(c3ccc(Cl)cc3)c4c1n(C)c(=O)n(C)c4=O)C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D08 compound treatment 1080.0 -279.0 -0.1 360.0 -336.0 -0.26 -0.2525 -0.9133 3119283 ChemDiv3_005706 OCCN1CCN(Cc2nc(O)c3ccccc3n2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D09 compound treatment 360.0 -999.0 -0.35 360.0 -336.0 -0.26 -0.4331 -0.9879 3119284 ChemDiv3_005707 COc1ccccc1N2CCN(CC2)C(=O)C(OC(=O)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D10 compound treatment 5600.0 4240.0 1.5 320.0 -376.0 -0.29 0.8596 0.5611 3025087 ChemDiv3_005708 CCOc1ccc(/C=c\2/sc3nnc(c4ccccc4C)n3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D11 compound treatment 320.0 -1040.0 -0.37 240.0 -456.0 -0.35 -0.5082 -0.9997 3119285 ChemDiv3_005709 Cc1cccc(c1)C(=O)OCCSc2nc(C)c3cc(C)c(C)cc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D12 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3025120 ChemDiv3_005710 CCOC(=O)c1ccc(Oc2nc(NC(C)(C)C)nc(n2)N(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D13 compound treatment 280.0 -1080.0 -0.38 400.0 -296.0 -0.23 -0.4314 -0.9691 3119286 ChemDiv3_005711 COC(=O)C1=C(C)N=C2SC(C)C(=O)N2C1c3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D14 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3025122 ChemDiv3_005712 COc1ccc(cc1CNC(=O)NC2CCCCC2)c3nn(C)c(=O)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D15 compound treatment 240.0 -1120.0 -0.4 280.0 -416.0 -0.32 -0.5066 -0.9942 3119287 ChemDiv3_005713 Cc1ccc(cc1)c2c(O)c3cc(C)c(C)cc3c4oc(=O)sc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D16 compound treatment 320.0 -1040.0 -0.37 240.0 -456.0 -0.35 -0.5082 -0.9997 1710143 ChemDiv3_005714 CN(C)S(=O)(=O)Nc1ccc(Oc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D17 compound treatment 400.0 -959.0 -0.34 240.0 -456.0 -0.35 -0.4882 -0.9999 3119288 ChemDiv3_005715 COC(=O)C1Sc2[nH]c(=O)sc2C(C1C(=O)OC)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D18 compound treatment 360.0 -999.0 -0.35 360.0 -336.0 -0.26 -0.4331 -0.9879 1126623 ChemDiv3_005716 Oc1ccc2ccccc2c1CN3CCc4ccccc4C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D19 compound treatment 360.0 -999.0 -0.35 240.0 -456.0 -0.35 -0.4982 -1.0 3119289 ChemDiv3_005717 Clc1ccc2oc(cc(=NCC3CCCO3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D20 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 1121936 ChemDiv3_005718 Cc1ccc(o1)C(=O)CC2(O)C(=O)Nc3ccccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D21 compound treatment 320.0 -1040.0 -0.37 400.0 -296.0 -0.23 -0.4214 -0.9731 3025125 ChemDiv3_005719 Clc1ccc2oc(c/c(=N\c3nccs3)/c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D22 compound treatment 240.0 -1120.0 -0.4 280.0 -416.0 -0.32 -0.5066 -0.9942 1496567 ChemDiv3_005720 C[N+]1(CC2COC(O2)c3ccco3)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D23 mock treatment 360.0 -999.0 -0.35 320.0 -376.0 -0.29 -0.4548 -0.9949 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 D24 mock treatment 400.0 -959.0 -0.34 320.0 -376.0 -0.29 -0.4447 -0.9967 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E01 compound treatment 1480.0 121.0 0.04 320.0 -376.0 -0.29 -0.1738 -0.5952 3119290 ChemDiv3_005721 Cc1nn(C)c(C)c1CNC(=O)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E02 compound treatment 3000.0 1640.0 0.58 360.0 -336.0 -0.26 0.2292 0.3598 1495208 ChemDiv3_005722 CCOC(=O)c1ccccc1NS(=O)(=O)c2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E03 compound treatment 3040.0 1680.0 0.6 1880.0 1180.0 0.91 1.0643 0.9791 3025127 ChemDiv3_005723 Fc1ccccc1CSc2nc(c3CCCc3c2C#N)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E04 compound treatment 1600.0 241.0 0.09 520.0 -176.0 -0.14 -0.0352 -0.2196 3119291 ChemDiv3_005724 Brc1ccc2ncnc(c3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E05 compound treatment 720.0 -639.0 -0.23 480.0 -216.0 -0.17 -0.2776 -0.9883 3119292 ChemDiv3_005725 CC(Oc1ccccc1)C(=O)Nc2scc3c2c(=O)oc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E06 compound treatment 640.0 -719.0 -0.25 360.0 -336.0 -0.26 -0.3628 -1.0 3025129 ChemDiv3_005726 CC(C)COc1ccc(cc1)C(=O)OCCN2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E07 compound treatment 600.0 -759.0 -0.27 640.0 -56.3 -0.04 -0.2209 -0.8102 3119293 ChemDiv3_005727 Cc1onc(c1C(=O)Oc2cccnc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E08 compound treatment 1040.0 -319.0 -0.11 400.0 -296.0 -0.23 -0.2408 -0.948 1605545 ChemDiv3_005728 CP(=O)(Nc1ccccn1)Oc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E09 compound treatment 1640.0 281.0 0.1 640.0 -56.3 -0.04 0.04 0.3681 1874575 ChemDiv3_005729 CCCC1(CN(CC2(CCC)CN(C1)C(=O)CC)C(=O)CC)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E10 compound treatment 680.0 -679.0 -0.24 440.0 -256.0 -0.2 -0.3094 -0.995 3119294 ChemDiv3_005730 O=C(COc1ccc(/C=c\2/sc3nc4ccccc4n3c2=O)cc1)N5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E11 compound treatment 1280.0 -78.8 -0.03 2280.0 1580.0 1.22 0.84 0.6907 3025179 ChemDiv3_005731 Cc1ccc(cc1)N2CCN(c3ccc(C)cc3)C24C(=O)c5ccccc5C4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E12 compound treatment 360.0 -999.0 -0.35 800.0 104.0 0.08 -0.1942 -0.5348 3119425 ChemDiv3_005732 C1CCC2(C1)N=C(C(=N2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E13 compound treatment 1160.0 -199.0 -0.07 520.0 -176.0 -0.14 -0.1455 -0.9538 3025181 ChemDiv3_005733 Clc1ccc2oc(nc2c1)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E14 compound treatment 1200.0 -159.0 -0.06 2560.0 1860.0 1.43 0.9719 0.6788 3119426 ChemDiv3_005734 CC1CCN(CC1)C(=O)c2ccc(NS(=O)(=O)c3cc(cc(C)c3C)C(C)(C)C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E15 compound treatment 1200.0 -159.0 -0.06 720.0 23.8 0.02 -0.0269 -0.4549 3025183 ChemDiv3_005735 CC(Sc1ccc(Br)c2cccc(C(=O)O)c12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E16 compound treatment 1280.0 -78.8 -0.03 560.0 -136.0 -0.1 -0.0937 -0.8656 3119427 ChemDiv3_005736 O=S(=O)(/C(=C\c1cn(nc1c2cc3ccccc3o2)c4ccccc4)/C#N)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E17 compound treatment 1080.0 -279.0 -0.1 320.0 -376.0 -0.29 -0.2742 -0.898 3025185 ChemDiv3_005737 CC(C)C[N+]1(C)Cc2ccccc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E18 compound treatment 1480.0 121.0 0.04 1000.0 304.0 0.23 0.1953 0.8236 3119428 ChemDiv3_005738 CC(C)n1c2ccc(C)cc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E19 compound treatment 1080.0 -279.0 -0.1 760.0 63.8 0.05 -0.0353 -0.3201 3025188 ChemDiv3_005739 CC1(C)CC(=O)CC(O1)C2(O)C(=O)N(Cc3ccccc3)c4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E20 compound treatment 5280.0 3920.0 1.39 880.0 184.0 0.14 1.0834 0.7748 1550690 ChemDiv3_005740 O=C1CSC(=O)N1CCN2C(=O)CSC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E21 compound treatment 4040.0 2680.0 0.95 1400.0 704.0 0.54 1.0546 0.9641 3119429 ChemDiv3_005741 COc1cc(C)c(cc1S(=O)(=O)N2CCN(CC2)c3cccc(Cl)c3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E22 compound treatment 2440.0 1080.0 0.38 440.0 -256.0 -0.2 0.1321 0.3065 3025192 ChemDiv3_005742 COc1ccc(NC(=O)CSc2nnc(Cc3c[nH]c4ccccc34)n2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E23 mock treatment 1920.0 561.0 0.2 560.0 -136.0 -0.1 0.0668 0.2971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 E24 mock treatment 360.0 -999.0 -0.35 1880.0 1180.0 0.91 0.3921 0.402 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F01 compound treatment 1000.0 -359.0 -0.13 800.0 104.0 0.08 -0.0337 -0.2243 3025134 ChemDiv3_005743 Clc1ccc(CSc2nnc(SCC(=O)N3CCc4ccccc4C3)s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F02 compound treatment 4200.0 2840.0 1.01 840.0 144.0 0.11 0.7907 0.7799 3119430 ChemDiv3_005744 OC(=O)c1cc2oc3ccccc3c4ccccc4oc2cc1C(=O)Nc5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F03 compound treatment 2720.0 1360.0 0.48 2920.0 2220.0 1.71 1.5486 0.8729 3025135 ChemDiv3_005745 Cc1cc(C)nc(NC2=NCCN2C(=O)Nc3ccc(Cl)c(Cl)c3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F04 compound treatment 3760.0 2400.0 0.85 1560.0 864.0 0.66 1.0712 0.9923 3119431 ChemDiv3_005746 Nc1ccccc1NC2=CC(=O)CC(C2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F05 compound treatment 5680.0 4320.0 1.53 1040.0 344.0 0.26 1.2706 0.8168 3119432 ChemDiv3_005747 NC(=N)NCCn1ccc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F06 compound treatment 920.0 -439.0 -0.16 760.0 63.8 0.05 -0.0755 -0.4624 3025138 ChemDiv3_005748 CC(=C1C(=O)c2ccccc2C1=O)NCCc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F07 compound treatment 1320.0 -38.8 -0.01 1000.0 304.0 0.23 0.1552 0.6643 3119433 ChemDiv3_005749 COC(=O)/C=C/1\SC(=NC1=O)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F08 compound treatment 920.0 -439.0 -0.16 680.0 -16.3 -0.01 -0.1189 -0.7613 1220960 ChemDiv3_005750 S=C(NCCN1CCOCC1)Nc2ccc(Nc3ccccc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F09 compound treatment 6160.0 4800.0 1.7 1640.0 944.0 0.72 1.7167 0.9275 3025143 ChemDiv3_005751 CC(=O)OC(C(=O)N1CCN(CC1)C(c2ccccc2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F10 compound treatment 2800.0 1440.0 0.51 920.0 224.0 0.17 0.483 0.8955 3119434 ChemDiv3_005752 COc1cc2CCN3COCC(=C3c2cc1OC)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F11 compound treatment 2080.0 721.0 0.26 7000.0 6300.0 4.84 3.603 0.7435 3119435 ChemDiv3_005753 CCOc1ccc2nc(NC(=O)Nc3ccc(F)cc3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F12 compound treatment 920.0 -439.0 -0.16 720.0 23.8 0.02 -0.0972 -0.62 3025194 ChemDiv3_005754 CCc1ccc(OC(C)C(=O)N(Cc2ccccc2)C3CCS(=O)(=O)C3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F13 compound treatment 640.0 -719.0 -0.25 1600.0 904.0 0.69 0.3103 0.4198 3119436 ChemDiv3_005755 CCC1SC2=NC(=C(C(N2C1=O)c3ccccc3Br)C(=O)OC)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F14 compound treatment 840.0 -519.0 -0.18 760.0 63.8 0.05 -0.0955 -0.5016 3025198 ChemDiv3_005756 COc1nnc(c2ccc(N3CCOCC3)c(NS(=O)(=O)c4ccc(C)cc4)c2)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F15 compound treatment 2880.0 1520.0 0.54 1760.0 1060.0 0.82 0.9591 0.9798 3119437 ChemDiv3_005757 O=C1N/C(=N/c2ccccc2)/CS1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F16 compound treatment 3000.0 1640.0 0.58 640.0 -56.3 -0.04 0.3812 0.6529 1202292 ChemDiv3_005758 CC1CCN(Cn2nc(oc2=S)c3ccccc3)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F17 compound treatment 3120.0 1760.0 0.62 920.0 224.0 0.17 0.5633 0.8693 3025202 ChemDiv3_005759 CCc1ccccc1Oc2coc3cc(OC(=O)c4ccccc4F)ccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F18 compound treatment 1120.0 -239.0 -0.08 440.0 -256.0 -0.2 -0.199 -0.9291 3119438 ChemDiv3_005760 CC(=O)Nc1ccc(/C=C/2\CCc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F19 compound treatment 1320.0 -38.8 -0.01 3760.0 3060.0 2.35 1.6535 0.703 3119439 ChemDiv3_005761 Clc1ccc2oc(cc(=NCCN3CCOCC3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F20 compound treatment 2280.0 921.0 0.33 360.0 -336.0 -0.26 0.0486 0.1166 3025205 ChemDiv3_005762 CC(C)N1CCc2c(C(=O)N)c(N)sc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F21 compound treatment 4640.0 3280.0 1.16 1440.0 744.0 0.57 1.2268 0.9463 3119440 ChemDiv3_005763 CCc1ccc2oc(cc(=NCc3cccnc3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F22 compound treatment 5320.0 3960.0 1.41 2400.0 1700.0 1.31 1.9185 0.9994 3026120 ChemDiv3_005764 C1CN2CCCN1C2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F23 mock treatment 3880.0 2520.0 0.89 1680.0 984.0 0.76 1.1665 0.9965 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 F24 mock treatment 3320.0 1960.0 0.7 2000.0 1300.0 1.0 1.1997 0.9842 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G01 compound treatment 880.0 -479.0 -0.17 920.0 224.0 0.17 0.0014 0.0057 3026121 ChemDiv3_005765 FC(F)(F)C1CC(Nc2cc(nn12)C(=O)NCCc3ccccc3)c4ccc(Br)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G02 compound treatment 360.0 -999.0 -0.35 1320.0 624.0 0.48 0.0881 0.1479 3026122 ChemDiv3_005766 O=S(=O)(NCCSc1ccccc1)c2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G03 compound treatment 5280.0 3920.0 1.39 280.0 -416.0 -0.32 0.7577 0.5308 3026123 ChemDiv3_005767 CCNS(=O)(=O)c1ccc(NC(=O)c2ccc(Cn3cc(Br)cn3)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G04 compound treatment 760.0 -599.0 -0.21 1160.0 464.0 0.36 0.1016 0.245 1181816 ChemDiv3_005768 CCOC(=O)c1sc2nc(N3CCCCC3)c4COC(C)(C)Cc4c2c1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G05 compound treatment 1680.0 321.0 0.11 1440.0 744.0 0.57 0.4843 0.8318 3026124 ChemDiv3_005769 Fc1ccc(cc1)N2CCN(CC2)C(=O)CC3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G06 compound treatment 760.0 -599.0 -0.21 680.0 -16.3 -0.01 -0.159 -0.7474 3026125 ChemDiv3_005770 CC(=O)Oc1ccc(cc1)C2OC(=O)c3ccccc3N2C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G07 compound treatment 880.0 -479.0 -0.17 1520.0 824.0 0.63 0.3271 0.4995 3119441 ChemDiv3_005771 CC1=C(C)CC(C(C1)C(=O)O)C(=O)NCc2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G08 compound treatment 760.0 -599.0 -0.21 1360.0 664.0 0.51 0.2101 0.3806 3026126 ChemDiv3_005772 Clc1ccc(cc1)S(=O)(=O)NCC(c2ccccc2)n3cc(nn3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G09 compound treatment 1360.0 1.25 0.0 1120.0 424.0 0.33 0.2304 0.7081 1391365 ChemDiv3_005773 CCCC1CN2CCC3=C(CCC3)C2(C)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G10 compound treatment 640.0 -719.0 -0.25 920.0 224.0 0.17 -0.0588 -0.1914 3119442 ChemDiv3_005774 CCCOc1ccc(cc1)C(=O)NCC2(CCOCC2)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G11 compound treatment 920.0 -439.0 -0.16 680.0 -16.3 -0.01 -0.1189 -0.7613 1049853 ChemDiv3_005775 CC(C)(C)C1CCc2[nH]c3ccccc3c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G12 compound treatment 680.0 -679.0 -0.24 800.0 104.0 0.08 -0.1139 -0.4493 3119443 ChemDiv3_005776 COc1ccc(cc1)C2Sc3nncn3N2Cc4ccc(C#N)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G13 compound treatment 360.0 -999.0 -0.35 440.0 -256.0 -0.2 -0.3896 -0.9615 1625614 ChemDiv3_005777 CC1=C(C(c2ccccc2)n3nc(nc3N1)c4ccccc4)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G14 compound treatment 640.0 -719.0 -0.25 480.0 -216.0 -0.17 -0.2977 -0.9784 1875792 ChemDiv3_005778 COC(=O)c1c(C)oc2ccc(cc12)N(C(=O)C3CCCCC3)S(=O)(=O)c4cc(C)c(C)cc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G15 compound treatment 1360.0 1.25 0.0 2040.0 1340.0 1.03 0.7298 0.7074 3026127 ChemDiv3_005779 CC(=O)Oc1csc2ccc(Br)c3cccc1c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G16 compound treatment 1920.0 561.0 0.2 1640.0 944.0 0.72 0.6531 0.8692 3119444 ChemDiv3_005780 Cc1ccc(cc1)S(=O)(=O)NC(O)C(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G17 compound treatment 880.0 -479.0 -0.17 1400.0 704.0 0.54 0.2619 0.4625 3026128 ChemDiv3_005781 C[N+]1(CC=C)Cc2ccccc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G18 compound treatment 7520.0 6160.0 2.19 360.0 -336.0 -0.26 1.363 0.6193 3119445 ChemDiv3_005782 Cc1ccc2n(Cc3ccccc3)c4nc5ccccc5nc4c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G19 compound treatment 1800.0 441.0 0.16 2920.0 2220.0 1.71 1.3179 0.7687 1377452 ChemDiv3_005783 CNC(=O)C1=NCCCc2cc(OC)c(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G20 compound treatment 1360.0 1.25 0.0 1760.0 1060.0 0.82 0.5778 0.7075 1867771 ChemDiv3_005784 CCCN1C(=O)SC(CC(=O)Nc2cccc3ccccc23)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G21 compound treatment 6800.0 5440.0 1.93 840.0 144.0 0.11 1.4429 0.7463 3119446 ChemDiv3_005785 COc1ccc(cc1)c2nc(N)n(n2)C(=O)CCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G22 compound treatment 600.0 -759.0 -0.27 720.0 23.8 0.02 -0.1774 -0.6577 3026129 ChemDiv3_005786 COc1ccccc1c2nnc3ccc4ccccc4n23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G23 mock treatment 1840.0 481.0 0.17 1000.0 304.0 0.23 0.2856 0.9882 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 G24 mock treatment 480.0 -879.0 -0.31 520.0 -176.0 -0.14 -0.3161 -0.9302 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H01 compound treatment 480.0 -879.0 -0.31 360.0 -336.0 -0.26 -0.403 -0.9956 3119447 ChemDiv3_005787 COc1ccc(cc1)c2cc(NC(=O)N3CCc4ccccc4C3)c5ccccc5n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H02 compound treatment 1200.0 -159.0 -0.06 960.0 264.0 0.2 0.1034 0.4918 3026130 ChemDiv3_005788 Cc1ccc(Oc2ccc3C(=O)N(CC(=O)O)C(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H03 compound treatment 520.0 -839.0 -0.3 680.0 -16.3 -0.01 -0.2192 -0.7361 3119448 ChemDiv3_005789 Cc1cc(C)nc(N/C(=N\S(=O)(=O)Cc2ccccc2)/Nc3ccccc3Br)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H04 compound treatment 3440.0 2080.0 0.74 7000.0 6300.0 4.84 3.9441 0.8057 3026131 ChemDiv3_005790 CCN/1C(=O)CS\C1=C(/C#N)\S(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H05 compound treatment 10760.0 9400.0 3.34 600.0 -96.3 -0.07 2.306 0.6913 3119585 ChemDiv3_005791 CC1CCc2ccccc2N1C(=N)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H06 compound treatment 1080.0 -279.0 -0.1 1280.0 584.0 0.45 0.247 0.5381 3119586 ChemDiv3_005792 Clc1ccc2[nH]c(=O)c(SCC(=O)NC3CCCC3)c(c4ccccc4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H07 compound treatment 2640.0 1280.0 0.45 560.0 -136.0 -0.1 0.2474 0.5305 3026132 ChemDiv3_005793 O=C(CN1C(=O)c2ccccc2C1=O)N3CCN=C3c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H08 compound treatment 6760.0 5400.0 1.92 560.0 -136.0 -0.1 1.2809 0.6675 3026133 ChemDiv3_005794 OC1CCN(CC1)C(=S)Nc2ccc(Nc3ccccc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H09 compound treatment 8280.0 6920.0 2.46 6800.0 6100.0 4.69 5.0496 0.9545 3119587 ChemDiv3_005795 O=C(C(Sc1nnc[nH]1)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H10 compound treatment 1160.0 -199.0 -0.07 440.0 -256.0 -0.2 -0.189 -0.9042 3119588 ChemDiv3_005796 COc1ccc(cc1)C(=O)/N=C/2\CCC(=C3N2CCc4cc(OC)c(OC)cc34)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H11 compound treatment 480.0 -879.0 -0.31 560.0 -136.0 -0.1 -0.2944 -0.8953 3026134 ChemDiv3_005797 CCCc1cc(=O)nc(NC(=N)Nc2cccc(C)c2)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H12 compound treatment 720.0 -639.0 -0.23 600.0 -96.3 -0.07 -0.2125 -0.8915 3119589 ChemDiv3_005798 COc1ccc(CN(C2CCS(=O)(=O)C2)C(=O)c3cccc(Cl)c3)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H13 compound treatment 1240.0 -119.0 -0.04 520.0 -176.0 -0.14 -0.1255 -0.8853 3026135 ChemDiv3_005799 CCSc1nc(cc(c1C#N)C(F)(F)F)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H14 compound treatment 840.0 -519.0 -0.18 480.0 -216.0 -0.17 -0.2475 -0.9987 3119590 ChemDiv3_005800 C(Oc1nnc(c2ccccc2)c3ccccc13)C4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H15 compound treatment 600.0 -759.0 -0.27 920.0 224.0 0.17 -0.0689 -0.2157 1579607 ChemDiv3_005801 Cc1c(N2C(=O)SC(CC(=O)O)C2=O)c(=O)n(c3ccccc3)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H16 compound treatment 1200.0 -159.0 -0.06 600.0 -96.3 -0.07 -0.0921 -0.991 3119591 ChemDiv3_005802 Cn1c(COc2ccccc2)n[nH]c1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H17 compound treatment 1560.0 201.0 0.07 440.0 -256.0 -0.2 -0.0886 -0.4235 3119592 ChemDiv3_005803 Cc1ccc2oc(cc(=NCCN3CCOCC3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H18 compound treatment 1120.0 -239.0 -0.08 720.0 23.8 0.02 -0.047 -0.5425 1678503 ChemDiv3_005804 O=C1NC(Oc2ccccc12)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H19 compound treatment 720.0 -639.0 -0.23 880.0 184.0 0.14 -0.0605 -0.2266 3119593 ChemDiv3_005805 Clc1ccc2oc(cc(=NCCCN3CCOCC3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H20 compound treatment 2800.0 1440.0 0.51 1040.0 344.0 0.26 0.5481 0.9527 3026136 ChemDiv3_005806 CS(=O)(=O)Nc1ccc2C(=O)NC(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H21 compound treatment 1920.0 561.0 0.2 2440.0 1740.0 1.34 1.0874 0.8034 3119594 ChemDiv3_005807 CCc1ccc2oc(cc(=NCC(=O)O)c2c1)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H22 compound treatment 800.0 -559.0 -0.2 5080.0 4380.0 3.37 2.2396 0.6643 3026137 ChemDiv3_005808 CC(C)CC1CCCCC1OC(=O)C[N+]2(C)CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H23 mock treatment 840.0 -519.0 -0.18 920.0 224.0 0.17 -0.0087 -0.0344 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 H24 mock treatment 640.0 -719.0 -0.25 1120.0 424.0 0.33 0.0497 0.1203 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I01 compound treatment 280.0 -1080.0 -0.38 2720.0 2020.0 1.55 0.828 0.5175 1254817 ChemDiv3_005809 CCCc1cc(C(=O)OC)c(NC(=O)CCCC(=O)O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I02 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 3119595 ChemDiv3_005810 COc1ccc(cc1)c2cc(c(C#N)c(SCCCn3c(=O)[nH]c4ccccc34)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I03 compound treatment 160.0 -1200.0 -0.43 320.0 -376.0 -0.29 -0.5049 -0.9822 3026138 ChemDiv3_005811 CN(C)c1ccc(NC(=O)C2(CC3CC4C2)CC(C3)(C4)n5cnc(Cl)n5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I04 compound treatment 1600.0 241.0 0.09 360.0 -336.0 -0.26 -0.122 -0.4487 1551640 ChemDiv3_005812 CCC1(C)Cc2c(C#N)c(N)sc(=S)c2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I05 compound treatment 520.0 -839.0 -0.3 2520.0 1820.0 1.4 0.7796 0.5447 3026139 ChemDiv3_005813 CN(Cc1c(C)nn(C)c1C)C(=O)c2cc(nc3ccc(Br)cc23)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I06 compound treatment 1120.0 -239.0 -0.08 4000.0 3300.0 2.54 1.7336 0.6831 3119596 ChemDiv3_005814 CCNc1nc(OCC)nc(n1)N2CCC(Cc3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I07 compound treatment 280.0 -1080.0 -0.38 360.0 -336.0 -0.26 -0.4531 -0.9816 3119597 ChemDiv3_005815 CS(=O)(=O)N1N=C(CC1c2ccccc2F)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I08 compound treatment 280.0 -1080.0 -0.38 320.0 -376.0 -0.29 -0.4748 -0.9904 3026140 ChemDiv3_005816 Clc1ccc(cc1)S(=O)(=O)NC2CCCCC2n3cc(nn3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I09 compound treatment 480.0 -879.0 -0.31 1560.0 864.0 0.66 0.2485 0.3391 3119598 ChemDiv3_005817 CCOc1ccc(Cc2nc(C)c(CC(=O)N3CCOCC3)c(O)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I10 compound treatment 240.0 -1120.0 -0.4 480.0 -216.0 -0.17 -0.398 -0.9252 3026141 ChemDiv3_005818 COC(=O)c1ccc(CN(Cc2ccc(o2)C(=O)OC)C(C)(C)C)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I11 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 1448703 ChemDiv3_005819 CCN(c1ccccc1)C2(O)C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I12 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 1324344 ChemDiv3_005820 COc1cc2CCN(C(c3ccccc3)c2cc1OC)C(=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I13 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 3026142 ChemDiv3_005821 Brc1ccc(cc1)C2C3=C(CCCC3=O)Nc4nc(nn24)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I14 compound treatment 600.0 -759.0 -0.27 520.0 -176.0 -0.14 -0.286 -0.9494 1875830 ChemDiv3_005822 O=C(C1CCCCC1)N(c2ccc3oc4CCCCc4c3c2)S(=O)(=O)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I15 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3119599 ChemDiv3_005823 Cc1cc(C)c2cccc(NC(=O)COc3ccc4oc5CCCCc5c4c3)c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I16 compound treatment 1800.0 441.0 0.16 280.0 -416.0 -0.32 -0.1153 -0.324 3026143 ChemDiv3_005824 OC(NC(=O)c1cccnc1)C(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I17 compound treatment 400.0 -959.0 -0.34 240.0 -456.0 -0.35 -0.4882 -0.9999 3026144 ChemDiv3_005825 C[N+]1(Cc2ccco2)Cc3ccccc3C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I18 compound treatment 320.0 -1040.0 -0.37 400.0 -296.0 -0.23 -0.4214 -0.9731 1286497 ChemDiv3_005826 COC(=O)CCn1cnc(c1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I19 compound treatment 880.0 -479.0 -0.17 560.0 -136.0 -0.1 -0.1941 -0.9729 3119600 ChemDiv3_005827 COC(=O)CSc1nc(N2CCOCC2)c3CSC(C)(C)Cc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I20 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 1867775 ChemDiv3_005828 CCCN1C(=O)SC(CC(=O)Nc2ccc(cc2)C(=O)OCC)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I21 compound treatment 280.0 -1080.0 -0.38 360.0 -336.0 -0.26 -0.4531 -0.9816 3119601 ChemDiv3_005829 Nc1nc(nn1C(=O)Cc2ccccc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I22 compound treatment 360.0 -999.0 -0.35 3880.0 3180.0 2.44 1.4778 0.5984 1344824 ChemDiv3_005830 C[N+](C)(C)CCOc1ccc2nc(N)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I23 mock treatment 2840.0 1480.0 0.53 360.0 -336.0 -0.26 0.189 0.3229 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 I24 mock treatment 1440.0 81.3 0.03 200.0 -496.0 -0.38 -0.249 -0.6517 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J01 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 3119602 ChemDiv3_005831 CCOC(=O)C1CCCN(Cc2nc(N)nc(Nc3ccc(Cl)cc3)n2)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J02 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 3119603 ChemDiv3_005832 COc1ccc(OCC(=O)NC(=S)N2CCCc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J03 compound treatment 360.0 -999.0 -0.35 480.0 -216.0 -0.17 -0.3679 -0.9403 3026145 ChemDiv3_005833 Cn1nc(SCC(=O)N2c3ccccc3CCc4ccccc24)sc1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J04 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 3119604 ChemDiv3_005834 CCCCc1ccc(cc1)N/2C(=O)CS\C2=C(\C#N)/S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J05 compound treatment 320.0 -1040.0 -0.37 760.0 63.8 0.05 -0.226 -0.6079 3026146 ChemDiv3_005835 CN(C)/C=N/c1c(C)[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J06 compound treatment 280.0 -1080.0 -0.38 360.0 -336.0 -0.26 -0.4531 -0.9816 3119605 ChemDiv3_005836 Clc1ccc2[nH]c(=O)c(SCC(=O)NCc3ccco3)c(c4ccccc4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J07 compound treatment 120.0 -1240.0 -0.44 240.0 -456.0 -0.35 -0.5584 -0.9937 1871803 ChemDiv3_005837 CC1CC(C)(C)Nc2ccc(OC(=O)c3ccco3)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J08 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 3119606 ChemDiv3_005838 NS(=O)(=O)c1ccc(NC(=S)N2CCC(O)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J09 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 3026147 ChemDiv3_005839 O=C(CSc1nnc2sc3ccccc3n12)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J10 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3119607 ChemDiv3_005840 COc1cc2CCN3C(=O)CCC(=C3c2cc1OC)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J11 compound treatment 320.0 -1040.0 -0.37 240.0 -456.0 -0.35 -0.5082 -0.9997 3026148 ChemDiv3_005841 COc1ccccc1c2nnc(SCC(=O)N3CCc4ccccc4C3)n2CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J12 compound treatment 400.0 -959.0 -0.34 360.0 -336.0 -0.26 -0.423 -0.9907 3026204 ChemDiv3_005842 CC(C)c1ccc(CN(C2CCS(=O)(=O)C2)C(=O)COc3cc(C)c(Cl)c(C)c3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J13 compound treatment 440.0 -919.0 -0.33 440.0 -256.0 -0.2 -0.3696 -0.9708 3026205 ChemDiv3_005843 CCOc1ccc(cc1)c2cc(c(C#N)c(SCC)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J14 compound treatment 800.0 -559.0 -0.2 360.0 -336.0 -0.26 -0.3227 -0.9915 3026206 ChemDiv3_005844 Cc1ccc(cc1)c2nnc(OCc3cccnc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J15 compound treatment 400.0 -959.0 -0.34 280.0 -416.0 -0.32 -0.4665 -0.9995 3026207 ChemDiv3_005845 COc1ccc(NC(=O)CC2SC(=NC2=O)Nc3ccc(OC)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J16 compound treatment 4360.0 3000.0 1.06 360.0 -336.0 -0.26 0.5703 0.5206 1585350 ChemDiv3_005846 Cc1ccc(cc1)C(=O)Cc2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J17 compound treatment 400.0 -959.0 -0.34 320.0 -376.0 -0.29 -0.4447 -0.9967 3026208 ChemDiv3_005847 CN(C)CCN=c1cc(oc2ccc(C)cc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J18 compound treatment 2000.0 641.0 0.23 9640.0 8940.0 6.87 5.016 0.7301 3026209 ChemDiv3_005848 O=C1CS/C(=N/c2ccccn2)/N1C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J19 compound treatment 400.0 -959.0 -0.34 400.0 -296.0 -0.23 -0.4013 -0.9809 3119739 ChemDiv3_005849 CN(C)CCN=c1cc(oc2ccc(Cl)cc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J20 compound treatment 2760.0 1400.0 0.5 320.0 -376.0 -0.29 0.1472 0.2561 1663031 ChemDiv3_005850 CC1C=C(C)C2C(C)C1COC2c3ccc(OC(=O)C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J21 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 3119740 ChemDiv3_005851 Cc1sc2ncn(CC(=O)O)c(=O)c2c1c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J22 compound treatment 1360.0 1.25 0.0 1040.0 344.0 0.26 0.1869 0.7083 3119741 ChemDiv3_005852 C[N+]1(CC(=O)OCCCC2CCCCC2)CCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J23 mock treatment 2040.0 681.0 0.24 320.0 -376.0 -0.29 -0.0334 -0.0886 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 J24 mock treatment 7480.0 6120.0 2.17 320.0 -376.0 -0.29 1.3312 0.6077 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K01 compound treatment 1360.0 1.25 0.0 760.0 63.8 0.05 0.0349 0.7135 3026210 ChemDiv3_005853 Nc1c(sc2nc(c3CCCCc3c12)C(F)(F)F)C(=O)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K02 compound treatment 4000.0 2640.0 0.94 1920.0 1220.0 0.94 1.3269 1.0 3119742 ChemDiv3_005854 OC(=O)CCSc1nc(cc(c1C#N)C(F)(F)F)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K03 compound treatment 440.0 -919.0 -0.33 720.0 23.8 0.02 -0.2176 -0.6665 1881588 ChemDiv3_005855 Fc1ccc(Cn2cc(NC(=O)c3cnccn3)cn2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K04 compound treatment 1080.0 -279.0 -0.1 480.0 -216.0 -0.17 -0.1873 -0.9694 3119743 ChemDiv3_005856 S=c1[nH]c(N2CCCC2)c3CCCCc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K05 compound treatment 1040.0 -319.0 -0.11 720.0 23.8 0.02 -0.0671 -0.5855 3119744 ChemDiv3_005857 CC(=O)NC1C(=O)N=C(S)N(C1=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K06 compound treatment 480.0 -879.0 -0.31 440.0 -256.0 -0.2 -0.3595 -0.9754 1344940 ChemDiv3_005858 CCNc1nc(nc(n1)N2CCC(Cc3ccccc3)CC2)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K07 compound treatment 720.0 -639.0 -0.23 760.0 63.8 0.05 -0.1256 -0.5419 3119745 ChemDiv3_005859 Cc1ccc(cc1)c2n(C)cc3n(C)c(=O)n(C)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K08 compound treatment 760.0 -599.0 -0.21 1080.0 384.0 0.29 0.0581 0.1601 3026211 ChemDiv3_005860 COc1ccc(/C=N/n2cnnc2S)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K09 compound treatment 320.0 -1040.0 -0.37 560.0 -136.0 -0.1 -0.3345 -0.8733 3119746 ChemDiv3_005861 Cc1cccc(C(CC(=O)N2CCCC2)c3ccccc3)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K10 compound treatment 800.0 -559.0 -0.2 520.0 -176.0 -0.14 -0.2358 -0.9827 3119747 ChemDiv3_005862 O=C(Nc1ccc(cc1)C(=O)NCC2OCCc3ccccc23)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K11 compound treatment 520.0 -839.0 -0.3 440.0 -256.0 -0.2 -0.3495 -0.9798 3026212 ChemDiv3_005863 FC(F)(F)c1cc(c2ccccc2)n3c4ccccc4nc3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K12 compound treatment 880.0 -479.0 -0.17 560.0 -136.0 -0.1 -0.1941 -0.9729 3119748 ChemDiv3_005864 C(Cc1ccccc1)Sc2nnc3sc4ccccc4n23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K13 compound treatment 2880.0 1520.0 0.54 2080.0 1380.0 1.06 1.1328 0.9507 3026213 ChemDiv3_005865 NS(=O)(=O)c1ccc(CCNC(=O)Nc2cccc(c2)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K14 compound treatment 1920.0 561.0 0.2 3520.0 2820.0 2.17 1.6737 0.7688 3119749 ChemDiv3_005866 Brc1ccc(NS(=O)(=O)c2ccc3SC(=O)c4cccc2c34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K15 compound treatment 7320.0 5960.0 2.11 2080.0 1380.0 1.06 2.2465 0.9493 3026214 ChemDiv3_005867 COC(=O)c1cc2sc3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K16 compound treatment 2200.0 841.0 0.3 1320.0 624.0 0.48 0.5496 0.9741 3119750 ChemDiv3_005868 CCOC(=O)c1c(oc2c(cc(O)cc12)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K17 compound treatment 7320.0 5960.0 2.11 560.0 -136.0 -0.1 1.4214 0.6713 3026215 ChemDiv3_005869 C[N+]1(CCOc2ccccc2)Cc3ccccc3C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K18 compound treatment 960.0 -399.0 -0.14 800.0 104.0 0.08 -0.0437 -0.2692 3119751 ChemDiv3_005870 C(Cn1c2ccccc2c3nc4ccccc4nc13)Oc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K19 compound treatment 880.0 -479.0 -0.17 360.0 -336.0 -0.26 -0.3026 -0.9794 3119752 ChemDiv3_005871 CC1(C)Cc2c(CO1)c(=O)n(c3ccccc3)c4ncnc(N)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K20 compound treatment 1360.0 1.25 0.0 720.0 23.8 0.02 0.0132 0.7241 1174145 ChemDiv3_005872 Cc1ccccc1NC(=O)CC2SC(=O)N(C2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K21 compound treatment 5680.0 4320.0 1.53 2800.0 2100.0 1.62 2.226 0.9997 3119753 ChemDiv3_005873 CC1=NN(C(=O)C1C(=O)c2ccccc2Br)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K22 compound treatment 600.0 -759.0 -0.27 680.0 -16.3 -0.01 -0.1991 -0.7391 3119754 ChemDiv3_005874 FC(F)(F)C1(N=C(CCC2CCCCC2)Nc3c1c(=O)[nH]c(=O)n3Cc4ccco4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K23 mock treatment 960.0 -399.0 -0.14 2440.0 1740.0 1.34 0.8466 0.6289 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 K24 mock treatment 1040.0 -319.0 -0.11 560.0 -136.0 -0.1 -0.1539 -0.9992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L01 compound treatment 4560.0 3200.0 1.14 960.0 264.0 0.2 0.9462 0.8202 3026216 ChemDiv3_005875 Cc1ccc(SCc2cc(=O)nc(NC(=N)Nc3ccccc3)[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L02 compound treatment 920.0 -439.0 -0.16 6560.0 5860.0 4.5 3.0731 0.6823 3026217 ChemDiv3_005876 CC1(C)CC(=O)c2cnc(NCc3ccccc3)nc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L03 compound treatment 1040.0 -319.0 -0.11 760.0 63.8 0.05 -0.0453 -0.3681 3119755 ChemDiv3_005877 COC(=O)C1=C(C)N/C(=C\c2ccc(cc2)C(C)(C)C)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L04 compound treatment 840.0 -519.0 -0.18 400.0 -296.0 -0.23 -0.2909 -0.9945 3119756 ChemDiv3_005878 Cn1c(=O)n(C)c2nc(NC3CCCC3)[nH]c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L05 compound treatment 760.0 -599.0 -0.21 4600.0 3900.0 3.0 1.969 0.6553 1476024 ChemDiv3_005879 S=C(CN1CCCC1=S)NCCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L06 compound treatment 1040.0 -319.0 -0.11 1160.0 464.0 0.36 0.1718 0.4599 3026218 ChemDiv3_005880 CN1CCN(CC1)C(=O)CSc2c(c3ccccc3)c4cc(Cl)ccc4[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L07 compound treatment 760.0 -599.0 -0.21 360.0 -336.0 -0.26 -0.3327 -0.9953 3119757 ChemDiv3_005881 COCc1cc(O)nc(NC(=N)Nc2ccccc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L08 compound treatment 520.0 -839.0 -0.3 680.0 -16.3 -0.01 -0.2192 -0.7361 3119758 ChemDiv3_005882 OC(C1CCN(CC1)C(=S)NCCc2ccccc2)(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L09 compound treatment 800.0 -559.0 -0.2 520.0 -176.0 -0.14 -0.2358 -0.9827 3026219 ChemDiv3_005883 CC1CCc2cc(F)ccc2N1C(=O)CN3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L10 compound treatment 520.0 -839.0 -0.3 520.0 -176.0 -0.14 -0.3061 -0.9364 3119759 ChemDiv3_005884 COc1cc2CCN3CN(CC(=O)O)CC(=C3c2cc1OC)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L11 compound treatment 1240.0 -119.0 -0.04 480.0 -216.0 -0.17 -0.1472 -0.8593 3026220 ChemDiv3_005885 CC1=CC(C)(C)Nc2ccc(OCC(=O)N3c4ccccc4Sc5ccccc35)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L12 compound treatment 520.0 -839.0 -0.3 560.0 -136.0 -0.1 -0.2844 -0.9016 3119760 ChemDiv3_005886 Cc1ccc2c(Cl)c(sc2c1)C(=O)N(Cc3cccs3)C4CCS(=O)(=O)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L13 compound treatment 880.0 -479.0 -0.17 1880.0 1180.0 0.91 0.5225 0.5652 3119761 ChemDiv3_005887 COc1cc(/C=c/2\sc3nc(nn3c2=O)c4ccccc4C)cc(Br)c1OC(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L14 compound treatment 800.0 -559.0 -0.2 640.0 -56.3 -0.04 -0.1707 -0.8414 3026221 ChemDiv3_005888 CCCNC(=O)CN1C(=O)COc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L15 compound treatment 1120.0 -239.0 -0.08 2400.0 1700.0 1.31 0.865 0.6599 3119762 ChemDiv3_005889 OC(=O)C1Sc2c(sc(=O)n2c3ccccc3)C4C1OC(=O)c5ccc(Br)cc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L16 compound treatment 600.0 -759.0 -0.27 600.0 -96.3 -0.07 -0.2426 -0.8691 1521472 ChemDiv3_005890 COc1ccc(C(=O)Cc2cc3ccccc3oc2=O)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L17 compound treatment 960.0 -399.0 -0.14 3160.0 2460.0 1.89 1.2374 0.6524 3119763 ChemDiv3_005891 Cc1ccc2oc(cc(=NCCO)c2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L18 compound treatment 720.0 -639.0 -0.23 5280.0 4580.0 3.52 2.3281 0.6602 1172536 ChemDiv3_005892 CCN(CC)C(=S)SCc1ccc(cc1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L19 compound treatment 1920.0 561.0 0.2 480.0 -216.0 -0.17 0.0234 0.0902 3119764 ChemDiv3_005893 OCCN=c1cc(oc2ccc(Cl)cc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L20 compound treatment 1760.0 401.0 0.14 1000.0 304.0 0.23 0.2655 0.972 1775901 ChemDiv3_005894 C(C1COC2(CCCCCCCCCCC2)O1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L21 compound treatment 2840.0 1480.0 0.53 920.0 224.0 0.17 0.493 0.8918 3119765 ChemDiv3_005895 C(Cn1nnc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L22 compound treatment 600.0 -759.0 -0.27 4400.0 3700.0 2.84 1.8203 0.6373 1155501 ChemDiv3_005896 C[N+]1(CC(O)c2ccccc2)CCCCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L23 mock treatment 640.0 -719.0 -0.25 1200.0 504.0 0.39 0.0932 0.2011 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 L24 mock treatment 2200.0 841.0 0.3 640.0 -56.3 -0.04 0.1805 0.5986 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M01 compound treatment 440.0 -919.0 -0.33 2000.0 1300.0 1.0 0.4773 0.4534 3119766 ChemDiv3_005897 COC(=O)c1ccc(C(=O)OC)c(NC(=O)Cn2nc(cc2C)C(F)(F)F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M02 compound treatment 560.0 -799.0 -0.28 440.0 -256.0 -0.2 -0.3395 -0.9841 3119767 ChemDiv3_005898 CCCC1C2CC(C)CC=C2C(=C(N)C1(C#N)C#N)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M03 compound treatment 2080.0 721.0 0.26 360.0 -336.0 -0.26 -0.0016 -0.0044 1202157 ChemDiv3_005899 COC(=O)c1c(NC(=O)C2CCCCC2C(=O)O)scc1c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M04 compound treatment 360.0 -999.0 -0.35 360.0 -336.0 -0.26 -0.4331 -0.9879 3119768 ChemDiv3_005900 COc1ccc(cc1)C(=O)OC(C)CN(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M05 compound treatment 400.0 -959.0 -0.34 4280.0 3580.0 2.75 1.705 0.615 3119904 ChemDiv3_005901 OC(=O)C1C(C2CCC1C2)C(=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M06 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 3026222 ChemDiv3_005902 Cc1cc(NC(=O)CSc2nccc(O)n2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M07 compound treatment 520.0 -839.0 -0.3 320.0 -376.0 -0.29 -0.4146 -0.9999 3119905 ChemDiv3_005903 CCc1nc2ccccc2c3nc(NC(=O)C(F)(F)F)nn13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M08 compound treatment 9280.0 7920.0 2.81 600.0 -96.3 -0.07 1.9347 0.6883 3026223 ChemDiv3_005904 CCOc1ncnc2c3cc4COC(C)(C)Cc4nc3sc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M09 compound treatment 2760.0 1400.0 0.5 360.0 -336.0 -0.26 0.169 0.3016 3119906 ChemDiv3_005905 OC(=O)CCc1ccc(c2ccccc2)n1CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M10 compound treatment 560.0 -799.0 -0.28 600.0 -96.3 -0.07 -0.2526 -0.8627 3119907 ChemDiv3_005906 COc1ccccc1C(CC(=O)NC2CCOC(C)(C)C2)c3ccc(OC(C)C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M11 compound treatment 760.0 -599.0 -0.21 320.0 -376.0 -0.29 -0.3544 -0.9886 1866129 ChemDiv3_005907 CC(=O)Nc1nc(C)cc2c3ccccc3oc(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M12 compound treatment 2680.0 1320.0 0.47 400.0 -296.0 -0.23 0.1706 0.3275 3026224 ChemDiv3_005908 CSc1nnc2nc(O)cc(N)n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M13 compound treatment 1720.0 361.0 0.13 2680.0 1980.0 1.52 1.1675 0.7639 3119908 ChemDiv3_005909 Cc1ccc(cc1)C(=O)C(OC(=O)c2c(C)cc(=O)oc2C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M14 compound treatment 480.0 -879.0 -0.31 2200.0 1500.0 1.15 0.5959 0.4983 3026225 ChemDiv3_005910 CCOC(=O)c1c2-c3ccccc3C(=O)c4c(Cl)ccc([nH]c1=O)c42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M15 compound treatment 440.0 -919.0 -0.33 360.0 -336.0 -0.26 -0.413 -0.9933 1535887 ChemDiv3_005911 Oc1ccc2OC3(CCCC3c2c1)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M16 compound treatment 960.0 -399.0 -0.14 360.0 -336.0 -0.26 -0.2826 -0.9599 3119909 ChemDiv3_005912 CCOC(=O)c1ccc(CC2S/C(=N\c3ccc(CC)cc3)/NC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M17 compound treatment 360.0 -999.0 -0.35 480.0 -216.0 -0.17 -0.3679 -0.9403 3026226 ChemDiv3_005913 COc1ccccc1C(CCNS(=O)(=O)c2ccc(C)cc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M18 compound treatment 3040.0 1680.0 0.6 840.0 144.0 0.11 0.4998 0.824 3119910 ChemDiv3_005914 C(COc1ccccc1)Cn2c3ccccc3c4nc5ccccc5nc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M19 compound treatment 720.0 -639.0 -0.23 1000.0 304.0 0.23 0.0047 0.0144 3119911 ChemDiv3_005915 COc1ccc(NC(c2c[nH]c3ccccc23)P4(=S)OCC(C)(C)CO4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M20 compound treatment 1000.0 -359.0 -0.13 400.0 -296.0 -0.23 -0.2508 -0.9624 1867787 ChemDiv3_005916 O=C1CSC(=O)N1Cc2ccc(CN3C(=O)CSC3=O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M21 compound treatment 960.0 -399.0 -0.14 640.0 -56.3 -0.04 -0.1306 -0.8828 3119912 ChemDiv3_005917 Cc1c2OC(C)(C)C(CO)c2c(C)c(OCc3ccccc3)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M22 compound treatment 920.0 -439.0 -0.16 760.0 63.8 0.05 -0.0755 -0.4624 3026227 ChemDiv3_005918 Fc1ccc2OCN(Cc2c1)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M23 mock treatment 2440.0 1080.0 0.38 720.0 23.8 0.02 0.2841 0.7399 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 M24 mock treatment 880.0 -479.0 -0.17 400.0 -296.0 -0.23 -0.2809 -0.9897 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N01 compound treatment 4240.0 2880.0 1.02 240.0 -456.0 -0.35 0.4751 0.4397 3119913 ChemDiv3_005919 CNC1=NC(=O)CC(S1)C(=O)Nc2ccc3ccccc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N02 compound treatment 360.0 -999.0 -0.35 400.0 -296.0 -0.23 -0.4114 -0.977 3026228 ChemDiv3_005920 O=C1CC(Cc2nc(NC3CC3)ncc12)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N03 compound treatment 240.0 -1120.0 -0.4 360.0 -336.0 -0.26 -0.4632 -0.9783 3119914 ChemDiv3_005921 Brc1ccccc1[C@@H]2Nc3ccccc3[C@@H]4C=CC[C@@H]42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N04 compound treatment 1560.0 201.0 0.07 840.0 144.0 0.11 0.1285 0.9778 3026281 ChemDiv3_005922 COC(=O)c1ccccc1NC(=C2C(=O)c3ccccc3C2=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N05 compound treatment 5360.0 4000.0 1.42 360.0 -336.0 -0.26 0.8212 0.5692 3026282 ChemDiv3_005923 NC(=O)c1c(N)c(C(=S)N)n2CCCc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N06 compound treatment 800.0 -559.0 -0.2 400.0 -296.0 -0.23 -0.301 -0.9977 3026283 ChemDiv3_005924 Cc1ccc(Sc2c(C)c3cc4OCOc4cc3[nH]c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N07 compound treatment 7600.0 6240.0 2.21 1640.0 944.0 0.72 2.0779 0.892 3026284 ChemDiv3_005925 Cc1ccccc1CSc2nnc3c4ccccc4[nH]c3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N08 compound treatment 480.0 -879.0 -0.31 320.0 -376.0 -0.29 -0.4247 -0.9993 3026285 ChemDiv3_005926 CCOc1ccc(/C=C/2\SC(=NC2=O)N3CCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N09 compound treatment 760.0 -599.0 -0.21 280.0 -416.0 -0.32 -0.3762 -0.9803 3026286 ChemDiv3_005927 COC(=O)c1cc(NC(=O)N2c3ccccc3Sc4ccccc24)cc(c1)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N10 compound treatment 1480.0 121.0 0.04 560.0 -136.0 -0.1 -0.0435 -0.3851 3026287 ChemDiv3_005928 COc1cc2CCN3CN(CC(=C3c2cc1OC)C#N)c4ccc(C)c(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N11 compound treatment 720.0 -639.0 -0.23 680.0 -16.3 -0.01 -0.169 -0.7449 3119915 ChemDiv3_005929 Nc1nc(CSc2nnc([nH]2)c3ccccc3)nc(Nc4ccccc4)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N12 compound treatment 920.0 -439.0 -0.16 600.0 -96.3 -0.07 -0.1623 -0.942 3026288 ChemDiv3_005930 O=C(/C=C/c1ccco1)N(Cc2cccs2)C3CCS(=O)(=O)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N13 compound treatment 400.0 -959.0 -0.34 480.0 -216.0 -0.17 -0.3579 -0.9456 3119916 ChemDiv3_005931 COc1ccccc1/C=C/C=c/2\sc3nc(nn3c2=O)c4cc(OC)c(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N14 compound treatment 2840.0 1480.0 0.53 480.0 -216.0 -0.17 0.2542 0.4612 3119917 ChemDiv3_005932 COc1ccc(cc1)C2=NC(=O)/C(=C\c3cc(OC)c(OC)c(OC)c3)/O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N15 compound treatment 440.0 -919.0 -0.33 480.0 -216.0 -0.17 -0.3479 -0.951 3026289 ChemDiv3_005933 OC(=O)C1Sc2[nH]c(=O)sc2C3C1C(=O)Oc4cc(O)ccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N16 compound treatment 400.0 -959.0 -0.34 800.0 104.0 0.08 -0.1842 -0.5272 1496915 ChemDiv3_005934 CCc1ccc(cc1)C(=O)Cc2cc3cccc(OC)c3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N17 compound treatment 920.0 -439.0 -0.16 360.0 -336.0 -0.26 -0.2926 -0.9707 3026290 ChemDiv3_005935 CCCN=c1cc(oc2ccc(C)cc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N18 compound treatment 960.0 -399.0 -0.14 600.0 -96.3 -0.07 -0.1523 -0.9541 3119918 ChemDiv3_005936 CC(C)c1ccc(NCc2nc(no2)c3ccc(Cl)cc3Cl)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N19 compound treatment 280.0 -1080.0 -0.38 360.0 -336.0 -0.26 -0.4531 -0.9816 3026291 ChemDiv3_005937 CC(O)CN=c1cc(oc2ccc(Cl)cc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N20 compound treatment 920.0 -439.0 -0.16 600.0 -96.3 -0.07 -0.1623 -0.942 1639224 ChemDiv3_005938 C[N+]1(CCCCC1)C2CCC3CCC2C3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N21 compound treatment 880.0 -479.0 -0.17 600.0 -96.3 -0.07 -0.1723 -0.9305 3026292 ChemDiv3_005939 Fc1ccc(Cn2nnc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N22 compound treatment 720.0 -639.0 -0.23 1000.0 304.0 0.23 0.0047 0.0144 3119919 ChemDiv3_005940 CC1(C)CCCC2=C1CC3C(C2)C(=O)N(CCC[N+](C)(C)C)C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N23 mock treatment 680.0 -679.0 -0.24 520.0 -176.0 -0.14 -0.2659 -0.9629 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 N24 mock treatment 720.0 -639.0 -0.23 800.0 104.0 0.08 -0.1039 -0.4326 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O01 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3026293 ChemDiv3_005941 Cc1cc(nn1C(=O)c2cccnc2Cl)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O02 compound treatment 240.0 -1120.0 -0.4 280.0 -416.0 -0.32 -0.5066 -0.9942 3119920 ChemDiv3_005942 COc1ccc(cc1OC)c2ccc3c(N)c(sc3n2)C(=O)Nc4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O03 compound treatment 440.0 -919.0 -0.33 320.0 -376.0 -0.29 -0.4347 -0.9982 1881926 ChemDiv3_005943 CC1CCc2c(C(=O)N)c(NC(=O)C3c4ccccc4Oc5ccccc35)sc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O04 compound treatment 280.0 -1080.0 -0.38 400.0 -296.0 -0.23 -0.4314 -0.9691 3026294 ChemDiv3_005944 COc1ccc(cc1)C(=O)OCC[N+]2(C)CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O05 compound treatment 360.0 -999.0 -0.35 320.0 -376.0 -0.29 -0.4548 -0.9949 3119921 ChemDiv3_005945 O=C(NC1CCCc2ccccc12)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O06 compound treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 3026295 ChemDiv3_005946 CCC(Sc1nc(C)cc(=O)[nH]1)C(=O)Nc2ccc(Cl)cn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O07 compound treatment 440.0 -919.0 -0.33 320.0 -376.0 -0.29 -0.4347 -0.9982 3119922 ChemDiv3_005947 Cc1ccc(cc1)c2nnc(NC(=O)c3cc4c5ccccc5[nH]c4c(C)n3)s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O08 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 1570877 ChemDiv3_005948 Oc1ccc(cc1)N2Cc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O09 compound treatment 360.0 -999.0 -0.35 360.0 -336.0 -0.26 -0.4331 -0.9879 3119923 ChemDiv3_005949 COC(=O)c1cccc(c1)n2c(CCC(=O)O)ccc2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O10 compound treatment 360.0 -999.0 -0.35 240.0 -456.0 -0.35 -0.4982 -1.0 3026296 ChemDiv3_005950 OC(=O)CCSc1nnc2sc3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O11 compound treatment 280.0 -1080.0 -0.38 240.0 -456.0 -0.35 -0.5183 -0.999 3119924 ChemDiv3_005951 CC(C)NS(=O)(=O)c1ccc(OCC(=O)N2CCC(Cc3ccccc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O12 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 3026297 ChemDiv3_005952 COc1cc2CCN(C(c3ccccc3)c2cc1OC)C(=O)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O13 compound treatment 320.0 -1040.0 -0.37 440.0 -256.0 -0.2 -0.3997 -0.9568 3119925 ChemDiv3_005953 Cn1c(=O)n(C)c2cc(CN)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O14 compound treatment 360.0 -999.0 -0.35 320.0 -376.0 -0.29 -0.4548 -0.9949 1875868 ChemDiv3_005954 COC(=O)c1c2C(=O)c3ccccc3C(=O)c2n4ccc(C)cc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O15 compound treatment 320.0 -1040.0 -0.37 240.0 -456.0 -0.35 -0.5082 -0.9997 3119926 ChemDiv3_005955 CCOC(=O)C1=CC2C(OC1=O)C=Cc3cc(Br)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O16 compound treatment 280.0 -1080.0 -0.38 360.0 -336.0 -0.26 -0.4531 -0.9816 3119927 ChemDiv3_005956 CCC1(C)Cc2ccccc2-c3c1c(=O)n(c4ccc(C)cc4)c5nncn35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O17 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 1224060 ChemDiv3_005957 CN(C)c1ccc(CN(CCC(c2ccco2)c3ccccc3)C(=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O18 compound treatment 360.0 -999.0 -0.35 320.0 -376.0 -0.29 -0.4548 -0.9949 1699767 ChemDiv3_005958 Cc1ccc(cc1)N(CC(=O)N)C2SC(=O)N(C2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O19 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 3026298 ChemDiv3_005959 COc1ccc(NC(=O)OC(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O20 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 1867846 ChemDiv3_005960 OC(=O)CCN1C(=O)SC(Nc2ccccc2)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O21 compound treatment 320.0 -1040.0 -0.37 320.0 -376.0 -0.29 -0.4648 -0.9927 3026299 ChemDiv3_005961 N=C1NC(=O)C(CC(=O)Nc2ccccc2)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O22 compound treatment 280.0 -1080.0 -0.38 360.0 -336.0 -0.26 -0.4531 -0.9816 1514101 ChemDiv3_005962 O=C1NC(C2=C(N1)c3ccccc3CC2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O23 mock treatment 200.0 -1160.0 -0.41 320.0 -376.0 -0.29 -0.4949 -0.9851 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 O24 mock treatment 320.0 -1040.0 -0.37 280.0 -416.0 -0.32 -0.4865 -0.9975 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P01 compound treatment 280.0 -1080.0 -0.38 280.0 -416.0 -0.32 -0.4966 -0.996 3120069 ChemDiv3_005963 COc1ccc(CNC(=O)C2CC(=O)N=C(N)S2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P02 compound treatment 320.0 -1040.0 -0.37 360.0 -336.0 -0.26 -0.4431 -0.9848 3026300 ChemDiv3_005964 COc1ccc(cc1)C2CC(=O)c3cnc(NCCc4ccccc4)nc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P03 compound treatment 240.0 -1120.0 -0.4 480.0 -216.0 -0.17 -0.398 -0.9252 3120070 ChemDiv3_005965 C1SCC1Oc2cccc(c2)[C@@H]3Nc4ccccc4[C@@H]5C=CC[C@@H]53 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P04 compound treatment 240.0 -1120.0 -0.4 360.0 -336.0 -0.26 -0.4632 -0.9783 3120071 ChemDiv3_005966 COc1cc(OC)nc(NC2OC(=O)c3ccccc23)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P05 compound treatment 440.0 -919.0 -0.33 480.0 -216.0 -0.17 -0.3479 -0.951 1615557 ChemDiv3_005967 Oc1cc(nc(Nc2nc3ccccc3o2)n1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P06 compound treatment 1960.0 601.0 0.21 280.0 -416.0 -0.32 -0.0751 -0.1956 3120072 ChemDiv3_005968 CCn1c(SCc2nc3ccccc3[nH]2)nc4cc(ccc4c1=O)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P07 compound treatment 2240.0 881.0 0.31 240.0 -456.0 -0.35 -0.0266 -0.0567 1279174 ChemDiv3_005969 O=C(CSc1nc2ccccc2o1)Nc3ccc(Oc4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P08 compound treatment 520.0 -839.0 -0.3 320.0 -376.0 -0.29 -0.4146 -0.9999 3120073 ChemDiv3_005970 CN(C)c1ccc(cc1)C(=S)N2CCN(CC2)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P09 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 3026301 ChemDiv3_005971 Cc1nc(SC(C(=O)c2ccccc2)c3ccccc3)nc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P10 compound treatment 2520.0 1160.0 0.41 240.0 -456.0 -0.35 0.0436 0.0807 3120074 ChemDiv3_005972 COc1cc2CCN3CN(CCc4ccccc4)CC(=C3c2cc1OC)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P11 compound treatment 2360.0 1000.0 0.36 280.0 -416.0 -0.32 0.0252 0.0527 3120075 ChemDiv3_005973 COC(=O)Cc1cc(=O)nc(/N=C(\N)/Nc2ccccc2)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P12 compound treatment 1880.0 521.0 0.18 280.0 -416.0 -0.32 -0.0952 -0.2579 3026302 ChemDiv3_005974 Cc1ccc(cc1CNC(=O)Nc2ccccc2)c3nn(C)c(=O)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P13 compound treatment 1600.0 241.0 0.09 1840.0 1140.0 0.88 0.6814 0.7724 3120076 ChemDiv3_005975 Cc1cccc(c1)c2nc3s/c(=C\C4=Cc5ccccc5OC4)/c(=O)n3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P14 compound treatment 520.0 -839.0 -0.3 320.0 -376.0 -0.29 -0.4146 -0.9999 3026303 ChemDiv3_005976 COc1ccc(cc1)C2=NC(=O)/C(=C\c3cccc(F)c3)/O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P15 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 3120077 ChemDiv3_005977 OC(=O)CC1S/C(=N/c2cccc(c2)C(F)(F)F)/NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P16 compound treatment 240.0 -1120.0 -0.4 640.0 -56.3 -0.04 -0.3112 -0.7794 1557885 ChemDiv3_005978 Brc1ccc(Cn2c(nc3ccccc23)S(=O)(=O)Cc4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P17 compound treatment 360.0 -999.0 -0.35 280.0 -416.0 -0.32 -0.4765 -0.9987 3120078 ChemDiv3_005979 Clc1ccc2oc(cc(=NCc3cccnc3)c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P18 compound treatment 280.0 -1080.0 -0.38 400.0 -296.0 -0.23 -0.4314 -0.9691 3120079 ChemDiv3_005980 COc1ccccc1N2C(=O)CCC2(C#N)c3ccc(OCc4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P19 compound treatment 2200.0 841.0 0.3 280.0 -416.0 -0.32 -0.0149 -0.0342 3026304 ChemDiv3_005981 Oc1ccc(/N=c/2\cc(oc3ccc(Cl)cc23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P20 compound treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 3120080 ChemDiv3_005982 CC1=NNC(C1)c2ccc(O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P21 compound treatment 360.0 -999.0 -0.35 200.0 -496.0 -0.38 -0.5199 -0.9993 3120081 ChemDiv3_005983 CCOC(=O)c1c(NC(=O)Cn2nnc3sc4CC(C)CCc4c3c2=O)sc5CCCCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P22 compound treatment 320.0 -1040.0 -0.37 200.0 -496.0 -0.38 -0.53 -0.9999 1635015 ChemDiv3_005984 COC(=O)c1ccc(C[N+]2(C)CCCCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P23 mock treatment 240.0 -1120.0 -0.4 320.0 -376.0 -0.29 -0.4849 -0.9878 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2017 P24 mock treatment 360.0 -999.0 -0.35 240.0 -456.0 -0.35 -0.4982 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A01 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 3026305 ChemDiv3_005985 CC1C=C(C)CC2C1C(=O)N(C2=O)c3ccc[n+](C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A02 compound treatment 280.0 -818.0 -0.29 720.0 -114.0 -0.09 -0.267 -0.8813 1470316 ChemDiv3_005986 CC1Cc2ccccc2N1C(=O)c3ccc(COc4ccc(C)c(C)c4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A03 compound treatment 240.0 -858.0 -0.3 440.0 -394.0 -0.3 -0.429 -1.0 3120082 ChemDiv3_005987 CC1CC(C)(C)OC(C[N+]2(C)CCCCC2)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A04 compound treatment 600.0 -498.0 -0.18 480.0 -354.0 -0.27 -0.317 -0.9781 3026306 ChemDiv3_005988 CN(C)c1ccc2sc(S)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A05 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3026307 ChemDiv3_005989 NNc1nc(cc(n1)C(F)(F)F)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A06 compound treatment 280.0 -818.0 -0.29 240.0 -594.0 -0.46 -0.5276 -0.9761 3120083 ChemDiv3_005990 OC(=O)c1ccc(N/C=C/C(=O)c2ccco2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A07 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3120084 ChemDiv3_005991 Nn1c(CCCc2nc3ccccc3c(=O)n2N)nc4ccccc4c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A08 compound treatment 840.0 -258.0 -0.09 320.0 -514.0 -0.39 -0.3437 -0.8483 3026308 ChemDiv3_005992 CC1CCC/C(=C\Nc2ccc(cc2C)C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A09 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 1620261 ChemDiv3_005993 COc1ccc(NC(=O)c2ccc(COc3ccc(cc3)C(C)C)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A10 compound treatment 360.0 -738.0 -0.26 240.0 -594.0 -0.46 -0.5075 -0.9652 3026309 ChemDiv3_005994 O=C(Nc1nncs1)C2CC(=O)OC2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A11 compound treatment 520.0 -578.0 -0.2 160.0 -674.0 -0.52 -0.5108 -0.9177 1567947 ChemDiv3_005995 Brc1cnn(Cc2ccc(o2)C(=O)NCc3ccccn3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A12 compound treatment 320.0 -778.0 -0.28 360.0 -474.0 -0.36 -0.4524 -0.9906 3026310 ChemDiv3_005996 Cc1cc(C)c2c(cc(O)nc2c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A13 compound treatment 480.0 -618.0 -0.22 320.0 -514.0 -0.39 -0.434 -0.9614 1123919 ChemDiv3_005997 COC(=O)c1ccc(COc2ccccc2OC)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A14 compound treatment 280.0 -818.0 -0.29 1200.0 366.0 0.28 -0.0064 -0.0159 3120085 ChemDiv3_005998 CC1(C)CC(=C(C(=O)C1)C(NC(=O)c2ccccc2)(C(F)(F)F)C(F)(F)F)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A15 compound treatment 280.0 -818.0 -0.29 520.0 -314.0 -0.24 -0.3756 -0.9958 1560602 ChemDiv3_005999 Cc1cccc2sc(NC(=O)c3ccc(COc4ccc5ccccc5c4)o3)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A16 compound treatment 280.0 -818.0 -0.29 1040.0 206.0 0.16 -0.0933 -0.2824 1019709 ChemDiv3_006000 C[N+]1(C)C2CCC1CC(C2)OC(=O)C(CO)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A17 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 1517127 ChemDiv3_006001 OC(=O)c1ccc(Cn2cccn2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A18 compound treatment 440.0 -658.0 -0.23 280.0 -554.0 -0.43 -0.4657 -0.96 3026361 ChemDiv3_006002 O=C1N(NS(=O)(=O)c2ccccc2)C(Nc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A19 compound treatment 400.0 -698.0 -0.25 400.0 -434.0 -0.33 -0.4106 -0.9893 3026362 ChemDiv3_006003 CC(C)c1ccc(OCc2ccc(cc2)C(=O)NCc3ccco3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A20 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3026363 ChemDiv3_006004 CSCCC(N1C(=O)/C(=C/c2cccnc2)/SC1=S)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A21 compound treatment 320.0 -778.0 -0.28 1920.0 1090.0 0.83 0.3945 0.4492 1636669 ChemDiv3_006005 Cc1ccc(OCc2ccc(o2)C(=O)Nc3nccs3)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A22 compound treatment 400.0 -698.0 -0.25 280.0 -554.0 -0.43 -0.4757 -0.9668 3026364 ChemDiv3_006006 Cc1nc(N)[nH]c(=O)c1CC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A23 mock treatment 360.0 -738.0 -0.26 840.0 5.93 0.0 -0.1818 -0.6947 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 A24 mock treatment 320.0 -778.0 -0.28 360.0 -474.0 -0.36 -0.4524 -0.9906 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B01 compound treatment 280.0 -818.0 -0.29 720.0 -114.0 -0.09 -0.267 -0.8813 3026365 ChemDiv3_006007 CC(C)(C)c1nc(c(NCc2ccccc2)o1)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B02 compound treatment 360.0 -738.0 -0.26 880.0 45.9 0.04 -0.1601 -0.6063 1058723 ChemDiv3_006008 COc1ccc(NCc2ccccc2O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B03 compound treatment 240.0 -858.0 -0.3 640.0 -194.0 -0.15 -0.3205 -0.9461 3120086 ChemDiv3_006009 Cc1cc(C)c(N(CC(O)Cn2c3ccccc3c4ccccc24)S(=O)(=O)C)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B04 compound treatment 400.0 -698.0 -0.25 280.0 -554.0 -0.43 -0.4757 -0.9668 3026366 ChemDiv3_006010 C=CCSc1n[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B05 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3026367 ChemDiv3_006011 NC(=O)C1CCCN(C1)C(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B06 compound treatment 320.0 -778.0 -0.28 400.0 -434.0 -0.33 -0.4307 -0.9956 3120087 ChemDiv3_006012 Cc1cccc(c1)N/2C3CS(=O)(=O)CC3S\C2=N\C(=O)c4ccc(Br)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B07 compound treatment 280.0 -818.0 -0.29 240.0 -594.0 -0.46 -0.5276 -0.9761 3026368 ChemDiv3_006013 COc1ccc(/C=C/C(=O)NCCNC2=NS(=O)(=O)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B08 compound treatment 240.0 -858.0 -0.3 480.0 -354.0 -0.27 -0.4073 -0.9984 3120088 ChemDiv3_006014 COc1ccc(cc1OC)S(=O)(=O)N2Cc3ccccc3CC2C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B09 compound treatment 480.0 -618.0 -0.22 4600.0 3770.0 2.89 1.8895 0.6517 3117797 ChemDiv3_006015 CCc1ccc(cc1)C2CC(c3ccccc3)n4ncnc4N2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B10 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3026369 ChemDiv3_006016 Cn1nnnc1SCC(=O)NCc2cccc(c2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B11 compound treatment 920.0 -178.0 -0.06 320.0 -514.0 -0.39 -0.3236 -0.8097 3117798 ChemDiv3_006017 COc1ccc(cc1OC)c2cn3c(n2)n(N)c4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B12 compound treatment 280.0 -818.0 -0.29 800.0 -34.1 -0.03 -0.2236 -0.7678 3026370 ChemDiv3_006018 COc1ccccc1CNc2ccc(O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B13 compound treatment 520.0 -578.0 -0.2 480.0 -354.0 -0.27 -0.3371 -0.9903 3117799 ChemDiv3_006019 Clc1ccc2[nH]c(=O)c(CN3CCCCC3)c(c4ccccc4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B14 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 3026371 ChemDiv3_006020 COc1cccc(CNC(C)c2ccccc2)c1OCc3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B15 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3117800 ChemDiv3_006021 CC1CCCN(CCC(=O)c2ccc(Br)cc2)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B16 compound treatment 240.0 -858.0 -0.3 440.0 -394.0 -0.3 -0.429 -1.0 3117801 ChemDiv3_006022 CCOc1ccc(cc1)c2nc(C#N)c(NCC(C)C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B17 compound treatment 480.0 -618.0 -0.22 320.0 -514.0 -0.39 -0.434 -0.9614 3026372 ChemDiv3_006023 CCOC(=O)c1sc(Nc2ccc(C)cc2C)nc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B18 compound treatment 280.0 -818.0 -0.29 240.0 -594.0 -0.46 -0.5276 -0.9761 3117802 ChemDiv3_006024 COc1ccc(CC(=O)Nc2ccc(cc2)c3nnc(S)s3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B19 compound treatment 400.0 -698.0 -0.25 360.0 -474.0 -0.36 -0.4323 -0.9823 3026373 ChemDiv3_006025 Cc1[nH]c2ccccc2c1C(=O)CSC(=S)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B20 compound treatment 360.0 -738.0 -0.26 3680.0 2850.0 2.18 1.3599 0.618 3117803 ChemDiv3_006026 Cc1ccc(cc1)C2=NNC(S2)c3cccc(C)n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B21 compound treatment 320.0 -778.0 -0.28 3640.0 2810.0 2.15 1.3282 0.6116 3117804 ChemDiv3_006027 Cc1ccc(cc1)C(=O)/C=c/2\[nH]c(=O)\c(=C\c3cccnc3)\s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B22 compound treatment 280.0 -818.0 -0.29 5320.0 4490.0 3.44 2.2302 0.6453 3026374 ChemDiv3_006028 COC(=O)c1c(NC(=O)CN2C(=O)c3cccc4cccc2c34)sc5CCCCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B23 mock treatment 840.0 -258.0 -0.09 440.0 -394.0 -0.3 -0.2785 -0.8813 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 B24 mock treatment 240.0 -858.0 -0.3 280.0 -554.0 -0.43 -0.5159 -0.9865 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C01 compound treatment 360.0 -738.0 -0.26 320.0 -514.0 -0.39 -0.4641 -0.9801 3117805 ChemDiv3_006029 C[N+]1(CCCC1)C2CCC3CCC2C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C02 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 1645761 ChemDiv3_006030 CN(C)S(=O)(=O)c1ccc(CCNC(=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C03 compound treatment 200.0 -898.0 -0.32 4600.0 3770.0 2.89 1.8192 0.6255 3117806 ChemDiv3_006031 C1OC(OCC12COC(OC2)c3ccncc3)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C04 compound treatment 400.0 -698.0 -0.25 400.0 -434.0 -0.33 -0.4106 -0.9893 1262889 ChemDiv3_006032 CC1CCC2(CC1)Nc3ccccc3C(=O)N2CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C05 compound treatment 240.0 -858.0 -0.3 440.0 -394.0 -0.3 -0.429 -1.0 3026375 ChemDiv3_006033 COc1nc(cc(n1)C(F)(F)F)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C06 compound treatment 360.0 -738.0 -0.26 240.0 -594.0 -0.46 -0.5075 -0.9652 3117807 ChemDiv3_006034 COc1ccccc1Oc2ccc(N/C=C/C(=O)c3ccco3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C07 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3026376 ChemDiv3_006035 Cc1nn(CC(=O)O)c(C)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C08 compound treatment 1320.0 223.0 0.08 480.0 -354.0 -0.27 -0.1364 -0.4819 3117808 ChemDiv3_006036 CN(C)c1ccc(/C=[N+]/2\[N-]C(=O)C(NC(=O)c3ccc(F)cc3)C2c4ccc(C)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C09 compound treatment 2440.0 1340.0 0.48 560.0 -274.0 -0.21 0.188 0.361 3026377 ChemDiv3_006037 CC1Cc2ccc(F)cc2CN1C(=O)c3ccc(COc4ccccc4Br)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C10 compound treatment 2240.0 1140.0 0.41 3200.0 2370.0 1.82 1.571 0.8441 3117809 ChemDiv3_006038 COc1ccc(C)cc1NC(=S)NC2(CN3CN4CN(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C11 compound treatment 3920.0 2820.0 1.0 240.0 -594.0 -0.46 0.3855 0.3504 1539793 ChemDiv3_006039 Brc1cnn(Cc2ccc(o2)C(=O)Nc3sc4CCCCCc4c3C#N)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C12 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3117810 ChemDiv3_006040 COc1ccc2c(cc(O)nc2c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C13 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 1482452 ChemDiv3_006041 COC(=O)c1ccc(COc2ccc3ccccc3c2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C14 compound treatment 280.0 -818.0 -0.29 360.0 -474.0 -0.36 -0.4624 -0.9937 3117811 ChemDiv3_006042 COc1ccc(cc1)C(=O)NC(c2c(C)[nH]n(c3ccccc3)c2=O)(C(F)(F)F)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C15 compound treatment 2080.0 983.0 0.35 320.0 -514.0 -0.39 -0.0326 -0.0619 1692576 ChemDiv3_006043 O=C(N1CCCCC1)c2ccc(COc3cccc4ccccc34)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C16 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 3117812 ChemDiv3_006044 Cn1c(=O)n(C)c2nc(SCC(=O)Nc3ccccc3F)n(Cc4ccccc4)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C17 compound treatment 400.0 -698.0 -0.25 320.0 -514.0 -0.39 -0.454 -0.9747 3117813 ChemDiv3_006045 O=C(OCCN1CCCCC1)c2cccc(COc3ccc4ccccc4c3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C18 compound treatment 320.0 -778.0 -0.28 2280.0 1450.0 1.11 0.5899 0.5157 3026378 ChemDiv3_006046 CC1(C)Nc2ccccc2C(=O)N1NS(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C19 compound treatment 320.0 -778.0 -0.28 360.0 -474.0 -0.36 -0.4524 -0.9906 3117814 ChemDiv3_006047 Cc1ccc(Cl)cc1NC(=O)c2ccc(Cn3cc(Cl)cn3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C20 compound treatment 320.0 -778.0 -0.28 360.0 -474.0 -0.36 -0.4524 -0.9906 3026379 ChemDiv3_006048 OC(=O)CC(N1C(=O)/C(=C\c2c[nH]c3ccccc23)/SC1=S)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C21 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3117815 ChemDiv3_006049 CC(C)OC(=O)c1ccc(NC(=O)c2ccc(Cn3cc(Cl)cn3)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C22 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 3117816 ChemDiv3_006050 CC(C)COC(=O)C1C2OC3(CN(Cc4cccs4)C(=O)C13)C=C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C23 mock treatment 2440.0 1340.0 0.48 320.0 -514.0 -0.39 0.0577 0.0933 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 C24 mock treatment 3800.0 2700.0 0.96 200.0 -634.0 -0.49 0.3337 0.3104 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D01 compound treatment 320.0 -778.0 -0.28 1200.0 366.0 0.28 0.0036 0.0092 3026380 ChemDiv3_006051 CCOc1ccc2nc(sc2c1)c3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D02 compound treatment 320.0 -778.0 -0.28 480.0 -354.0 -0.27 -0.3872 -1.0 3026381 ChemDiv3_006052 Cc1ccccc1NCc2ccccc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D03 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 1362120 ChemDiv3_006053 Cc1cccc(OCC(=O)NS(=O)(=O)c2ccc(Cl)cc2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D04 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3117817 ChemDiv3_006054 O=C1N(C(c2c1oc3ccccc3c2=O)c4ccccc4)c5nccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D05 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 1533324 ChemDiv3_006055 CC(=C)c1cccc(c1)C(C)(C)NC(=O)N2CCCC(C2)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D06 compound treatment 240.0 -858.0 -0.3 240.0 -594.0 -0.46 -0.5376 -0.9806 3117818 ChemDiv3_006056 COc1ccc2c3c4c(=O)n(C)c(=O)n(C)c4cn3ccc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D07 compound treatment 400.0 -698.0 -0.25 360.0 -474.0 -0.36 -0.4323 -0.9823 3026382 ChemDiv3_006057 Cc1cccc(NC(=O)Cn2c(=O)oc3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D08 compound treatment 2280.0 1180.0 0.42 440.0 -394.0 -0.3 0.0827 0.1599 3117819 ChemDiv3_006058 CC(C)CC(NS(=O)(=O)c1cccs1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D09 compound treatment 2240.0 1140.0 0.41 320.0 -514.0 -0.39 0.0075 0.0133 3117820 ChemDiv3_006059 Cc1ccc(cc1)C2CC(c3c(F)cccc3Cl)n4nc(N)nc4N2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D10 compound treatment 440.0 -658.0 -0.23 520.0 -314.0 -0.24 -0.3354 -0.9999 3026383 ChemDiv3_006060 FC(F)(F)c1cccc(NC(=O)Cn2cnc(SCc3ccccc3)n2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D11 compound treatment 440.0 -658.0 -0.23 360.0 -474.0 -0.36 -0.4223 -0.9769 3117821 ChemDiv3_006061 O=C(Nc1ccc2[nH]c(nc2c1)c3ccccn3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D12 compound treatment 400.0 -698.0 -0.25 280.0 -554.0 -0.43 -0.4757 -0.9668 3026384 ChemDiv3_006062 CCOc1ccc(CNc2ccc(O)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D13 compound treatment 240.0 -858.0 -0.3 240.0 -594.0 -0.46 -0.5376 -0.9806 1136263 ChemDiv3_006063 Fc1ccc(cc1)S(=O)(=O)N2CCc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D14 compound treatment 360.0 -738.0 -0.26 320.0 -514.0 -0.39 -0.4641 -0.9801 3117822 ChemDiv3_006064 CC(C)(C)NC(=O)COc1ccc(CNC2C3CC4CC(C3)CC2C4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D15 compound treatment 360.0 -738.0 -0.26 480.0 -354.0 -0.27 -0.3772 -0.9998 3026385 ChemDiv3_006065 CC1CCCC(C)N1C(=O)c2ccc(NC(=O)C(O)(c3ccccc3)c4ccccc4)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D16 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3117952 ChemDiv3_006066 CCOc1ccc(cc1)c2nc(C#N)c(NCCCN(CC)CC)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D17 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3026386 ChemDiv3_006067 FC(F)(F)c1cc(nc(NC(=N)Nc2cccc(Cl)c2)n1)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D18 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3117953 ChemDiv3_006068 CCCCc1c(C)nc(SCc2ccccc2)nc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D19 compound treatment 480.0 -618.0 -0.22 360.0 -474.0 -0.36 -0.4123 -0.9705 1283248 ChemDiv3_006069 Cc1[nH]c2ccccc2c1C(=O)CSc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D20 compound treatment 360.0 -738.0 -0.26 360.0 -474.0 -0.36 -0.4424 -0.9869 3117954 ChemDiv3_006070 Cc1ccc(NS(=O)(=O)c2ccc(NC(=O)CN3C(=O)c4cccc5cccc3c45)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D21 compound treatment 240.0 -858.0 -0.3 360.0 -474.0 -0.36 -0.4725 -0.996 3026387 ChemDiv3_006071 O=C(Cn1cc(/C=N/n2cnnc2)c3ccccc13)Nc4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D22 compound treatment 280.0 -818.0 -0.29 5040.0 4210.0 3.23 2.0782 0.641 3117955 ChemDiv3_006072 Clc1cccc(c1)N2CCN(CC2)C(=O)CN3C(=O)c4ccccc4S3(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D23 mock treatment 240.0 -858.0 -0.3 360.0 -474.0 -0.36 -0.4725 -0.996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 D24 mock treatment 520.0 -578.0 -0.2 320.0 -514.0 -0.39 -0.4239 -0.9534 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E01 compound treatment 520.0 -578.0 -0.2 1520.0 686.0 0.53 0.2275 0.4026 1119813 ChemDiv3_006073 OC(=O)C1C(C2CC1C=C2)C(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E02 compound treatment 720.0 -378.0 -0.13 4960.0 4130.0 3.17 2.1451 0.6766 3117956 ChemDiv3_006074 Sc1nnc(Cn2cnc3ccccc23)n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E03 compound treatment 600.0 -498.0 -0.18 640.0 -194.0 -0.15 -0.2301 -0.9965 3026388 ChemDiv3_006075 CCN(CC)CC(=O)OCC1C(C)CC(=CC1C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E04 compound treatment 1920.0 823.0 0.29 1200.0 366.0 0.28 0.405 0.9998 3117957 ChemDiv3_006076 Nc1nc2CCCCc2c(c1C#N)c3ccncc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E05 compound treatment 560.0 -538.0 -0.19 720.0 -114.0 -0.09 -0.1968 -0.9377 3117958 ChemDiv3_006077 FC(F)(F)c1cc(C2CC2)n(CCC(=O)NCCC3=CCCCC3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E06 compound treatment 840.0 -258.0 -0.09 480.0 -354.0 -0.27 -0.2568 -0.8955 3026389 ChemDiv3_006078 Cc1ccc(O)c(N/C=C\2/CCCC2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E07 compound treatment 600.0 -498.0 -0.18 480.0 -354.0 -0.27 -0.317 -0.9781 3026390 ChemDiv3_006079 CCOC(=O)Cn1nc(c(Br)c1C2CC2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E08 compound treatment 1000.0 -97.5 -0.03 1840.0 1010.0 0.77 0.5216 0.6748 3117959 ChemDiv3_006080 COc1ccc(cc1)c2ccc(CCC(=O)O)n2Cc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E09 compound treatment 2360.0 1260.0 0.45 880.0 45.9 0.04 0.3416 0.7604 3117960 ChemDiv3_006081 Nn1c(CSc2ccccn2)nc3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E10 compound treatment 440.0 -658.0 -0.23 440.0 -394.0 -0.3 -0.3789 -0.9917 3117961 ChemDiv3_006082 NC(=O)Nc1nc2ccccc2[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E11 compound treatment 3840.0 2740.0 0.97 280.0 -554.0 -0.43 0.3872 0.3646 3026510 ChemDiv3_006083 FC(F)(F)c1ccc(NC(=O)c2ccc(Cn3cc(Br)cn3)o2)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E12 compound treatment 440.0 -658.0 -0.23 480.0 -354.0 -0.27 -0.3571 -0.9971 3117962 ChemDiv3_006084 CN1C=C/C(=C\c2cc[n+](C)c3ccccc23)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E13 compound treatment 560.0 -538.0 -0.19 640.0 -194.0 -0.15 -0.2402 -0.9926 3026511 ChemDiv3_006085 COC(=O)c1ccc(COc2cc(C)cc(C)c2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E14 compound treatment 1680.0 583.0 0.21 3200.0 2370.0 1.82 1.4305 0.7825 1191701 ChemDiv3_006086 O=C1N(CN2CCCCCC2)c3ccccc3C41OCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E15 compound treatment 800.0 -298.0 -0.11 1040.0 206.0 0.16 0.0372 0.1955 1130164 ChemDiv3_006087 COC(=O)c1ccc(COc2cccc(Cl)c2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E16 compound treatment 800.0 -298.0 -0.11 2600.0 1770.0 1.36 0.884 0.6501 3117963 ChemDiv3_006088 COC(=O)c1cccc(Oc2nc(Nc3ccccc3F)nc(n2)N4CCC5C=CC=CC5C4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E17 compound treatment 800.0 -298.0 -0.11 7480.0 6650.0 5.1 3.5332 0.6923 3026512 ChemDiv3_006089 FC(F)(F)COCc1ccc(cc1)C(=O)Nc2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E18 compound treatment 960.0 -138.0 -0.05 1200.0 366.0 0.28 0.1642 0.5757 3117964 ChemDiv3_006090 CC(=O)NN1C(Nc2ccccc2C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E19 compound treatment 1840.0 743.0 0.26 1200.0 366.0 0.28 0.3849 0.9995 3117965 ChemDiv3_006091 CC(C)c1ccc(C)cc1OCc2ccc(o2)C(=O)Nc3ccccc3C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E20 compound treatment 640.0 -458.0 -0.16 1160.0 326.0 0.25 0.0622 0.2085 3026513 ChemDiv3_006092 CCC1(C)CC2=C(CO1)Cc3c(N2)nc(SCC(=C)C)n(c4ccccc4)c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E21 compound treatment 1200.0 103.0 0.04 4400.0 3570.0 2.74 1.9615 0.7164 1473483 ChemDiv3_006093 Brc1ccccc1OCc2ccc(cc2)C(=O)N3CCc4ccccc4C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E22 compound treatment 1080.0 -17.5 -0.01 1600.0 766.0 0.59 0.4114 0.6996 3117966 ChemDiv3_006094 CCc1ccc(cc1)N2CC3(OC4C=C3)C(C4C(=O)OC)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E23 mock treatment 880.0 -218.0 -0.08 480.0 -354.0 -0.27 -0.2468 -0.8733 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 E24 mock treatment 6760.0 5660.0 2.01 520.0 -314.0 -0.24 1.2499 0.6178 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F01 compound treatment 4240.0 3140.0 1.11 920.0 85.9 0.07 0.8349 0.7476 3026514 ChemDiv3_006095 COc1cc(cc(OC)c1OC)c2nc3ccccc3n2CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F02 compound treatment 840.0 -258.0 -0.09 4480.0 3650.0 2.8 1.9146 0.6837 3026515 ChemDiv3_006096 Cc1cccc(NCc2ccccc2O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F03 compound treatment 1520.0 423.0 0.15 1320.0 486.0 0.37 0.3698 0.9197 3117967 ChemDiv3_006097 CCc1ccc(cc1)N2C(=O)CN(CC(=O)OC)C2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F04 compound treatment 2360.0 1260.0 0.45 1640.0 806.0 0.62 0.7542 0.9874 3117968 ChemDiv3_006098 O=c1c(/C=C(\C#N)/S(=O)(=O)c2ccccc2)c(Oc3ccccc3)nc4ccccn14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F05 compound treatment 2400.0 1300.0 0.46 1600.0 766.0 0.59 0.7425 0.9929 3026516 ChemDiv3_006099 CC1CCN(CC1)C(=O)NC(C)(C)c2cccc(c2)C(=C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F06 compound treatment 800.0 -298.0 -0.11 1040.0 206.0 0.16 0.0372 0.1955 1004614 ChemDiv3_006100 OC(=O)CNS(=O)(=O)c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F07 compound treatment 1000.0 -97.5 -0.03 1280.0 446.0 0.34 0.2176 0.6324 3117969 ChemDiv3_006101 Cc1cccc(c1)c2noc(COc3ccccc3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F08 compound treatment 800.0 -298.0 -0.11 1000.0 166.0 0.13 0.0154 0.0934 3026517 ChemDiv3_006102 C(Sc1nc2ccccc2[nH]1)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F09 compound treatment 7040.0 5940.0 2.11 6200.0 5370.0 4.12 4.4036 0.9516 3117970 ChemDiv3_006103 Cc1ccc(cc1)C2CC(c3ccccc3C)n4nc(N)nc4N2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F10 compound treatment 800.0 -298.0 -0.11 960.0 126.0 0.1 -0.0063 -0.0438 3026518 ChemDiv3_006104 Cc1cc(C)c(Cn2c(nc3ccccc23)S(=O)(=O)Cc4ccccc4)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F11 compound treatment 1440.0 343.0 0.12 2240.0 1410.0 1.08 0.8491 0.7818 3117971 ChemDiv3_006105 COC(=O)c1ccc(cc1)C(=O)Nc2ccc3[nH]c(nc3c2)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F12 compound treatment 1040.0 -57.5 -0.02 2280.0 1450.0 1.11 0.7705 0.694 3026519 ChemDiv3_006106 CC(C)(CO)NCc1cccs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F13 compound treatment 1000.0 -97.5 -0.03 1240.0 406.0 0.31 0.1959 0.6248 3117972 ChemDiv3_006107 Cc1ccc2NC(CC(N3CCCC3=O)c2c1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F14 compound treatment 680.0 -418.0 -0.15 920.0 85.9 0.07 -0.0581 -0.3582 3026520 ChemDiv3_006108 COc1cc(CNC(C)(C)C)ccc1OCC(=O)NC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F15 compound treatment 600.0 -498.0 -0.18 7560.0 6730.0 5.16 3.5264 0.6825 3117973 ChemDiv3_006109 COC(=O)[C@@]1(C)CCCC2(C)C1CCc3cc(ccc32)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F16 compound treatment 2040.0 943.0 0.33 2760.0 1930.0 1.48 1.2819 0.8457 3026553 ChemDiv3_006110 CCOc1ccc(cc1)c2nc(C#N)c(o2)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F17 compound treatment 1120.0 22.5 0.01 1040.0 206.0 0.16 0.1174 0.7419 3117974 ChemDiv3_006111 N=C(NCCc1c[nH]c2ccccc12)NC(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F18 compound treatment 680.0 -418.0 -0.15 2760.0 1930.0 1.48 0.9408 0.6331 3117975 ChemDiv3_006112 Cc1ccc(Cl)cc1N2CCN(CC2)C(=O)c3ccccc3N(Cc4ccccc4)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F19 compound treatment 2840.0 1740.0 0.62 2160.0 1330.0 1.02 1.1569 0.9714 3026554 ChemDiv3_006113 COc1ccc(/C=C/C(=O)N2C(OCc3ccccc23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F20 compound treatment 2800.0 1700.0 0.6 4200.0 3370.0 2.58 2.2543 0.8495 3117976 ChemDiv3_006114 CCN1C(=O)N/C(=C/c2cn(Cc3ccccc3)c4ccccc24)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F21 compound treatment 960.0 -138.0 -0.05 1720.0 886.0 0.68 0.4464 0.6547 2117939 ChemDiv3_006115 Cc1cc(/C=N/O)nc(O)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F22 compound treatment 480.0 -618.0 -0.22 4520.0 3690.0 2.83 1.846 0.6504 3117977 ChemDiv3_006116 COc1ccc(cc1)S(=O)(=O)Nc2ccccc2C(=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F23 mock treatment 2360.0 1260.0 0.45 4760.0 3930.0 3.01 2.4479 0.8034 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 F24 mock treatment 800.0 -298.0 -0.11 4680.0 3850.0 2.95 2.0132 0.6814 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G01 compound treatment 1200.0 103.0 0.04 840.0 5.93 0.0 0.0289 0.7894 1118910 ChemDiv3_006117 Nc1ccc(cc1)S(=O)(=O)NCCC2=CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G02 compound treatment 760.0 -338.0 -0.12 1000.0 166.0 0.13 0.0054 0.031 1155616 ChemDiv3_006118 CC(=O)NCCc1ccc(cc1)S(=O)(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G03 compound treatment 760.0 -338.0 -0.12 800.0 -34.1 -0.03 -0.1032 -0.8417 3026556 ChemDiv3_006119 CC(C)CC1(C)OCC(C[N+]2(C)CCCCC2)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G04 compound treatment 480.0 -618.0 -0.22 520.0 -314.0 -0.24 -0.3254 -0.9989 3118114 ChemDiv3_006120 Cc1c(nc(N)c(C#N)c1c2ccco2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G05 compound treatment 320.0 -778.0 -0.28 400.0 -434.0 -0.33 -0.4307 -0.9956 3026557 ChemDiv3_006121 C[N+]1(CC2COC(O2)C3CCC=CC3)CCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G06 compound treatment 360.0 -738.0 -0.26 1640.0 806.0 0.62 0.2525 0.3759 3118115 ChemDiv3_006122 CN(C)c1ccc(N/C=C\2/CCCC2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G07 compound treatment 480.0 -618.0 -0.22 480.0 -354.0 -0.27 -0.3471 -0.9943 3118116 ChemDiv3_006123 CS(=O)c1nc(cc(n1)C(F)(F)F)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G08 compound treatment 320.0 -778.0 -0.28 400.0 -434.0 -0.33 -0.4307 -0.9956 3118117 ChemDiv3_006124 COc1ccccc1/C=[N+]/2\[N-]C(=O)C(NC(=O)c3cccc(C)c3)C2c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G09 compound treatment 1200.0 103.0 0.04 1320.0 486.0 0.37 0.2895 0.7724 3026558 ChemDiv3_006125 CC(C1OCC(C[N+]2(C)CCCCC2)O1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G10 compound treatment 560.0 -538.0 -0.19 680.0 -154.0 -0.12 -0.2185 -0.9736 3026559 ChemDiv3_006126 NC(=S)Nc1nc2ccccc2[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G11 compound treatment 640.0 -458.0 -0.16 920.0 85.9 0.07 -0.0681 -0.3888 1437584 ChemDiv3_006127 Cc1nn(Cc2ccc(o2)C(=O)NCc3ccc(C)cc3)c(C)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G12 compound treatment 360.0 -738.0 -0.26 760.0 -74.1 -0.06 -0.2252 -0.8412 3026560 ChemDiv3_006128 CC(=S)Nc1c(O)[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G13 compound treatment 600.0 -498.0 -0.18 2160.0 1330.0 1.02 0.595 0.5759 1641981 ChemDiv3_006129 Cc1cc(NC(=O)c2ccc(COc3ccc(Cl)c(C)c3)o2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G14 compound treatment 1280.0 183.0 0.06 680.0 -154.0 -0.12 -0.0379 -0.2808 3026561 ChemDiv3_006130 CC1SC2(CCCCC2)N(C1=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G15 compound treatment 640.0 -458.0 -0.16 520.0 -314.0 -0.24 -0.2853 -0.9814 1387920 ChemDiv3_006131 CC1Cc2ccccc2N1C(=O)c3cccc(COc4ccc(Cl)cc4)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G16 compound treatment 1120.0 22.5 0.01 920.0 85.9 0.07 0.0523 0.7869 3026562 ChemDiv3_006132 CS(=O)(=O)c1nnnn1c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G17 compound treatment 360.0 -738.0 -0.26 1360.0 526.0 0.4 0.1005 0.2089 3118118 ChemDiv3_006133 FC(F)(F)COCc1ccc(cc1)C(=O)NCc2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G18 compound treatment 1440.0 343.0 0.12 640.0 -194.0 -0.15 -0.0194 -0.1011 3118119 ChemDiv3_006134 O=C(NN1C(Nc2ccccc2C1=O)c3ccccn3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G19 compound treatment 480.0 -618.0 -0.22 960.0 126.0 0.1 -0.0865 -0.3614 3026563 ChemDiv3_006135 Cn1cc(Cl)c(n1)C(=O)NCC(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G20 compound treatment 680.0 -418.0 -0.15 800.0 -34.1 -0.03 -0.1232 -0.8193 1552729 ChemDiv3_006136 CCC1(C)Cc2c(CO1)sc3nc(SC)n4c(SCc5ccccc5)nnc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G21 compound treatment 1520.0 423.0 0.15 1040.0 206.0 0.16 0.2178 0.9996 1129557 ChemDiv3_006137 CCOc1ccc(OCc2ccc(o2)C(=O)NN)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G22 compound treatment 560.0 -538.0 -0.19 1720.0 886.0 0.68 0.3461 0.49 1160784 ChemDiv3_006138 CC(C)N1CC2(OC3C=C2)C(C3C(=O)O)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G23 mock treatment 400.0 -698.0 -0.25 1120.0 286.0 0.22 -0.0197 -0.0597 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 G24 mock treatment 840.0 -258.0 -0.09 7600.0 6770.0 5.19 3.6084 0.6946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H01 compound treatment 560.0 -538.0 -0.19 1240.0 406.0 0.31 0.0855 0.2341 3026564 ChemDiv3_006139 CCCCn1c2ccccc2c3nnc(SCC(=O)NC4=NC(=O)CS4)nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H02 compound treatment 720.0 -378.0 -0.13 1000.0 166.0 0.13 -0.0046 -0.025 1508512 ChemDiv3_006140 CC(=O)N1N=C(OC1(C)C)c2ccc(cc2)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H03 compound treatment 7440.0 6340.0 2.25 840.0 5.93 0.0 1.5942 0.7085 3118120 ChemDiv3_006141 OC(=O)CC1(CC(=O)Nc2ccc(Cl)cc2)CCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H04 compound treatment 520.0 -578.0 -0.2 560.0 -274.0 -0.21 -0.2936 -0.9999 3026565 ChemDiv3_006142 S=C1NC(C2=C(N1)C3CCN2CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H05 compound treatment 520.0 -578.0 -0.2 640.0 -194.0 -0.15 -0.2502 -0.9878 3118121 ChemDiv3_006143 Cc1cc(=O)n(CC=C)c(O)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H06 compound treatment 400.0 -698.0 -0.25 520.0 -314.0 -0.24 -0.3455 -0.9999 3026566 ChemDiv3_006144 CC1(C)N(C(=O)N(C1=N)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H07 compound treatment 6200.0 5100.0 1.81 480.0 -354.0 -0.27 1.0877 0.5943 1251296 ChemDiv3_006145 O=S(=O)(NCc1ccc2OCOc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H08 compound treatment 720.0 -378.0 -0.13 680.0 -154.0 -0.12 -0.1783 -0.9981 3118122 ChemDiv3_006146 O=C(NC1=C(N(Cc2ccccc2)S(=O)(=O)c3ccccc13)C(=O)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H09 compound treatment 600.0 -498.0 -0.18 640.0 -194.0 -0.15 -0.2301 -0.9965 3026567 ChemDiv3_006147 Cc1cc(OCc2nc(no2)c3ccc(OCC(=O)N)cc3)cc(C)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H10 compound treatment 520.0 -578.0 -0.2 600.0 -234.0 -0.18 -0.2719 -0.9979 1494546 ChemDiv3_006148 CC(NCc1cccnc1)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H11 compound treatment 440.0 -658.0 -0.23 720.0 -114.0 -0.09 -0.2269 -0.9105 3026602 ChemDiv3_006149 Cc1nc2cc(ccc2[nH]1)c3nc4cc(NC(=O)c5cccs5)ccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H12 compound treatment 1040.0 -57.5 -0.02 1000.0 166.0 0.13 0.0757 0.5864 3118123 ChemDiv3_006150 COc1cccc(CNC(C)(C)CO)c1OCc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H13 compound treatment 600.0 -498.0 -0.18 4080.0 3250.0 2.49 1.6373 0.6554 3026603 ChemDiv3_006151 C1C[C@@H]2[C@H](O1)c3ccccc3N[C@@H]2c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H14 compound treatment 440.0 -658.0 -0.23 720.0 -114.0 -0.09 -0.2269 -0.9105 3118124 ChemDiv3_006152 COc1cc(CNc2ccc3[nH]c(=O)[nH]c3c2)cc(Br)c1OCC(=O)NC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H15 compound treatment 720.0 -378.0 -0.13 1120.0 286.0 0.22 0.0605 0.2354 3026604 ChemDiv3_006153 Cc1ccc(c(C)c1C)S(=O)(=O)N2CCN(C/C=C/c3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H16 compound treatment 440.0 -658.0 -0.23 520.0 -314.0 -0.24 -0.3354 -0.9999 3118125 ChemDiv3_006154 CN(C)CCCNc1oc(nc1C#N)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H17 compound treatment 3000.0 1900.0 0.67 560.0 -274.0 -0.21 0.3284 0.4646 3118126 ChemDiv3_006155 Cc1cc(C)nc(NC(=N)NCCc2c[nH]c3ccccc23)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H18 compound treatment 600.0 -498.0 -0.18 760.0 -74.1 -0.06 -0.165 -0.8899 3026605 ChemDiv3_006156 O=C(CN1C(=O)CSC1=O)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H19 compound treatment 560.0 -538.0 -0.19 6400.0 5570.0 4.27 2.8867 0.6749 3026606 ChemDiv3_006157 CCc1ccc(cc1)n2c(=O)oc3ccc(Cl)cc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H20 compound treatment 640.0 -458.0 -0.16 760.0 -74.1 -0.06 -0.155 -0.9012 3118127 ChemDiv3_006158 CCN1C(=O)N/C(=C/c2ccc(OCc3ccc(cc3)C(=O)O)cc2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H21 compound treatment 480.0 -618.0 -0.22 1040.0 206.0 0.16 -0.0431 -0.1596 3026607 ChemDiv3_006159 C[N+](C)(C)CCC(O)c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H22 compound treatment 2200.0 1100.0 0.39 1920.0 1090.0 0.83 0.8661 0.9405 3118128 ChemDiv3_006160 O=C(CC1SC2=NCCN2C1=O)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H23 mock treatment 640.0 -458.0 -0.16 800.0 -34.1 -0.03 -0.1333 -0.8106 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 H24 mock treatment 880.0 -218.0 -0.08 2920.0 2090.0 1.6 1.0778 0.6723 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I01 compound treatment 280.0 -818.0 -0.29 4440.0 3610.0 2.77 1.7524 0.6296 3118129 ChemDiv3_006161 O=C1C2C3CC(C=C3)C2C(=O)N1CCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I02 compound treatment 320.0 -778.0 -0.28 400.0 -434.0 -0.33 -0.4307 -0.9956 1625760 ChemDiv3_006162 OC(=O)c1ccc(CSC2CCCCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I03 compound treatment 880.0 -218.0 -0.08 280.0 -554.0 -0.43 -0.3553 -0.822 3026608 ChemDiv3_006163 Oc1ccc(cc1CC=C)C(=O)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I04 compound treatment 400.0 -698.0 -0.25 280.0 -554.0 -0.43 -0.4757 -0.9668 3118130 ChemDiv3_006164 CCSC1(SCC)N=C(N)C2(C#N)C(c3ccc(F)cc3)C21C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I05 compound treatment 600.0 -498.0 -0.18 400.0 -434.0 -0.33 -0.3604 -0.9558 3026609 ChemDiv3_006165 CC1CCc2nc(NN)nc(c2C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I06 compound treatment 520.0 -578.0 -0.2 320.0 -514.0 -0.39 -0.4239 -0.9534 3118131 ChemDiv3_006166 CC1(O)CC(=NN1S(=O)(=O)c2ccccc2)C(F)(F)OC(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I07 compound treatment 400.0 -698.0 -0.25 240.0 -594.0 -0.46 -0.4975 -0.9587 3118132 ChemDiv3_006167 O=C(CN1C(=O)C2C3CC(C=C3)C2C1=O)OCCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I08 compound treatment 1680.0 583.0 0.21 280.0 -554.0 -0.43 -0.1547 -0.3271 3026610 ChemDiv3_006168 CCOC(=O)Cc1c(C)nc2c(c(nn2c1C)C(F)(F)F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I09 compound treatment 360.0 -738.0 -0.26 280.0 -554.0 -0.43 -0.4858 -0.9727 3118133 ChemDiv3_006169 C[N+]1(CC(=O)OCCCc2ccccc2)CCOCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I10 compound treatment 280.0 -818.0 -0.29 240.0 -594.0 -0.46 -0.5276 -0.9761 3026611 ChemDiv3_006170 CC1=NC(=O)CN1c2ccc(N)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I11 compound treatment 440.0 -658.0 -0.23 200.0 -634.0 -0.49 -0.5091 -0.9432 3118134 ChemDiv3_006171 Cc1cc(nn1Cc2ccc(o2)C(=O)NCc3ccco3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I12 compound treatment 640.0 -458.0 -0.16 280.0 -554.0 -0.43 -0.4155 -0.9127 3026612 ChemDiv3_006172 Cc1ccc2S/C(=C\c3sc4ccccc4[n+]3C)/N(CCO)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I13 compound treatment 840.0 -258.0 -0.09 360.0 -474.0 -0.36 -0.3219 -0.858 1573342 ChemDiv3_006173 CCN(CC)C(=O)c1ccc(COc2cccc3ccccc23)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I14 compound treatment 360.0 -738.0 -0.26 320.0 -514.0 -0.39 -0.4641 -0.9801 3118261 ChemDiv3_006174 O=C(CCN1C(=O)c2ccccc2C1=O)N3CCC(C3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I15 compound treatment 280.0 -818.0 -0.29 480.0 -354.0 -0.27 -0.3973 -0.9995 1720015 ChemDiv3_006175 Clc1ccccc1OCc2cccc(c2)C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I16 compound treatment 360.0 -738.0 -0.26 4120.0 3290.0 2.52 1.5988 0.6304 3118262 ChemDiv3_006176 CCN1C(=O)N/C(=C/c2ccc(Sc3ccc(C)cc3)o2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I17 compound treatment 560.0 -538.0 -0.19 840.0 5.93 0.0 -0.1316 -0.69 3026613 ChemDiv3_006177 CCn1nccc1C(=O)Nc2cc(Cl)ccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I18 compound treatment 320.0 -778.0 -0.28 640.0 -194.0 -0.15 -0.3004 -0.9582 3118263 ChemDiv3_006178 O=C(COc1ccc(cc1)C2Nc3cccc4cccc(N2)c34)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I19 compound treatment 400.0 -698.0 -0.25 400.0 -434.0 -0.33 -0.4106 -0.9893 3026614 ChemDiv3_006179 CCn1nccc1C(=O)NC2=C(CCC2)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I20 compound treatment 400.0 -698.0 -0.25 1120.0 286.0 0.22 -0.0197 -0.0597 3118264 ChemDiv3_006180 COc1ccc(CSc2nnc3c4c5CC(C)(C)OCc5sc4nc(SC)n23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I21 compound treatment 600.0 -498.0 -0.18 320.0 -514.0 -0.39 -0.4039 -0.9342 1646334 ChemDiv3_006181 O=C(NCc1cccnc1)c2ccc(COc3cccc4ccccc34)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I22 compound treatment 320.0 -778.0 -0.28 3480.0 2650.0 2.03 1.2413 0.6055 3118265 ChemDiv3_006182 CCOC(=O)C1C2OC3(CN(C(C)C)C(=O)C13)C=C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I23 mock treatment 800.0 -298.0 -0.11 960.0 126.0 0.1 -0.0063 -0.0438 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 I24 mock treatment 360.0 -738.0 -0.26 1320.0 486.0 0.37 0.0788 0.1729 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J01 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3118266 ChemDiv3_006183 CC(N1C(=O)/C(=C\2/C(=O)N(C)c3ccccc23)/SC1=S)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J02 compound treatment 440.0 -658.0 -0.23 360.0 -474.0 -0.36 -0.4223 -0.9769 1213293 ChemDiv3_006184 COc1ccc(CC2(C)OC(=NN2C(=O)C)c3ccncc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J03 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3118267 ChemDiv3_006185 COc1ccc(NC(=O)CC2(CC(=O)O)CCCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J04 compound treatment 280.0 -818.0 -0.29 400.0 -434.0 -0.33 -0.4407 -0.9976 1515449 ChemDiv3_006186 COc1ccc2C3=NN(C(C3CCc2c1)c4ccccc4)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J05 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3118268 ChemDiv3_006187 Clc1ccc(OCCN2CCNCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J06 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3026615 ChemDiv3_006188 Cc1ccccc1Nc2nnc(C)c(=O)n2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J07 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3118269 ChemDiv3_006189 Fc1ccccc1N2CCN(CC2)C(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J08 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3118270 ChemDiv3_006190 CN1C(=C(OC(=O)C)c2ccccc2S1(=O)=O)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J09 compound treatment 360.0 -738.0 -0.26 800.0 -34.1 -0.03 -0.2035 -0.7739 3026616 ChemDiv3_006191 C(c1ccccc1)n2c3nc(nn3c4ccccc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J10 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3118271 ChemDiv3_006192 CC(NCc1ccc(F)cc1)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J11 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 3026654 ChemDiv3_006193 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3nc([nH]c3c2)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J12 compound treatment 320.0 -778.0 -0.28 480.0 -354.0 -0.27 -0.3872 -1.0 3118272 ChemDiv3_006194 COc1cc(CNC(C)(C)CO)cc(Br)c1OCc2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J13 compound treatment 560.0 -538.0 -0.19 400.0 -434.0 -0.33 -0.3705 -0.9649 3026655 ChemDiv3_006195 CCc1cccc2C(C)CC3(CCCC3)Nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J14 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 3118273 ChemDiv3_006196 CCOc1cc(CNc2ccc(OC)cc2)ccc1OCC(=O)NC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J15 compound treatment 320.0 -778.0 -0.28 4200.0 3370.0 2.58 1.6322 0.6281 3118274 ChemDiv3_006197 COc1cccc(NC(=S)NC(=N)Nc2nc(C)c3ccccc3n2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J16 compound treatment 1800.0 703.0 0.25 2680.0 1850.0 1.42 1.1783 0.8189 1490556 ChemDiv3_006198 COc1ccc(Nc2oc(nc2C#N)c3ccc(OC)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J17 compound treatment 400.0 -698.0 -0.25 400.0 -434.0 -0.33 -0.4106 -0.9893 3118275 ChemDiv3_006199 CCNC(=S)N1CCN=C1Nc2nc(C)cc(C)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J18 compound treatment 280.0 -818.0 -0.29 360.0 -474.0 -0.36 -0.4624 -0.9937 3026656 ChemDiv3_006200 S=C(N1CCCCC1)c2cn(Cc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J19 compound treatment 840.0 -258.0 -0.09 280.0 -554.0 -0.43 -0.3654 -0.8398 1547515 ChemDiv3_006201 COC(=O)c1ccc(NC(=O)c2cccc(c2)C(=O)Nc3ccc(cc3)C(=O)OC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J20 compound treatment 320.0 -778.0 -0.28 240.0 -594.0 -0.46 -0.5175 -0.971 3026657 ChemDiv3_006202 CCN1C(=O)N/C(=C/c2cccn2c3ccc(cc3)C(=O)O)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J21 compound treatment 360.0 -738.0 -0.26 360.0 -474.0 -0.36 -0.4424 -0.9869 3118276 ChemDiv3_006203 CNS(=O)(=O)c1ccc2c(c1)oc(=O)c3cc(ccc32)S(=O)(=O)NC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J22 compound treatment 440.0 -658.0 -0.23 400.0 -434.0 -0.33 -0.4006 -0.9848 3118277 ChemDiv3_006204 Fc1ccc(CN2C(=O)SC(C3SC(=O)N(Cc4ccc(F)cc4)C3=O)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J23 mock treatment 360.0 -738.0 -0.26 1320.0 486.0 0.37 0.0788 0.1729 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 J24 mock treatment 320.0 -778.0 -0.28 5080.0 4250.0 3.26 2.1099 0.645 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K01 compound treatment 1160.0 62.5 0.02 1120.0 286.0 0.22 0.1709 0.7746 1399766 ChemDiv3_006205 OC(=O)c1ccc(COc2ccccc2CC=C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K02 compound treatment 640.0 -458.0 -0.16 960.0 126.0 0.1 -0.0464 -0.2456 3118278 ChemDiv3_006206 COc1cc(OC)c(/N=C/2\C=C(O)C(=O)c3ccccc23)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K03 compound treatment 520.0 -578.0 -0.2 480.0 -354.0 -0.27 -0.3371 -0.9903 3026658 ChemDiv3_006207 COC(=O)c1ccc(COc2ccc(cc2OC)C3OC(C)CC(C)(C)O3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K04 compound treatment 760.0 -338.0 -0.12 840.0 5.93 0.0 -0.0814 -0.6797 3118279 ChemDiv3_006208 COc1ccc(cc1)C2C3(C#N)C(=NC4(OCCO4)C23C#N)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K05 compound treatment 520.0 -578.0 -0.2 800.0 -34.1 -0.03 -0.1634 -0.791 3026659 ChemDiv3_006209 CC1CCc2nc(NCCO)nc(c2C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K06 compound treatment 1000.0 -97.5 -0.03 720.0 -114.0 -0.09 -0.0864 -0.9174 3118280 ChemDiv3_006210 OC(=O)c1ccccc1N/C=C\2/CCCCC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K07 compound treatment 280.0 -818.0 -0.29 720.0 -114.0 -0.09 -0.267 -0.8813 3118281 ChemDiv3_006211 CC1=NN(C(C1)c2ccc(OCC(=O)NCCC3=CCCCC3)cc2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K08 compound treatment 400.0 -698.0 -0.25 560.0 -274.0 -0.21 -0.3237 -0.9967 3026660 ChemDiv3_006212 CCOc1ccc(NC2=CC(=O)CCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K09 compound treatment 400.0 -698.0 -0.25 920.0 85.9 0.07 -0.1283 -0.5011 3026661 ChemDiv3_006213 C[N+]1(CC(=O)OC2CCCCCCCCCCC2)CCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K10 compound treatment 840.0 -258.0 -0.09 1040.0 206.0 0.16 0.0472 0.2585 3118282 ChemDiv3_006214 CSc1[n+](C)ccc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K11 compound treatment 480.0 -618.0 -0.22 1080.0 246.0 0.19 -0.0214 -0.074 1702476 ChemDiv3_006215 CCc1ccc(OCc2ccc(o2)C(=O)OC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K12 compound treatment 800.0 -298.0 -0.11 1160.0 326.0 0.25 0.1023 0.3767 3026662 ChemDiv3_006216 Cc1cc2N=C(CC(c3ccccc3)n2n1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K13 compound treatment 440.0 -658.0 -0.23 7320.0 6490.0 4.98 3.356 0.6732 3118283 ChemDiv3_006217 CCn1ccc(n1)C(=O)Nc2nccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K14 compound treatment 2840.0 1740.0 0.62 920.0 85.9 0.07 0.4837 0.7781 3118284 ChemDiv3_006218 O=C(/C=C/c1ccccc1)N2CCC(C2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K15 compound treatment 320.0 -778.0 -0.28 640.0 -194.0 -0.15 -0.3004 -0.9582 3026663 ChemDiv3_006219 CCn1ccc(n1)C(=O)Nc2ccccc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K16 compound treatment 520.0 -578.0 -0.2 1200.0 366.0 0.28 0.0538 0.1547 3026664 ChemDiv3_006220 CCOC(=O)NN1CNc2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K17 compound treatment 480.0 -618.0 -0.22 880.0 45.9 0.04 -0.13 -0.5858 3118285 ChemDiv3_006221 OC(=O)c1cccc(COCC(F)(F)F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K18 compound treatment 800.0 -298.0 -0.11 800.0 -34.1 -0.03 -0.0931 -0.8565 3118286 ChemDiv3_006222 COc1ccc(cc1OC)c2nnc3s/c(=C\c4ccco4)/c(=O)n23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K19 compound treatment 560.0 -538.0 -0.19 480.0 -354.0 -0.27 -0.327 -0.985 3026665 ChemDiv3_006223 CC1CN(CC(C)O1)C(=O)c2ccc(COCC(F)(F)F)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K20 compound treatment 600.0 -498.0 -0.18 720.0 -114.0 -0.09 -0.1867 -0.9477 3118287 ChemDiv3_006224 CCn1c(=O)c2c3CCCCc3sc2n4c(SCc5ccc(OC)cc5)nnc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K21 compound treatment 480.0 -618.0 -0.22 480.0 -354.0 -0.27 -0.3471 -0.9943 1606512 ChemDiv3_006225 CCOc1ccc(OCc2ccc(o2)C(=O)NC(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K22 compound treatment 640.0 -458.0 -0.16 520.0 -314.0 -0.24 -0.2853 -0.9814 3118288 ChemDiv3_006226 CCOC(=O)C1C2OC3(CN(CC(C)C)C(=O)C13)C=C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K23 mock treatment 800.0 -298.0 -0.11 680.0 -154.0 -0.12 -0.1583 -0.9984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 K24 mock treatment 640.0 -458.0 -0.16 1360.0 526.0 0.4 0.1707 0.3924 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L01 compound treatment 4120.0 3020.0 1.07 680.0 -154.0 -0.12 0.6745 0.6253 1377574 ChemDiv3_006227 Cc1ccc(CCNc2ccccc2)cn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L02 compound treatment 560.0 -538.0 -0.19 320.0 -514.0 -0.39 -0.4139 -0.9443 2076714 ChemDiv3_006228 CCOC(=O)CSc1nnnn1c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L03 compound treatment 1080.0 -17.5 -0.01 880.0 45.9 0.04 0.0205 0.5738 3118409 ChemDiv3_006229 OC(=O)CC1(CC(=O)Nc2cccnc2)CCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L04 compound treatment 6840.0 5740.0 2.04 840.0 5.93 0.0 1.4437 0.7087 3026666 ChemDiv3_006230 CCc1ccc2[nH]c3nc(C)cc(C)c3c(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L05 compound treatment 760.0 -338.0 -0.12 2200.0 1370.0 1.05 0.6568 0.6223 3118410 ChemDiv3_006231 CC(C)c1ccc(OCCN2CCNCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L06 compound treatment 1320.0 223.0 0.08 440.0 -394.0 -0.3 -0.1581 -0.5057 3118411 ChemDiv3_006232 Cc1nnc(NCc2ccccc2)n(N)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L07 compound treatment 480.0 -618.0 -0.22 600.0 -234.0 -0.18 -0.282 -0.9952 3026667 ChemDiv3_006233 CN(C(=O)N1c2ccccc2Sc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L08 compound treatment 1160.0 62.5 0.02 400.0 -434.0 -0.33 -0.22 -0.6586 1467460 ChemDiv3_006234 O=C(Cn1n(CC(=O)N2CCOCC2)c(=O)n(c3ccccc3)c1=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L09 compound treatment 600.0 -498.0 -0.18 440.0 -394.0 -0.3 -0.3387 -0.9671 3118412 ChemDiv3_006235 COc1ccc(cc1OC)C(=O)Cn2c(=O)c(CCC(=O)O)nn3c4ccccc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L10 compound treatment 280.0 -818.0 -0.29 800.0 -34.1 -0.03 -0.2236 -0.7678 3118413 ChemDiv3_006236 CN(C)c1ccc(NCc2cccc(Br)c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L11 compound treatment 600.0 -498.0 -0.18 1800.0 966.0 0.74 0.3996 0.5242 3118414 ChemDiv3_006237 COC(=O)CN1C(c2ccccc2)c3cc(C)ccc3N=C1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L12 compound treatment 720.0 -378.0 -0.13 4120.0 3290.0 2.52 1.6891 0.6686 3026716 ChemDiv3_006238 CCOc1ccc(CNc2ccc(cc2)N3CCN(Cc4ccccc4)CC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L13 compound treatment 1400.0 303.0 0.11 1040.0 206.0 0.16 0.1877 0.9822 1024590 ChemDiv3_006239 COc1ccc(cc1)C(=O)CCN2CCC(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L14 compound treatment 520.0 -578.0 -0.2 920.0 85.9 0.07 -0.0982 -0.4563 3026717 ChemDiv3_006240 CCOc1cc(CNc2nc[nH]n2)ccc1OCC(=O)NC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L15 compound treatment 680.0 -418.0 -0.15 720.0 -114.0 -0.09 -0.1667 -0.9686 3118415 ChemDiv3_006241 CC1=Nc2ccccc2N=C(N)C1c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L16 compound treatment 640.0 -458.0 -0.16 1360.0 526.0 0.4 0.1707 0.3924 1485170 ChemDiv3_006242 COc1ccc(cc1)c2nc(C#N)c(o2)N3CCN(C)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L17 compound treatment 680.0 -418.0 -0.15 8240.0 7410.0 5.69 3.9156 0.6885 3026718 ChemDiv3_006243 N=C(NC(=O)c1ccccc1)N2N=CCC2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L18 compound treatment 360.0 -738.0 -0.26 680.0 -154.0 -0.12 -0.2686 -0.9356 1548077 ChemDiv3_006244 OC(=O)C1CC=CCC1C(=O)Nc2ccccc2S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L19 compound treatment 680.0 -418.0 -0.15 720.0 -114.0 -0.09 -0.1667 -0.9686 3118416 ChemDiv3_006245 COC(Cn1c(cc(C2=C(O)CC(C)(C)CC2=O)c1c3ccccc3)c4ccccc4)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L20 compound treatment 400.0 -698.0 -0.25 800.0 -34.1 -0.03 -0.1935 -0.7775 3026719 ChemDiv3_006246 Cc1ccc2cccc(OCc3ccc(Br)cc3)c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L21 compound treatment 840.0 -258.0 -0.09 680.0 -154.0 -0.12 -0.1482 -0.9918 3026720 ChemDiv3_006247 CN(C)c1ccc(CNc2cc(C)ccn2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L22 compound treatment 400.0 -698.0 -0.25 3080.0 2250.0 1.72 1.0443 0.5995 3118417 ChemDiv3_006248 COC(=O)c1cc2ccc(OC)c(OC)c2c(=O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L23 mock treatment 1120.0 22.5 0.01 640.0 -194.0 -0.15 -0.0997 -0.6683 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 L24 mock treatment 400.0 -698.0 -0.25 3360.0 2530.0 1.94 1.1963 0.6119 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M01 compound treatment 560.0 -538.0 -0.19 920.0 85.9 0.07 -0.0882 -0.4371 3026721 ChemDiv3_006249 CC1CC(CC(C)(C)C1)OC(=O)CN2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M02 compound treatment 3560.0 2460.0 0.87 800.0 -34.1 -0.03 0.5992 0.6856 1691540 ChemDiv3_006250 Fc1ccccc1C2N(Cc3ccccc3)CCCN2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M03 compound treatment 440.0 -658.0 -0.23 400.0 -434.0 -0.33 -0.4006 -0.9848 3118418 ChemDiv3_006251 FC(F)(F)c1cc(nc(SCC(=O)OCCCc2ccccc2)n1)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M04 compound treatment 2720.0 1620.0 0.58 720.0 -114.0 -0.09 0.3451 0.5927 3026722 ChemDiv3_006252 COc1ccc(cc1)C2C3(C#N)C(=NC(OC)(OC)C23C#N)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M05 compound treatment 440.0 -658.0 -0.23 360.0 -474.0 -0.36 -0.4223 -0.9769 3118419 ChemDiv3_006253 FC(F)(F)c1nc(SCC(=O)NCCC2=CCCCC2)nc3CCCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M06 compound treatment 720.0 -378.0 -0.13 480.0 -354.0 -0.27 -0.2869 -0.9468 3026723 ChemDiv3_006254 CC1CCC/C(=C/Nc2ccc3OCOc3c2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M07 compound treatment 1680.0 583.0 0.21 1040.0 206.0 0.16 0.2579 0.9913 3118420 ChemDiv3_006255 CC1=NN(C(C1)c2ccc(OCC(=O)N3CCCC3)cc2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M08 compound treatment 280.0 -818.0 -0.29 400.0 -434.0 -0.33 -0.4407 -0.9976 3118421 ChemDiv3_006256 C/N=C/1\S/C(=C/c2cccn2c3ccc(cc3)N(C)C)/C(=O)N1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M09 compound treatment 360.0 -738.0 -0.26 240.0 -594.0 -0.46 -0.5075 -0.9652 3026724 ChemDiv3_006257 CCOC(=O)C1CCCN(CCP(=O)(c2ccccc2)c3ccccc3)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M10 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 3118422 ChemDiv3_006258 Cc1ccccc1/N=C/2\Nc3ccc4ccccc4c3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M11 compound treatment 440.0 -658.0 -0.23 320.0 -514.0 -0.39 -0.444 -0.9685 1171394 ChemDiv3_006259 Clc1cnn(Cc2cccc(c2)C(=O)NC3CCCCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M12 compound treatment 440.0 -658.0 -0.23 480.0 -354.0 -0.27 -0.3571 -0.9971 3118423 ChemDiv3_006260 NCCn1c(N)c(C#N)c2nc3ccccc3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M13 compound treatment 320.0 -778.0 -0.28 400.0 -434.0 -0.33 -0.4307 -0.9956 1308018 ChemDiv3_006261 Cc1ccc(OCc2ccc(o2)C(=O)NC(c3ccccc3)c4ccccc4)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M14 compound treatment 640.0 -458.0 -0.16 1160.0 326.0 0.25 0.0622 0.2085 1706518 ChemDiv3_006262 O=C(CCN1CCc2ccccc2C1)c3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M15 compound treatment 240.0 -858.0 -0.3 480.0 -354.0 -0.27 -0.4073 -0.9984 3118424 ChemDiv3_006263 COC(=O)c1ccc(Cn2nc(cc2C)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M16 compound treatment 400.0 -698.0 -0.25 480.0 -354.0 -0.27 -0.3672 -0.9989 3026725 ChemDiv3_006264 CCOC(=O)NN1C(Nc2ccccc2C1=O)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M17 compound treatment 560.0 -538.0 -0.19 800.0 -34.1 -0.03 -0.1533 -0.7967 3118425 ChemDiv3_006265 FC(F)(F)COCc1ccc(o1)C(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M18 compound treatment 560.0 -538.0 -0.19 960.0 126.0 0.1 -0.0665 -0.3109 3026726 ChemDiv3_006266 N(c1nc2ccccc2[nH]1)n3cnnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M19 compound treatment 360.0 -738.0 -0.26 840.0 5.93 0.0 -0.1818 -0.6947 3118426 ChemDiv3_006267 FC(F)(F)COCc1cccc(c1)C(=O)N/C=N/c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M20 compound treatment 3200.0 2100.0 0.75 920.0 85.9 0.07 0.574 0.7667 1375388 ChemDiv3_006268 CCCOc1ccc(cc1)c2cnc(S)nc2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M21 compound treatment 3480.0 2380.0 0.85 1040.0 206.0 0.16 0.7094 0.8251 3118427 ChemDiv3_006269 FC(F)(F)COC(=O)c1ccc(COc2ccc3ccccc3c2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M22 compound treatment 2480.0 1380.0 0.49 560.0 -274.0 -0.21 0.198 0.371 3118428 ChemDiv3_006270 CCN1C(=O)/C(=C/c2cn(CC)c3ccccc23)/NC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M23 mock treatment 560.0 -538.0 -0.19 1080.0 246.0 0.19 -0.0013 -0.0049 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 M24 mock treatment 1640.0 543.0 0.19 5000.0 4170.0 3.2 2.3976 0.7483 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N01 compound treatment 2680.0 1580.0 0.56 3760.0 2930.0 2.25 1.9853 0.8575 1348089 ChemDiv3_006271 OCc1ccccc1CN2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N02 compound treatment 1000.0 -97.5 -0.03 800.0 -34.1 -0.03 -0.043 -0.9905 3026727 ChemDiv3_006272 CCCSc1nnc(N)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N03 compound treatment 360.0 -738.0 -0.26 1200.0 366.0 0.28 0.0136 0.0356 3118429 ChemDiv3_006273 OC(=O)CC1(CC(=O)Nc2cccc(c2)C(F)(F)F)CCCC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N04 compound treatment 560.0 -538.0 -0.19 760.0 -74.1 -0.06 -0.175 -0.8797 3118430 ChemDiv3_006274 Cc1cccc(c1)N2C3CS(=O)(=O)CC3N(C2=O)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N05 compound treatment 400.0 -698.0 -0.25 320.0 -514.0 -0.39 -0.454 -0.9747 3026728 ChemDiv3_006275 COc1cccc(OCCCN2CCNCC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N06 compound treatment 480.0 -618.0 -0.22 760.0 -74.1 -0.06 -0.1951 -0.8621 3026729 ChemDiv3_006276 Cc1nnc(NCCc2ccccc2)n(N)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N07 compound treatment 480.0 -618.0 -0.22 320.0 -514.0 -0.39 -0.434 -0.9614 1129689 ChemDiv3_006277 COc1cc2c(cc1NC(=O)CCC3CCCCC3)oc4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N08 compound treatment 240.0 -858.0 -0.3 200.0 -634.0 -0.49 -0.5593 -0.9744 3118431 ChemDiv3_006278 OC(=O)Cn1nnnc1SCC(=O)Nc2ccccc2F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N09 compound treatment 320.0 -778.0 -0.28 1440.0 606.0 0.47 0.1339 0.2476 3025868 ChemDiv3_006279 C(N1CCOCC1)c2c(nc3c4ccccc4ccn23)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N10 compound treatment 640.0 -458.0 -0.16 3720.0 2890.0 2.22 1.4519 0.6536 3025869 ChemDiv3_006280 CC(=O)N(Cc1cccc(Br)c1)c2ccc3oc(nc3c2)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N11 compound treatment 560.0 -538.0 -0.19 800.0 -34.1 -0.03 -0.1533 -0.7967 1668136 ChemDiv3_006281 COC(=O)CN1C(c2ccccc2)c3cc(Cl)ccc3NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N12 compound treatment 640.0 -458.0 -0.16 440.0 -394.0 -0.3 -0.3287 -0.9574 3118551 ChemDiv3_006282 O=C(N1CCN(CC1)c2ccc(NCc3ccc4OCOc4c3)cc2)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N13 compound treatment 2760.0 1660.0 0.59 160.0 -674.0 -0.52 0.0511 0.0651 3025870 ChemDiv3_006283 CCOC(=O)N1CCN(CCC(=O)c2ccc(OC)cc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N14 compound treatment 600.0 -498.0 -0.18 600.0 -234.0 -0.18 -0.2519 -1.0 3118552 ChemDiv3_006284 CN(C)CCCNc1oc(nc1C#N)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N15 compound treatment 360.0 -738.0 -0.26 680.0 -154.0 -0.12 -0.2686 -0.9356 3025871 ChemDiv3_006285 COc1ccc(cc1)C(=O)NC2=Nc3ccccc3N=C(C)C2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N16 compound treatment 240.0 -858.0 -0.3 480.0 -354.0 -0.27 -0.4073 -0.9984 3118553 ChemDiv3_006286 CCOC(=O)N1CCC(CC1)Nc2nc(OC)nc(OC)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N17 compound treatment 800.0 -298.0 -0.11 760.0 -74.1 -0.06 -0.1148 -0.9579 3118554 ChemDiv3_006287 CN1CCN(CC1)C(=S)SCC(=O)Nc2nc(=O)c3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N18 compound treatment 2080.0 983.0 0.35 640.0 -194.0 -0.15 0.1411 0.3722 1736377 ChemDiv3_006288 OC(=O)CCC(=O)Nc1cccc(O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N19 compound treatment 360.0 -738.0 -0.26 840.0 5.93 0.0 -0.1818 -0.6947 3118555 ChemDiv3_006289 CCOCC(=O)NC1CCSC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N20 compound treatment 320.0 -778.0 -0.28 560.0 -274.0 -0.21 -0.3438 -0.9911 3025872 ChemDiv3_006290 O=C(CN1C(=O)c2ccccc2S1(=O)=O)Nc3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N21 compound treatment 520.0 -578.0 -0.2 640.0 -194.0 -0.15 -0.2502 -0.9878 3118556 ChemDiv3_006291 CCCn1c(NCc2ccc(OC)cc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N22 compound treatment 1640.0 543.0 0.19 720.0 -114.0 -0.09 0.0742 0.3507 3025873 ChemDiv3_006292 CC(C)C1CCC(C)CC1OCC[N+](C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N23 mock treatment 3880.0 2780.0 0.99 720.0 -114.0 -0.09 0.636 0.6418 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 N24 mock treatment 560.0 -538.0 -0.19 920.0 85.9 0.07 -0.0882 -0.4371 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O01 compound treatment 400.0 -698.0 -0.25 320.0 -514.0 -0.39 -0.454 -0.9747 1217799 ChemDiv3_006293 OC(=O)c1cccc(COc2ccccc2CC=C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O02 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 1711668 ChemDiv3_006294 OC(=O)c1ccc(CSCC(=O)Nc2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O03 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3025874 ChemDiv3_006295 Cc1ccc(cc1)S(=O)(=O)CC(N2CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O04 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3118557 ChemDiv3_006296 CCSC1(SCC)N=C(N)C2(C#N)C(c3ccc(OC)cc3)C21C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O05 compound treatment 360.0 -738.0 -0.26 280.0 -554.0 -0.43 -0.4858 -0.9727 3025875 ChemDiv3_006297 CCn1cc(Br)c(n1)c2nc3ccccc3c(=O)n2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O06 compound treatment 400.0 -698.0 -0.25 320.0 -514.0 -0.39 -0.454 -0.9747 3118558 ChemDiv3_006298 CCOc1ccc(N/C=C\2/CCCC(C)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O07 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 3118559 ChemDiv3_006299 CCOC(=O)COc1ccc(cc1)C2CC(=NN2c3ccccc3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O08 compound treatment 240.0 -858.0 -0.3 360.0 -474.0 -0.36 -0.4725 -0.996 3025876 ChemDiv3_006300 Cc1ccc(cc1)C2=C/C(=C/c3ccc(o3)c4cccc(c4)C(=O)O)/C(=O)O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O09 compound treatment 280.0 -818.0 -0.29 200.0 -634.0 -0.49 -0.5493 -0.9694 3118560 ChemDiv3_006301 COC(=O)c1ccc(Cn2cc(Cl)cn2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O10 compound treatment 400.0 -698.0 -0.25 520.0 -314.0 -0.24 -0.3455 -0.9999 3025877 ChemDiv3_006302 Cc1cc(C)c2nc(O)cc(C(=O)O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O11 compound treatment 280.0 -818.0 -0.29 400.0 -434.0 -0.33 -0.4407 -0.9976 1294303 ChemDiv3_006303 CCCc1ccc(OCc2ccc(cc2)C(=O)n3cc(Br)cn3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O12 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3118561 ChemDiv3_006304 Cc1nn(c(N)c1C(NC(=O)c2ccccc2)(C(F)(F)F)C(F)(F)F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O13 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3025878 ChemDiv3_006305 O=C(NC1CCOC1=O)c2ccc(COc3ccc4ccccc4c3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O14 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 1507755 ChemDiv3_006306 OC1(CN(CCC(=O)c2ccc3OCCOc3c2)CCc4ccccc41)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O15 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3025879 ChemDiv3_006307 O=C(Nc1ccncc1)c2cccc(COc3ccc4ccccc4c3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O16 compound treatment 400.0 -698.0 -0.25 320.0 -514.0 -0.39 -0.454 -0.9747 3118562 ChemDiv3_006308 CS(=O)(=O)NN1C(=O)c2ccccc2NC31CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O17 compound treatment 200.0 -898.0 -0.32 320.0 -514.0 -0.39 -0.5042 -0.9943 3025880 ChemDiv3_006309 CC(C)(C)NC(=O)c1ccc(COCC(F)(F)F)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O18 compound treatment 400.0 -698.0 -0.25 440.0 -394.0 -0.3 -0.3889 -0.995 3118563 ChemDiv3_006310 OC(=O)C(N1C(=O)/C(=C/c2ccncc2)/SC1=S)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O19 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 3118564 ChemDiv3_006311 COC(=O)c1ccccc1NC(=O)c2ccc(Cn3cc(Cl)cn3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O20 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3025881 ChemDiv3_006312 OC(=O)CC1N(C(=S)N(C1=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O21 compound treatment 280.0 -818.0 -0.29 200.0 -634.0 -0.49 -0.5493 -0.9694 1248802 ChemDiv3_006313 CCOc1ccc(OCc2cccc(c2)C(=O)N3CCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O22 compound treatment 720.0 -378.0 -0.13 320.0 -514.0 -0.39 -0.3738 -0.8968 3025882 ChemDiv3_006314 COc1cccc(c1)c2nc(c(o2)N(C)C)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O23 mock treatment 440.0 -658.0 -0.23 240.0 -594.0 -0.46 -0.4874 -0.9515 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 O24 mock treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P01 compound treatment 320.0 -778.0 -0.28 360.0 -474.0 -0.36 -0.4524 -0.9906 1267325 ChemDiv3_006315 CC1CCN(Cc2ccccc2CO)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P02 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3025883 ChemDiv3_006316 O=c1n(CCSc2nnnn2c3ccccc3)nnn1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P03 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3118565 ChemDiv3_006317 Cc1cc(c2c(nn(c3ccccc3)c2n1)c4ccccc4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P04 compound treatment 360.0 -738.0 -0.26 400.0 -434.0 -0.33 -0.4206 -0.9928 3118566 ChemDiv3_006318 OC(=O)Cn1c(nc(=S)c2CCCCc21)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P05 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 1877641 ChemDiv3_006319 COc1ccc2C(NC(=O)c3cnn(c3N)c4ccccc4)OC(=O)c2c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P06 compound treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 3118567 ChemDiv3_006320 Cc1nn2N=C(CSc2nc1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P07 compound treatment 280.0 -818.0 -0.29 360.0 -474.0 -0.36 -0.4624 -0.9937 1851771 ChemDiv3_006321 CCCC(=O)Nc1ccc2n(CC)c3ccccc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P08 compound treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 3025884 ChemDiv3_006322 CCSc1nc2ccccc2n1S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P09 compound treatment 200.0 -898.0 -0.32 360.0 -474.0 -0.36 -0.4825 -0.9978 3025939 ChemDiv3_006323 CC(C)(C)c1cn2c(n1)n(N)c3ccccc32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P10 compound treatment 240.0 -858.0 -0.3 400.0 -434.0 -0.33 -0.4507 -0.999 3118568 ChemDiv3_006324 Clc1ccccc1COc2cccc(CNCc3cccnc3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P11 compound treatment 240.0 -858.0 -0.3 200.0 -634.0 -0.49 -0.5593 -0.9744 3025940 ChemDiv3_006325 Clc1ccc2N=C3CNC(=O)CN3C(c4ccccc4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P12 compound treatment 360.0 -738.0 -0.26 160.0 -674.0 -0.52 -0.5509 -0.9501 3118569 ChemDiv3_006326 COc1cc(CNc2ccc(cc2)C(=O)O)ccc1OCc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P13 compound treatment 280.0 -818.0 -0.29 280.0 -554.0 -0.43 -0.5058 -0.9826 3025941 ChemDiv3_006327 CCOC(=O)N1CCN(CCC(=O)c2ccc(Br)cc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P14 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 1294667 ChemDiv3_006328 Fc1ccc(cc1)c2nc(C#N)c(NC3CCCCC3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P15 compound treatment 440.0 -658.0 -0.23 320.0 -514.0 -0.39 -0.444 -0.9685 3118570 ChemDiv3_006329 CN(C1CCCCC1)C(=S)SCC(=O)c2c(C)[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P16 compound treatment 1040.0 -57.5 -0.02 320.0 -514.0 -0.39 -0.2935 -0.7427 3025942 ChemDiv3_006330 Cc1ccc(cc1)C(=O)CC(C(=O)O)c2cn(CCC#N)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P17 compound treatment 360.0 -738.0 -0.26 320.0 -514.0 -0.39 -0.4641 -0.9801 3118571 ChemDiv3_006331 Clc1ccc2[nH]c(=O)c(SC(=S)N3CCOCC3)c(c4ccccc4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P18 compound treatment 240.0 -858.0 -0.3 240.0 -594.0 -0.46 -0.5376 -0.9806 3025943 ChemDiv3_006332 OC(=O)Cn1cc(C(=S)N2CCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P19 compound treatment 240.0 -858.0 -0.3 320.0 -514.0 -0.39 -0.4942 -0.9917 3118572 ChemDiv3_006333 Clc1ccc(cc1)C(=O)/C=c/2\[nH]c(=O)\c(=C\c3cccnc3)\s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P20 compound treatment 240.0 -858.0 -0.3 280.0 -554.0 -0.43 -0.5159 -0.9865 1860014 ChemDiv3_006334 Cc1c(NC(=O)CCSc2ccc(C)cc2)c(=O)n(c3ccccc3)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P21 compound treatment 320.0 -778.0 -0.28 280.0 -554.0 -0.43 -0.4958 -0.978 1074405 ChemDiv3_006335 Oc1ccccc1CNc2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P22 compound treatment 360.0 -738.0 -0.26 280.0 -554.0 -0.43 -0.4858 -0.9727 3025944 ChemDiv3_006336 CC[N+]1(C)CC2CCC(C)(C1)C2(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P23 mock treatment 320.0 -778.0 -0.28 320.0 -514.0 -0.39 -0.4741 -0.9847 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2018 P24 mock treatment 280.0 -818.0 -0.29 320.0 -514.0 -0.39 -0.4841 -0.9885 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A01 compound treatment 280.0 -826.0 -0.29 440.0 -407.0 -0.31 -0.4281 -0.9995 3118695 ChemDiv3_006337 CNC(=O)COc1ccc(cc1)c2nn(C)c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A02 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3118696 ChemDiv3_006338 CCOC(=O)N1CCC(CC1)NC(=O)C(Cc2ccccc2)NC(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A03 compound treatment 480.0 -626.0 -0.22 320.0 -527.0 -0.4 -0.4431 -0.9602 3025945 ChemDiv3_006339 COc1nnc(c2ccc(N3CCCCC3)c(NC(=O)C)c2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A04 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3118697 ChemDiv3_006340 O=C(CSc1nnc2ccc3ccccc3n12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A05 compound treatment 360.0 -746.0 -0.26 440.0 -407.0 -0.31 -0.4081 -0.9966 3025946 ChemDiv3_006341 CC(C)Nc1nc(NC(C)C)nc(Sc2nn(C)c(=S)s2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A06 compound treatment 3600.0 2490.0 0.88 920.0 73.1 0.06 0.6652 0.7505 3118698 ChemDiv3_006342 CCC(=O)c1c(OCC(=O)N)ccc2c(C)cc(=O)oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A07 compound treatment 440.0 -666.0 -0.24 720.0 -127.0 -0.1 -0.236 -0.9232 3118699 ChemDiv3_006343 CCOc1ccc(Nc2nc(N)nc(CN3CC(C)CC(C)C3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A08 compound treatment 360.0 -746.0 -0.26 3480.0 2630.0 2.02 1.2422 0.6093 3025947 ChemDiv3_006344 CCOc1ccc(Nc2oc(COc3ccccc3Cl)nc2C#N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A09 compound treatment 360.0 -746.0 -0.26 920.0 73.1 0.06 -0.1475 -0.5451 3118700 ChemDiv3_006345 Cc1nc(SCSc2nc3ccccc3s2)nc4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A10 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3025948 ChemDiv3_006346 Cc1cccc(c1)c2nc3SC(CC(=O)n3n2)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A11 compound treatment 440.0 -666.0 -0.24 200.0 -647.0 -0.5 -0.5183 -0.9423 3118701 ChemDiv3_006347 Cc1cc(C)c2CN(Cc3ccc(Cl)cc3)COc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A12 compound treatment 360.0 -746.0 -0.26 1040.0 193.0 0.15 -0.0824 -0.2715 3118702 ChemDiv3_006348 O=C(Cn1cc(/C=C\2/C(=O)Nc3ccccc23)c4ccccc14)NCC5CCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A13 compound treatment 280.0 -826.0 -0.29 240.0 -607.0 -0.47 -0.5367 -0.975 3025949 ChemDiv3_006349 CC1CC(C)N(C(C)C1)C(=O)CSc2nc(c3CCc4ccccc4-c3n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A14 compound treatment 440.0 -666.0 -0.24 560.0 -287.0 -0.22 -0.3229 -0.9994 3118703 ChemDiv3_006350 COc1ccc(cc1)C2(CCOCC2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A15 compound treatment 600.0 -506.0 -0.18 640.0 -207.0 -0.16 -0.2393 -0.9981 3118704 ChemDiv3_006351 Cc1cc(nc(SCCNC(=O)Cc2ccc(F)cc2)n1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A16 compound treatment 400.0 -706.0 -0.25 320.0 -527.0 -0.4 -0.4632 -0.9735 3025950 ChemDiv3_006352 CCOC(=O)c1ccc(NC(=O)CCC(C)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A17 compound treatment 240.0 -866.0 -0.31 280.0 -567.0 -0.44 -0.525 -0.9855 3118705 ChemDiv3_006353 COc1cccc(NC(=O)C(C)Sc2nc(cc(n2)C(F)(F)F)c3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A18 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 1220163 ChemDiv3_006354 COc1cc2c(C(=O)N3CCN(CC3)c4ccccc4C)c(C)oc2cc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A19 compound treatment 1200.0 93.8 0.03 400.0 -447.0 -0.34 -0.2191 -0.6356 3118706 ChemDiv3_006355 CC1Cc2ccccc2N1C(=O)CSc3nc(cc(n3)C(F)(F)F)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A20 compound treatment 3320.0 2210.0 0.79 360.0 -487.0 -0.37 0.291 0.3346 3118707 ChemDiv3_006356 Cc1ccc(Sc2c(CS(=O)(=O)c3ccccc3)[nH]c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A21 compound treatment 480.0 -626.0 -0.22 400.0 -447.0 -0.34 -0.3997 -0.9779 3025951 ChemDiv3_006357 COc1ccc(cc1)c2cc(nc(SCCC(=O)N3CCCC3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A22 compound treatment 400.0 -706.0 -0.25 760.0 -86.9 -0.07 -0.2243 -0.8652 3118708 ChemDiv3_006358 O=C(c1ccncc1)n2nc3-c4ccccc4C(=O)c5cccc2c35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A23 mock treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 A24 mock treatment 480.0 -626.0 -0.22 280.0 -567.0 -0.44 -0.4648 -0.9513 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B01 compound treatment 360.0 -746.0 -0.26 480.0 -367.0 -0.28 -0.3864 -0.9995 3025952 ChemDiv3_006359 CCC(=O)n1nc(nc1SC)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B02 compound treatment 280.0 -826.0 -0.29 400.0 -447.0 -0.34 -0.4499 -0.9969 3118709 ChemDiv3_006360 CN1C(=O)/C(=C/c2ccc(o2)c3ccc(cc3)C(=O)O)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B03 compound treatment 400.0 -706.0 -0.25 320.0 -527.0 -0.4 -0.4632 -0.9735 3025953 ChemDiv3_006361 Nc1nc2ccccc2n1C(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B04 compound treatment 360.0 -746.0 -0.26 240.0 -607.0 -0.47 -0.5167 -0.9641 1713239 ChemDiv3_006362 NCCC(=O)N1c2ccccc2Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B05 compound treatment 280.0 -826.0 -0.29 240.0 -607.0 -0.47 -0.5367 -0.975 3118710 ChemDiv3_006363 CCC1(C2c3cc(Br)ccc3OC(=O)C21C(=O)c4ccco4)C(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B06 compound treatment 400.0 -706.0 -0.25 440.0 -407.0 -0.31 -0.398 -0.994 3118711 ChemDiv3_006364 Cc1cccc(C)c1NC(=O)Cn2c(nc3ccccc23)S(=O)(=O)CC(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B07 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3025954 ChemDiv3_006365 COc1ccc(cc1)c2c/c(=N\c3ccc(OC)c(OC)c3)/c4ccccc4o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B08 compound treatment 800.0 -306.0 -0.11 280.0 -567.0 -0.44 -0.3846 -0.8573 3118712 ChemDiv3_006366 FC(F)(F)c1ccccc1NC(=O)Cn2cc(C(=O)c3cccs3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B09 compound treatment 320.0 -786.0 -0.28 400.0 -447.0 -0.34 -0.4398 -0.9947 3026005 ChemDiv3_006367 C=CCOc1nnc(OCC=C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B10 compound treatment 320.0 -786.0 -0.28 520.0 -327.0 -0.25 -0.3747 -0.9986 3026006 ChemDiv3_006368 Cc1cc(Oc2ccccc2)nc(SCc3ccccc3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B11 compound treatment 320.0 -786.0 -0.28 440.0 -407.0 -0.31 -0.4181 -0.9984 3118713 ChemDiv3_006369 Nn1c(=O)c2ccccc2n3c(SCC(=O)N(c4ccccc4)c5ccccc5)nnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B12 compound treatment 640.0 -466.0 -0.17 320.0 -527.0 -0.4 -0.403 -0.9221 3026007 ChemDiv3_006370 COc1ccccc1CN2CCCC(C2)C(=O)N(C)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B13 compound treatment 1440.0 334.0 0.12 520.0 -327.0 -0.25 -0.0937 -0.3378 3118714 ChemDiv3_006371 O=S(=O)(/N=C(/Nc1cc(ncn1)N2CCOCC2)\c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B14 compound treatment 720.0 -386.0 -0.14 280.0 -567.0 -0.44 -0.4046 -0.8868 3118715 ChemDiv3_006372 Cc1ccc(cc1)C(=O)Nc2nonc2NC(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B15 compound treatment 520.0 -586.0 -0.21 520.0 -327.0 -0.25 -0.3245 -0.9956 3026008 ChemDiv3_006373 CS(=O)(=O)Nc1nc2NC(=CC(c3ccccc3)n2n1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B16 compound treatment 760.0 -346.0 -0.12 280.0 -567.0 -0.44 -0.3946 -0.8726 1138557 ChemDiv3_006374 Nc1nonc1n2nnc(C(=O)O)c2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B17 compound treatment 440.0 -666.0 -0.24 240.0 -607.0 -0.47 -0.4966 -0.9505 3026009 ChemDiv3_006375 CCOC=C1C(=O)c2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B18 compound treatment 400.0 -706.0 -0.25 320.0 -527.0 -0.4 -0.4632 -0.9735 3118716 ChemDiv3_006376 COc1cccc2c3nc(nc(NC(=O)C)c3c(=O)oc12)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B19 compound treatment 360.0 -746.0 -0.26 320.0 -527.0 -0.4 -0.4732 -0.9789 1327186 ChemDiv3_006377 CCCc1nnc(NC(=O)C(CC)Sc2nnc3c4ccccc4[nH]c3n2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B20 compound treatment 360.0 -746.0 -0.26 240.0 -607.0 -0.47 -0.5167 -0.9641 3026010 ChemDiv3_006378 CC(C)(C)c1ccc2OCN(Cc2c1)c3cccc(c3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B21 compound treatment 240.0 -866.0 -0.31 4360.0 3510.0 2.7 1.6898 0.6225 3118717 ChemDiv3_006379 CCOC(=O)Cc1cc(sc1c2ccc(OC)cc2)C(=O)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B22 compound treatment 520.0 -586.0 -0.21 320.0 -527.0 -0.4 -0.4331 -0.9522 3026011 ChemDiv3_006380 Cc1ccc2NC(=O)/C(=C/3\SC(=O)N(CC(=O)O)C3=O)/c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B23 mock treatment 3880.0 2770.0 0.98 280.0 -567.0 -0.44 0.388 0.3606 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 B24 mock treatment 1560.0 454.0 0.16 200.0 -647.0 -0.5 -0.2374 -0.4546 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C01 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3118718 ChemDiv3_006381 Cn1nc(c2ccc(OCC(=O)N3CCN(Cc4ccccc4)CC3)cc2)c5ccccc5c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C02 compound treatment 280.0 -826.0 -0.29 360.0 -487.0 -0.37 -0.4716 -0.9928 3026012 ChemDiv3_006382 CN(C)S(=O)(=O)N1CCN(CC1)S(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C03 compound treatment 280.0 -826.0 -0.29 200.0 -647.0 -0.5 -0.5584 -0.9684 3118719 ChemDiv3_006383 CCNc1nc(Oc2ccc(O)nn2)nc(n1)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C04 compound treatment 400.0 -706.0 -0.25 360.0 -487.0 -0.37 -0.4415 -0.9811 3026013 ChemDiv3_006384 Clc1ccc(cc1)c2csc3nnc(SCC(=O)c4ccc5OCOc5c4)n23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C05 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3118720 ChemDiv3_006385 CCNc1nc(NCC)nc(n1)C(=O)OCCO 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C06 compound treatment 280.0 -826.0 -0.29 440.0 -407.0 -0.31 -0.4281 -0.9995 1634799 ChemDiv3_006386 CCc1c(oc2c(C)c3oc(=O)cc(C)c3cc12)C(=O)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C07 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3026014 ChemDiv3_006387 COC(=O)/C=C/1\NC2CCCCC2NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C08 compound treatment 360.0 -746.0 -0.26 240.0 -607.0 -0.47 -0.5167 -0.9641 3118855 ChemDiv3_006388 Clc1cccc(OCc2nc(C#N)c(o2)N3CCCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C09 compound treatment 280.0 -826.0 -0.29 360.0 -487.0 -0.37 -0.4716 -0.9928 3026015 ChemDiv3_006389 S=C(SCSc1nc2ccccc2s1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C10 compound treatment 280.0 -826.0 -0.29 480.0 -367.0 -0.28 -0.4064 -0.9998 3118856 ChemDiv3_006390 Cc1ccc(Nc2ccc(NCc3ccccc3)nn2)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C11 compound treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 3026016 ChemDiv3_006391 Cc1ccc(cc1C)N2NC(=O)/C(=N/O)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C12 compound treatment 400.0 -706.0 -0.25 360.0 -487.0 -0.37 -0.4415 -0.9811 3118857 ChemDiv3_006392 O=C/1Nc2ccccc2\C1=C/C3=Cc4ccccc4OC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C13 compound treatment 3920.0 2810.0 1.0 600.0 -247.0 -0.19 0.5718 0.5628 3026017 ChemDiv3_006393 COc1ccc(cc1)c2cc(nc(SCC(=O)N)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C14 compound treatment 4520.0 3410.0 1.21 360.0 -487.0 -0.37 0.592 0.4671 1220737 ChemDiv3_006394 CCOC(=O)c1c(c2ccccc2)n(Cc3ccccc3)c4ccc(O)c(CN(C)C)c14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C15 compound treatment 440.0 -666.0 -0.24 360.0 -487.0 -0.37 -0.4314 -0.9756 3026018 ChemDiv3_006395 CCOC(=O)CS(=O)(=O)c1nc(cc(n1)C(F)(F)F)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C16 compound treatment 1160.0 53.8 0.02 320.0 -527.0 -0.4 -0.2725 -0.673 3118858 ChemDiv3_006396 COC(=O)c1ccc(NC(=O)CC(CC(=O)O)c2ccccc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C17 compound treatment 880.0 -226.0 -0.08 280.0 -567.0 -0.44 -0.3645 -0.8236 3118859 ChemDiv3_006397 CCCNC(=O)CSc1nc(cc(n1)C(F)(F)F)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C18 compound treatment 360.0 -746.0 -0.26 320.0 -527.0 -0.4 -0.4732 -0.9789 1323060 ChemDiv3_006398 CC1CCN(Cc2c(O)ccc3occ(C(=O)c4ccccc4)c23)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C19 compound treatment 640.0 -466.0 -0.17 320.0 -527.0 -0.4 -0.403 -0.9221 3118860 ChemDiv3_006399 COC(=O)c1c(NC(=O)CSc2nc(cc(n2)C(F)(F)F)c3ccco3)sc4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C20 compound treatment 320.0 -786.0 -0.28 520.0 -327.0 -0.25 -0.3747 -0.9986 1256796 ChemDiv3_006400 O=c1[nH]c(CSc2ccccn2)nc3c4ccccc4oc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C21 compound treatment 240.0 -866.0 -0.31 520.0 -327.0 -0.25 -0.3948 -0.9949 3118861 ChemDiv3_006401 COc1ccc(cc1)c2cc(nc(SCCC(=O)NCCc3ccccc3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C22 compound treatment 280.0 -826.0 -0.29 680.0 -167.0 -0.13 -0.2979 -0.9311 3026019 ChemDiv3_006402 O=C(Cc1ccccc1)n2nc3-c4ccccc4C(=O)c5cccc2c35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C23 mock treatment 400.0 -706.0 -0.25 840.0 -6.9 -0.01 -0.1809 -0.7219 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 C24 mock treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D01 compound treatment 280.0 -826.0 -0.29 360.0 -487.0 -0.37 -0.4716 -0.9928 3118862 ChemDiv3_006403 CSc1nc(nn1C(=O)c2ccccc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D02 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3118863 ChemDiv3_006404 CN1C(=O)/C(=C/c2cn(Cc3ccccc3)c4ccccc24)/c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D03 compound treatment 440.0 -666.0 -0.24 320.0 -527.0 -0.4 -0.4532 -0.9673 1476567 ChemDiv3_006405 CCOc1ccc(NC(=O)CSC2=NCCS2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D04 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3118864 ChemDiv3_006406 CCOC(=O)C1=C(N)c2ccccc2CC1(C)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D05 compound treatment 240.0 -866.0 -0.31 360.0 -487.0 -0.37 -0.4816 -0.9953 3026020 ChemDiv3_006407 COC(=O)C(C)(C)C1C(C(=O)N2CCOCC2)C(=O)Oc3ccc(Br)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D06 compound treatment 480.0 -626.0 -0.22 360.0 -487.0 -0.37 -0.4214 -0.9691 3118865 ChemDiv3_006408 COC(=O)c1ccccc1NC(=O)CS(=O)(=O)c2nnnn2c3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D07 compound treatment 240.0 -866.0 -0.31 440.0 -407.0 -0.31 -0.4382 -1.0 3118866 ChemDiv3_006409 COc1ccc(OC)c(/N=c/2\cc(oc3ccccc23)c4ccc5OCOc5c4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D08 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3026021 ChemDiv3_006410 Cc1ccc(OCCn2cc(C(=O)c3ccccc3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D09 compound treatment 240.0 -866.0 -0.31 320.0 -527.0 -0.4 -0.5033 -0.9908 3118867 ChemDiv3_006411 Cc1cc(C)c(C#N)c(SCC(=O)Nc2nsc(n2)c3ccc(Cl)cc3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D10 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3026022 ChemDiv3_006412 Cc1cc(C)nc(n1)N2CC(=O)N(CCOc3ccc(Br)cc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D11 compound treatment 360.0 -746.0 -0.26 280.0 -567.0 -0.44 -0.4949 -0.9716 3026072 ChemDiv3_006413 Nn1c(=O)c2ccccc2n3c(SCC(=O)c4ccccc4)nnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D12 compound treatment 320.0 -786.0 -0.28 400.0 -447.0 -0.34 -0.4398 -0.9947 3118868 ChemDiv3_006414 O=C(NCn1nnc(n1)c2ccncc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D13 compound treatment 2680.0 1570.0 0.56 360.0 -487.0 -0.37 0.1304 0.1942 3026073 ChemDiv3_006415 CCOC(=O)NC1(Nc2ccccc2Cl)Oc3ccccc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D14 compound treatment 800.0 -306.0 -0.11 320.0 -527.0 -0.4 -0.3629 -0.8663 3118869 ChemDiv3_006416 O=C(COc1ccccc1)Nc2nonc2NC(=O)COc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D15 compound treatment 400.0 -706.0 -0.25 360.0 -487.0 -0.37 -0.4415 -0.9811 3118870 ChemDiv3_006417 NS(=O)(=O)c1ccc(cc1)S(=O)(=O)NCCc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D16 compound treatment 920.0 -186.0 -0.07 480.0 -367.0 -0.28 -0.2459 -0.8499 3026074 ChemDiv3_006418 OC(=O)CC(c1ccccc1)c2cc(Cl)ccc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D17 compound treatment 15400.0 14300.0 5.07 5360.0 4510.0 3.46 6.0355 0.9828 1472447 ChemDiv3_006419 OC1(NC(=O)c2ccccc2)C(=O)c3ccccc3C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D18 compound treatment 520.0 -586.0 -0.21 280.0 -567.0 -0.44 -0.4548 -0.9429 3118871 ChemDiv3_006420 O=C1CSC2(N1c3ccccc3)C(=O)N(CN4CCCCC4)c5ccccc52 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D19 compound treatment 480.0 -626.0 -0.22 320.0 -527.0 -0.4 -0.4431 -0.9602 3026075 ChemDiv3_006421 CCCSc1nnc2c3ccccc3n(CC)c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D20 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 1015796 ChemDiv3_006422 CC(C)(C)c1ccc2OCN(Cc2c1)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D21 compound treatment 1320.0 214.0 0.08 240.0 -607.0 -0.47 -0.2758 -0.5843 3118872 ChemDiv3_006423 CCOc1ccc(NC(=O)c2sc(C)c(CC(=O)Nc3ccc(Cl)cc3)c2O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D22 compound treatment 400.0 -706.0 -0.25 360.0 -487.0 -0.37 -0.4415 -0.9811 3118873 ChemDiv3_006424 OC(=O)CC12CSc3[nH]c(=O)sc3C2c4ccccc4OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D23 mock treatment 400.0 -706.0 -0.25 3040.0 2190.0 1.68 1.0134 0.5953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 D24 mock treatment 2320.0 1210.0 0.43 560.0 -287.0 -0.22 0.1487 0.3075 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E01 compound treatment 320.0 -786.0 -0.28 1080.0 233.0 0.18 -0.0707 -0.2133 3026076 ChemDiv3_006425 CN(CCO)C(=O)c1ccc(cc1)c2nn(C)c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E02 compound treatment 320.0 -786.0 -0.28 520.0 -327.0 -0.25 -0.3747 -0.9986 3118874 ChemDiv3_006426 CN(C(=O)N1CCN(CC1)c2ccccn2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E03 compound treatment 2000.0 894.0 0.32 3320.0 2470.0 1.9 1.5667 0.8139 3026077 ChemDiv3_006427 CCOc1ccc(Oc2nc(NCC(C)C)nc(OC)n2)nn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E04 compound treatment 640.0 -466.0 -0.17 360.0 -487.0 -0.37 -0.3813 -0.9328 3118875 ChemDiv3_006428 Cc1ccccc1C2C3=C(Nc4c2c(=O)n(C)c(=O)n4C)c5ccccc5C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E05 compound treatment 320.0 -786.0 -0.28 920.0 73.1 0.06 -0.1575 -0.5537 3026078 ChemDiv3_006429 CC(C)(C)Nc1nc(nc(n1)C(=O)O)N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E06 compound treatment 1640.0 534.0 0.19 880.0 33.1 0.03 0.1519 0.7949 3118876 ChemDiv3_006430 CCC(=O)c1cc2c(C)cc(=O)oc2c(C)c1C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E07 compound treatment 440.0 -666.0 -0.24 2080.0 1230.0 0.95 0.5023 0.5148 3118877 ChemDiv3_006431 O=C(CSc1nn(c2ccccc2)c(=S)s1)N3N=CCC3c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E08 compound treatment 280.0 -826.0 -0.29 560.0 -287.0 -0.22 -0.363 -0.9901 3026079 ChemDiv3_006432 CC1CN(CC(C)O1)c2oc(COc3ccc(C)cc3)nc2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E09 compound treatment 1040.0 -66.3 -0.02 1560.0 713.0 0.55 0.3705 0.6761 3118878 ChemDiv3_006433 CCOC(=O)c1cnc(SCSc2nc3ccccc3s2)nc1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E10 compound treatment 2000.0 894.0 0.32 320.0 -527.0 -0.4 -0.0618 -0.1203 3026080 ChemDiv3_006434 CC(=O)Nc1ccc(cc1)c2cn3cccc(C)c3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E11 compound treatment 520.0 -586.0 -0.21 800.0 -46.9 -0.04 -0.1725 -0.8174 1483046 ChemDiv3_006435 CC(C)OC(=O)c1ccc2[nH]c3CCCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E12 compound treatment 2960.0 1850.0 0.66 4920.0 4070.0 3.13 2.6761 0.8375 3118879 ChemDiv3_006436 O=C(Cn1cc(/C=C\2/C(=O)Nc3ccccc23)c4ccccc14)N5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E13 compound treatment 760.0 -346.0 -0.12 1440.0 593.0 0.46 0.2351 0.4985 3026081 ChemDiv3_006437 CCOC(=O)CSc1nc(cc(n1)C(F)(F)F)c2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E14 compound treatment 760.0 -346.0 -0.12 920.0 73.1 0.06 -0.0472 -0.3493 3026082 ChemDiv3_006438 CCOc1ccc(c2ccccc12)S(=O)(=O)n3ccc(C)n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E15 compound treatment 760.0 -346.0 -0.12 1080.0 233.0 0.18 0.0397 0.1828 3118880 ChemDiv3_006439 CCOC(=O)CS(=O)c1nc(c2CCc3ccccc3-c2n1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E16 compound treatment 520.0 -586.0 -0.21 720.0 -127.0 -0.1 -0.2159 -0.9403 3118998 ChemDiv3_006440 OC(=O)c1ccc(NC(=O)C2CC(=O)OC2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E17 compound treatment 840.0 -266.0 -0.09 4000.0 3150.0 2.42 1.6449 0.679 3026083 ChemDiv3_006441 CN(C(=O)CSc1nc(cc(n1)C(F)(F)F)c2cccs2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E18 compound treatment 3600.0 2490.0 0.88 2360.0 1510.0 1.16 1.4469 0.991 3118999 ChemDiv3_006442 CCCCN1CCc2c(C1)c3ccccc3n2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E19 compound treatment 760.0 -346.0 -0.12 1520.0 673.0 0.52 0.2785 0.5244 3119000 ChemDiv3_006443 FC(F)(F)C1CC(Nc2cc(nn12)C(=O)N3CCCCC3)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E20 compound treatment 1640.0 534.0 0.19 1680.0 833.0 0.64 0.5861 0.8787 3026084 ChemDiv3_006444 COc1cccc(OC)c1C2=NCC(=O)Nc3c2oc4ccc(Br)cc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E21 compound treatment 1240.0 134.0 0.05 560.0 -287.0 -0.22 -0.1222 -0.5423 3119001 ChemDiv3_006445 COc1ccc(cc1)c2cc(nc(SCCC(=O)N(C)Cc3ccccc3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E22 compound treatment 1520.0 414.0 0.15 240.0 -607.0 -0.47 -0.2257 -0.462 3025905 ChemDiv3_006446 O=C(c1ccco1)n2nc3-c4ccccc4C(=O)c5cccc2c35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E23 mock treatment 960.0 -146.0 -0.05 2160.0 1310.0 1.01 0.6761 0.6698 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 E24 mock treatment 840.0 -266.0 -0.09 6080.0 5230.0 4.02 2.7741 0.6903 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F01 compound treatment 720.0 -386.0 -0.14 1200.0 353.0 0.27 0.0948 0.3121 3119002 ChemDiv3_006447 CSc1nc(nn1S(=O)(=O)C)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F02 compound treatment 760.0 -346.0 -0.12 5040.0 4190.0 3.22 2.1894 0.6796 3119003 ChemDiv3_006448 CCN(CC)C(=O)Cn1cc(/C=C\2/C(=O)N(C)c3ccccc23)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F03 compound treatment 1240.0 134.0 0.05 1320.0 473.0 0.36 0.2904 0.7927 3025907 ChemDiv3_006449 FC(F)(F)c1ccccc1NC(=O)CSC2=NCCS2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F04 compound treatment 1560.0 454.0 0.16 1040.0 193.0 0.15 0.2186 0.9992 3119004 ChemDiv3_006450 O=C(C1CN2C(=C(C1)C(=O)c3ccccc3)Sc4ccccc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F05 compound treatment 960.0 -146.0 -0.05 5000.0 4150.0 3.19 2.2179 0.6955 3025910 ChemDiv3_006451 CC(C1C(C(=O)c2ccccc2)C(=O)Oc3ccc(Br)cc13)C(=O)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F06 compound treatment 1120.0 13.8 0.0 1480.0 633.0 0.49 0.3471 0.7142 3119005 ChemDiv3_006452 OC(=O)CSc1ncnc2scc(c3ccc(Br)cc3)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F07 compound treatment 1040.0 -66.3 -0.02 4120.0 3270.0 2.51 1.7602 0.7005 3119006 ChemDiv3_006453 Nc1ccccc1/N=c/2\cc(oc3ccccc23)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F08 compound treatment 440.0 -666.0 -0.24 3040.0 2190.0 1.68 1.0234 0.6019 3025912 ChemDiv3_006454 Fc1ccc(Cn2cc(C(=O)c3ccccc3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F09 compound treatment 2040.0 934.0 0.33 2480.0 1630.0 1.25 1.1208 0.8643 3119007 ChemDiv3_006455 Cc1ccc(C)c(c1)S(=O)(=O)NCC(=O)Nc2nsc(n2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F10 compound treatment 680.0 -426.0 -0.15 1400.0 553.0 0.42 0.1933 0.4289 3025914 ChemDiv3_006456 CSc1nc(C)cc(OCC(=O)N2CCCCC2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F11 compound treatment 720.0 -386.0 -0.14 4840.0 3990.0 3.07 2.0708 0.6748 3119008 ChemDiv3_006457 CC(=O)Nc1sc-2c(CCc3ccccc23)c1C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F12 compound treatment 1080.0 -26.3 -0.01 6320.0 5470.0 4.2 2.9645 0.7055 3025917 ChemDiv3_006458 Clc1ccc(cc1)N(CCOC(=O)c2cccs2)C3=NS(=O)(=O)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F13 compound treatment 600.0 -506.0 -0.18 1600.0 753.0 0.58 0.2818 0.4655 3119009 ChemDiv3_006459 FC(F)(F)C1(NS(=O)(=O)c2ccccc2)OCCO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F14 compound treatment 640.0 -466.0 -0.17 6360.0 5510.0 4.23 2.8759 0.679 3119010 ChemDiv3_006460 COc1ccc(cc1)C(=O)Nc2nonc2NC(=O)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F15 compound treatment 1240.0 134.0 0.05 840.0 -6.9 -0.01 0.0298 0.6243 3025920 ChemDiv3_006461 COc1ccc(NC(=O)C2CCCN2c3cccc(c3)C(F)(F)F)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F16 compound treatment 560.0 -546.0 -0.19 480.0 -367.0 -0.28 -0.3362 -0.9833 3119011 ChemDiv3_006462 COc1cc2CCN(CCC(=O)N)C(C)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F17 compound treatment 600.0 -506.0 -0.18 1440.0 593.0 0.46 0.195 0.3984 3119012 ChemDiv3_006463 CCC(N)CC1(CC2CC3CC(C2)C1)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F18 compound treatment 1120.0 13.8 0.0 960.0 113.0 0.09 0.0648 0.7457 1787529 ChemDiv3_006464 COc1ccc(OC)c(c1)c2nc(Nc3ccccc3F)sc2CC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F19 compound treatment 720.0 -386.0 -0.14 1280.0 433.0 0.33 0.1382 0.3844 1696294 ChemDiv3_006465 CCC(Sc1nnc2c3ccccc3n(CC)c2n1)C(=O)NC(C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F20 compound treatment 1880.0 774.0 0.27 4360.0 3510.0 2.7 2.1012 0.7751 3025978 ChemDiv3_006466 CC(C)(C)N1COc2ccc(cc2C1)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F21 compound treatment 4160.0 3050.0 1.08 1760.0 913.0 0.7 1.2617 0.9778 3119013 ChemDiv3_006467 Clc1ccc(Nc2nnns2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F22 compound treatment 2720.0 1610.0 0.57 600.0 -247.0 -0.19 0.2708 0.449 3119014 ChemDiv3_006468 CCC(C)c1ccc(OCCCN2CCN(C)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F23 mock treatment 1760.0 654.0 0.23 1640.0 793.0 0.61 0.5945 0.9125 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 F24 mock treatment 400.0 -706.0 -0.25 5360.0 4510.0 3.46 2.2728 0.6543 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G01 compound treatment 5040.0 3930.0 1.4 1120.0 273.0 0.21 1.135 0.8043 3025980 ChemDiv3_006469 Cn1nc(c2ccc(cc2)C(=O)NCC3CCCO3)c4ccccc4c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G02 compound treatment 360.0 -746.0 -0.26 680.0 -167.0 -0.13 -0.2778 -0.9445 3119015 ChemDiv3_006470 Cc1ccc(cc1)C(=O)CC(C(=O)O)n2cccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G03 compound treatment 400.0 -706.0 -0.25 480.0 -367.0 -0.28 -0.3763 -0.9983 3119016 ChemDiv3_006471 C(Cn1c2ccccc2c3nc4ccccc4nc13)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G04 compound treatment 1080.0 -26.3 -0.01 680.0 -167.0 -0.13 -0.0972 -0.7565 3025983 ChemDiv3_006472 CCn1c2NC3=C(C(c4ccsc4)c2c(=O)[nH]c1=O)C(=O)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G05 compound treatment 1880.0 774.0 0.27 880.0 33.1 0.03 0.2121 0.7693 3119017 ChemDiv3_006473 CCNc1cc(nc(Oc2ccc(OCCOc3ccccc3C)nn2)n1)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G06 compound treatment 1080.0 -26.3 -0.01 400.0 -447.0 -0.34 -0.2492 -0.726 3119018 ChemDiv3_006474 CCc1c(oc2ccc3c(C)cc(=O)oc3c12)C(C)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G07 compound treatment 800.0 -306.0 -0.11 1160.0 313.0 0.24 0.0932 0.3531 3025986 ChemDiv3_006475 Cc1ccnc(SCC(=O)N2N=CCC2c3ccccc3)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G08 compound treatment 480.0 -626.0 -0.22 1960.0 1110.0 0.85 0.4472 0.5064 3026041 ChemDiv3_006476 CN(C)CCNc1oc(COc2ccc(C)cc2)nc1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G09 compound treatment 2360.0 1250.0 0.44 1160.0 313.0 0.24 0.4845 0.9583 3119019 ChemDiv3_006477 COC(=O)/C=c\1/sc2=NC(C)(C)C=C(C)n2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G10 compound treatment 520.0 -586.0 -0.21 1440.0 593.0 0.46 0.1749 0.3494 3026044 ChemDiv3_006478 CC(=O)NCCSc1nc(cc(c1C#N)c2ccc(F)cc2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G11 compound treatment 1040.0 -66.3 -0.02 520.0 -327.0 -0.25 -0.1941 -0.77 3119020 ChemDiv3_006479 FC(F)(F)c1nn(CC(=O)N(Cc2ccccc2)Cc3ccccc3)c4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G12 compound treatment 1280.0 174.0 0.06 4560.0 3710.0 2.85 2.0593 0.7222 3119021 ChemDiv3_006480 CC1CCCC(C)N1C(=O)Cn2cc(/C=C\3/C(=O)N(C)c4ccccc34)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G13 compound treatment 440.0 -666.0 -0.24 560.0 -287.0 -0.22 -0.3229 -0.9994 3026047 ChemDiv3_006481 COc1ccc(cc1)c2cc(nc(SCC(=O)N(C)C3CCCCC3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G14 compound treatment 1360.0 254.0 0.09 720.0 -127.0 -0.1 -0.0052 -0.0395 3119022 ChemDiv3_006482 CCc1ccc(cc1)n2cc3C(=O)CC(C)(C)Cc3c(C#N)c2=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G15 compound treatment 4680.0 3570.0 1.27 480.0 -367.0 -0.28 0.6973 0.5369 3026050 ChemDiv3_006483 CC(Sc1nc(cc(n1)C(F)(F)F)c2ccccc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G16 compound treatment 400.0 -706.0 -0.25 680.0 -167.0 -0.13 -0.2678 -0.9515 3119023 ChemDiv3_006484 CC1(C)CC(CCc2nnc(S)[nH]2)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G17 compound treatment 1280.0 174.0 0.06 1920.0 1070.0 0.82 0.6261 0.7579 3119024 ChemDiv3_006485 FC(F)(F)c1cc(nc(SCC(=O)NCc2ccncc2)n1)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G18 compound treatment 560.0 -546.0 -0.19 760.0 -86.9 -0.07 -0.1842 -0.8988 3026052 ChemDiv3_006486 CCOC(=O)c1oc2ccccc2c1CN3CCN(CC3)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G19 compound treatment 360.0 -746.0 -0.26 560.0 -287.0 -0.22 -0.3429 -0.9958 3119025 ChemDiv3_006487 CC(C)CNC(=O)c1cc2NC(CC(n2n1)C(F)(F)F)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G20 compound treatment 2360.0 1250.0 0.44 1760.0 913.0 0.7 0.8102 0.9759 3026055 ChemDiv3_006488 Cc1cc(C)nc(SCCc2ccncc2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G21 compound treatment 520.0 -586.0 -0.21 1880.0 1030.0 0.79 0.4138 0.5046 3119026 ChemDiv3_006489 COc1ccc(cc1)c2cc(nc(SCCC(=O)N(C)c3ccccc3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G22 compound treatment 2840.0 1730.0 0.62 960.0 113.0 0.09 0.4963 0.799 3026105 ChemDiv3_006490 O=C(C1CCCCC1)n2nc3-c4ccccc4C(=O)c5cccc2c35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G23 mock treatment 1000.0 -106.0 -0.04 920.0 73.1 0.06 0.013 0.1928 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 G24 mock treatment 1440.0 334.0 0.12 800.0 -46.9 -0.04 0.0583 0.4708 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H01 compound treatment 800.0 -306.0 -0.11 600.0 -247.0 -0.19 -0.2109 -0.9651 3119150 ChemDiv3_006491 CSc1nc(nn1S(=O)(=O)c2ccc(Cl)cc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H02 compound treatment 560.0 -546.0 -0.19 440.0 -407.0 -0.31 -0.3579 -0.9736 3119151 ChemDiv3_006492 CCc1cccc2c(/C=C\3/C(=O)N(C)c4ccccc34)cn(CC(=O)NC5CCCC5)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H03 compound treatment 440.0 -666.0 -0.24 1600.0 753.0 0.58 0.2417 0.387 3026108 ChemDiv3_006493 O=C(CSC1=NCCS1)N2CCN(CC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H04 compound treatment 640.0 -466.0 -0.17 480.0 -367.0 -0.28 -0.3161 -0.9678 3026109 ChemDiv3_006494 CC(CN(C)Cc1ccccc1)OC(=O)c2cc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H05 compound treatment 560.0 -546.0 -0.19 1760.0 913.0 0.7 0.3587 0.4931 3119152 ChemDiv3_006495 CC1(C2c3cc(Br)ccc3OC(=O)C21C(=O)N4CCCCC4)C(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H06 compound treatment 560.0 -546.0 -0.19 2160.0 1310.0 1.01 0.5758 0.5609 1700700 ChemDiv3_006496 CC(C(=O)O)n1cnc2scc(c3ccc(Cl)cc3)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H07 compound treatment 1080.0 -26.3 -0.01 4280.0 3430.0 2.64 1.8571 0.7046 3119153 ChemDiv3_006497 Cc1cc2c3c(C)n(C4CCCCC4)c(C)c3c(C)nn2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H08 compound treatment 2200.0 1090.0 0.39 720.0 -127.0 -0.1 0.2055 0.5136 3119154 ChemDiv3_006498 O=C(c1cn(CCCOc2ccccc2)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H09 compound treatment 1000.0 -106.0 -0.04 400.0 -447.0 -0.34 -0.2693 -0.7801 3026112 ChemDiv3_006499 CCC(C)c1ccc(OCC(=O)Nc2cccc(c3nc4ncccc4o3)c2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H10 compound treatment 320.0 -786.0 -0.28 440.0 -407.0 -0.31 -0.4181 -0.9984 3119155 ChemDiv3_006500 COc1ccc(cc1OC)c2nc3ccccc3n2C(=O)c4ccccc4C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H11 compound treatment 400.0 -706.0 -0.25 1040.0 193.0 0.15 -0.0723 -0.2485 3119156 ChemDiv3_006501 Cn1cc(C2CC(=O)N(C2=O)c3ccc(Br)cc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H12 compound treatment 840.0 -266.0 -0.09 720.0 -127.0 -0.1 -0.1357 -0.9999 3026114 ChemDiv3_006502 FC(F)(F)c1cccc(c1)c2ccc(o2)c3nn4c(nnc4s3)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H13 compound treatment 3000.0 1890.0 0.67 440.0 -407.0 -0.31 0.2541 0.343 3119157 ChemDiv3_006503 COC(=O)c1ccc(NC(=O)NC(=O)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H14 compound treatment 320.0 -786.0 -0.28 920.0 73.1 0.06 -0.1575 -0.5537 3026116 ChemDiv3_006504 Clc1cccc(Cl)c1COC(=O)CCc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H15 compound treatment 440.0 -666.0 -0.24 480.0 -367.0 -0.28 -0.3663 -0.9962 3119158 ChemDiv3_006505 Cc1cc(C)c(N2CCCC2C(=O)Nc3cccc(c3)C(F)(F)F)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H16 compound treatment 2440.0 1330.0 0.47 2480.0 1630.0 1.25 1.2211 0.9112 1253000 ChemDiv3_006506 OC(=O)Cn1cnc(c1)c2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H17 compound treatment 680.0 -426.0 -0.15 6120.0 5270.0 4.05 2.7556 0.6802 3119159 ChemDiv3_006507 CC(C)(CN)C1(CC2CC3CC(C2)C1)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H18 compound treatment 680.0 -426.0 -0.15 1040.0 193.0 0.15 -0.0021 -0.0099 3026118 ChemDiv3_006508 COc1ccc2-c3nc(NC(=O)c4ccc(OC)c(Br)c4)sc3Cc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H19 compound treatment 1240.0 134.0 0.05 960.0 113.0 0.09 0.0949 0.9596 3119160 ChemDiv3_006509 CCCn1c2ccccc2c3nnc(SC(CC)C(=O)Nc4nc(C)c(s4)C(=O)OCC)nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H20 compound treatment 680.0 -426.0 -0.15 800.0 -46.9 -0.04 -0.1324 -0.8517 3119161 ChemDiv3_006510 CC(=O)Nc1ccc(cc1)N2COc3ccc(NC(=O)C)cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H21 compound treatment 680.0 -426.0 -0.15 800.0 -46.9 -0.04 -0.1324 -0.8517 3026188 ChemDiv3_006511 Cc1ccc(Nc2nnns2)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H22 compound treatment 400.0 -706.0 -0.25 480.0 -367.0 -0.28 -0.3763 -0.9983 3026189 ChemDiv3_006512 Cc1ccc(OCCn2ncc3ccccc3c2=O)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H23 mock treatment 400.0 -706.0 -0.25 2560.0 1710.0 1.32 0.7528 0.5623 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 H24 mock treatment 5560.0 4450.0 1.58 3880.0 3030.0 2.33 2.7637 0.9821 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I01 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3119162 ChemDiv3_006513 CC1CCN(CC1)C(=O)c2ccc(cc2)c3nn(C)c(=O)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I02 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3026192 ChemDiv3_006514 COc1ccc(cc1)c2c(C#N)c(SCC(=O)c3ccccc3)nc4CC(C)(C)CC(=O)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I03 compound treatment 360.0 -746.0 -0.26 360.0 -487.0 -0.37 -0.4515 -0.9857 3119163 ChemDiv3_006515 CCCn1c2ccc(CC)cc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I04 compound treatment 320.0 -786.0 -0.28 240.0 -607.0 -0.47 -0.5267 -0.9699 3119164 ChemDiv3_006516 CCC(=O)c1ccc(N2CCN(CC2)C(=O)c3ccco3)c(F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I05 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3026195 ChemDiv3_006517 O=C(CN1C(=O)C2C3CC(C=C3)C2C1=O)Nc4ccc5ncccc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I06 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3119165 ChemDiv3_006518 CC(Nc1oc(COc2ccccc2C)nc1C#N)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I07 compound treatment 320.0 -786.0 -0.28 400.0 -447.0 -0.34 -0.4398 -0.9947 3119166 ChemDiv3_006519 O=C(NCc1ccccc1)C2CC(=O)NC(=N2)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I08 compound treatment 3320.0 2210.0 0.79 3680.0 2830.0 2.18 2.0933 0.9052 3026198 ChemDiv3_006520 COc1ccc(OCc2nc(C#N)c(o2)N3CCOCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I09 compound treatment 3000.0 1890.0 0.67 1000.0 153.0 0.12 0.5581 0.8184 3119167 ChemDiv3_006521 Cc1nc(NC2=NCN(Cc3ccccc3)CN2)nc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I10 compound treatment 520.0 -586.0 -0.21 200.0 -647.0 -0.5 -0.4982 -0.9254 3026200 ChemDiv3_006522 CC(C)Cn1c(=O)oc2ccc(C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I11 compound treatment 280.0 -826.0 -0.29 800.0 -46.9 -0.04 -0.2327 -0.788 3119168 ChemDiv3_006523 CN(C(=O)Cn1nc(c2CCCCc21)C(F)(F)F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I12 compound treatment 1080.0 -26.3 -0.01 280.0 -567.0 -0.44 -0.3143 -0.7221 3026203 ChemDiv3_006524 CN1C(=O)/C(=C/c2cn(CC(=O)N3CCCC3)c4ccccc24)/c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I13 compound treatment 360.0 -746.0 -0.26 1000.0 153.0 0.12 -0.1041 -0.3593 3119169 ChemDiv3_006525 COc1ccc(cc1)c2cc(nc(SCC(=O)N3CC4(C)CC3CC(C)(C)C4)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I14 compound treatment 360.0 -746.0 -0.26 280.0 -567.0 -0.44 -0.4949 -0.9716 3026268 ChemDiv3_006526 Cc1[nH]c2ccccc2c1Cc3n[nH]c(=S)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I15 compound treatment 320.0 -786.0 -0.28 760.0 -86.9 -0.07 -0.2444 -0.8522 3119170 ChemDiv3_006527 CC(Sc1nc(cc(n1)C(F)(F)F)c2ccccc2)C(=O)Nc3cc(C)on3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I16 compound treatment 480.0 -626.0 -0.22 360.0 -487.0 -0.37 -0.4214 -0.9691 3119171 ChemDiv3_006528 CC(CC1CC(C)(C)OC1=O)c2nnc(S)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I17 compound treatment 1280.0 174.0 0.06 480.0 -367.0 -0.28 -0.1556 -0.5396 3026271 ChemDiv3_006529 FC(F)(F)c1cc(nc(SCC(=O)N2CCSCC2)n1)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I18 compound treatment 4320.0 3210.0 1.14 440.0 -407.0 -0.31 0.5853 0.4951 3119172 ChemDiv3_006530 OC(=O)c1oc2ccc(Br)cc2c1n3cccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I19 compound treatment 1640.0 534.0 0.19 360.0 -487.0 -0.37 -0.1304 -0.3113 3119173 ChemDiv3_006531 FC(F)(F)C1CC(Nc2cc(nn12)C(=O)NCc3ccncc3)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I20 compound treatment 800.0 -306.0 -0.11 360.0 -487.0 -0.37 -0.3411 -0.8764 3026273 ChemDiv3_006532 COc1ccc2oc(C(=O)CCC(=O)O)c(N)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I21 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3119174 ChemDiv3_006533 COc1ccc(cc1)c2cc(nc(SCCC(=O)Nc3ccccc3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I22 compound treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 3026275 ChemDiv3_006534 CN(C)CCN1C(=O)C(=C(C(=O)c2ccc(C)cc2)C13C(=O)N(C)c4ccccc43)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I23 mock treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 I24 mock treatment 1000.0 -106.0 -0.04 320.0 -527.0 -0.4 -0.3127 -0.7697 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J01 compound treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 3119175 ChemDiv3_006535 CCS(=O)(=O)n1nc(nc1SC)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J02 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3026278 ChemDiv3_006536 CN1C(=O)/C(=C/c2cn(CC(=O)O)c3ccccc23)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J03 compound treatment 440.0 -666.0 -0.24 440.0 -407.0 -0.31 -0.388 -0.9905 3119176 ChemDiv3_006537 CC(Nc1nc(nc2ccccc12)N3CCNCC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J04 compound treatment 400.0 -706.0 -0.25 280.0 -567.0 -0.44 -0.4849 -0.9656 3119177 ChemDiv3_006538 CC(CN(C)Cc1ccccc1)OC(=O)C2COc3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J05 compound treatment 360.0 -746.0 -0.26 360.0 -487.0 -0.37 -0.4515 -0.9857 3026280 ChemDiv3_006539 OC1(C(OC(=O)C21CCCCC2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J06 compound treatment 280.0 -826.0 -0.29 240.0 -607.0 -0.47 -0.5367 -0.975 3119178 ChemDiv3_006540 Cc1ccc(OCCn2cc(/C=C\3/C(=O)Nc4cc(Cl)ccc34)c5ccccc25)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J07 compound treatment 280.0 -826.0 -0.29 600.0 -247.0 -0.19 -0.3413 -0.9777 3026350 ChemDiv3_006541 CCOc1ccc(cc1)C2C(=C(N)Oc3c2ccc(=O)c4c(C)oc(C)c34)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J08 compound treatment 480.0 -626.0 -0.22 280.0 -567.0 -0.44 -0.4648 -0.9513 3119295 ChemDiv3_006542 CC1CCCCN1C(=O)Cn2cc(C(=O)c3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J09 compound treatment 2920.0 1810.0 0.64 320.0 -527.0 -0.4 0.1689 0.2223 3026352 ChemDiv3_006543 COc1ccc(C[N+](C)(C)C2CCCCC2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J10 compound treatment 400.0 -706.0 -0.25 320.0 -527.0 -0.4 -0.4632 -0.9735 3119296 ChemDiv3_006544 Cc1ccc(Cn2c(nc3ccccc23)C4CN(C(=O)C4)c5ccccc5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J11 compound treatment 320.0 -786.0 -0.28 440.0 -407.0 -0.31 -0.4181 -0.9984 1183983 ChemDiv3_006545 CC1(CN2CC3(C)CN(C1)C2c4ccccc4)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J12 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 3119297 ChemDiv3_006546 Clc1ccc(cc1)S(=O)(=O)NC2CCCCC2SC3=NCCS3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J13 compound treatment 320.0 -786.0 -0.28 560.0 -287.0 -0.22 -0.353 -0.9932 3119298 ChemDiv3_006547 CC(C)C1CCC(C)CC1OC(=O)NC(=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J14 compound treatment 320.0 -786.0 -0.28 400.0 -447.0 -0.34 -0.4398 -0.9947 3026356 ChemDiv3_006548 CCc1ccc(cc1)C2N(C(=O)c3oc4ccccc4c(=O)c23)c5ccccn5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J15 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 1556642 ChemDiv3_006549 OC(=O)CCC(=O)N1CCN(CC1)c2nc(c3ccccc3)c4cc(Br)ccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J16 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3026357 ChemDiv3_006550 CCCN(CCC)Cc1c(nnn1c2nonc2N)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J17 compound treatment 800.0 -306.0 -0.11 840.0 -6.9 -0.01 -0.0806 -0.7407 1720359 ChemDiv3_006551 Cc1c(CCNS(=O)(=O)c2ccc(Br)cc2)c3ccccc3n1Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J18 compound treatment 760.0 -346.0 -0.12 280.0 -567.0 -0.44 -0.3946 -0.8726 3119299 ChemDiv3_006552 COc1ccc2-c3nc(NC(=O)c4cc(OC)c(OC)c(OC)c4)sc3CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J19 compound treatment 1040.0 -66.3 -0.02 320.0 -527.0 -0.4 -0.3026 -0.7469 3026360 ChemDiv3_006553 Cc1c(NC(=O)CSc2ccccn2)c(=O)n(c3ccccc3)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J20 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 1032134 ChemDiv3_006554 Brc1ccc2OCN(Cc2c1)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J21 compound treatment 560.0 -546.0 -0.19 400.0 -447.0 -0.34 -0.3796 -0.9634 1787632 ChemDiv3_006555 Cc1ccc(cc1)c2nc(Nc3ccc(C)c(Cl)c3)sc2CC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J22 compound treatment 360.0 -746.0 -0.26 280.0 -567.0 -0.44 -0.4949 -0.9716 3025861 ChemDiv3_006556 CC1CCN(CCCOc2c(C)cccc2CC=C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J23 mock treatment 280.0 -826.0 -0.29 360.0 -487.0 -0.37 -0.4716 -0.9928 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 J24 mock treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K01 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3119300 ChemDiv3_006557 CCC(=O)N1CCN(CC1)c2nnc(c3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K02 compound treatment 2360.0 1250.0 0.44 1200.0 353.0 0.27 0.5062 0.9718 3025864 ChemDiv3_006558 CCc1c(C#N)c(SCC(=O)c2ccc3OCOc3c2)nc4CC(C)(C)CC(=O)c14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K03 compound treatment 480.0 -626.0 -0.22 3440.0 2590.0 1.99 1.2506 0.6243 3119301 ChemDiv3_006559 COc1ccc(CC(=O)n2nc(C)cc2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K04 compound treatment 520.0 -586.0 -0.21 1000.0 153.0 0.12 -0.0639 -0.2677 3119302 ChemDiv3_006560 COc1ccc(NC(=O)C(C)Oc2ccc3c(C)c(CCC(C)C)c(=O)oc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K05 compound treatment 480.0 -626.0 -0.22 480.0 -367.0 -0.28 -0.3563 -0.9931 3025867 ChemDiv3_006561 Cc1ccc(cc1)S(=O)(=O)/N=C(/Nc2nc(C)cc(C)n2)\N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K06 compound treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 3119303 ChemDiv3_006562 Fc1ccccc1OCc2nc(C#N)c(NCC=C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K07 compound treatment 280.0 -826.0 -0.29 2080.0 1230.0 0.95 0.4621 0.4663 3119304 ChemDiv3_006563 C(N1CNC(=NC1)Nc2nc3ccccc3o2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K08 compound treatment 480.0 -626.0 -0.22 840.0 -6.9 -0.01 -0.1608 -0.7238 3025924 ChemDiv3_006564 Cc1cccc(OCc2nc(C#N)c(NCCc3ccccc3)o2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K09 compound treatment 1440.0 334.0 0.12 520.0 -327.0 -0.25 -0.0937 -0.3378 3119305 ChemDiv3_006565 COC(=O)CC1N(CCNC1=O)C(=O)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K10 compound treatment 560.0 -546.0 -0.19 720.0 -127.0 -0.1 -0.2059 -0.9494 3119306 ChemDiv3_006566 CCOC(=O)Cn1c(=O)oc2ccc(C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K11 compound treatment 600.0 -506.0 -0.18 1080.0 233.0 0.18 -4.0E-4 -0.0018 3025928 ChemDiv3_006567 COc1cccc(c1)c2cc(n3ncc(C(=O)N(C)CCc4ccccn4)c3n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K12 compound treatment 1320.0 214.0 0.08 760.0 -86.9 -0.07 0.0064 0.0638 3119307 ChemDiv3_006568 COc1ccc(cc1)C(=O)Nc2ccc(cc2)c3nnc(S)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K13 compound treatment 320.0 -786.0 -0.28 1440.0 593.0 0.46 0.1247 0.2336 3119308 ChemDiv3_006569 CC(C)NC(=O)CSc1nc(cc(n1)C(F)(F)F)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K14 compound treatment 760.0 -346.0 -0.12 520.0 -327.0 -0.25 -0.2643 -0.946 3025932 ChemDiv3_006570 Cc1[nH]c2ccccc2c1Cc3nnc(SCC=C)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K15 compound treatment 600.0 -506.0 -0.18 1000.0 153.0 0.12 -0.0439 -0.2044 3119309 ChemDiv3_006571 CC(Sc1nc(cc(n1)C(F)(F)F)c2ccccc2)C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K16 compound treatment 480.0 -626.0 -0.22 600.0 -247.0 -0.19 -0.2911 -0.9969 3025934 ChemDiv3_006572 CC1CC(CCC(=O)Nc2ccc(cc2)S(=O)(=O)N)C(=O)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K17 compound treatment 560.0 -546.0 -0.19 640.0 -207.0 -0.16 -0.2493 -0.9951 3119310 ChemDiv3_006573 NC(=O)c1c(NC(=O)CSc2nc(cc(n2)C(F)(F)F)c3cccs3)sc4CCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K18 compound treatment 560.0 -546.0 -0.19 360.0 -487.0 -0.37 -0.4013 -0.9532 3025938 ChemDiv3_006574 COC(=O)CCC(=O)c1oc2ccc(OC)cc2c1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K19 compound treatment 520.0 -586.0 -0.21 1160.0 313.0 0.24 0.0229 0.0721 3119311 ChemDiv3_006575 COc1ccc(cc1OC)c2cc(nc(SCC(=O)N(C)Cc3cn(C)nc3C)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K20 compound treatment 560.0 -546.0 -0.19 1320.0 473.0 0.36 0.1198 0.291 3025991 ChemDiv3_006576 CCOC(=O)c1c(CSC(=N)N)n(c2ccccc2)c3cc(Br)c(OC(=O)C)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K21 compound treatment 640.0 -466.0 -0.17 920.0 73.1 0.06 -0.0773 -0.4424 3119312 ChemDiv3_006577 CCN1C(=O)c2ccc(cc2C1=O)c3nc4cc(Cl)ccc4c(=O)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K22 compound treatment 840.0 -266.0 -0.09 640.0 -207.0 -0.16 -0.1791 -0.9692 3025994 ChemDiv3_006578 COCCN1C(=O)C(=C(C(=O)c2ccccc2)C13C(=O)N(CC=C)c4ccccc43)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K23 mock treatment 5640.0 4530.0 1.61 440.0 -407.0 -0.31 0.9164 0.5593 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 K24 mock treatment 1040.0 -66.3 -0.02 640.0 -207.0 -0.16 -0.1289 -0.803 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L01 compound treatment 400.0 -706.0 -0.25 840.0 -6.9 -0.01 -0.1809 -0.7219 3119313 ChemDiv3_006579 Nc1nc(nn1S(=O)(=O)c2ccc(Cl)cc2)C(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L02 compound treatment 2680.0 1570.0 0.56 440.0 -407.0 -0.31 0.1739 0.2718 3119314 ChemDiv3_006580 CCn1cc(/C=C\2/C(=O)N(c3ccccc23)c4ccccc4)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L03 compound treatment 1680.0 574.0 0.2 3680.0 2830.0 2.18 1.6819 0.7699 3025997 ChemDiv3_006581 OC1=NC(Nc2sc3CCCCc3c12)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L04 compound treatment 600.0 -506.0 -0.18 320.0 -527.0 -0.4 -0.413 -0.9332 3025999 ChemDiv3_006582 OC(=O)CCNC1=NC(=O)CS1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L05 compound treatment 360.0 -746.0 -0.26 1200.0 353.0 0.27 0.0045 0.0119 3119315 ChemDiv3_006583 O=C1N(NC(c2ccco2)C31CCCCC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L06 compound treatment 840.0 -266.0 -0.09 320.0 -527.0 -0.4 -0.3528 -0.8494 3119316 ChemDiv3_006584 O=C(Cn1cc(C(=O)C2CC2)c3ccccc13)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L07 compound treatment 400.0 -706.0 -0.25 680.0 -167.0 -0.13 -0.2678 -0.9515 3026002 ChemDiv3_006585 Cc1cc2c3c(C)n(Cc4ccccc4)c(C)c3c(C)nn2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L08 compound treatment 1000.0 -106.0 -0.04 400.0 -447.0 -0.34 -0.2693 -0.7801 3119317 ChemDiv3_006586 COc1ccc(OCc2nnc3SCC(=Nn23)c4ccc(Br)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L09 compound treatment 640.0 -466.0 -0.17 520.0 -327.0 -0.25 -0.2944 -0.9795 1874485 ChemDiv3_006587 Cc1ccc(cc1)S(=O)(=O)N2CCCC3(CCCCC3)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L10 compound treatment 360.0 -746.0 -0.26 4880.0 4030.0 3.1 2.0022 0.6443 3119318 ChemDiv3_006588 O=C(N1CCC(CC1)N(CCc2ccccc2)Cc3ccccc3)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L11 compound treatment 520.0 -586.0 -0.21 480.0 -367.0 -0.28 -0.3462 -0.9889 3026058 ChemDiv3_006589 Cc1ccc(cc1)S(=O)(=O)N2CC3(C)CN(CC(C)(C2)C3)S(=O)(=O)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L12 compound treatment 360.0 -746.0 -0.26 440.0 -407.0 -0.31 -0.4081 -0.9966 3119319 ChemDiv3_006590 Clc1ccc(cc1)S(=O)(=O)NC2CCCCC2Sc3nc4ccccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L13 compound treatment 520.0 -586.0 -0.21 1160.0 313.0 0.24 0.0229 0.0721 3119320 ChemDiv3_006591 OC(CSc1cccc2cccnc12)Cn3c4ccccc4c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L14 compound treatment 480.0 -626.0 -0.22 1320.0 473.0 0.36 0.0997 0.2343 3026062 ChemDiv3_006592 Fc1ccccc1c2n[nH]c(=S)n2CCCN3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L15 compound treatment 760.0 -346.0 -0.12 760.0 -86.9 -0.07 -0.134 -0.9589 3026063 ChemDiv3_006593 Clc1ccc2c(c1)c(nc3nncn32)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L16 compound treatment 280.0 -826.0 -0.29 4280.0 3430.0 2.64 1.6564 0.6246 3119449 ChemDiv3_006594 CCOC(=O)c1nnn(c2nonc2N)c1c3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L17 compound treatment 680.0 -426.0 -0.15 480.0 -367.0 -0.28 -0.3061 -0.9575 3026067 ChemDiv3_006595 OC1=NN(CC1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L18 compound treatment 320.0 -786.0 -0.28 520.0 -327.0 -0.25 -0.3747 -0.9986 3119450 ChemDiv3_006596 COc1ccc2CCc3sc(NC(=O)c4ccccc4Br)nc3-c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L19 compound treatment 560.0 -546.0 -0.19 2080.0 1230.0 0.95 0.5324 0.5509 3119451 ChemDiv3_006597 Cc1ccc(cc1)S(=O)(=O)/N=C\2/S\C(=C/c3ccc4ccccc4n3)\C(=O)N2CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L20 compound treatment 320.0 -786.0 -0.28 880.0 33.1 0.03 -0.1793 -0.64 3026070 ChemDiv3_006598 CC(=O)Nc1ccc(cc1)N2COc3ccc(Cl)cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L21 compound treatment 760.0 -346.0 -0.12 600.0 -247.0 -0.19 -0.2209 -0.9779 3119452 ChemDiv3_006599 Cc1ccc(cc1)c2nc(Nc3cccc(c3)C(F)(F)F)sc2CC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L22 compound treatment 800.0 -306.0 -0.11 2920.0 2070.0 1.59 1.0486 0.6573 3027037 ChemDiv3_006600 CC1CCN(CCCOc2ccc(Br)cc2C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L23 mock treatment 800.0 -306.0 -0.11 880.0 33.1 0.03 -0.0589 -0.5275 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 L24 mock treatment 720.0 -386.0 -0.14 680.0 -167.0 -0.13 -0.1875 -0.9994 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M01 compound treatment 360.0 -746.0 -0.26 640.0 -207.0 -0.16 -0.2995 -0.9701 3027038 ChemDiv3_006601 O=C(Nc1ccccc1)N2CCN(CC2)c3nnc(c4ccccc4)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M02 compound treatment 560.0 -546.0 -0.19 2760.0 1910.0 1.47 0.9015 0.6085 3027039 ChemDiv3_006602 C(Sc1nnc2ccccn12)c3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M03 compound treatment 400.0 -706.0 -0.25 800.0 -46.9 -0.04 -0.2026 -0.8005 3027040 ChemDiv3_006603 NS(=O)(=O)c1ccc(NC2=NC(=O)C(CC(=O)Nc3ccccc3)S2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M04 compound treatment 4000.0 2890.0 1.03 1760.0 913.0 0.7 1.2216 0.9827 1240987 ChemDiv3_006604 CCc1cc2c(C)cc(=O)oc2c(CC=C)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M05 compound treatment 1440.0 334.0 0.12 2120.0 1270.0 0.98 0.7748 0.787 3027041 ChemDiv3_006605 Cc1ccc(Nc2nc(N)nc(CSc3ncccn3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M06 compound treatment 400.0 -706.0 -0.25 680.0 -167.0 -0.13 -0.2678 -0.9515 3027042 ChemDiv3_006606 COc1ccccc1OCc2nc(C#N)c(o2)N3CC(C)CC(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M07 compound treatment 280.0 -826.0 -0.29 560.0 -287.0 -0.22 -0.363 -0.9901 3119453 ChemDiv3_006607 C(N1CNC(=NC1)Nc2nc3ccccc3s2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M08 compound treatment 240.0 -866.0 -0.31 560.0 -287.0 -0.22 -0.373 -0.9867 3119454 ChemDiv3_006608 Clc1ccc(OCc2nc(C#N)c(NCCc3ccccc3)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M09 compound treatment 640.0 -466.0 -0.17 520.0 -327.0 -0.25 -0.2944 -0.9795 3027043 ChemDiv3_006609 COC(=O)CC1N(CCNC1=O)C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M10 compound treatment 360.0 -746.0 -0.26 680.0 -167.0 -0.13 -0.2778 -0.9445 3119455 ChemDiv3_006610 Cc1cccc(c1)N(C2CS(=O)(=O)C=C2)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M11 compound treatment 400.0 -706.0 -0.25 880.0 33.1 0.03 -0.1592 -0.6321 3027044 ChemDiv3_006611 NC(=O)CSc1nc(c2CCc3ccccc3-c2n1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M12 compound treatment 880.0 -226.0 -0.08 1000.0 153.0 0.12 0.0264 0.1852 3119456 ChemDiv3_006612 Cc1ccc(cc1)C(=O)NCC2OCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M13 compound treatment 3720.0 2610.0 0.93 280.0 -567.0 -0.44 0.3479 0.3397 3119457 ChemDiv3_006613 CC(C)CNC(=O)CSc1nc(cc(n1)C(F)(F)F)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M14 compound treatment 400.0 -706.0 -0.25 1000.0 153.0 0.12 -0.094 -0.3398 3027045 ChemDiv3_006614 CCOC(=O)c1ccc(cc1)N2C(=O)C(C)C(Cc3cc(C)cc(C)c3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M15 compound treatment 1320.0 214.0 0.08 560.0 -287.0 -0.22 -0.1021 -0.4384 3119458 ChemDiv3_006615 CC(Sc1nc(cc(n1)C(F)(F)F)c2ccccc2)C(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M16 compound treatment 480.0 -626.0 -0.22 960.0 113.0 0.09 -0.0957 -0.4012 3027046 ChemDiv3_006616 Oc1ccc(Br)cc1C(CC(=O)NCCCN2CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M17 compound treatment 520.0 -586.0 -0.21 880.0 33.1 0.03 -0.1291 -0.6161 3119459 ChemDiv3_006617 FC(F)(F)c1cc(nc(SCC(=O)N(Cc2ccccc2)Cc3ccccc3)n1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M18 compound treatment 360.0 -746.0 -0.26 640.0 -207.0 -0.16 -0.2995 -0.9701 3027047 ChemDiv3_006618 Cc1nc(SCCC(=O)O)c2oc3ccccc3c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M19 compound treatment 600.0 -506.0 -0.18 880.0 33.1 0.03 -0.109 -0.6011 3119460 ChemDiv3_006619 COc1ccc(cc1OC)c2cc(nc(SCC(=O)Nc3cn(C)nc3C)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M20 compound treatment 400.0 -706.0 -0.25 1840.0 993.0 0.76 0.362 0.451 3119461 ChemDiv3_006620 CCOC(=O)c1c(CSc2nc3ccccc3[nH]2)n(c4ccccc4)c5ccc(OC(=O)C)cc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M21 compound treatment 3520.0 2410.0 0.86 4040.0 3190.0 2.45 2.3389 0.9007 3027048 ChemDiv3_006621 Clc1ccc(CC(=O)NC2=NCCS2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M22 compound treatment 480.0 -626.0 -0.22 1560.0 713.0 0.55 0.23 0.3893 3119462 ChemDiv3_006622 CN1C(=O)C2(N(CC3CCCO3)C(=O)C(=C2C(=O)c4ccc(OCC=C)cc4)O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M23 mock treatment 600.0 -506.0 -0.18 640.0 -207.0 -0.16 -0.2393 -0.9981 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 M24 mock treatment 600.0 -506.0 -0.18 3120.0 2270.0 1.75 1.107 0.631 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N01 compound treatment 800.0 -306.0 -0.11 1160.0 313.0 0.24 0.0932 0.3531 3027049 ChemDiv3_006623 COc1ccc(CNc2nc(N)n(n2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N02 compound treatment 360.0 -746.0 -0.26 720.0 -127.0 -0.1 -0.2561 -0.9078 3119463 ChemDiv3_006624 COCCn1c(C)cc(/C=C\2/C(=O)N(c3ccccc23)c4ccccc4)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N03 compound treatment 520.0 -586.0 -0.21 720.0 -127.0 -0.1 -0.2159 -0.9403 3027050 ChemDiv3_006625 CCOC(=O)N1CCc2c(C1)sc3NC(N=C(O)c23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N04 compound treatment 520.0 -586.0 -0.21 600.0 -247.0 -0.19 -0.2811 -0.9989 3119464 ChemDiv3_006626 COC(=O)c1ccc(cc1)n2nnnc2SCCCC(=O)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N05 compound treatment 360.0 -746.0 -0.26 680.0 -167.0 -0.13 -0.2778 -0.9445 3027051 ChemDiv3_006627 COC(=O)CNc1c(F)c(F)nc(F)c1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N06 compound treatment 640.0 -466.0 -0.17 1000.0 153.0 0.12 -0.0338 -0.1668 3119465 ChemDiv3_006628 Cc1ccccc1OCCCn2cc(C(=O)C3CC3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N07 compound treatment 840.0 -266.0 -0.09 640.0 -207.0 -0.16 -0.1791 -0.9692 3027052 ChemDiv3_006629 Cc1ccc(cc1)c2nn(CCC(=O)O)cc2/C=C/3\SC(=N)NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N08 compound treatment 1040.0 -66.3 -0.02 560.0 -287.0 -0.22 -0.1724 -0.7781 3119466 ChemDiv3_006630 Cc1ccc2n(CC(O)CNCc3ccccc3)c4CCCCc4c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N09 compound treatment 640.0 -466.0 -0.17 1120.0 273.0 0.21 0.0313 0.1172 1369071 ChemDiv3_006631 Cc1cc(NC(=O)C2COc3ccccc3O2)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N10 compound treatment 680.0 -426.0 -0.15 600.0 -247.0 -0.19 -0.241 -0.9937 3027053 ChemDiv3_006632 COc1ccc(CN2CCC(CC2)N(C)Cc3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N11 compound treatment 440.0 -666.0 -0.24 640.0 -207.0 -0.16 -0.2794 -0.9813 3119467 ChemDiv3_006633 FC(F)(F)C1(NC(=O)Sc2ccccc2)Oc3ccccc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N12 compound treatment 800.0 -306.0 -0.11 1040.0 193.0 0.15 0.028 0.1524 3119468 ChemDiv3_006634 Cc1cc(C)n2c(SC(CNS(=O)(=O)c3ccccc3)c4ccccc4)nnc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N13 compound treatment 440.0 -666.0 -0.24 800.0 -46.9 -0.04 -0.1926 -0.8055 3027054 ChemDiv3_006635 CN1C(=O)CN(C2CCCCC2)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N14 compound treatment 240.0 -866.0 -0.31 640.0 -207.0 -0.16 -0.3296 -0.9528 3027055 ChemDiv3_006636 CCCCc1c(C)nc(SCC(=O)O)nc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N15 compound treatment 560.0 -546.0 -0.19 400.0 -447.0 -0.34 -0.3796 -0.9634 3119469 ChemDiv3_006637 CN(C)/C=C/C=C/1\CCc2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N16 compound treatment 760.0 -346.0 -0.12 480.0 -367.0 -0.28 -0.286 -0.9308 3027056 ChemDiv3_006638 COc1c(F)c(F)c(C(=O)O)c(Nc2ccc(C)cc2C)c1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N17 compound treatment 720.0 -386.0 -0.14 2760.0 1910.0 1.47 0.9417 0.6384 3119470 ChemDiv3_006639 CC1CN(N=C1O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N18 compound treatment 640.0 -466.0 -0.17 840.0 -6.9 -0.01 -0.1207 -0.7294 3119471 ChemDiv3_006640 CC(=O)Nc1ccc2OCN(Cc3ccc(Cl)cc3)Cc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N19 compound treatment 400.0 -706.0 -0.25 720.0 -127.0 -0.1 -0.246 -0.9153 3027057 ChemDiv3_006641 Cc1oc2ccccc2c1c3csc(n3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N20 compound treatment 440.0 -666.0 -0.24 880.0 33.1 0.03 -0.1492 -0.6275 3119472 ChemDiv3_006642 COc1ccc2cc(sc(=O)c2c1OC)C(=O)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N21 compound treatment 920.0 -186.0 -0.07 760.0 -86.9 -0.07 -0.0939 -1.0 3027058 ChemDiv3_006643 COC(=O)c1cn(CCOc2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N22 compound treatment 1880.0 774.0 0.27 600.0 -247.0 -0.19 0.0601 0.1801 3119473 ChemDiv3_006644 CC(C)c1ccc(C)cc1OCCN2CC(C)CC(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N23 mock treatment 480.0 -626.0 -0.22 720.0 -127.0 -0.1 -0.226 -0.9316 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 N24 mock treatment 320.0 -786.0 -0.28 1120.0 273.0 0.21 -0.049 -0.1403 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O01 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3119474 ChemDiv3_006645 O=C(C1CCCCC1)N2CCN(CC2)c3nnc(c4ccccc4)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O02 compound treatment 400.0 -706.0 -0.25 1920.0 1070.0 0.82 0.4054 0.4708 3027059 ChemDiv3_006646 COCCn1c(C)cc(C(=O)CSc2nnc3ccccn23)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O03 compound treatment 400.0 -706.0 -0.25 280.0 -567.0 -0.44 -0.4849 -0.9656 3027060 ChemDiv3_006647 CSC1=NN1c2cc(C)nc(N)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O04 compound treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 1195811 ChemDiv3_006648 O=c1ccc2ccc(OCc3ccccc3)cc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O05 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3119475 ChemDiv3_006649 Cc1ccc(Nc2nc(N)nc(CN3CCC(Cc4ccccc4)CC3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O06 compound treatment 360.0 -746.0 -0.26 320.0 -527.0 -0.4 -0.4732 -0.9789 3027061 ChemDiv3_006650 CCN1CCN(CC1)c2oc(COc3ccccc3C)nc2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O07 compound treatment 400.0 -706.0 -0.25 360.0 -487.0 -0.37 -0.4415 -0.9811 3119608 ChemDiv3_006651 OC(=O)c1cccnc1SCC(=O)N2c3ccccc3CCc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O08 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3027062 ChemDiv3_006652 COc1ccccc1OCc2nc(C#N)c(o2)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O09 compound treatment 4480.0 3370.0 1.2 520.0 -327.0 -0.25 0.6688 0.5469 3119609 ChemDiv3_006653 CC1=Nc2ccccc2N=C(NC(=O)/C=C/C(=O)O)C1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O10 compound treatment 520.0 -586.0 -0.21 320.0 -527.0 -0.4 -0.4331 -0.9522 3027063 ChemDiv3_006654 CC1CCCC(C)N1C(=O)Cn2cc(/C=C\3/C(=O)Nc4ccccc34)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O11 compound treatment 3560.0 2450.0 0.87 160.0 -687.0 -0.53 0.2426 0.2384 3119610 ChemDiv3_006655 CN(Cc1ccccc1)C(=O)CSc2nc(c3CCc4ccccc4-c3n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O12 compound treatment 440.0 -666.0 -0.24 360.0 -487.0 -0.37 -0.4314 -0.9756 3119611 ChemDiv3_006656 COc1ccc(cc1)C2(CCOCC2)C(=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O13 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3027064 ChemDiv3_006657 Cc1cc(nc(SCCNC(=O)c2ccccc2F)n1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O14 compound treatment 280.0 -826.0 -0.29 360.0 -487.0 -0.37 -0.4716 -0.9928 3119612 ChemDiv3_006658 COc1ccc2oc(CS(=O)c3ccccc3)c(C(=O)O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O15 compound treatment 360.0 -746.0 -0.26 800.0 -46.9 -0.04 -0.2126 -0.7959 3119613 ChemDiv3_006659 CC(Sc1nc(cc(n1)C(F)(F)F)c2ccccc2)C(=O)NCCCn3ccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O16 compound treatment 560.0 -546.0 -0.19 200.0 -647.0 -0.5 -0.4882 -0.9158 3027065 ChemDiv3_006660 COc1nc(NC(C)(C)C)nc(Oc2ccc(=O)n(C)n2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O17 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3119614 ChemDiv3_006661 CC1CN(CC(C)O1)C(=O)CSc2nc(cc(n2)C(F)(F)F)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O18 compound treatment 320.0 -786.0 -0.28 360.0 -487.0 -0.37 -0.4615 -0.9896 3027066 ChemDiv3_006662 CCOC(=O)c1c(CN(CC)CC)n(c2ccccc2)c3ccc(O)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O19 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3119615 ChemDiv3_006663 COc1ccc(cc1)c2cc(nc(SCCC(=O)NC(C)C)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O20 compound treatment 240.0 -866.0 -0.31 240.0 -607.0 -0.47 -0.5468 -0.9796 3027067 ChemDiv3_006664 O=C(ON1C(=O)c2cccc3cccc(C1=O)c23)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O21 compound treatment 280.0 -826.0 -0.29 440.0 -407.0 -0.31 -0.4281 -0.9995 3027068 ChemDiv3_006665 Cc1cc(C)n(n1)c2nncc(n2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O22 compound treatment 200.0 -906.0 -0.32 280.0 -567.0 -0.44 -0.5351 -0.9889 3119616 ChemDiv3_006666 CN1C(=O)C2(N(CCCN3CCOCC3)C(=O)C(=C2C(=O)c4ccc(C)c(F)c4)O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O23 mock treatment 360.0 -746.0 -0.26 280.0 -567.0 -0.44 -0.4949 -0.9716 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 O24 mock treatment 360.0 -746.0 -0.26 280.0 -567.0 -0.44 -0.4949 -0.9716 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P01 compound treatment 320.0 -786.0 -0.28 400.0 -447.0 -0.34 -0.4398 -0.9947 3027069 ChemDiv3_006667 Nc1nc(NCc2c(F)cccc2Cl)nn1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P02 compound treatment 240.0 -866.0 -0.31 560.0 -287.0 -0.22 -0.373 -0.9867 3119617 ChemDiv3_006668 CCN(CC)CCSc1nc(O)c(C)c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P03 compound treatment 360.0 -746.0 -0.26 240.0 -607.0 -0.47 -0.5167 -0.9641 3119618 ChemDiv3_006669 CCCCN1C(=O)C(O)(CC(=O)c2c(C)coc2C)c3cc(Br)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P04 compound treatment 240.0 -866.0 -0.31 240.0 -607.0 -0.47 -0.5468 -0.9796 3027070 ChemDiv3_006670 COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)OCc4ccccn4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P05 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3119619 ChemDiv3_006671 COc1cccc(=O)c2c(C)n(CC(=O)c3ccccc3)c(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P06 compound treatment 440.0 -666.0 -0.24 280.0 -567.0 -0.44 -0.4749 -0.9588 3027071 ChemDiv3_006672 O=C(c1cccs1)c2cn(CCOc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P07 compound treatment 440.0 -666.0 -0.24 400.0 -447.0 -0.34 -0.4097 -0.9835 3119620 ChemDiv3_006673 CC(C)OC(=O)C1C2C3CCCCC3(NC1=O)Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P08 compound treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 3119621 ChemDiv3_006674 Cc1ccc2n(CC(O)CN(CC=C)CC=C)c3CCCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P09 compound treatment 400.0 -706.0 -0.25 320.0 -527.0 -0.4 -0.4632 -0.9735 1148562 ChemDiv3_006675 Cc1c(sc(=S)n1CCOc2ccccc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P10 compound treatment 600.0 -506.0 -0.18 160.0 -687.0 -0.53 -0.4999 -0.8973 3119622 ChemDiv3_006676 CN(Cc1ccccc1)C(=O)C2CCCN(Cc3ccc(Cl)cc3)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P11 compound treatment 1680.0 574.0 0.2 320.0 -527.0 -0.4 -0.1421 -0.3138 3027072 ChemDiv3_006677 FC(F)(F)C(=O)NC(=O)N1CCCc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P12 compound treatment 4640.0 3530.0 1.25 280.0 -567.0 -0.44 0.5787 0.4361 3119623 ChemDiv3_006678 Cc1cc(C)n2c(SC3CCCCC3NS(=O)(=O)c4ccccc4)nnc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P13 compound treatment 360.0 -746.0 -0.26 200.0 -647.0 -0.5 -0.5384 -0.9566 3027134 ChemDiv3_006679 Cc1cc(=O)n2nc(nc2[nH]1)N3C(=O)c4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P14 compound treatment 280.0 -826.0 -0.29 320.0 -527.0 -0.4 -0.4933 -0.9875 3027135 ChemDiv3_006680 Clc1ccc2OC(=O)CC(c3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P15 compound treatment 280.0 -826.0 -0.29 280.0 -567.0 -0.44 -0.515 -0.9815 1922162 ChemDiv3_006681 CN(C)/C=C/C=C1C(=O)CCCC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P16 compound treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 3027136 ChemDiv3_006682 C(Nc1ccccn1)c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P17 compound treatment 280.0 -826.0 -0.29 240.0 -607.0 -0.47 -0.5367 -0.975 1722485 ChemDiv3_006683 Cc1cc(N)n(n1)c2ccccc2C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P18 compound treatment 200.0 -906.0 -0.32 240.0 -607.0 -0.47 -0.5568 -0.9836 3027137 ChemDiv3_006684 CC(=O)Nc1ccc2OCN(Cc2c1)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P19 compound treatment 480.0 -626.0 -0.22 280.0 -567.0 -0.44 -0.4648 -0.9513 3027138 ChemDiv3_006685 CC(C)c1ccc(C)cc1OCC(=O)Nc2cc(ccc2Cl)c3nc4ncccc4o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P20 compound treatment 400.0 -706.0 -0.25 400.0 -447.0 -0.34 -0.4198 -0.9881 3027139 ChemDiv3_006686 OCCNC(=O)c1cc2ccccc2c(=O)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P21 compound treatment 240.0 -866.0 -0.31 280.0 -567.0 -0.44 -0.525 -0.9855 3027140 ChemDiv3_006687 CCc1cccc2c(/C=C\3/C(=O)N(C)c4ccccc34)c[nH]c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P22 compound treatment 200.0 -906.0 -0.32 240.0 -607.0 -0.47 -0.5568 -0.9836 3119624 ChemDiv3_006688 CC(C)(c1ccccc1)c2ccc(OCCN3CCOCC3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P23 mock treatment 320.0 -786.0 -0.28 320.0 -527.0 -0.4 -0.4833 -0.9835 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2019 P24 mock treatment 320.0 -786.0 -0.28 280.0 -567.0 -0.44 -0.505 -0.9769 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A01 compound treatment 360.0 -776.0 -0.28 6560.0 5940.0 4.56 3.0302 0.6632 3119625 ChemDiv3_006689 Cc1nn2c(nnc2c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A02 compound treatment 360.0 -776.0 -0.28 680.0 60.6 0.05 -0.1618 -0.5793 3027141 ChemDiv3_006690 Clc1ccc(cc1)c2noc(CCCN3C(=O)c4ccccc4C3=O)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A03 compound treatment 280.0 -856.0 -0.3 1080.0 461.0 0.35 0.0353 0.0757 3119626 ChemDiv3_006691 CCC(CO)NS(=O)(=O)c1cc(ccc1OC)c2nnc3c4ccccc4c(C)nn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A04 compound treatment 320.0 -816.0 -0.29 240.0 -379.0 -0.29 -0.4107 -1.0 3027142 ChemDiv3_006692 CCc1nc2cc3sc(CC)nc3cc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A05 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 1191945 ChemDiv3_006693 CCOP(=S)(OCC)C(Nc1ccccc1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A06 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 3027143 ChemDiv3_006694 CC(=O)n1nc(nc1N)c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A07 compound treatment 280.0 -856.0 -0.3 360.0 -259.0 -0.2 -0.3556 -0.979 3119627 ChemDiv3_006695 Nc1cc(=O)[nH]c2nnc(SCc3ccc(Br)cc3)n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A08 compound treatment 400.0 -736.0 -0.26 280.0 -339.0 -0.26 -0.3689 -1.0 3027144 ChemDiv3_006696 O=C(COc1ccccc1)Nc2c(oc3ccccc23)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A09 compound treatment 400.0 -736.0 -0.26 320.0 -299.0 -0.23 -0.3472 -0.998 3119628 ChemDiv3_006697 CC(C)(C)C(=O)Oc1ccc2cc(c3ccc4ccccc4n3)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A10 compound treatment 440.0 -696.0 -0.25 920.0 301.0 0.23 -0.0114 -0.0338 3119629 ChemDiv3_006698 COc1ccc(cc1c2nnc3c4ccccc4c(C)nn23)S(=O)(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A11 compound treatment 440.0 -696.0 -0.25 680.0 60.6 0.05 -0.1417 -0.5639 3027145 ChemDiv3_006699 O=C1CSC(N1)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A12 compound treatment 1280.0 144.0 0.05 920.0 301.0 0.23 0.1993 0.843 1492220 ChemDiv3_006700 CCOC(=O)c1nn(c2ccc(OC)cc2)c(=O)c3c(N)scc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A13 compound treatment 3440.0 2300.0 0.82 3320.0 2700.0 2.07 2.0439 0.9171 3027146 ChemDiv3_006701 CN1CCc2nc(SCc3cccc(c3)C(F)(F)F)c(C#N)cc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A14 compound treatment 1320.0 184.0 0.07 1040.0 421.0 0.32 0.2744 0.833 3119630 ChemDiv3_006702 COc1ccc(CN2CNc3nc4ccccc4n3C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A15 compound treatment 520.0 -616.0 -0.22 640.0 20.6 0.02 -0.1434 -0.6541 3027147 ChemDiv3_006703 Cc1cc(SCc2ccccc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A16 compound treatment 360.0 -776.0 -0.28 440.0 -179.0 -0.14 -0.2921 -0.9487 3119631 ChemDiv3_006704 CC1(Nc2ccccc2-c3nc4ccccc4n31)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A17 compound treatment 520.0 -616.0 -0.22 400.0 -219.0 -0.17 -0.2737 -0.9917 3119632 ChemDiv3_006705 COC(=O)C1=CN(C=C(C1c2ccc(OC)c(O)c2)C(=O)OC)c3cc(C)cc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A18 compound treatment 280.0 -856.0 -0.3 480.0 -139.0 -0.11 -0.2904 -0.9019 3027148 ChemDiv3_006706 OC(=O)c1ccc(cc1)n2nnnc2Oc3ccccc3C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A19 compound treatment 440.0 -696.0 -0.25 320.0 -299.0 -0.23 -0.3372 -0.9994 1643940 ChemDiv3_006707 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3oc(=O)sc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A20 compound treatment 6320.0 5180.0 1.84 360.0 -259.0 -0.2 1.1595 0.6269 1197258 ChemDiv3_006708 CC1(C)Cc2c(C#N)c(NC3CCCCC3)nc(c4ccco4)c2CO1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A21 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3119633 ChemDiv3_006709 COc1ccc(Nc2nc(N)nc(CSC(=S)N(C)C3CCCCC3)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A22 compound treatment 400.0 -736.0 -0.26 280.0 -339.0 -0.26 -0.3689 -1.0 3119769 ChemDiv3_006710 COc1cc2CC[N+](C)(C)C3CC4(C=CC(=O)C=C4)c(c32)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A23 mock treatment 280.0 -856.0 -0.3 240.0 -379.0 -0.29 -0.4207 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 A24 mock treatment 320.0 -816.0 -0.29 320.0 -299.0 -0.23 -0.3673 -0.9934 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B01 compound treatment 320.0 -816.0 -0.29 360.0 -259.0 -0.2 -0.3455 -0.9833 3027149 ChemDiv3_006711 C1COC(O1)c2cccn2c3ccc4noc(c5ccccc5)c4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B02 compound treatment 360.0 -776.0 -0.28 240.0 -379.0 -0.29 -0.4007 -0.9996 3119770 ChemDiv3_006712 Cc1nn(c2cc(ccc2N)N3CCCCC3)c(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B03 compound treatment 1560.0 424.0 0.15 440.0 -179.0 -0.14 0.0089 0.0438 3027150 ChemDiv3_006713 COc1ccc(cc1)C2N=C(SC(=C2C#N)N)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B04 compound treatment 520.0 -616.0 -0.22 320.0 -299.0 -0.23 -0.3171 -0.9997 3119771 ChemDiv3_006714 Fc1ccc(CSc2ncnc3n(CC=C)c(=S)sc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B05 compound treatment 760.0 -376.0 -0.13 360.0 -259.0 -0.2 -0.2352 -0.9811 3027151 ChemDiv3_006715 Cc1cc(C)c(c2cc(no2)C(F)(F)F)c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B06 compound treatment 1360.0 224.0 0.08 240.0 -379.0 -0.29 -0.1498 -0.4963 3119772 ChemDiv3_006716 CCC(Sc1nnc2sc3ccccc3n12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B07 compound treatment 280.0 -856.0 -0.3 480.0 -139.0 -0.11 -0.2904 -0.9019 3119773 ChemDiv3_006717 COc1ccccc1C2N(C(=O)N3CCCN23)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B08 compound treatment 320.0 -816.0 -0.29 240.0 -379.0 -0.29 -0.4107 -1.0 3027152 ChemDiv3_006718 CCN1/C(=C\2/N(C(=NC2=O)C)c3ccccc3)/C=Cc4ccc(C)cc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B09 compound treatment 280.0 -856.0 -0.3 200.0 -419.0 -0.32 -0.4424 -0.9996 3119774 ChemDiv3_006719 Oc1ccccc1N2CC=C(NC2=O)c3ccc(cc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B10 compound treatment 520.0 -616.0 -0.22 320.0 -299.0 -0.23 -0.3171 -0.9997 3027153 ChemDiv3_006720 CCc1cc(C(=O)N2CCOCC2)c(NC3=NS(=O)(=O)c4ccccc34)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B11 compound treatment 640.0 -496.0 -0.18 720.0 101.0 0.08 -0.0698 -0.3633 3119775 ChemDiv3_006721 CC(N/C=C/1\C(=O)Oc2ccccc2C1=O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B12 compound treatment 3120.0 1980.0 0.7 3400.0 2780.0 2.13 2.0071 0.8929 3119776 ChemDiv3_006722 O/N=C/c1ccc(cn1)C(=O)NCc2ccccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B13 compound treatment 444640.0 444000.0 157.33 373440.0 373000.0 286.22 313.639 0.9603 1466284 ChemDiv3_006723 CCn1nc(N)c2c(O)nc(O)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B14 compound treatment 4440.0 3300.0 1.17 3800.0 3180.0 2.44 2.5554 0.9435 3119777 ChemDiv3_006724 COCc1cc(C)n(CC(=O)Nc2cc(Cl)ccc2OC)c(=O)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B15 compound treatment 680.0 -456.0 -0.16 680.0 60.6 0.05 -0.0815 -0.4841 3027154 ChemDiv3_006725 NCCC1COc2ccccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B16 compound treatment 1920.0 784.0 0.28 5840.0 5220.0 4.01 3.0307 0.7543 3119778 ChemDiv3_006726 CC(C)c1ccc(cc1)S(=O)(=O)/N=C\2/C=C(Sc3nc[nH]n3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B17 compound treatment 240.0 -896.0 -0.32 360.0 -259.0 -0.2 -0.3656 -0.9746 3027155 ChemDiv3_006727 CC(C)C(NC(=O)c1cc(oc1C)c2ccc3OCCOc3c2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B18 compound treatment 440.0 -696.0 -0.25 320.0 -299.0 -0.23 -0.3372 -0.9994 3119779 ChemDiv3_006728 Cc1ccc(cc1)C2CC(=O)n3nc(N)nc3N2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B19 compound treatment 4360.0 3220.0 1.14 360.0 -259.0 -0.2 0.6679 0.5753 3027156 ChemDiv3_006729 OP(=O)(CN1CCOCC1)C2Cc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B20 compound treatment 360.0 -776.0 -0.28 400.0 -219.0 -0.17 -0.3138 -0.9722 3119780 ChemDiv3_006730 Cc1cc2-c3cccc(C)c3NC(c4cccc(O)c4O)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B21 compound treatment 520.0 -616.0 -0.22 280.0 -339.0 -0.26 -0.3388 -0.9962 3119781 ChemDiv3_006731 CC1=CS(=O)(=O)CC1Sc2nc(C)n[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B22 compound treatment 240.0 -896.0 -0.32 320.0 -299.0 -0.23 -0.3873 -0.9873 3027157 ChemDiv3_006732 OC(=O)Cn1cc(C(=O)c2ccccc2F)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B23 mock treatment 440.0 -696.0 -0.25 320.0 -299.0 -0.23 -0.3372 -0.9994 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 B24 mock treatment 560.0 -576.0 -0.2 320.0 -299.0 -0.23 -0.3071 -0.9983 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C01 compound treatment 5960.0 4820.0 1.71 760.0 141.0 0.11 1.2864 0.7502 1224449 ChemDiv3_006733 c1ccc(cc1)c2nnc3c4ccccc4c(nn23)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C02 compound treatment 360.0 -776.0 -0.28 400.0 -219.0 -0.17 -0.3138 -0.9722 3027158 ChemDiv3_006734 CCCC(=O)N1N=C(OC1c2ccc(OC)cc2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C03 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3119782 ChemDiv3_006735 CCC(=O)Nc1cccc(c1)c2nnc3c4ccccc4c(C)nn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C04 compound treatment 240.0 -896.0 -0.32 280.0 -339.0 -0.26 -0.409 -0.9951 3027159 ChemDiv3_006736 CC(C)c1nc2cc3sc(nc3cc2s1)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C05 compound treatment 320.0 -816.0 -0.29 320.0 -299.0 -0.23 -0.3673 -0.9934 3119783 ChemDiv3_006737 CCOC(=O)c1snc2c(=O)[nH]cnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C06 compound treatment 280.0 -856.0 -0.3 240.0 -379.0 -0.29 -0.4207 -0.9998 3027160 ChemDiv3_006738 Cc1cc(C)nc(n1)N2CC(=O)NC2=N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C07 compound treatment 800.0 -336.0 -0.12 280.0 -339.0 -0.26 -0.2686 -0.9373 3119784 ChemDiv3_006739 Nc1cc(=O)[nH]c2nnc(SCC=C)n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C08 compound treatment 440.0 -696.0 -0.25 360.0 -259.0 -0.2 -0.3154 -0.9943 3119785 ChemDiv3_006740 COc1cc(cc(OC)c1OC)C(=O)Nc2c(oc3ccccc23)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C09 compound treatment 440.0 -696.0 -0.25 480.0 -139.0 -0.11 -0.2503 -0.9299 3027161 ChemDiv3_006741 Cc1c(O)ccc(c2n[nH]cc2c3nc4ccccc4s3)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C10 compound treatment 360.0 -776.0 -0.28 440.0 -179.0 -0.14 -0.2921 -0.9487 3119786 ChemDiv3_006742 COc1ccc(cc1c2nnc3c4ccccc4c(C)nn23)S(=O)(=O)N(C)CCO 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C11 compound treatment 560.0 -576.0 -0.2 880.0 261.0 0.2 -0.0031 -0.0107 3027162 ChemDiv3_006743 COc1ccc(Cn2c(=O)oc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C12 compound treatment 920.0 -216.0 -0.08 720.0 101.0 0.08 4.0E-4 0.0036 3119787 ChemDiv3_006744 Cc1ccc2nsnc2c1S(=O)(=O)NC3CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C13 compound treatment 7280.0 6140.0 2.18 6080.0 5460.0 4.19 4.5055 0.9536 3027163 ChemDiv3_006745 Brc1ccccc1CSc2nc3C4CCN(CC4)c3cc2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C14 compound treatment 880.0 -256.0 -0.09 1120.0 501.0 0.38 0.2075 0.5254 3119788 ChemDiv3_006746 C1CCC(CC1)N2CNc3nc4ccccc4n3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C15 compound treatment 440.0 -696.0 -0.25 480.0 -139.0 -0.11 -0.2503 -0.9299 3027164 ChemDiv3_006747 COCc1ccc2oc(cc2c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C16 compound treatment 360.0 -776.0 -0.28 1240.0 621.0 0.48 0.1422 0.2584 1298113 ChemDiv3_006748 CCC1(C)Nc2ccccc2-c3nc4ccccc4n31 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C17 compound treatment 520.0 -616.0 -0.22 680.0 60.6 0.05 -0.1217 -0.5443 3119789 ChemDiv3_006749 Cc1ccc2nc(NCn3nc(oc3=S)c4ccccc4)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C18 compound treatment 520.0 -616.0 -0.22 960.0 341.0 0.26 0.0303 0.089 3027165 ChemDiv3_006750 CCn1cc(C2N3CC4(C)CN2CC(C)(C3)C4O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C19 compound treatment 480.0 -656.0 -0.23 5520.0 4900.0 3.76 2.4957 0.6621 3119790 ChemDiv3_006751 O=C(N(c1ccc2oc(=O)sc2c1)S(=O)(=O)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C20 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 1249288 ChemDiv3_006752 CCN(CC)CCNc1nc(c2ccco2)c3COC(C)(C)Cc3c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C21 compound treatment 4720.0 3580.0 1.27 240.0 -379.0 -0.29 0.693 0.5314 3027166 ChemDiv3_006753 COc1ccccc1Nc2nc(N)nc(CN3CCC(C)CC3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C22 compound treatment 1360.0 224.0 0.08 280.0 -339.0 -0.26 -0.1281 -0.4703 3119791 ChemDiv3_006754 O=C(Cn1cc(C(=O)C2CCCCC2)c3ccccc13)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C23 mock treatment 360.0 -776.0 -0.28 440.0 -179.0 -0.14 -0.2921 -0.9487 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 C24 mock treatment 360.0 -776.0 -0.28 280.0 -339.0 -0.26 -0.3789 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D01 compound treatment 4400.0 3260.0 1.16 360.0 -259.0 -0.2 0.6779 0.577 3027167 ChemDiv3_006755 COc1cc(ccc1O)C2N(Cc3ccccc3)C(=O)c4oc5ccccc5c(=O)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D02 compound treatment 320.0 -816.0 -0.29 2360.0 1740.0 1.34 0.7402 0.5413 1400123 ChemDiv3_006756 Cc1cccn2cc(nc12)c3cccc(NC(=O)c4ccccc4)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D03 compound treatment 280.0 -856.0 -0.3 240.0 -379.0 -0.29 -0.4207 -0.9998 3027168 ChemDiv3_006757 CSc1nnc-2c(OC=Nc3ccc(Cl)cc32)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D04 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3119792 ChemDiv3_006758 C=CCn1c(=S)sc2c(SCC(=O)N3CCc4ccccc34)ncnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D05 compound treatment 360.0 -776.0 -0.28 160.0 -459.0 -0.35 -0.4441 -0.9925 3119793 ChemDiv3_006759 CCOC(=O)C1SC2(CC1(O)c3c(C)cc(C)nc3O2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D06 compound treatment 360.0 -776.0 -0.28 280.0 -339.0 -0.26 -0.3789 -0.9996 3027169 ChemDiv3_006760 Nc1ccc2[nH]c(nc2c1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D07 compound treatment 440.0 -696.0 -0.25 280.0 -339.0 -0.26 -0.3589 -0.9996 1726077 ChemDiv3_006761 COc1ccc(cc1)C2N3CC(C)(C)CN23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D08 compound treatment 280.0 -856.0 -0.3 200.0 -419.0 -0.32 -0.4424 -0.9996 3027219 ChemDiv3_006762 CCN1C=C/C(=C\c2cc[n+](CC)c3ccccc23)/c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D09 compound treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 3027220 ChemDiv3_006763 c1ccc(cc1)c2nn3c(nnc3s2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D10 compound treatment 280.0 -856.0 -0.3 480.0 -139.0 -0.11 -0.2904 -0.9019 3027221 ChemDiv3_006764 CCc1ccc(NC(=O)Cn2c(=O)oc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D11 compound treatment 320.0 -816.0 -0.29 440.0 -179.0 -0.14 -0.3021 -0.9422 3027222 ChemDiv3_006765 O=C(Cn1c(nc2ccccc12)c3ccccn3)NCCCn4ccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D12 compound treatment 920.0 -216.0 -0.08 600.0 -19.4 -0.01 -0.0648 -0.8287 3027223 ChemDiv3_006766 C/C(=N\O)/C(=O)NCCc1c[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D13 compound treatment 720.0 -416.0 -0.15 560.0 -59.4 -0.05 -0.1366 -0.8842 3027224 ChemDiv3_006767 O=c1[nH]c2ccc(cc2[nH]1)S(=O)(=O)NC3CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D14 compound treatment 520.0 -616.0 -0.22 600.0 -19.4 -0.01 -0.1651 -0.7534 3027225 ChemDiv3_006768 Clc1ccc(cc1)c2nnc(SC3CCOC3=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D15 compound treatment 480.0 -656.0 -0.23 480.0 -139.0 -0.11 -0.2403 -0.9378 1057023 ChemDiv3_006769 OC(=O)CCC1COc2ccccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D16 compound treatment 680.0 -456.0 -0.16 400.0 -219.0 -0.17 -0.2335 -0.9998 3119794 ChemDiv3_006770 O=C1C(=C/C(=N/S(=O)(=O)c2cccs2)/c3ccccc13)Sc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D17 compound treatment 440.0 -696.0 -0.25 360.0 -259.0 -0.2 -0.3154 -0.9943 3027226 ChemDiv3_006771 Cc1cccc(OCCCn2c(=O)sc3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D18 compound treatment 360.0 -776.0 -0.28 320.0 -299.0 -0.23 -0.3572 -0.996 3119928 ChemDiv3_006772 Clc1ccc(cc1)C2CC(=O)n3c(N2)nc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D19 compound treatment 280.0 -856.0 -0.3 400.0 -219.0 -0.17 -0.3339 -0.9613 3027227 ChemDiv3_006773 OP(=O)(CN1CCCCCC1)C2Cc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D20 compound treatment 320.0 -816.0 -0.29 320.0 -299.0 -0.23 -0.3673 -0.9934 3119929 ChemDiv3_006774 Cc1cc2-c3cccc(C)c3NC(c4ccsc4)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D21 compound treatment 3720.0 2580.0 0.92 320.0 -299.0 -0.23 0.4856 0.5139 1438487 ChemDiv3_006775 Cc1cccc(NC2CS(=O)(=O)CC2O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D22 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3027228 ChemDiv3_006776 CC1CCCCN1C(=O)CSc2nc(cc(n2)C(F)(F)F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D23 mock treatment 360.0 -776.0 -0.28 200.0 -419.0 -0.32 -0.4224 -0.997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 D24 mock treatment 240.0 -896.0 -0.32 320.0 -299.0 -0.23 -0.3873 -0.9873 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E01 compound treatment 1240.0 104.0 0.04 400.0 -219.0 -0.17 -0.0931 -0.5398 3119930 ChemDiv3_006777 CNS(=O)(=O)c1ccc(C)c(c1)c2nnc3c4ccccc4c(C)nn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E02 compound treatment 9840.0 8700.0 3.09 920.0 301.0 0.23 2.3465 0.7579 3027229 ChemDiv3_006778 OCN1C(=O)c2ccncc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E03 compound treatment 560.0 -576.0 -0.2 1560.0 941.0 0.72 0.3661 0.4878 1238985 ChemDiv3_006779 CC1OP(=S)(OC1C)C(Nc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E04 compound treatment 760.0 -376.0 -0.13 520.0 -99.4 -0.08 -0.1483 -0.9648 3027230 ChemDiv3_006780 COCC(=O)n1nc(nc1NCc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E05 compound treatment 400.0 -736.0 -0.26 560.0 -59.4 -0.05 -0.2169 -0.8181 3119931 ChemDiv3_006781 COc1ccc(cc1)C2OC(=NN2C(=O)C)c3ccc(cc3)S(=O)(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E06 compound treatment 1480.0 344.0 0.12 960.0 341.0 0.26 0.2711 0.9397 3119932 ChemDiv3_006782 Cc1ccc(cc1)C(=O)c2oc3ccccc3c2NC(=O)C4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E07 compound treatment 1200.0 63.8 0.02 1000.0 381.0 0.29 0.2226 0.7596 3027231 ChemDiv3_006783 CCOC(=O)c1oc2cc(O)c(CC)cc2c(=O)c1c3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E08 compound treatment 1280.0 144.0 0.05 480.0 -139.0 -0.11 -0.0396 -0.3341 3119933 ChemDiv3_006784 CC(C)C(=O)Nc1c(oc2ccccc12)C(=O)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E09 compound treatment 1200.0 63.8 0.02 1840.0 1220.0 0.94 0.6786 0.724 3027232 ChemDiv3_006785 O=C(Oc1ccc2c(=O)c(coc2c1)c3ccccc3)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E10 compound treatment 1320.0 184.0 0.07 1160.0 541.0 0.42 0.3396 0.8082 3119934 ChemDiv3_006786 COc1ccc(cc1c2nnc3c4ccccc4c(C)nn23)S(=O)(=O)NCCN5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E11 compound treatment 840.0 -296.0 -0.11 720.0 101.0 0.08 -0.0197 -0.1508 1785240 ChemDiv3_006787 OC(=O)Cc1c(c2ccccc2)c3cc(Cl)ccc3[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E12 compound treatment 3160.0 2020.0 0.72 400.0 -219.0 -0.17 0.3886 0.5269 3119935 ChemDiv3_006788 COC(=O)C1=NOC2C1C(=O)N(C2=O)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E13 compound treatment 1040.0 -96.3 -0.03 1160.0 541.0 0.42 0.2694 0.6468 3027233 ChemDiv3_006789 Cc1cc(nc2snc(Br)c12)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E14 compound treatment 640.0 -496.0 -0.18 4320.0 3700.0 2.84 1.8844 0.662 3119936 ChemDiv3_006790 NC1=NC(c2ccncc2)n3c(N1)nc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E15 compound treatment 1320.0 184.0 0.07 720.0 101.0 0.08 0.1007 0.9964 3027234 ChemDiv3_006791 CC(C)COc1ccc(cc1)S(=O)(=O)n2cc(F)c(=O)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E16 compound treatment 520.0 -616.0 -0.22 680.0 60.6 0.05 -0.1217 -0.5443 3119937 ChemDiv3_006792 Oc1ccccc1C2Nc3ccccc3-c4nc5ccccc5n24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E17 compound treatment 3480.0 2340.0 0.83 840.0 221.0 0.17 0.7077 0.834 3119938 ChemDiv3_006793 CN(C)c1nc(Oc2ccc(=O)n(C)n2)nc(n1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E18 compound treatment 1360.0 224.0 0.08 720.0 101.0 0.08 0.1108 0.9999 3027235 ChemDiv3_006794 CC1(CN2CC3(C)CN(C1)C2C4C(=O)Nc5ccccc45)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E19 compound treatment 1760.0 624.0 0.22 680.0 60.6 0.05 0.1894 0.8376 3119939 ChemDiv3_006795 CC(=O)N(c1ccc2oc(=O)sc2c1)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E20 compound treatment 840.0 -296.0 -0.11 1520.0 901.0 0.69 0.4146 0.5928 3119940 ChemDiv3_006796 CCCCc1nc2sc3c(NCC=C)ncnc3c2c4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E21 compound treatment 7440.0 6300.0 2.24 4040.0 3420.0 2.63 3.4382 0.9968 3027236 ChemDiv3_006797 COc1ccccc1Nc2nc(N)nc(CN3CCc4ccccc4C3)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E22 compound treatment 720.0 -416.0 -0.15 600.0 -19.4 -0.01 -0.1149 -0.7744 3119941 ChemDiv3_006798 O=C(Cn1cc(C(=O)c2ccco2)c3ccccc13)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E23 mock treatment 1120.0 -16.3 -0.01 600.0 -19.4 -0.01 -0.0146 -0.915 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 E24 mock treatment 2760.0 1620.0 0.58 4520.0 3900.0 2.99 2.5248 0.8279 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F01 compound treatment 4680.0 3540.0 1.26 560.0 -59.4 -0.05 0.8567 0.681 3027237 ChemDiv3_006799 CN(C)S(=O)(=O)c1ccc2c(c1)oc(=O)c3cc(ccc32)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F02 compound treatment 2160.0 1020.0 0.36 1080.0 461.0 0.35 0.5069 0.9999 3119942 ChemDiv3_006800 Cc1ccn2cc(nc2c1)c3cccc(NS(=O)(=O)c4cc(C)c(C)cc4C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F03 compound treatment 2280.0 1140.0 0.41 4200.0 3580.0 2.75 2.2307 0.8028 3119943 ChemDiv3_006801 On1c(nc2CCCCc21)C(=O)c3ccc(Oc4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F04 compound treatment 5640.0 4500.0 1.6 680.0 60.6 0.05 1.1627 0.7274 3027238 ChemDiv3_006802 NC(=O)CSc1ncnc2n(CC=C)c(=S)sc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F05 compound treatment 2800.0 1660.0 0.59 440.0 -179.0 -0.14 0.32 0.528 2117441 ChemDiv3_006803 OC(=O)C1CCCN1Cc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F06 compound treatment 4600.0 3460.0 1.23 480.0 -139.0 -0.11 0.7932 0.6431 3027239 ChemDiv3_006804 Nc1ncnc2n(CCOc3ccccc3)cnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F07 compound treatment 5800.0 4660.0 1.65 1120.0 501.0 0.38 1.4416 0.8488 3119944 ChemDiv3_006805 O=C(OCc1ccccc1)C2=NNC3C2C(=O)N(C3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F08 compound treatment 600.0 -536.0 -0.19 720.0 101.0 0.08 -0.0799 -0.389 3027240 ChemDiv3_006806 CCN(CC)CCNc1nc(C)cc(C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F09 compound treatment 1320.0 184.0 0.07 760.0 141.0 0.11 0.1224 0.9708 1107523 ChemDiv3_006807 C(Oc1ccccc1)c2nn3c(nnc3s2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F10 compound treatment 1440.0 304.0 0.11 680.0 60.6 0.05 0.1091 0.9296 3119945 ChemDiv3_006808 CC(C)COc1ccc(cc1)C(=O)Nc2ccc(cc2)C(=O)NCC3(CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F11 compound treatment 2760.0 1620.0 0.58 800.0 181.0 0.14 0.5054 0.853 3027241 ChemDiv3_006809 COc1cccc(c1)c2nn3c(Cc4ccccc4)nnc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F12 compound treatment 3400.0 2260.0 0.8 1640.0 1020.0 0.78 1.1219 0.9999 3027242 ChemDiv3_006810 O=C(NCCc1c[nH]c2ccccc12)c3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F13 compound treatment 4040.0 2900.0 1.03 6040.0 5420.0 4.16 3.671 0.8563 3119946 ChemDiv3_006811 CC(C)C1Cc2[nH]c(=O)c(cc2CO1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F14 compound treatment 1400.0 264.0 0.09 720.0 101.0 0.08 0.1208 0.9955 3027243 ChemDiv3_006812 COc1ccc(cc1)c2nnc(SC3CCOC3=O)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F15 compound treatment 5400.0 4260.0 1.51 680.0 60.6 0.05 1.1025 0.7285 3119947 ChemDiv3_006813 OC(=O)CCC1CCC(=O)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F16 compound treatment 5640.0 4500.0 1.6 1080.0 461.0 0.35 1.3798 0.8432 3119948 ChemDiv3_006814 OC(=O)c1ccc(cc1)S(=O)(=O)Nc2ccc3oc4CCCC(=O)c4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F17 compound treatment 5800.0 4660.0 1.65 640.0 20.6 0.02 1.1811 0.7138 3027244 ChemDiv3_006815 Clc1ccccc1OCCCn2c(=O)sc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F18 compound treatment 2080.0 944.0 0.33 640.0 20.6 0.02 0.2479 0.7398 3119949 ChemDiv3_006816 COC(=O)C1=NNC(C1c2ccc(OC)cc2)C(=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F19 compound treatment 2120.0 984.0 0.35 2560.0 1940.0 1.49 1.3003 0.8497 3027245 ChemDiv3_006817 OC(c1ccco1)P(=O)(O)C2Cc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F20 compound treatment 1400.0 264.0 0.09 1280.0 661.0 0.51 0.4248 0.8237 3119950 ChemDiv3_006818 CC(NC(=O)Cn1cc(C(=O)C2CCCCC2)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F21 compound treatment 2560.0 1420.0 0.51 840.0 221.0 0.17 0.4769 0.8953 1147731 ChemDiv3_006819 COc1ccc(cc1)N2C(=S)SC3CS(=O)(=O)CC32C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F22 compound treatment 920.0 -216.0 -0.08 1000.0 381.0 0.29 0.1524 0.5044 3119951 ChemDiv3_006820 FC(F)(F)c1nc(SCC(=O)N2CCCC2)nc-3c1CCc4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F23 mock treatment 640.0 -496.0 -0.18 1680.0 1060.0 0.81 0.4513 0.5417 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 F24 mock treatment 1280.0 144.0 0.05 1520.0 901.0 0.69 0.525 0.7572 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G01 compound treatment 7360.0 6220.0 2.21 360.0 -259.0 -0.2 1.4204 0.6407 3119952 ChemDiv3_006821 Cc1ccc(cc1c2nnc3c4ccccc4c(C)nn23)S(=O)(=O)NC5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G02 compound treatment 10480.0 9340.0 3.31 960.0 341.0 0.26 2.5287 0.7605 1307285 ChemDiv3_006822 C1C2N(N=C1c3ccco3)C(Oc4ccccc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G03 compound treatment 1720.0 584.0 0.21 600.0 -19.4 -0.01 0.1359 0.6547 3120089 ChemDiv3_006823 CCOP(=S)(OCC)C1(CCCCC1)Nc2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G04 compound treatment 560.0 -576.0 -0.2 960.0 341.0 0.26 0.0404 0.1216 3027246 ChemDiv3_006824 CCC(=O)n1nc(nc1NCc2ccco2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G05 compound treatment 640.0 -496.0 -0.18 680.0 60.6 0.05 -0.0916 -0.5028 3120090 ChemDiv3_006825 O=S(=O)(N1CCN(CCC#N)CC1)c2ccc(C#N)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G06 compound treatment 1200.0 63.8 0.02 920.0 301.0 0.23 0.1792 0.7727 1874090 ChemDiv3_006826 Cc1ccc(cc1)C(=O)c2oc3ccccc3c2NC(=O)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G07 compound treatment 2800.0 1660.0 0.59 880.0 261.0 0.2 0.5588 0.8967 3120091 ChemDiv3_006827 COc1ccc(cc1OC)c2c(C)[nH]nc2c3ccc(O)cc3O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G08 compound treatment 720.0 -416.0 -0.15 480.0 -139.0 -0.11 -0.1801 -0.9875 3120092 ChemDiv3_006828 CCC(=O)Nc1ccc2n3CCN(Cc4ccccc4)Cc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G09 compound treatment 480.0 -656.0 -0.23 520.0 -99.4 -0.08 -0.2186 -0.8921 3027247 ChemDiv3_006829 COc1cccc(Oc2c(oc3cc(OC)ccc3c2=O)C(F)(F)F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G10 compound treatment 800.0 -336.0 -0.12 440.0 -179.0 -0.14 -0.1817 -0.9974 3120093 ChemDiv3_006830 COc1cccc(c1)C2N(CCCN3CCOCC3)C(=O)c4oc5ccccc5c(=O)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G11 compound treatment 800.0 -336.0 -0.12 400.0 -219.0 -0.17 -0.2034 -0.9857 3027248 ChemDiv3_006831 Clc1cccc(NC(=O)C2=CC(=O)N3CCCN=C3S2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G12 compound treatment 680.0 -456.0 -0.16 480.0 -139.0 -0.11 -0.1901 -0.9798 1212660 ChemDiv3_006832 COc1cccc(C2Nc3cccc4cccc(N2)c34)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G13 compound treatment 9160.0 8020.0 2.85 1040.0 421.0 0.32 2.2411 0.7823 1600675 ChemDiv3_006833 CCCc1noc2NC(=C(C#N)C(c12)c3cc(Br)ccc3F)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G14 compound treatment 760.0 -376.0 -0.13 680.0 60.6 0.05 -0.0615 -0.4348 3027249 ChemDiv3_006834 O=C(CC1OCCN(Cc2ccccc2)C1=O)Nc3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G15 compound treatment 760.0 -376.0 -0.13 400.0 -219.0 -0.17 -0.2135 -0.9934 3120094 ChemDiv3_006835 CN(Cc1nc(no1)c2ccc(Cl)cc2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G16 compound treatment 920.0 -216.0 -0.08 440.0 -179.0 -0.14 -0.1516 -0.9619 3027250 ChemDiv3_006836 N1C(/C=C/c2ccccc2)n3c(nc4ccccc34)-c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G17 compound treatment 440.0 -696.0 -0.25 840.0 221.0 0.17 -0.0549 -0.1832 3120095 ChemDiv3_006837 CCOc1ccc(Oc2cc(C)nc(SC)n2)nn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G18 compound treatment 960.0 -176.0 -0.06 1360.0 741.0 0.57 0.3579 0.6256 3120096 ChemDiv3_006838 Cc1ccc(cc1)S(=O)(=O)CC2CSc3ncnc4ncn2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G19 compound treatment 760.0 -376.0 -0.13 1040.0 421.0 0.32 0.134 0.3834 3027251 ChemDiv3_006839 Cc1ccc(c(C)c1)S(=O)(=O)N(C(=O)C2CCCCC2)c3ccc4oc(=O)sc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G20 compound treatment 1240.0 104.0 0.04 1480.0 861.0 0.66 0.4932 0.7453 1136208 ChemDiv3_006840 COc1cc2CCNC3Cc4ccc(O)cc4-c(c1OC)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G21 compound treatment 280.0 -856.0 -0.3 440.0 -179.0 -0.14 -0.3121 -0.936 3027309 ChemDiv3_006841 Cc1ccnc(Nc2nc3ccccc3o2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G22 compound treatment 2600.0 1460.0 0.52 400.0 -219.0 -0.17 0.2481 0.4545 3027310 ChemDiv3_006842 Clc1ccccc1OCCn2cc(C(=O)c3ccco3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G23 mock treatment 560.0 -576.0 -0.2 760.0 141.0 0.11 -0.0682 -0.295 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 G24 mock treatment 1040.0 -96.3 -0.03 440.0 -179.0 -0.14 -0.1215 -0.8565 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H01 compound treatment 640.0 -496.0 -0.18 800.0 181.0 0.14 -0.0264 -0.1179 1707309 ChemDiv3_006843 COc1ccc(CN(C)CCc2ccccn2)c(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H02 compound treatment 4680.0 3540.0 1.26 640.0 20.6 0.02 0.9001 0.716 3027311 ChemDiv3_006844 CC(C)(C)c1cc2nc(cc(N)n2n1)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H03 compound treatment 320.0 -816.0 -0.29 600.0 -19.4 -0.01 -0.2153 -0.7424 3027312 ChemDiv3_006845 COc1ccc(OCC(=O)c2c(O)c3ccccc3oc2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H04 compound treatment 280.0 -856.0 -0.3 400.0 -219.0 -0.17 -0.3339 -0.9613 1225575 ChemDiv3_006846 NS(=O)(=O)c1ccc(CCNC2=CC(=O)OC32CCCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H05 compound treatment 560.0 -576.0 -0.2 360.0 -259.0 -0.2 -0.2853 -0.9999 3027313 ChemDiv3_006847 COc1ccc(Nc2nc(nc3ccccc23)N4CCN(C)CC4)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H06 compound treatment 640.0 -496.0 -0.18 2080.0 1460.0 1.12 0.6684 0.5889 3120097 ChemDiv3_006848 Nc1ncnc2n(Cc3ccccc3)c(SCC(=O)O)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H07 compound treatment 4680.0 3540.0 1.26 640.0 20.6 0.02 0.9001 0.716 3027314 ChemDiv3_006849 CCc1c(O)nc(SCC(=O)N2CCc3ccccc23)n(c4ccc(F)cc4)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H08 compound treatment 800.0 -336.0 -0.12 480.0 -139.0 -0.11 -0.16 -0.9985 1407492 ChemDiv3_006850 COc1cccc(Nc2nc(=O)[nH]nc2C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H09 compound treatment 560.0 -576.0 -0.2 960.0 341.0 0.26 0.0404 0.1216 3027315 ChemDiv3_006851 C1Oc2ccc(cc2O1)c3nn4c(nnc4s3)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H10 compound treatment 560.0 -576.0 -0.2 1440.0 821.0 0.63 0.3009 0.4544 3120098 ChemDiv3_006852 OC(=O)CCNC(=O)c1ccc(NC(=O)Cc2ccc(Cl)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H11 compound treatment 680.0 -456.0 -0.16 920.0 301.0 0.23 0.0488 0.173 3120099 ChemDiv3_006853 COc1ccc(Cc2nn3c(Cc4ccccc4)nnc3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H12 compound treatment 360.0 -776.0 -0.28 560.0 -59.4 -0.05 -0.2269 -0.8131 3027316 ChemDiv3_006854 CCCn1nnnc1NCc2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H13 compound treatment 720.0 -416.0 -0.15 440.0 -179.0 -0.14 -0.2018 -0.9994 3120100 ChemDiv3_006855 Clc1ccc(COc2ccc3OC(=O)CCc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H14 compound treatment 680.0 -456.0 -0.16 520.0 -99.4 -0.08 -0.1684 -0.9411 3027317 ChemDiv3_006856 O=C1NN=C(CC1c2cn(CCC#N)c3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H15 compound treatment 680.0 -456.0 -0.16 440.0 -179.0 -0.14 -0.2118 -0.9968 3120101 ChemDiv3_006857 O=C(Cn1c(=O)n2ncnc2c3c4CCCCc4sc13)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H16 compound treatment 840.0 -296.0 -0.11 480.0 -139.0 -0.11 -0.15 -1.0 3120102 ChemDiv3_006858 CN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc4ccc(O)c(c4)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H17 compound treatment 600.0 -536.0 -0.19 4440.0 3820.0 2.93 1.9396 0.6599 3027318 ChemDiv3_006859 CC(C)(C)c1ccc(OCCCn2c(=O)sc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H18 compound treatment 640.0 -496.0 -0.18 1000.0 381.0 0.29 0.0822 0.2408 3120103 ChemDiv3_006860 Cc1cc2-c3ccccc3NC(c4cccs4)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H19 compound treatment 480.0 -656.0 -0.23 400.0 -219.0 -0.17 -0.2837 -0.9874 3027319 ChemDiv3_006861 FC(F)(F)c1cccc(NC(=O)C2CCCNC2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H20 compound treatment 4120.0 2980.0 1.06 560.0 -59.4 -0.05 0.7162 0.676 3120104 ChemDiv3_006862 OC(=O)Cn1cc(C(=O)C2CC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H21 compound treatment 960.0 -176.0 -0.06 440.0 -179.0 -0.14 -0.1416 -0.9362 3120105 ChemDiv3_006863 CN(C)c1cccc(c1)N2C3CS(=O)(=O)CC3SC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H22 compound treatment 1160.0 23.8 0.01 1720.0 1100.0 0.84 0.6035 0.7141 3027320 ChemDiv3_006864 FC(F)(F)c1cc(nc(SCCC(=O)N2CCCCC2)n1)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H23 mock treatment 1800.0 664.0 0.24 400.0 -219.0 -0.17 0.0474 0.1638 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 H24 mock treatment 1800.0 664.0 0.24 2080.0 1460.0 1.12 0.9594 0.8373 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I01 compound treatment 600.0 -536.0 -0.19 3800.0 3180.0 2.44 1.5921 0.65 3120106 ChemDiv3_006865 Cc1ccc(cc1c2nnc3c4ccccc4c(C)nn23)S(=O)(=O)N5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I02 compound treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 3027321 ChemDiv3_006866 CC1CCC2(CC1)Oc3ccccc3C4CC(=NN42)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I03 compound treatment 280.0 -856.0 -0.3 360.0 -259.0 -0.2 -0.3556 -0.979 3120107 ChemDiv3_006867 CCOP(=S)(OCC)C(O)c1ccccc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I04 compound treatment 400.0 -736.0 -0.26 240.0 -379.0 -0.29 -0.3906 -0.9985 3120108 ChemDiv3_006868 O=C(c1ccccc1)n2nc(nc2NCc3ccco3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I05 compound treatment 320.0 -816.0 -0.29 480.0 -139.0 -0.11 -0.2804 -0.9083 3027322 ChemDiv3_006869 Oc1nc(nc2n(Cc3ccccc3)nnc12)C(=O)NCc4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I06 compound treatment 320.0 -816.0 -0.29 240.0 -379.0 -0.29 -0.4107 -1.0 3120109 ChemDiv3_006870 O=C(Nc1c(oc2ccccc12)C(=O)c3ccccc3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I07 compound treatment 360.0 -776.0 -0.28 320.0 -299.0 -0.23 -0.3572 -0.996 3120110 ChemDiv3_006871 CCc1cc2c(=O)c(coc2c(CN3CCCC(C)C3)c1O)c4nc5ccccc5[nH]4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I08 compound treatment 400.0 -736.0 -0.26 400.0 -219.0 -0.17 -0.3038 -0.9775 3027323 ChemDiv3_006872 O=C(Nc1ccc2n3CCN(Cc4ccccc4)Cc3nc2c1)C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I09 compound treatment 400.0 -736.0 -0.26 280.0 -339.0 -0.26 -0.3689 -1.0 3120111 ChemDiv3_006873 COc1ccc(Oc2coc3cc(OC(=O)N4CCOCC4)ccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I10 compound treatment 440.0 -696.0 -0.25 320.0 -299.0 -0.23 -0.3372 -0.9994 3120112 ChemDiv3_006874 COCCN1C(c2c(oc3ccccc3c2=O)C1=O)c4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I11 compound treatment 920.0 -216.0 -0.08 360.0 -259.0 -0.2 -0.195 -0.914 3027324 ChemDiv3_006875 OC(=O)CSc1nc(ccc1C#N)c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I12 compound treatment 400.0 -736.0 -0.26 400.0 -219.0 -0.17 -0.3038 -0.9775 3027325 ChemDiv3_006876 CC(C)(C)OC(=O)N1C[C@H]2[C@H](NC(=O)c3nsc(Cl)c3Cl)[C@H]2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I13 compound treatment 280.0 -856.0 -0.3 240.0 -379.0 -0.29 -0.4207 -0.9998 3120113 ChemDiv3_006877 NC1=C(CC(=O)N1c2cccc(c2)C(F)(F)F)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I14 compound treatment 920.0 -216.0 -0.08 520.0 -99.4 -0.08 -0.1082 -1.0 3120114 ChemDiv3_006878 Cc1cc(C)nc(Nc2n[nH]c(n2)c3ccccc3C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I15 compound treatment 680.0 -456.0 -0.16 320.0 -299.0 -0.23 -0.277 -0.9853 3027326 ChemDiv3_006879 Cc1cc(Oc2ccc(=O)n(C)n2)nc(SCC(=O)N)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I16 compound treatment 4600.0 3460.0 1.23 280.0 -339.0 -0.26 0.6846 0.5451 3120115 ChemDiv3_006880 OC(=O)CCN1CN(CCC(=O)O)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I17 compound treatment 360.0 -776.0 -0.28 400.0 -219.0 -0.17 -0.3138 -0.9722 3027327 ChemDiv3_006881 CN(C)c1nc(OCCNS(=O)(=O)c2ccc(C)cc2)nc(n1)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I18 compound treatment 360.0 -776.0 -0.28 320.0 -299.0 -0.23 -0.3572 -0.996 1732213 ChemDiv3_006882 Cc1nc2sc3c(NC4CCCCC4)ncnc3c2c5CC(C)(C)OCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I19 compound treatment 400.0 -736.0 -0.26 360.0 -259.0 -0.2 -0.3255 -0.991 3117823 ChemDiv3_006883 COc1ccc(cc1OC)S(=O)(=O)N(C(=O)C2CCCCC2)c3ccc4oc(=O)sc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I20 compound treatment 440.0 -696.0 -0.25 320.0 -299.0 -0.23 -0.3372 -0.9994 1788191 ChemDiv3_006884 COc1cc2CCN(C3Cc4ccc(OC(=O)C)cc4-c(c1OC)c32)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I21 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 3117824 ChemDiv3_006885 CCOC(=O)c1cnc(Nc2nc3ccccc3o2)nc1CSc4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I22 compound treatment 360.0 -776.0 -0.28 360.0 -259.0 -0.2 -0.3355 -0.9873 3027328 ChemDiv3_006886 O=C(c1ccco1)c2cn(Cc3ccccc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I23 mock treatment 960.0 -176.0 -0.06 400.0 -219.0 -0.17 -0.1633 -0.909 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 I24 mock treatment 2040.0 904.0 0.32 320.0 -299.0 -0.23 0.0642 0.1627 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J01 compound treatment 5920.0 4780.0 1.7 760.0 141.0 0.11 1.2763 0.7506 3117825 ChemDiv3_006887 CN(CCc1ccccn1)Cc2ccccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J02 compound treatment 400.0 -736.0 -0.26 800.0 181.0 0.14 -0.0866 -0.2929 3117826 ChemDiv3_006888 Cc1nnc2sc(nn12)c3ccc(NC(=O)COc4ccc(C)cc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J03 compound treatment 400.0 -736.0 -0.26 280.0 -339.0 -0.26 -0.3689 -1.0 3027329 ChemDiv3_006889 Nc1c(cc(C#N)c2nc3ccccc3n12)c4nc5ccccc5[nH]4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J04 compound treatment 360.0 -776.0 -0.28 320.0 -299.0 -0.23 -0.3572 -0.996 3117827 ChemDiv3_006890 CCCN(CCC)S(=O)(=O)c1cccc(c1)c2cn3ccc(C)cc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J05 compound treatment 320.0 -816.0 -0.29 360.0 -259.0 -0.2 -0.3455 -0.9833 3027330 ChemDiv3_006891 COC(=O)c1n[nH]c2C(=O)N(C(=O)c12)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J06 compound treatment 320.0 -816.0 -0.29 360.0 -259.0 -0.2 -0.3455 -0.9833 1190486 ChemDiv3_006892 Sc1nc2ccc(cc2o1)S(=O)(=O)Nc3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J07 compound treatment 320.0 -816.0 -0.29 560.0 -59.4 -0.05 -0.237 -0.8084 3027331 ChemDiv3_006893 CCCCn1cc(C2CC(=O)N(C2=O)c3ccc(Br)cc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J08 compound treatment 400.0 -736.0 -0.26 440.0 -179.0 -0.14 -0.282 -0.9553 3117828 ChemDiv3_006894 CC1CN(CC(C)O1)S(=O)(=O)c2ccc3NC(=O)c4cccc2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J09 compound treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 3117829 ChemDiv3_006895 COc1cc(cc(OC)c1OC)c2nn3c(nnc3s2)c4ccc(cc4)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J10 compound treatment 320.0 -816.0 -0.29 480.0 -139.0 -0.11 -0.2804 -0.9083 3027332 ChemDiv3_006896 OC(=O)CCNC(=O)c1ccc(NC(=O)C(c2ccccc2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J11 compound treatment 440.0 -696.0 -0.25 360.0 -259.0 -0.2 -0.3154 -0.9943 3117830 ChemDiv3_006897 Cc1nn(c(O)c1C2OC(=O)c3ccccc23)c4nc5ccccc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J12 compound treatment 440.0 -696.0 -0.25 240.0 -379.0 -0.29 -0.3806 -0.9966 3117831 ChemDiv3_006898 CCOc1ccc(CNc2ccc(CNc3ncn[nH]3)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J13 compound treatment 3360.0 2220.0 0.79 600.0 -19.4 -0.01 0.5473 0.6937 3027333 ChemDiv3_006899 OC(=O)C1OC(=NC21CC2)c3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J14 compound treatment 560.0 -576.0 -0.2 320.0 -299.0 -0.23 -0.3071 -0.9983 3117832 ChemDiv3_006900 COC(=O)C(CC(=O)c1ccc(Br)cc1)n2cncn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J15 compound treatment 5720.0 4580.0 1.63 480.0 -139.0 -0.11 1.0742 0.6592 3027334 ChemDiv3_006901 CCC1CC(CSc2nnc[nH]2)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J16 compound treatment 480.0 -656.0 -0.23 400.0 -219.0 -0.17 -0.2837 -0.9874 3117833 ChemDiv3_006902 CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NC(Cc4c[nH]c5ccccc45)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J17 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3027335 ChemDiv3_006903 Cc1ccc(cc1)S(=O)(=O)n2c(=O)sc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J18 compound treatment 400.0 -736.0 -0.26 200.0 -419.0 -0.32 -0.4123 -0.9946 3117834 ChemDiv3_006904 Cc1cc2-c3ccccc3NC(c4cccnc4)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J19 compound treatment 320.0 -816.0 -0.29 320.0 -299.0 -0.23 -0.3673 -0.9934 3027336 ChemDiv3_006905 FC(F)(F)c1ccccc1NC(=O)C2CCCNC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J20 compound treatment 480.0 -656.0 -0.23 360.0 -259.0 -0.2 -0.3054 -0.997 3117835 ChemDiv3_006906 CC(C)NC(=O)Cn1cc(C(=O)C(C)(C)C)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J21 compound treatment 360.0 -776.0 -0.28 400.0 -219.0 -0.17 -0.3138 -0.9722 3027337 ChemDiv3_006907 FC(F)(F)c1ccccc1Nc2nc(cs2)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J22 compound treatment 400.0 -736.0 -0.26 360.0 -259.0 -0.2 -0.3255 -0.991 3117836 ChemDiv3_006908 FC(F)(F)c1cc(nc(SCCC(=O)N2CCCc3ccccc23)n1)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J23 mock treatment 3280.0 2140.0 0.76 360.0 -259.0 -0.2 0.397 0.505 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 J24 mock treatment 1120.0 -16.3 -0.01 320.0 -299.0 -0.23 -0.1666 -0.7246 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K01 compound treatment 1600.0 464.0 0.16 880.0 261.0 0.2 0.2578 0.9953 3117837 ChemDiv3_006909 CN(C1CCCCC1)S(=O)(=O)c2ccc(C)c(c2)c3nnc4c5ccccc5c(C)nn34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K02 compound treatment 800.0 -336.0 -0.12 1240.0 621.0 0.48 0.2526 0.5142 3027338 ChemDiv3_006910 Cc1ccc(cc1)N2C(=O)C3SC(=C(C#N)C(C3C2=O)c4ccco4)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K03 compound treatment 11400.0 10300.0 3.64 800.0 181.0 0.14 2.6727 0.7335 3117838 ChemDiv3_006911 CCOc1ccc(cc1)C(Nc2ccccc2)P3(=S)OCCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K04 compound treatment 2640.0 1500.0 0.53 600.0 -19.4 -0.01 0.3667 0.6871 3027339 ChemDiv3_006912 CC(C)C(=O)n1nc(nc1NCc2ccccc2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K05 compound treatment 960.0 -176.0 -0.06 560.0 -59.4 -0.05 -0.0764 -0.9879 3117839 ChemDiv3_006913 Cc1ccc(CNC(=O)c2nc(O)c3nnn(Cc4ccco4)c3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K06 compound treatment 680.0 -456.0 -0.16 920.0 301.0 0.23 0.0488 0.173 3027340 ChemDiv3_006914 CC(C)C(=O)Nc1c(oc2ccccc12)C(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K07 compound treatment 880.0 -256.0 -0.09 480.0 -139.0 -0.11 -0.1399 -0.9967 3117840 ChemDiv3_006915 Nc1oc2c(CN3CCCCCC3)c(O)ccc2c(=O)c1c4nc5ccccc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K08 compound treatment 1240.0 104.0 0.04 1000.0 381.0 0.29 0.2327 0.7899 3117841 ChemDiv3_006916 CS(=O)(=O)Nc1ccc2n3CCN(Cc4ccccc4)Cc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K09 compound treatment 600.0 -536.0 -0.19 4720.0 4100.0 3.15 2.0916 0.6632 3027341 ChemDiv3_006917 COc1cccc(Oc2coc3cc(OC(=O)N(C)C)ccc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K10 compound treatment 1000.0 -136.0 -0.05 640.0 20.6 0.02 -0.023 -0.4516 3117842 ChemDiv3_006918 Cc1nc(sc1C(=O)OCC=C)N2C(c3c(oc4ccc(F)cc4c3=O)C2=O)c5ccc(O)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K11 compound treatment 1240.0 104.0 0.04 440.0 -179.0 -0.14 -0.0713 -0.5005 1615206 ChemDiv3_006919 N#Cc1ccc(nc1SCCN2CCCCC2)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K12 compound treatment 800.0 -336.0 -0.12 1200.0 581.0 0.45 0.2309 0.5003 3117843 ChemDiv3_006920 CCN1CNC(=NC1)Nc2nc(C)c3cc(C)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K13 compound treatment 680.0 -456.0 -0.16 440.0 -179.0 -0.14 -0.2118 -0.9968 3027494 ChemDiv3_006921 CCOc1csc2nc(C)cc(C)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K14 compound treatment 1680.0 544.0 0.19 640.0 20.6 0.02 0.1476 0.7626 3117844 ChemDiv3_006922 CCc1ccc(cc1)C2C3=C(CCCC3=O)Nc4nn(c(O)c24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K15 compound treatment 1960.0 824.0 0.29 480.0 -139.0 -0.11 0.131 0.4209 3027495 ChemDiv3_006923 Cc1ccccc1OC2C(N(CCc3ccc(F)cc3)C2=O)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K16 compound treatment 1280.0 144.0 0.05 400.0 -219.0 -0.17 -0.083 -0.4718 3117845 ChemDiv3_006924 Cn1c2ccc(F)cc2c3nnc(NN)nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K17 compound treatment 640.0 -496.0 -0.18 2080.0 1460.0 1.12 0.6684 0.5889 3117846 ChemDiv3_006925 Cc1nc(NS(=O)(=O)c2ccccc2)sc1NC(=O)Nc3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K18 compound treatment 4840.0 3700.0 1.31 360.0 -259.0 -0.2 0.7883 0.5932 1216864 ChemDiv3_006926 CC(C)CNc1ncnc2c1sc3nc(C(C)C)c4COC(C)(C)Cc4c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K19 compound treatment 4240.0 3100.0 1.1 520.0 -99.4 -0.08 0.7246 0.6565 3117847 ChemDiv3_006927 Cc1ccc(c(C)c1)S(=O)(=O)N(C(=O)Oc2ccccc2)c3ccc4oc(=O)sc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K20 compound treatment 3120.0 1980.0 0.7 5720.0 5100.0 3.92 3.2665 0.821 3027496 ChemDiv3_006928 CC1(C)Oc2ccc3ccc(=O)oc3c2C(/C=N/O)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K21 compound treatment 18040.0 16900.0 6.0 20320.0 19700.0 15.12 14.9349 0.9179 3117978 ChemDiv3_006929 CC1(C)CC(=O)C2=C(C1)NC(=NC2c3ccccc3)Nc4nc5ccccc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K22 compound treatment 1160.0 23.8 0.01 640.0 20.6 0.02 0.0172 0.9563 3027497 ChemDiv3_006930 CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)CC)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K23 mock treatment 7520.0 6380.0 2.26 560.0 -59.4 -0.05 1.5691 0.6927 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 K24 mock treatment 720.0 -416.0 -0.15 720.0 101.0 0.08 -0.0498 -0.2987 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L01 compound treatment 5120.0 3980.0 1.41 960.0 341.0 0.26 1.1842 0.824 3117979 ChemDiv3_006931 CC(C)n1cc(cn1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L02 compound treatment 6960.0 5820.0 2.07 1040.0 421.0 0.32 1.6892 0.8078 3117980 ChemDiv3_006932 COc1ccc(cc1)C2NC(=O)c3c4CCCc4sc3N2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L03 compound treatment 680.0 -456.0 -0.16 560.0 -59.4 -0.05 -0.1467 -0.8723 3027540 ChemDiv3_006933 CC(C)CC(NS(=O)(=O)c1ccc2[nH]c(=O)c(=O)[nH]c2c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L04 compound treatment 600.0 -536.0 -0.19 360.0 -259.0 -0.2 -0.2753 -0.9997 3117981 ChemDiv3_006934 O=S(=O)(N1CCCCC1)c2cccc(c2)c3cn4ccccc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L05 compound treatment 680.0 -456.0 -0.16 640.0 20.6 0.02 -0.1032 -0.6348 3027541 ChemDiv3_006935 COC(=O)c1n[nH]c2C(=O)N(C3CCCCC3)C(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L06 compound treatment 680.0 -456.0 -0.16 440.0 -179.0 -0.14 -0.2118 -0.9968 3117982 ChemDiv3_006936 Cn1c(=O)n(C)c2cc(ccc12)S(=O)(=O)NCCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L07 compound treatment 4200.0 3060.0 1.09 640.0 20.6 0.02 0.7797 0.7173 1330090 ChemDiv3_006937 COc1cc2CCN(CCC(=O)O)Cc2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L08 compound treatment 560.0 -576.0 -0.2 600.0 -19.4 -0.01 -0.1551 -0.7565 3117983 ChemDiv3_006938 OC(=O)c1ccc2nc(sc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L09 compound treatment 960.0 -176.0 -0.06 520.0 -99.4 -0.08 -0.0981 -0.9951 3117984 ChemDiv3_006939 C(c1nnc2sc(Nc3ccccc3)nn12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L10 compound treatment 6920.0 5780.0 2.05 600.0 -19.4 -0.01 1.4403 0.702 3027542 ChemDiv3_006940 O/N=C(/C(=O)NCC1CCNCC1)\c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L11 compound treatment 600.0 -536.0 -0.19 280.0 -339.0 -0.26 -0.3187 -0.9881 3117985 ChemDiv3_006941 Cc1nonc1OCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L12 compound treatment 480.0 -656.0 -0.23 480.0 -139.0 -0.11 -0.2403 -0.9378 3117986 ChemDiv3_006942 COC(=O)c1ccccc1NC(=O)C(C)N2c3cccc4cccc(c34)S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L13 compound treatment 8520.0 7380.0 2.62 400.0 -219.0 -0.17 1.7331 0.6603 3027543 ChemDiv3_006943 Cc1ccccc1N2C(=O)c3ccccc3S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L14 compound treatment 1160.0 23.8 0.01 520.0 -99.4 -0.08 -0.048 -0.6252 3117987 ChemDiv3_006944 OCCN1CCOC2(O)C1=C/C(=N\S(=O)(=O)c3ccccc3)/c4ccccc42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L15 compound treatment 5480.0 4340.0 1.54 5040.0 4420.0 3.39 3.4894 0.9362 3027544 ChemDiv3_006945 CC(C)CNCC1COc2ccccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L16 compound treatment 640.0 -496.0 -0.18 520.0 -99.4 -0.08 -0.1784 -0.9299 3117988 ChemDiv3_006946 OC(=O)C1CCCN1S(=O)(=O)c2ccc3NC(=O)c4cccc2c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L17 compound treatment 400.0 -736.0 -0.26 480.0 -139.0 -0.11 -0.2603 -0.9224 3027545 ChemDiv3_006947 OC(=O)c1ccc(NC(=O)CSC2c3ccccc3Oc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L18 compound treatment 720.0 -416.0 -0.15 480.0 -139.0 -0.11 -0.1801 -0.9875 3117989 ChemDiv3_006948 COc1ccc(cc1)C2Nc3ccccc3-c4cc(C)nn24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L19 compound treatment 1040.0 -96.3 -0.03 6600.0 5980.0 4.59 3.2225 0.7018 3027546 ChemDiv3_006949 CC(=O)N1CCc2cc3nc(C)cc(C)c3cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L20 compound treatment 800.0 -336.0 -0.12 600.0 -19.4 -0.01 -0.0949 -0.7891 3117990 ChemDiv3_006950 COc1ccc(OCCn2cc(C(=O)C(C)(C)C)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L21 compound treatment 1080.0 -56.3 -0.02 800.0 181.0 0.14 0.084 0.5992 3027547 ChemDiv3_006951 Cc1oc(cc1c2nn3c(nnc3s2)c4ccco4)c5ccc(Cl)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L22 compound treatment 640.0 -496.0 -0.18 760.0 141.0 0.11 -0.0481 -0.2331 3117991 ChemDiv3_006952 FC(F)(F)c1cc(nc(SCCC(=O)NCCc2ccccc2)n1)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L23 mock treatment 1200.0 63.8 0.02 480.0 -139.0 -0.11 -0.0597 -0.5456 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 L24 mock treatment 1000.0 -136.0 -0.05 1680.0 1060.0 0.81 0.5416 0.664 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M01 compound treatment 720.0 -416.0 -0.15 1000.0 381.0 0.29 0.1022 0.3122 3027548 ChemDiv3_006953 CCCCN(C)S(=O)(=O)c1ccc(C)c(c1)c2nnc3c4ccccc4c(C)nn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M02 compound treatment 520.0 -616.0 -0.22 480.0 -139.0 -0.11 -0.2302 -0.946 3117992 ChemDiv3_006954 Cc1ccc2nc(oc2c1)c3cccc(n3)c4nc5ccc(C)cc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M03 compound treatment 3760.0 2620.0 0.93 280.0 -339.0 -0.26 0.4739 0.4903 3117993 ChemDiv3_006955 Cc1ccc(NC(=O)CC2(C(=O)c3ccccc3C2=O)c4ccc(Br)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M04 compound treatment 800.0 -336.0 -0.12 560.0 -59.4 -0.05 -0.1166 -0.9129 3027549 ChemDiv3_006956 CC(=O)n1nc(nc1NCc2ccc(F)cc2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M05 compound treatment 1640.0 504.0 0.18 520.0 -99.4 -0.08 0.0724 0.3728 3117994 ChemDiv3_006957 Oc1nc(nc2n(Cc3ccc4OCOc4c3)nnc12)C(=O)Nc5ccccc5Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M06 compound treatment 600.0 -536.0 -0.19 680.0 60.6 0.05 -0.1016 -0.5187 3027550 ChemDiv3_006958 COc1ccc(cc1)C(=O)c2oc3ccccc3c2NC(=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M07 compound treatment 600.0 -536.0 -0.19 640.0 20.6 0.02 -0.1233 -0.646 3117995 ChemDiv3_006959 CCOC(=O)c1oc2c(CN3CCN(C)CC3)c(O)ccc2c(=O)c1c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M08 compound treatment 920.0 -216.0 -0.08 640.0 20.6 0.02 -0.043 -0.5494 3027551 ChemDiv3_006960 Clc1ccc(NC(=O)CN2C(=O)COc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M09 compound treatment 1040.0 -96.3 -0.03 640.0 20.6 0.02 -0.0129 -0.3437 3117996 ChemDiv3_006961 CCOc1ccccc1Oc2c(C)oc3cc(O)ccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M10 compound treatment 880.0 -256.0 -0.09 440.0 -179.0 -0.14 -0.1616 -0.9797 3117997 ChemDiv3_006962 Cc1ccc(nc1)N2C(c3c(oc4cc(C)c(C)cc4c3=O)C2=O)c5ccc(O)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M11 compound treatment 760.0 -376.0 -0.13 1600.0 981.0 0.75 0.438 0.5728 1531927 ChemDiv3_006963 N#Cc1ccc(nc1SCc2ccccn2)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M12 compound treatment 600.0 -536.0 -0.19 520.0 -99.4 -0.08 -0.1885 -0.9195 3117998 ChemDiv3_006964 CCCCN1CNC(=NC1)Nc2nc(C)c3ccccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M13 compound treatment 1440.0 304.0 0.11 760.0 141.0 0.11 0.1525 1.0 3027552 ChemDiv3_006965 CCC1CCc2[nH]c(=S)c(C#N)c(c2C1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M14 compound treatment 800.0 -336.0 -0.12 840.0 221.0 0.17 0.0354 0.171 3117999 ChemDiv3_006966 O=C(CN1C(=O)CSC1=O)Nc2ccccc2N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M15 compound treatment 2880.0 1740.0 0.62 680.0 60.6 0.05 0.4703 0.7582 3118000 ChemDiv3_006967 COc1ccc(OC2C(N(Cc3ccc(F)cc3)C2=O)c4ccc(OC)c(OC)c4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M16 compound treatment 760.0 -376.0 -0.13 360.0 -259.0 -0.2 -0.2352 -0.9811 3027553 ChemDiv3_006968 CCn1c2ccc(F)cc2c3nnc(NN)nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M17 compound treatment 880.0 -256.0 -0.09 520.0 -99.4 -0.08 -0.1182 -0.9962 3118001 ChemDiv3_006969 Oc1ccc(NC(=O)C2(CCCC2)c3ccccc3)cc1c4nc5ccccc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M18 compound treatment 920.0 -216.0 -0.08 600.0 -19.4 -0.01 -0.0648 -0.8287 1296351 ChemDiv3_006970 CCN(CC)CCNc1ncnc2c1sc3nc(C(C)C)c4CCCCc4c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M19 compound treatment 1160.0 23.8 0.01 920.0 301.0 0.23 0.1692 0.7324 3118002 ChemDiv3_006971 COc1ccc(cc1OC)S(=O)(=O)N(C(=O)Oc2ccccc2)c3ccc4oc(=O)sc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M20 compound treatment 400.0 -736.0 -0.26 800.0 181.0 0.14 -0.0866 -0.2929 3027554 ChemDiv3_006972 CN/C=C/1\C(=O)C(C)(C)Oc2ccc3ccc(=O)oc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M21 compound treatment 1160.0 23.8 0.01 760.0 141.0 0.11 0.0823 0.76 3118003 ChemDiv3_006973 COc1ccccc1C2C(=C3N=C(N)c4ccccc4N3C5=C2C(=O)CCC5)C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M22 compound treatment 880.0 -256.0 -0.09 640.0 20.6 0.02 -0.0531 -0.5751 3027555 ChemDiv3_006974 Fc1cnc(nc1N2CCc3ccccc23)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M23 mock treatment 760.0 -376.0 -0.13 720.0 101.0 0.08 -0.0397 -0.2577 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 M24 mock treatment 880.0 -256.0 -0.09 880.0 261.0 0.2 0.0772 0.3513 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N01 compound treatment 1280.0 144.0 0.05 960.0 341.0 0.26 0.221 0.8294 1879463 ChemDiv3_006975 CSc1nnc2nc3n(C)c4ccccc4c3nn12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N02 compound treatment 1400.0 264.0 0.09 560.0 -59.4 -0.05 0.0339 0.3261 3118004 ChemDiv3_006976 COc1ccc(cc1)c2nc(SC)c3COC(C)(C)Cc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N03 compound treatment 600.0 -536.0 -0.19 560.0 -59.4 -0.05 -0.1667 -0.8524 3027605 ChemDiv3_006977 OC(=O)C(Cc1ccccc1)NS(=O)(=O)c2ccc3[nH]c(=O)c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N04 compound treatment 1000.0 -136.0 -0.05 560.0 -59.4 -0.05 -0.0664 -0.9996 3118005 ChemDiv3_006978 CCOc1cc(ccc1O)C2N(CCc3ccc(OC)cc3)C(=O)c4oc5ccc(F)cc5c(=O)c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N05 compound treatment 1320.0 184.0 0.07 560.0 -59.4 -0.05 0.0139 0.1744 3027606 ChemDiv3_006979 COC(=O)c1n[nH]c2C(=O)N(Cc3ccccc3)C(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N06 compound treatment 760.0 -376.0 -0.13 600.0 -19.4 -0.01 -0.1049 -0.781 3118006 ChemDiv3_006980 COc1ccc(cc1)N(C(=O)C(C)C)S(=O)(=O)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N07 compound treatment 480.0 -656.0 -0.23 480.0 -139.0 -0.11 -0.2403 -0.9378 1477484 ChemDiv3_006981 CNCc1cc2ccccc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N08 compound treatment 480.0 -656.0 -0.23 480.0 -139.0 -0.11 -0.2403 -0.9378 3118135 ChemDiv3_006982 COc1ccccc1C(CCNCc2ccccc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N09 compound treatment 600.0 -536.0 -0.19 760.0 141.0 0.11 -0.0582 -0.2659 3027607 ChemDiv3_006983 C(Cc1ccccc1)c2nn3c(COc4ccccc4)nnc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N10 compound treatment 960.0 -176.0 -0.06 600.0 -19.4 -0.01 -0.0547 -0.8514 3118136 ChemDiv3_006984 O/N=C/c1ccc(cn1)C(=O)NCC2CCCO2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N11 compound treatment 800.0 -336.0 -0.12 720.0 101.0 0.08 -0.0297 -0.209 1579314 ChemDiv3_006985 COc1cccc(Nc2cc(C)c3ccccc3n2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N12 compound treatment 880.0 -256.0 -0.09 640.0 20.6 0.02 -0.0531 -0.5751 3118137 ChemDiv3_006986 CC(N1c2cccc3cccc(c23)S1(=O)=O)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N13 compound treatment 560.0 -576.0 -0.2 640.0 20.6 0.02 -0.1333 -0.6503 3118138 ChemDiv3_006987 COc1ccc(cc1)N2C(=O)c3ccccc3S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N14 compound treatment 1040.0 -96.3 -0.03 720.0 101.0 0.08 0.0305 0.361 3027608 ChemDiv3_006988 Cc1oc2ccc(NS(=O)(=O)c3ccccc3)cc2c1C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N15 compound treatment 720.0 -416.0 -0.15 720.0 101.0 0.08 -0.0498 -0.2987 3118139 ChemDiv3_006989 Cc1ccc2nc(O)c(cc2c1)c3noc(n3)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N16 compound treatment 760.0 -376.0 -0.13 680.0 60.6 0.05 -0.0615 -0.4348 3118140 ChemDiv3_006990 CCC(NCC(O)Cn1c2ccccc2c3ccccc13)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N17 compound treatment 720.0 -416.0 -0.15 600.0 -19.4 -0.01 -0.1149 -0.7744 3027609 ChemDiv3_006991 O=C1C(Oc2ccccc2)C(N1C3CCCC3)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N18 compound treatment 800.0 -336.0 -0.12 680.0 60.6 0.05 -0.0514 -0.4016 3118141 ChemDiv3_006992 Cc1cc2-c3cc(C)ccc3NC(c4cccnc4)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N19 compound treatment 6800.0 5660.0 2.01 680.0 60.6 0.05 1.4536 0.7233 1141558 ChemDiv3_006993 C=CC1CN2CCC1CC2C(OC(=O)c3ccco3)c4ccnc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N20 compound treatment 1160.0 23.8 0.01 680.0 60.6 0.05 0.0389 0.8217 3027610 ChemDiv3_006994 Cc1ccccc1OCCCn2cc(C(=O)C(C)(C)C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N21 compound treatment 1120.0 -16.3 -0.01 560.0 -59.4 -0.05 -0.0363 -0.7903 3118142 ChemDiv3_006995 Clc1ccc2nc(NC3=NCN(CCN4CCOCC4)CN3)nc(c5ccccc5)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N22 compound treatment 840.0 -296.0 -0.11 720.0 101.0 0.08 -0.0197 -0.1508 3118143 ChemDiv3_006996 FC(F)(F)c1cc(nc(SCCC(=O)NCc2ccncc2)n1)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N23 mock treatment 640.0 -496.0 -0.18 800.0 181.0 0.14 -0.0264 -0.1179 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 N24 mock treatment 960.0 -176.0 -0.06 680.0 60.6 0.05 -0.0113 -0.1448 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O01 compound treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 3027611 ChemDiv3_006997 COc1ccc(cc1S(=O)(=O)NC(C)(C)C)c2nnc3c4ccccc4c(C)nn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O02 compound treatment 320.0 -816.0 -0.29 200.0 -419.0 -0.32 -0.4324 -0.9986 3118144 ChemDiv3_006998 C(c1ccc2[nH]cnc2c1)c3ccc4[nH]cnc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O03 compound treatment 240.0 -896.0 -0.32 200.0 -419.0 -0.32 -0.4525 -1.0 3027612 ChemDiv3_006999 NC(=N)NC(=N)Nc1ccccc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O04 compound treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 3118145 ChemDiv3_007000 COc1ccc(CC(=O)n2nc(nc2NCc3ccco3)c4ccc(Cl)cc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O05 compound treatment 3720.0 2580.0 0.92 440.0 -179.0 -0.14 0.5508 0.5942 3027613 ChemDiv3_007001 CCc1nnc(Cn2nnc3c(O)nc(nc23)C(=O)Nc4ccc(C)cc4)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O06 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3118146 ChemDiv3_007002 Clc1ccc(cc1)C(=O)Nc2c(oc3ccccc23)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O07 compound treatment 280.0 -856.0 -0.3 440.0 -179.0 -0.14 -0.3121 -0.936 3118147 ChemDiv3_007003 COc1ccc(cc1)c2c(C)oc3c(CN4CCN(C)CC4)c(O)ccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O08 compound treatment 400.0 -736.0 -0.26 360.0 -259.0 -0.2 -0.3255 -0.991 3027614 ChemDiv3_007004 Cc1nn2c(nnc2c3ccccc13)c4ccc(NC(=O)c5ccccc5Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O09 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 3118148 ChemDiv3_007005 Cc1ccc(OCC(O)Cn2c(=N)n(CC=C)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O10 compound treatment 360.0 -776.0 -0.28 280.0 -339.0 -0.26 -0.3789 -0.9996 3027615 ChemDiv3_007006 Cc1ccc(Cn2cc(CO)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O11 compound treatment 360.0 -776.0 -0.28 240.0 -379.0 -0.29 -0.4007 -0.9996 1633269 ChemDiv3_007007 CC(C)(C)C(=O)CSc1nc2C3CCN(CC3)c2cc1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O12 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 3027616 ChemDiv3_007008 CCCCN1CNC(=NC1)Nc2nc3ccccc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O13 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 3118149 ChemDiv3_007009 Cc1[nH]nc2OC(=C(C#N)C3(CCN(CC3)C(=O)c4ccccc4)c12)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O14 compound treatment 360.0 -776.0 -0.28 320.0 -299.0 -0.23 -0.3572 -0.996 3027617 ChemDiv3_007010 CCN1C(c2ccccc2)n3c(nc4ccccc34)-c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O15 compound treatment 200.0 -936.0 -0.33 280.0 -339.0 -0.26 -0.4191 -0.9928 3118150 ChemDiv3_007011 COC(=O)c1ccc(cc1)C2C(Oc3ccc(OC)cc3)C(=O)N2Cc4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O16 compound treatment 360.0 -776.0 -0.28 560.0 -59.4 -0.05 -0.2269 -0.8131 3027618 ChemDiv3_007012 FC(F)(F)c1cccc2c3nc4ccccc4nc3[nH]c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O17 compound treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 3118151 ChemDiv3_007013 COC(=O)C1=NN(C2C1C(=O)N(C2=O)c3ccccc3OC)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O18 compound treatment 280.0 -856.0 -0.3 200.0 -419.0 -0.32 -0.4424 -0.9996 1305651 ChemDiv3_007014 CC(C)c1nc2sc3c(NCC4CCCO4)ncnc3c2c5CCCCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O19 compound treatment 400.0 -736.0 -0.26 320.0 -299.0 -0.23 -0.3472 -0.998 3027619 ChemDiv3_007015 CC(C)C(=O)N(c1ccc2oc(=O)sc2c1)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O20 compound treatment 280.0 -856.0 -0.3 360.0 -259.0 -0.2 -0.3556 -0.979 1486140 ChemDiv3_007016 CC1=C(Cc2cc3ccc(=O)oc3cc2O)CC(C)(C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O21 compound treatment 400.0 -736.0 -0.26 240.0 -379.0 -0.29 -0.3906 -0.9985 3118152 ChemDiv3_007017 CC1(C)CC(=O)C2=C(C1)N3C(=C(C#N)C2c4cccnc4)N=C(N)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O22 compound treatment 320.0 -816.0 -0.29 320.0 -299.0 -0.23 -0.3673 -0.9934 3027672 ChemDiv3_007018 OC(=O)Cn1c2ccc(Br)cc2c3nc4ccccc4nc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O23 mock treatment 280.0 -856.0 -0.3 320.0 -299.0 -0.23 -0.3773 -0.9905 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 O24 mock treatment 280.0 -856.0 -0.3 360.0 -259.0 -0.2 -0.3556 -0.979 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P01 compound treatment 440.0 -696.0 -0.25 320.0 -299.0 -0.23 -0.3372 -0.9994 3118153 ChemDiv3_007019 C(Sc1nnc-2c(OC=Nc3ccccc32)n1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P02 compound treatment 160.0 -976.0 -0.35 280.0 -339.0 -0.26 -0.4291 -0.9902 3027673 ChemDiv3_007020 Cc1cc(C)nc(SCc2cnc(C)nc2N)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P03 compound treatment 240.0 -896.0 -0.32 240.0 -379.0 -0.29 -0.4308 -0.999 3118154 ChemDiv3_007021 Cc1cc(C)c(C(=O)/C=C(\N2CCCC2)/C(F)(F)F)c(=O)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P04 compound treatment 280.0 -856.0 -0.3 240.0 -379.0 -0.29 -0.4207 -0.9998 1726419 ChemDiv3_007022 Cc1[nH]c2ccc(cc2c1CC(=O)O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P05 compound treatment 440.0 -696.0 -0.25 360.0 -259.0 -0.2 -0.3154 -0.9943 3118155 ChemDiv3_007023 COc1ccc(cc1)C2N(OC(=O)N2c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P06 compound treatment 360.0 -776.0 -0.28 240.0 -379.0 -0.29 -0.4007 -0.9996 3027674 ChemDiv3_007024 CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)/Sc4cc(OC)ccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P07 compound treatment 240.0 -896.0 -0.32 280.0 -339.0 -0.26 -0.409 -0.9951 3118156 ChemDiv3_007025 COc1ccc(cc1OC)c2onc3ccc4c5ccccc5oc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P08 compound treatment 240.0 -896.0 -0.32 360.0 -259.0 -0.2 -0.3656 -0.9746 3118157 ChemDiv3_007026 Cc1ccc(cc1)S(=O)(=O)NCCC(c2ccco2)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P09 compound treatment 320.0 -816.0 -0.29 400.0 -219.0 -0.17 -0.3238 -0.9667 3027675 ChemDiv3_007027 OC(=O)CCN/C=C/1\C(=O)Oc2ccccc2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P10 compound treatment 320.0 -816.0 -0.29 280.0 -339.0 -0.26 -0.389 -0.9986 3027676 ChemDiv3_007028 O/N=C/C(=O)NCc1ccccn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P11 compound treatment 600.0 -536.0 -0.19 360.0 -259.0 -0.2 -0.2753 -0.9997 3118158 ChemDiv3_007029 COc1ccc(Nc2nc3ccc(C)cc3nc2Nc4ccc(OC)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P12 compound treatment 240.0 -896.0 -0.32 200.0 -419.0 -0.32 -0.4525 -1.0 3118159 ChemDiv3_007030 CC(N1c2cccc3cccc(c23)S1(=O)=O)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P13 compound treatment 320.0 -816.0 -0.29 360.0 -259.0 -0.2 -0.3455 -0.9833 3027677 ChemDiv3_007031 COCc1cc(C)nc2sc(C(=O)N3CCN(CC3)c4ccccc4)c(N)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P14 compound treatment 280.0 -856.0 -0.3 280.0 -339.0 -0.26 -0.399 -0.9971 3118160 ChemDiv3_007032 Oc1ccc(NS(=O)(=O)c2ccccc2)cc1Sc3nc[nH]n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P15 compound treatment 320.0 -816.0 -0.29 400.0 -219.0 -0.17 -0.3238 -0.9667 1714084 ChemDiv3_007033 COc1ccc(Br)cc1S(=O)(=O)N2CCN(Cc3ccc4OCOc4c3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P16 compound treatment 360.0 -776.0 -0.28 320.0 -299.0 -0.23 -0.3572 -0.996 3118289 ChemDiv3_007034 CSc1nc2NC(C)(C)CC(=O)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P17 compound treatment 2600.0 1460.0 0.52 360.0 -259.0 -0.2 0.2264 0.4071 3118290 ChemDiv3_007035 COC(=O)c1ccc(cc1)C2C(Oc3ccccc3)C(=O)N2CCc4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P18 compound treatment 200.0 -936.0 -0.33 320.0 -299.0 -0.23 -0.3974 -0.9838 3027678 ChemDiv3_007036 Cc1cc2-c3cccc(C)c3NC(/C=C\c4ccccc4)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P19 compound treatment 360.0 -776.0 -0.28 360.0 -259.0 -0.2 -0.3355 -0.9873 1446881 ChemDiv3_007037 CCOC(=O)NC1CCS(=O)(=O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P20 compound treatment 520.0 -616.0 -0.22 160.0 -459.0 -0.35 -0.4039 -0.9736 3027679 ChemDiv3_007038 CC(C)(C)C(=O)c1cn(CC(=O)O)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P21 compound treatment 2600.0 1460.0 0.52 280.0 -339.0 -0.26 0.1829 0.3149 3118291 ChemDiv3_007039 COC(=O)CC1N(CCNC1=O)C(=O)NS(=O)(=O)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P22 compound treatment 480.0 -656.0 -0.23 280.0 -339.0 -0.26 -0.3488 -0.9984 3118292 ChemDiv3_007040 FC(F)(F)c1cc(nc(SCCC(=O)Nc2ccccc2)n1)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P23 mock treatment 480.0 -656.0 -0.23 440.0 -179.0 -0.14 -0.262 -0.9686 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2020 P24 mock treatment 320.0 -816.0 -0.29 240.0 -379.0 -0.29 -0.4107 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A01 compound treatment 360.0 -543.0 -0.19 3080.0 2310.0 1.77 1.1177 0.6267 1539835 ChemDiv3_007393 Fc1ccccc1C(=O)NCCn2cc(SCC(=O)N3CCCCC3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A02 compound treatment 360.0 -543.0 -0.19 7080.0 6310.0 4.84 3.2892 0.6785 3119324 ChemDiv3_007394 O=C(NCCCN1CCCCC1)c2ccc3c(=O)n4CCCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A03 compound treatment 600.0 -303.0 -0.11 360.0 -410.0 -0.32 -0.2986 -0.8973 3119325 ChemDiv3_007395 COc1ccc(cc1Cl)n2nc(C(=O)NCC(=O)NC3CCCCCC3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A04 compound treatment 760.0 -143.0 -0.05 240.0 -530.0 -0.41 -0.3236 -0.7888 3027601 ChemDiv3_007396 Cc1c(sc2nc3CCCn3c(=O)c12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A05 compound treatment 560.0 -343.0 -0.12 360.0 -410.0 -0.32 -0.3087 -0.9142 3027602 ChemDiv3_007397 CC(=O)Nn1cc(C(=O)O)c2ccccc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A06 compound treatment 360.0 -543.0 -0.19 560.0 -210.0 -0.16 -0.2503 -0.9962 3119326 ChemDiv3_007398 CC1CC(C)(C)NC(=S)N1CCC(=O)Nc2c(C)n(C)n(c3ccccc3)c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A07 compound treatment 360.0 -543.0 -0.19 360.0 -410.0 -0.32 -0.3588 -0.9721 3119327 ChemDiv3_007399 COc1ccc(NC(=O)Cn2ccc3ccccc3c2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A08 compound treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 3119328 ChemDiv3_007400 CN(Cc1ccccc1)S(=O)(=O)c2cc(Br)cc3CCN(C(=O)C)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A09 compound treatment 400.0 -503.0 -0.18 240.0 -530.0 -0.41 -0.4139 -0.9313 3027661 ChemDiv3_007401 COC(=O)Cn1cnc2sc(C)c(c2c1=O)S(=O)(=O)N3CC(C)CC(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A10 compound treatment 320.0 -583.0 -0.21 800.0 29.7 0.02 -0.13 -0.6254 3119329 ChemDiv3_007402 CC(C)CCNC(=O)c1cc(Sc2ccc(F)cc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A11 compound treatment 360.0 -543.0 -0.19 280.0 -490.0 -0.38 -0.4023 -0.9515 3119330 ChemDiv3_007403 COc1ccccc1N2CCN(CC2)C(=O)c3cnc(Nc4ccc(C)c(Cl)c4)c5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A12 compound treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 1295744 ChemDiv3_007404 COC(=O)C(C)Sc1ncnc2n(cc(c3ccccc3)c12)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A13 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3119331 ChemDiv3_007405 COc1cccc(c1)C2C(C(=O)O)c3ccccc3C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A14 compound treatment 240.0 -663.0 -0.24 240.0 -530.0 -0.41 -0.4541 -0.9659 3027666 ChemDiv3_007406 COc1ccc(cc1)n2nc(C(=O)NCC(=O)N3CCCC3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A15 compound treatment 360.0 -543.0 -0.19 520.0 -250.0 -0.19 -0.272 -1.0 3119332 ChemDiv3_007407 O=C(CCNC(=O)Cn1ccc2ccccc2c1=O)NC3CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A16 compound treatment 320.0 -583.0 -0.21 280.0 -490.0 -0.38 -0.4123 -0.9601 1729397 ChemDiv3_007408 CCC(=O)N1CC(=O)Nc2ccc(F)cc2C1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A17 compound treatment 2640.0 1740.0 0.62 200.0 -570.0 -0.44 0.1262 0.167 3027669 ChemDiv3_007409 O=C(NCCC1=CCCCC1)c2cc3c(=O)[nH]c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A18 compound treatment 3240.0 2340.0 0.83 400.0 -370.0 -0.28 0.3853 0.4396 1492777 ChemDiv3_007410 COc1ccccc1c2nnc(NC(=O)c3ccc(cc3)S(=O)(=O)N4CC(C)OC(C)C4)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A19 compound treatment 280.0 -623.0 -0.22 360.0 -410.0 -0.32 -0.3789 -0.9849 3119333 ChemDiv3_007411 CC1CCCN(C1)C(=O)Cc2cn(Cc3cccc(Cl)c3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A20 compound treatment 520.0 -383.0 -0.14 440.0 -330.0 -0.25 -0.2753 -0.9571 3027725 ChemDiv3_007412 COCc1nnc(NC(=O)c2ccc(cc2)S(=O)(=O)N(CC=C)CC=C)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A21 compound treatment 240.0 -663.0 -0.24 480.0 -290.0 -0.22 -0.3238 -0.9996 3119334 ChemDiv3_007413 COc1ccc(CCNC(=O)CSc2cc(Cl)nc3ccc(C)cc23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A22 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3027727 ChemDiv3_007414 O=C(CCN1C(=O)C2C3CC(C=C3)C2C1=O)NC(c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A23 mock treatment 360.0 -543.0 -0.19 280.0 -490.0 -0.38 -0.4023 -0.9515 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 A24 mock treatment 360.0 -543.0 -0.19 320.0 -450.0 -0.35 -0.3805 -0.9618 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B01 compound treatment 360.0 -543.0 -0.19 280.0 -490.0 -0.38 -0.4023 -0.9515 3119335 ChemDiv3_007415 CC(C)Cc1ccc(cc1)S(=O)(=O)N2CCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B02 compound treatment 560.0 -343.0 -0.12 360.0 -410.0 -0.32 -0.3087 -0.9142 3119336 ChemDiv3_007416 CCCCn1/c(=N\C(=O)C(C)(C)C)/c(cc2c(=O)n3ccccc3nc12)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B03 compound treatment 4280.0 3380.0 1.2 360.0 -410.0 -0.32 0.6245 0.5041 1729864 ChemDiv3_007417 COc1ccc(cc1OC)S(=O)(=O)Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B04 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3119337 ChemDiv3_007418 CCC(=O)Oc1c(Sc2ccc(C)cc2)c(C)nn1C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B05 compound treatment 480.0 -423.0 -0.15 280.0 -490.0 -0.38 -0.3722 -0.9185 3027732 ChemDiv3_007419 Cc1ccc(CN(Cc2ccco2)C(=S)Nc3c(C)cc(C)cc3C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B06 compound treatment 4040.0 3140.0 1.11 800.0 29.7 0.02 0.8031 0.7214 3119338 ChemDiv3_007420 Clc1ccc2[nH]c3CCN(Cc4ccccc4)Cc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B07 compound treatment 2080.0 1180.0 0.42 240.0 -530.0 -0.41 0.0075 0.0128 3119339 ChemDiv3_007421 CC(C)c1ccc(NC(=O)C(N(C)c2ccccc2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B08 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3027734 ChemDiv3_007422 O=C(CCS(=O)(=O)c1cccc2nsnc12)NC(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B09 compound treatment 280.0 -623.0 -0.22 200.0 -570.0 -0.44 -0.4658 -0.9498 3119340 ChemDiv3_007423 CC(C)c1ccc(NC(=O)C(N(C)C(=O)Cc2cccs2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B10 compound treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 3119341 ChemDiv3_007424 CC1CCCC(NC(=O)C2(O)N(C(=O)Nc3ccccc32)c4ccc(C)c(C)c4)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B11 compound treatment 320.0 -583.0 -0.21 480.0 -290.0 -0.22 -0.3037 -0.9993 3027737 ChemDiv3_007425 CCC(C)(N(C(=O)C)c1ccc(C)cc1)C(=O)NC2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B12 compound treatment 240.0 -663.0 -0.24 240.0 -530.0 -0.41 -0.4541 -0.9659 3027738 ChemDiv3_007426 CCOc1ccc(cc1)N(CC)S(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B13 compound treatment 240.0 -663.0 -0.24 320.0 -450.0 -0.35 -0.4106 -0.9823 3119342 ChemDiv3_007427 Cc1cccc(OCC(=O)Nc2ccc3nc(cc(C)c3c2)N4CCCCC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B14 compound treatment 320.0 -583.0 -0.21 240.0 -530.0 -0.41 -0.434 -0.9506 3026787 ChemDiv3_007428 CCC(C)NC(=O)C1C(N(C)C(=O)c2cc(OC)c(OC)cc12)c3ccc(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B15 compound treatment 400.0 -503.0 -0.18 1000.0 230.0 0.18 -0.0014 -0.0054 3119476 ChemDiv3_007429 CCCN1CCN(CC1)C(=O)Cn2cnc3sc(C)c(c3c2=O)S(=O)(=O)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B16 compound treatment 320.0 -583.0 -0.21 440.0 -330.0 -0.25 -0.3254 -0.9948 1498334 ChemDiv3_007430 CCSc1nc2NC3=C(C(c4ccccc4)c2c(=O)[nH]1)C(=O)CCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B17 compound treatment 680.0 -223.0 -0.08 400.0 -370.0 -0.28 -0.2568 -0.8705 3026790 ChemDiv3_007431 COc1ccc(cc1)C2C(C(=O)Nc3ccc(OC)c(OC)c3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B18 compound treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 3119477 ChemDiv3_007432 CCN(Cc1ccccc1)C(=O)CSc2nc3nc(C)c(Cc4ccccc4Cl)c(C)n3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B19 compound treatment 400.0 -503.0 -0.18 240.0 -530.0 -0.41 -0.4139 -0.9313 3026791 ChemDiv3_007433 COc1ccc(cc1)C2C(C(=O)Nc3cc(C)c(Cl)cc3OC)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B20 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3119478 ChemDiv3_007434 COc1ccc(cc1)N2C(C(CCC2=O)C(=O)N3CCCCC3)c4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B21 compound treatment 600.0 -303.0 -0.11 240.0 -530.0 -0.41 -0.3638 -0.864 3119479 ChemDiv3_007435 CC1CCCCN1C(=O)NC2(Oc3ccccc3O2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B22 compound treatment 480.0 -423.0 -0.15 280.0 -490.0 -0.38 -0.3722 -0.9185 3026794 ChemDiv3_007436 CCc1ccc(NC(=O)c2cnc(Nc3ccc(OC)cc3)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B23 mock treatment 520.0 -383.0 -0.14 240.0 -530.0 -0.41 -0.3838 -0.8944 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 B24 mock treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C01 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 1729621 ChemDiv3_007437 CC(Sc1cn(CCNC(=O)c2cccs2)c3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C02 compound treatment 480.0 -423.0 -0.15 360.0 -410.0 -0.32 -0.3287 -0.9423 3119480 ChemDiv3_007438 O=C(NCc1ccccc1)c2ccc3c(=O)n4CCCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C03 compound treatment 1560.0 658.0 0.23 400.0 -370.0 -0.28 -0.0361 -0.0982 3026797 ChemDiv3_007439 COc1ccc(cc1)N(C)C(=O)c2cnc(N3CCN(CC3)c4ncccn4)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C04 compound treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 3119481 ChemDiv3_007440 Cn1c2ccccc2c3cnn(CNC(=O)Nc4ccc(F)cc4)c(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C05 compound treatment 400.0 -503.0 -0.18 240.0 -530.0 -0.41 -0.4139 -0.9313 3119482 ChemDiv3_007441 CCc1ccc(NC(=O)C2CCC(=O)N(C2c3ccc(OC)cc3)c4ccc(OC)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C06 compound treatment 4520.0 3620.0 1.28 320.0 -450.0 -0.35 0.663 0.4988 3026800 ChemDiv3_007442 CC1CC(C)(C)NC(=S)N1CC(=O)N(C)Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C07 compound treatment 480.0 -423.0 -0.15 280.0 -490.0 -0.38 -0.3722 -0.9185 3119483 ChemDiv3_007443 COc1ccc(CNC(=O)C2C(N(C)C(=O)c3ccccc23)c4cccs4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C08 compound treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 3026854 ChemDiv3_007444 Cc1cc(NC(=O)CCS(=O)(=O)c2nc(cc(n2)C(F)(F)F)c3ccc4OCOc4c3)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C09 compound treatment 280.0 -623.0 -0.22 160.0 -610.0 -0.47 -0.4875 -0.9411 3119484 ChemDiv3_007445 COc1ccc(cc1)N(C)C(=O)c2cn(CC(C)C)c(=O)c3cc(OC)c(OC)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C10 compound treatment 360.0 -543.0 -0.19 320.0 -450.0 -0.35 -0.3805 -0.9618 3026857 ChemDiv3_007446 Fc1ccc(Sc2cc(C(=O)NCCC3=CCCCC3)c4ccccc4n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C11 compound treatment 280.0 -623.0 -0.22 360.0 -410.0 -0.32 -0.3789 -0.9849 3119485 ChemDiv3_007447 CCN(C(=O)c1coc(=O)c2ccccc12)c3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C12 compound treatment 280.0 -623.0 -0.22 280.0 -490.0 -0.38 -0.4223 -0.9677 1182380 ChemDiv3_007448 CCOc1ccc(cc1)n2cc(c3ccccc3)c4c(SCC)ncnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C13 compound treatment 320.0 -583.0 -0.21 280.0 -490.0 -0.38 -0.4123 -0.9601 3026859 ChemDiv3_007449 CN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C14 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3119486 ChemDiv3_007450 COc1ccc(cc1)n2nc(C(=O)NCC(=O)NCc3ccccc3OC)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C15 compound treatment 240.0 -663.0 -0.24 360.0 -410.0 -0.32 -0.3889 -0.9896 3026861 ChemDiv3_007451 CCc1ccc(NC(=O)c2cc3c(=O)oc4ccccc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C16 compound treatment 320.0 -583.0 -0.21 480.0 -290.0 -0.22 -0.3037 -0.9993 1329624 ChemDiv3_007452 Fc1ccc2NC(=O)CN(C(c3ccccc3)c2c1)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C17 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3119487 ChemDiv3_007453 COc1ccc2cc(/C=N/Cc3ccc(C)cc3)c(nc2c1)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C18 compound treatment 320.0 -583.0 -0.21 240.0 -530.0 -0.41 -0.434 -0.9506 1251410 ChemDiv3_007454 COc1cccc(c1)c2nnc(NC(=O)c3ccc(cc3)S(=O)(=O)N(C)C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C19 compound treatment 320.0 -583.0 -0.21 240.0 -530.0 -0.41 -0.434 -0.9506 3119488 ChemDiv3_007455 Clc1cccc(Cn2cc(CC(=O)Nc3nc4ccccc4s3)c5ccccc25)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C20 compound treatment 1640.0 738.0 0.26 200.0 -570.0 -0.44 -0.1246 -0.2443 3026866 ChemDiv3_007456 CCN(Cc1ccccc1)S(=O)(=O)c2ccc(cc2)C(=O)Nc3nnc(COC)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C21 compound treatment 1840.0 938.0 0.33 440.0 -330.0 -0.25 0.0558 0.1335 3119489 ChemDiv3_007457 FC(F)(F)c1cccc(NC(=S)Nc2ccc3nc4CCCCCn4c(=O)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C22 compound treatment 360.0 -543.0 -0.19 240.0 -530.0 -0.41 -0.424 -0.9415 3026868 ChemDiv3_007458 CCN(C(=O)Cn1c(=O)oc2ccccc12)c3cccc(c3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C23 mock treatment 3080.0 2180.0 0.77 440.0 -330.0 -0.25 0.3669 0.4513 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 C24 mock treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D01 compound treatment 360.0 -543.0 -0.19 440.0 -330.0 -0.25 -0.3154 -0.9907 1212159 ChemDiv3_007459 COc1ccc(OC)c(c1)S(=O)(=O)N2CC(C)OC(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D02 compound treatment 1480.0 578.0 0.2 400.0 -370.0 -0.28 -0.0562 -0.1603 3119490 ChemDiv3_007460 CCCCn1/c(=N\C(=O)c2ccccc2)/c(cc3c(=O)n4ccccc4nc13)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D03 compound treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 1880067 ChemDiv3_007461 CC1CN(C(C)CN1S(=O)(=O)c2ccc(F)cc2)S(=O)(=O)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D04 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3026919 ChemDiv3_007462 CC(=O)Oc1c(Sc2c(F)c(F)c(F)c(F)c2F)c(C)nn1C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D05 compound treatment 4160.0 3260.0 1.16 320.0 -450.0 -0.35 0.5727 0.4748 3119491 ChemDiv3_007463 COc1cc(Cl)c(C)cc1NC(=S)N(Cc2ccco2)Cc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D06 compound treatment 440.0 -463.0 -0.16 280.0 -490.0 -0.38 -0.3822 -0.9307 3026921 ChemDiv3_007464 CCc1ccc(NC(=O)CCS(=O)(=O)c2cccc3nonc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D07 compound treatment 280.0 -623.0 -0.22 560.0 -210.0 -0.16 -0.2703 -0.9882 3119492 ChemDiv3_007465 CC(C)c1ccc(NC(=O)C(N2CCc3ccccc23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D08 compound treatment 320.0 -583.0 -0.21 200.0 -570.0 -0.44 -0.4557 -0.9413 3119493 ChemDiv3_007466 O=C(CCNS(=O)(=O)c1cccc2nsnc12)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D09 compound treatment 240.0 -663.0 -0.24 400.0 -370.0 -0.28 -0.3672 -0.9955 3026924 ChemDiv3_007467 CC(C)c1ccc(NC(=O)C(NC(=O)/C=C/c2ccc3OCOc3c2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D10 compound treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 3119494 ChemDiv3_007468 CC(C)NC(=O)C1(O)N(C(=O)Nc2ccccc21)c3ccc(Cl)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D11 compound treatment 920.0 17.5 0.01 360.0 -410.0 -0.32 -0.2184 -0.693 3119495 ChemDiv3_007469 CCC(C)(N(C)C(=O)c1ccccn1)C(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D12 compound treatment 320.0 -583.0 -0.21 240.0 -530.0 -0.41 -0.434 -0.9506 3026926 ChemDiv3_007470 CCN(c1ccc(F)cc1)S(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D13 compound treatment 1240.0 338.0 0.12 440.0 -330.0 -0.25 -0.0947 -0.3375 3119496 ChemDiv3_007471 Cc1cc(nc2ccc(NC(=O)CCC3CCCC3)cc12)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D14 compound treatment 680.0 -223.0 -0.08 360.0 -410.0 -0.32 -0.2786 -0.8578 3026928 ChemDiv3_007472 COC(=O)c1cn(NC(=O)c2cccc(OC)c2)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D15 compound treatment 240.0 -663.0 -0.24 360.0 -410.0 -0.32 -0.3889 -0.9896 3119634 ChemDiv3_007473 COCCN1C(C(C(=O)NCc2ccccc2OC)c3ccccc3C1=O)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D16 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3119635 ChemDiv3_007474 CCOC(=O)C1=C(C)NC2=C(C1c3ccccc3)C(=O)C(C(C)C2)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D17 compound treatment 360.0 -543.0 -0.19 200.0 -570.0 -0.44 -0.4457 -0.9319 3026931 ChemDiv3_007475 COc1ccc(cc1)C2C(C(=O)Nc3ccc(cc3)C(F)(F)F)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D18 compound treatment 720.0 -183.0 -0.06 240.0 -530.0 -0.41 -0.3337 -0.8094 3119636 ChemDiv3_007476 Cc1cccc(CN2C(=O)CSc3ccc(cc23)C(=O)NCc4c(F)cc(F)cc4F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D19 compound treatment 360.0 -543.0 -0.19 320.0 -450.0 -0.35 -0.3805 -0.9618 3119637 ChemDiv3_007477 COc1ccc(cc1)C2C(C(=O)NCCCN3CCC(C)CC3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D20 compound treatment 480.0 -423.0 -0.15 320.0 -450.0 -0.35 -0.3504 -0.93 3119638 ChemDiv3_007478 COc1ccc(cc1)N2C(C(CCC2=O)C(=O)N3CCN(CC3)c4ccccc4)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D21 compound treatment 2000.0 1100.0 0.39 320.0 -450.0 -0.35 0.0308 0.0592 3026981 ChemDiv3_007479 FC(F)(F)C1(NC(=O)N2CCCc3ccccc23)Oc4ccccc4O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D22 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3119639 ChemDiv3_007480 COc1ccc(CCC(=O)Nc2ccc3nc(cc(C)c3c2)N4CCC(C)CC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D23 mock treatment 440.0 -463.0 -0.16 240.0 -530.0 -0.41 -0.4039 -0.9202 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 D24 mock treatment 440.0 -463.0 -0.16 240.0 -530.0 -0.41 -0.4039 -0.9202 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E01 compound treatment 400.0 -503.0 -0.18 560.0 -210.0 -0.16 -0.2402 -0.9988 3026983 ChemDiv3_007481 COC(=O)COc1nsnc1N2CCOCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E02 compound treatment 1360.0 458.0 0.16 2000.0 1230.0 0.94 0.7823 0.8167 3119640 ChemDiv3_007482 COc1ccccc1Nc2c3CCCCc3nc4ccc(NC(=O)/C=C/c5cccs5)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E03 compound treatment 2520.0 1620.0 0.57 480.0 -290.0 -0.22 0.2481 0.4031 3026984 ChemDiv3_007483 CCN(C(=O)c1cnc(N2CCN(CC2)c3ncccn3)c4ccccc14)c5cccc(Cl)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E04 compound treatment 880.0 -22.5 -0.01 3480.0 2710.0 2.08 1.4653 0.7044 3119641 ChemDiv3_007484 Cc1cc2ccccc2c(=O)n1CC(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E05 compound treatment 2120.0 1220.0 0.43 1080.0 310.0 0.24 0.4735 0.9604 3026987 ChemDiv3_007485 COc1ccc(cc1)C2C(CCC(=O)N2c3ccc(OC)cc3)C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E06 compound treatment 320.0 -583.0 -0.21 680.0 -90.3 -0.07 -0.1951 -0.8953 3119642 ChemDiv3_007486 CC1CC(C)(C)NC(=S)N1CC(=O)Nc2ccccc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E07 compound treatment 760.0 -143.0 -0.05 3640.0 2870.0 2.2 1.5221 0.6907 3119643 ChemDiv3_007487 COc1ccccc1CNC(=O)Cn2cnc3ccc(cc3c2=O)S(=O)(=O)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E08 compound treatment 680.0 -223.0 -0.08 520.0 -250.0 -0.19 -0.1917 -0.9227 3026990 ChemDiv3_007488 COc1ccccc1c2cc(nc(n2)S(=O)(=O)CCCC(=O)N3CCCCC3C)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E09 compound treatment 600.0 -303.0 -0.11 1040.0 270.0 0.21 0.0705 0.3024 3119644 ChemDiv3_007489 COc1ccc(CNC(=O)c2cn(CC(C)C)c(=O)c3cc(OC)c(OC)cc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E10 compound treatment 800.0 -103.0 -0.04 440.0 -330.0 -0.25 -0.205 -0.8003 3119645 ChemDiv3_007490 CCC(C)N1C(C(=O)NC2CCCC(C)C2C)C3(OC4C=C3)C(C4C(=O)Nc5cccc(C)c5)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E11 compound treatment 800.0 -103.0 -0.04 1040.0 270.0 0.21 0.1207 0.5741 3026993 ChemDiv3_007491 CN(C(=O)c1coc(=O)c2ccccc12)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E12 compound treatment 480.0 -423.0 -0.15 440.0 -330.0 -0.25 -0.2853 -0.9685 3026995 ChemDiv3_007492 Cn1c(C(=O)O)c(CC(=O)Nc2cnc3ccccc3c2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E13 compound treatment 1360.0 458.0 0.16 640.0 -130.0 -0.1 0.044 0.2309 3028013 ChemDiv3_007493 COc1ccc(CNC(=O)c2cc3c(=O)oc4ccccc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E14 compound treatment 600.0 -303.0 -0.11 1120.0 350.0 0.27 0.1139 0.3941 3028014 ChemDiv3_007494 COc1ccc(cc1)n2nc(C(=O)NCC(=O)NC3CCCC(C)C3C)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E15 compound treatment 840.0 -62.5 -0.02 320.0 -450.0 -0.35 -0.2601 -0.7509 3028015 ChemDiv3_007495 CCc1ccc(CNC(=O)c2coc(=O)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E16 compound treatment 2120.0 1220.0 0.43 1120.0 350.0 0.27 0.4952 0.9738 1175664 ChemDiv3_007496 COc1ccc(cc1)n2nc3CS(=O)Cc3c2NC(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E17 compound treatment 3280.0 2380.0 0.84 440.0 -330.0 -0.25 0.4171 0.4736 3028016 ChemDiv3_007497 CCc1ccc(Nc2nc3cc(OC)ccc3cc2C#N)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E18 compound treatment 760.0 -143.0 -0.05 560.0 -210.0 -0.16 -0.1499 -0.8861 1274303 ChemDiv3_007498 COc1cccc(c1)c2nnc(NC(=O)c3ccc(cc3)S(=O)(=O)N4CCCCC4C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E19 compound treatment 440.0 -463.0 -0.16 480.0 -290.0 -0.22 -0.2736 -0.9886 3119646 ChemDiv3_007499 CCC1CCCCN1C(=O)Cc2cn(Cc3cccc(Cl)c3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E20 compound treatment 800.0 -103.0 -0.04 1320.0 550.0 0.42 0.2727 0.6438 3119647 ChemDiv3_007500 FC(F)(F)c1ccc(NC(=O)CCCN2C(=O)c3cccnc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E21 compound treatment 1880.0 978.0 0.35 1560.0 790.0 0.61 0.6739 0.9649 3028017 ChemDiv3_007501 Cc1cccc(CCNC(=S)Nc2ccc3nc4CCCCCn4c(=O)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E22 compound treatment 920.0 17.5 0.01 1240.0 470.0 0.36 0.2594 0.7192 3119648 ChemDiv3_007502 CC1CC(C)(C)NC(=S)N1CCC(=O)Nc2ccc3OCCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E23 mock treatment 840.0 -62.5 -0.02 560.0 -210.0 -0.16 -0.1299 -0.7967 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 E24 mock treatment 1440.0 538.0 0.19 1760.0 990.0 0.76 0.6721 0.858 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F01 compound treatment 1080.0 178.0 0.06 4120.0 3350.0 2.57 1.8629 0.7242 1624488 ChemDiv3_007503 COc1ccc(OC)c(c1)S(=O)(=O)N2CCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F02 compound treatment 440.0 -463.0 -0.16 2720.0 1950.0 1.5 0.9424 0.6258 3119649 ChemDiv3_007504 CCCCn1/c(=N\C(=O)C(C)Oc2ccccc2)/c(cc3c(=O)n4ccccc4nc13)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F03 compound treatment 880.0 -22.5 -0.01 1000.0 230.0 0.18 0.119 0.6744 3119650 ChemDiv3_007505 CCc1ccc(NC(=S)N(CCCN2CCCCC2)Cc3cccs3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F04 compound treatment 2240.0 1340.0 0.47 5080.0 4310.0 3.31 2.675 0.8003 3028018 ChemDiv3_007506 CC1CC(C)CN(C1)c2nc3n(C)c(=O)n(C)c(=O)c3n2CCSc4nnc(C)s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F05 compound treatment 1320.0 418.0 0.15 640.0 -130.0 -0.1 0.034 0.1901 3119651 ChemDiv3_007507 CSc1cccc(NC(=S)N(CCN2CCCCC2)Cc3ccco3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F06 compound treatment 520.0 -383.0 -0.14 1040.0 270.0 0.21 0.0504 0.2038 3028019 ChemDiv3_007508 CC1CCCCN1C(=O)CCS(=O)(=O)c2cccc3nonc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F07 compound treatment 5080.0 4180.0 1.48 880.0 110.0 0.08 1.1074 0.7461 3119652 ChemDiv3_007509 COc1ccc(cc1)C(NC(=O)Cc2cc3ccccc3[nH]2)C(=O)Nc4ccc5OCCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F08 compound treatment 1600.0 698.0 0.25 1760.0 990.0 0.76 0.7122 0.8913 3028020 ChemDiv3_007510 CCc1ccc(NC(=O)CCNS(=O)(=O)c2cccc3nsnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F09 compound treatment 1080.0 178.0 0.06 3120.0 2350.0 1.8 1.3201 0.7313 3119653 ChemDiv3_007511 COc1ccc(cc1)C(N(Cc2ccco2)C(=O)c3cnccn3)C(=O)Nc4ccc(cc4)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F10 compound treatment 640.0 -263.0 -0.09 1560.0 790.0 0.61 0.3628 0.5916 1174354 ChemDiv3_007512 CNC(=S)N1CCc2cc(OC)c(OC)cc2C1COc3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F11 compound treatment 480.0 -423.0 -0.15 1640.0 870.0 0.67 0.3661 0.5351 3028021 ChemDiv3_007513 CCC(C)(N(C)C(=O)Cc1cccs1)C(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F12 compound treatment 640.0 -263.0 -0.09 7480.0 6710.0 5.15 3.5766 0.6942 1379326 ChemDiv3_007514 O=C(CN1C(=O)c2ccccc2S1(=O)=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F13 compound treatment 2640.0 1740.0 0.62 1040.0 270.0 0.21 0.5822 0.8955 3119654 ChemDiv3_007515 COc1ccc(/C=C/C(=O)Nc2ccc3nc(cc(C)c3c2)N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F14 compound treatment 600.0 -303.0 -0.11 640.0 -130.0 -0.1 -0.1466 -0.9994 3028022 ChemDiv3_007516 COC(=O)c1cn(NC(=O)C(C2CCCC2)c3ccccc3)c(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F15 compound treatment 600.0 -303.0 -0.11 1920.0 1150.0 0.88 0.5482 0.6166 3119655 ChemDiv3_007517 CCN1CCCC1CNC(=O)C2C(N(CCOC)C(=O)c3ccccc23)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F16 compound treatment 1400.0 498.0 0.18 840.0 69.7 0.05 0.1626 0.8818 1872278 ChemDiv3_007518 CC1CCN(CC1)/C(=C/c2nsc(Nc3ccc(F)c(Cl)c3)n2)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F17 compound treatment 1080.0 178.0 0.06 6320.0 5550.0 4.26 3.0572 0.7175 3119656 ChemDiv3_007519 COc1ccc(cc1)C2C(C(=O)NC3CCCC(C)C3C)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F18 compound treatment 760.0 -143.0 -0.05 1840.0 1070.0 0.82 0.5449 0.6623 3119795 ChemDiv3_007520 COc1ccccc1CNC(=O)c2ccc3SCC(=O)N(Cc4ccc(F)cc4Cl)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F19 compound treatment 680.0 -223.0 -0.08 1240.0 470.0 0.36 0.1992 0.5395 3028024 ChemDiv3_007521 CCCCN(C)C(=O)C1C(N(Cc2ccc(F)cc2)C(=O)c3ccccc13)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F20 compound treatment 840.0 -62.5 -0.02 3360.0 2590.0 1.99 1.3902 0.6992 3119796 ChemDiv3_007522 COc1ccc(cc1)N2C(C(CCC2=O)C(=O)NCC3CCCO3)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F21 compound treatment 3360.0 2460.0 0.87 680.0 -90.3 -0.07 0.5674 0.6488 3028025 ChemDiv3_007523 CC(C)CNC(=O)NC1(Oc2ccc(Cl)cc2O1)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F22 compound treatment 2080.0 1180.0 0.42 3200.0 2430.0 1.87 1.6143 0.8445 3119797 ChemDiv3_007524 CC1CCN(CC1)c2cc(C)c3cc(NC(=O)c4ccc5OCOc5c4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F23 mock treatment 1680.0 778.0 0.28 1240.0 470.0 0.36 0.45 0.9912 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 F24 mock treatment 720.0 -183.0 -0.06 6240.0 5470.0 4.2 2.9235 0.6961 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G01 compound treatment 4640.0 3740.0 1.33 520.0 -250.0 -0.19 0.8016 0.5984 3119798 ChemDiv3_007525 CCOC(=O)C1CCN(CC1)C(=O)c2n[nH]c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G02 compound treatment 1560.0 658.0 0.23 560.0 -210.0 -0.16 0.0508 0.1789 3028026 ChemDiv3_007526 COc1ccccc1Nc2c3CCCCc3nc4ccc(NC(=O)CCN5CCOCC5)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G03 compound treatment 560.0 -343.0 -0.12 560.0 -210.0 -0.16 -0.2001 -0.9902 3119799 ChemDiv3_007527 COc1ccc(cc1)C2C(C(=O)NC3CCCCC3)c4ccccc4C(=O)N2c5ccc(OC)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G04 compound treatment 520.0 -383.0 -0.14 760.0 -10.3 -0.01 -0.1016 -0.7471 3119800 ChemDiv3_007528 CC(C)c1ccc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G05 compound treatment 360.0 -543.0 -0.19 560.0 -210.0 -0.16 -0.2503 -0.9962 3028027 ChemDiv3_007529 COc1ccc(cc1)C2C(CCC(=O)N2c3ccc(OC)cc3)C(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G06 compound treatment 280.0 -623.0 -0.22 440.0 -330.0 -0.25 -0.3355 -0.9976 3119801 ChemDiv3_007530 CC1CC(C)(C)NC(=S)N1CC(=O)N2CCC(Cc3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G07 compound treatment 480.0 -423.0 -0.15 640.0 -130.0 -0.1 -0.1767 -0.9807 3119802 ChemDiv3_007531 CCCCN(CC)C(=O)Cn1cnc2ccc(cc2c1=O)S(=O)(=O)N3CCC(C)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G08 compound treatment 520.0 -383.0 -0.14 1120.0 350.0 0.27 0.0939 0.3121 3028028 ChemDiv3_007532 COC(=O)CCS(=O)(=O)c1nc(cc(n1)C(F)(F)F)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G09 compound treatment 1760.0 858.0 0.3 640.0 -130.0 -0.1 0.1444 0.4508 3119803 ChemDiv3_007533 COc1ccc(CNC(=O)c2cnc(Nc3ccccc3OC)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G10 compound treatment 3000.0 2100.0 0.74 440.0 -330.0 -0.25 0.3468 0.4412 3119804 ChemDiv3_007534 CCC(C)N1C(C(=O)NC2CCCCC2)C3(OC4C=C3)C(C4C(=O)Nc5cccc(Cl)c5)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G11 compound treatment 880.0 -22.5 -0.01 520.0 -250.0 -0.19 -0.1415 -0.7358 3028029 ChemDiv3_007535 CN(C(=O)c1coc(=O)c2ccccc12)c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G12 compound treatment 320.0 -583.0 -0.21 800.0 29.7 0.02 -0.13 -0.6254 3028030 ChemDiv3_007536 Cn1c(C(=O)O)c(CC(=O)N2CCCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G13 compound treatment 1400.0 498.0 0.18 720.0 -50.3 -0.04 0.0975 0.5395 3119805 ChemDiv3_007537 FC(F)(F)c1cccc(c1)N2CCN(CC2)C(=O)c3cc4c(=O)oc5ccccc5c4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G14 compound treatment 1320.0 418.0 0.15 960.0 190.0 0.15 0.2077 1.0 1158320 ChemDiv3_007538 Cc1ccc2NC(=O)CN(C(c3ccc(F)cc3)c2c1)C(=O)COc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G15 compound treatment 360.0 -543.0 -0.19 600.0 -170.0 -0.13 -0.2285 -0.9823 3119806 ChemDiv3_007539 Cc1ccc(CNC(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G16 compound treatment 640.0 -263.0 -0.09 400.0 -370.0 -0.28 -0.2669 -0.8921 1232646 ChemDiv3_007540 CCC(=O)Nc1c2CS(=O)Cc2nn1c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G17 compound treatment 680.0 -223.0 -0.08 440.0 -330.0 -0.25 -0.2351 -0.8853 3028031 ChemDiv3_007541 CC(C)NC(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G18 compound treatment 600.0 -303.0 -0.11 720.0 -50.3 -0.04 -0.1032 -0.9048 1173970 ChemDiv3_007542 COc1ccc(c2nnc(NC(=O)c3ccc(cc3)S(=O)(=O)N4CCC(C)CC4)o2)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G19 compound treatment 640.0 -263.0 -0.09 1120.0 350.0 0.27 0.124 0.4363 3028032 ChemDiv3_007543 COC(=O)c1cc2c(Cl)nc3ccc(C)cc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G20 compound treatment 560.0 -343.0 -0.12 7800.0 7030.0 5.4 3.7302 0.691 3119807 ChemDiv3_007544 COc1ccc(NC(=O)CN2C(=O)C3C4CC(C=C4)C3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G21 compound treatment 360.0 -543.0 -0.19 7560.0 6790.0 5.21 3.5498 0.6805 3028033 ChemDiv3_007545 O=c1n2CCCCCc2nc3ccc(NC(=S)NC4CCCCCC4)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G22 compound treatment 2240.0 1340.0 0.47 1040.0 270.0 0.21 0.4819 0.9309 3119808 ChemDiv3_007546 CC1Cc2ccccc2N1C(=O)CCN3C(C)CC(C)(C)NC3=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G23 mock treatment 1480.0 578.0 0.2 2080.0 1310.0 1.01 0.8558 0.834 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 G24 mock treatment 400.0 -503.0 -0.18 840.0 69.7 0.05 -0.0882 -0.474 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H01 compound treatment 2720.0 1820.0 0.64 640.0 -130.0 -0.1 0.3852 0.5903 3028034 ChemDiv3_007547 COc1ccc(OC)c(c1)S(=O)(=O)N2CCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H02 compound treatment 440.0 -463.0 -0.16 3240.0 2470.0 1.9 1.2247 0.6435 3119809 ChemDiv3_007548 CCOC(=O)c/1cc2c(=O)n3ccccc3nc2n(C4CCCCC4)\c1=N/C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H03 compound treatment 640.0 -263.0 -0.09 640.0 -130.0 -0.1 -0.1366 -0.9994 3119810 ChemDiv3_007549 CCc1ccc(NC(=S)N(CCCN2CCCC2)Cc3ccco3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H04 compound treatment 720.0 -183.0 -0.06 360.0 -410.0 -0.32 -0.2685 -0.835 3028035 ChemDiv3_007550 CN(Cc1ccccc1)c2nc3n(C)c(=O)n(C)c(=O)c3n2CCSc4nc5ccccc5o4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H05 compound treatment 600.0 -303.0 -0.11 1960.0 1190.0 0.91 0.5699 0.6198 3119811 ChemDiv3_007551 Clc1ccccc1NC(=S)N(CCN2CCCCCC2)Cc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H06 compound treatment 1760.0 858.0 0.3 400.0 -370.0 -0.28 0.0141 0.0338 3028036 ChemDiv3_007552 COc1ccccc1CNC(=O)CCS(=O)(=O)c2cccc3nonc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H07 compound treatment 520.0 -383.0 -0.14 440.0 -330.0 -0.25 -0.2753 -0.9571 3119812 ChemDiv3_007553 CN(C(C(=O)Nc1ccc2OCOc2c1)c3ccccc3)C(=O)/C=C\c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H08 compound treatment 1200.0 298.0 0.11 280.0 -490.0 -0.38 -0.1916 -0.49 3119813 ChemDiv3_007554 O=C(CCNS(=O)(=O)c1cccc2nsnc12)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H09 compound treatment 320.0 -583.0 -0.21 960.0 190.0 0.15 -0.0431 -0.1707 3028037 ChemDiv3_007555 CC(C)c1ccc(NC(=O)C(N2CC(=O)Nc3ccccc23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H10 compound treatment 640.0 -263.0 -0.09 440.0 -330.0 -0.25 -0.2452 -0.9075 1434209 ChemDiv3_007556 COc1cc2CCN(C(COc3ccc(F)cc3)c2cc1OC)C(=S)Nc4cccc(C)c4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H11 compound treatment 400.0 -503.0 -0.18 920.0 150.0 0.11 -0.0448 -0.2112 3119814 ChemDiv3_007557 CCC(C)(N(C(=O)c1ccccn1)c2ccccc2)C(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H12 compound treatment 1160.0 258.0 0.09 8160.0 7390.0 5.67 4.0761 0.7184 3028038 ChemDiv3_007558 COc1ccc(CN(C(=O)CN2C(=O)c3ccccc3S2(=O)=O)c4ccccc4O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H13 compound treatment 2560.0 1660.0 0.59 560.0 -210.0 -0.16 0.3016 0.4946 3119815 ChemDiv3_007559 CCN1CCN(CC1)c2cc(C)c3cc(NC(=O)c4ccncc4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H14 compound treatment 2920.0 2020.0 0.72 520.0 -250.0 -0.19 0.3702 0.4995 3028039 ChemDiv3_007560 COC(=O)c1cn(NC(=O)Cc2ccccc2OC)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H15 compound treatment 5560.0 4660.0 1.65 560.0 -210.0 -0.16 1.0541 0.635 3119816 ChemDiv3_007561 COCCN1C(C(C(=O)N2CCN(CC2)c3ccccn3)c4ccccc4C1=O)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H16 compound treatment 3320.0 2420.0 0.86 560.0 -210.0 -0.16 0.4922 0.5641 3119817 ChemDiv3_007562 C/C(=C\c1nsc(Nc2ccc(Cl)cc2)n1)/NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H17 compound treatment 560.0 -343.0 -0.12 680.0 -90.3 -0.07 -0.1349 -0.9646 3028040 ChemDiv3_007563 COc1ccc(cc1)C2C(C(=O)NCC3CCCO3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H18 compound treatment 680.0 -223.0 -0.08 7200.0 6430.0 4.94 3.4346 0.6957 3119953 ChemDiv3_007564 Cc1ccc(CNC(=O)C2C3OC4(CN(Cc5cccs5)C(=O)C24)C=C3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H19 compound treatment 640.0 -263.0 -0.09 720.0 -50.3 -0.04 -0.0932 -0.9241 3119954 ChemDiv3_007565 COc1ccc(cc1)C2C(C(=O)N3CCCCC3)c4ccccc4C(=O)N2Cc5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H20 compound treatment 1200.0 298.0 0.11 4480.0 3710.0 2.85 2.0885 0.7328 3028095 ChemDiv3_007566 COc1cc(OC)cc(c1)C(=O)Nn2cc(C(=O)N3CCN(C)CC3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H21 compound treatment 360.0 -543.0 -0.19 640.0 -130.0 -0.1 -0.2068 -0.9536 3028096 ChemDiv3_007567 FC(F)(F)C1(NC(=O)N2CCCCC2)Oc3ccc(Cl)cc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H22 compound treatment 560.0 -343.0 -0.12 1360.0 590.0 0.45 0.2342 0.4996 3028097 ChemDiv3_007568 FC(F)(F)c1cc(nc(n1)N2CCCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H23 mock treatment 680.0 -223.0 -0.08 520.0 -250.0 -0.19 -0.1917 -0.9227 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 H24 mock treatment 3400.0 2500.0 0.89 2400.0 1630.0 1.25 1.5112 0.9857 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I01 compound treatment 280.0 -623.0 -0.22 360.0 -410.0 -0.32 -0.3789 -0.9849 3028098 ChemDiv3_007569 COc1ccc(CCNC(=O)c2n[nH]c(=O)c3ccccc23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I02 compound treatment 240.0 -663.0 -0.24 440.0 -330.0 -0.25 -0.3455 -0.9993 3028099 ChemDiv3_007570 CCOC(=O)c1n[nH]c-2c1COc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I03 compound treatment 200.0 -703.0 -0.25 320.0 -450.0 -0.35 -0.4207 -0.9871 3028100 ChemDiv3_007571 COc1ccc(cc1)C2C(C(=O)Nc3cccc(C)n3)c4ccccc4C(=O)N2c5ccc(OC)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I04 compound treatment 280.0 -623.0 -0.22 280.0 -490.0 -0.38 -0.4223 -0.9677 3119955 ChemDiv3_007572 CC1CCN(CCCNC(=O)Cn2c(C)cc3ccccc3c2=O)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I05 compound treatment 280.0 -623.0 -0.22 440.0 -330.0 -0.25 -0.3355 -0.9976 3028101 ChemDiv3_007573 COc1ccc(cc1)C2C(CCC(=O)N2c3ccc(OC)cc3)C(=O)N4CC(C)CC(C)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I06 compound treatment 320.0 -583.0 -0.21 280.0 -490.0 -0.38 -0.4123 -0.9601 3119956 ChemDiv3_007574 CCc1ccc(NC(=O)CCCN2C(C)CC(C)(C)NC2=S)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I07 compound treatment 4080.0 3180.0 1.13 360.0 -410.0 -0.32 0.5743 0.4907 3119957 ChemDiv3_007575 CCN(C(=O)c1cn(CC)c(=O)c2cc(OC)c(OC)cc12)c3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I08 compound treatment 440.0 -463.0 -0.16 320.0 -450.0 -0.35 -0.3605 -0.942 3028102 ChemDiv3_007576 CCOC(=O)N1CCC(CC1)NC(=O)c2cc(Sc3ccc(Cl)cc3)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I09 compound treatment 440.0 -463.0 -0.16 1080.0 310.0 0.24 0.0521 0.1803 3119958 ChemDiv3_007577 O=C(NC1CCCCC1)C2C3N(CCc4ccccc34)C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I10 compound treatment 280.0 -623.0 -0.22 240.0 -530.0 -0.41 -0.444 -0.9587 3119959 ChemDiv3_007578 CCCCN1C(C(=O)NC2CCCCC2)C3(OC4C=C3)C(C4C(=O)Nc5ccc(cc5)C(C)C)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I11 compound treatment 440.0 -463.0 -0.16 400.0 -370.0 -0.28 -0.317 -0.9659 3028103 ChemDiv3_007579 COc1ccc(cc1)N(C)C(=O)c2cc3c(=O)oc4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I12 compound treatment 560.0 -343.0 -0.12 720.0 -50.3 -0.04 -0.1132 -0.8881 3119960 ChemDiv3_007580 Cn1c(C(=O)O)c(CC(=O)NCc2cccnc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I13 compound treatment 440.0 -463.0 -0.16 360.0 -410.0 -0.32 -0.3388 -0.9538 3028104 ChemDiv3_007581 CC1CC(C)CN(CCCNC(=O)c2cnc(Nc3ccc(C)c(Cl)c3)c4ccccc24)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I14 compound treatment 480.0 -423.0 -0.15 240.0 -530.0 -0.41 -0.3939 -0.9079 1310972 ChemDiv3_007582 Fc1ccc(CC(=O)N2CC(=O)Nc3ccc(F)cc3C2c4ccc(F)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I15 compound treatment 360.0 -543.0 -0.19 840.0 69.7 0.05 -0.0983 -0.4919 3119961 ChemDiv3_007583 Cc1ccc(CNC(=O)CCC(=O)Nc2ccc3nc(cc(C)c3c2)N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I16 compound treatment 360.0 -543.0 -0.19 600.0 -170.0 -0.13 -0.2285 -0.9823 1525579 ChemDiv3_007584 CCCCC(=O)Nc1c2CS(=O)Cc2nn1C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I17 compound treatment 280.0 -623.0 -0.22 3680.0 2910.0 2.23 1.4234 0.6341 3119962 ChemDiv3_007585 CCOC(=O)CSc1cc(=O)n(CC)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I18 compound treatment 360.0 -543.0 -0.19 320.0 -450.0 -0.35 -0.3805 -0.9618 1682890 ChemDiv3_007586 CC(C)CN(CC(C)C)S(=O)(=O)c1ccc(cc1)C(=O)Nc2nnc(o2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I19 compound treatment 3760.0 2860.0 1.01 360.0 -410.0 -0.32 0.494 0.4654 3119963 ChemDiv3_007587 COC(=O)c1cc2COc3ccccc3-c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I20 compound treatment 4120.0 3220.0 1.14 440.0 -330.0 -0.25 0.6278 0.5369 3119964 ChemDiv3_007588 Fc1cccc(NC(=O)CN2C(=O)C3C4CC(C=C4)C3C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I21 compound treatment 360.0 -543.0 -0.19 360.0 -410.0 -0.32 -0.3588 -0.9721 3028105 ChemDiv3_007589 O=c1n2CCCCCc2nc3ccc(NC(=S)NCc4ccccn4)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I22 compound treatment 560.0 -343.0 -0.12 320.0 -450.0 -0.35 -0.3304 -0.9016 3119965 ChemDiv3_007590 CC1CC(C)(C)NC(=S)N1CC(=O)NCc2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I23 mock treatment 600.0 -303.0 -0.11 360.0 -410.0 -0.32 -0.2986 -0.8973 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 I24 mock treatment 280.0 -623.0 -0.22 240.0 -530.0 -0.41 -0.444 -0.9587 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J01 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3028106 ChemDiv3_007591 O=S(=O)(N1CCCCCC1)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J02 compound treatment 320.0 -583.0 -0.21 280.0 -490.0 -0.38 -0.4123 -0.9601 3119966 ChemDiv3_007592 CCOC(=O)c/1cc2c(=O)n3ccccc3nc2n(Cc4ccco4)\c1=N/C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J03 compound treatment 400.0 -503.0 -0.18 360.0 -410.0 -0.32 -0.3488 -0.9637 3119967 ChemDiv3_007593 CCc1ccc(NC(=S)N(Cc2cccs2)C3CCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J04 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3028107 ChemDiv3_007594 Cc1nnc(NN2CCOCC2)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J05 compound treatment 360.0 -543.0 -0.19 160.0 -610.0 -0.47 -0.4674 -0.9227 3119968 ChemDiv3_007595 CCOC(=O)N1CCN(CC1)c2cc(NCCC(=O)O)c3C(=O)c4ccccc4-c5onc2c53 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J06 compound treatment 440.0 -463.0 -0.16 280.0 -490.0 -0.38 -0.3822 -0.9307 3028108 ChemDiv3_007596 O=C(CCS(=O)(=O)c1cccc2nonc12)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J07 compound treatment 720.0 -183.0 -0.06 360.0 -410.0 -0.32 -0.2685 -0.835 3119969 ChemDiv3_007597 COc1ccc(NC(=O)C(N(C)C(=O)Cc2c[nH]c3ccccc23)c4ccc(OC)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J08 compound treatment 2040.0 1140.0 0.4 240.0 -530.0 -0.41 -0.0026 -0.0045 3028109 ChemDiv3_007598 CC1CCN(CC1)C(=O)CCNS(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J09 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3119970 ChemDiv3_007599 CN(C(C(=O)NC1CCCC1)c2ccc(Cl)cc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J10 compound treatment 280.0 -623.0 -0.22 280.0 -490.0 -0.38 -0.4223 -0.9677 1345440 ChemDiv3_007600 CC(C)(C)NS(=O)(=O)c1cccc2nsnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J11 compound treatment 400.0 -503.0 -0.18 560.0 -210.0 -0.16 -0.2402 -0.9988 3119971 ChemDiv3_007601 O=C(NC1CCCC1)C2(CCCCC2)N(Cc3cccs3)C(=O)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J12 compound treatment 360.0 -543.0 -0.19 440.0 -330.0 -0.25 -0.3154 -0.9907 3028110 ChemDiv3_007602 Cc1cc2ccccc2c(=O)n1CC(=O)NCC(=O)Nc3nc4ccccc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J13 compound treatment 480.0 -423.0 -0.15 320.0 -450.0 -0.35 -0.3504 -0.93 3119972 ChemDiv3_007603 CCN1CCN(CC1)c2cc(C)c3cc(NC(=O)CC4CCCCC4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J14 compound treatment 200.0 -703.0 -0.25 280.0 -490.0 -0.38 -0.4424 -0.9799 3028111 ChemDiv3_007604 COC(=O)c1cn(NC(=O)CCC2CCCC2)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J15 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3119973 ChemDiv3_007605 COCCN1C(C(C(=O)NCC2COc3ccccc3O2)c4ccccc4C1=O)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J16 compound treatment 360.0 -543.0 -0.19 280.0 -490.0 -0.38 -0.4023 -0.9515 3028112 ChemDiv3_007606 CCN/C(=C/c1nsc(Nc2ccc(Cl)c(Cl)c2)n1)/C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J17 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3119974 ChemDiv3_007607 COc1ccc(cc1)C2C(C(=O)NCCc3ccc(OC)c(OC)c3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J18 compound treatment 320.0 -583.0 -0.21 640.0 -130.0 -0.1 -0.2169 -0.9446 3119975 ChemDiv3_007608 O=C(NC1CCCCC1)C2C3OC4(CN(Cc5cccs5)C(=O)C24)C=C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J19 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3028113 ChemDiv3_007609 CC(C)c1ccc(NC(=O)NC2(Oc3ccccc3O2)C(F)(F)F)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J20 compound treatment 360.0 -543.0 -0.19 320.0 -450.0 -0.35 -0.3805 -0.9618 3119976 ChemDiv3_007610 CCN(CC)c1cc(C)c2cc(NC(=O)c3ccc(Br)c(OC)c3)ccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J21 compound treatment 320.0 -583.0 -0.21 920.0 150.0 0.11 -0.0649 -0.2743 3028114 ChemDiv3_007611 CCOC(=O)c/1cc2c(=O)n3ccccc3nc2n(C)\c1=N/C(=O)\C=C\c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J22 compound treatment 200.0 -703.0 -0.25 200.0 -570.0 -0.44 -0.4858 -0.9643 3119977 ChemDiv3_007612 FC(F)(F)c1cc(nc(n1)N2CCN(CC2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J23 mock treatment 240.0 -663.0 -0.24 840.0 69.7 0.05 -0.1284 -0.5325 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 J24 mock treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K01 compound treatment 920.0 17.5 0.01 1080.0 310.0 0.24 0.1725 0.7253 3120116 ChemDiv3_007613 O=C(NCCC1=CCCCC1)c2n[nH]c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K02 compound treatment 1280.0 378.0 0.13 600.0 -170.0 -0.13 0.0022 0.0119 3028115 ChemDiv3_007614 CCOC(=O)c1sc2nc3CCCCn3c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K03 compound treatment 640.0 -263.0 -0.09 640.0 -130.0 -0.1 -0.1366 -0.9994 3120117 ChemDiv3_007615 COc1ccc(cc1)C2C(C(=O)N3CC(C)CC(C)C3)c4ccccc4C(=O)N2c5ccc(OC)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K04 compound treatment 960.0 57.5 0.02 520.0 -250.0 -0.19 -0.1215 -0.6285 3028116 ChemDiv3_007616 CC1CC(C)(C)NC(=S)N1CCC(=O)Nc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K05 compound treatment 640.0 -263.0 -0.09 1840.0 1070.0 0.82 0.5148 0.6229 3120118 ChemDiv3_007617 COc1ccc(cc1)C2C(CCC(=O)N2c3ccc(OC)cc3)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K06 compound treatment 4240.0 3340.0 1.18 920.0 150.0 0.11 0.9184 0.7721 3028117 ChemDiv3_007618 CC1CC(C)(C)NC(=S)N1CCCC(=O)N2CCN(CC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K07 compound treatment 680.0 -223.0 -0.08 360.0 -410.0 -0.32 -0.2786 -0.8578 3120119 ChemDiv3_007619 CCn1cc(C(=O)NCCC(C)C)c2cc(OC)c(OC)cc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K08 compound treatment 840.0 -62.5 -0.02 720.0 -50.3 -0.04 -0.043 -0.9653 3120120 ChemDiv3_007620 Clc1ccc(Sc2cc(C(=O)N3CCC4(CC3)OCCO4)c5ccccc5n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K09 compound treatment 360.0 -543.0 -0.19 3840.0 3070.0 2.36 1.5303 0.6472 3028118 ChemDiv3_007621 COc1ccc(cc1O)c2c(C(=O)O)c3cc(OC)c(OC)cc3c(=O)n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K10 compound treatment 480.0 -423.0 -0.15 800.0 29.7 0.02 -0.0899 -0.5928 3120121 ChemDiv3_007622 CCOc1ccc(NC(=O)C2C3OC4(C=C3)C(N(C(C)C)C(=O)C24)C(=O)NC5CCCCC5C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K11 compound treatment 880.0 -22.5 -0.01 760.0 -10.3 -0.01 -0.0112 -1.0 3028119 ChemDiv3_007623 CN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K12 compound treatment 1080.0 178.0 0.06 3000.0 2230.0 1.71 1.2549 0.7326 3120122 ChemDiv3_007624 CC1CC(C)CN(CCCNC(=O)Cc2c(C(=O)O)n(C)c3ccccc23)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K13 compound treatment 1640.0 738.0 0.26 1120.0 350.0 0.27 0.3748 0.9999 3028120 ChemDiv3_007625 CCN1CCN(CC1)C(=O)Cc2c([nH]c3ccccc23)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K14 compound treatment 840.0 -62.5 -0.02 600.0 -170.0 -0.13 -0.1081 -0.8154 1389024 ChemDiv3_007626 CCCC(=O)N1CC(=O)Nc2ccc(C)cc2C1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K15 compound treatment 480.0 -423.0 -0.15 400.0 -370.0 -0.28 -0.307 -0.9553 3028121 ChemDiv3_007627 COc1ccc2cc(C#N)c(Cl)nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K16 compound treatment 760.0 -143.0 -0.05 2040.0 1270.0 0.97 0.6535 0.6695 1517473 ChemDiv3_007628 CC(C)(C)C(=O)Nc1c2CS(=O)Cc2nn1c3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K17 compound treatment 920.0 17.5 0.01 1880.0 1110.0 0.85 0.6068 0.7122 3028122 ChemDiv3_007629 Clc1cccc(NC(=O)c2ccc3c(Cl)c4CCCCc4nc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K18 compound treatment 1160.0 258.0 0.09 2800.0 2030.0 1.56 1.1664 0.7473 1180917 ChemDiv3_007630 CCCCN(CC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2nnc(o2)c3ccc(Cl)s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K19 compound treatment 1040.0 138.0 0.05 840.0 69.7 0.05 0.0723 0.9989 3028123 ChemDiv3_007631 Cc1ccc2cc3c(NCc4ccc(F)cc4Cl)n[nH]c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K20 compound treatment 840.0 -62.5 -0.02 720.0 -50.3 -0.04 -0.043 -0.9653 3120123 ChemDiv3_007632 O=C(CN1C(=O)C2C3CC(C=C3)C2C1=O)NC4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K21 compound treatment 920.0 17.5 0.01 720.0 -50.3 -0.04 -0.0229 -0.586 3120124 ChemDiv3_007633 O=c1n2CCCCCc2nc3ccc(NC(=S)N4CCCC4)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K22 compound treatment 560.0 -343.0 -0.12 600.0 -170.0 -0.13 -0.1784 -0.9993 3028124 ChemDiv3_007634 Fc1ccc(cc1)S(=O)(=O)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K23 mock treatment 1480.0 578.0 0.2 840.0 69.7 0.05 0.1827 0.8628 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 K24 mock treatment 1560.0 658.0 0.23 880.0 110.0 0.08 0.2245 0.9052 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L01 compound treatment 520.0 -383.0 -0.14 880.0 110.0 0.08 -0.0364 -0.228 3028125 ChemDiv3_007635 Brc1ccc(s1)S(=O)(=O)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L02 compound treatment 760.0 -143.0 -0.05 1160.0 390.0 0.3 0.1758 0.5794 1281251 ChemDiv3_007636 CCCC(=O)Oc1c(Sc2ccccc2)c(C)nn1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L03 compound treatment 520.0 -383.0 -0.14 1320.0 550.0 0.42 0.2024 0.4567 3120125 ChemDiv3_007637 Cc1cccc(NC(=S)N(CCN2CCCCCC2)Cc3cccs3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L04 compound treatment 320.0 -583.0 -0.21 4720.0 3950.0 3.03 1.998 0.6574 1420486 ChemDiv3_007638 O=c1cnnc(Nc2ccccc2)[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L05 compound treatment 1040.0 138.0 0.05 960.0 190.0 0.15 0.1375 0.8951 3120126 ChemDiv3_007639 C=CCN(C(C(=O)Nc1ccc2OCCOc2c1)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L06 compound treatment 680.0 -223.0 -0.08 760.0 -10.3 -0.01 -0.0614 -0.7742 3028126 ChemDiv3_007640 Clc1ccc(CNC(=O)CCS(=O)(=O)c2cccc3nonc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L07 compound treatment 520.0 -383.0 -0.14 720.0 -50.3 -0.04 -0.1233 -0.8737 3028179 ChemDiv3_007641 COc1ccc(NC(=O)C(N(C)C(=O)c2ccc(=O)[nH]c2)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L08 compound treatment 480.0 -423.0 -0.15 480.0 -290.0 -0.22 -0.2636 -0.9814 3028180 ChemDiv3_007642 Cc1ccc(CNC(=O)C2(O)N(C(=O)Nc3ccccc32)c4ccc(C)c(C)c4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L09 compound treatment 320.0 -583.0 -0.21 600.0 -170.0 -0.13 -0.2386 -0.9756 3028181 ChemDiv3_007643 CCN(C(C(=O)NC1CCCC1)c2ccccc2)c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L10 compound treatment 480.0 -423.0 -0.15 800.0 29.7 0.02 -0.0899 -0.5928 3028182 ChemDiv3_007644 Cc1c(Cl)cccc1NS(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L11 compound treatment 4080.0 3180.0 1.13 1760.0 990.0 0.76 1.3343 0.9816 3028183 ChemDiv3_007645 CC(=O)NC1(CCCCC1)C(=O)NC2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L12 compound treatment 2680.0 1780.0 0.63 1560.0 790.0 0.61 0.8746 0.9998 3028184 ChemDiv3_007646 CN(C1CCCCC1)C(=O)CNC(=O)Cn2c(C)cc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L13 compound treatment 1840.0 938.0 0.33 600.0 -170.0 -0.13 0.1427 0.3993 3120127 ChemDiv3_007647 CCN1CCN(CC1)c2cc(C)c3cc(NC(=O)COc4ccc(Cl)cc4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L14 compound treatment 440.0 -463.0 -0.16 600.0 -170.0 -0.13 -0.2085 -0.9937 3028185 ChemDiv3_007648 COC(=O)c1cn(NC(=O)C2CCCCC2)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L15 compound treatment 1000.0 97.5 0.03 9400.0 8630.0 6.63 4.7092 0.7108 3120128 ChemDiv3_007649 COCCN1C(C(C(=O)Nc2ccc(cc2)C(C)C)c3ccccc3C1=O)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L16 compound treatment 480.0 -423.0 -0.15 680.0 -90.3 -0.07 -0.155 -0.9387 3028186 ChemDiv3_007650 COc1ccc(CN/C(=C/c2nsc(Nc3ccc(F)cc3)n2)/C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L17 compound treatment 1000.0 97.5 0.03 320.0 -450.0 -0.35 -0.22 -0.6332 3120129 ChemDiv3_007651 COc1ccc(cc1)C2C(C(=O)NCc3ccccn3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L18 compound treatment 680.0 -223.0 -0.08 360.0 -410.0 -0.32 -0.2786 -0.8578 3120130 ChemDiv3_007652 O=C(NCCCN1CCOCC1)C2C3OC4(CN(Cc5cccs5)C(=O)C24)C=C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L19 compound treatment 440.0 -463.0 -0.16 1240.0 470.0 0.36 0.139 0.3508 3028187 ChemDiv3_007653 FC(F)(F)C1(NC(=O)NCc2ccccc2)Oc3ccccc3O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L20 compound treatment 400.0 -503.0 -0.18 640.0 -130.0 -0.1 -0.1968 -0.9627 3120131 ChemDiv3_007654 CCN(CC)c1cc(C)c2cc(NC(=O)/C(=C\c3ccccc3)/C)ccc2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L21 compound treatment 840.0 -62.5 -0.02 3600.0 2830.0 2.17 1.5204 0.6999 3028188 ChemDiv3_007655 CCOC(=O)c/1cc2c(=O)n3ccccc3nc2n(C)\c1=N/C(=O)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L22 compound treatment 1000.0 97.5 0.03 1080.0 310.0 0.24 0.1926 0.8015 3120132 ChemDiv3_007656 CN(Cc1ccccc1)c2nc(cc(n2)C(F)(F)F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L23 mock treatment 880.0 -22.5 -0.01 1720.0 950.0 0.73 0.5099 0.6993 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 L24 mock treatment 1080.0 178.0 0.06 320.0 -450.0 -0.35 -0.1999 -0.569 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M01 compound treatment 2560.0 1660.0 0.59 2280.0 1510.0 1.16 1.2353 0.9505 3120133 ChemDiv3_007657 CCN1CCN(CCCNC(=O)c2n[nH]c(=O)c3ccccc23)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M02 compound treatment 1120.0 218.0 0.08 400.0 -370.0 -0.28 -0.1465 -0.4972 3028189 ChemDiv3_007658 Cc1cc(NC2CCCCC2)nc3ccc(N)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M03 compound treatment 640.0 -263.0 -0.09 1040.0 270.0 0.21 0.0806 0.3548 3120134 ChemDiv3_007659 COc1ccc(cc1)C2C(C(=O)NCc3cccnc3)c4ccccc4C(=O)N2c5ccc(OC)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M04 compound treatment 1160.0 258.0 0.09 640.0 -130.0 -0.1 -0.0062 -0.0454 3028190 ChemDiv3_007660 COc1ccc(CCNC(=O)CCN2C(C)CC(C)(C)NC2=S)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M05 compound treatment 1400.0 498.0 0.18 480.0 -290.0 -0.22 -0.0328 -0.1154 3120135 ChemDiv3_007661 COc1ccc(CCNC(=O)Cn2ccc3ccccc3c2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M06 compound treatment 520.0 -383.0 -0.14 680.0 -90.3 -0.07 -0.145 -0.9514 3120136 ChemDiv3_007662 CC1CC(C)(C)NC(=S)N1CCCC(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M07 compound treatment 2160.0 1260.0 0.45 800.0 29.7 0.02 0.3315 0.7423 3028191 ChemDiv3_007663 COc1ccc(CNC(=O)Cn2ccc3ccccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M08 compound treatment 400.0 -503.0 -0.18 1840.0 1070.0 0.82 0.4546 0.541 3120137 ChemDiv3_007664 Fc1ccc(Sc2cc(C(=O)NCc3ccccn3)c4ccccc4n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M09 compound treatment 760.0 -143.0 -0.05 960.0 190.0 0.15 0.0672 0.4361 3028192 ChemDiv3_007665 Cc1ccc(Nc2ncc(C(=O)NCCC3=CCCCC3)c4ccccc24)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M10 compound treatment 560.0 -343.0 -0.12 720.0 -50.3 -0.04 -0.1132 -0.8881 1477396 ChemDiv3_007666 CCSc1ncnc2n(cc(c3ccccc3)c12)c4cccc(F)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M11 compound treatment 560.0 -343.0 -0.12 1120.0 350.0 0.27 0.1039 0.3526 3117848 ChemDiv3_007667 CC(C)CCNC(=O)c1cc2c(=O)oc3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M12 compound treatment 560.0 -343.0 -0.12 2480.0 1710.0 1.31 0.8422 0.6389 3028193 ChemDiv3_007668 CC(C)c1ccc(cc1)N(C)C(=O)Cc2c(C(=O)O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M13 compound treatment 920.0 17.5 0.01 640.0 -130.0 -0.1 -0.0664 -0.662 3117849 ChemDiv3_007669 COc1ccccc1NC(=O)c2cnc(Nc3ccc(C)c(Cl)c3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M14 compound treatment 760.0 -143.0 -0.05 680.0 -90.3 -0.07 -0.0848 -0.9879 1453585 ChemDiv3_007670 Cc1ccc2NC(=O)CN(C(c3ccccc3)c2c1)C(=O)c4ccc(C)c(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M15 compound treatment 600.0 -303.0 -0.11 480.0 -290.0 -0.22 -0.2335 -0.9439 1354186 ChemDiv3_007671 COc1ccc2nc3sc(cc3cc2c1)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M16 compound treatment 760.0 -143.0 -0.05 480.0 -290.0 -0.22 -0.1933 -0.846 1356549 ChemDiv3_007672 Clc1cccc(c1)n2nc3CS(=O)Cc3c2NC(=O)c4cccc(Br)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M17 compound treatment 720.0 -183.0 -0.06 560.0 -210.0 -0.16 -0.16 -0.9195 3117850 ChemDiv3_007673 CCn1c(=O)cc(SCC(=O)NCCc2ccc(C)cc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M18 compound treatment 760.0 -143.0 -0.05 560.0 -210.0 -0.16 -0.1499 -0.8861 3117851 ChemDiv3_007674 CCc1nnc(NC(=O)c2ccc(cc2)S(=O)(=O)N(C)c3ccccc3)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M19 compound treatment 720.0 -183.0 -0.06 1880.0 1110.0 0.85 0.5566 0.6515 3028194 ChemDiv3_007675 COC(=O)CSc1cc(Cl)nc2ccc(C)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M20 compound treatment 600.0 -303.0 -0.11 2440.0 1670.0 1.28 0.8305 0.6457 3117852 ChemDiv3_007676 O=C(CN1C(=O)C2C3CC(C=C3)C2C1=O)NCCN4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M21 compound treatment 560.0 -343.0 -0.12 4000.0 3230.0 2.48 1.6673 0.6717 3028195 ChemDiv3_007677 O=c1n2CCCCCc2nc3ccc(NC(=S)NCC4CCCO4)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M22 compound treatment 600.0 -303.0 -0.11 800.0 29.7 0.02 -0.0598 -0.5448 1876488 ChemDiv3_007678 CC(C)Cc1ccc(cc1)S(=O)(=O)N2CC(C)CC(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M23 mock treatment 1920.0 1020.0 0.36 560.0 -210.0 -0.16 0.1411 0.3567 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 M24 mock treatment 840.0 -62.5 -0.02 2520.0 1750.0 1.34 0.9342 0.6953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N01 compound treatment 840.0 -62.5 -0.02 680.0 -90.3 -0.07 -0.0647 -0.8889 3028196 ChemDiv3_007679 O=S(=O)(N1CCc2ccccc12)c3ccc(cc3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N02 compound treatment 360.0 -543.0 -0.19 960.0 190.0 0.15 -0.0331 -0.1372 1535908 ChemDiv3_007680 Cc1nn(c(OC(=O)c2cccs2)c1Sc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N03 compound treatment 7000.0 6100.0 2.16 1480.0 710.0 0.54 1.9148 0.8584 3117853 ChemDiv3_007681 CCc1ccccc1NC(=S)N(CCN(C)C)Cc2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N04 compound treatment 1680.0 778.0 0.28 440.0 -330.0 -0.25 0.0157 0.0419 1505679 ChemDiv3_007682 Cc1ccc2n(CCC#N)c3CC[N+](C)(C)Cc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N05 compound treatment 440.0 -463.0 -0.16 320.0 -450.0 -0.35 -0.3605 -0.942 3117854 ChemDiv3_007683 CCN(C(C(=O)Nc1ccc2OCCOc2c1)c3ccccc3)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N06 compound treatment 520.0 -383.0 -0.14 720.0 -50.3 -0.04 -0.1233 -0.8737 3028197 ChemDiv3_007684 CN(C(=O)CCS(=O)(=O)c1cccc2nonc12)c3cc(C)ccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N07 compound treatment 640.0 -263.0 -0.09 1400.0 630.0 0.48 0.276 0.5606 3117855 ChemDiv3_007685 COc1ccc(NC(=O)C(NC(=O)c2ccc(=O)[nH]c2)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N08 compound treatment 760.0 -143.0 -0.05 840.0 69.7 0.05 0.0021 0.0283 3117856 ChemDiv3_007686 OC1(N(C(=O)Nc2ccccc21)c3c(F)cccc3F)C(=O)NCc4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N09 compound treatment 680.0 -223.0 -0.08 680.0 -90.3 -0.07 -0.1048 -0.9979 3028198 ChemDiv3_007687 CN(C(C(=O)NC1CCCCC1)c2ccc(C)cc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N10 compound treatment 640.0 -263.0 -0.09 320.0 -450.0 -0.35 -0.3103 -0.8667 3117857 ChemDiv3_007688 CCCCN(Cc1ccccc1)S(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N11 compound treatment 640.0 -263.0 -0.09 1120.0 350.0 0.27 0.124 0.4363 3028199 ChemDiv3_007689 CC(=O)N(Cc1ccco1)C2(CCCCC2)C(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N12 compound treatment 600.0 -303.0 -0.11 5200.0 4430.0 3.4 2.3288 0.6845 3117858 ChemDiv3_007690 COc1ccc(cc1)N2CCN(CC2)C(=O)CNC(=O)Cn3c(C)cc4ccccc4c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N13 compound treatment 560.0 -343.0 -0.12 1200.0 430.0 0.33 0.1473 0.4191 3117859 ChemDiv3_007691 COc1ccc(C(=O)Nc2ccc3nc(cc(C)c3c2)N4CCN(CC4)c5ncccn5)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N14 compound treatment 760.0 -143.0 -0.05 640.0 -130.0 -0.1 -0.1065 -0.95 3028200 ChemDiv3_007692 COC(=O)c1cn(NC(=O)C2CCCO2)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N15 compound treatment 720.0 -183.0 -0.06 1320.0 550.0 0.42 0.2526 0.5917 3117860 ChemDiv3_007693 COCCN1C(C(C(=O)NCCCN2CCC(C)CC2)c3ccccc3C1=O)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N16 compound treatment 760.0 -143.0 -0.05 680.0 -90.3 -0.07 -0.0848 -0.9879 3028201 ChemDiv3_007694 C/C(=C\c1nsc(Nc2ccccc2)n1)/NCc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N17 compound treatment 640.0 -263.0 -0.09 520.0 -250.0 -0.19 -0.2017 -0.9447 3117861 ChemDiv3_007695 CCCCN(C)C(=O)C1C(N(C)C(=O)c2ccccc12)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N18 compound treatment 760.0 -143.0 -0.05 1400.0 630.0 0.48 0.3061 0.6297 3117862 ChemDiv3_007696 Clc1ccccc1CN2CC3(OC4C=C3)C(C4C(=O)NC5CC5)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N19 compound treatment 760.0 -143.0 -0.05 640.0 -130.0 -0.1 -0.1065 -0.95 3028202 ChemDiv3_007697 COc1ccc(CCNC(=O)NC2(Oc3ccccc3O2)C(F)(F)F)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N20 compound treatment 680.0 -223.0 -0.08 2200.0 1430.0 1.1 0.7203 0.6546 3117863 ChemDiv3_007698 CCc1ccc2nc(sc2c1)N3CCC(CC3)C(=O)NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N21 compound treatment 320.0 -583.0 -0.21 680.0 -90.3 -0.07 -0.1951 -0.8953 3028203 ChemDiv3_007699 CCCn1/c(=N\C(=O)C(CC)c2ccccc2)/c(cc3c(=O)n4ccccc4nc13)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N22 compound treatment 480.0 -423.0 -0.15 4240.0 3470.0 2.66 1.7776 0.6663 3117864 ChemDiv3_007700 FC(F)(F)c1cc(nc(NCCc2ccccc2)n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N23 mock treatment 1200.0 298.0 0.11 2040.0 1270.0 0.97 0.7639 0.7791 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 N24 mock treatment 760.0 -143.0 -0.05 640.0 -130.0 -0.1 -0.1065 -0.95 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O01 compound treatment 440.0 -463.0 -0.16 360.0 -410.0 -0.32 -0.3388 -0.9538 3117865 ChemDiv3_007701 NC(=O)C1CCN(CC1)C(=O)c2n[nH]c(=O)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O02 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3028204 ChemDiv3_007702 OC(=O)C1C(N(C2CCCC2)C(=O)c3ccccc13)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O03 compound treatment 520.0 -383.0 -0.14 200.0 -570.0 -0.44 -0.4056 -0.8847 3117866 ChemDiv3_007703 COc1ccc(cc1)C2C(C(=O)N3CCCCC3)c4ccccc4C(=O)N2c5ccc(OC)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O04 compound treatment 280.0 -623.0 -0.22 240.0 -530.0 -0.41 -0.444 -0.9587 3028205 ChemDiv3_007704 CC1CC(C)(C)NC(=S)N1CCC(=O)N2CCc3ccccc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O05 compound treatment 320.0 -583.0 -0.21 200.0 -570.0 -0.44 -0.4557 -0.9413 3117867 ChemDiv3_007705 O=C(Cn1ccc2ccccc2c1=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O06 compound treatment 240.0 -663.0 -0.24 320.0 -450.0 -0.35 -0.4106 -0.9823 3117868 ChemDiv3_007706 CC1CC(C)(C)NC(=S)N1CCCC(=O)Nc2nc3ccccc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O07 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3028206 ChemDiv3_007707 COc1cc2c(cn(C)c(=O)c2cc1OC)C(=O)NCCC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O08 compound treatment 400.0 -503.0 -0.18 280.0 -490.0 -0.38 -0.3922 -0.9417 3117869 ChemDiv3_007708 COc1ccc(CCNC(=O)c2cc(Sc3ccc(F)cc3)nc4ccccc24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O09 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3117870 ChemDiv3_007709 Cc1ccc(Nc2ncc(C(=O)N3CCCCCC3)c4ccccc24)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O10 compound treatment 320.0 -583.0 -0.21 400.0 -370.0 -0.28 -0.3471 -0.9877 1167034 ChemDiv3_007710 COc1ccccc1n2cc(c3ccccc3)c4c(SCC(C)C)ncnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O11 compound treatment 280.0 -623.0 -0.22 400.0 -370.0 -0.28 -0.3572 -0.9922 3118007 ChemDiv3_007711 CCN(C(=O)c1coc(=O)c2ccccc12)c3cc(OC)ccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O12 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3028207 ChemDiv3_007712 COc1ccc(cc1)n2nc(C(=O)NCC(=O)Nc3cccc(OC)c3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O13 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3118008 ChemDiv3_007713 CCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O14 compound treatment 280.0 -623.0 -0.22 360.0 -410.0 -0.32 -0.3789 -0.9849 1720471 ChemDiv3_007714 CC(=O)N1CC(=O)Nc2ccc(Cl)cc2C1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O15 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3028208 ChemDiv3_007715 O=C(NC1CCCCC1)c2cc3c(=O)[nH]c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O16 compound treatment 440.0 -463.0 -0.16 400.0 -370.0 -0.28 -0.317 -0.9659 1267933 ChemDiv3_007716 CN(C)S(=O)(=O)c1ccc(cc1)C(=O)Nc2c3CS(=O)Cc3nn2C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O17 compound treatment 280.0 -623.0 -0.22 200.0 -570.0 -0.44 -0.4658 -0.9498 3028263 ChemDiv3_007717 COc1cc(NC(=O)c2ccc3c(c4CCCCc4nc3c2)n5ccnc5)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O18 compound treatment 280.0 -623.0 -0.22 280.0 -490.0 -0.38 -0.4223 -0.9677 3028264 ChemDiv3_007718 CCc1nnc(NC(=O)c2ccc(cc2)S(=O)(=O)N3CCCC3)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O19 compound treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 3028265 ChemDiv3_007719 CN(C1CCCCC1)C(=O)c2ccc3c(=O)n4CCCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O20 compound treatment 280.0 -623.0 -0.22 400.0 -370.0 -0.28 -0.3572 -0.9922 3028266 ChemDiv3_007720 CC1Cc2ccccc2N1C(=O)CCN3C(=O)C4C5CC(C=C5)C4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O21 compound treatment 320.0 -583.0 -0.21 1480.0 710.0 0.54 0.2391 0.4104 3118009 ChemDiv3_007721 CCCCN(C)C(=S)Nc1ccc2nc3CCCCCn3c(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O22 compound treatment 280.0 -623.0 -0.22 320.0 -450.0 -0.35 -0.4006 -0.9766 3028267 ChemDiv3_007722 CC(C)Cc1ccc(cc1)S(=O)(=O)N2C(C)Cc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O23 mock treatment 320.0 -583.0 -0.21 240.0 -530.0 -0.41 -0.434 -0.9506 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 O24 mock treatment 280.0 -623.0 -0.22 200.0 -570.0 -0.44 -0.4658 -0.9498 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P01 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3118010 ChemDiv3_007723 CC(C)Cc1ccc(cc1)S(=O)(=O)n2cccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P02 compound treatment 2600.0 1700.0 0.6 320.0 -450.0 -0.35 0.1813 0.2612 1702898 ChemDiv3_007724 Cc1nn(c(OC(=O)c2ccccc2)c1Sc3ccccc3)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P03 compound treatment 2200.0 1300.0 0.46 280.0 -490.0 -0.38 0.0593 0.0997 3118011 ChemDiv3_007725 CCc1ccccc1NC(=S)N(CCCN2CCOCC2)Cc3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P04 compound treatment 280.0 -623.0 -0.22 280.0 -490.0 -0.38 -0.4223 -0.9677 3028268 ChemDiv3_007726 Cc1ccc2[nH]c3CC[N+](C)(Cc4ccccc4)Cc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P05 compound treatment 320.0 -583.0 -0.21 320.0 -450.0 -0.35 -0.3906 -0.9697 3118012 ChemDiv3_007727 Cc1ccc(NC(=O)C(N2CCc3ccccc23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P06 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3118013 ChemDiv3_007728 O=C(CCS(=O)(=O)c1cccc2nsnc12)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P07 compound treatment 280.0 -623.0 -0.22 200.0 -570.0 -0.44 -0.4658 -0.9498 3028269 ChemDiv3_007729 CC(C)c1ccc(NC(=O)C(NC(=O)Cc2cccs2)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P08 compound treatment 2680.0 1780.0 0.63 360.0 -410.0 -0.32 0.2231 0.3166 3118014 ChemDiv3_007730 OC1(N(C(=O)Nc2ccccc21)c3ccccc3)C(=O)NC4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P09 compound treatment 320.0 -583.0 -0.21 360.0 -410.0 -0.32 -0.3689 -0.9791 3118015 ChemDiv3_007731 O=C(NC1CCCCC1)C(N2CCc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P10 compound treatment 400.0 -503.0 -0.18 240.0 -530.0 -0.41 -0.4139 -0.9313 3028270 ChemDiv3_007732 CN(c1cccc(C)c1)S(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P11 compound treatment 280.0 -623.0 -0.22 360.0 -410.0 -0.32 -0.3789 -0.9849 3118016 ChemDiv3_007733 CO/C(=N\C1CCCCC1)/C(O)c2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P12 compound treatment 440.0 -463.0 -0.16 320.0 -450.0 -0.35 -0.3605 -0.942 3028271 ChemDiv3_007734 Cc1cc2ccccc2c(=O)n1CC(=O)NCC(=O)NCC3COc4ccccc4O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P13 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3118017 ChemDiv3_007735 CC1CCN(CC1)S(=O)(=O)c2c(C)sc3ncn(CC(=O)NC4CCCC(C)C4C)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P14 compound treatment 320.0 -583.0 -0.21 280.0 -490.0 -0.38 -0.4123 -0.9601 3118018 ChemDiv3_007736 COC(=O)c1cn(NC(=O)/C(=C/c2ccccc2)/C)c(=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P15 compound treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 3028272 ChemDiv3_007737 COc1ccc(cc1)C2C(C(=O)NCCC3=CCCCC3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P16 compound treatment 240.0 -663.0 -0.24 240.0 -530.0 -0.41 -0.4541 -0.9659 3118019 ChemDiv3_007738 C/C(=C\c1nsc(Nc2ccccc2)n1)/NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P17 compound treatment 400.0 -503.0 -0.18 320.0 -450.0 -0.35 -0.3705 -0.9525 3118020 ChemDiv3_007739 COc1ccc(cc1)C2C(C(=O)N3CCCCC3)c4ccccc4C(=O)N2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P18 compound treatment 280.0 -623.0 -0.22 240.0 -530.0 -0.41 -0.444 -0.9587 3028273 ChemDiv3_007740 Cc1ccc(CN2CC3(OC4C=C3)C(C4C(=O)NCCc5ccc(Cl)cc5)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P19 compound treatment 240.0 -663.0 -0.24 280.0 -490.0 -0.38 -0.4324 -0.9743 3118021 ChemDiv3_007741 CCN(C1CCCCC1)C(=O)NC2(Oc3ccccc3O2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P20 compound treatment 400.0 -503.0 -0.18 240.0 -530.0 -0.41 -0.4139 -0.9313 3118022 ChemDiv3_007742 CCc1ccc2nc(sc2c1)N3CCC(CC3)C(=O)NCC4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P21 compound treatment 280.0 -623.0 -0.22 280.0 -490.0 -0.38 -0.4223 -0.9677 3028274 ChemDiv3_007743 CCOC(=O)c/1cc2c(=O)n3ccccc3nc2n(C(C)C)\c1=N\C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P22 compound treatment 280.0 -623.0 -0.22 160.0 -610.0 -0.47 -0.4875 -0.9411 3118023 ChemDiv3_007744 FC(F)(F)c1cc(nc(NC2CCCC2)n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P23 mock treatment 320.0 -583.0 -0.21 240.0 -530.0 -0.41 -0.434 -0.9506 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2022 P24 mock treatment 400.0 -503.0 -0.18 240.0 -530.0 -0.41 -0.4139 -0.9313 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A01 compound treatment 1600.0 571.0 0.2 240.0 -388.0 -0.3 -0.0671 -0.1863 3028275 ChemDiv3_007745 FC(F)(F)c1cc(nc(NCc2cccnc2)n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A02 compound treatment 3320.0 2290.0 0.81 360.0 -268.0 -0.21 0.4295 0.5123 3118024 ChemDiv3_007746 Clc1cccc(/C=C\2/Cc3ccccc3C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A03 compound treatment 880.0 -149.0 -0.05 280.0 -348.0 -0.27 -0.226 -0.8309 3118025 ChemDiv3_007747 CC1(CC2CC(C)(C)C1)CN2c3nc(cc(n3)C(F)(F)F)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A04 compound treatment 480.0 -549.0 -0.19 360.0 -268.0 -0.21 -0.2829 -0.9996 3028276 ChemDiv3_007748 O=C1/C(=C/c2ccc(cc2)N3CCOCC3)/Cc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A05 compound treatment 320.0 -709.0 -0.25 680.0 52.5 0.04 -0.1493 -0.5863 3118026 ChemDiv3_007749 O=C(CCS(=O)(=O)c1cccs1)NC2CCCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A06 compound treatment 200.0 -829.0 -0.29 320.0 -308.0 -0.24 -0.3748 -0.9941 3028277 ChemDiv3_007750 O=C/1C(CC\C1=C/c2ccc(cc2)N3CCOCC3)C4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A07 compound treatment 680.0 -349.0 -0.12 280.0 -348.0 -0.27 -0.2761 -0.939 3118027 ChemDiv3_007751 COc1ccc(cc1)C2C(CCC(=O)N2c3ccc4OCOc4c3)C(=O)NCc5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A08 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3118028 ChemDiv3_007752 COc1ccccc1OCCn2cc(/C=C/3\Cc4ccccc4C3=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A09 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 3028278 ChemDiv3_007753 CCOC(=O)N1CCN(CC1)C(=O)C2CC(=O)N(C2c3ccc(OC)cc3)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A10 compound treatment 200.0 -829.0 -0.29 280.0 -348.0 -0.27 -0.3965 -0.9988 3118029 ChemDiv3_007754 COc1ccc(/C=C/2\CC(C/C(=C/c3ccc(OC)cc3OC)/C2=O)C(C)(C)C)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A11 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 1213232 ChemDiv3_007755 COc1cccc(NC(=O)CSc2nc3c4ccccc4[nH]c3c(=O)n2C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A12 compound treatment 440.0 -589.0 -0.21 360.0 -268.0 -0.21 -0.2929 -1.0 3118030 ChemDiv3_007756 CN1C/C(=C\c2ccc(F)c(F)c2)/C(=O)\C(=C\c3ccc(F)c(F)c3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A13 compound treatment 240.0 -789.0 -0.28 360.0 -268.0 -0.21 -0.3431 -0.9884 1398001 ChemDiv3_007757 CCOc1ccc(cc1)n2c(SCC)nc3c4ccccc4[nH]c3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A14 compound treatment 720.0 -309.0 -0.11 240.0 -388.0 -0.3 -0.2878 -0.9079 3028279 ChemDiv3_007758 CC(C)/C=C/1\CC/C(=C\c2ccc(cc2)N(C)C)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A15 compound treatment 280.0 -749.0 -0.27 360.0 -268.0 -0.21 -0.333 -0.9919 1343294 ChemDiv3_007759 CC(NCc1nc2ccccc2n1C)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A16 compound treatment 280.0 -749.0 -0.27 240.0 -388.0 -0.3 -0.3982 -0.9984 3028280 ChemDiv3_007760 CC(C)CCNC(=O)c1oc2ccc(cc2c1C)S(=O)(=O)N3CCC4(CC3)OCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A17 compound treatment 280.0 -749.0 -0.27 360.0 -268.0 -0.21 -0.333 -0.9919 3118031 ChemDiv3_007761 C=CCN1C(=O)C(CC(=O)Nc2ccccc2)N(Cc3ccccn3)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A18 compound treatment 360.0 -669.0 -0.24 240.0 -388.0 -0.3 -0.3781 -0.9937 3120677 ChemDiv3_007762 CN1C(C(C(=O)N2CCCCC2)c3ccccc3C1=O)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A19 compound treatment 240.0 -789.0 -0.28 280.0 -348.0 -0.27 -0.3865 -0.9997 3028281 ChemDiv3_007763 CN1C/C(=C\c2ccc3ccccc3c2)/C(=O)\C(=C/c4cccc5ccccc45)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A20 compound treatment 360.0 -669.0 -0.24 320.0 -308.0 -0.24 -0.3347 -1.0 3120678 ChemDiv3_007764 CC(C)C(NC(=O)C1CCC(C)CC1)C(=O)Nc2ccc(F)c(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A21 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 3028282 ChemDiv3_007765 CN(C)c1ccc(/C=C/2\Cc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A22 compound treatment 160.0 -869.0 -0.31 2240.0 1610.0 1.24 0.6574 0.5153 3120679 ChemDiv3_007766 COc1ccc(NC(=O)C(NC(=O)C2CCCCC2)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A23 mock treatment 240.0 -789.0 -0.28 400.0 -228.0 -0.17 -0.3214 -0.9743 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 A24 mock treatment 200.0 -829.0 -0.29 360.0 -268.0 -0.21 -0.3531 -0.9846 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B01 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 3120680 ChemDiv3_007767 CC(C)CC(NC(=O)C1CCC(C)CC1)C(=O)Nc2cccc(C)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B02 compound treatment 440.0 -589.0 -0.21 360.0 -268.0 -0.21 -0.2929 -1.0 3028283 ChemDiv3_007768 O=C(CCc1nc2sc3CCCCc3c2c(=O)[nH]1)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B03 compound treatment 320.0 -709.0 -0.25 400.0 -228.0 -0.17 -0.3013 -0.9842 3120681 ChemDiv3_007769 CCOC(=O)N1CCC(CC1)NC(=O)C(NC(=O)C2CCC(C)CC2)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B04 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3028284 ChemDiv3_007770 CCCn1c(CCNC(=O)c2cccc(C)c2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B05 compound treatment 280.0 -749.0 -0.27 360.0 -268.0 -0.21 -0.333 -0.9919 3120682 ChemDiv3_007771 CCN(CC)S(=O)(=O)c1ccc(cc1)C(=O)NCCSc2c[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B06 compound treatment 360.0 -669.0 -0.24 320.0 -308.0 -0.24 -0.3347 -1.0 3028285 ChemDiv3_007772 C=CCn1c(nc2ccccc12)C(Cc3ccccc3)NC(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B07 compound treatment 440.0 -589.0 -0.21 440.0 -188.0 -0.14 -0.2495 -0.9835 3120683 ChemDiv3_007773 O=C(NCCSc1c([nH]c2ccccc12)c3ccccc3)c4ccc(cc4)N5C(=O)CCC5=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B08 compound treatment 280.0 -749.0 -0.27 440.0 -188.0 -0.14 -0.2896 -0.9586 3120684 ChemDiv3_007774 O=C(CSc1oc(nc1S(=O)(=O)c2ccccc2)c3cccs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B09 compound treatment 240.0 -789.0 -0.28 200.0 -428.0 -0.33 -0.4299 -0.9968 3028286 ChemDiv3_007775 Oc1nc(nc(c1C#N)c2ccccc2)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B10 compound treatment 320.0 -709.0 -0.25 360.0 -268.0 -0.21 -0.323 -0.995 3120685 ChemDiv3_007776 Cc1nc2nc(SCC(=O)N3CCC4(CC3)OCCO4)nn2c(C)c1Cc5ccccc5Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B11 compound treatment 240.0 -789.0 -0.28 240.0 -388.0 -0.3 -0.4082 -0.9995 3028287 ChemDiv3_007777 CC(C)c1ccc(NC(=O)c2ccc(NS(=O)(=O)c3cccs3)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B12 compound treatment 840.0 -189.0 -0.07 280.0 -348.0 -0.27 -0.236 -0.858 3120686 ChemDiv3_007778 COc1cccc(NC(=O)c2cc3c(=O)oc4ccccc4c3s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B13 compound treatment 320.0 -709.0 -0.25 520.0 -108.0 -0.08 -0.2361 -0.8924 3028288 ChemDiv3_007779 CN(Cc1ccccc1)C(=O)CNC(=O)Cn2ccc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B14 compound treatment 720.0 -309.0 -0.11 360.0 -268.0 -0.21 -0.2227 -0.9567 3120687 ChemDiv3_007780 O=C(Nc1c(nc2ccccn12)c3cccs3)C(c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B15 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3120688 ChemDiv3_007781 CCn1cc(C(=O)N(C)Cc2ccccc2)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B16 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3028289 ChemDiv3_007782 Cc1ccc(C)c(NC(=O)CS(=O)(=O)c2c[nH]c3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B17 compound treatment 320.0 -709.0 -0.25 160.0 -468.0 -0.36 -0.4316 -0.9848 3120689 ChemDiv3_007783 COc1cc2c(cn(CC(C)C)c(=O)c2cc1OC)C(=O)N3CCC4(CC3)OCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B18 compound treatment 240.0 -789.0 -0.28 240.0 -388.0 -0.3 -0.4082 -0.9995 3028290 ChemDiv3_007784 Clc1ccc(Cn2cc(c3ccccc23)S(=O)(=O)CC(=O)N4CCc5ccccc45)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B19 compound treatment 4280.0 3250.0 1.15 360.0 -268.0 -0.21 0.6703 0.5722 3120690 ChemDiv3_007785 NC(=O)C[n+]1ccn2c(NC3CCCCC3)c(nc2c1)c4ccccc4O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B20 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3028291 ChemDiv3_007786 COCCn1c(=O)[nH]c2cc(ccc2c1=O)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B21 compound treatment 480.0 -549.0 -0.19 240.0 -388.0 -0.3 -0.348 -0.9789 3120691 ChemDiv3_007787 COC(CNC(=O)Cc1ccc(cc1)n2c(=O)[nH]c3ccsc3c2=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B22 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3120692 ChemDiv3_007788 CCOC(=O)C1CCCN(C1)C(=O)Cc2c([nH]c3ccccc23)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B23 mock treatment 320.0 -709.0 -0.25 2520.0 1890.0 1.45 0.8496 0.5762 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 B24 mock treatment 240.0 -789.0 -0.28 360.0 -268.0 -0.21 -0.3431 -0.9884 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C01 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3028292 ChemDiv3_007789 CCN(CC)c1nc(cc(n1)C(F)(F)F)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C02 compound treatment 320.0 -709.0 -0.25 400.0 -228.0 -0.17 -0.3013 -0.9842 3120693 ChemDiv3_007790 O=C/1C(CC\C1=C/c2ccccc2)C3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C03 compound treatment 360.0 -669.0 -0.24 360.0 -268.0 -0.21 -0.313 -0.9974 1221975 ChemDiv3_007791 COc1ccc(CN2C(=O)c3ccc(F)cc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C04 compound treatment 600.0 -429.0 -0.15 240.0 -388.0 -0.3 -0.3179 -0.9515 3120694 ChemDiv3_007792 O=C/1/C(=C/c2ccc(cc2)N3CCOCC3)/CC\C1=C/c4ccc(cc4)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C05 compound treatment 480.0 -549.0 -0.19 280.0 -348.0 -0.27 -0.3263 -0.988 3028413 ChemDiv3_007793 O=C(CNS(=O)(=O)c1cccs1)NC(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C06 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3120695 ChemDiv3_007794 O=C1/C(=C/c2ccc(cc2)N3CCOCC3)/CCc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C07 compound treatment 240.0 -789.0 -0.28 240.0 -388.0 -0.3 -0.4082 -0.9995 3028414 ChemDiv3_007795 COc1cc2C(C(N(C)C(=O)c2cc1OC)c3cccs3)C(=O)NCCN(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C08 compound treatment 320.0 -709.0 -0.25 360.0 -268.0 -0.21 -0.323 -0.995 3120696 ChemDiv3_007796 COc1cccc(/C=C/2\CC/C(=C\c3cccc(OC)c3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C09 compound treatment 280.0 -749.0 -0.27 240.0 -388.0 -0.3 -0.3982 -0.9984 3120697 ChemDiv3_007797 COc1ccc(cc1)C2C(CC(=O)N2c3ccc(OC)cc3)C(=O)N(C)c4ccc(cc4)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C10 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3028415 ChemDiv3_007798 CCC1C/C(=C\c2ccccc2OC)/C(=O)\C(=C/c3ccccc3OC)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C11 compound treatment 400.0 -629.0 -0.22 360.0 -268.0 -0.21 -0.3029 -0.9991 1164510 ChemDiv3_007799 Cn1c(SCc2ccccc2)nc3c4ccccc4[nH]c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C12 compound treatment 360.0 -669.0 -0.24 200.0 -428.0 -0.33 -0.3998 -0.9873 3028416 ChemDiv3_007800 CN1C/C(=C\c2cc(Br)cs2)/C(=O)\C(=C\c3cc(Br)cs3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C13 compound treatment 320.0 -709.0 -0.25 360.0 -268.0 -0.21 -0.323 -0.995 1215694 ChemDiv3_007801 CCCSc1nc2c3ccccc3[nH]c2c(=O)n1c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C14 compound treatment 320.0 -709.0 -0.25 280.0 -348.0 -0.27 -0.3664 -0.9996 3120698 ChemDiv3_007802 CC(C)/C=C/1\CC/C(=C\c2ccc(Cl)cc2)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C15 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3028417 ChemDiv3_007803 Cc1ccc(NCc2nc3ccccc3n2C)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C16 compound treatment 400.0 -629.0 -0.22 360.0 -268.0 -0.21 -0.3029 -0.9991 3120699 ChemDiv3_007804 CC1CC(C)CN(C1)S(=O)(=O)c2ccc3oc(C(=O)NC4CCCc5ccccc45)c(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C17 compound treatment 1920.0 891.0 0.32 360.0 -268.0 -0.21 0.0783 0.2078 3028418 ChemDiv3_007805 CCc1ccc(NC(=O)c2sc3[nH]c(=O)c(cc3c2N)C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C18 compound treatment 240.0 -789.0 -0.28 240.0 -388.0 -0.3 -0.4082 -0.9995 3120700 ChemDiv3_007806 CCc1ccc(NC(=O)C2C(N(C)C(=O)c3ccccc23)c4cccs4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C19 compound treatment 2280.0 1250.0 0.44 280.0 -348.0 -0.27 0.1252 0.2418 3028419 ChemDiv3_007807 CC1C/C(=C\c2ccco2)/C(=O)\C(=C/c3ccco3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C20 compound treatment 3120.0 2090.0 0.74 320.0 -308.0 -0.24 0.3576 0.4594 3120701 ChemDiv3_007808 CC(C)C(NC(=O)C1CCCCC1)C(=O)N2CCN(CC2)c3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C21 compound treatment 320.0 -709.0 -0.25 200.0 -428.0 -0.33 -0.4099 -0.9913 3028420 ChemDiv3_007809 O=C1/C(=C/c2ccco2)/Cc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C22 compound treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 3120881 ChemDiv3_007810 CC(C)C(NC(=O)c1ccc(cc1)C2(CC3CC4CC(C3)C2)C4)C(=O)NCC5CCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C23 mock treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 C24 mock treatment 240.0 -789.0 -0.28 200.0 -428.0 -0.33 -0.4299 -0.9968 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D01 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3120882 ChemDiv3_007811 CCOC(=O)N1CCN(CC1)C(=O)C(NC(=O)c2ccc(cc2)C3(CC4CC5CC(C4)C3)C5)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D02 compound treatment 320.0 -709.0 -0.25 280.0 -348.0 -0.27 -0.3664 -0.9996 3028421 ChemDiv3_007812 CCCn1c(CNC(=O)CC)nc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D03 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3120883 ChemDiv3_007813 CCc1cccc(NC(=O)C(NC(=O)C2CCC(C)CC2)C(C)C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D04 compound treatment 240.0 -789.0 -0.28 400.0 -228.0 -0.17 -0.3214 -0.9743 3028422 ChemDiv3_007814 CCCCn1c(CCNC(=O)c2ccc(Cl)cc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D05 compound treatment 360.0 -669.0 -0.24 1040.0 413.0 0.32 0.0562 0.142 3120884 ChemDiv3_007815 O=C(NCCSc1c[nH]c2ccccc12)c3ccc(cc3)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D06 compound treatment 320.0 -709.0 -0.25 280.0 -348.0 -0.27 -0.3664 -0.9996 3028423 ChemDiv3_007816 COc1cc(cc(OC)c1OC)C(=O)NC(Cc2ccccc2)c3nc4ccccc4[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D07 compound treatment 320.0 -709.0 -0.25 2360.0 1730.0 1.33 0.7627 0.5635 3120885 ChemDiv3_007817 CC(C)C(=O)NCCSc1c([nH]c2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D08 compound treatment 520.0 -509.0 -0.18 1480.0 853.0 0.65 0.3352 0.4937 3120886 ChemDiv3_007818 Cc1ccc(cc1)S(=O)(=O)c2nc(oc2SCc3ccccc3F)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D09 compound treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 3028424 ChemDiv3_007819 FC(F)(F)c1nc(nc2CCCCCc12)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D10 compound treatment 240.0 -789.0 -0.28 360.0 -268.0 -0.21 -0.3431 -0.9884 3120887 ChemDiv3_007820 CCc1ccc(NC(=O)c2ccc(NC(=O)C3CCCO3)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D11 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3028447 ChemDiv3_007821 O=C(NC1CCN(Cc2ccccc2)CC1)c3ccc(NS(=O)(=O)c4cccs4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D12 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3120888 ChemDiv3_007822 CCC(C)NC(=O)C1CCC(=O)N(C1c2ccc(OC)cc2)c3cc(OC)c(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D13 compound treatment 280.0 -749.0 -0.27 360.0 -268.0 -0.21 -0.333 -0.9919 3028448 ChemDiv3_007823 O=C(CNC(=O)Cn1ccc2ccccc2c1=O)NC3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D14 compound treatment 240.0 -789.0 -0.28 400.0 -228.0 -0.17 -0.3214 -0.9743 3120889 ChemDiv3_007824 FC(F)(F)c1cccc(c1)C(=O)Nc2c(nc3ccccn23)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D15 compound treatment 320.0 -709.0 -0.25 240.0 -388.0 -0.3 -0.3881 -0.9965 3120890 ChemDiv3_007825 CCn1cc(C(=O)NC2CCCC(C)C2C)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D16 compound treatment 320.0 -709.0 -0.25 280.0 -348.0 -0.27 -0.3664 -0.9996 3028449 ChemDiv3_007826 Cc1cccc(NC(=O)CS(=O)(=O)c2cn(C)c3ccccc23)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D17 compound treatment 2800.0 1770.0 0.63 280.0 -348.0 -0.27 0.2557 0.3745 3120891 ChemDiv3_007827 COC(=O)CNC(=O)c1cn(CC(C)C)c(=O)c2cc(OC)c(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D18 compound treatment 1720.0 691.0 0.25 320.0 -308.0 -0.24 0.0065 0.019 3028450 ChemDiv3_007828 Clc1ccc(Cn2cc(c3ccccc23)S(=O)(=O)CC(=O)Nc4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D19 compound treatment 440.0 -589.0 -0.21 2440.0 1810.0 1.39 0.8362 0.5943 3120892 ChemDiv3_007829 Cc1ccc(Nc2c(nc3c[n+](CC(=O)N)ccn23)c4c[nH]c5ccccc45)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D20 compound treatment 400.0 -629.0 -0.22 360.0 -268.0 -0.21 -0.3029 -0.9991 3120893 ChemDiv3_007830 COc1cc2[nH]c(=O)n(CCCC(=O)NC3CCCC3)c(=O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D21 compound treatment 4920.0 3890.0 1.38 480.0 -148.0 -0.11 0.896 0.6469 3028451 ChemDiv3_007831 CC(C)CCNC(=O)c1ccc(Cn2c(=O)[nH]c3ccsc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D22 compound treatment 960.0 -68.8 -0.02 360.0 -268.0 -0.21 -0.1625 -0.7856 3120894 ChemDiv3_007832 CCN(CC)C(=O)Cc1c([nH]c2ccccc12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D23 mock treatment 400.0 -629.0 -0.22 280.0 -348.0 -0.27 -0.3464 -0.996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 D24 mock treatment 320.0 -709.0 -0.25 680.0 52.5 0.04 -0.1493 -0.5863 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E01 compound treatment 1040.0 11.3 0.0 920.0 293.0 0.22 0.1616 0.7196 3028452 ChemDiv3_007833 COc1ccc(cc1)c2cc(nc(n2)N3CCOCC3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E02 compound treatment 320.0 -709.0 -0.25 1080.0 453.0 0.35 0.0679 0.1582 3120895 ChemDiv3_007834 CN(C)c1ccc(/C=C/2\CCC(C3CCCC3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E03 compound treatment 560.0 -469.0 -0.17 360.0 -268.0 -0.21 -0.2628 -0.9945 1786811 ChemDiv3_007835 CCOC(=O)N1CCN(CC1)C(=O)C2COc3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E04 compound treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 3120896 ChemDiv3_007836 CN1CCCc2cc(/C=C/3\CC/C(=C/c4ccc5CCCN(C)c5c4)/C3=O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E05 compound treatment 360.0 -669.0 -0.24 2880.0 2250.0 1.73 1.055 0.6044 3120897 ChemDiv3_007837 Cc1ccc2nc(NC(=O)CCNS(=O)(=O)c3cccs3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E06 compound treatment 320.0 -709.0 -0.25 480.0 -148.0 -0.11 -0.2579 -0.9351 3028453 ChemDiv3_007838 Brc1ccccc1/C=C/2\Cc3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E07 compound treatment 1520.0 491.0 0.17 440.0 -188.0 -0.14 0.0214 0.0949 3120898 ChemDiv3_007839 COc1cc2C(C(N(C)C(=O)c2cc1OC)c3cccs3)C(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E08 compound treatment 7000.0 5970.0 2.12 840.0 213.0 0.16 1.6132 0.7593 3028454 ChemDiv3_007840 Cc1ccc(/C=C/2\CC/C(=C\c3ccc(C)o3)/C2=O)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E09 compound treatment 560.0 -469.0 -0.17 560.0 -67.5 -0.05 -0.1542 -0.8855 3120899 ChemDiv3_007841 CCOC(=O)C(C)Sc1ncnc2[nH]cnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E10 compound treatment 4000.0 2970.0 1.05 680.0 52.5 0.04 0.7738 0.7336 3028455 ChemDiv3_007842 COc1ccc(Br)cc1C2CC(=O)C(C)C(N2)c3cc(Br)ccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E11 compound treatment 2560.0 1530.0 0.54 880.0 253.0 0.19 0.5212 0.9036 1491562 ChemDiv3_007843 COC(=O)C(C)Sc1nc2c3ccccc3[nH]c2c(=O)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E12 compound treatment 600.0 -429.0 -0.15 440.0 -188.0 -0.14 -0.2093 -0.9996 3120900 ChemDiv3_007844 COc1ccc(/C=C/2\CCC(C3CCCC3)C2=O)cc1Cn4cccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E13 compound treatment 3720.0 2690.0 0.95 1120.0 493.0 0.38 0.9424 0.9178 1479023 ChemDiv3_007845 Clc1cccc(c1)n2c(SCC(=O)N3CCCCCC3)nc4c5ccccc5[nH]c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E14 compound treatment 680.0 -349.0 -0.12 1680.0 1050.0 0.81 0.4839 0.5919 3120901 ChemDiv3_007846 COc1ccc(/C=C/2\CC/C(=C\CC(C)C)/C2=O)cc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E15 compound treatment 440.0 -589.0 -0.21 680.0 52.5 0.04 -0.1192 -0.5603 3028456 ChemDiv3_007847 Clc1ccc(Cn2c(CNc3ccccc3)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E16 compound treatment 440.0 -589.0 -0.21 520.0 -108.0 -0.08 -0.206 -0.9175 3120902 ChemDiv3_007848 CCN(CC)S(=O)(=O)c1ccc2oc(C(=O)NC3CCCCC3C)c(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E17 compound treatment 5200.0 4170.0 1.48 1600.0 973.0 0.75 1.5743 0.9498 3120903 ChemDiv3_007849 Cc1cccc(NC(=O)c2sc3[nH]c(=O)c(cc3c2N)C(=O)O)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E18 compound treatment 2120.0 1090.0 0.39 1200.0 573.0 0.44 0.5845 0.998 3028457 ChemDiv3_007850 COc1cc2c(cn(C)c(=O)c2cc1OC)C(=O)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E19 compound treatment 14720.0 13700.0 4.86 2480.0 1850.0 1.42 4.44 0.8773 3120904 ChemDiv3_007851 CC1C/C(=C\c2ccncc2)/C(=O)\C(=C/c3ccncc3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E20 compound treatment 480.0 -549.0 -0.19 1200.0 573.0 0.44 0.1731 0.3602 3120905 ChemDiv3_007852 CC(=O)Nc1ccc(NC(=O)C(Cc2ccccc2)NC(=O)C3CCCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E21 compound treatment 1480.0 451.0 0.16 520.0 -108.0 -0.08 0.0548 0.3045 3028458 ChemDiv3_007853 COc1ccc2C(=O)/C(=C\c3ccco3)/CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E22 compound treatment 680.0 -349.0 -0.12 1440.0 813.0 0.62 0.3536 0.556 3121298 ChemDiv3_007854 CCN1CCCC1CNC(=O)C(NC(=O)c2ccc(cc2)C3(CC4CC5CC(C4)C3)C5)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E23 mock treatment 480.0 -549.0 -0.19 560.0 -67.5 -0.05 -0.1743 -0.8652 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 E24 mock treatment 1520.0 491.0 0.17 880.0 253.0 0.19 0.2603 0.9986 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F01 compound treatment 1400.0 371.0 0.13 2080.0 1450.0 1.12 0.8816 0.7852 3028459 ChemDiv3_007855 CC(C)CC(NC(=O)c1ccc(cc1)C2(CC3CC4CC(C3)C2)C4)C(=O)NCc5cccnc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F02 compound treatment 1760.0 731.0 0.26 920.0 293.0 0.22 0.3422 0.9974 3121092 ChemDiv3_007856 CCCn1c(CNC(=O)c2cc(OC)c(OC)c(OC)c2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F03 compound treatment 1040.0 11.3 0.0 320.0 -308.0 -0.24 -0.1641 -0.6951 3028460 ChemDiv3_007857 CCCC1CCC(CC1)C(=O)NC(C(C)C)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F04 compound treatment 520.0 -509.0 -0.18 1400.0 773.0 0.59 0.2917 0.4706 3121093 ChemDiv3_007858 COc1cc(cc(OC)c1OC)C(=O)NCCc2nc3ccccc3n2CC(=C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F05 compound treatment 760.0 -269.0 -0.1 760.0 133.0 0.1 0.0045 0.0324 3028487 ChemDiv3_007859 COc1cc(/C=C/C(=O)NCCSc2c[nH]c3ccccc23)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F06 compound treatment 4640.0 3610.0 1.28 680.0 52.5 0.04 0.9344 0.729 3121094 ChemDiv3_007860 CCOC(=O)c1[nH]c2ccccc2c1NC(=S)Nc3cccc(C)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F07 compound treatment 3600.0 2570.0 0.91 2760.0 2130.0 1.64 1.8026 0.9619 3121095 ChemDiv3_007861 Cc1[nH]c2ccccc2c1SCCNC(=O)c3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F08 compound treatment 3000.0 1970.0 0.7 2160.0 1530.0 1.18 1.3264 0.9691 3028488 ChemDiv3_007862 Clc1ccc(cc1)S(=O)(=O)c2nc(oc2SCC(=O)NC3CCCCC3)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F09 compound treatment 840.0 -189.0 -0.07 2160.0 1530.0 1.18 0.7846 0.6658 3121096 ChemDiv3_007863 FC(F)(F)c1nc(NCc2ccccc2)nc3CCCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F10 compound treatment 520.0 -509.0 -0.18 1120.0 493.0 0.38 0.1397 0.3335 3121097 ChemDiv3_007864 CCOC(=O)N1CCC(CC1)NC(=O)c2ccc(NC(=O)C3CCCO3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F11 compound treatment 840.0 -189.0 -0.07 1320.0 693.0 0.53 0.3286 0.6132 3028489 ChemDiv3_007865 COc1ccc(cc1)N2CCN(CC2)C(=O)c3ccc(NS(=O)(=O)c4cccs4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F12 compound treatment 720.0 -309.0 -0.11 760.0 133.0 0.1 -0.0055 -0.0369 3121098 ChemDiv3_007866 CCCCN(C)C(=O)C1CCC(=O)N(C1c2ccc(OC)cc2)c3cc(OC)c(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F13 compound treatment 480.0 -549.0 -0.19 6920.0 6290.0 4.83 3.2783 0.6781 3028490 ChemDiv3_007867 O=C(Cn1ccc2ccccc2c1=O)NCC(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F14 compound treatment 640.0 -389.0 -0.14 840.0 213.0 0.16 0.0178 0.0835 3121099 ChemDiv3_007868 Cc1ccn2c(NC(=O)C3CCCCC3)c(nc2c1)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F15 compound treatment 760.0 -269.0 -0.1 3000.0 2370.0 1.82 1.2205 0.6692 3028491 ChemDiv3_007869 CCn1cc(C(=O)NCc2cccnc2)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F16 compound treatment 1080.0 51.3 0.02 1040.0 413.0 0.32 0.2368 0.7465 3121100 ChemDiv3_007870 CCn1cc(c2ccccc12)S(=O)(=O)CC(=O)Nc3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F17 compound treatment 1040.0 11.3 0.0 3480.0 2850.0 2.19 1.5513 0.7084 3121101 ChemDiv3_007871 COc1cc2c(cn(CC(C)C)c(=O)c2cc1OC)C(=O)NCCCN3CCN(C)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F18 compound treatment 1200.0 171.0 0.06 840.0 213.0 0.16 0.1583 0.9094 3028492 ChemDiv3_007872 Fc1ccc(CS(=O)(=O)c2cn(Cc3ccccc3Cl)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F19 compound treatment 1360.0 331.0 0.12 1360.0 733.0 0.56 0.4807 0.8368 3121102 ChemDiv3_007873 Cc1cccc(C)c1/N=C/2\Oc3ccccc3N(C(=O)C(F)(F)F)C2(C)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F20 compound treatment 840.0 -189.0 -0.07 2800.0 2170.0 1.67 1.132 0.6782 3028493 ChemDiv3_007874 COc1cc2[nH]c(=O)n(CCCC(=O)N3CCN(CC3)c4cccc(Cl)c4)c(=O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F21 compound treatment 680.0 -349.0 -0.12 800.0 173.0 0.13 0.0062 0.034 3121103 ChemDiv3_007875 O=C(N1CCCCC1)c2ccc(Cn3c(=O)[nH]c4ccsc4c3=O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F22 compound treatment 720.0 -309.0 -0.11 1360.0 733.0 0.56 0.3202 0.5589 3121104 ChemDiv3_007876 CC1CC(C)CN(CCCNC(=O)Cc2c([nH]c3ccccc23)C(=O)O)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F23 mock treatment 1000.0 -28.8 -0.01 680.0 52.5 0.04 0.0213 0.512 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 F24 mock treatment 2440.0 1410.0 0.5 1120.0 493.0 0.38 0.6214 0.9904 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G01 compound treatment 5600.0 4570.0 1.62 320.0 -308.0 -0.24 0.9797 0.5979 3028494 ChemDiv3_007877 COc1ccc(cc1)c2cc(nc(n2)N3CCCCCC3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G02 compound treatment 840.0 -189.0 -0.07 480.0 -148.0 -0.11 -0.1274 -0.9686 3121105 ChemDiv3_007878 O=C1/C(=C\c2ccccn2)/Cc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G03 compound treatment 400.0 -629.0 -0.22 320.0 -308.0 -0.24 -0.3246 -0.9996 1773605 ChemDiv3_007879 CCOc1ccc(OCC)c(NC(=O)C2COc3ccccc3O2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G04 compound treatment 3000.0 1970.0 0.7 440.0 -188.0 -0.14 0.3927 0.55 3121106 ChemDiv3_007880 Cn1cccc1/C=C/2\CCc3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G05 compound treatment 1640.0 611.0 0.22 360.0 -268.0 -0.21 0.0081 0.0272 3121107 ChemDiv3_007881 CCC(=O)N1CCc2cc(Br)cc(c12)S(=O)(=O)NCc3ccccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G06 compound treatment 1320.0 291.0 0.1 1920.0 1290.0 0.99 0.7747 0.7765 3028495 ChemDiv3_007882 CCn1c2ccccc2c3cc(/C=C/4\Cc5ccccc5C4=O)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G07 compound treatment 520.0 -509.0 -0.18 520.0 -108.0 -0.08 -0.186 -0.9371 3121108 ChemDiv3_007883 COc1ccccc1Nc2ncc(C(=O)NCCc3ccc(OC)c(OC)c3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G08 compound treatment 480.0 -549.0 -0.19 560.0 -67.5 -0.05 -0.1743 -0.8652 3028496 ChemDiv3_007884 CCN1C/C(=C\c2ccccc2)/C(=O)\C(=C\c3ccccc3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G09 compound treatment 720.0 -309.0 -0.11 1960.0 1330.0 1.02 0.6459 0.6278 3121109 ChemDiv3_007885 O=C(CSc1nc2CCSc2c(=O)n1c3ccccc3)N4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G10 compound treatment 640.0 -389.0 -0.14 1400.0 773.0 0.59 0.3218 0.5286 3121110 ChemDiv3_007886 O=C/1/C(=C/c2ccccn2)/CC(C\C1=C/c3ccccn3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G11 compound treatment 1440.0 411.0 0.15 520.0 -108.0 -0.08 0.0448 0.2673 1364356 ChemDiv3_007887 CCC1CCCCN1C(=O)CSc2nc3c4ccccc4[nH]c3c(=O)n2c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G12 compound treatment 1800.0 771.0 0.27 480.0 -148.0 -0.11 0.1134 0.3829 3121111 ChemDiv3_007888 COc1ccc(/C=C/2\CCc3ccccc3C2=O)cc1Cn4cccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G13 compound treatment 1800.0 771.0 0.27 1600.0 973.0 0.75 0.7214 0.9072 1642950 ChemDiv3_007889 NC(=O)CSc1nc2c3ccccc3[nH]c2c(=O)n1c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G14 compound treatment 400.0 -629.0 -0.22 800.0 173.0 0.13 -0.0641 -0.247 3028497 ChemDiv3_007890 CSc1ccc(/C=C/2\CC/C(=C\C(C)C)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G15 compound treatment 840.0 -189.0 -0.07 720.0 92.5 0.07 0.0029 0.0294 3121112 ChemDiv3_007891 COc1ccc(NCc2nc3ccccc3n2CCOc4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G16 compound treatment 1080.0 51.3 0.02 400.0 -228.0 -0.17 -0.1106 -0.6301 3028498 ChemDiv3_007892 Cc1c(oc2ccc(cc12)S(=O)(=O)N3CCCC3)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G17 compound treatment 6200.0 5170.0 1.83 360.0 -268.0 -0.21 1.152 0.6241 3121113 ChemDiv3_007893 Nc1c(sc2[nH]c(=O)c(cc12)C(=O)O)C(=O)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G18 compound treatment 1680.0 651.0 0.23 400.0 -228.0 -0.17 0.0399 0.1376 3028499 ChemDiv3_007894 COc1cc2c(cn(C)c(=O)c2cc1OC)C(=O)N3CCCCC3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G19 compound treatment 2480.0 1450.0 0.51 520.0 -108.0 -0.08 0.3057 0.5863 3121114 ChemDiv3_007895 COc1cccc(/C=C/2\CN(C)C/C(=C\c3cccc(OC)c3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G20 compound treatment 1520.0 491.0 0.17 920.0 293.0 0.22 0.282 0.9921 3121115 ChemDiv3_007896 CC(C)CC(NC(=O)C1CCC(C)CC1)C(=O)Nc2ccc(Br)c(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G21 compound treatment 720.0 -309.0 -0.11 840.0 213.0 0.16 0.0379 0.1929 3028500 ChemDiv3_007897 Cc1ccccc1/C=C/2\Cc3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G22 compound treatment 560.0 -469.0 -0.17 880.0 253.0 0.19 0.0195 0.0763 3121116 ChemDiv3_007898 CC(C)C(NC(=O)c1ccc(cc1)C2(CC3CC4CC(C3)C2)C4)C(=O)Nc5cccc(C)n5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G23 mock treatment 920.0 -109.0 -0.04 680.0 52.5 0.04 0.0012 0.0219 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 G24 mock treatment 2200.0 1170.0 0.42 720.0 92.5 0.07 0.344 0.8161 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H01 compound treatment 8240.0 7210.0 2.56 600.0 -27.5 -0.02 1.794 0.7012 3121117 ChemDiv3_007899 COc1cc(NC(=O)C2CCCN2C(=O)C3CCC(C)CC3)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H02 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3028537 ChemDiv3_007900 CC(C)n1c(CNC(=O)c2ccccc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H03 compound treatment 640.0 -389.0 -0.14 480.0 -148.0 -0.11 -0.1776 -0.9952 3121299 ChemDiv3_007901 CCOC(=O)N1CCC(CC1)NC(=O)C2CCCCN2S(=O)(=O)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H04 compound treatment 480.0 -549.0 -0.19 360.0 -268.0 -0.21 -0.2829 -0.9996 3121300 ChemDiv3_007902 CCCn1c(CCCNC(=O)c2ccc(OC)c(OC)c2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H05 compound treatment 440.0 -589.0 -0.21 400.0 -228.0 -0.17 -0.2712 -0.996 3028538 ChemDiv3_007903 Cc1ccc(cc1)c2[nH]c3ccccc3c2SCCNC(=O)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H06 compound treatment 680.0 -349.0 -0.12 360.0 -268.0 -0.21 -0.2327 -0.9706 3121301 ChemDiv3_007904 CCOC(=O)c1[nH]c2ccccc2c1NC(=O)c3ccc(cc3)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H07 compound treatment 7040.0 6010.0 2.13 760.0 133.0 0.1 1.5798 0.74 3028539 ChemDiv3_007905 CCc1ccc(cc1)C2NC(=O)NC3=C2C(=O)CCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H08 compound treatment 1360.0 331.0 0.12 920.0 293.0 0.22 0.2419 0.9544 3121302 ChemDiv3_007906 N(c1c(nc2ccccn12)c3ccco3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H09 compound treatment 720.0 -309.0 -0.11 400.0 -228.0 -0.17 -0.2009 -0.9747 3028540 ChemDiv3_007907 FC(F)(F)c1nc(NCCc2ccccc2)nc3CCCCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H10 compound treatment 680.0 -349.0 -0.12 440.0 -188.0 -0.14 -0.1893 -0.9972 3121303 ChemDiv3_007908 O=C(Nc1ccc(cc1)C(=O)NCC2COc3ccccc3O2)C4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H11 compound treatment 280.0 -749.0 -0.27 520.0 -108.0 -0.08 -0.2462 -0.8851 1521576 ChemDiv3_007909 Clc1ccc(s1)c2cc(C(=O)NCC3CCCO3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H12 compound treatment 440.0 -589.0 -0.21 400.0 -228.0 -0.17 -0.2712 -0.996 3028541 ChemDiv3_007910 Cc1ccc(NS(=O)(=O)c2ccc3[nH]c(=O)sc3c2)cc1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H13 compound treatment 1800.0 771.0 0.27 920.0 293.0 0.22 0.3522 0.9952 3121304 ChemDiv3_007911 CCc1ccc(NC(=O)CNC(=O)Cn2ccc3ccccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H14 compound treatment 2480.0 1450.0 0.51 480.0 -148.0 -0.11 0.284 0.5387 3028542 ChemDiv3_007912 Cc1ccn2c(NC(=O)C(C)(C)Oc3ccc(Cl)cc3)c(nc2c1)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H15 compound treatment 560.0 -469.0 -0.17 800.0 173.0 0.13 -0.0239 -0.1126 3121305 ChemDiv3_007913 CCCCN(CC)C(=O)c1cn(CC)c(=O)c2cc(OC)c(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H16 compound treatment 320.0 -709.0 -0.25 360.0 -268.0 -0.21 -0.323 -0.995 3121306 ChemDiv3_007914 CCOC(=O)c1c(NC(=O)CS(=O)(=O)c2cn(CC)c3ccccc23)sc4CCCCc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H17 compound treatment 1600.0 571.0 0.2 520.0 -108.0 -0.08 0.0849 0.3882 3028543 ChemDiv3_007915 CC(C)c1ccc(Nc2c(nc3cnccn23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H18 compound treatment 600.0 -429.0 -0.15 800.0 173.0 0.13 -0.0139 -0.069 3121307 ChemDiv3_007916 COCCn1c(=O)[nH]c2cc(ccc2c1=O)C(=O)N3CCN(Cc4ccc5OCOc5c4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H19 compound treatment 520.0 -509.0 -0.18 480.0 -148.0 -0.11 -0.2077 -0.9748 3028544 ChemDiv3_007917 CCc1cccc(C)c1Nc2c(nc3cnccn23)c4ccsc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H20 compound treatment 600.0 -429.0 -0.15 680.0 52.5 0.04 -0.079 -0.5024 3121308 ChemDiv3_007918 CCOc1ccccc1C2NC(=S)NC(c3ccccc3OCC)C24C(=O)NC(=O)NC4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H21 compound treatment 560.0 -469.0 -0.17 360.0 -268.0 -0.21 -0.2628 -0.9945 3028545 ChemDiv3_007919 O=C(CCCCn1c(=O)[nH]c2ccsc2c1=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H22 compound treatment 600.0 -429.0 -0.15 440.0 -188.0 -0.14 -0.2093 -0.9996 3121309 ChemDiv3_007920 CCc1ccccc1N(C)C(=O)Cc2c([nH]c3ccccc23)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H23 mock treatment 560.0 -469.0 -0.17 720.0 92.5 0.07 -0.0674 -0.3726 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 H24 mock treatment 640.0 -389.0 -0.14 920.0 293.0 0.22 0.0613 0.2325 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I01 compound treatment 520.0 -509.0 -0.18 280.0 -348.0 -0.27 -0.3163 -0.9819 3121310 ChemDiv3_007921 COc1ccc(cc1)c2cc(nc(NCC3CCCO3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I02 compound treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 3028546 ChemDiv3_007922 COc1ccccc1/C=C/2\CC/C(=C\c3ccccc3OC)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I03 compound treatment 280.0 -749.0 -0.27 360.0 -268.0 -0.21 -0.333 -0.9919 3121311 ChemDiv3_007923 COc1ccc2nc(NC(=O)CNS(=O)(=O)c3cccs3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I04 compound treatment 400.0 -629.0 -0.22 240.0 -388.0 -0.3 -0.3681 -0.9899 3028547 ChemDiv3_007924 COc1cccc(/C=C/2\CCC(C3CCCC3)C2=O)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I05 compound treatment 320.0 -709.0 -0.25 400.0 -228.0 -0.17 -0.3013 -0.9842 3121312 ChemDiv3_007925 CN(C1CCCCC1)S(=O)(=O)c2cc(Br)cc3CCN(C(=O)C4CC4)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I06 compound treatment 280.0 -749.0 -0.27 640.0 12.5 0.01 -0.181 -0.6811 3121313 ChemDiv3_007926 CC(C)Cc1nn(cc1/C=C/2\Cc3ccccc3C2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I07 compound treatment 1040.0 11.3 0.0 360.0 -268.0 -0.21 -0.1424 -0.6932 3028548 ChemDiv3_007927 COc1ccccc1Nc2ncc(C(=O)NCCCN3CCC(C)CC3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I08 compound treatment 360.0 -669.0 -0.24 320.0 -308.0 -0.24 -0.3347 -1.0 3121314 ChemDiv3_007928 O=C/1/C(=C/c2ccco2)/CC(C\C1=C/c3ccco3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I09 compound treatment 440.0 -589.0 -0.21 560.0 -67.5 -0.05 -0.1843 -0.8566 3028549 ChemDiv3_007929 CCSc1nc2CCSc2c(=O)n1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I10 compound treatment 440.0 -589.0 -0.21 480.0 -148.0 -0.11 -0.2278 -0.9586 3121315 ChemDiv3_007930 CC(C)(C)C1C/C(=C\c2ccccn2)/C(=O)\C(=C/c3ccccn3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I11 compound treatment 5840.0 4810.0 1.71 1040.0 413.0 0.32 1.4308 0.8242 1726170 ChemDiv3_007931 O=C(CSc1nc2c3ccccc3[nH]c2c(=O)n1c4ccccc4)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I12 compound treatment 320.0 -709.0 -0.25 960.0 333.0 0.26 0.0027 0.0076 3028550 ChemDiv3_007932 CCN(CC)c1ccc(/C=C/2\CCc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I13 compound treatment 400.0 -629.0 -0.22 2800.0 2170.0 1.67 1.0216 0.6071 1390633 ChemDiv3_007933 CCOC(=O)C(C)Sc1nc2c3ccccc3[nH]c2c(=O)n1c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I14 compound treatment 440.0 -589.0 -0.21 520.0 -108.0 -0.08 -0.206 -0.9175 3028551 ChemDiv3_007934 CC(C)/C=C/1\CC/C(=C\c2ccc(cc2)C(F)(F)F)/C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I15 compound treatment 440.0 -589.0 -0.21 280.0 -348.0 -0.27 -0.3363 -0.9927 3121316 ChemDiv3_007935 Cn1c(CSC2=NCCN2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I16 compound treatment 520.0 -509.0 -0.18 320.0 -308.0 -0.24 -0.2945 -0.9912 3028552 ChemDiv3_007936 CCN(CC)C(=O)c1oc2ccc(cc2c1C)S(=O)(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I17 compound treatment 360.0 -669.0 -0.24 360.0 -268.0 -0.21 -0.313 -0.9974 1495115 ChemDiv3_007937 COc1ccc(cc1)C2NC(C(C)C(=O)C2C)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I18 compound treatment 320.0 -709.0 -0.25 480.0 -148.0 -0.11 -0.2579 -0.9351 3121317 ChemDiv3_007938 CCN(CC)C(=O)c1cn(C)c(=O)c2cc(OC)c(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I19 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3028587 ChemDiv3_007939 O=C/1/C(=C\c2ccsc2)/CC\C1=C\c3ccsc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I20 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3121318 ChemDiv3_007940 CC(C)CC(NC(=O)C1CCCCC1)C(=O)NC2CCC(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I21 compound treatment 200.0 -829.0 -0.29 280.0 -348.0 -0.27 -0.3965 -0.9988 3028588 ChemDiv3_007941 Fc1ccccc1/C=C/2\Cc3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I22 compound treatment 240.0 -789.0 -0.28 280.0 -348.0 -0.27 -0.3865 -0.9997 3121319 ChemDiv3_007942 CC(C)C(NC(=O)C1CCC(C)CC1)C(=O)N2CCC3(CC2)OCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I23 mock treatment 360.0 -669.0 -0.24 320.0 -308.0 -0.24 -0.3347 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 I24 mock treatment 3280.0 2250.0 0.8 440.0 -188.0 -0.14 0.4629 0.5705 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J01 compound treatment 200.0 -829.0 -0.29 280.0 -348.0 -0.27 -0.3965 -0.9988 3121320 ChemDiv3_007943 CCc1cccc(NC(=O)C(Cc2ccccc2)NC(=O)C3CCC(C)CC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J02 compound treatment 280.0 -749.0 -0.27 640.0 12.5 0.01 -0.181 -0.6811 3028589 ChemDiv3_007944 CCCn1c(nc2ccccc12)C(C)NC(=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J03 compound treatment 360.0 -669.0 -0.24 240.0 -388.0 -0.3 -0.3781 -0.9937 3121696 ChemDiv3_007945 COc1ccc(cc1)c2[nH]c3ccccc3c2SCCNC(=O)c4ccc(OC)c(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J04 compound treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 3028590 ChemDiv3_007946 CC(=C)Cn1c(CCCNC(=O)c2ccc(F)cc2)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J05 compound treatment 3480.0 2450.0 0.87 360.0 -268.0 -0.21 0.4697 0.5257 3121494 ChemDiv3_007947 Cc1[nH]c2ccccc2c1SCCNC(=O)/C=C/c3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J06 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3028591 ChemDiv3_007948 Fc1ccc(NC(=O)CSc2oc(nc2S(=O)(=O)c3ccccc3)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J07 compound treatment 280.0 -749.0 -0.27 400.0 -228.0 -0.17 -0.3113 -0.9793 3121495 ChemDiv3_007949 O=C1CCCC2=C1C(NC(=S)N2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J08 compound treatment 400.0 -629.0 -0.22 320.0 -308.0 -0.24 -0.3246 -0.9996 3121496 ChemDiv3_007950 Fc1ccc(Nc2c(nc3ccccn23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J09 compound treatment 280.0 -749.0 -0.27 240.0 -388.0 -0.3 -0.3982 -0.9984 3028592 ChemDiv3_007951 COc1ccc(CCNc2nc(c3CC(C)CCc3n2)C(F)(F)F)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J10 compound treatment 400.0 -629.0 -0.22 360.0 -268.0 -0.21 -0.3029 -0.9991 3121497 ChemDiv3_007952 COc1ccc(cc1)N2CCN(CCNC(=O)c3ccc(NC(=O)C4CCCO4)cc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J11 compound treatment 360.0 -669.0 -0.24 400.0 -228.0 -0.17 -0.2913 -0.9887 3121498 ChemDiv3_007953 CC1CCCCC1NC(=O)c2cc(nc3ccccc23)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J12 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3028593 ChemDiv3_007954 O=C(Cn1c(=O)sc2ccccc12)NCc3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J13 compound treatment 1080.0 51.3 0.02 280.0 -348.0 -0.27 -0.1758 -0.6574 3121499 ChemDiv3_007955 CCn1cc(C(=O)NCCC2=CCCCC2)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J14 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 3028594 ChemDiv3_007956 Cc1ccn2c(NC(=O)c3ccc(C)c(C)c3)c(nc2c1)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J15 compound treatment 320.0 -709.0 -0.25 360.0 -268.0 -0.21 -0.323 -0.995 3121500 ChemDiv3_007957 CCn1cc(C(=O)N2CCCCC2)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J16 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3028595 ChemDiv3_007958 CCCn1cc(c2ccccc12)S(=O)(=O)CC(=O)Nc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J17 compound treatment 480.0 -549.0 -0.19 360.0 -268.0 -0.21 -0.2829 -0.9996 3121501 ChemDiv3_007959 Clc1ccc(cc1)c2nc3cnccn3c2NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J18 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 3121502 ChemDiv3_007960 COc1ccc(Cn2c(=O)[nH]c3cc(ccc3c2=O)C(=O)NC4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J19 compound treatment 280.0 -749.0 -0.27 560.0 -67.5 -0.05 -0.2245 -0.8294 3028596 ChemDiv3_007961 NC(=O)C[n+]1ccn2c(NC3CCCCC3)c(nc2c1)c4ccc(cc4)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J20 compound treatment 440.0 -589.0 -0.21 840.0 213.0 0.16 -0.0323 -0.122 3121503 ChemDiv3_007962 Clc1ccc(cc1)C2NC(=S)NC(c3ccc(Cl)cc3)C24C(=O)NC(=O)NC4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J21 compound treatment 360.0 -669.0 -0.24 640.0 12.5 0.01 -0.161 -0.6779 3121504 ChemDiv3_007963 O=C(CCCCn1c(=O)[nH]c2ccsc2c1=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J22 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3028597 ChemDiv3_007964 COc1ccc(cc1)N(C)C(=O)Cc2c([nH]c3ccccc23)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J23 mock treatment 240.0 -789.0 -0.28 280.0 -348.0 -0.27 -0.3865 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 J24 mock treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K01 compound treatment 1040.0 11.3 0.0 1040.0 413.0 0.32 0.2268 0.716 3121505 ChemDiv3_007965 COc1ccccc1c2cc(nc(NCc3ccco3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K02 compound treatment 320.0 -709.0 -0.25 560.0 -67.5 -0.05 -0.2144 -0.8353 3028598 ChemDiv3_007966 Cn1cccc1/C=C/2\CC/C(=C\c3cccn3C)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K03 compound treatment 6520.0 5490.0 1.95 320.0 -308.0 -0.24 1.2105 0.6169 3121506 ChemDiv3_007967 O=C(CNS(=O)(=O)c1cccs1)N2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K04 compound treatment 520.0 -509.0 -0.18 360.0 -268.0 -0.21 -0.2728 -0.9979 3121507 ChemDiv3_007968 CN1CCCc2cc(/C=C/3\CCC(C4CCCC4)C3=O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K05 compound treatment 400.0 -629.0 -0.22 360.0 -268.0 -0.21 -0.3029 -0.9991 3028599 ChemDiv3_007969 CCc1cccc(NS(=O)(=O)c2cc(Br)cc3CCN(C(=O)C4CC4)c32)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K06 compound treatment 400.0 -629.0 -0.22 240.0 -388.0 -0.3 -0.3681 -0.9899 3121508 ChemDiv3_007970 CCn1c2ccccc2c3cc(/C=C/4\CCC(C5CCCC5)C4=O)ccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K07 compound treatment 360.0 -669.0 -0.24 480.0 -148.0 -0.11 -0.2478 -0.9427 3028600 ChemDiv3_007971 COc1ccccc1Nc2ncc(C(=O)N(C)c3ccc(Cl)cc3)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K08 compound treatment 720.0 -309.0 -0.11 520.0 -108.0 -0.08 -0.1358 -0.9903 3121509 ChemDiv3_007972 COc1ccc(OC)c(/C=C/2\CC(C/C(=C\c3cc(OC)ccc3OC)/C2=O)c4ccccc4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K09 compound treatment 360.0 -669.0 -0.24 680.0 52.5 0.04 -0.1393 -0.5787 3121510 ChemDiv3_007973 CCOc1ccc(cc1)n2c(SCC(=O)NCc3ccco3)nc4CCSc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K10 compound treatment 480.0 -549.0 -0.19 360.0 -268.0 -0.21 -0.2829 -0.9996 3028601 ChemDiv3_007974 CCC1C/C(=C\c2sccc2C)/C(=O)\C(=C\c3sccc3C)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K11 compound treatment 520.0 -509.0 -0.18 360.0 -268.0 -0.21 -0.2728 -0.9979 1415020 ChemDiv3_007975 CCC(C)Sc1nc2c3ccccc3[nH]c2c(=O)n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K12 compound treatment 2040.0 1010.0 0.36 480.0 -148.0 -0.11 0.1736 0.4615 3028602 ChemDiv3_007976 Brc1csc(/C=C/2\CCC(C3CCCC3)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K13 compound treatment 400.0 -629.0 -0.22 840.0 213.0 0.16 -0.0424 -0.1533 3121511 ChemDiv3_007977 CSC1=NSC2=NC(=O)/C(=C\c3cccs3)/C(=N)N12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K14 compound treatment 920.0 -109.0 -0.04 480.0 -148.0 -0.11 -0.1074 -0.8974 3027776 ChemDiv3_007978 CC1CCN(CC1)S(=O)(=O)c2ccc3oc(C(=O)NCCc4ccc(Cl)cc4)c(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K15 compound treatment 480.0 -549.0 -0.19 320.0 -308.0 -0.24 -0.3046 -0.9954 3121512 ChemDiv3_007979 Clc1ccccc1Cn2c(CSC3=NCCN3)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K16 compound treatment 680.0 -349.0 -0.12 400.0 -228.0 -0.17 -0.211 -0.9857 3121513 ChemDiv3_007980 Cc1c(oc2ccc(cc12)S(=O)(=O)N3CCCC3)C(=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K17 compound treatment 440.0 -589.0 -0.21 480.0 -148.0 -0.11 -0.2278 -0.9586 3027777 ChemDiv3_007981 O=C/1/C(=C/c2ccco2)/CN(Cc3ccccc3)C\C1=C/c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K18 compound treatment 5280.0 4250.0 1.51 400.0 -228.0 -0.17 0.9429 0.6211 3121514 ChemDiv3_007982 CC1CCC(CC1)C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)NCc4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K19 compound treatment 1440.0 411.0 0.15 560.0 -67.5 -0.05 0.0665 0.4296 3027778 ChemDiv3_007983 O=C/1/C(=C/c2ccc3nccnc3c2)/CCC\C1=C/c4ccc5nccnc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K20 compound treatment 3640.0 2610.0 0.93 240.0 -388.0 -0.3 0.4447 0.457 3121515 ChemDiv3_007984 CC(C)CC(NC(=O)C1CCCCC1)C(=O)N2CCN(CC2)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K21 compound treatment 520.0 -509.0 -0.18 400.0 -228.0 -0.17 -0.2511 -0.9999 3027779 ChemDiv3_007985 CCc1ccc(/C=C/2\Cc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K22 compound treatment 520.0 -509.0 -0.18 400.0 -228.0 -0.17 -0.2511 -0.9999 3121516 ChemDiv3_007986 CC(C)C(NC(=O)c1ccc(cc1)C2(CC3CC4CC(C3)C2)C4)C(=O)N(C)Cc5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K23 mock treatment 2480.0 1450.0 0.51 920.0 293.0 0.22 0.5228 0.9308 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 K24 mock treatment 680.0 -349.0 -0.12 1200.0 573.0 0.44 0.2233 0.4891 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L01 compound treatment 840.0 -189.0 -0.07 480.0 -148.0 -0.11 -0.1274 -0.9686 3027780 ChemDiv3_007987 Fc1ccc(cc1)S(=O)(=O)N2CCCCC2C(=O)N3CCN(CC3)c4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L02 compound treatment 360.0 -669.0 -0.24 320.0 -308.0 -0.24 -0.3347 -1.0 3121517 ChemDiv3_007988 COCC(=O)NC(C)c1nc2ccccc2n1Cc3cc(C)ccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L03 compound treatment 400.0 -629.0 -0.22 360.0 -268.0 -0.21 -0.3029 -0.9991 3121518 ChemDiv3_007989 Brc1ccc(cc1)c2[nH]c3ccccc3c2SCCNC(=O)c4ccncc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L04 compound treatment 320.0 -709.0 -0.25 400.0 -228.0 -0.17 -0.3013 -0.9842 3027781 ChemDiv3_007990 COc1ccccc1C(=O)NCCCc2nc3ccccc3n2CC(=C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L05 compound treatment 480.0 -549.0 -0.19 360.0 -268.0 -0.21 -0.2829 -0.9996 3121519 ChemDiv3_007991 COc1cccc(C(=O)NCCSc2c[nH]c3ccccc23)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L06 compound treatment 440.0 -589.0 -0.21 320.0 -308.0 -0.24 -0.3146 -0.9981 3121697 ChemDiv3_007992 CCOc1ccc(NC(=O)CSc2oc(nc2S(=O)(=O)c3ccccc3)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L07 compound treatment 880.0 -149.0 -0.05 320.0 -308.0 -0.24 -0.2042 -0.8443 3027782 ChemDiv3_007993 CCc1ccc(cc1)C2NC(=O)NC3=C2C(=O)CC(C)(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L08 compound treatment 480.0 -549.0 -0.19 480.0 -148.0 -0.11 -0.2177 -0.9668 3121698 ChemDiv3_007994 C1CN(CCO1)c2ccc(cc2)c3nc4ccccn4c3Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L09 compound treatment 360.0 -669.0 -0.24 480.0 -148.0 -0.11 -0.2478 -0.9427 3027783 ChemDiv3_007995 CC1CCc2nc(nc(c2C1)C(F)(F)F)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L10 compound treatment 480.0 -549.0 -0.19 400.0 -228.0 -0.17 -0.2612 -0.9985 3121699 ChemDiv3_007996 CCC(=O)N1CCc2cc(Br)cc(c12)S(=O)(=O)CCC(=O)NCC3CCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L11 compound treatment 480.0 -549.0 -0.19 760.0 133.0 0.1 -0.0657 -0.2992 3027784 ChemDiv3_007997 CCN(CC)S(=O)(=O)c1ccc(NC(=O)c2cc(nc3ccccc23)c4cccs4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L12 compound treatment 1040.0 11.3 0.0 480.0 -148.0 -0.11 -0.0772 -0.6818 3121700 ChemDiv3_007998 COc1ccc(CC(=O)Nc2c(nc3ccccn23)c4ccc(F)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L13 compound treatment 520.0 -509.0 -0.18 440.0 -188.0 -0.14 -0.2294 -0.9937 3121701 ChemDiv3_007999 CCn1cc(C(=O)Nc2cccc(OC)c2)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L14 compound treatment 1080.0 51.3 0.02 440.0 -188.0 -0.14 -0.0889 -0.6129 3027785 ChemDiv3_008000 CCC(CC)C(=O)Nc1c(nc2cc(C)ccn12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L15 compound treatment 560.0 -469.0 -0.17 320.0 -308.0 -0.24 -0.2845 -0.9853 3121702 ChemDiv3_008001 COc1cc2c(cn(CC(C)C)c(=O)c2cc1OC)C(=O)Nc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L16 compound treatment 480.0 -549.0 -0.19 400.0 -228.0 -0.17 -0.2612 -0.9985 3027786 ChemDiv3_008002 Fc1cccc(Cn2cc(c3ccccc23)S(=O)(=O)CC(=O)NC4CCCCC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L17 compound treatment 680.0 -349.0 -0.12 360.0 -268.0 -0.21 -0.2327 -0.9706 3121703 ChemDiv3_008003 Cc1ccc(o1)c2nc3cnccn3c2NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L18 compound treatment 520.0 -509.0 -0.18 480.0 -148.0 -0.11 -0.2077 -0.9748 3121704 ChemDiv3_008004 COc1ccc(Cn2c(=O)[nH]c3cc(ccc3c2=O)C(=O)NCc4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L19 compound treatment 720.0 -309.0 -0.11 360.0 -268.0 -0.21 -0.2227 -0.9567 3027787 ChemDiv3_008005 COc1ccc(Cl)cc1N2C(=O)C3C(NN(C3C2=O)C(=O)c4ccc(C)cc4)c5ccccc5F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L20 compound treatment 680.0 -349.0 -0.12 320.0 -308.0 -0.24 -0.2544 -0.9545 3121705 ChemDiv3_008006 O=C(Cn1ccc2ccccc2c1=O)NCCC(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L21 compound treatment 480.0 -549.0 -0.19 1920.0 1290.0 0.99 0.564 0.5578 3121706 ChemDiv3_008007 CC1CCCCC1NC(=O)CCCn2c(=O)[nH]c3ccsc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L22 compound treatment 1040.0 11.3 0.0 880.0 253.0 0.19 0.1399 0.7215 3027788 ChemDiv3_008008 CNC(=S)N(CCc1c(C)[nH]c2ccccc12)Cc3cc(OC)c(OC)c(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L23 mock treatment 480.0 -549.0 -0.19 400.0 -228.0 -0.17 -0.2612 -0.9985 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 L24 mock treatment 1920.0 891.0 0.32 720.0 92.5 0.07 0.2738 0.8449 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M01 compound treatment 1520.0 491.0 0.17 1000.0 373.0 0.29 0.3254 0.9718 3121707 ChemDiv3_008009 COc1ccc(cc1OC)c2cc(nc(n2)N3CCc4ccccc4C3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M02 compound treatment 440.0 -589.0 -0.21 400.0 -228.0 -0.17 -0.2712 -0.996 3121708 ChemDiv3_008010 CSc1ccc(/C=C/2\CC/C(=C\c3ccc(SC)cc3)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M03 compound treatment 2160.0 1130.0 0.4 560.0 -67.5 -0.05 0.2471 0.6107 3027789 ChemDiv3_008011 CCC1CCCCN1S(=O)(=O)c2cc(Br)cc3CCN(C(=O)CC)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M04 compound treatment 640.0 -389.0 -0.14 160.0 -468.0 -0.36 -0.3513 -0.9137 3121709 ChemDiv3_008012 CCc1ccc(/C=C/2\CCc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M05 compound treatment 760.0 -269.0 -0.1 400.0 -228.0 -0.17 -0.1909 -0.9595 3027790 ChemDiv3_008013 Clc1ccccc1CCNS(=O)(=O)c2cc(Br)cc3CCN(C(=O)C4CC4)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M06 compound treatment 1760.0 731.0 0.26 840.0 213.0 0.16 0.2988 0.975 3121710 ChemDiv3_008014 CC(C)Cc1nn(cc1/C=C/2\CCC(C3CCCC3)C2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M07 compound treatment 880.0 -149.0 -0.05 640.0 12.5 0.01 -0.0305 -0.5692 3121711 ChemDiv3_008015 COc1cc(cc(OC)c1OC)C(=O)Nc2ccc3nc(cc(C)c3c2)N4CCN(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M08 compound treatment 1080.0 51.3 0.02 760.0 133.0 0.1 0.0848 0.8205 3027791 ChemDiv3_008016 CC(C)(C)C1C/C(=C\c2ccco2)/C(=O)\C(=C/c3ccco3)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M09 compound treatment 640.0 -389.0 -0.14 600.0 -27.5 -0.02 -0.1124 -0.806 3121712 ChemDiv3_008017 CCOC(=O)C(C)(C)Sc1nc2CCSc2c(=O)n1c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M10 compound treatment 9280.0 8250.0 2.93 720.0 92.5 0.07 2.12 0.724 3121713 ChemDiv3_008018 COc1ccc(/C=C/2\CC/C(=C\c3ccc(OC)c(Cn4cccn4)c3)/C2=O)cc1Cn5cccn5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M11 compound treatment 1000.0 -28.8 -0.01 760.0 133.0 0.1 0.0647 0.633 1638612 ChemDiv3_008019 Cc1ccc(cc1)n2c(SCC(=O)N3CCCCC3)nc4c5ccccc5[nH]c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M12 compound treatment 840.0 -189.0 -0.07 600.0 -27.5 -0.02 -0.0623 -0.887 3027839 ChemDiv3_008020 Brc1csc(/C=C/2\CCC/C(=C\c3cc(Br)cs3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M13 compound treatment 6000.0 4970.0 1.76 3160.0 2530.0 1.94 2.6218 0.9988 3121714 ChemDiv3_008021 CCSC1=NSC2=NC(=O)/C(=C\c3ccc(OC(=O)c4ccco4)c(Cl)c3)/C(=N)N12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M14 compound treatment 400.0 -629.0 -0.22 600.0 -27.5 -0.02 -0.1726 -0.7706 3027840 ChemDiv3_008022 CN(C1CCCCC1)S(=O)(=O)c2ccc3oc(C(=O)NCc4ccccc4)c(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M15 compound treatment 520.0 -509.0 -0.18 600.0 -27.5 -0.02 -0.1425 -0.7845 3121715 ChemDiv3_008023 CCOc1ccc(cc1)N2C(=O)C(CC(=O)Nc3ccccc3)N(CCN4CCN(C)CC4)C2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M16 compound treatment 680.0 -349.0 -0.12 560.0 -67.5 -0.05 -0.1241 -0.9254 3027841 ChemDiv3_008024 CC(C)NC(=O)c1oc2ccc(cc2c1C)S(=O)(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M17 compound treatment 640.0 -389.0 -0.14 440.0 -188.0 -0.14 -0.1993 -0.9998 3121716 ChemDiv3_008025 Clc1cccc(/C=C/2\CC/C(=C\c3cccc(Cl)c3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M18 compound treatment 480.0 -549.0 -0.19 640.0 12.5 0.01 -0.1309 -0.6714 3121717 ChemDiv3_008026 CC1CCC(CC1)C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)NC4CCCCC4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M19 compound treatment 840.0 -189.0 -0.07 840.0 213.0 0.16 0.068 0.3857 3027842 ChemDiv3_008027 CCOc1ccc(/C=C/2\CC/C(=C\c3ccc(OCC)cc3)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M20 compound treatment 400.0 -629.0 -0.22 600.0 -27.5 -0.02 -0.1726 -0.7706 3121718 ChemDiv3_008028 CCc1cccc(NC(=O)C(CC(C)C)NC(=O)C2CCCCC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M21 compound treatment 640.0 -389.0 -0.14 480.0 -148.0 -0.11 -0.1776 -0.9952 3027843 ChemDiv3_008029 O=C1/C(=C/c2ccsc2)/Cc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M22 compound treatment 2760.0 1730.0 0.61 600.0 -27.5 -0.02 0.4193 0.6824 3121719 ChemDiv3_008030 COc1ccc(cc1OC)S(=O)(=O)N2CCCCC2C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M23 mock treatment 1480.0 451.0 0.16 680.0 52.5 0.04 0.1417 0.8584 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 M24 mock treatment 6640.0 5610.0 1.99 960.0 333.0 0.26 1.588 0.7913 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N01 compound treatment 3280.0 2250.0 0.8 480.0 -148.0 -0.11 0.4846 0.6008 3027844 ChemDiv3_008031 COc1ccc(NC(=O)C2CCCCN2S(=O)(=O)c3ccc(cc3)C(C)(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N02 compound treatment 840.0 -189.0 -0.07 480.0 -148.0 -0.11 -0.1274 -0.9686 3121720 ChemDiv3_008032 CCC(=O)NC(C)c1nc2ccccc2n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N03 compound treatment 480.0 -549.0 -0.19 680.0 52.5 0.04 -0.1092 -0.5491 3121721 ChemDiv3_008033 COc1ccc(CC(=O)NCCSc2c([nH]c3ccccc23)c4ccccc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N04 compound treatment 5520.0 4490.0 1.59 560.0 -67.5 -0.05 1.09 0.6837 3027845 ChemDiv3_008034 COc1ccccc1C(=O)NCCCc2nc3ccccc3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N05 compound treatment 960.0 -68.8 -0.02 400.0 -228.0 -0.17 -0.1407 -0.7981 3121722 ChemDiv3_008035 CCC(=O)NCCSc1c[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N06 compound treatment 640.0 -389.0 -0.14 1640.0 1010.0 0.78 0.4521 0.5727 3122110 ChemDiv3_008036 Clc1ccc(cc1)S(=O)(=O)c2nc(oc2SCC(=O)NCC3CCCO3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N07 compound treatment 640.0 -389.0 -0.14 2280.0 1650.0 1.27 0.7996 0.6266 3027846 ChemDiv3_008037 Nc1n[nH]c2nc(nc(c3ccccc3)c12)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N08 compound treatment 600.0 -429.0 -0.15 680.0 52.5 0.04 -0.079 -0.5024 3121904 ChemDiv3_008038 CCCNC(=O)CSc1nc2nc(C)c(Cc3cccc(C)c3)c(C)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N09 compound treatment 560.0 -469.0 -0.17 2680.0 2050.0 1.58 0.9966 0.629 3027847 ChemDiv3_008039 Brc1ccc(NC(=O)C(Cc2ccccc2)NS(=O)(=O)c3cccs3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N10 compound treatment 2800.0 1770.0 0.63 680.0 52.5 0.04 0.4728 0.7509 3121905 ChemDiv3_008040 Clc1ccc(cc1)n2cc(nc2S(=O)(=O)CC(=O)Nc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N11 compound treatment 680.0 -349.0 -0.12 1800.0 1170.0 0.9 0.549 0.6042 3121906 ChemDiv3_008041 O=C(Nc1ccc(cc1)S(=O)(=O)N2CCCCC2)c3cc(nc4ccccc34)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N12 compound treatment 5680.0 4650.0 1.65 520.0 -108.0 -0.08 1.1084 0.6709 3027848 ChemDiv3_008042 Fc1ccc(cc1)c2nc3ccccn3c2NC(=O)COc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N13 compound treatment 880.0 -149.0 -0.05 1240.0 613.0 0.47 0.2952 0.6238 3121907 ChemDiv3_008043 CCC(C)NC(=O)c1cn(CC)c(=O)c2cc(OC)c(OC)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N14 compound treatment 800.0 -229.0 -0.08 720.0 92.5 0.07 -0.0072 -0.0665 3027849 ChemDiv3_008044 CCC(C(=O)Nc1c(nc2cc(C)ccn12)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N15 compound treatment 640.0 -389.0 -0.14 960.0 333.0 0.26 0.083 0.286 3121908 ChemDiv3_008045 COc1cc2c(cn(CC(C)C)c(=O)c2cc1OC)C(=O)N3CCN(CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N16 compound treatment 600.0 -429.0 -0.15 640.0 12.5 0.01 -0.1008 -0.6612 3121909 ChemDiv3_008046 Cc1ccccc1Cn2cc(c3ccccc23)S(=O)(=O)CC(=O)Nc4ccc5OCCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N17 compound treatment 800.0 -229.0 -0.08 640.0 12.5 0.01 -0.0506 -0.6192 3027850 ChemDiv3_008047 Cc1ccccc1Nc2c(nc3c[n+](CC(=O)N)ccn23)c4ccsc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N18 compound treatment 600.0 -429.0 -0.15 800.0 173.0 0.13 -0.0139 -0.069 3121910 ChemDiv3_008048 CCC(C)NC(=O)c1ccc2c(=O)n(Cc3ccc(OC)cc3)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N19 compound treatment 640.0 -389.0 -0.14 560.0 -67.5 -0.05 -0.1342 -0.9106 3027851 ChemDiv3_008049 Cc1cccc(N2CCN(CC2)C(=O)Cc3ccc(cc3)n4c(=O)[nH]c5ccsc5c4=O)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N20 compound treatment 1800.0 771.0 0.27 680.0 52.5 0.04 0.222 0.8026 3121911 ChemDiv3_008050 CCc1ccc(NC(=O)CCNC(=O)Cn2ccc3ccccc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N21 compound treatment 2000.0 971.0 0.34 680.0 52.5 0.04 0.2721 0.7845 3121912 ChemDiv3_008051 Cc1ccc(CCNC(=O)C2CCC(Cn3c(=O)[nH]c4ccsc4c3=O)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N22 compound treatment 760.0 -269.0 -0.1 840.0 213.0 0.16 0.0479 0.2537 3027852 ChemDiv3_008052 COc1ccc2[nH]c(C)c(CCN(Cc3cccs3)C(=S)NC4CCCCC4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N23 mock treatment 880.0 -149.0 -0.05 560.0 -67.5 -0.05 -0.074 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 N24 mock treatment 720.0 -309.0 -0.11 320.0 -308.0 -0.24 -0.2444 -0.939 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O01 compound treatment 280.0 -749.0 -0.27 360.0 -268.0 -0.21 -0.333 -0.9919 3121913 ChemDiv3_008053 COc1ccc(cc1OC)c2cc(nc(NC(C)c3ccccc3)n2)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O02 compound treatment 320.0 -709.0 -0.25 240.0 -388.0 -0.3 -0.3881 -0.9965 3027853 ChemDiv3_008054 CC1C/C(=C\c2cccn2C)/C(=O)\C(=C/c3cccn3C)\C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O03 compound treatment 320.0 -709.0 -0.25 400.0 -228.0 -0.17 -0.3013 -0.9842 3121914 ChemDiv3_008055 CCCNS(=O)(=O)c1cc(Br)cc2CCN(C(=O)CC)c21 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O04 compound treatment 360.0 -669.0 -0.24 320.0 -308.0 -0.24 -0.3347 -1.0 3121915 ChemDiv3_008056 COc1cc(/C=C/2\CCc3ccccc3C2=O)ccc1OCCC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O05 compound treatment 240.0 -789.0 -0.28 360.0 -268.0 -0.21 -0.3431 -0.9884 3027854 ChemDiv3_008057 CCN(c1ccc(C)c(C)c1)S(=O)(=O)c2cc(Br)cc3CC(C)N(C(=O)C)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O06 compound treatment 360.0 -669.0 -0.24 200.0 -428.0 -0.33 -0.3998 -0.9873 3121916 ChemDiv3_008058 Cc1cc(/C=C/2\CCC(C3CCCC3)C2=O)c(C)n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O07 compound treatment 560.0 -469.0 -0.17 240.0 -388.0 -0.3 -0.3279 -0.9622 3121917 ChemDiv3_008059 CN1CCN(CC1)c2cc(C)c3cc(NC(=O)C4CCC(CC4)C(C)(C)C)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O08 compound treatment 240.0 -789.0 -0.28 200.0 -428.0 -0.33 -0.4299 -0.9968 3121918 ChemDiv3_008060 COc1cccc(/C=C/2\CC(C/C(=C/c3cccc(OC)c3OC)/C2=O)C(C)(C)C)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O09 compound treatment 360.0 -669.0 -0.24 160.0 -468.0 -0.36 -0.4215 -0.9798 3027902 ChemDiv3_008061 Clc1ccc(cc1)n2c(SCC(=O)Nc3nccs3)nc4CCSc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O10 compound treatment 320.0 -709.0 -0.25 240.0 -388.0 -0.3 -0.3881 -0.9965 3121919 ChemDiv3_008062 Fc1ccc(/C=C/2\CCC/C(=C\c3ccc(F)c(F)c3)/C2=O)cc1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O11 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 1129536 ChemDiv3_008063 CCCSc1nc2c3ccccc3[nH]c2c(=O)n1c4cc(C)cc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O12 compound treatment 480.0 -549.0 -0.19 360.0 -268.0 -0.21 -0.2829 -0.9996 3121920 ChemDiv3_008064 CN1C/2CCC1/C(=C/c3ccccc3)/C(=O)\C2=C\c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O13 compound treatment 240.0 -789.0 -0.28 280.0 -348.0 -0.27 -0.3865 -0.9997 1241030 ChemDiv3_008065 COc1ccc(cc1)C(O)C(Nc2ccccc2)c3nc4ccccc4n3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O14 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3027903 ChemDiv3_008066 CN(C1CCCCC1)S(=O)(=O)c2ccc3oc(C(=O)NC4CCCC4)c(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O15 compound treatment 400.0 -629.0 -0.22 200.0 -428.0 -0.33 -0.3898 -0.9823 3121921 ChemDiv3_008067 CCN1C(=O)C(CC(=O)Nc2ccc(Br)cc2)N(CCNC(=O)C)C1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O16 compound treatment 240.0 -789.0 -0.28 280.0 -348.0 -0.27 -0.3865 -0.9997 3027904 ChemDiv3_008068 CN(Cc1ccccc1)C(=O)C2C(N(C)C(=O)c3ccccc23)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O17 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3121922 ChemDiv3_008069 O=C/1/C(=C/c2cccnc2)/CC\C1=C/c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O18 compound treatment 280.0 -749.0 -0.27 400.0 -228.0 -0.17 -0.3113 -0.9793 3121923 ChemDiv3_008070 CC(C)C(NC(=O)C1CCC(C)CC1)C(=O)NC2CCC(C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O19 compound treatment 240.0 -789.0 -0.28 360.0 -268.0 -0.21 -0.3431 -0.9884 3027905 ChemDiv3_008071 Brc1ccc(/C=C\2/CC\C(=C\c3ccc(Br)o3)\C2=O)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O20 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3121924 ChemDiv3_008072 CC(C)CC(NC(=O)C1CCCCC1)C(=O)NCc2ccccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O21 compound treatment 280.0 -749.0 -0.27 160.0 -468.0 -0.36 -0.4416 -0.989 3027906 ChemDiv3_008073 CN1CCCc2cc(/C=C/3\Cc4ccccc4C3=O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O22 compound treatment 320.0 -709.0 -0.25 240.0 -388.0 -0.3 -0.3881 -0.9965 1198561 ChemDiv3_008074 OC(=O)C1CCCCN1S(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O23 mock treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 O24 mock treatment 440.0 -589.0 -0.21 400.0 -228.0 -0.17 -0.2712 -0.996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P01 compound treatment 200.0 -829.0 -0.29 320.0 -308.0 -0.24 -0.3748 -0.9941 3121925 ChemDiv3_008075 CC(C)C(NC(=O)C1CCC(C)CC1)C(=O)NCc2ccccn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P02 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3027907 ChemDiv3_008076 CCCC(=O)NCCc1nc2ccccc2n1CCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P03 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3121926 ChemDiv3_008077 COc1ccc(cc1)c2[nH]c3ccccc3c2SCCNC(=O)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P04 compound treatment 440.0 -589.0 -0.21 280.0 -348.0 -0.27 -0.3363 -0.9927 3027908 ChemDiv3_008078 Cn1c(nc2ccccc12)C(Cc3ccccc3)NC(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P05 compound treatment 320.0 -709.0 -0.25 360.0 -268.0 -0.21 -0.323 -0.995 3121927 ChemDiv3_008079 Cc1[nH]c2ccccc2c1SCCNC(=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P06 compound treatment 320.0 -709.0 -0.25 400.0 -228.0 -0.17 -0.3013 -0.9842 3121928 ChemDiv3_008080 Cc1ccc(cc1)c2nc(c(SCC(=O)N)o2)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P07 compound treatment 280.0 -749.0 -0.27 320.0 -308.0 -0.24 -0.3547 -0.9983 3027909 ChemDiv3_008081 CC(C)c1ccc(cc1)c2nc(nc3nn4c(C)cc(C)nc4c23)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P08 compound treatment 240.0 -789.0 -0.28 280.0 -348.0 -0.27 -0.3865 -0.9997 3122111 ChemDiv3_008082 CC1CCCC(NC(=O)CSc2nc3nc(C)c(Cc4ccccc4Cl)c(C)n3n2)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P09 compound treatment 1080.0 51.3 0.02 240.0 -388.0 -0.3 -0.1975 -0.6627 3027910 ChemDiv3_008083 CC1CCCN(C1)C(=O)c2ccc(NS(=O)(=O)c3cccs3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P10 compound treatment 240.0 -789.0 -0.28 320.0 -308.0 -0.24 -0.3648 -0.9964 3122112 ChemDiv3_008084 CC(=O)NC1=NN(C(S1)/C=C/c2ccccc2)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P11 compound treatment 200.0 -829.0 -0.29 320.0 -308.0 -0.24 -0.3748 -0.9941 3122113 ChemDiv3_008085 O=C(NCCN1CCCc2ccccc12)c3cc(nc4ccccc34)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P12 compound treatment 560.0 -469.0 -0.17 360.0 -268.0 -0.21 -0.2628 -0.9945 3027911 ChemDiv3_008086 Fc1ccc(cc1)c2nc3ccccn3c2NC(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P13 compound treatment 360.0 -669.0 -0.24 280.0 -348.0 -0.27 -0.3564 -0.9983 3122114 ChemDiv3_008087 CCn1cc(C(=O)N(C)C2CCCCC2)c3cc(OC)c(OC)cc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P14 compound treatment 280.0 -749.0 -0.27 480.0 -148.0 -0.11 -0.2679 -0.9278 3027912 ChemDiv3_008088 COc1ccc(NC(=O)CS(=O)(=O)c2c[nH]c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P15 compound treatment 280.0 -749.0 -0.27 280.0 -348.0 -0.27 -0.3765 -1.0 3122115 ChemDiv3_008089 COc1ccc(CCNC(=O)c2cn(CC(C)C)c(=O)c3cc(OC)c(OC)cc23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P16 compound treatment 320.0 -709.0 -0.25 480.0 -148.0 -0.11 -0.2579 -0.9351 3027913 ChemDiv3_008090 Clc1ccc(Cn2cc(c3ccccc23)S(=O)(=O)CC(=O)N4CCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P17 compound treatment 320.0 -709.0 -0.25 280.0 -348.0 -0.27 -0.3664 -0.9996 3122116 ChemDiv3_008091 COc1ccc(Nc2c(nc3cnccn23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P18 compound treatment 320.0 -709.0 -0.25 320.0 -308.0 -0.24 -0.3447 -0.9995 3122117 ChemDiv3_008092 CCOC(=O)N1CCN(CC1)C(=O)c2ccc3c(=O)n(CCc4ccccc4)c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P19 compound treatment 2160.0 1130.0 0.4 280.0 -348.0 -0.27 0.0951 0.1974 3027914 ChemDiv3_008093 Clc1ccc(CNC(=O)c2ccc(Cn3c(=O)[nH]c4ccsc4c3=O)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P20 compound treatment 1000.0 -28.8 -0.01 960.0 333.0 0.26 0.1733 0.6783 3122118 ChemDiv3_008094 OC(=O)c1[nH]c2ccccc2c1CC(=O)N3CCN(CC3)c4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P21 compound treatment 240.0 -789.0 -0.28 760.0 133.0 0.1 -0.1259 -0.423 3027915 ChemDiv3_008095 Cc1ccc(NC(=O)CCn2c(=O)[nH]c3ccsc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P22 compound treatment 2280.0 1250.0 0.44 280.0 -348.0 -0.27 0.1252 0.2418 3122119 ChemDiv3_008096 COc1ccc2[nH]c(C)c(CCN(Cc3cccs3)C(=S)Nc4cccc(C)c4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P23 mock treatment 320.0 -709.0 -0.25 640.0 12.5 0.01 -0.171 -0.6796 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2023 P24 mock treatment 360.0 -669.0 -0.24 240.0 -388.0 -0.3 -0.3781 -0.9937 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A01 compound treatment 400.0 -538.0 -0.19 640.0 47.5 0.04 -0.109 -0.5617 3122120 ChemDiv3_008097 CCNC(=S)N1CCc2cc(OC)c(OC)cc2C1COc3ccc4c(C)cc(=O)oc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A02 compound treatment 320.0 -618.0 -0.22 880.0 288.0 0.22 0.0012 0.0038 3027916 ChemDiv3_008098 COc1ccc(cc1OC)c2csc3ncc(c(=O)n23)S(=O)(=O)c4ccc(F)c(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A03 compound treatment 640.0 -298.0 -0.11 240.0 -353.0 -0.27 -0.266 -0.9157 3122121 ChemDiv3_008099 Cc1sc2n(CC(=O)NC3CCCCC3)c(=O)n(c4ccc(Cl)cc4)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A04 compound treatment 280.0 -658.0 -0.23 720.0 128.0 0.1 -0.0957 -0.3784 1870274 ChemDiv3_008100 Fc1ccc(cc1)C2CC(=Nc3nc(cn23)c4ccccc4)c5ccc(Cl)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A05 compound treatment 400.0 -538.0 -0.19 600.0 7.5 0.01 -0.1308 -0.6854 3122122 ChemDiv3_008101 O=C(Cn1c(=O)[nH]c2ccsc2c1=O)NC3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A06 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3027917 ChemDiv3_008102 CC(C)CC1CC(=O)NC(=N1)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A07 compound treatment 320.0 -618.0 -0.22 400.0 -193.0 -0.15 -0.2594 -0.9816 3122123 ChemDiv3_008103 Nc1c(nnn1c2ccc(OC(F)(F)F)cc2)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A08 compound treatment 4720.0 3780.0 1.34 360.0 -233.0 -0.18 0.8226 0.6077 3027963 ChemDiv3_008104 CCN(c1ccccc1)S(=O)(=O)c2ccc(CC(C)C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A09 compound treatment 1200.0 263.0 0.09 320.0 -273.0 -0.21 -0.0821 -0.3585 3122124 ChemDiv3_008105 CCN(c1ccccc1)c2nc3ccsc3c(=O)s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A10 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3027964 ChemDiv3_008106 C=CCNS(=O)(=O)c1cccs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A11 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3122125 ChemDiv3_008107 COC(=O)c1sccc1NC(=S)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A12 compound treatment 560.0 -378.0 -0.13 400.0 -193.0 -0.15 -0.1992 -0.9988 1255510 ChemDiv3_008108 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(Cl)s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A13 compound treatment 440.0 -498.0 -0.18 240.0 -353.0 -0.27 -0.3162 -0.9785 3122126 ChemDiv3_008109 COc1ccc(cc1)N2CCN(CCCn3c(NN)nc4ccsc4c3=O)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A14 compound treatment 320.0 -618.0 -0.22 880.0 288.0 0.22 0.0012 0.0038 3122127 ChemDiv3_008110 COc1ccc(CNC(=O)c2cc(=O)[nH]c3ccc(cc23)S(=O)(=O)N4CCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A15 compound treatment 520.0 -418.0 -0.15 880.0 288.0 0.22 0.0513 0.1932 3027965 ChemDiv3_008111 COc1ccc(Cl)cc1NC2=NC3CS(=O)(=O)CC3S2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A16 compound treatment 280.0 -658.0 -0.23 240.0 -353.0 -0.27 -0.3563 -0.9973 3122128 ChemDiv3_008112 CC1(C)CC(=O)c2cc(OCC(=O)NCCN3CCOCC3)ccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A17 compound treatment 280.0 -658.0 -0.23 3000.0 2410.0 1.85 1.142 0.613 3027966 ChemDiv3_008113 CCOC(=O)C1=C(Cn2nnc(C(=O)OC)c2C(=O)OC)NC(=O)NC1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A18 compound treatment 400.0 -538.0 -0.19 440.0 -153.0 -0.12 -0.2176 -0.9726 3122129 ChemDiv3_008114 CCN(CC)c1ccc(CNc2ccc3n(cnc3c2)C(C)(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A19 compound treatment 680.0 -258.0 -0.09 360.0 -233.0 -0.18 -0.1908 -0.9516 3122130 ChemDiv3_008115 COc1cc2nc(n3nc(C)cc3C)n4nc(nc4c2cc1OC)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A20 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3027967 ChemDiv3_008116 Cc1nc2c(cnn2c(O)c1Cc3ccccc3F)C(=O)NC4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A21 compound treatment 240.0 -698.0 -0.25 280.0 -313.0 -0.24 -0.3446 -0.9999 3122131 ChemDiv3_008117 O=c1oc2ccccc2cc1c3nc(no3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A22 compound treatment 320.0 -618.0 -0.22 240.0 -353.0 -0.27 -0.3463 -0.9945 3027968 ChemDiv3_008118 CN(c1cccc(C)c1)S(=O)(=O)c2ccc3NC(=O)CCc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A23 mock treatment 560.0 -378.0 -0.13 280.0 -313.0 -0.24 -0.2643 -0.9621 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 A24 mock treatment 480.0 -458.0 -0.16 320.0 -273.0 -0.21 -0.2627 -0.9921 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B01 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3122132 ChemDiv3_008119 CCCNS(=O)(=O)c1cccc2cccnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B02 compound treatment 280.0 -658.0 -0.23 440.0 -153.0 -0.12 -0.2477 -0.9492 3122133 ChemDiv3_008120 O=C(Nc1cccnc1)c2noc3CCCCc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B03 compound treatment 240.0 -698.0 -0.25 160.0 -433.0 -0.33 -0.4097 -0.9895 3027969 ChemDiv3_008121 Cc1ccc(Cl)cc1N2CCN(CC2)C(=O)C3CCN(CC3)S(=O)(=O)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B04 compound treatment 200.0 -738.0 -0.26 320.0 -273.0 -0.21 -0.3329 -0.9939 3122134 ChemDiv3_008122 CCCNC(=O)c1noc-2c1CCc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B05 compound treatment 280.0 -658.0 -0.23 3280.0 2690.0 2.06 1.294 0.6232 3122135 ChemDiv3_008123 FC(F)(F)c1cccc(NC(=O)CCS(=O)(=O)c2ccc(Br)s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B06 compound treatment 360.0 -578.0 -0.2 400.0 -193.0 -0.15 -0.2494 -0.9872 3027970 ChemDiv3_008124 COCC(C)NC(=O)c1noc-2c1CCc3cc(OC)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B07 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3122136 ChemDiv3_008125 Fc1ccc(cc1)c2cc(no2)C(=O)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B08 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3122137 ChemDiv3_008126 CCc1ccc(NC(=O)CCC(=O)Nc2ccc3nc(cc(C)c3c2)N4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B09 compound treatment 360.0 -578.0 -0.2 280.0 -313.0 -0.24 -0.3145 -0.9969 3027971 ChemDiv3_008127 COc1ccc(cc1)c2cc(no2)C(=O)N3CCN(C)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B10 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3027972 ChemDiv3_008128 COc1ccc(cc1)c2cn(c3ccc(Br)cc3)c(=O)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B11 compound treatment 320.0 -618.0 -0.22 240.0 -353.0 -0.27 -0.3463 -0.9945 3122534 ChemDiv3_008129 COc1ccccc1c2cc(no2)C(=O)NCc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B12 compound treatment 440.0 -498.0 -0.18 360.0 -233.0 -0.18 -0.251 -1.0 3122319 ChemDiv3_008130 CCC(C)NC(=O)c1cn(CCOC)c(=O)c2n(C)c3ccccc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B13 compound treatment 440.0 -498.0 -0.18 2880.0 2290.0 1.76 1.117 0.6329 3027973 ChemDiv3_008131 O=C(NC1CCCCC1)c2cc(on2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B14 compound treatment 240.0 -698.0 -0.25 640.0 47.5 0.04 -0.1492 -0.5965 3122320 ChemDiv3_008132 Cc1cccc(C)c1Nc2c(nc3[nH]cnn23)c4cc(Br)ccc4O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B15 compound treatment 1160.0 223.0 0.08 480.0 -113.0 -0.09 -0.0053 -0.0449 3027974 ChemDiv3_008133 COCC(C)NC(=O)c1cc(on1)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B16 compound treatment 280.0 -658.0 -0.23 480.0 -113.0 -0.09 -0.226 -0.9086 3122321 ChemDiv3_008134 O=C(C1C2N(CCc3ccccc23)C(=O)c4ccccc14)N5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B17 compound treatment 360.0 -578.0 -0.2 280.0 -313.0 -0.24 -0.3145 -0.9969 3027975 ChemDiv3_008135 Oc1ccccc1c2cc(no2)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B18 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3122322 ChemDiv3_008136 Cc1ccc(cc1)n2c(=O)n(CC(=O)N(CC=C)c3ccccc3)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B19 compound treatment 400.0 -538.0 -0.19 240.0 -353.0 -0.27 -0.3262 -0.9853 3027976 ChemDiv3_008137 O=C(N1CCc2ccccc2C1)c3cc(on3)C4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B20 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3122323 ChemDiv3_008138 CCOC(=O)c1ccccc1NC(=O)Cn2c(=O)n(c3cc(C)cc(C)c3)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B21 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3027977 ChemDiv3_008139 CC(C)Cc1cc(no1)C(=O)NCc2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B22 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3122324 ChemDiv3_008140 CCC(C)NC(=O)Cn1c(=O)n(CC(=O)NCc2ccc(C)cc2)c(=O)c3sccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B23 mock treatment 320.0 -618.0 -0.22 1040.0 448.0 0.34 0.088 0.2161 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 B24 mock treatment 240.0 -698.0 -0.25 720.0 128.0 0.1 -0.1057 -0.3974 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C01 compound treatment 2760.0 1820.0 0.65 280.0 -313.0 -0.24 0.2875 0.4169 3027978 ChemDiv3_008141 COc1cc2CCN(C(COc3ccc4c(C)cc(=O)oc4c3)c2cc1OC)C(=O)C5CC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C02 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3122325 ChemDiv3_008142 O=c1n(CCc2c[nH]c3ccccc23)c(=S)[nH]c4nccnc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C03 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 1228727 ChemDiv3_008143 Nc1c(oc2ccccc12)C(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C04 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 1226922 ChemDiv3_008144 CCOC(=O)C1=C(C)Nc2nc3ccccc3n2C1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C05 compound treatment 240.0 -698.0 -0.25 360.0 -233.0 -0.18 -0.3012 -0.9872 3122326 ChemDiv3_008145 Fc1ccc(cc1)N2CCN(CCCNC(=O)c3cccn4c(=O)c5ccccc5nc34)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C06 compound treatment 240.0 -698.0 -0.25 320.0 -273.0 -0.21 -0.3229 -0.9965 3027979 ChemDiv3_008146 O=C(Nc1ccc(Oc2ccccc2)cc1)c3ccc(Cn4c(=O)[nH]c5ccsc5c4=O)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C07 compound treatment 1560.0 623.0 0.22 240.0 -353.0 -0.27 -0.0352 -0.1008 3122327 ChemDiv3_008147 CCOC(=O)c1c(NC(=O)NCc2ccccc2)sc3CCCc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C08 compound treatment 520.0 -418.0 -0.15 280.0 -313.0 -0.24 -0.2744 -0.9731 3122328 ChemDiv3_008148 CC(C)Cc1ccc(cc1)S(=O)(=O)N2C(C)CCc3ccc(F)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C09 compound treatment 280.0 -658.0 -0.23 400.0 -193.0 -0.15 -0.2694 -0.9758 3122329 ChemDiv3_008149 Clc1ccc(cc1)N2CCN(CC2)c3nc4ccsc4c(=O)s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C10 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3027767 ChemDiv3_008150 O=S(=O)(c1cccs1)n2ccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C11 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3027768 ChemDiv3_008151 O=C(Nn1c(=O)[nH]c2ccsc2c1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C12 compound treatment 240.0 -698.0 -0.25 360.0 -233.0 -0.18 -0.3012 -0.9872 3122330 ChemDiv3_008152 CC(C)NS(=O)(=O)c1ccc(Cl)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C13 compound treatment 240.0 -698.0 -0.25 360.0 -233.0 -0.18 -0.3012 -0.9872 3122331 ChemDiv3_008153 Cc1nc2c3ccccc3nc(NN4C(=O)CCC4=O)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C14 compound treatment 400.0 -538.0 -0.19 360.0 -233.0 -0.18 -0.261 -0.9995 3027812 ChemDiv3_008154 CCN(c1cccc(C)c1)S(=O)(=O)c2c(C)[nH]c(=O)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C15 compound treatment 360.0 -578.0 -0.2 280.0 -313.0 -0.24 -0.3145 -0.9969 3122332 ChemDiv3_008155 O=C(Nc1ccccc1)c2ccc(NC3=NC4CS(=O)(=O)CC4S3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C16 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3027813 ChemDiv3_008156 CC1(C)CC(=O)c2cc(OCC(=O)NCc3ccccc3)ccc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C17 compound treatment 360.0 -578.0 -0.2 240.0 -353.0 -0.27 -0.3362 -0.9906 3122333 ChemDiv3_008157 O=C(NCc1ccccc1)C2CCCN(C2)c3nc4ccsc4c(=O)s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C18 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 3027815 ChemDiv3_008158 CCCn1cnc2cc(NCc3ccccc3O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C19 compound treatment 320.0 -618.0 -0.22 240.0 -353.0 -0.27 -0.3463 -0.9945 3122334 ChemDiv3_008159 Cc1ccc(cc1)c2nnn3c2[nH]c(=O)c4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C20 compound treatment 200.0 -738.0 -0.26 360.0 -233.0 -0.18 -0.3112 -0.9826 3122335 ChemDiv3_008160 CCOC(=O)C1CCCN(C1)C(=O)c2cnn3c(O)c(Cc4ccc(Cl)cc4)c(C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C21 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3027818 ChemDiv3_008161 COc1ccc(cc1)c2noc(n2)c/3cc4ccccc4o\c3=N/c5ccc(NC(=O)C)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C22 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3122336 ChemDiv3_008162 O=C1CCc2cc(ccc2N1)S(=O)(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C23 mock treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 C24 mock treatment 3360.0 2420.0 0.86 320.0 -273.0 -0.21 0.4597 0.5198 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D01 compound treatment 3800.0 2860.0 1.02 280.0 -313.0 -0.24 0.5484 0.5256 3027820 ChemDiv3_008163 COC(CNS(=O)(=O)c1cccc2cccnc12)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D02 compound treatment 360.0 -578.0 -0.2 400.0 -193.0 -0.15 -0.2494 -0.9872 3122337 ChemDiv3_008164 O=C(NC1CCCCC1)c2noc3CCCCCc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D03 compound treatment 280.0 -658.0 -0.23 360.0 -233.0 -0.18 -0.2911 -0.9913 3122338 ChemDiv3_008165 O=C(NC1CCCc2ccccc12)C3CCN(CC3)S(=O)(=O)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D04 compound treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 3027824 ChemDiv3_008166 CCc1ccccc1NC(=O)c2noc-3c2CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D05 compound treatment 480.0 -458.0 -0.16 360.0 -233.0 -0.18 -0.241 -0.9989 3122339 ChemDiv3_008167 Brc1ccc(s1)S(=O)(=O)CCC(=O)NC2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D06 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3122340 ChemDiv3_008168 COc1ccc2-c3onc(C(=O)Nc4cccnc4)c3CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D07 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3027875 ChemDiv3_008169 CN(Cc1ccccc1)C(=O)c2cc(on2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D08 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 3122341 ChemDiv3_008170 CC1CCN(CC1)C(=O)CCC(=O)Nc2ccc3nc(cc(C)c3c2)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D09 compound treatment 520.0 -418.0 -0.15 280.0 -313.0 -0.24 -0.2744 -0.9731 3027878 ChemDiv3_008171 COc1ccc(cc1)c2cc(no2)C(=O)N(C)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D10 compound treatment 400.0 -538.0 -0.19 240.0 -353.0 -0.27 -0.3262 -0.9853 3122342 ChemDiv3_008172 CC1CC(C)CN(C1)c2cc(C)c3cc(NC(=O)CCC(=O)Nc4ccc(F)cc4Cl)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D11 compound treatment 520.0 -418.0 -0.15 440.0 -153.0 -0.12 -0.1875 -0.9932 3027880 ChemDiv3_008173 COc1ccccc1c2cc(no2)C(=O)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D12 compound treatment 440.0 -498.0 -0.18 280.0 -313.0 -0.24 -0.2944 -0.9886 3122343 ChemDiv3_008174 COCCn1cc(C(=O)N2CCC(C)CC2)c3c4ccccc4n(C)c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D13 compound treatment 520.0 -418.0 -0.15 360.0 -233.0 -0.18 -0.2309 -0.9957 3027882 ChemDiv3_008175 O=C(NCCc1ccccc1)c2cc(on2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D14 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3122344 ChemDiv3_008176 Cc1cccc(C)c1Nc2c(nc3sccn23)c4ccsc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D15 compound treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 3122345 ChemDiv3_008177 O=C(Nc1sc2CCCc2c1C#N)c3cc(on3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D16 compound treatment 400.0 -538.0 -0.19 360.0 -233.0 -0.18 -0.261 -0.9995 3027885 ChemDiv3_008178 COc1ccccc1CNC(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D17 compound treatment 360.0 -578.0 -0.2 2200.0 1610.0 1.23 0.7278 0.5818 3122535 ChemDiv3_008179 Cc1cc(no1)C(=O)NCc2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D18 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3122536 ChemDiv3_008180 O=C(Cn1c(=O)n(c2ccccc2)c(=O)c3sccc13)NCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D19 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3027936 ChemDiv3_008181 CC(C)c1cc(no1)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D20 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3122537 ChemDiv3_008182 CCc1ccc(NC(=O)Cn2c(=O)n(CCC(=O)NCc3ccccc3)c(=O)c4sccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D21 compound treatment 1600.0 663.0 0.24 320.0 -273.0 -0.21 0.0183 0.058 3027939 ChemDiv3_008183 CC(C)Cc1cc(no1)C(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D22 compound treatment 2520.0 1580.0 0.56 280.0 -313.0 -0.24 0.2273 0.3723 3122538 ChemDiv3_008184 CN(C1CCCCC1)C(=O)Cn2c(=O)n(CC(=O)NCCc3ccccc3)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D23 mock treatment 320.0 -618.0 -0.22 360.0 -233.0 -0.18 -0.2811 -0.9948 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 D24 mock treatment 600.0 -338.0 -0.12 400.0 -193.0 -0.15 -0.1892 -0.9945 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E01 compound treatment 1920.0 983.0 0.35 280.0 -313.0 -0.24 0.0768 0.1815 3122539 ChemDiv3_008185 O=C(NCCNc1ccc2ccccc2c1)c3cccn4c(=O)c5sccc5nc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E02 compound treatment 960.0 22.5 0.01 2080.0 1490.0 1.14 0.8131 0.712 3027942 ChemDiv3_008186 COC(=O)c1ccccc1NC(=O)Cn2c(=O)c3ccccc3n4nncc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E03 compound treatment 1400.0 463.0 0.16 320.0 -273.0 -0.21 -0.0319 -0.12 3122540 ChemDiv3_008187 COc1cc(OC)cc(c1)n2c(=O)n(Cc3cc(=O)n4ccccc4n3)c5ccccc5c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E04 compound treatment 840.0 -97.5 -0.03 360.0 -233.0 -0.18 -0.1507 -0.8287 3027944 ChemDiv3_008188 NC1=C(C#N)C(Nc2nc3ccccc3n12)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E05 compound treatment 1280.0 343.0 0.12 400.0 -193.0 -0.15 -0.0186 -0.0971 3122541 ChemDiv3_008189 COc1ccc(OC)c(c1)C2NC(C3C2C(=O)N(C3=O)c4cccc(c4)C(=O)O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E06 compound treatment 520.0 -418.0 -0.15 760.0 168.0 0.13 -0.0138 -0.0703 3027947 ChemDiv3_008190 CCc1cccc(NC(=O)CCCn2c(=O)[nH]c3ccsc3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E07 compound treatment 2760.0 1820.0 0.65 1040.0 448.0 0.34 0.7001 0.9562 3122542 ChemDiv3_008191 COc1ccc(CC(=O)NC(=S)Nc2cccnc2Cl)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E08 compound treatment 360.0 -578.0 -0.2 840.0 248.0 0.19 -0.0105 -0.0376 3027949 ChemDiv3_008192 CNS(=O)(=O)c1cc(OC)ccc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E09 compound treatment 640.0 -298.0 -0.11 1520.0 928.0 0.71 0.4289 0.5958 3122543 ChemDiv3_008193 COc1ccc(cc1OC)c2cn(c3ccc(C)cc3C)c(=S)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E10 compound treatment 920.0 -17.5 -0.01 1280.0 688.0 0.53 0.3688 0.6987 1624330 ChemDiv3_008194 COc1ccccc1CNS(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E11 compound treatment 1080.0 143.0 0.05 560.0 -32.5 -0.02 0.0181 0.3211 3122544 ChemDiv3_008195 COC(=O)c1ccc(C(=O)OC)c(NC(=S)N2CC(C)CC(C)C2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E12 compound treatment 840.0 -97.5 -0.03 360.0 -233.0 -0.18 -0.1507 -0.8287 3027999 ChemDiv3_008196 Clc1ccc(s1)S(=O)(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E13 compound treatment 440.0 -498.0 -0.18 280.0 -313.0 -0.24 -0.2944 -0.9886 3122545 ChemDiv3_008197 CN(C)C(=O)c1sc2[nH]c(=O)n(c3ccccc3C(F)(F)F)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E14 compound treatment 1200.0 263.0 0.09 3960.0 3370.0 2.59 1.8939 0.7321 3028001 ChemDiv3_008198 CCCCN(CC)S(=O)(=O)c1c(C)[nH]c(=O)[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E15 compound treatment 1120.0 183.0 0.06 440.0 -153.0 -0.12 -0.037 -0.2766 3122546 ChemDiv3_008199 CCN(Cc1ccccc1)C(=O)Cn2c(=O)n(NC(=O)c3ccccc3)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E16 compound treatment 840.0 -97.5 -0.03 800.0 208.0 0.16 0.0882 0.541 3028003 ChemDiv3_008200 CC(C)NC(=O)COc1ccc2OC(C)(C)CC(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E17 compound treatment 960.0 22.5 0.01 840.0 248.0 0.19 0.14 0.7362 3122547 ChemDiv3_008201 COC(=O)c1cccnc1n2c(=O)n(Cc3ccccc3F)c4ncccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E18 compound treatment 5520.0 4580.0 1.63 1880.0 1290.0 0.99 1.8484 0.9716 3028005 ChemDiv3_008202 CC(C)n1cnc2cc(NCc3ccccc3O)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E19 compound treatment 600.0 -338.0 -0.12 880.0 288.0 0.22 0.0714 0.2844 3122548 ChemDiv3_008203 Cc1ccc(cc1)S(=O)(=O)c2c[nH]c(=S)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E20 compound treatment 1280.0 343.0 0.12 400.0 -193.0 -0.15 -0.0186 -0.0971 3122549 ChemDiv3_008204 Cc1nc2c(cnn2c(O)c1Cc3ccc(F)cc3Cl)C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E21 compound treatment 1600.0 663.0 0.24 1760.0 1170.0 0.9 0.8 0.8633 3028009 ChemDiv3_008205 CC1CCN(CC1)C(=O)c2ccc3c(=O)[nH]c4c(nnn4c3c2)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E22 compound treatment 600.0 -338.0 -0.12 680.0 87.5 0.07 -0.0372 -0.2707 1571875 ChemDiv3_008206 CC1Cc2ccccc2N1S(=O)(=O)c3ccc4[nH]c(=O)c(=O)[nH]c4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E23 mock treatment 1200.0 263.0 0.09 1080.0 488.0 0.37 0.3305 0.8569 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 E24 mock treatment 280.0 -658.0 -0.23 1200.0 608.0 0.47 0.1649 0.3161 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F01 compound treatment 1160.0 223.0 0.08 600.0 7.5 0.01 0.0599 0.7567 3028011 ChemDiv3_008207 CC(C)CN(CC(C)C)S(=O)(=O)c1cccc2cccnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F02 compound treatment 3800.0 2860.0 1.02 1040.0 448.0 0.34 0.961 0.8964 3122550 ChemDiv3_008208 O=C(NCCc1ccccc1)c2noc3CCCCCc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F03 compound treatment 1280.0 343.0 0.12 920.0 328.0 0.25 0.2637 0.9443 3122551 ChemDiv3_008209 Clc1cccc(c1)N2CCN(CC2)C(=O)C(NS(=O)(=O)c3cccs3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F04 compound treatment 2120.0 1180.0 0.42 1040.0 448.0 0.34 0.5396 0.9951 3028078 ChemDiv3_008210 Brc1ccc(NC(=O)c2noc-3c2CCc4ccccc34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F05 compound treatment 5320.0 4380.0 1.55 680.0 87.5 0.07 1.1468 0.737 3122552 ChemDiv3_008211 CCOC(=O)N1CCN(CC1)C(=O)CCS(=O)(=O)c2ccc(Br)s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F06 compound treatment 1840.0 903.0 0.32 960.0 368.0 0.28 0.4259 0.998 3028081 ChemDiv3_008212 Nc1nc(cc(n1)C(F)(F)F)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F07 compound treatment 1200.0 263.0 0.09 760.0 168.0 0.13 0.1568 0.9874 3122553 ChemDiv3_008213 CC1CCCC(C)N1C(=O)c2cc(on2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F08 compound treatment 800.0 -138.0 -0.05 1360.0 768.0 0.59 0.3822 0.6464 3028083 ChemDiv3_008214 Brc1ccc(s1)c2cc(C(=O)NCCN3CCc4ccccc4C3)c5ccccc5n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F09 compound treatment 1240.0 303.0 0.11 1040.0 448.0 0.34 0.3188 0.8858 3122554 ChemDiv3_008215 COc1ccc(cc1)c2cc(no2)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F10 compound treatment 1160.0 223.0 0.08 760.0 168.0 0.13 0.1467 0.9725 3122555 ChemDiv3_008216 CC1CC(C)CN(C1)c2cc(C)c3cc(NC(=O)CCC(=O)N4CCCC4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F11 compound treatment 2120.0 1180.0 0.42 560.0 -32.5 -0.02 0.279 0.6639 3028086 ChemDiv3_008217 COc1ccc(cc1OC)c2cc(no2)C(=O)NCC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F12 compound treatment 4280.0 3340.0 1.19 1840.0 1250.0 0.96 1.5157 0.9944 3122556 ChemDiv3_008218 COCCn1cc(C(=O)NC2CCCCCC2)c3c4ccccc4n(C)c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F13 compound treatment 1320.0 383.0 0.14 680.0 87.5 0.07 0.1434 0.9474 3028088 ChemDiv3_008219 O=C(NCc1ccccc1)c2cc(on2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F14 compound treatment 360.0 -578.0 -0.2 2120.0 1530.0 1.17 0.6844 0.5749 3122557 ChemDiv3_008220 Cc1cccc(NC(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F15 compound treatment 1600.0 663.0 0.24 2880.0 2290.0 1.76 1.408 0.7947 3028090 ChemDiv3_008221 CCC1CCCCN1C(=O)c2cc(on2)c3ccc(Cl)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F16 compound treatment 2080.0 1140.0 0.41 520.0 -72.5 -0.06 0.2472 0.6043 3122558 ChemDiv3_008222 CCOc1ccc(CCNC(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25)cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F17 compound treatment 1640.0 703.0 0.25 1680.0 1090.0 0.83 0.7666 0.8798 3028091 ChemDiv3_008223 Cc1cc(no1)C(=O)NC2CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F18 compound treatment 960.0 22.5 0.01 800.0 208.0 0.16 0.1183 0.7416 3122559 ChemDiv3_008224 Cc1cccc(Cn2c(=O)n(c3ccccc3)c(=O)c4sccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F19 compound treatment 840.0 -97.5 -0.03 1120.0 528.0 0.4 0.2619 0.6444 3028094 ChemDiv3_008225 CC(C)c1cc(no1)C(=O)NCc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F20 compound treatment 600.0 -338.0 -0.12 1480.0 888.0 0.68 0.3971 0.5741 3122944 ChemDiv3_008226 Cc1ccc(CNC(=O)CCCn2c(=O)n(Cc3ccc(F)cc3Cl)c4ccsc4c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F21 compound treatment 1720.0 783.0 0.28 1480.0 888.0 0.68 0.6781 0.9216 3028165 ChemDiv3_008227 CCCNC(=O)c1cc(CC(C)C)on1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F22 compound treatment 2000.0 1060.0 0.38 600.0 7.5 0.01 0.2706 0.7178 3122742 ChemDiv3_008228 Fc1cccc(NC(=O)Cn2c(=O)n(CC(=O)NCCc3ccccc3)c(=O)c4sccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F23 mock treatment 1360.0 423.0 0.15 600.0 7.5 0.01 0.1101 0.7337 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 F24 mock treatment 1280.0 343.0 0.12 760.0 168.0 0.13 0.1768 0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G01 compound treatment 520.0 -418.0 -0.15 1240.0 648.0 0.5 0.2468 0.4758 3028167 ChemDiv3_008229 O=C(NCc1ccccc1)c2ccc3nc4ccccc4c(=O)n3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G02 compound treatment 720.0 -218.0 -0.08 400.0 -193.0 -0.15 -0.1591 -0.9541 3122743 ChemDiv3_008230 Cc1ccc(cc1)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G03 compound treatment 880.0 -57.5 -0.02 680.0 87.5 0.07 0.0331 0.4712 3122744 ChemDiv3_008231 CC1CCCCN1C(=O)Cn2c(=O)n(c3ccc(Cl)cc3)c(=O)c4c(C)c(C)sc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G04 compound treatment 1160.0 223.0 0.08 1200.0 608.0 0.47 0.3856 0.8152 3028170 ChemDiv3_008232 NC1=C(C#N)C(Nc2ncnn12)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G05 compound treatment 520.0 -418.0 -0.15 520.0 -72.5 -0.06 -0.1441 -0.9107 3122745 ChemDiv3_008233 COc1cccc(C2NC(C3C2C(=O)N(C3=O)c4cccc(c4)C(=O)O)C(=O)O)c1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G06 compound treatment 440.0 -498.0 -0.18 480.0 -113.0 -0.09 -0.1859 -0.946 3028171 ChemDiv3_008234 O=C(Cc1ccc(cc1)n2c(=O)[nH]c3ccsc3c2=O)Nc4ccc(cc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G07 compound treatment 840.0 -97.5 -0.03 360.0 -233.0 -0.18 -0.1507 -0.8287 3122746 ChemDiv3_008235 Clc1ncccc1NC(=S)NC(=O)/C=C/c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G08 compound treatment 520.0 -418.0 -0.15 520.0 -72.5 -0.06 -0.1441 -0.9107 1632740 ChemDiv3_008236 COc1ccc(OC)c(c1)S(=O)(=O)NC2CCN(Cc3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G09 compound treatment 520.0 -418.0 -0.15 280.0 -313.0 -0.24 -0.2744 -0.9731 3122747 ChemDiv3_008237 COc1ccc(cc1OC)c2cn(c3ccc(C)c(Cl)c3)c(=S)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G10 compound treatment 720.0 -218.0 -0.08 400.0 -193.0 -0.15 -0.1591 -0.9541 3028174 ChemDiv3_008238 CNS(=O)(=O)c1cccs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G11 compound treatment 8880.0 7940.0 2.82 400.0 -193.0 -0.15 1.8878 0.6691 3122748 ChemDiv3_008239 COC(=O)c1sccc1NC(=S)N(C)CCC#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G12 compound treatment 600.0 -338.0 -0.12 320.0 -273.0 -0.21 -0.2326 -0.9649 3028177 ChemDiv3_008240 CC(C)CN(CC(C)C)S(=O)(=O)c1ccc(Br)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G13 compound treatment 320.0 -618.0 -0.22 360.0 -233.0 -0.18 -0.2811 -0.9948 3122749 ChemDiv3_008241 CCc1cccc(NC(=O)NC(=O)Cn2nnc(C(=O)OC)c2C(=O)OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G14 compound treatment 600.0 -338.0 -0.12 1160.0 568.0 0.44 0.2234 0.4945 3122750 ChemDiv3_008242 COc1ccc(cc1)N(C)S(=O)(=O)c2c(C)[nH]c(=O)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G15 compound treatment 880.0 -57.5 -0.02 280.0 -313.0 -0.24 -0.1841 -0.7645 3122751 ChemDiv3_008243 Cc1cc(C)c(Cn2c(=O)n(NC(=O)c3ccccc3)c(=O)c4sccc24)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G16 compound treatment 1520.0 583.0 0.21 4360.0 3770.0 2.89 2.1913 0.7557 3028247 ChemDiv3_008244 CCN(CC)C(=O)COc1ccc2OC(C)(C)CC(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G17 compound treatment 360.0 -578.0 -0.2 880.0 288.0 0.22 0.0112 0.0372 3028249 ChemDiv3_008245 OC1=C(NS(=O)(=O)c2ccccc12)C(=O)c3ccc(Cl)s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G18 compound treatment 600.0 -338.0 -0.12 400.0 -193.0 -0.15 -0.1892 -0.9945 3122752 ChemDiv3_008246 CCCn1cnc2cc(NCc3cccc(OC)c3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G19 compound treatment 520.0 -418.0 -0.15 480.0 -113.0 -0.09 -0.1658 -0.967 3122753 ChemDiv3_008247 Fc1ccc(cc1)S(=O)(=O)c2c[nH]c(=S)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G20 compound treatment 880.0 -57.5 -0.02 1600.0 1010.0 0.77 0.5325 0.6882 3028251 ChemDiv3_008248 CC(C)C(NS(=O)(=O)c1cccs1)C(=O)NC2CCCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G21 compound treatment 1840.0 903.0 0.32 320.0 -273.0 -0.21 0.0785 0.2051 3122754 ChemDiv3_008249 COc1cccc(CN2CCc3[nH]c(=S)[nH]c(=O)c3C2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G22 compound treatment 8080.0 7140.0 2.53 720.0 128.0 0.1 1.8609 0.7339 3028254 ChemDiv3_008250 O=S(=O)(NCCC1=CCCCC1)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G23 mock treatment 480.0 -458.0 -0.16 560.0 -32.5 -0.02 -0.1324 -0.8063 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 G24 mock treatment 520.0 -418.0 -0.15 920.0 328.0 0.25 0.0731 0.2504 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H01 compound treatment 18600.0 17700.0 6.27 440.0 -153.0 -0.12 4.3477 0.6938 3122755 ChemDiv3_008251 CCCCN(C)S(=O)(=O)c1cccc2cccnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H02 compound treatment 1440.0 503.0 0.18 840.0 248.0 0.19 0.2604 0.9995 3122756 ChemDiv3_008252 CC(C)(C)C1CCc2onc(C(=O)NCc3ccc(F)cc3)c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H03 compound treatment 4200.0 3260.0 1.16 840.0 248.0 0.19 0.9527 0.8123 3028256 ChemDiv3_008253 O=C(NCc1ccccc1)C(NS(=O)(=O)c2cccs2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H04 compound treatment 680.0 -258.0 -0.09 800.0 208.0 0.16 0.0481 0.2617 3122757 ChemDiv3_008254 Cc1ccc(Cn2ccc(NC(=O)c3noc-4c3CCc5ccccc45)n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H05 compound treatment 680.0 -258.0 -0.09 600.0 7.5 0.01 -0.0605 -0.6612 3028258 ChemDiv3_008255 Cc1ccc(CNC(=O)CCS(=O)(=O)c2ccc(Br)s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H06 compound treatment 400.0 -538.0 -0.19 560.0 -32.5 -0.02 -0.1525 -0.7929 3122758 ChemDiv3_008256 Fc1ccc(cc1)c2cc(nc(n2)n3cccn3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H07 compound treatment 880.0 -57.5 -0.02 320.0 -273.0 -0.21 -0.1624 -0.7724 3028261 ChemDiv3_008257 CC(C)NC(=O)c1cc(on1)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H08 compound treatment 600.0 -338.0 -0.12 920.0 328.0 0.25 0.0931 0.3344 1377023 ChemDiv3_008258 O=C(NC1CCCC1)C2COc3ccccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H09 compound treatment 680.0 -258.0 -0.09 280.0 -313.0 -0.24 -0.2342 -0.9124 3122759 ChemDiv3_008259 COc1ccc(cc1)c2cc(no2)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H10 compound treatment 640.0 -298.0 -0.11 560.0 -32.5 -0.02 -0.0923 -0.8508 3122760 ChemDiv3_008260 CC(C)Cn1cc(C(=O)N2CCCC2)c3c4ccccc4n(C)c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H11 compound treatment 720.0 -218.0 -0.08 520.0 -72.5 -0.06 -0.0939 -0.9872 3027825 ChemDiv3_008261 CCN(CC)C(=O)c1cc(on1)c2ccc(OC)c(OC)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H12 compound treatment 760.0 -178.0 -0.06 2160.0 1570.0 1.2 0.8064 0.6692 3027827 ChemDiv3_008262 Cc1cccc(C)c1Nc2c(CN3C(=O)c4ccccc4C3=O)nc5ccc(Br)cn25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H13 compound treatment 880.0 -57.5 -0.02 1960.0 1370.0 1.05 0.7279 0.6932 3122761 ChemDiv3_008263 CCCNC(=O)c1cc(on1)c2ccco2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H14 compound treatment 600.0 -338.0 -0.12 440.0 -153.0 -0.12 -0.1674 -0.9999 3122762 ChemDiv3_008264 COc1cccc(NC(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H15 compound treatment 680.0 -258.0 -0.09 320.0 -273.0 -0.21 -0.2125 -0.931 3027829 ChemDiv3_008265 CN(C(=O)c1cc(on1)c2ccc(Cl)c(Cl)c2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H16 compound treatment 800.0 -138.0 -0.05 400.0 -193.0 -0.15 -0.139 -0.8931 3122763 ChemDiv3_008266 CCC1CCCCN1C(=O)Cn2c(=O)n(c3cc(F)ccc3F)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H17 compound treatment 560.0 -378.0 -0.13 1880.0 1290.0 0.99 0.6042 0.6058 3027831 ChemDiv3_008267 Cc1cc(no1)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H18 compound treatment 800.0 -138.0 -0.05 520.0 -72.5 -0.06 -0.0738 -0.9978 3122764 ChemDiv3_008268 Cc1ccc(cc1F)n2c(=O)n(CC(=O)NCC3CCCO3)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H19 compound treatment 440.0 -498.0 -0.18 320.0 -273.0 -0.21 -0.2727 -0.9964 3027833 ChemDiv3_008269 COc1ccc(CNC(=O)c2cc(on2)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H20 compound treatment 720.0 -218.0 -0.08 560.0 -32.5 -0.02 -0.0722 -0.8904 3122765 ChemDiv3_008270 Fc1ccc(Cn2c(=O)n(CCCC(=O)NCc3ccc4OCOc4c3)c(=O)c5sccc25)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H21 compound treatment 560.0 -378.0 -0.13 440.0 -153.0 -0.12 -0.1775 -0.9978 3027835 ChemDiv3_008271 CC(C)Cc1cc(no1)C(=O)Nc2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H22 compound treatment 880.0 -57.5 -0.02 720.0 128.0 0.1 0.0548 0.548 3122766 ChemDiv3_008272 Clc1cccc(Cn2c(=O)n(CC(=O)NCc3ccco3)c(=O)c4sccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H23 mock treatment 640.0 -298.0 -0.11 480.0 -113.0 -0.09 -0.1357 -0.995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 H24 mock treatment 4880.0 3940.0 1.4 600.0 7.5 0.01 0.993 0.71 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I01 compound treatment 8040.0 7100.0 2.52 360.0 -233.0 -0.18 1.6554 0.6554 3027838 ChemDiv3_008273 Clc1ccc(CNC(=O)c2ccc3c(=O)n(c4ccccc4)c(=O)[nH]c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I02 compound treatment 520.0 -418.0 -0.15 360.0 -233.0 -0.18 -0.2309 -0.9957 3027888 ChemDiv3_008274 CC1C(NC(C(C)C1=O)c2ccc(Br)cc2)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I03 compound treatment 280.0 -658.0 -0.23 360.0 -233.0 -0.18 -0.2911 -0.9913 3122767 ChemDiv3_008275 Cc1sc2n(CC(=O)NCc3ccc(C)cc3)c(=O)n(c4ccc(C)c(C)c4)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I04 compound treatment 360.0 -578.0 -0.2 520.0 -72.5 -0.06 -0.1842 -0.8678 3027890 ChemDiv3_008276 CC(C)C1C2=C(CC(C)(C)CC2=O)Nc3nc(SCc4cccc(C)c4)[nH]c(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I05 compound treatment 360.0 -578.0 -0.2 1240.0 648.0 0.5 0.2066 0.3843 3122768 ChemDiv3_008277 COc1ccc(NC(=O)CCCn2c(=O)n(Cc3ccccc3)c4ccsc4c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I06 compound treatment 240.0 -698.0 -0.25 360.0 -233.0 -0.18 -0.3012 -0.9872 3122945 ChemDiv3_008278 CC1CCCCC1NC(=O)CN2C(=O)COc3ccc(C)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I07 compound treatment 400.0 -538.0 -0.19 280.0 -313.0 -0.24 -0.3045 -0.9935 3027892 ChemDiv3_008279 Fc1ccc(cc1)C(=O)c2c[nH]c3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I08 compound treatment 360.0 -578.0 -0.2 520.0 -72.5 -0.06 -0.1842 -0.8678 3027894 ChemDiv3_008280 Brc1cccc(NS(=O)(=O)c2cccs2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I09 compound treatment 240.0 -698.0 -0.25 1040.0 448.0 0.34 0.068 0.1605 3122946 ChemDiv3_008281 COC(=O)c1ccc(C(=O)OC)c(NC(=S)N2CCCCC2C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I10 compound treatment 360.0 -578.0 -0.2 560.0 -32.5 -0.02 -0.1625 -0.7874 3027898 ChemDiv3_008282 CSc1cccc(NS(=O)(=O)c2cccs2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I11 compound treatment 200.0 -738.0 -0.26 280.0 -313.0 -0.24 -0.3546 -0.9991 3122947 ChemDiv3_008283 COC(=O)c1sccc1NC(=S)N2CC(C)CC(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I12 compound treatment 320.0 -618.0 -0.22 3080.0 2490.0 1.91 1.1955 0.6219 3027900 ChemDiv3_008284 O=C(CCn1c(=O)oc2ccccc12)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I13 compound treatment 280.0 -658.0 -0.23 640.0 47.5 0.04 -0.1391 -0.5894 3122948 ChemDiv3_008285 O=C(CCn1c(=O)c2sc3ccccc3c2[nH]c1=S)NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I14 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3122949 ChemDiv3_008286 CCOC(=O)C1=C(NC(=C(C#N)C1c2ccco2)SCC(=O)Nc3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I15 compound treatment 280.0 -658.0 -0.23 360.0 -233.0 -0.18 -0.2911 -0.9913 3027952 ChemDiv3_008287 COc1ccc(CCn2c(NN)nc3ccsc3c2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I16 compound treatment 160.0 -778.0 -0.28 400.0 -193.0 -0.15 -0.2995 -0.9572 3122950 ChemDiv3_008288 CCCCn1cnc2cc(NCc3ccc(C)cc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I17 compound treatment 240.0 -698.0 -0.25 280.0 -313.0 -0.24 -0.3446 -0.9999 3122951 ChemDiv3_008289 COC(=O)c1nnn(CC(=O)N(Cc2ccccc2)c3ccc(Br)cc3)c1C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I18 compound treatment 280.0 -658.0 -0.23 360.0 -233.0 -0.18 -0.2911 -0.9913 3027956 ChemDiv3_008290 CCCn1cnc2cc(NCc3ccc(Cl)cc3Cl)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I19 compound treatment 240.0 -698.0 -0.25 320.0 -273.0 -0.21 -0.3229 -0.9965 3027957 ChemDiv3_008291 CCCCN1CCc2[nH]c(=S)[nH]c(=O)c2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I20 compound treatment 520.0 -418.0 -0.15 320.0 -273.0 -0.21 -0.2527 -0.9857 3122952 ChemDiv3_008292 CC(C)C(NS(=O)(=O)c1cccs1)C(=O)Nc2cccc(C)c2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I21 compound treatment 360.0 -578.0 -0.2 240.0 -353.0 -0.27 -0.3362 -0.9906 1293215 ChemDiv3_008293 O=c1n(c2ccccc2)c(=S)[nH]c3c4ccccc4oc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I22 compound treatment 240.0 -698.0 -0.25 360.0 -233.0 -0.18 -0.3012 -0.9872 3027960 ChemDiv3_008294 C=CCN(c1ccccc1)S(=O)(=O)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I23 mock treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 I24 mock treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J01 compound treatment 320.0 -618.0 -0.22 720.0 128.0 0.1 -0.0857 -0.3571 3122953 ChemDiv3_008295 O=S(=O)(N(CCc1ccccc1)Cc2ccccc2)c3cccc4cccnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J02 compound treatment 440.0 -498.0 -0.18 480.0 -113.0 -0.09 -0.1859 -0.946 3028950 ChemDiv3_008296 CCc1c(C)sc(NC(=O)c2noc3CCC(Cc23)C(C)(C)C)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J03 compound treatment 320.0 -618.0 -0.22 160.0 -433.0 -0.33 -0.3897 -0.9796 3028951 ChemDiv3_008297 Cc1cccc(NC(=O)CNS(=O)(=O)c2ccc(Br)s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J04 compound treatment 320.0 -618.0 -0.22 240.0 -353.0 -0.27 -0.3463 -0.9945 3028952 ChemDiv3_008298 Cc1nn(Cc2ccccc2)c(C)c1NC(=O)c3noc-4c3CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J05 compound treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 3028953 ChemDiv3_008299 Brc1ccc(s1)S(=O)(=O)CCC(=O)NC(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J06 compound treatment 360.0 -578.0 -0.2 400.0 -193.0 -0.15 -0.2494 -0.9872 3028954 ChemDiv3_008300 Cc1nccn1c2nc(cc(n2)C(F)(F)F)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J07 compound treatment 8160.0 7220.0 2.56 3600.0 3010.0 2.31 3.4444 0.9987 3028955 ChemDiv3_008301 CC(C)CNC(=O)c1cc(on1)c2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J08 compound treatment 240.0 -698.0 -0.25 720.0 128.0 0.1 -0.1057 -0.3974 3028956 ChemDiv3_008302 CSc1cccc(NC(=O)C2COc3ccccc3O2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J09 compound treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 3122954 ChemDiv3_008303 COc1cccc(c1)c2cc(no2)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J10 compound treatment 280.0 -658.0 -0.23 360.0 -233.0 -0.18 -0.2911 -0.9913 3122955 ChemDiv3_008304 CC(C)Cn1cc(C(=O)NCc2ccco2)c3c4ccccc4n(C)c3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J11 compound treatment 360.0 -578.0 -0.2 1200.0 608.0 0.47 0.1849 0.363 3028957 ChemDiv3_008305 O=C(N1CCOCC1)c2cc(on2)c3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J12 compound treatment 280.0 -658.0 -0.23 2000.0 1410.0 1.08 0.5991 0.542 3122956 ChemDiv3_008306 Brc1ccc2nc(CN3C(=O)c4ccccc4C3=O)c(NC5CCCCC5)n2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J13 compound treatment 200.0 -738.0 -0.26 480.0 -113.0 -0.09 -0.2461 -0.8931 3028958 ChemDiv3_008307 O=C(N(C1CCCCC1)C2CCCCC2)c3cc(on3)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J14 compound treatment 280.0 -658.0 -0.23 360.0 -233.0 -0.18 -0.2911 -0.9913 3122957 ChemDiv3_008308 Cc1cc(Br)ccc1NC(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J15 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3028959 ChemDiv3_008309 CCN(CC)C(=O)c1cc(on1)c2ccc(Cl)c(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J16 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 3122958 ChemDiv3_008310 COc1cccc(c1)n2c(=O)n(Cc3ccc(F)cc3Cl)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J17 compound treatment 280.0 -658.0 -0.23 240.0 -353.0 -0.27 -0.3563 -0.9973 3028960 ChemDiv3_008311 Cc1cc(no1)C(=O)N(C2CCCCC2)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J18 compound treatment 880.0 -57.5 -0.02 360.0 -233.0 -0.18 -0.1406 -0.7828 3122959 ChemDiv3_008312 COc1cccc(c1)n2c(=O)n(Cc3ccc(cc3)C(C)(C)C)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J19 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3028961 ChemDiv3_008313 CCCNC(=O)c1cc(on1)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J20 compound treatment 320.0 -618.0 -0.22 240.0 -353.0 -0.27 -0.3463 -0.9945 3122960 ChemDiv3_008314 CC1CC(C)CN(C1)C(=O)Cn2c(=O)n(CCCC(=O)NCc3ccco3)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J21 compound treatment 640.0 -298.0 -0.11 280.0 -313.0 -0.24 -0.2443 -0.932 3028962 ChemDiv3_008315 O=C(NCc1cccnc1)c2noc3CCCCc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J22 compound treatment 360.0 -578.0 -0.2 560.0 -32.5 -0.02 -0.1625 -0.7874 3122961 ChemDiv3_008316 CCN(Cc1ccccc1)C(=O)Cn2c(=O)n(CC(=O)NCc3ccco3)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J23 mock treatment 1160.0 223.0 0.08 440.0 -153.0 -0.12 -0.027 -0.191 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 J24 mock treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K01 compound treatment 1040.0 103.0 0.04 1400.0 808.0 0.62 0.4641 0.7473 3028963 ChemDiv3_008317 Clc1ccc(CCNC(=O)c2ccc3c(=O)n(c4ccccc4)c(=O)[nH]c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K02 compound treatment 960.0 22.5 0.01 400.0 -193.0 -0.15 -0.0989 -0.6679 3122962 ChemDiv3_008318 CC(C)C1CCC(C)CC1OC(=O)C2=C(C)Nc3nnnn3C2c4ccc(Br)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K03 compound treatment 2560.0 1620.0 0.58 560.0 -32.5 -0.02 0.3894 0.6758 3122963 ChemDiv3_008319 O=C(Cn1c(=O)n(Cc2ccccc2)c(=O)c3ccccc13)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K04 compound treatment 840.0 -97.5 -0.03 920.0 328.0 0.25 0.1533 0.6041 3028964 ChemDiv3_008320 O=C(CC1SC(=NC1=O)N2N=C(CC2c3ccccc3)c4ccccc4)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K05 compound treatment 1000.0 62.5 0.02 360.0 -233.0 -0.18 -0.1105 -0.6146 3122964 ChemDiv3_008321 COc1ccc(NC(=O)CCCn2c(=O)n(CC(=O)C(C)(C)C)c3ccsc3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K06 compound treatment 800.0 -138.0 -0.05 760.0 168.0 0.13 0.0564 0.4104 3122965 ChemDiv3_008322 CC1CCC(CC1)NC(=O)CCN2C(=O)COc3ccc(C)cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K07 compound treatment 840.0 -97.5 -0.03 560.0 -32.5 -0.02 -0.0421 -0.9872 3028965 ChemDiv3_008323 COC(=O)c1nnn(CC(=O)Nc2ccc(OC)cc2)c1N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K08 compound treatment 880.0 -57.5 -0.02 440.0 -153.0 -0.12 -0.0972 -0.818 1741953 ChemDiv3_008324 COc1ccc(C)cc1NS(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K09 compound treatment 4160.0 3220.0 1.14 600.0 7.5 0.01 0.8124 0.7107 3122966 ChemDiv3_008325 COC(=O)c1ccc(C(=O)OC)c(NC(=S)N2CCCC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K10 compound treatment 1120.0 183.0 0.06 2600.0 2010.0 1.54 1.1356 0.7362 3028966 ChemDiv3_008326 CCN(c1ccccc1)S(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K11 compound treatment 640.0 -298.0 -0.11 560.0 -32.5 -0.02 -0.0923 -0.8508 3122967 ChemDiv3_008327 CCN(CC)C(=S)Nc1ccsc1C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K12 compound treatment 840.0 -97.5 -0.03 400.0 -193.0 -0.15 -0.129 -0.8496 3122968 ChemDiv3_008328 CC1CCCCC1NC(=O)CCn2c(=O)oc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K13 compound treatment 1640.0 703.0 0.25 360.0 -233.0 -0.18 0.05 0.1631 3028967 ChemDiv3_008329 CCOC(=O)c1ccccc1NC(=S)N2CC(C)CC(C)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K14 compound treatment 2360.0 1420.0 0.5 2120.0 1530.0 1.17 1.186 0.929 3122969 ChemDiv3_008330 CC(=O)N1CCC2(CC1)CC(=O)c3cc(OCC(=O)N4CCCC4)ccc3O2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K15 compound treatment 600.0 -338.0 -0.12 360.0 -233.0 -0.18 -0.2109 -0.9811 3028968 ChemDiv3_008331 Cc1ccc(CSC2=NS(=O)(=O)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K16 compound treatment 760.0 -178.0 -0.06 680.0 87.5 0.07 0.003 0.0323 3123352 ChemDiv3_008332 CC(C)n1cnc2cc(NCc3ccc(Br)cc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K17 compound treatment 480.0 -458.0 -0.16 680.0 87.5 0.07 -0.0673 -0.3829 3028969 ChemDiv3_008333 Clc1ccc(cc1)c2nnn3c2nc(Cl)c4ccccc43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K18 compound treatment 880.0 -57.5 -0.02 440.0 -153.0 -0.12 -0.0972 -0.818 3123148 ChemDiv3_008334 COc1cccc(CNc2ccc3n(cnc3c2)C(C)(C)C)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K19 compound treatment 760.0 -178.0 -0.06 560.0 -32.5 -0.02 -0.0622 -0.9179 3123149 ChemDiv3_008335 CCOC(=O)c1[nH]c2ccc(OC)cc2c1NC(=S)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K20 compound treatment 640.0 -298.0 -0.11 440.0 -153.0 -0.12 -0.1574 -0.9987 3028970 ChemDiv3_008336 CCOc1ccc(OCC)c(NC(=O)C(NS(=O)(=O)c2cccs2)C(C)C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K21 compound treatment 760.0 -178.0 -0.06 560.0 -32.5 -0.02 -0.0622 -0.9179 3123150 ChemDiv3_008337 Cc1noc(n1)c2cc3cc(Br)ccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K22 compound treatment 1480.0 543.0 0.19 920.0 328.0 0.25 0.3139 0.9913 3028971 ChemDiv3_008338 O=S(=O)(NN1CCOCC1)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K23 mock treatment 520.0 -418.0 -0.15 440.0 -153.0 -0.12 -0.1875 -0.9932 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 K24 mock treatment 600.0 -338.0 -0.12 480.0 -113.0 -0.09 -0.1457 -0.9872 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L01 compound treatment 880.0 -57.5 -0.02 760.0 168.0 0.13 0.0765 0.5876 3123151 ChemDiv3_008339 CCCCN(c1ccccc1)S(=O)(=O)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L02 compound treatment 1480.0 543.0 0.19 1560.0 968.0 0.74 0.6613 0.8619 3123152 ChemDiv3_008340 Cc1nn(Cc2c(Cl)cccc2Cl)c(C)c1NC(=O)c3noc4CCC(Cc34)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L03 compound treatment 600.0 -338.0 -0.12 440.0 -153.0 -0.12 -0.1674 -0.9999 3028972 ChemDiv3_008341 Brc1ccc(s1)S(=O)(=O)NCC(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L04 compound treatment 480.0 -458.0 -0.16 2440.0 1850.0 1.42 0.8882 0.6221 3123153 ChemDiv3_008342 COc1ccc2-c3onc(C(=O)N4C(C)CCCC4C)c3CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L05 compound treatment 680.0 -258.0 -0.09 480.0 -113.0 -0.09 -0.1257 -0.9996 3028973 ChemDiv3_008343 CCc1ccc(NC(=O)c2ccc(NC(=O)CCS(=O)(=O)c3cccs3)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L06 compound treatment 520.0 -418.0 -0.15 440.0 -153.0 -0.12 -0.1875 -0.9932 3123154 ChemDiv3_008344 COc1cccc(c1)c2cc(nc(n2)n3cccn3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L07 compound treatment 360.0 -578.0 -0.2 440.0 -153.0 -0.12 -0.2276 -0.9648 3028974 ChemDiv3_008345 Brc1ccc(cc1)c2cc(no2)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L08 compound treatment 440.0 -498.0 -0.18 440.0 -153.0 -0.12 -0.2076 -0.9801 3123155 ChemDiv3_008346 Clc1ccc(s1)c2cc(C(=O)NC3CCCC3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L09 compound treatment 760.0 -178.0 -0.06 480.0 -113.0 -0.09 -0.1056 -0.9879 3123156 ChemDiv3_008347 COc1cccc(c1)c2cc(no2)C(=O)N3CCCCC3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L10 compound treatment 800.0 -138.0 -0.05 280.0 -313.0 -0.24 -0.2041 -0.8338 3028975 ChemDiv3_008348 CCOc1ccc(NC(=O)c2cn(CC(C)C)c(=O)c3n(C)c4ccccc4c23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L11 compound treatment 600.0 -338.0 -0.12 480.0 -113.0 -0.09 -0.1457 -0.9872 3123157 ChemDiv3_008349 Cc1cc(NC(=O)c2cc(on2)c3ccc4OCOc4c3)n(n1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L12 compound treatment 760.0 -178.0 -0.06 440.0 -153.0 -0.12 -0.1273 -0.9577 3028976 ChemDiv3_008350 CSc1ccc(cc1)c2nc3ccc(C)cn3c2NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L13 compound treatment 760.0 -178.0 -0.06 520.0 -72.5 -0.06 -0.0839 -0.9981 3123158 ChemDiv3_008351 O=C(NCc1cccs1)c2cc(on2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L14 compound treatment 880.0 -57.5 -0.02 640.0 47.5 0.04 0.0114 0.2719 3123159 ChemDiv3_008352 CCC(C)NC(=O)C1C2N(CCc3ccccc23)C(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L15 compound treatment 760.0 -178.0 -0.06 400.0 -193.0 -0.15 -0.149 -0.9277 3028977 ChemDiv3_008353 Clc1ccc(cc1Cl)c2cc(no2)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L16 compound treatment 600.0 -338.0 -0.12 1160.0 568.0 0.44 0.2234 0.4945 3123160 ChemDiv3_008354 CCN(Cc1ccccc1)C(=O)Cn2c(=O)n(c3cccc(OC)c3)c(=O)c4sccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L17 compound treatment 1000.0 62.5 0.02 600.0 7.5 0.01 0.0197 0.8621 3028978 ChemDiv3_008355 Cc1cc(no1)C(=O)Nc2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L18 compound treatment 1240.0 303.0 0.11 360.0 -233.0 -0.18 -0.0503 -0.2417 3123161 ChemDiv3_008356 CCOc1ccc(cc1)n2c(=O)n(CC(=O)Nc3cccc(c3)C(F)(F)F)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L19 compound treatment 520.0 -418.0 -0.15 760.0 168.0 0.13 -0.0138 -0.0703 3028979 ChemDiv3_008357 CC(C)NC(=O)c1cc(on1)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L20 compound treatment 640.0 -298.0 -0.11 2880.0 2290.0 1.76 1.1672 0.6634 3123162 ChemDiv3_008358 CC(C)(C)C(=O)Cn1c(=O)n(CCCC(=O)NCc2ccco2)c(=O)c3sccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L21 compound treatment 1200.0 263.0 0.09 600.0 7.5 0.01 0.0699 0.7494 3028980 ChemDiv3_008359 O=C(NCCCn1ccnc1)c2noc3CCCCc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L22 compound treatment 1000.0 62.5 0.02 520.0 -72.5 -0.06 -0.0237 -0.3952 3123163 ChemDiv3_008360 COc1cc(OC)cc(c1)n2c(=O)n(CC(=O)c3ccc(Cl)cc3)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L23 mock treatment 440.0 -498.0 -0.18 560.0 -32.5 -0.02 -0.1424 -0.7991 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 L24 mock treatment 720.0 -218.0 -0.08 1600.0 1010.0 0.77 0.4924 0.6334 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M01 compound treatment 5040.0 4100.0 1.46 1000.0 408.0 0.31 1.2503 0.8399 3028981 ChemDiv3_008361 CN1C(=O)/C(=C(\O)/C=C/c2ccc(C)cc2)/C3CC1(C)Oc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M02 compound treatment 520.0 -418.0 -0.15 320.0 -273.0 -0.21 -0.2527 -0.9857 3123164 ChemDiv3_008362 CCOc1ccccc1C2C(=C(C)Nc3nc4ccccc4n23)C(=O)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M03 compound treatment 440.0 -498.0 -0.18 600.0 7.5 0.01 -0.1207 -0.6837 3028982 ChemDiv3_008363 O=c1n(Cc2ccccc2)c(=O)c3ccccc3n1Cc4ccccc4C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M04 compound treatment 440.0 -498.0 -0.18 1680.0 1090.0 0.83 0.4656 0.5456 3123165 ChemDiv3_008364 NC(=O)C1C(C=C(NC1=O)c2ccccc2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M05 compound treatment 320.0 -618.0 -0.22 400.0 -193.0 -0.15 -0.2594 -0.9816 3028983 ChemDiv3_008365 CCCN1C(=S)NC2C(C)C1(C)Oc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M06 compound treatment 360.0 -578.0 -0.2 560.0 -32.5 -0.02 -0.1625 -0.7874 3123166 ChemDiv3_008366 CCC1Oc2ccc(C)cc2N(CC(=O)NCC3COc4ccccc4O3)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M07 compound treatment 280.0 -658.0 -0.23 960.0 368.0 0.28 0.0346 0.0944 3123167 ChemDiv3_008367 COC(=O)c1ccc2c(=O)n(c(Nc3ccccc3)nc2c1)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M08 compound treatment 360.0 -578.0 -0.2 520.0 -72.5 -0.06 -0.1842 -0.8678 3028984 ChemDiv3_008368 CCC(C)NS(=O)(=O)c1cccs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M09 compound treatment 840.0 -97.5 -0.03 360.0 -233.0 -0.18 -0.1507 -0.8287 3028985 ChemDiv3_008369 CCN(CC)C(=S)Nc1cc(ccc1C(=O)OC)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M10 compound treatment 520.0 -418.0 -0.15 320.0 -273.0 -0.21 -0.2527 -0.9857 3123168 ChemDiv3_008370 CC1CCc2ccc(F)cc2N1S(=O)(=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M11 compound treatment 360.0 -578.0 -0.2 680.0 87.5 0.07 -0.0974 -0.4516 3123169 ChemDiv3_008371 O=C(CCCn1c(=O)c2sc3ccccc3c2[nH]c1=S)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M12 compound treatment 520.0 -418.0 -0.15 840.0 248.0 0.19 0.0296 0.123 3028986 ChemDiv3_008372 Fc1ccc(cc1)N2CCN(CCCNC(=O)CCn3c(=O)oc4ccccc34)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M13 compound treatment 720.0 -218.0 -0.08 520.0 -72.5 -0.06 -0.0939 -0.9872 1074952 ChemDiv3_008373 Nc1c(nnn1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M14 compound treatment 600.0 -338.0 -0.12 400.0 -193.0 -0.15 -0.1892 -0.9945 3029045 ChemDiv3_008374 O=C(COc1ccc2OC3(CCCCC3)CC(=O)c2c1)NCc4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M15 compound treatment 720.0 -218.0 -0.08 2320.0 1730.0 1.33 0.8832 0.6648 3029046 ChemDiv3_008375 O=C1CCC(=O)N1Nc2nc3ccccc3c4nc(nn24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M16 compound treatment 360.0 -578.0 -0.2 1400.0 808.0 0.62 0.2935 0.4495 3029047 ChemDiv3_008376 CCCCn1cnc2cc(NCc3ccc(Br)cc3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M17 compound treatment 480.0 -458.0 -0.16 640.0 47.5 0.04 -0.089 -0.5349 3029048 ChemDiv3_008377 Clc1nc2c(nnn2c3ccccc13)S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M18 compound treatment 280.0 -658.0 -0.23 560.0 -32.5 -0.02 -0.1826 -0.7783 3029049 ChemDiv3_008378 CC(C)(C)n1cnc2cc(NCc3ccccn3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M19 compound treatment 560.0 -378.0 -0.13 680.0 87.5 0.07 -0.0472 -0.315 1548756 ChemDiv3_008379 CCOC(=O)CC(=O)Nc1ccsc1C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M20 compound treatment 920.0 -17.5 -0.01 640.0 47.5 0.04 0.0214 0.5784 3029050 ChemDiv3_008380 Cc1ccc(C)c(c1)N2CCN(CC2)S(=O)(=O)c3ccc4NC(=O)CCc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M21 compound treatment 4040.0 3100.0 1.1 600.0 7.5 0.01 0.7823 0.7108 3123170 ChemDiv3_008381 Cc1ccc(cc1)c2csc(n2)c3ccccc3N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M22 compound treatment 880.0 -57.5 -0.02 600.0 7.5 0.01 -0.0104 -0.4884 1619066 ChemDiv3_008382 O=S(=O)(NC1CCCC1)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M23 mock treatment 760.0 -178.0 -0.06 760.0 168.0 0.13 0.0464 0.3241 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 M24 mock treatment 1000.0 62.5 0.02 1200.0 608.0 0.47 0.3455 0.7399 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N01 compound treatment 840.0 -97.5 -0.03 480.0 -113.0 -0.09 -0.0855 -0.9193 3029051 ChemDiv3_008383 CC1CC(C)CN(CCCNS(=O)(=O)c2cccc3cccnc23)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N02 compound treatment 800.0 -138.0 -0.05 360.0 -233.0 -0.18 -0.1607 -0.8685 3123171 ChemDiv3_008384 O=C(NCCc1ccccc1)c2noc-3c2CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N03 compound treatment 400.0 -538.0 -0.19 520.0 -72.5 -0.06 -0.1742 -0.8769 3123172 ChemDiv3_008385 CCOc1ccc(NC(=O)CCNS(=O)(=O)c2ccc(Br)s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N04 compound treatment 1520.0 583.0 0.21 280.0 -313.0 -0.24 -0.0235 -0.0743 3029052 ChemDiv3_008386 COc1ccc2-c3onc(C(=O)N4CCCC4)c3CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N05 compound treatment 680.0 -258.0 -0.09 520.0 -72.5 -0.06 -0.1039 -0.9718 3123173 ChemDiv3_008387 O=C(CCS(=O)(=O)c1cccs1)Nc2ccc(cc2)C(=O)NCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N06 compound treatment 320.0 -618.0 -0.22 720.0 128.0 0.1 -0.0857 -0.3571 3029053 ChemDiv3_008388 COc1cccc(c1)c2cc(nc(n2)n3cc(C)c(=O)[nH]c3=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N07 compound treatment 280.0 -658.0 -0.23 560.0 -32.5 -0.02 -0.1826 -0.7783 3123174 ChemDiv3_008389 Oc1ccc(cc1)c2cc(no2)C(=O)N3CCN(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N08 compound treatment 280.0 -658.0 -0.23 760.0 168.0 0.13 -0.074 -0.2778 3123353 ChemDiv3_008390 COc1ccccc1N2C(=O)C3C(NC(Cc4ccccc4)(C3C2=O)C(=O)O)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N09 compound treatment 440.0 -498.0 -0.18 1160.0 568.0 0.44 0.1833 0.3899 3029054 ChemDiv3_008391 COc1cccc(c1)c2cc(no2)C(=O)N(C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N10 compound treatment 480.0 -458.0 -0.16 760.0 168.0 0.13 -0.0238 -0.1151 3123354 ChemDiv3_008392 CCOc1ccc(CCNC(=O)c2cn(CC(C)C)c(=O)c3n(C)c4ccccc4c23)cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N11 compound treatment 720.0 -218.0 -0.08 760.0 168.0 0.13 0.0364 0.2425 3029055 ChemDiv3_008393 CCOC(=O)c1c(NC(=O)c2cc(on2)c3ccc4OCOc4c3)sc5CCCCc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N12 compound treatment 840.0 -97.5 -0.03 560.0 -32.5 -0.02 -0.0421 -0.9872 3123355 ChemDiv3_008394 NNC(=O)CNc1c(nc2ccccn12)c3ccsc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N13 compound treatment 1640.0 703.0 0.25 640.0 47.5 0.04 0.202 0.802 3029056 ChemDiv3_008395 O=C(N1CCCc2ccccc12)c3cc(on3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N14 compound treatment 760.0 -178.0 -0.06 680.0 87.5 0.07 0.003 0.0323 3123356 ChemDiv3_008396 CN(C1CCCCC1)C(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N15 compound treatment 920.0 -17.5 -0.01 600.0 7.5 0.01 -3.0E-4 -0.0376 3029057 ChemDiv3_008397 CC(C)CNC(=O)c1cc(on1)c2ccccc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N16 compound treatment 960.0 22.5 0.01 1520.0 928.0 0.71 0.5091 0.715 3123357 ChemDiv3_008398 CCOc1ccc(cc1)n2c(=O)n(CC(=O)NC3CCCC3)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N17 compound treatment 840.0 -97.5 -0.03 800.0 208.0 0.16 0.0882 0.541 3029058 ChemDiv3_008399 O=C(NCc1ccccc1)c2cc(on2)C3CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N18 compound treatment 720.0 -218.0 -0.08 560.0 -32.5 -0.02 -0.0722 -0.8904 3123358 ChemDiv3_008400 Cc1ccc(cc1F)n2c(=O)n(CC(=O)c3ccc(Br)cc3)c4ccsc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N19 compound treatment 680.0 -258.0 -0.09 680.0 87.5 0.07 -0.0171 -0.1507 3029059 ChemDiv3_008401 CC(C)c1cc(no1)C(=O)Nc2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N20 compound treatment 1600.0 663.0 0.24 1000.0 408.0 0.31 0.3874 0.9901 3123359 ChemDiv3_008402 COc1ccc(CNC(=O)CCn2c(=O)n(Cc3cc(C)ccc3C)c4ccsc4c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N21 compound treatment 560.0 -378.0 -0.13 800.0 208.0 0.16 0.0179 0.0863 3029060 ChemDiv3_008403 O=C(N1CCCCC1)c2noc3CCCCc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N22 compound treatment 720.0 -218.0 -0.08 800.0 208.0 0.16 0.0581 0.3282 3123360 ChemDiv3_008404 O=C(NCc1ccco1)c2ccc(Cn3c(=O)n(Cc4ccccc4C#N)c5ccsc5c3=O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N23 mock treatment 600.0 -338.0 -0.12 640.0 47.5 0.04 -0.0589 -0.4704 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 N24 mock treatment 760.0 -178.0 -0.06 680.0 87.5 0.07 0.003 0.0323 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O01 compound treatment 440.0 -498.0 -0.18 240.0 -353.0 -0.27 -0.3162 -0.9785 3029061 ChemDiv3_008405 CC1(CC2NC(=O)N1Cc3ccccc3)Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O02 compound treatment 320.0 -618.0 -0.22 480.0 -113.0 -0.09 -0.216 -0.9172 3123361 ChemDiv3_008406 CC1=C(C(c2ccc(Br)cc2)n3c(N1)nc4ccccc34)C(=O)N5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O03 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3123362 ChemDiv3_008407 CC(NC(=O)CCCn1c(=O)[nH]c2ccsc2c1=O)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O04 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 3029062 ChemDiv3_008408 NC1=NC(CC(=O)N1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O05 compound treatment 360.0 -578.0 -0.2 240.0 -353.0 -0.27 -0.3362 -0.9906 3029063 ChemDiv3_008409 COc1ccc(NC(=O)Cn2c(cn(c3ccc(C)cc3)c2=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O06 compound treatment 240.0 -698.0 -0.25 280.0 -313.0 -0.24 -0.3446 -0.9999 3123363 ChemDiv3_008410 CC(C)Cc1ccc(cc1)S(=O)(=O)NC2CCCCC2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O07 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3123364 ChemDiv3_008411 O=c1sc(nc2ccsc12)N3CCN(CC3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O08 compound treatment 280.0 -658.0 -0.23 240.0 -353.0 -0.27 -0.3563 -0.9973 3029064 ChemDiv3_008412 CC(C)(C)NS(=O)(=O)c1cccs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O09 compound treatment 240.0 -698.0 -0.25 360.0 -233.0 -0.18 -0.3012 -0.9872 3029065 ChemDiv3_008413 COC(=O)c1sccc1NC(=S)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O10 compound treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 1674734 ChemDiv3_008414 NC(=O)c1ccccc1NS(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O11 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3123365 ChemDiv3_008415 CCOC(=O)c1ccccc1NC(=S)N(C)Cc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O12 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3029066 ChemDiv3_008416 O=C(NC1CCCC1)c2cc(=O)[nH]c3ccc(cc23)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O13 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3123366 ChemDiv3_008417 Cc1cccc(C)c1NC2=NC3CS(=O)(=O)CC3S2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O14 compound treatment 320.0 -618.0 -0.22 320.0 -273.0 -0.21 -0.3028 -0.9997 3123367 ChemDiv3_008418 Cc1ccc(CNC(=O)COc2ccc3OC4(CCCCC4)CC(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O15 compound treatment 280.0 -658.0 -0.23 440.0 -153.0 -0.12 -0.2477 -0.9492 3029067 ChemDiv3_008419 O=c1[nH]c2ccccc2c3nc(nn13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O16 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3123368 ChemDiv3_008420 CCc1ccc(CNc2ccc3n(C)cnc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O17 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 3029068 ChemDiv3_008421 CN(Cc1ccccc1)c2nc3c(nnn3c4ccccc24)S(=O)(=O)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O18 compound treatment 320.0 -618.0 -0.22 680.0 87.5 0.07 -0.1074 -0.4687 3123369 ChemDiv3_008422 CCCn1cnc2cc(NCc3cccs3)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O19 compound treatment 320.0 -618.0 -0.22 360.0 -233.0 -0.18 -0.2811 -0.9948 3123370 ChemDiv3_008423 Fc1ccc(Cn2c(=O)c3ccccc3n4c(=O)[nH]nc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O20 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3029069 ChemDiv3_008424 CCc1cccc(NS(=O)(=O)c2ccc3NC(=O)CCc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O21 compound treatment 480.0 -458.0 -0.16 280.0 -313.0 -0.24 -0.2844 -0.9819 3123371 ChemDiv3_008425 Cc1ccc(NC(=O)CSC2=NC3(CCCCC3)Nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O22 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3029070 ChemDiv3_008426 COC(CN(C)S(=O)(=O)c1cccc2cccnc12)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O23 mock treatment 4480.0 3540.0 1.26 360.0 -233.0 -0.18 0.7624 0.6006 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 O24 mock treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P01 compound treatment 320.0 -618.0 -0.22 280.0 -313.0 -0.24 -0.3245 -0.999 3123372 ChemDiv3_008427 CCOc1ccccc1N(C)S(=O)(=O)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P02 compound treatment 280.0 -658.0 -0.23 280.0 -313.0 -0.24 -0.3346 -0.9999 3029071 ChemDiv3_008428 O=C(NCc1ccccc1)c2noc-3c2CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P03 compound treatment 360.0 -578.0 -0.2 320.0 -273.0 -0.21 -0.2928 -0.9999 3123373 ChemDiv3_008429 COc1ccc(cc1)N2CCN(CC2)C(=O)CCNS(=O)(=O)c3ccc(Br)s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P04 compound treatment 360.0 -578.0 -0.2 240.0 -353.0 -0.27 -0.3362 -0.9906 3123374 ChemDiv3_008430 COc1ccc2-c3onc(C(=O)N(C)c4ccccc4)c3CCc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P05 compound treatment 320.0 -618.0 -0.22 440.0 -153.0 -0.12 -0.2377 -0.9569 3029072 ChemDiv3_008431 Cn1c2ccccc2c3c(cn(C)c(=O)c13)C(=O)NCCCN4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P06 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3123375 ChemDiv3_008432 FC(F)(F)c1cc(nc(n1)n2cccn2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P07 compound treatment 400.0 -538.0 -0.19 320.0 -273.0 -0.21 -0.2828 -0.9989 3029073 ChemDiv3_008433 CC(C)NC(=O)c1cc(on1)c2ccc(O)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P08 compound treatment 720.0 -218.0 -0.08 280.0 -313.0 -0.24 -0.2242 -0.8896 3123376 ChemDiv3_008434 COc1ccc(cc1)C2NC(CC(C)C)(C3C2C(=O)N(C3=O)c4ccccc4OC)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P09 compound treatment 360.0 -578.0 -0.2 360.0 -233.0 -0.18 -0.2711 -0.9976 3029074 ChemDiv3_008435 COc1cccc(c1)c2cc(no2)C(=O)NC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P10 compound treatment 280.0 -658.0 -0.23 240.0 -353.0 -0.27 -0.3563 -0.9973 3123377 ChemDiv3_008436 CC(C)CCNC(=O)c1cn(CC(C)C)c(=O)c2n(C)c3ccccc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P11 compound treatment 280.0 -658.0 -0.23 320.0 -273.0 -0.21 -0.3129 -0.9985 3123378 ChemDiv3_008437 Cc1nn(Cc2ccc(F)cc2)c(C)c1NC(=O)c3cc(on3)c4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P12 compound treatment 400.0 -538.0 -0.19 280.0 -313.0 -0.24 -0.3045 -0.9935 3029075 ChemDiv3_008438 CC(C)c1ccc(Nc2c(nc3[nH]cnn23)c4ccc(cc4)N(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P13 compound treatment 280.0 -658.0 -0.23 920.0 328.0 0.25 0.0129 0.0375 3029076 ChemDiv3_008439 CC(C)CNC(=O)c1cc(on1)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P14 compound treatment 320.0 -618.0 -0.22 360.0 -233.0 -0.18 -0.2811 -0.9948 3120512 ChemDiv3_008440 CCOC(=O)C1CCN(CC1)C(=O)C2C3N(CCc4ccccc34)C(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P15 compound treatment 360.0 -578.0 -0.2 400.0 -193.0 -0.15 -0.2494 -0.9872 3029077 ChemDiv3_008441 CCN(CC)C(=O)c1cc(on1)c2ccccc2O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P16 compound treatment 360.0 -578.0 -0.2 440.0 -153.0 -0.12 -0.2276 -0.9648 3120313 ChemDiv3_008442 FC(F)(F)c1cccc(c1)n2c(=O)n(CC(=O)N3CCCc4ccccc34)c5ccsc5c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P17 compound treatment 480.0 -458.0 -0.16 280.0 -313.0 -0.24 -0.2844 -0.9819 3029078 ChemDiv3_008443 CCC(C)NC(=O)c1cc(on1)C2CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P18 compound treatment 6760.0 5820.0 2.07 240.0 -353.0 -0.27 1.2692 0.6093 3120314 ChemDiv3_008444 Cc1cccc(NC(=O)Cn2c(=O)n(c3ccc(F)cc3)c(=O)c4sccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P19 compound treatment 320.0 -618.0 -0.22 240.0 -353.0 -0.27 -0.3463 -0.9945 3029079 ChemDiv3_008445 CCCc1cc(no1)C(=O)N(C2CCCCC2)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P20 compound treatment 160.0 -778.0 -0.28 240.0 -353.0 -0.27 -0.3864 -1.0 3120315 ChemDiv3_008446 COc1ccc(CNC(=O)CCn2c(=O)n(CC(=O)N3CCCCC3C)c4ccsc4c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P21 compound treatment 1840.0 903.0 0.32 280.0 -313.0 -0.24 0.0567 0.1418 3029080 ChemDiv3_008447 O=C(N(C1CCCCC1)C2CCCCC2)c3noc4CCCCc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P22 compound treatment 400.0 -538.0 -0.19 280.0 -313.0 -0.24 -0.3045 -0.9935 3120316 ChemDiv3_008448 Cc1ccc(CNC(=O)Cc2ccc(cc2)n3c(=O)n(Cc4ccccc4)c5ccsc5c3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P23 mock treatment 360.0 -578.0 -0.2 400.0 -193.0 -0.15 -0.2494 -0.9872 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2024 P24 mock treatment 480.0 -458.0 -0.16 200.0 -393.0 -0.3 -0.3278 -0.9579 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A01 compound treatment 5080.0 3840.0 1.36 600.0 -286.0 -0.22 0.8079 0.5857 3120317 ChemDiv3_008449 O=C(Cc1ccc(cc1)n2c(=O)n(Cc3ccccc3C#N)c4ccsc4c2=O)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A02 compound treatment 4000.0 2760.0 0.98 3160.0 2270.0 1.75 1.9267 0.9625 3029081 ChemDiv3_008450 CN(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A03 compound treatment 3280.0 2040.0 0.72 520.0 -366.0 -0.28 0.313 0.4034 3029082 ChemDiv3_008451 O=C(Nc1ccccc1)c2cc3c(=O)n4ccccc4nc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A04 compound treatment 760.0 -481.0 -0.17 360.0 -526.0 -0.4 -0.406 -0.9268 3029144 ChemDiv3_008452 CCN(Cc1ccccc1)C(=O)Cn2c(=O)n(c3ccc(C)cc3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A05 compound treatment 320.0 -921.0 -0.33 200.0 -686.0 -0.53 -0.6032 -0.9737 1281503 ChemDiv3_008453 CCCCn1c(=O)c2ccccc2c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A06 compound treatment 440.0 -801.0 -0.28 320.0 -566.0 -0.43 -0.508 -0.9789 3029145 ChemDiv3_008454 O=C(CCn1c(=O)n(Cc2ccccc2)c3ccccc3c1=O)NCc4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A07 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029146 ChemDiv3_008455 COC(=O)CSc1nnc(CNC(=O)c2cccs2)n1c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A08 compound treatment 280.0 -961.0 -0.34 360.0 -526.0 -0.4 -0.5264 -0.9965 3029147 ChemDiv3_008456 Fc1ccc(cc1)C(=O)Cn2c(=O)n(CCCC(=O)NC3CCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A09 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3029148 ChemDiv3_008457 CC1(CC2/C(=C(/O)\C=C\c3ccccc3)/C(=O)N1)Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A10 compound treatment 520.0 -721.0 -0.26 280.0 -606.0 -0.46 -0.5096 -0.9604 3120318 ChemDiv3_008458 CN(C1CCCCC1)C(=O)Cn2c(=O)n(CCC(=O)NCCc3ccccc3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A11 compound treatment 1040.0 -201.0 -0.07 320.0 -566.0 -0.43 -0.3575 -0.8125 3029149 ChemDiv3_008459 O=C/1/C(=C/c2cccnc2)/CS\C1=C/c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A12 compound treatment 400.0 -841.0 -0.3 4520.0 3630.0 2.79 1.762 0.6279 3120319 ChemDiv3_008460 CCCCN(CC)C(=O)Cn1c(=O)n(Cc2ccccc2Cl)c(=O)c3cc(OC)c(OC)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A13 compound treatment 560.0 -681.0 -0.24 360.0 -526.0 -0.4 -0.4562 -0.97 3029150 ChemDiv3_008461 CCCSC1=N/C(=C/c2cccs2)/C(=O)N1c3ccc(F)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A14 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3120320 ChemDiv3_008462 CCc1ccc(NS(=O)(=O)c2ccc3[nH]c(nc3c2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A15 compound treatment 3640.0 2400.0 0.85 320.0 -566.0 -0.43 0.2947 0.3085 3120321 ChemDiv3_008463 CC1(C)N=C(SCC(=O)Nc2ccccc2)C(=N1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A16 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3029151 ChemDiv3_008464 CCOC(=O)c1ccc(NC(=O)CSc2nccn2c3cccc(C)c3C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A17 compound treatment 840.0 -401.0 -0.14 520.0 -366.0 -0.28 -0.2991 -0.9505 3120322 ChemDiv3_008465 Clc1ccc(cc1)C(=O)CSC2=NN3CCCC(=O)N=C3S2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A18 compound treatment 360.0 -881.0 -0.31 1160.0 274.0 0.21 -0.0721 -0.1911 3120323 ChemDiv3_008466 CCN1CCN(CC1)c2cc(C)c3cc(NC(=S)N(C)Cc4ccccc4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A19 compound treatment 320.0 -921.0 -0.33 440.0 -446.0 -0.34 -0.473 -0.9997 3029152 ChemDiv3_008467 Clc1ccc(cc1)S(=O)(=O)C2(CC2)C(=O)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A20 compound treatment 560.0 -681.0 -0.24 360.0 -526.0 -0.4 -0.4562 -0.97 3120324 ChemDiv3_008468 CC1CCCC(C)N1CCNC(=O)Nc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A21 compound treatment 520.0 -721.0 -0.26 360.0 -526.0 -0.4 -0.4662 -0.9759 3029153 ChemDiv3_008469 CCN(CC)C(=O)Cn1c(=O)n(Cc2ccccc2)c(=O)c3c4CCCc4sc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A22 compound treatment 520.0 -721.0 -0.26 320.0 -566.0 -0.43 -0.4879 -0.9682 3120325 ChemDiv3_008470 Clc1ccc(NC(=O)NCCN2CCN(CC2)c3cccc(Cl)c3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A23 mock treatment 360.0 -881.0 -0.31 1040.0 154.0 0.12 -0.1372 -0.4103 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 A24 mock treatment 280.0 -961.0 -0.34 480.0 -406.0 -0.31 -0.4613 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B01 compound treatment 360.0 -881.0 -0.31 3760.0 2870.0 2.21 1.3394 0.6009 3120326 ChemDiv3_008471 C(C1COC(O1)(c2ccccc2)c3ccccc3)n4cncn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B02 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 3029154 ChemDiv3_008472 Fc1ccc(cc1)C(=O)NCCn2ccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B03 compound treatment 280.0 -961.0 -0.34 6440.0 5550.0 4.26 2.7742 0.6485 3120327 ChemDiv3_008473 CC(C)CCNC(=O)C1C(N(C)C(=O)c2ccccc12)c3cn(C)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B04 compound treatment 360.0 -881.0 -0.31 3400.0 2510.0 1.93 1.1439 0.585 3029155 ChemDiv3_008474 Cc1cc2ccccc2n1CCNC(=O)C3(CCCC3)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B05 compound treatment 280.0 -961.0 -0.34 320.0 -566.0 -0.43 -0.5481 -0.9929 3120328 ChemDiv3_008475 Brc1ccc(s1)S(=O)(=O)NC(C(=O)N2CCOCC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B06 compound treatment 920.0 -321.0 -0.11 320.0 -566.0 -0.43 -0.3876 -0.8635 1299511 ChemDiv3_008476 CC1CCCC(N1C(=O)CCS)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B07 compound treatment 280.0 -961.0 -0.34 240.0 -646.0 -0.5 -0.5916 -0.9834 3120329 ChemDiv3_008477 COc1ccc2nc(NC(=O)C3CCCN(C3)S(=O)(=O)c4cccc5nonc45)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B08 compound treatment 200.0 -1040.0 -0.37 800.0 -85.5 -0.07 -0.3076 -0.8199 3029156 ChemDiv3_008478 CCOC(=O)C1C(CC(=CC1=O)c2cccc(OC)c2)c3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B09 compound treatment 240.0 -1000.0 -0.36 440.0 -446.0 -0.34 -0.493 -0.9998 3120330 ChemDiv3_008479 Clc1ccccc1CN2COc3cc4OCOc4cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B10 compound treatment 200.0 -1040.0 -0.37 200.0 -686.0 -0.53 -0.6333 -0.985 3120331 ChemDiv3_008480 CC1CC(C)CN(C1)C(=O)Cc2c([nH]c3ccc(Cl)cc23)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B11 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029157 ChemDiv3_008481 COC(=O)C1C(C)Cc2[nH]c(C(=O)OC(C)C)c(C)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B12 compound treatment 360.0 -881.0 -0.31 640.0 -246.0 -0.19 -0.3543 -0.9707 3120332 ChemDiv3_008482 CC1CC(C)CN(C1)C(=O)CSc2nnc(o2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B13 compound treatment 320.0 -921.0 -0.33 2320.0 1430.0 1.1 0.5476 0.4767 3029158 ChemDiv3_008483 CCCc1c([nH]c2CC(C)(C)CC(=O)c12)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B14 compound treatment 320.0 -921.0 -0.33 320.0 -566.0 -0.43 -0.5381 -0.9902 3120333 ChemDiv3_008484 CCOC(=O)N1CCN(CC1)C(=O)CSc2nnc(COc3ccc(Cl)cc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B15 compound treatment 320.0 -921.0 -0.33 800.0 -85.5 -0.07 -0.2775 -0.8325 3029159 ChemDiv3_008485 Cc1cccc(c1)C2CC(=O)NC3=C2C(=O)CC(C3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B16 compound treatment 320.0 -921.0 -0.33 4040.0 3150.0 2.42 1.4813 0.6062 3120334 ChemDiv3_008486 COc1ccc(OC)c(c1)C(N2CCN(CC2)c3ccccc3)c4c(O)[nH]c(=S)[nH]c4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B17 compound treatment 400.0 -841.0 -0.3 2160.0 1270.0 0.98 0.4808 0.47 3120335 ChemDiv3_008487 Cc1cc2cc(CCNC(=O)/C=C\c3ccccc3)c(=O)[nH]c2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B18 compound treatment 680.0 -561.0 -0.2 720.0 -166.0 -0.13 -0.2306 -0.9765 3029160 ChemDiv3_008488 CCOc1ccc(cc1)C(=O)/C=C(/Nc2cccc(C)c2)\C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B19 compound treatment 320.0 -921.0 -0.33 6440.0 5550.0 4.26 2.7842 0.651 3120336 ChemDiv3_008489 COc1cc(/C=C\C(=O)NCCc2cc3ccc(C)cc3[nH]c2=O)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B20 compound treatment 240.0 -1000.0 -0.36 400.0 -486.0 -0.37 -0.5147 -0.9997 3029161 ChemDiv3_008490 O=C(/C=C/1\Nc2ccccc2NC1=O)c3ccc(cc3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B21 compound treatment 880.0 -361.0 -0.13 5680.0 4790.0 3.68 2.5121 0.6821 3120337 ChemDiv3_008491 COc1ccc(cc1)S(=O)(=O)NCCc2cc3ccc(OC)cc3[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B22 compound treatment 480.0 -761.0 -0.27 320.0 -566.0 -0.43 -0.498 -0.9739 3029162 ChemDiv3_008492 O=C(/C=C\1/Nc2ccccc2NC1=O)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B23 mock treatment 520.0 -721.0 -0.26 520.0 -366.0 -0.28 -0.3794 -0.9989 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 B24 mock treatment 360.0 -881.0 -0.31 360.0 -526.0 -0.4 -0.5063 -0.9921 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C01 compound treatment 760.0 -481.0 -0.17 3520.0 2630.0 2.02 1.3094 0.6451 3120338 ChemDiv3_008493 NC(=O)Cn1c(=O)n(CCC(=O)NCCc2ccc(Cl)cc2)c(=O)c3sccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C02 compound treatment 360.0 -881.0 -0.31 360.0 -526.0 -0.4 -0.5063 -0.9921 3029163 ChemDiv3_008494 CN(CC(=O)NCc1ccc(C)cc1)S(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C03 compound treatment 320.0 -921.0 -0.33 2200.0 1310.0 1.01 0.4825 0.4548 3120513 ChemDiv3_008495 CN(Cc1ccccc1)C(=O)c2cc3c(=O)n4cccc(C)c4nc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C04 compound treatment 240.0 -1000.0 -0.36 400.0 -486.0 -0.37 -0.5147 -0.9997 3120514 ChemDiv3_008496 COc1cc(cc(OC)c1OC)n2c(=O)n(CC(=O)NCc3ccc(C)cc3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C05 compound treatment 280.0 -961.0 -0.34 440.0 -446.0 -0.34 -0.483 -1.0 1065885 ChemDiv3_008497 O=c1n(c2ccccc2)c(=O)c3ccccc3c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C06 compound treatment 280.0 -961.0 -0.34 320.0 -566.0 -0.43 -0.5481 -0.9929 3120515 ChemDiv3_008498 O=C(CCCCn1c(=O)n(Cc2ccccc2C#N)c3ccccc3c1=O)NCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C07 compound treatment 240.0 -1000.0 -0.36 240.0 -646.0 -0.5 -0.6016 -0.9867 3029164 ChemDiv3_008499 COC(=O)CSc1nnc(CNC(=O)c2ccccc2OC)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C08 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3120516 ChemDiv3_008500 O=C(CCn1c(=O)n(CC(=O)NCc2ccco2)c3ccccc3c1=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C09 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3120517 ChemDiv3_008501 COc1ccc(/C=C/C(=C/2\C3C4CCCCC4(NC2=O)Oc5ccccc35)/O)c(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C10 compound treatment 520.0 -721.0 -0.26 480.0 -406.0 -0.31 -0.4011 -0.9953 3029165 ChemDiv3_008502 O=C(CCn1c(=O)n(CC(=O)Nc2ccccc2)c3ccccc3c1=O)NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C11 compound treatment 360.0 -881.0 -0.31 280.0 -606.0 -0.46 -0.5498 -0.9814 3029166 ChemDiv3_008503 COc1ccc(cc1)N2C(=O)/C(=C/c3ccccc3)/N=C2SCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C12 compound treatment 280.0 -961.0 -0.34 360.0 -526.0 -0.4 -0.5264 -0.9965 3120518 ChemDiv3_008504 Brc1ccc(NC(=O)Cn2c(=O)n(CC(=O)NC3CCCC3)c(=O)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C13 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3120519 ChemDiv3_008505 CCOC(=O)CSC1=N/C(=C/c2ccsc2)/C(=O)N1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C14 compound treatment 400.0 -841.0 -0.3 280.0 -606.0 -0.46 -0.5397 -0.977 1371701 ChemDiv3_008506 Cc1ccc(C)c(c1)N2CCN(CC2)S(=O)(=O)c3ccc4[nH]c(nc4c3)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C15 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3120520 ChemDiv3_008507 O=C(N1C(=S)C(=NC21CCCC2)c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C16 compound treatment 280.0 -961.0 -0.34 440.0 -446.0 -0.34 -0.483 -1.0 3120521 ChemDiv3_008508 COc1cccc(c1)n2ccnc2SCC(=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C17 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3029167 ChemDiv3_008509 CCOc1ccc2nc(NC(=O)C3(CC3)S(=O)(=O)c4ccc(C)cc4)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C18 compound treatment 240.0 -1000.0 -0.36 320.0 -566.0 -0.43 -0.5582 -0.995 3120522 ChemDiv3_008510 CCOc1ccc(cc1)N(CC)C(=S)Nc2ccc3nc(cc(C)c3c2)N4CCN(CC)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C19 compound treatment 360.0 -881.0 -0.31 360.0 -526.0 -0.4 -0.5063 -0.9921 3029168 ChemDiv3_008511 Clc1ccc(cc1)S(=O)(=O)C2(CC2)C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C20 compound treatment 360.0 -881.0 -0.31 400.0 -486.0 -0.37 -0.4846 -0.9962 3120523 ChemDiv3_008512 Fc1ccc(NC(=S)NCCCN2CCCCCC2)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C21 compound treatment 240.0 -1000.0 -0.36 440.0 -446.0 -0.34 -0.493 -0.9998 3120524 ChemDiv3_008513 Cc1ccc(Cn2c(=O)n(Cc3ccccc3)c(=O)c4c5CCCc5sc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C22 compound treatment 320.0 -921.0 -0.33 2880.0 1990.0 1.53 0.8516 0.5439 3029169 ChemDiv3_008514 Cc1cccc(N2CCN(CCNC(=S)Nc3c(C)cccc3C)CC2)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C23 mock treatment 320.0 -921.0 -0.33 400.0 -486.0 -0.37 -0.4947 -0.9979 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 C24 mock treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D01 compound treatment 320.0 -921.0 -0.33 240.0 -646.0 -0.5 -0.5815 -0.9796 1483037 ChemDiv3_008515 OC(=O)CC1(C(=O)c2ccccc2C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D02 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3120525 ChemDiv3_008516 O=C(CC(c1ccccc1)c2ccccc2)NCCn3ccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D03 compound treatment 440.0 -801.0 -0.28 320.0 -566.0 -0.43 -0.508 -0.9789 3120526 ChemDiv3_008517 CN1C(C(C(=O)NCCCN2CCCC2=O)c3ccccc3C1=O)c4cn(C)c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D04 compound treatment 240.0 -1000.0 -0.36 280.0 -606.0 -0.46 -0.5799 -0.9912 3029170 ChemDiv3_008518 CCOc1ccc(CC(=O)NCCn2c(C)cc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D05 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029171 ChemDiv3_008519 Brc1ccc(s1)S(=O)(=O)N2CCC(CC2)C(=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D06 compound treatment 160.0 -1080.0 -0.38 440.0 -446.0 -0.34 -0.5131 -0.9984 3120527 ChemDiv3_008520 CC(=O)N1CCc2cc(Br)cc(c12)S(=O)(=O)CC(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D07 compound treatment 280.0 -961.0 -0.34 2680.0 1790.0 1.38 0.733 0.5165 3120528 ChemDiv3_008521 COc1ccc(CCNC(=O)C2CCCN(C2)S(=O)(=O)c3cccc4nonc34)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D08 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029172 ChemDiv3_008522 CCOC(=O)C1C(CC(=CC1=O)c2ccco2)c3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D09 compound treatment 320.0 -921.0 -0.33 440.0 -446.0 -0.34 -0.473 -0.9997 3120529 ChemDiv3_008523 COc1ccc(CN2COc3ccc(OC)cc3C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D10 compound treatment 360.0 -881.0 -0.31 400.0 -486.0 -0.37 -0.4846 -0.9962 3120530 ChemDiv3_008524 OC(=O)c1[nH]c2ccc(Cl)cc2c1CC(=O)NCC3COc4ccccc4O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D11 compound treatment 240.0 -1000.0 -0.36 320.0 -566.0 -0.43 -0.5582 -0.995 3029173 ChemDiv3_008525 CCOc1ccc(Br)cc1C2CC(=O)Nc3c(C)c(C)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D12 compound treatment 240.0 -1000.0 -0.36 320.0 -566.0 -0.43 -0.5582 -0.995 3120531 ChemDiv3_008526 COc1cccc(c1)c2nnc(SCC(=O)N3CCCC(C)C3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D13 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 3029234 ChemDiv3_008527 CCOc1ccccc1C2CC(=O)Nc3c2c(=O)n(C)c(=O)n3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D14 compound treatment 360.0 -881.0 -0.31 320.0 -566.0 -0.43 -0.5281 -0.987 3029235 ChemDiv3_008528 O=C(CSc1nnc(o1)C2COc3ccccc3O2)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D15 compound treatment 440.0 -801.0 -0.28 280.0 -606.0 -0.46 -0.5297 -0.9721 3029236 ChemDiv3_008529 FC(F)(F)c1ccccc1C2CC(=O)NC3=C2C(=O)CC(C3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D16 compound treatment 240.0 -1000.0 -0.36 360.0 -526.0 -0.4 -0.5364 -0.998 3029237 ChemDiv3_008530 COc1cccc(C(N2CCOCC2)c3c(O)[nH]c(=S)[nH]c3=O)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D17 compound treatment 440.0 -801.0 -0.28 320.0 -566.0 -0.43 -0.508 -0.9789 3029238 ChemDiv3_008531 Cc1ccc(cc1)C(=O)NCCc2cc3cc(C)c(C)cc3[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D18 compound treatment 240.0 -1000.0 -0.36 360.0 -526.0 -0.4 -0.5364 -0.998 3029239 ChemDiv3_008532 CCOc1ccc(cc1)C(=O)/C=C(\O)/C(=O)Nc2ccc(cc2)S(=O)(=O)NC(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D19 compound treatment 520.0 -721.0 -0.26 400.0 -486.0 -0.37 -0.4445 -0.9832 3120532 ChemDiv3_008533 CN(C)S(=O)(=O)c1ccc(cc1)C(=O)NCCc2cc3ccc(C)cc3[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D20 compound treatment 280.0 -961.0 -0.34 480.0 -406.0 -0.31 -0.4613 -0.999 3120533 ChemDiv3_008534 COc1cccc(c1)C(=O)/C=C/2\Nc3ccc(cc3NC2=O)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D21 compound treatment 360.0 -881.0 -0.31 3000.0 2110.0 1.62 0.9268 0.5606 3029240 ChemDiv3_008535 CC1Cc2nc(SC/C=C/c3ccccc3)n(C)c(=O)c2S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D22 compound treatment 280.0 -961.0 -0.34 7880.0 6990.0 5.37 3.5559 0.6609 3120534 ChemDiv3_008536 Cc1ccc2nsnc2c1NC(=O)CC3(C[C@H]4C[C@@H]5C[C@H](C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D23 mock treatment 320.0 -921.0 -0.33 4960.0 4070.0 3.13 1.9808 0.6298 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 D24 mock treatment 280.0 -961.0 -0.34 440.0 -446.0 -0.34 -0.483 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E01 compound treatment 3160.0 1920.0 0.68 1960.0 1070.0 0.82 1.0646 0.9954 3029241 ChemDiv3_008537 COc1cccc(c1)n2c(=O)n(CC(=O)NCCC3=CCCCC3)c4sc(C)c(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E02 compound treatment 360.0 -881.0 -0.31 560.0 -326.0 -0.25 -0.3978 -0.9938 3120535 ChemDiv3_008538 CN(CC(=O)Nc1ccc(cc1)C(F)(F)F)S(=O)(=O)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E03 compound treatment 760.0 -481.0 -0.17 720.0 -166.0 -0.13 -0.2106 -0.9894 3120536 ChemDiv3_008539 CCCNC(=O)c1cc2c(=O)n3cccc(C)c3nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E04 compound treatment 640.0 -601.0 -0.21 5960.0 5070.0 3.9 2.6039 0.6674 3029242 ChemDiv3_008540 CCN(Cc1ccccc1)C(=O)Cn2c(=O)n(C3CCCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E05 compound treatment 1520.0 279.0 0.1 1720.0 834.0 0.64 0.5229 0.8067 3120537 ChemDiv3_008541 COC(=O)CSc1nnc(c2ccncc2)n1c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E06 compound treatment 560.0 -681.0 -0.24 800.0 -85.5 -0.07 -0.2173 -0.8677 3120702 ChemDiv3_008542 CCC1CCCCN1C(=O)Cn2c(=O)n(C3CCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E07 compound treatment 360.0 -881.0 -0.31 760.0 -126.0 -0.1 -0.2892 -0.884 3029243 ChemDiv3_008543 COC(=O)CSc1nnc(CNC(=O)c2ccc(cc2)S(=O)(=O)N3CCCCC3)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E08 compound treatment 2040.0 799.0 0.28 1720.0 834.0 0.64 0.6534 0.9327 3120703 ChemDiv3_008544 CCN(C(=O)Cn1c(=O)n(Cc2ccc3OCOc3c2)c(=O)c4ccccc14)c5cccc(C)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E09 compound treatment 1280.0 38.7 0.01 400.0 -486.0 -0.37 -0.2539 -0.6806 3029244 ChemDiv3_008545 FC(F)(F)C(=O)Nc1ccc2nc3c(=O)[nH]c(=O)[nH]c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E10 compound treatment 1000.0 -241.0 -0.09 1680.0 794.0 0.61 0.3708 0.602 3120704 ChemDiv3_008546 Cc1ccc(C)c(Cn2c(=O)n(CCCC(=O)NCc3ccccc3Cl)c(=O)c4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E11 compound treatment 1360.0 119.0 0.04 1400.0 514.0 0.39 0.3091 0.7781 3029245 ChemDiv3_008547 COc1ccccc1/C=C/2\CS/C(=C\c3ccccc3OC)/C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E12 compound treatment 680.0 -561.0 -0.2 1120.0 234.0 0.18 -0.0135 -0.0503 3120705 ChemDiv3_008548 Cc1ccccc1Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E13 compound treatment 640.0 -601.0 -0.21 1080.0 194.0 0.15 -0.0453 -0.1738 3029246 ChemDiv3_008549 CC1(C)NC(=S)C(=N1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E14 compound treatment 2480.0 1240.0 0.44 1760.0 874.0 0.67 0.7854 0.9789 1177109 ChemDiv3_008550 CC1Cc2ccccc2N1S(=O)(=O)c3ccc4[nH]c(nc4c3)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E15 compound treatment 1400.0 159.0 0.06 1080.0 194.0 0.15 0.1454 0.9111 3029247 ChemDiv3_008551 CC1(C)N=C(C(=S)N1C(=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E16 compound treatment 560.0 -681.0 -0.24 800.0 -85.5 -0.07 -0.2173 -0.8677 3120706 ChemDiv3_008552 CCC(=O)Oc1c(c(C)nn1C(C)(C)C)S(=O)(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E17 compound treatment 3720.0 2480.0 0.88 800.0 -85.5 -0.07 0.5753 0.6525 3029248 ChemDiv3_008553 Cc1ccc(CNC(=O)C2(CC2)S(=O)(=O)c3ccc(C)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E18 compound treatment 920.0 -321.0 -0.11 400.0 -486.0 -0.37 -0.3442 -0.883 3120707 ChemDiv3_008554 CCN1CCN(CC1)c2cc(C)c3cc(NC(=S)NCc4ccc(C)cc4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E19 compound treatment 880.0 -361.0 -0.13 1280.0 394.0 0.3 0.1235 0.3756 3120708 ChemDiv3_008555 CC1CCN(CCCNC(=O)C2(CC2)S(=O)(=O)c3ccc(Cl)cc3)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E20 compound treatment 760.0 -481.0 -0.17 680.0 -206.0 -0.16 -0.2323 -0.9992 3029249 ChemDiv3_008556 CCOc1ccc(CCNC(=O)Nc2ccc(C)c(C)c2)cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E21 compound treatment 800.0 -441.0 -0.16 4640.0 3750.0 2.88 1.9275 0.6677 3120709 ChemDiv3_008557 CCC1CCCCN1C(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c4c5CCCc5sc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E22 compound treatment 680.0 -561.0 -0.2 3560.0 2670.0 2.05 1.3111 0.6356 3029250 ChemDiv3_008558 COc1ccc(cc1)N2CCN(CCCNC(=S)Nc3c(C)cccc3C)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E23 mock treatment 800.0 -441.0 -0.16 1120.0 234.0 0.18 0.0166 0.0696 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 E24 mock treatment 2360.0 1120.0 0.4 3560.0 2670.0 2.05 1.7325 0.8284 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F01 compound treatment 2440.0 1200.0 0.43 1000.0 114.0 0.09 0.3628 0.8356 3120710 ChemDiv3_008559 CCOc1ccc(NC(=S)NCCCn2ccnc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F02 compound treatment 480.0 -761.0 -0.27 2640.0 1750.0 1.35 0.7615 0.5543 3120711 ChemDiv3_008560 O=C(NCCn1ccc2ccccc12)c3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F03 compound treatment 1160.0 -81.3 -0.03 2240.0 1350.0 1.04 0.7149 0.6872 1594156 ChemDiv3_008561 CCCCc1nnc(NC(=O)Nc2ccc(C)cc2)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F04 compound treatment 1480.0 239.0 0.08 1160.0 274.0 0.21 0.2089 0.9198 3120712 ChemDiv3_008562 Cc1cc(C)c2c(nn3c(cc(nc23)C(F)(F)F)C4CC4)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F05 compound treatment 800.0 -441.0 -0.16 1440.0 554.0 0.43 0.1903 0.4196 3120713 ChemDiv3_008563 CC(C)c1ccc(NC(=O)C2CCC(CNS(=O)(=O)c3cccs3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F06 compound treatment 1760.0 519.0 0.18 840.0 -45.5 -0.03 0.1054 0.5628 3029251 ChemDiv3_008564 COc1ccc(OC)c(NC(=O)CS(=O)(=O)c2cccc3nsnc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F07 compound treatment 1000.0 -241.0 -0.09 2440.0 1550.0 1.19 0.7833 0.6547 3120714 ChemDiv3_008565 Cc1cccc(N2CCN(CC2)C(=O)C3CCCN(C3)S(=O)(=O)c4cccc5nonc45)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F08 compound treatment 640.0 -601.0 -0.21 1280.0 394.0 0.3 0.0633 0.1709 3029252 ChemDiv3_008566 CCOC(=O)C1C(CC(=CC1=O)c2ccc(C)cc2)c3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F09 compound treatment 880.0 -361.0 -0.13 680.0 -206.0 -0.16 -0.2022 -0.9947 3120715 ChemDiv3_008567 COc1ccccc1C2CC(=O)Nc3cc4CCCc4cc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F10 compound treatment 1160.0 -81.3 -0.03 1840.0 954.0 0.73 0.4978 0.6788 3029253 ChemDiv3_008568 CCN(C(=O)Cc1c([nH]c2ccc(Cl)cc12)C(=O)O)c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F11 compound treatment 520.0 -721.0 -0.26 1280.0 394.0 0.3 0.0332 0.0838 3120716 ChemDiv3_008569 Cc1c([nH]c2CC(CC(=O)c12)c3ccc(cc3)C(C)(C)C)C(=O)Nc4ccc(C)c(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F12 compound treatment 560.0 -681.0 -0.24 7000.0 6110.0 4.69 3.1484 0.6698 3120717 ChemDiv3_008570 CCC1CCCCN1C(=O)CSc2nnc(o2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F13 compound treatment 800.0 -441.0 -0.16 1480.0 594.0 0.46 0.212 0.4394 3029254 ChemDiv3_008571 CCOc1ccccc1C2CC(=O)NC(=C2C(=O)OCC3CCCCC3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F14 compound treatment 480.0 -761.0 -0.27 1280.0 394.0 0.3 0.0232 0.0571 3120718 ChemDiv3_008572 COCCN1C(C(C(=O)NCc2ccco2)c3ccccc3C1=O)c4c[nH]c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F15 compound treatment 1160.0 -81.3 -0.03 1120.0 234.0 0.18 0.1069 0.5864 3029255 ChemDiv3_008573 CCc1ccc(cc1)C2CC(=O)NC3=C2C(=O)CCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F16 compound treatment 720.0 -521.0 -0.18 1520.0 634.0 0.49 0.2137 0.4101 3120719 ChemDiv3_008574 COc1ccccc1C(N(Cc2ccccc2)C(C)C)c3c(O)[nH]c(=S)[nH]c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F17 compound treatment 840.0 -401.0 -0.14 920.0 34.5 0.03 -0.0819 -0.5659 3029256 ChemDiv3_008575 CCC(=O)NCCc1cc2cc(C)c(C)cc2[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F18 compound treatment 360.0 -881.0 -0.31 480.0 -406.0 -0.31 -0.4412 -1.0 3120720 ChemDiv3_008576 Cc1ccc(cc1C)C(=O)/C=C(\O)/C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F19 compound treatment 1280.0 38.7 0.01 800.0 -85.5 -0.07 -0.0367 -0.5474 3120721 ChemDiv3_008577 CCCC(=O)NCCc1cc2ccc(OC)cc2[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F20 compound treatment 2560.0 1320.0 0.47 1240.0 354.0 0.27 0.5232 0.9668 3029257 ChemDiv3_008578 CC(C)CC(=O)NC(=S)Nc1cccc2nsnc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F21 compound treatment 41280.0 40000.0 14.2 2000.0 1110.0 0.86 10.6484 0.7483 3120722 ChemDiv3_008579 CCc1ccc(NC(=O)CSc2nc3CC(C)Sc3c(=O)n2CC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F22 compound treatment 1520.0 279.0 0.1 1320.0 434.0 0.33 0.3058 0.8789 3029258 ChemDiv3_008580 O=C(CC1(C[C@H]2C[C@@H]3C[C@H](C2)C1)C3)Nc4ccc5C(=O)OCc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F23 mock treatment 5960.0 4720.0 1.67 3480.0 2590.0 1.99 2.5921 0.9963 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 F24 mock treatment 1120.0 -121.0 -0.04 2280.0 1390.0 1.07 0.7266 0.6781 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G01 compound treatment 400.0 -841.0 -0.3 1600.0 714.0 0.55 0.1768 0.2832 3120723 ChemDiv3_008581 Cc1sc2n(Cc3cccc(C)c3)c(=O)n(Cc4ccccc4)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G02 compound treatment 520.0 -721.0 -0.26 1520.0 634.0 0.49 0.1635 0.2972 3120724 ChemDiv3_008582 COc1ccc2nc(NC(=O)CN(C)S(=O)(=O)c3cccs3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G03 compound treatment 640.0 -601.0 -0.21 680.0 -206.0 -0.16 -0.2624 -0.989 3029259 ChemDiv3_008583 CCN(CC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G04 compound treatment 640.0 -601.0 -0.21 720.0 -166.0 -0.13 -0.2407 -0.9694 3120725 ChemDiv3_008584 CCc1ccc(cc1)n2c(=O)n(CC(=O)C(C)(C)C)c3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G05 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 3029260 ChemDiv3_008585 CCn1c(COc2cccc3cccnc23)nnc1SCC(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G06 compound treatment 680.0 -561.0 -0.2 520.0 -366.0 -0.28 -0.3392 -0.9859 3120726 ChemDiv3_008586 CC1CCCCN1C(=O)Cn2c(=O)n(C3CCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G07 compound treatment 600.0 -641.0 -0.23 560.0 -326.0 -0.25 -0.3376 -0.9989 3029261 ChemDiv3_008587 Brc1cccc(c1)c2nnc3sc(CN4CCc5ccccc45)cn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G08 compound treatment 5520.0 4280.0 1.52 400.0 -486.0 -0.37 0.8097 0.5181 3120906 ChemDiv3_008588 CC1CCCC(NC(=O)CCCn2c(=O)[nH]c3cc(Cl)ccc3c2=O)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G09 compound treatment 320.0 -921.0 -0.33 560.0 -326.0 -0.25 -0.4078 -0.9912 3029262 ChemDiv3_008589 CN(C)/C=N/c1cc2nc3[nH]c(=O)n(CC=C)c(=O)c3nc2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G10 compound treatment 960.0 -281.0 -0.1 1280.0 394.0 0.3 0.1436 0.4503 3120907 ChemDiv3_008590 COc1ccc(CCn2c(=O)n(CC(=O)N(C)c3ccccc3)c4ccccc4c2=O)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G11 compound treatment 520.0 -721.0 -0.26 640.0 -246.0 -0.19 -0.3142 -0.9887 3120908 ChemDiv3_008591 Fc1ccc(cc1)c2n[nH]cc2/C=C/3\CS/C(=C\c4c[nH]nc4c5ccc(F)cc5)/C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G12 compound treatment 640.0 -601.0 -0.21 920.0 34.5 0.03 -0.1321 -0.6146 3029263 ChemDiv3_008592 Cc1ccccc1NC(=O)Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G13 compound treatment 360.0 -881.0 -0.31 760.0 -126.0 -0.1 -0.2892 -0.884 3120909 ChemDiv3_008593 S=C1NC2(CCCC2)N=C1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G14 compound treatment 1560.0 319.0 0.11 720.0 -166.0 -0.13 -0.0099 -0.0582 3120910 ChemDiv3_008594 Clc1ccccc1NS(=O)(=O)c2ccc3[nH]c(nc3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G15 compound treatment 360.0 -881.0 -0.31 360.0 -526.0 -0.4 -0.5063 -0.9921 3029264 ChemDiv3_008595 C(Sc1ncnc2c3ccccc3oc12)/C=C/c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G16 compound treatment 560.0 -681.0 -0.24 680.0 -206.0 -0.16 -0.2825 -0.9786 3120911 ChemDiv3_008596 CC(=O)Oc1c(c(C)nn1c2ccccc2)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G17 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 3029265 ChemDiv3_008597 Cc1ccc(cc1)S(=O)(=O)C2(CC2)C(=O)N3CCN(CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G18 compound treatment 520.0 -721.0 -0.26 800.0 -85.5 -0.07 -0.2274 -0.8607 3120912 ChemDiv3_008598 CN1CCN(CC1)c2cc(C)c3cc(NC(=S)N4CCCCC4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G19 compound treatment 320.0 -921.0 -0.33 400.0 -486.0 -0.37 -0.4947 -0.9979 3120913 ChemDiv3_008599 CCOc1ccc(cc1)n2c(=O)n(CC(=O)NCC3CCCO3)c4sc5CCCCc5c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G20 compound treatment 1600.0 359.0 0.13 680.0 -206.0 -0.16 -0.0216 -0.1065 3029266 ChemDiv3_008600 CCOc1ccc(NC(=O)NCCN2C(C)CCCC2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G21 compound treatment 1800.0 559.0 0.2 400.0 -486.0 -0.37 -0.1234 -0.2924 3120914 ChemDiv3_008601 CCc1ccc(cc1)n2c(=O)n(CC(=O)N(C)C3CCCCC3)c4sc5CCCc5c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G22 compound treatment 600.0 -641.0 -0.23 520.0 -366.0 -0.28 -0.3593 -0.9946 3029392 ChemDiv3_008602 CCN1CCN(CCNC(=O)Nc2ccc(Cl)cc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G23 mock treatment 840.0 -401.0 -0.14 640.0 -246.0 -0.19 -0.2339 -0.9904 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 G24 mock treatment 680.0 -561.0 -0.2 8720.0 7830.0 6.01 4.1122 0.6833 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H01 compound treatment 680.0 -561.0 -0.2 2040.0 1150.0 0.89 0.4859 0.5349 3120915 ChemDiv3_008603 CSc1ccc(NC(=O)NCCCN2CCC(Cc3ccccc3)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H02 compound treatment 6440.0 5200.0 1.84 400.0 -486.0 -0.37 1.0405 0.553 3029393 ChemDiv3_008604 COc1cc(/C=C/C(=O)NCCn2ccc3ccccc23)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H03 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 2106390 ChemDiv3_008605 COc1ccc(/C=C/2\N=C(NC2=O)SC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H04 compound treatment 1680.0 439.0 0.16 560.0 -326.0 -0.25 -0.0667 -0.2264 3029394 ChemDiv3_008606 O=c1[nH]cc(/C=N/CCN2CCOCC2)c(Nc3ccccc3)c1C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H05 compound treatment 440.0 -801.0 -0.28 1040.0 154.0 0.12 -0.1171 -0.3803 3120917 ChemDiv3_008607 CCc1ccc(NC(=O)C2CCN(CC2)S(=O)(=O)c3c(C)[nH]c(=O)[nH]c3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H06 compound treatment 480.0 -761.0 -0.27 600.0 -286.0 -0.22 -0.346 -0.9946 3029395 ChemDiv3_008608 Cc1cc(C)cc(NC(=O)CS(=O)(=O)c2cccc3nsnc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H07 compound treatment 5520.0 4280.0 1.52 840.0 -45.5 -0.03 1.0486 0.6906 3120918 ChemDiv3_008609 CC(NC(=O)C1CCCN(C1)S(=O)(=O)c2cccc3nonc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H08 compound treatment 560.0 -681.0 -0.24 840.0 -45.5 -0.03 -0.1956 -0.801 3120919 ChemDiv3_008610 CCOc1cc2CCN3C(C(C(=O)N(C)Cc4ccccc4)c5ccccc5C3=O)c2cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H09 compound treatment 480.0 -761.0 -0.27 520.0 -366.0 -0.28 -0.3894 -0.9998 3029396 ChemDiv3_008611 COC(=O)c1[nH]c2CC(CC(=O)c2c1C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H10 compound treatment 520.0 -721.0 -0.26 1800.0 914.0 0.7 0.3155 0.4222 3120920 ChemDiv3_008612 Cc1ccc(cc1)c2noc(CCC(=O)NCCCN3CCN(CC3)c4ccc(F)cc4)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H11 compound treatment 440.0 -801.0 -0.28 640.0 -246.0 -0.19 -0.3343 -0.9801 3029438 ChemDiv3_008613 COc1cc(OC)c2C(CC(=O)Nc2c1)c3ccccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H12 compound treatment 400.0 -841.0 -0.3 600.0 -286.0 -0.22 -0.366 -0.9885 3120921 ChemDiv3_008614 CC1CCCCN1C(=O)CSc2nnc(o2)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H13 compound treatment 760.0 -481.0 -0.17 600.0 -286.0 -0.22 -0.2757 -0.9924 3120922 ChemDiv3_008615 CC1=C(C(CC(=O)N1)c2cc3OCOc3cc2Br)C(=O)OCc4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H14 compound treatment 360.0 -881.0 -0.31 680.0 -206.0 -0.16 -0.3326 -0.9499 3029439 ChemDiv3_008616 CCc1ccc(NC(=O)C2C(N(CCOC)C(=O)c3ccccc23)c4c[nH]c5ccccc45)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H15 compound treatment 520.0 -721.0 -0.26 400.0 -486.0 -0.37 -0.4445 -0.9832 3120923 ChemDiv3_008617 CC1=C(C(CC(=O)N1)c2ccccc2C(F)(F)F)C(=O)OC3CCCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H16 compound treatment 560.0 -681.0 -0.24 640.0 -246.0 -0.19 -0.3042 -0.9924 3120924 ChemDiv3_008618 CCc1ccc(cc1)N2C(=S)N(C3CC2(C)Oc4ccccc34)C(=O)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H17 compound treatment 1520.0 279.0 0.1 2760.0 1870.0 1.44 1.0875 0.7539 3029440 ChemDiv3_008619 COc1ccc(OC)c2[nH]c(=O)c(CCNC(=O)/C=C\c3ccc4OCOc4c3)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H18 compound treatment 1400.0 159.0 0.06 10360.0 9470.0 7.27 5.1831 0.7126 3120925 ChemDiv3_008620 Clc1ccc(cc1)C(=O)/C=C/2\Nc3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H19 compound treatment 600.0 -641.0 -0.23 760.0 -126.0 -0.1 -0.229 -0.9269 3120926 ChemDiv3_008621 COc1ccc2cc(CCNC(=O)COc3ccc4ccccc4c3)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H20 compound treatment 400.0 -841.0 -0.3 1120.0 234.0 0.18 -0.0837 -0.2403 3029441 ChemDiv3_008622 Cc1cc(N2CCN(CC2)c3ccccc3)n4ncnc4n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H21 compound treatment 600.0 -641.0 -0.23 2480.0 1590.0 1.22 0.7047 0.566 3029397 ChemDiv3_008623 CCCSc1nc2CC(C)Sc2c(=O)n1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H22 compound treatment 560.0 -681.0 -0.24 1920.0 1030.0 0.79 0.3907 0.4706 3120927 ChemDiv3_008624 CCc1ccc(cc1)C(=O)/C=C/2\Sc3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H23 mock treatment 880.0 -361.0 -0.13 840.0 -45.5 -0.03 -0.1153 -0.8682 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 H24 mock treatment 3800.0 2560.0 0.91 1880.0 994.0 0.76 1.1817 0.9963 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I01 compound treatment 360.0 -881.0 -0.31 320.0 -566.0 -0.43 -0.5281 -0.987 3029398 ChemDiv3_008625 CCC(C)NC(=O)Cn1c(=O)n(c2ccc(Cl)c(Cl)c2)c(=O)c3c(C)c(C)sc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I02 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 3120928 ChemDiv3_008626 O=C(NC1CCCC1)C2CCN(CC2)S(=O)(=O)c3cccc4nonc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I03 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3120929 ChemDiv3_008627 Cc1cccn2c(=O)c3cc(sc3nc12)C(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I04 compound treatment 440.0 -801.0 -0.28 320.0 -566.0 -0.43 -0.508 -0.9789 3029399 ChemDiv3_008628 CC(C)(C)c1ccc(Cn2c(=O)n(Cc3ccc4OCOc4c3)c(=O)c5ccccc25)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I05 compound treatment 320.0 -921.0 -0.33 360.0 -526.0 -0.4 -0.5164 -0.9945 3120930 ChemDiv3_008629 COC(=O)CSc1nnc(CNC(=O)Cc2ccccc2)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I06 compound treatment 2240.0 999.0 0.35 280.0 -606.0 -0.46 -0.0782 -0.1338 3120931 ChemDiv3_008630 Cc1ccccc1Cn2c(=O)n(CCCCC(=O)NC3CCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I07 compound treatment 520.0 -721.0 -0.26 400.0 -486.0 -0.37 -0.4445 -0.9832 3029400 ChemDiv3_008631 Brc1cccc(c1)c2nnc3sc(CN4CCc5ccccc5C4)cn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I08 compound treatment 320.0 -921.0 -0.33 320.0 -566.0 -0.43 -0.5381 -0.9902 3120932 ChemDiv3_008632 Clc1ccc2c(=O)n(CCCC(=O)NC3CCCCCCC3)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I09 compound treatment 840.0 -401.0 -0.14 280.0 -606.0 -0.46 -0.4294 -0.8832 3029401 ChemDiv3_008633 CCC(=O)Nc1cc2nc3[nH]c(=O)n(C4CCCCCC4)c(=O)c3nc2cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I10 compound treatment 360.0 -881.0 -0.31 280.0 -606.0 -0.46 -0.5498 -0.9814 3121118 ChemDiv3_008634 COc1cc2n(CC(=O)NC3CCCCC3)c(=O)n(Cc4ccccc4Cl)c(=O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I11 compound treatment 440.0 -801.0 -0.28 360.0 -526.0 -0.4 -0.4863 -0.9853 3029402 ChemDiv3_008635 CCSC1=N/C(=C\c2ccccc2)/C(=O)N1c3ccc(C)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I12 compound treatment 280.0 -961.0 -0.34 360.0 -526.0 -0.4 -0.5264 -0.9965 3121119 ChemDiv3_008636 COc1cccc(c1)C(=O)Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I13 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3029442 ChemDiv3_008637 CC1(C)NC(=O)C(=N1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I14 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029443 ChemDiv3_008638 COc1ccc(NC(=O)CSc2nccn2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I15 compound treatment 440.0 -801.0 -0.28 360.0 -526.0 -0.4 -0.4863 -0.9853 3121120 ChemDiv3_008639 CCOC(=O)C(C)Sc1ncnc2c3ccccc3oc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I16 compound treatment 360.0 -881.0 -0.31 440.0 -446.0 -0.34 -0.4629 -0.999 3121121 ChemDiv3_008640 COc1cc2CCN3C(C(C(=O)NC4CCCC(C)C4C)c5ccccc5C3=O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I17 compound treatment 520.0 -721.0 -0.26 320.0 -566.0 -0.43 -0.4879 -0.9682 3029444 ChemDiv3_008641 CN(C1CCCCC1)C(=O)C2(CC2)S(=O)(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I18 compound treatment 360.0 -881.0 -0.31 800.0 -85.5 -0.07 -0.2675 -0.8373 3121122 ChemDiv3_008642 CCN1CCN(CCCNC(=S)Nc2ccc3nc(cc(C)c3c2)N4CCN(C)CC4)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I19 compound treatment 320.0 -921.0 -0.33 2360.0 1470.0 1.13 0.5693 0.4832 3029445 ChemDiv3_008643 COc1ccc(c(OC)c1)n2c(=O)n(CC(=O)Nc3cc(C)[nH]n3)c4sc5CCCCc5c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I20 compound treatment 3040.0 1800.0 0.64 600.0 -286.0 -0.22 0.2962 0.439 1912372 ChemDiv3_008644 O=C(OCC1CC2CC1C=C2)c3cc4ccccc4oc3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I21 compound treatment 400.0 -841.0 -0.3 1040.0 154.0 0.12 -0.1272 -0.396 3121123 ChemDiv3_008645 CCOc1ccc(cc1)n2c(=O)n(CC(=O)N(CC)CC)c3sc4CCCCCc4c3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I22 compound treatment 480.0 -761.0 -0.27 400.0 -486.0 -0.37 -0.4545 -0.9875 3121124 ChemDiv3_008646 Cc1c(NC(=O)NCc2ccccc2)c(=O)n(c3ccccc3)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I23 mock treatment 2840.0 1600.0 0.57 360.0 -526.0 -0.4 0.1157 0.1663 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 I24 mock treatment 336320.0 335000.0 118.87 4960.0 4070.0 3.13 86.2641 0.7255 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J01 compound treatment 320.0 -921.0 -0.33 400.0 -486.0 -0.37 -0.4947 -0.9979 3029446 ChemDiv3_008647 O=c1n(CCN2CCCCC2)c(=S)[nH]c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J02 compound treatment 2080.0 839.0 0.3 360.0 -526.0 -0.4 -0.0749 -0.1494 3121125 ChemDiv3_008648 Cc1ccc(cc1)C(=O)NCCn2ccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J03 compound treatment 320.0 -921.0 -0.33 2720.0 1830.0 1.41 0.7648 0.529 3029447 ChemDiv3_008649 CSC1=N/C(=C\c2ccccc2Cl)/C(=O)N1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J04 compound treatment 320.0 -921.0 -0.33 320.0 -566.0 -0.43 -0.5381 -0.9902 3121126 ChemDiv3_008650 CCc1ccc(N/C=C/2\C(=O)Nc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J05 compound treatment 200.0 -1040.0 -0.37 360.0 -526.0 -0.4 -0.5465 -0.999 3121127 ChemDiv3_008651 CC(NC(=O)C1CCN(CC1)S(=O)(=O)c2c(C)[nH]c(=O)[nH]c2=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J06 compound treatment 480.0 -761.0 -0.27 280.0 -606.0 -0.46 -0.5197 -0.9666 3029448 ChemDiv3_008652 Cc1cc(Br)ccc1NC(=O)CS(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J07 compound treatment 320.0 -921.0 -0.33 360.0 -526.0 -0.4 -0.5164 -0.9945 3121128 ChemDiv3_008653 Fc1ccc(cc1)N2CCN(CC2)C(=O)C3CCCN(C3)S(=O)(=O)c4cccc5nonc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J08 compound treatment 280.0 -961.0 -0.34 720.0 -166.0 -0.13 -0.331 -0.9095 3029449 ChemDiv3_008654 CCOc1cc2CCN3C(C(C(=O)N4CCCCC4)c5ccccc5C3=O)c2cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J09 compound treatment 320.0 -921.0 -0.33 480.0 -406.0 -0.31 -0.4512 -0.9997 1610300 ChemDiv3_008655 COc1ccc(cc1)N2COc3ccc(OC)cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J10 compound treatment 280.0 -961.0 -0.34 440.0 -446.0 -0.34 -0.483 -1.0 3029450 ChemDiv3_008656 CCCN(C(=O)CCc1nc(no1)c2ccccc2F)c3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J11 compound treatment 280.0 -961.0 -0.34 400.0 -486.0 -0.37 -0.5047 -0.999 3121129 ChemDiv3_008657 Cc1cc(C)c2C(CC(=O)Nc2c1)c3cccc(Cl)c3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J12 compound treatment 360.0 -881.0 -0.31 240.0 -646.0 -0.5 -0.5715 -0.9753 3121130 ChemDiv3_008658 O=C(CSc1nnc(o1)c2ccco2)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J13 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029451 ChemDiv3_008659 COc1ccccc1C2CC(=O)NC(=C2C(=O)OC3CCCC3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J14 compound treatment 400.0 -841.0 -0.3 440.0 -446.0 -0.34 -0.4529 -0.9977 3121131 ChemDiv3_008660 COCCN1C(C(C(=O)NCCc2cccc(C)c2)c3ccccc3C1=O)c4c[nH]c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J15 compound treatment 320.0 -921.0 -0.33 320.0 -566.0 -0.43 -0.5381 -0.9902 3121132 ChemDiv3_008661 COc1ccc(cc1)C2CC(=O)C3=C(C2)NC(=O)CC3c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J16 compound treatment 160.0 -1080.0 -0.38 320.0 -566.0 -0.43 -0.5782 -0.9981 3029452 ChemDiv3_008662 CC1(CC2N(C(=O)c3cccc(F)c3)C(=S)N1c4ccccc4)Oc5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J17 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3121133 ChemDiv3_008663 CCC(=O)NCCc1cc2c(OC)ccc(OC)c2[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J18 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029453 ChemDiv3_008664 COc1ccccc1C(=O)/C=C/2\Nc3cc4n(C)c(=O)n(C)c4cc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J19 compound treatment 360.0 -881.0 -0.31 400.0 -486.0 -0.37 -0.4846 -0.9962 3121134 ChemDiv3_008665 COc1ccc2cc(CCNC(=O)c3ccccc3)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J20 compound treatment 440.0 -801.0 -0.28 280.0 -606.0 -0.46 -0.5297 -0.9721 3121135 ChemDiv3_008666 COc1cccc(c1)C(=O)/C=C(\Nc2ccc3C(=O)OCc3c2)/C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J21 compound treatment 400.0 -841.0 -0.3 720.0 -166.0 -0.13 -0.3009 -0.9276 3029454 ChemDiv3_008667 COCCn1c(SCC(=O)N2CCOCC2)nc3CC(C)Sc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J22 compound treatment 560.0 -681.0 -0.24 280.0 -606.0 -0.46 -0.4996 -0.9536 3121136 ChemDiv3_008668 O=C(/C=C\1/Nc2nonc2NC1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J23 mock treatment 840.0 -401.0 -0.14 600.0 -286.0 -0.22 -0.2557 -0.9782 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 J24 mock treatment 6640.0 5400.0 1.92 480.0 -406.0 -0.31 1.1341 0.5845 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K01 compound treatment 1320.0 78.7 0.03 720.0 -166.0 -0.13 -0.0701 -0.5389 3029455 ChemDiv3_008669 CC(C)CCNC(=O)c1cc2c(=O)n3ccccc3nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K02 compound treatment 440.0 -801.0 -0.28 800.0 -85.5 -0.07 -0.2474 -0.8481 3121137 ChemDiv3_008670 CCN(C(=O)C1CCN(CC1)S(=O)(=O)c2cccc3nonc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K03 compound treatment 720.0 -521.0 -0.18 520.0 -366.0 -0.28 -0.3292 -0.9795 3121138 ChemDiv3_008671 CC(NC(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K04 compound treatment 640.0 -601.0 -0.21 1280.0 394.0 0.3 0.0633 0.1709 3029456 ChemDiv3_008672 Cc1cccc2nc(Cn3c(=O)n(CCC(=O)NCc4ccco4)c(=O)c5ccccc35)cc(=O)n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K05 compound treatment 360.0 -881.0 -0.31 720.0 -166.0 -0.13 -0.3109 -0.9213 3121139 ChemDiv3_008673 COC(=O)CSc1nnc(CNC(=O)c2ccccc2F)n1Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K06 compound treatment 320.0 -921.0 -0.33 520.0 -366.0 -0.28 -0.4295 -0.9971 3121140 ChemDiv3_008674 Cc1ccc(Cn2c(=O)n(CCC(=O)N3CCc4ccccc4C3)c(=O)c5ccccc25)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K07 compound treatment 1080.0 -161.0 -0.06 800.0 -85.5 -0.07 -0.0869 -0.9977 3029457 ChemDiv3_008675 Brc1cccc(c1)c2nnc3sc(CNCCc4ccccc4)cn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K08 compound treatment 320.0 -921.0 -0.33 720.0 -166.0 -0.13 -0.321 -0.9153 3121141 ChemDiv3_008676 COc1cccc(c1)C(=O)Cn2c(=O)n(CCc3ccccc3)c(=O)c4cc(OC)c(OC)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K09 compound treatment 240.0 -1000.0 -0.36 800.0 -85.5 -0.07 -0.2976 -0.8238 3029499 ChemDiv3_008677 C=CCN1C(=O)/C(=C\c2ccccc2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K10 compound treatment 480.0 -761.0 -0.27 920.0 34.5 0.03 -0.1722 -0.6348 3029500 ChemDiv3_008678 CCC1CCCCN1C(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c4cc(OC)c(OC)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K11 compound treatment 360.0 -881.0 -0.31 480.0 -406.0 -0.31 -0.4412 -1.0 3029501 ChemDiv3_008679 CCSC1=N/C(=C\c2cccnc2)/C(=O)N1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K12 compound treatment 960.0 -281.0 -0.1 600.0 -286.0 -0.22 -0.2256 -0.9365 3029502 ChemDiv3_008680 Cc1ccc(cc1)n2c(=O)n(Cc3cccc(C)c3)c4cc(ccc4c2=O)C(=O)NCc5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K13 compound treatment 480.0 -761.0 -0.27 920.0 34.5 0.03 -0.1722 -0.6348 3029503 ChemDiv3_008681 O=C1NC2(CCCC2)N=C1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K14 compound treatment 400.0 -841.0 -0.3 600.0 -286.0 -0.22 -0.366 -0.9885 3029504 ChemDiv3_008682 Fc1ccccc1NC(=O)CSc2nccn2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K15 compound treatment 440.0 -801.0 -0.28 1600.0 714.0 0.55 0.1869 0.3025 3029505 ChemDiv3_008683 O=C(CSc1ncnc2c3ccccc3oc12)OCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K16 compound treatment 600.0 -641.0 -0.23 1080.0 194.0 0.15 -0.0553 -0.2032 3121142 ChemDiv3_008684 CCN(CC)C(=O)C1C2N(CCc3cc(OC)c(OC)cc23)C(=O)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K17 compound treatment 360.0 -881.0 -0.31 720.0 -166.0 -0.13 -0.3109 -0.9213 3029506 ChemDiv3_008685 CSc1cccc(NC(=O)C2(CC2)S(=O)(=O)c3ccc(C)cc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K18 compound treatment 2080.0 839.0 0.3 720.0 -166.0 -0.13 0.1205 0.3726 3121143 ChemDiv3_008686 CN1CCN(CC1)c2cc(C)c3cc(NC(=S)NC4CC4)ccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K19 compound treatment 520.0 -721.0 -0.26 600.0 -286.0 -0.22 -0.3359 -0.997 3121321 ChemDiv3_008687 Clc1cccc(Cn2c(=O)n(c3ccccc3)c(=O)c4c5CCCc5sc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K20 compound treatment 960.0 -281.0 -0.1 880.0 -5.52 0.0 -0.0736 -0.7365 3029507 ChemDiv3_008688 Clc1ccc(cc1)c2cc(NC(=S)Nc3cccc(Cl)c3)n[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K21 compound treatment 720.0 -521.0 -0.18 800.0 -85.5 -0.07 -0.1772 -0.9029 3121322 ChemDiv3_008689 CCC(C)NC(=O)Cn1c(=O)n(CCc2ccccc2)c(=O)c3c4CCCCc4sc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K22 compound treatment 440.0 -801.0 -0.28 520.0 -366.0 -0.28 -0.3994 -1.0 1315204 ChemDiv3_008690 Cc1c(n2c(=O)c3ccccc3[nH]c2=S)c(=O)n(c4ccccc4)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K23 mock treatment 560.0 -681.0 -0.24 480.0 -406.0 -0.31 -0.391 -0.9922 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 K24 mock treatment 2400.0 1160.0 0.41 800.0 -85.5 -0.07 0.2442 0.5867 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L01 compound treatment 1080.0 -161.0 -0.06 1200.0 314.0 0.24 0.1303 0.525 3121323 ChemDiv3_008691 FC(F)(F)c1ccccc1NC(=O)NCCN2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L02 compound treatment 4960.0 3720.0 1.32 440.0 -446.0 -0.34 0.691 0.507 3029508 ChemDiv3_008692 FC(F)(F)c1cc(cc(c1)C(F)(F)F)C(=O)NCCn2ccc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L03 compound treatment 600.0 -641.0 -0.23 840.0 -45.5 -0.03 -0.1856 -0.8063 3121324 ChemDiv3_008693 Clc1ccc2nc(c(Nc3ccccc3)n2c1)c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L04 compound treatment 280.0 -961.0 -0.34 440.0 -446.0 -0.34 -0.483 -1.0 3121325 ChemDiv3_008694 CCCOc1ccc2oc(=O)c3N(CCCc3c2c1)C(=O)CN(C)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L05 compound treatment 280.0 -961.0 -0.34 520.0 -366.0 -0.28 -0.4396 -0.9953 3029509 ChemDiv3_008695 COc1ccc(NC(=O)C2CCCN(C2)S(=O)(=O)c3ccc(Br)s3)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L06 compound treatment 440.0 -801.0 -0.28 560.0 -326.0 -0.25 -0.3777 -0.9979 3121326 ChemDiv3_008696 O=C(CS(=O)(=O)c1cccc2nsnc12)N3CC(=O)N(CCc4ccccc4)C(=O)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L07 compound treatment 520.0 -721.0 -0.26 680.0 -206.0 -0.16 -0.2925 -0.973 3121327 ChemDiv3_008697 CCC(C)NC(=O)C1C(N(C)C(=O)c2ccccc12)c3c[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L08 compound treatment 440.0 -801.0 -0.28 680.0 -206.0 -0.16 -0.3126 -0.9614 3029510 ChemDiv3_008698 CCOc1cc2CCN3C(C(C(=O)NCCC(C)C)c4ccccc4C3=O)c2cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L09 compound treatment 440.0 -801.0 -0.28 640.0 -246.0 -0.19 -0.3343 -0.9801 3121328 ChemDiv3_008699 Cc1c([nH]c2CCCC(=O)c12)C(=O)OC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L10 compound treatment 360.0 -881.0 -0.31 520.0 -366.0 -0.28 -0.4195 -0.9985 3029511 ChemDiv3_008700 COc1ccc(N(C)C(=O)CCc2nc(no2)c3ccccc3F)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L11 compound treatment 1520.0 279.0 0.1 400.0 -486.0 -0.37 -0.1937 -0.5022 3121329 ChemDiv3_008701 CCc1ccc(cc1)C2CC(=O)NC3=C2C(=O)CC(C)(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L12 compound treatment 480.0 -761.0 -0.27 680.0 -206.0 -0.16 -0.3025 -0.9672 3121330 ChemDiv3_008702 Cc1cc(NC(=O)CSc2nnc(o2)c3ccco3)no1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L13 compound treatment 800.0 -441.0 -0.16 1480.0 594.0 0.46 0.212 0.4394 3029512 ChemDiv3_008703 Clc1ccc(cc1)C2CC(=O)NC3=C2C(=O)CC(C3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L14 compound treatment 640.0 -601.0 -0.21 400.0 -486.0 -0.37 -0.4144 -0.9649 3121331 ChemDiv3_008704 COCCN1C(C(C(=O)NCCN2CCOCC2)c3ccccc3C1=O)c4cn(C)c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L15 compound treatment 560.0 -681.0 -0.24 760.0 -126.0 -0.1 -0.239 -0.9187 3121332 ChemDiv3_008705 CC1=C(C(CC(=O)N1)c2cccc(Cl)c2)C(=O)OC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L16 compound treatment 520.0 -721.0 -0.26 1080.0 194.0 0.15 -0.0754 -0.2544 3029513 ChemDiv3_008706 CC1(CC2N(C(=O)c3ccccc3)C(=O)N1c4ccccc4)Oc5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L17 compound treatment 360.0 -881.0 -0.31 840.0 -45.5 -0.03 -0.2458 -0.7813 3121333 ChemDiv3_008707 Cc1ccc2cc(CCNC(=O)Cc3ccccc3)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L18 compound treatment 400.0 -841.0 -0.3 2600.0 1710.0 1.32 0.7197 0.5332 1922455 ChemDiv3_008708 O/C(=C\C(=O)c1ccccc1)/C(=O)Nc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L19 compound treatment 480.0 -761.0 -0.27 560.0 -326.0 -0.25 -0.3677 -0.9992 3029514 ChemDiv3_008709 Cc1ccc(C)c2[nH]c(=O)c(CCNC(=O)C(C)(C)Oc3ccc(Cl)cc3)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L20 compound treatment 400.0 -841.0 -0.3 280.0 -606.0 -0.46 -0.5397 -0.977 3121334 ChemDiv3_008710 OC(=O)/C(=C/C(=O)c1ccc(F)cc1)/Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L21 compound treatment 640.0 -601.0 -0.21 680.0 -206.0 -0.16 -0.2624 -0.989 3121335 ChemDiv3_008711 CCC1CCCCN1C(=O)CSc2nc3CC(C)Sc3c(=O)n2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L22 compound treatment 440.0 -801.0 -0.28 880.0 -5.52 0.0 -0.204 -0.7176 3029515 ChemDiv3_008712 O=C(CC1(CC2CC3CC(C2)C1)C3)Nc4ccc5[nH]c(=O)[nH]c5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L23 mock treatment 400.0 -841.0 -0.3 760.0 -126.0 -0.1 -0.2792 -0.8902 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 L24 mock treatment 1000.0 -241.0 -0.09 840.0 -45.5 -0.03 -0.0852 -0.9219 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M01 compound treatment 800.0 -441.0 -0.16 680.0 -206.0 -0.16 -0.2223 -1.0 3121336 ChemDiv3_008713 Cc1cccc(NC(=O)c2cc3c(=O)n4ccccc4nc3s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M02 compound treatment 640.0 -601.0 -0.21 2240.0 1350.0 1.04 0.5845 0.5506 3121337 ChemDiv3_008714 O=C(NCc1ccccc1)C2CCN(CC2)S(=O)(=O)c3cccc4nonc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M03 compound treatment 440.0 -801.0 -0.28 760.0 -126.0 -0.1 -0.2691 -0.8967 3029516 ChemDiv3_008715 CCN(C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M04 compound treatment 520.0 -721.0 -0.26 1160.0 274.0 0.21 -0.0319 -0.0963 3121338 ChemDiv3_008716 Cc1cccc(NC(=O)Cn2c(=O)n(CCC(=O)NCc3ccco3)c(=O)c4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M05 compound treatment 320.0 -921.0 -0.33 1440.0 554.0 0.43 0.0699 0.1303 3029517 ChemDiv3_008717 CCOC(=O)CSc1nnc(CNC(=O)c2cccs2)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M06 compound treatment 400.0 -841.0 -0.3 920.0 34.5 0.03 -0.1923 -0.6419 3121339 ChemDiv3_008718 O=C(Cn1c(=O)n(Cc2ccc(cc2)C(=O)NC3CCCC3)c(=O)c4ccccc14)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M07 compound treatment 440.0 -801.0 -0.28 1080.0 194.0 0.15 -0.0954 -0.2972 3029518 ChemDiv3_008719 Brc1ccc(cc1)c2nnc3sc(CN4CCC5(CC4)OCCO5)cn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M08 compound treatment 320.0 -921.0 -0.33 840.0 -45.5 -0.03 -0.2558 -0.7783 3121340 ChemDiv3_008720 Cc1ccccc1Cn2c(=O)n(CC3CCC(CC3)C(=O)NCc4ccccc4)c(=O)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M09 compound treatment 360.0 -881.0 -0.31 3240.0 2350.0 1.81 1.0571 0.5763 3029519 ChemDiv3_008721 Fc1ccc(/C=C/2\CS/C(=C\c3ccc(F)cc3)/C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M10 compound treatment 600.0 -641.0 -0.23 440.0 -446.0 -0.34 -0.4027 -0.9804 3121341 ChemDiv3_008722 CCC(C)NC(=O)Cn1c(=O)n(Cc2ccccc2Cl)c(=O)c3cc(OC)c(OC)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M11 compound treatment 440.0 -801.0 -0.28 560.0 -326.0 -0.25 -0.3777 -0.9979 3029520 ChemDiv3_008723 Fc1cccc(/C=C/2\CS/C(=C\c3cccc(F)c3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M12 compound treatment 720.0 -521.0 -0.18 640.0 -246.0 -0.19 -0.264 -1.0 3121342 ChemDiv3_008724 CC(C)(C)NS(=O)(=O)c1ccc2[nH]c(nc2c1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M13 compound treatment 480.0 -761.0 -0.27 1120.0 234.0 0.18 -0.0637 -0.1962 3029521 ChemDiv3_008725 CC(C)CC1(C)NC(=S)C(=N1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M14 compound treatment 600.0 -641.0 -0.23 960.0 74.5 0.06 -0.1204 -0.5134 3121343 ChemDiv3_008726 Cc1cccc(c1)n2ccnc2SCC(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M15 compound treatment 560.0 -681.0 -0.24 880.0 -5.52 0.0 -0.1739 -0.7194 3121344 ChemDiv3_008727 CCc1ccc(NC(=O)CSC2=NN3CCCC(=O)N=C3S2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M16 compound treatment 680.0 -561.0 -0.2 1000.0 114.0 0.09 -0.0786 -0.3613 3029522 ChemDiv3_008728 CC1CCN(CC1)S(=O)(=O)c2cn(CC(=O)N(C)Cc3ccccc3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M17 compound treatment 840.0 -401.0 -0.14 880.0 -5.52 0.0 -0.1037 -0.7278 3121345 ChemDiv3_008729 Clc1ccc(NC(=O)C2(CC2)S(=O)(=O)c3ccc(Cl)cc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M18 compound treatment 560.0 -681.0 -0.24 960.0 74.5 0.06 -0.1305 -0.5253 3029523 ChemDiv3_008730 CCOc1ccc(NC(=O)NCCCN2CCCC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M19 compound treatment 680.0 -561.0 -0.2 960.0 74.5 0.06 -0.1004 -0.4845 3121346 ChemDiv3_008731 CCCN(CCC)C(=O)Cn1c(=O)n(c2ccc(Cl)cc2)c(=O)c3c4CCCc4sc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M20 compound treatment 760.0 -481.0 -0.17 800.0 -85.5 -0.07 -0.1672 -0.9138 3029524 ChemDiv3_008732 Cc1c(CO)[nH]c2ccc(Cl)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M21 compound treatment 560.0 -681.0 -0.24 720.0 -166.0 -0.13 -0.2607 -0.9549 3121347 ChemDiv3_008733 COc1ccc(NC(=O)Cn2c(=O)n(c3ccccc3)c(=O)c4c5CCCCc5sc24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M22 compound treatment 840.0 -401.0 -0.14 920.0 34.5 0.03 -0.0819 -0.5659 3029525 ChemDiv3_008734 Cc1ccc(NC(=S)NCCCN2CCN(CC2)c3cc(Cl)ccc3C)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M23 mock treatment 960.0 -281.0 -0.1 880.0 -5.52 0.0 -0.0736 -0.7365 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 M24 mock treatment 1280.0 38.7 0.01 600.0 -286.0 -0.22 -0.1453 -0.6615 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N01 compound treatment 720.0 -521.0 -0.18 520.0 -366.0 -0.28 -0.3292 -0.9795 3121520 ChemDiv3_008735 CCc1nnc(NC(=O)Nc2ccccc2C(F)(F)F)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N02 compound treatment 800.0 -441.0 -0.16 3360.0 2470.0 1.9 1.2326 0.6466 3121521 ChemDiv3_008736 Cc1cc2ccccc2n1CCNC(=O)Cc3cccc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N03 compound treatment 320.0 -921.0 -0.33 800.0 -85.5 -0.07 -0.2775 -0.8325 3029526 ChemDiv3_008737 Cc1ccc(Nc2c(nc3ccccn23)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N04 compound treatment 1040.0 -201.0 -0.07 920.0 34.5 0.03 -0.0318 -0.4172 3121522 ChemDiv3_008738 CCCOc1ccc2oc(=O)c3N(CCCc3c2c1)C(=O)CN4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N05 compound treatment 440.0 -801.0 -0.28 520.0 -366.0 -0.28 -0.3994 -1.0 3029527 ChemDiv3_008739 COc1ccc(C)cc1NC(=O)CN(C)S(=O)(=O)c2ccc(Br)s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N06 compound treatment 520.0 -721.0 -0.26 1120.0 234.0 0.18 -0.0536 -0.1715 3121523 ChemDiv3_008740 CCOC(=O)C1C(CC(=CC1=O)c2ccc(F)cc2)c3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N07 compound treatment 440.0 -801.0 -0.28 480.0 -406.0 -0.31 -0.4211 -0.999 3121524 ChemDiv3_008741 CN1C(C(C(=O)NCc2ccc(F)cc2)c3ccccc3C1=O)c4c[nH]c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N08 compound treatment 680.0 -561.0 -0.2 960.0 74.5 0.06 -0.1004 -0.4845 3029528 ChemDiv3_008742 CCCCN(C)C(=O)Cc1c([nH]c2ccc(Cl)cc12)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N09 compound treatment 720.0 -521.0 -0.18 680.0 -206.0 -0.16 -0.2423 -0.9969 3029529 ChemDiv3_008743 CCCOC(=O)c1[nH]c2CCCC(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N10 compound treatment 520.0 -721.0 -0.26 560.0 -326.0 -0.25 -0.3576 -0.9999 3121525 ChemDiv3_008744 CCN(C(=O)CCc1nc(no1)c2ccccc2F)c3cc(Cl)ccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N11 compound treatment 600.0 -641.0 -0.23 840.0 -45.5 -0.03 -0.1856 -0.8063 3121526 ChemDiv3_008745 Cc1c([nH]c2CC(CC(=O)c12)c3ccc(Cl)cc3)C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N12 compound treatment 640.0 -601.0 -0.21 920.0 34.5 0.03 -0.1321 -0.6146 1375150 ChemDiv3_008746 COc1cc(cc(OC)c1OC)c2nnc(SCC(=O)N3CCCCC3C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N13 compound treatment 680.0 -561.0 -0.2 760.0 -126.0 -0.1 -0.2089 -0.9445 3121527 ChemDiv3_008747 Fc1ccc(cc1)C2CC(=O)C3=C(C2)NC(=O)CC3c4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N14 compound treatment 560.0 -681.0 -0.24 680.0 -206.0 -0.16 -0.2825 -0.9786 3029530 ChemDiv3_008748 CC1CCCN(C1)C(c2ccc(F)cc2)c3c(O)[nH]c(=O)[nH]c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N15 compound treatment 1000.0 -241.0 -0.09 880.0 -5.52 0.0 -0.0635 -0.7412 3121528 ChemDiv3_008749 CC(C)SC1=NSC2=NC(=O)/C(=C\c3ccc(OC(=O)C)cc3)/C(=N)N12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N16 compound treatment 640.0 -601.0 -0.21 1080.0 194.0 0.15 -0.0453 -0.1738 3121529 ChemDiv3_008750 Brc1cc2CCN(C(=O)C3CC3)c2c(c1)S(=O)(=O)CCC(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N17 compound treatment 480.0 -761.0 -0.27 760.0 -126.0 -0.1 -0.2591 -0.9036 3029531 ChemDiv3_008751 CCCC(=O)NCCc1cc2ccc(C)cc2[nH]c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N18 compound treatment 840.0 -401.0 -0.14 800.0 -85.5 -0.07 -0.1471 -0.9382 3029574 ChemDiv3_008752 Cc1ccc(cc1C)C(=O)/C=C/2\Nc3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N19 compound treatment 440.0 -801.0 -0.28 720.0 -166.0 -0.13 -0.2909 -0.9341 3029575 ChemDiv3_008753 Cc1ccc2cc(CCNC(=O)C3(CC4CC5CC(C4)C3)C5)c(=O)[nH]c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N20 compound treatment 600.0 -641.0 -0.23 1240.0 354.0 0.27 0.0316 0.089 3029576 ChemDiv3_008754 Cc1c[n+]([O-])n(n1)c2ccc(cc2)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N21 compound treatment 600.0 -641.0 -0.23 720.0 -166.0 -0.13 -0.2507 -0.9622 3029577 ChemDiv3_008755 CCOC(=O)N1CCN(CC1)C(=O)CSc2nc3CC(C)Sc3c(=O)n2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N22 compound treatment 400.0 -841.0 -0.3 400.0 -486.0 -0.37 -0.4746 -0.9939 3029578 ChemDiv3_008756 Clc1ccc(cc1)c2cc3Nc4ccccc4Nc3nn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N23 mock treatment 640.0 -601.0 -0.21 720.0 -166.0 -0.13 -0.2407 -0.9694 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 N24 mock treatment 600.0 -641.0 -0.23 680.0 -206.0 -0.16 -0.2724 -0.984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O01 compound treatment 400.0 -841.0 -0.3 440.0 -446.0 -0.34 -0.4529 -0.9977 3029579 ChemDiv3_008757 CC(C)CN(CC(C)C)C(=O)c1cc2c(=O)n3ccccc3nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O02 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3121530 ChemDiv3_008758 O=C(NC1CCCCC1)C2CCCN(C2)S(=O)(=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O03 compound treatment 480.0 -761.0 -0.27 360.0 -526.0 -0.4 -0.4762 -0.9809 3029580 ChemDiv3_008759 Cc1cccn2c(=O)c3cc(sc3nc12)C(=O)NC4CCSC4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O04 compound treatment 440.0 -801.0 -0.28 360.0 -526.0 -0.4 -0.4863 -0.9853 3121531 ChemDiv3_008760 COc1ccccc1CNC(=O)CCn2c(=O)n(Cc3ccc(F)cc3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O05 compound treatment 200.0 -1040.0 -0.37 320.0 -566.0 -0.43 -0.5682 -0.9968 3029581 ChemDiv3_008761 CCOC(=O)CSc1nnc(CNC(=O)c2cccs2)n1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O06 compound treatment 600.0 -641.0 -0.23 520.0 -366.0 -0.28 -0.3593 -0.9946 3121532 ChemDiv3_008762 CN(C1CCCCC1)C(=O)Cn2c(=O)n(CCCCC(=O)NC3CCCC3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O07 compound treatment 320.0 -921.0 -0.33 320.0 -566.0 -0.43 -0.5381 -0.9902 3121533 ChemDiv3_008763 Brc1ccc(cc1)c2nnc3sc(CNCc4ccc5OCOc5c4)cn23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O08 compound treatment 400.0 -841.0 -0.3 360.0 -526.0 -0.4 -0.4963 -0.989 3029582 ChemDiv3_008764 Cc1ccccc1Cn2c(=O)n(CCC(=O)NCCc3ccccc3)c(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O09 compound treatment 440.0 -801.0 -0.28 440.0 -446.0 -0.34 -0.4429 -0.9958 3121534 ChemDiv3_008765 Cc1cccc(/C=C/2\CS/C(=C\c3cccc(C)c3)/C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O10 compound treatment 360.0 -881.0 -0.31 920.0 34.5 0.03 -0.2023 -0.6449 3121535 ChemDiv3_008766 COc1cc2n(CC(=O)N3CC(C)CC(C)C3)c(=O)n(Cc4ccccc4Cl)c(=O)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O11 compound treatment 280.0 -961.0 -0.34 320.0 -566.0 -0.43 -0.5481 -0.9929 3029583 ChemDiv3_008767 CCOc1ccc(cc1)N2C(=O)/C(=C/c3ccc(F)cc3)/N=C2SC(CC)C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O12 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3121536 ChemDiv3_008768 Clc1ccccc1CNS(=O)(=O)c2ccc3[nH]c(nc3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O13 compound treatment 360.0 -881.0 -0.31 400.0 -486.0 -0.37 -0.4846 -0.9962 3029584 ChemDiv3_008769 O=C(CSC1=NC2(CCCC2)N=C1c3ccccc3)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O14 compound treatment 320.0 -921.0 -0.33 280.0 -606.0 -0.46 -0.5598 -0.9851 3121537 ChemDiv3_008770 Cc1cccc(c1)n2ccnc2SCC(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O15 compound treatment 320.0 -921.0 -0.33 400.0 -486.0 -0.37 -0.4947 -0.9979 3029585 ChemDiv3_008771 Fc1ccccc1CSC2=NN3CCCC(=O)N=C3S2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O16 compound treatment 320.0 -921.0 -0.33 440.0 -446.0 -0.34 -0.473 -0.9997 3121538 ChemDiv3_008772 CCOc1ccccc1NC(=O)Cn2cc(c3ccccc3c2=O)S(=O)(=O)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O17 compound treatment 360.0 -881.0 -0.31 280.0 -606.0 -0.46 -0.5498 -0.9814 3121539 ChemDiv3_008773 Clc1ccc(cc1)S(=O)(=O)C2(CC2)C(=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O18 compound treatment 280.0 -961.0 -0.34 320.0 -566.0 -0.43 -0.5481 -0.9929 3029586 ChemDiv3_008774 CCc1ccc(NC(=O)NCCN2CCc3ccccc3C2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O19 compound treatment 200.0 -1040.0 -0.37 400.0 -486.0 -0.37 -0.5248 -1.0 3121540 ChemDiv3_008775 CC1CC(C)CN(C1)C(=O)Cn2c(=O)n(c3ccc(Cl)cc3)c(=O)c4c5CCCc5sc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O20 compound treatment 280.0 -961.0 -0.34 240.0 -646.0 -0.5 -0.5916 -0.9834 3029587 ChemDiv3_008776 Nc1cc(c2ccccc2)n(n1)C(=O)Nc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O21 compound treatment 240.0 -1000.0 -0.36 240.0 -646.0 -0.5 -0.6016 -0.9867 3121541 ChemDiv3_008777 CCc1ccc(NC(=O)Cn2c(=O)n(CCc3ccccc3)c(=O)c4c5CCCCc5sc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O22 compound treatment 280.0 -961.0 -0.34 360.0 -526.0 -0.4 -0.5264 -0.9965 3029588 ChemDiv3_008778 CCN1CCN(Cc2ccc(NC(=O)Nc3ccccc3)cc2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O23 mock treatment 280.0 -961.0 -0.34 320.0 -566.0 -0.43 -0.5481 -0.9929 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 O24 mock treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P01 compound treatment 360.0 -881.0 -0.31 360.0 -526.0 -0.4 -0.5063 -0.9921 3121542 ChemDiv3_008779 CN1C(C(C(=O)NCc2ccco2)c3ccccc3C1=O)c4cn(C)c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P02 compound treatment 440.0 -801.0 -0.28 520.0 -366.0 -0.28 -0.3994 -1.0 3121543 ChemDiv3_008780 Cc1cc2ccccc2n1CCNC(=O)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P03 compound treatment 880.0 -361.0 -0.13 320.0 -566.0 -0.43 -0.3976 -0.8784 3029589 ChemDiv3_008781 C1Oc2ccc(Nc3c(nc4ccccn34)c5ccccc5)cc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P04 compound treatment 240.0 -1000.0 -0.36 280.0 -606.0 -0.46 -0.5799 -0.9912 3121544 ChemDiv3_008782 OC(=O)c1ccccc1N/C=C/2\C(=O)Nc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P05 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3029590 ChemDiv3_008783 Cc1[nH]c(=O)[nH]c(=O)c1S(=O)(=O)N2CCCC(C2)C(=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P06 compound treatment 320.0 -921.0 -0.33 240.0 -646.0 -0.5 -0.5815 -0.9796 3121545 ChemDiv3_008784 CCOC(=O)C1C(CC(=CC1=O)c2cccs2)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P07 compound treatment 240.0 -1000.0 -0.36 280.0 -606.0 -0.46 -0.5799 -0.9912 3121546 ChemDiv3_008785 Cc1ccc(cc1C)N2COc3cc4OCOc4cc3C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P08 compound treatment 520.0 -721.0 -0.26 560.0 -326.0 -0.25 -0.3576 -0.9999 3029591 ChemDiv3_008786 OC(=O)c1[nH]c2ccc(Cl)cc2c1CC(=O)N3CCC4(CC3)OCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P09 compound treatment 480.0 -761.0 -0.27 280.0 -606.0 -0.46 -0.5197 -0.9666 3121723 ChemDiv3_008787 CCCc1c([nH]c2CC(CC(=O)c12)c3ccccc3)C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P10 compound treatment 840.0 -401.0 -0.14 280.0 -606.0 -0.46 -0.4294 -0.8832 3121724 ChemDiv3_008788 CC1CCCCN1C(=O)CSc2nnc(o2)c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P11 compound treatment 1520.0 279.0 0.1 320.0 -566.0 -0.43 -0.2371 -0.5324 3029592 ChemDiv3_008789 CCOC(=O)c1[nH]c2CC(CC(=O)c2c1c3ccccc3)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P12 compound treatment 4440.0 3200.0 1.13 240.0 -646.0 -0.5 0.4519 0.365 1558672 ChemDiv3_008790 O=C(CSc1nnc(Cc2ccccc2)o1)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P13 compound treatment 320.0 -921.0 -0.33 240.0 -646.0 -0.5 -0.5815 -0.9796 3121725 ChemDiv3_008791 COC(=O)C1C(C)CC2=C(C(CC(=O)N2)c3cccc(OC)c3)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P14 compound treatment 1640.0 399.0 0.14 240.0 -646.0 -0.5 -0.2504 -0.4859 3029593 ChemDiv3_008792 Cc1ccc(cc1)C(N2CCCCC2)c3c(O)[nH]c(=S)[nH]c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P15 compound treatment 280.0 -961.0 -0.34 280.0 -606.0 -0.46 -0.5698 -0.9884 3121726 ChemDiv3_008793 COc1cc(/C=C\2/C(=N)N3C(=NSC3=NC2=O)SC(C)C)ccc1O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P16 compound treatment 360.0 -881.0 -0.31 240.0 -646.0 -0.5 -0.5715 -0.9753 3029594 ChemDiv3_008794 CC1CCCN(C1)C(=O)CCS(=O)(=O)c2cc(Br)cc3CCN(C(=O)C4CC4)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P17 compound treatment 280.0 -961.0 -0.34 240.0 -646.0 -0.5 -0.5916 -0.9834 3121727 ChemDiv3_008795 Cc1ccc2cc(CCNC(=O)c3ccc(Cl)cc3Cl)c(=O)[nH]c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P18 compound treatment 320.0 -921.0 -0.33 520.0 -366.0 -0.28 -0.4295 -0.9971 3121728 ChemDiv3_008796 COc1ccccc1C(=O)/C=C(\O)/C(=O)Nc2sc3CCCc3c2C#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P19 compound treatment 240.0 -1000.0 -0.36 800.0 -85.5 -0.07 -0.2976 -0.8238 3029595 ChemDiv3_008797 Cc1ccc(cc1)S(=O)(=O)NCCc2cc3ccc(C)cc3[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P20 compound treatment 400.0 -841.0 -0.3 360.0 -526.0 -0.4 -0.4963 -0.989 1082215 ChemDiv3_008798 O=C(c1nc2ccccc2[nH]1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P21 compound treatment 4440.0 3200.0 1.13 360.0 -526.0 -0.4 0.5171 0.4294 3121729 ChemDiv3_008799 CC1Cc2nc(SCC(=O)NCc3ccco3)n(Cc4ccccc4)c(=O)c2S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P22 compound treatment 440.0 -801.0 -0.28 240.0 -646.0 -0.5 -0.5514 -0.9652 3029596 ChemDiv3_008800 CCN1CCN(CCCNC(=O)c2ccc3N/C(=C\C(=O)c4ccc(OC)cc4)/C(=O)Nc3c2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P23 mock treatment 240.0 -1000.0 -0.36 240.0 -646.0 -0.5 -0.6016 -0.9867 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2025 P24 mock treatment 320.0 -921.0 -0.33 320.0 -566.0 -0.43 -0.5381 -0.9902 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A01 compound treatment 920.0 376.0 0.13 1760.0 1050.0 0.81 0.6657 0.8129 3121730 ChemDiv3_008801 COc1cccc(c1)C(=O)/C=C/2\Nc3ccc(cc3NC2=O)C(=O)Nc4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A02 compound treatment 3400.0 2860.0 1.01 920.0 212.0 0.16 0.8318 0.8105 3029597 ChemDiv3_008802 C1CCC(CC1)Sc2nc3ccccc3n4cnnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A03 compound treatment 2640.0 2100.0 0.74 520.0 -188.0 -0.14 0.424 0.5598 3121731 ChemDiv3_008803 Cc1cc(C)n(CCC(=O)Nc2ccc(C)cc2C)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A04 compound treatment 320.0 -224.0 -0.08 1680.0 972.0 0.75 0.4718 0.6284 3121732 ChemDiv3_008804 Cc1ccc(CNC(=O)c2cccc(Nc3nc4ccccc4n5cnnc35)c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A05 compound treatment 720.0 176.0 0.06 1600.0 892.0 0.69 0.5287 0.7684 3029598 ChemDiv3_008805 Cc1cc(C)n(n1)c2nc3ccccc3nc2NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A06 compound treatment 280.0 -264.0 -0.09 520.0 -188.0 -0.14 -0.168 -0.9782 3121733 ChemDiv3_008806 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc3oc(=O)c4ncn(CC)c4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A07 compound treatment 480.0 -63.8 -0.02 480.0 -228.0 -0.17 -0.1395 -0.792 3029599 ChemDiv3_008807 CCc1ccc(NC(=O)CCc2nc3ccccc3[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A08 compound treatment 240.0 -304.0 -0.11 400.0 -308.0 -0.24 -0.2432 -0.9368 3121734 ChemDiv3_008808 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A09 compound treatment 480.0 -63.8 -0.02 1000.0 292.0 0.22 0.1427 0.6327 1119277 ChemDiv3_008809 Clc1cnn(c(=O)c1Cl)C2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A10 compound treatment 2240.0 1700.0 0.6 360.0 -348.0 -0.27 0.2368 0.3597 3121735 ChemDiv3_008810 CCCCN(CC)C(=O)c1cc2cc3cc(OC)ccc3nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A11 compound treatment 2560.0 2020.0 0.72 240.0 -468.0 -0.36 0.2519 0.3148 3121736 ChemDiv3_008811 OC(=O)C1(CC2CC3C1)CC(C2)(C3)n4ncc(NCCc5ccccc5)c(Cl)c4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A12 compound treatment 1520.0 976.0 0.35 800.0 92.4 0.07 0.2951 0.8346 3029600 ChemDiv3_008812 CC1=Nc2cc(ccc2Sc3ccccc13)C(=O)NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A13 compound treatment 440.0 -104.0 -0.04 840.0 132.0 0.1 0.0459 0.4242 3121737 ChemDiv3_008813 Cc1cc(Nc2cnn(c3nc4ccccc4o3)c(=O)c2Cl)ccc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A14 compound treatment 320.0 -224.0 -0.08 600.0 -108.0 -0.08 -0.1145 -0.9998 3029601 ChemDiv3_008814 CCCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)NC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A15 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3121738 ChemDiv3_008815 O=C(NCCc1ccccc1)c2nnc(o2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A16 compound treatment 920.0 376.0 0.13 280.0 -428.0 -0.33 -0.1377 -0.3887 3029602 ChemDiv3_008816 Fc1ccc(CN2CCN(CC(=O)NCc3ccc(Cl)cc3)C2=O)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A17 compound treatment 320.0 -224.0 -0.08 320.0 -388.0 -0.3 -0.2665 -0.8655 3121739 ChemDiv3_008817 CC(C)NC(=O)c1nnc(Cc2cccc(Cl)c2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A18 compound treatment 400.0 -144.0 -0.05 520.0 -188.0 -0.14 -0.1379 -0.9026 3121740 ChemDiv3_008818 CC(NC(=O)/C=C/1\Sc2ccccc2NC1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A19 compound treatment 240.0 -304.0 -0.11 720.0 12.4 0.01 -0.0695 -0.6421 3029603 ChemDiv3_008819 COc1ccccc1N2CCN(CCCNC(=O)c3nnc(Cc4ccccc4Cl)o3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A20 compound treatment 360.0 -184.0 -0.07 1160.0 452.0 0.35 0.1995 0.5645 3121741 ChemDiv3_008820 CN1C(=O)/C(=C/c2ccc(cc2)C(=O)NC3CCCC3)/Oc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A21 compound treatment 200.0 -344.0 -0.12 240.0 -468.0 -0.36 -0.3401 -0.897 1139900 ChemDiv3_008821 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A22 compound treatment 320.0 -224.0 -0.08 1560.0 852.0 0.65 0.4066 0.6168 3029604 ChemDiv3_008822 CN1C(=O)/C(=C\c2ccccc2)/Sc3ccc(cc13)C(=O)NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A23 mock treatment 360.0 -184.0 -0.07 360.0 -348.0 -0.27 -0.2348 -0.8547 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 A24 mock treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B01 compound treatment 640.0 96.3 0.03 840.0 132.0 0.1 0.096 0.8954 3121742 ChemDiv3_008823 COc1ccc(/C=C/2\Oc3ccccc3N(CC(=O)NC(C)c4ccccc4)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B02 compound treatment 400.0 -144.0 -0.05 360.0 -348.0 -0.27 -0.2247 -0.8273 3029605 ChemDiv3_008824 O=C1C(N=C2N1C(=S)Nc3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B03 compound treatment 480.0 -63.8 -0.02 320.0 -388.0 -0.3 -0.2264 -0.7587 3121743 ChemDiv3_008825 Clc1ccc(/C=C\2/Sc3ccccc3N(CC(=O)NCC4CCCO4)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B04 compound treatment 320.0 -224.0 -0.08 320.0 -388.0 -0.3 -0.2665 -0.8655 3121744 ChemDiv3_008826 COc1cccc(c1)N2C(=S)NC3C(C)C2(C)Oc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B05 compound treatment 1120.0 576.0 0.2 440.0 -268.0 -0.21 -7.0E-4 -0.0025 3029651 ChemDiv3_008827 Cc1cc(NC(=O)/C=C\c2ccccc2)nc3c4ccccc4oc(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B06 compound treatment 760.0 216.0 0.08 240.0 -468.0 -0.36 -0.1996 -0.5437 3121745 ChemDiv3_008828 Cc1ccccc1NS(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B07 compound treatment 1400.0 856.0 0.3 280.0 -428.0 -0.33 -0.0173 -0.0388 3029652 ChemDiv3_008829 Cn1cc(CC(=O)N2CCN(CC2)c3ccc(Cl)cc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B08 compound treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 1700577 ChemDiv3_008830 CC(Oc1ccccc1)C(=O)OCn2nnc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B09 compound treatment 840.0 296.0 0.11 320.0 -388.0 -0.3 -0.1361 -0.4313 3121746 ChemDiv3_008831 COc1ccc2n(C)/c(=N/C(=O)CSCC(=O)Nc3nc(cs3)c4ccccc4)/sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B10 compound treatment 440.0 -104.0 -0.04 280.0 -428.0 -0.33 -0.2581 -0.7815 3029654 ChemDiv3_008832 CCOC(=O)Cn1nc(c2ccccc2)c3cnc4ccc(CC)cc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B11 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 3121929 ChemDiv3_008833 Cc1n[nH]c(C)c1S(=O)(=O)Nc2cccc(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B12 compound treatment 640.0 96.3 0.03 280.0 -428.0 -0.33 -0.208 -0.6302 3029655 ChemDiv3_008834 CSc1ccc(Cn2cccc2C3=NC(CO3)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B13 compound treatment 800.0 256.0 0.09 360.0 -348.0 -0.27 -0.1244 -0.4413 3121930 ChemDiv3_008835 Cc1noc(C)c1S(=O)(=O)NCCN2CCN(CC2)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B14 compound treatment 5760.0 5220.0 1.85 440.0 -268.0 -0.21 1.1632 0.6248 3121931 ChemDiv3_008836 CCS(=O)(=O)C1=NSC2=NC(=O)/C(=C\c3ccc(OCc4ccc(C)cc4)c(OC)c3)/C(=N)N12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B15 compound treatment 2080.0 1540.0 0.54 280.0 -428.0 -0.33 0.1532 0.2409 3029658 ChemDiv3_008837 Cc1cc(C)n2c(Nc3c(C)cccc3C)c(nc2n1)c4ccc(Cl)s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B16 compound treatment 3000.0 2460.0 0.87 240.0 -468.0 -0.36 0.3623 0.3844 3121932 ChemDiv3_008838 CCC(=O)N1C(C)Cc2cc(ccc12)S(=O)(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B17 compound treatment 2040.0 1500.0 0.53 200.0 -508.0 -0.39 0.0998 0.1515 3029659 ChemDiv3_008839 COCC(=O)N1N=C(CC1c2ccccc2C)c3cccc(NS(=O)(=O)C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B18 compound treatment 560.0 16.3 0.01 360.0 -348.0 -0.27 -0.1846 -0.6917 3121933 ChemDiv3_008840 O=C(C1CCC1)N2CCc3cc(ccc23)S(=O)(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B19 compound treatment 480.0 -63.8 -0.02 240.0 -468.0 -0.36 -0.2698 -0.7502 3029660 ChemDiv3_008841 O=C(CSc1nnc(CNC(=O)c2ccco2)o1)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B20 compound treatment 320.0 -224.0 -0.08 3160.0 2450.0 1.88 1.2752 0.6767 3121934 ChemDiv3_008842 COC(CNC(=O)C1CCN(CC1)S(=O)(=O)c2cccc3nsnc23)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B21 compound treatment 520.0 -23.8 -0.01 280.0 -428.0 -0.33 -0.2381 -0.725 3121935 ChemDiv3_008843 CN(C(=O)c1cn(C2CCCC2)c(=O)c3n(C)c4ccccc4c13)c5cccc(c5)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B22 compound treatment 280.0 -264.0 -0.09 400.0 -308.0 -0.24 -0.2331 -0.9179 3029662 ChemDiv3_008844 CCCN(C(=O)c1cc2cc3ccc(C)cc3nc2o1)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B23 mock treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 B24 mock treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C01 compound treatment 400.0 -144.0 -0.05 2040.0 1330.0 1.02 0.6873 0.671 3121936 ChemDiv3_008845 COc1ccc(cc1OC)C(=O)/C=C/2\Nc3ccc(cc3NC2=O)C(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C02 compound treatment 520.0 -23.8 -0.01 280.0 -428.0 -0.33 -0.2381 -0.725 3029663 ChemDiv3_008846 Cc1nnn(n1)C2(CC3CC4CC(C3)(C2)C(=O)NC5CCCCCC5)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C03 compound treatment 1440.0 896.0 0.32 480.0 -228.0 -0.17 0.1013 0.2791 3121937 ChemDiv3_008847 Cc1ccc(C)c(c1)N2CCN(CC2)C(=O)CN3CC(CC3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C04 compound treatment 2720.0 2180.0 0.77 240.0 -468.0 -0.36 0.2921 0.343 3029664 ChemDiv3_008848 O=c1oc2ccccc2c(N3CCN(CC3)c4ccccc4)c1CN5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C05 compound treatment 1880.0 1340.0 0.47 280.0 -428.0 -0.33 0.1031 0.1788 3121938 ChemDiv3_008849 Cc1nccn1CCC(=O)Nc2ccc(C)c(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C06 compound treatment 400.0 -144.0 -0.05 280.0 -428.0 -0.33 -0.2682 -0.8073 3121939 ChemDiv3_008850 Cc1ccc2cc3cc(sc3nc2c1)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C07 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3028694 ChemDiv3_008851 CC(=O)OC1C(N(N=C1c2ccccc2)C(=O)C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C08 compound treatment 2560.0 2020.0 0.72 360.0 -348.0 -0.27 0.3171 0.4153 3028696 ChemDiv3_008852 CCOc1ccccc1N(C)C(=O)c2cc3cc4ccc(OC)cc4nc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C09 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3028697 ChemDiv3_008853 CCc1ccc(NC(=O)C2NC(=O)CC2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C10 compound treatment 400.0 -144.0 -0.05 240.0 -468.0 -0.36 -0.2899 -0.7995 3028699 ChemDiv3_008854 COc1ccc2nc3sc(cc3cc2c1)C(=O)N(C)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C11 compound treatment 2600.0 2060.0 0.73 240.0 -468.0 -0.36 0.262 0.3222 3028700 ChemDiv3_008855 Cc1nnn(n1)C2(CC3CC4CC(CC(=O)Nc5ccc(Cl)cc5)(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C12 compound treatment 3400.0 2860.0 1.01 520.0 -188.0 -0.14 0.6146 0.6006 3028703 ChemDiv3_008856 CCOC(=O)N1CCC(CC1)NC(=O)c2ccc3Sc4ccccc4C(=Nc3c2)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C13 compound treatment 440.0 -104.0 -0.04 840.0 132.0 0.1 0.0459 0.4242 3028704 ChemDiv3_008857 Cc1ccc(c(C)c1)S(=O)(=O)Nc2ccc3C(=O)OCc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C14 compound treatment 400.0 -144.0 -0.05 240.0 -468.0 -0.36 -0.2899 -0.7995 3121940 ChemDiv3_008858 CCC(C)NC(=O)c1ccc2Sc3ccc(Cl)cc3C(=Nc2c1)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C15 compound treatment 400.0 -144.0 -0.05 280.0 -428.0 -0.33 -0.2682 -0.8073 3028705 ChemDiv3_008859 COc1cc(Cc2nnc(o2)C(=O)NC(C)C)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C16 compound treatment 1000.0 456.0 0.16 200.0 -508.0 -0.39 -0.1611 -0.3818 3121941 ChemDiv3_008860 O=C(CN1CCN(Cc2ccccc2)C1=O)NC3CCCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C17 compound treatment 3400.0 2860.0 1.01 360.0 -348.0 -0.27 0.5278 0.5037 3028708 ChemDiv3_008861 O=C1OCc2cc(NS(=O)(=O)c3ccc(cc3)C4CCCCC4)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C18 compound treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 3121942 ChemDiv3_008862 COC(CNC(=O)/C=C/1\Sc2ccccc2NC1=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C19 compound treatment 1080.0 536.0 0.19 280.0 -428.0 -0.33 -0.0976 -0.2573 3121943 ChemDiv3_008863 Clc1cccc(c1)c2nnc(o2)C(=O)NC3CCCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C20 compound treatment 3160.0 2620.0 0.93 320.0 -388.0 -0.3 0.4459 0.4575 3028711 ChemDiv3_008864 CN1C(=O)/C(=C/c2ccc(cc2)C(=O)NCc3ccccc3)/Oc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C21 compound treatment 1040.0 496.0 0.18 280.0 -428.0 -0.33 -0.1076 -0.289 3121944 ChemDiv3_008865 CCOC(=O)c1nnc(Cc2ccc(C)cc2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C22 compound treatment 960.0 416.0 0.15 320.0 -388.0 -0.3 -0.106 -0.3191 3121945 ChemDiv3_008866 CC1CC(C)CN(C1)C(=O)c2ccc3S/C(=C\c4cccc(Cl)c4)/C(=O)N(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C23 mock treatment 440.0 -104.0 -0.04 280.0 -428.0 -0.33 -0.2581 -0.7815 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 C24 mock treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D01 compound treatment 3440.0 2900.0 1.03 1160.0 452.0 0.35 0.9721 0.8963 3028714 ChemDiv3_008867 COc1ccc(/C=C/2\Oc3ccccc3N(CC(=O)N4CCOCC4)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D02 compound treatment 1720.0 1180.0 0.42 360.0 -348.0 -0.27 0.1064 0.2147 3121946 ChemDiv3_008868 NC(=O)CSC1=Nc2ccccc2C3=NC(C(=O)N31)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D03 compound treatment 360.0 -184.0 -0.07 200.0 -508.0 -0.39 -0.3216 -0.8141 3121947 ChemDiv3_008869 CC(NC(=O)CN1C(=O)/C(=C/c2ccccc2C)/Sc3ccccc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D04 compound treatment 440.0 -104.0 -0.04 360.0 -348.0 -0.27 -0.2147 -0.7971 3028717 ChemDiv3_008870 CC(C)NC(=S)Nc1ccc2nc(cc(C)c2c1)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D05 compound treatment 2520.0 1980.0 0.7 280.0 -428.0 -0.33 0.2636 0.3405 3121948 ChemDiv3_008871 Cc1cc(NC(=O)CC2CCCCC2)nc3c4ccccc4oc(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D06 compound treatment 2040.0 1500.0 0.53 320.0 -388.0 -0.3 0.1649 0.271 3028719 ChemDiv3_008872 Cc1ccc(cc1)N2C(=O)C3C4OC(CNC(=S)Nc5ccc(Br)cc5)(C=C4)C3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D07 compound treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 3028774 ChemDiv3_008873 Cn1cc(CC(=O)NCCN2CCN(CC2)c3cccc(Cl)c3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D08 compound treatment 400.0 -144.0 -0.05 320.0 -388.0 -0.3 -0.2465 -0.8164 1464635 ChemDiv3_008874 O=C(OCn1nnc2ccccc2c1=O)C3(CC4CC5CC(C4)C3)C5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D09 compound treatment 2640.0 2100.0 0.74 280.0 -428.0 -0.33 0.2937 0.3613 3028776 ChemDiv3_008875 COCCn1/c(=N/C(=O)CSCC(=O)N2CCCc3ccccc23)/sc4cc(OC)ccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D10 compound treatment 520.0 -23.8 -0.01 640.0 -67.6 -0.05 -0.0426 -0.8113 3028777 ChemDiv3_008876 Cc1ccc(cc1)c2nn(c3cccc(F)c3)c4c2cnc5cc(F)c(F)cc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D11 compound treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 3028778 ChemDiv3_008877 CSc1cccc(NC(=O)C2CCN(CC2)S(=O)(=O)c3c(C)n[nH]c3C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D12 compound treatment 440.0 -104.0 -0.04 360.0 -348.0 -0.27 -0.2147 -0.7971 3028780 ChemDiv3_008878 CC1COC(=N1)c2cccn2Cc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D13 compound treatment 3320.0 2780.0 0.98 320.0 -388.0 -0.3 0.486 0.4724 3121949 ChemDiv3_008879 CC1CCCCN1S(=O)(=O)c2ccc3N(CCc3c2)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D14 compound treatment 2200.0 1660.0 0.59 360.0 -348.0 -0.27 0.2268 0.3514 3028783 ChemDiv3_008880 CS(=O)(=O)C1=NN2C(=NC(=O)/C(=C/c3ccco3)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D15 compound treatment 240.0 -304.0 -0.11 400.0 -308.0 -0.24 -0.2432 -0.9368 3121950 ChemDiv3_008881 CC(C)Nc1c(nc2nc(C)cc(C)n12)c3ccc(C)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D16 compound treatment 2360.0 1820.0 0.64 320.0 -388.0 -0.3 0.2452 0.3455 3028785 ChemDiv3_008882 CN(Cc1ccccc1)S(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D17 compound treatment 3080.0 2540.0 0.9 360.0 -348.0 -0.27 0.4475 0.4769 3121951 ChemDiv3_008883 CS(=O)(=O)Nc1cccc(c1)C2=NN(C(C2)c3cccs3)C(=O)CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D18 compound treatment 2320.0 1780.0 0.63 520.0 -188.0 -0.14 0.3437 0.5318 3121952 ChemDiv3_008884 Cc1ccccc1NS(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D19 compound treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 3028790 ChemDiv3_008885 O=C(CSc1nnc(CNC(=O)c2ccco2)o1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D20 compound treatment 2200.0 1660.0 0.59 240.0 -468.0 -0.36 0.1616 0.2347 3121953 ChemDiv3_008886 COc1ccc(cc1)N(C)C(=O)C2CCN(CC2)S(=O)(=O)c3cccc4nsnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D21 compound treatment 2160.0 1620.0 0.57 320.0 -388.0 -0.3 0.195 0.3019 3028792 ChemDiv3_008887 CC(C)NC(=O)c1cn(C2CCCCC2)c(=O)c3n(C)c4ccccc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D22 compound treatment 4080.0 3540.0 1.25 240.0 -468.0 -0.36 0.6332 0.4853 3121954 ChemDiv3_008888 Cc1ccc2cc3cc(oc3nc2c1)C(=O)N4CCN(CC4)c5cc(Cl)ccc5C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D23 mock treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 D24 mock treatment 320.0 -224.0 -0.08 320.0 -388.0 -0.3 -0.2665 -0.8655 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E01 compound treatment 2560.0 2020.0 0.72 600.0 -108.0 -0.08 0.4474 0.6213 3121955 ChemDiv3_008889 CC1CC(C)CN(C1)S(=O)(=O)c2ccc(NC(=O)C3COc4ccccc4O3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E02 compound treatment 360.0 -184.0 -0.07 1320.0 612.0 0.47 0.2864 0.6033 3028849 ChemDiv3_008890 CC(C)Sc1nc2ccccc2n3cnnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E03 compound treatment 800.0 256.0 0.09 440.0 -268.0 -0.21 -0.081 -0.3605 3028852 ChemDiv3_008891 COc1ccc(cc1)C(=O)/C=C/2\Nc3ccc(cc3NC2=O)C(=O)NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E04 compound treatment 440.0 -104.0 -0.04 400.0 -308.0 -0.24 -0.193 -0.8076 3028853 ChemDiv3_008892 COc1ccc(cc1OC)S(=O)(=O)Nc2c(O)c3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E05 compound treatment 760.0 216.0 0.08 360.0 -348.0 -0.27 -0.1344 -0.4842 3028857 ChemDiv3_008893 OC1C(NN=C1c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E06 compound treatment 560.0 16.3 0.01 640.0 -67.6 -0.05 -0.0326 -0.6247 3028859 ChemDiv3_008894 CCN(C(=O)c1cc2cc3ccc(C)cc3nc2s1)c4ccc(C)c(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E07 compound treatment 480.0 -63.8 -0.02 800.0 92.4 0.07 0.0342 0.459 3028862 ChemDiv3_008895 CC(NC(=O)CCc1nc2ccccc2[nH]1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E08 compound treatment 680.0 136.0 0.05 4600.0 3890.0 2.99 2.1472 0.7184 3028864 ChemDiv3_008896 CCCN(C(=O)c1cc2cc3ccc(OC)cc3nc2s1)c4ccc(CC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E09 compound treatment 720.0 176.0 0.06 520.0 -188.0 -0.14 -0.0576 -0.367 3121956 ChemDiv3_008897 C(Nc1nc2ccccc2n3nnnc13)C4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E10 compound treatment 7280.0 6740.0 2.39 840.0 132.0 0.1 1.7616 0.7365 3122138 ChemDiv3_008898 COc1ccc2nc3sc(cc3cc2c1)C(=O)N(C)c4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E11 compound treatment 880.0 336.0 0.12 560.0 -148.0 -0.11 0.0042 0.0257 3028868 ChemDiv3_008899 OC(=O)C1(CC2CC3C1)CC(C2)(C3)n4ncc(NCc5ccc(F)cc5)c(Cl)c4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E12 compound treatment 440.0 -104.0 -0.04 480.0 -228.0 -0.17 -0.1496 -0.8377 3122139 ChemDiv3_008900 CCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)NCC(OC)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E13 compound treatment 560.0 16.3 0.01 440.0 -268.0 -0.21 -0.1412 -0.687 3122140 ChemDiv3_008901 COc1ccccc1Cc2nnc(o2)C(=O)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E14 compound treatment 720.0 176.0 0.06 3680.0 2970.0 2.28 1.6578 0.7262 3028927 ChemDiv3_008902 CN(Cc1ccccc1)C(=O)c2ccc3Sc4ccc(Cl)cc4C(=Nc3c2)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E15 compound treatment 880.0 336.0 0.12 640.0 -67.6 -0.05 0.0477 0.3664 3028930 ChemDiv3_008903 CCOC(=O)c1[nH]c2ccc(OC)cc2c1C(SCC(=O)O)c3ccc(cc3)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E16 compound treatment 560.0 16.3 0.01 720.0 12.4 0.01 0.0108 0.971 3028931 ChemDiv3_008904 COC(CNC(=O)CN1CCN(Cc2ccccc2)C1=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E17 compound treatment 560.0 16.3 0.01 360.0 -348.0 -0.27 -0.1846 -0.6917 3028935 ChemDiv3_008905 Cc1ccc(C)c(c1)N2CCN(CCCNC(=O)c3nnc(Cc4c(F)cccc4Cl)o3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E18 compound treatment 400.0 -144.0 -0.05 360.0 -348.0 -0.27 -0.2247 -0.8273 3028936 ChemDiv3_008906 CC1CCCC(NC(=O)/C=C/2\Sc3ccccc3NC2=O)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E19 compound treatment 600.0 56.3 0.02 640.0 -67.6 -0.05 -0.0226 -0.4062 3028938 ChemDiv3_008907 OCCNC(=O)c1nnc(o1)c2cccc(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E20 compound treatment 1320.0 776.0 0.28 560.0 -148.0 -0.11 0.1146 0.3849 3122141 ChemDiv3_008908 COc1cccc(c1)N2CCN(CC2)C(=O)c3ccc(/C=C/4\Oc5ccccc5N(C)C4=O)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E21 compound treatment 560.0 16.3 0.01 1360.0 652.0 0.5 0.3582 0.7152 3028941 ChemDiv3_008909 Cc1cc(C)n(n1)c2nc3ccccc3nc2N4CCN(CC4)S(=O)(=O)c5ccc(F)c(C)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E22 compound treatment 920.0 376.0 0.13 1480.0 772.0 0.59 0.5137 0.8451 3122142 ChemDiv3_008910 CN1C(=O)/C(=C/c2cccc(Cl)c2)/Sc3ccc(cc13)C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E23 mock treatment 2920.0 2380.0 0.84 1040.0 332.0 0.26 0.7765 0.8817 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 E24 mock treatment 1480.0 936.0 0.33 480.0 -228.0 -0.17 0.1113 0.2966 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F01 compound treatment 1000.0 456.0 0.16 1760.0 1050.0 0.81 0.6858 0.8322 3028944 ChemDiv3_008911 Clc1cccc(/C=C\2/Oc3ccccc3N(CC(=O)NCC4COc5ccccc5O4)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F02 compound treatment 640.0 96.3 0.03 640.0 -67.6 -0.05 -0.0125 -0.202 3122143 ChemDiv3_008912 CCC(SC1=Nc2ccccc2C3=NC(C(=O)N31)c4ccccc4)C(=O)Nc5cccc(OC)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F03 compound treatment 600.0 56.3 0.02 1560.0 852.0 0.65 0.4769 0.7283 3028946 ChemDiv3_008913 CNC(=O)CN1C(=O)/C(=C/c2ccccc2C)/Sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F04 compound treatment 2760.0 2220.0 0.79 1680.0 972.0 0.75 1.0838 0.9997 3122144 ChemDiv3_008914 Cc1cc(nc2ccc(NC(=S)NCCN3CCOCC3)cc12)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F05 compound treatment 1880.0 1340.0 0.47 920.0 212.0 0.16 0.4505 0.8987 3122145 ChemDiv3_008915 CC(C)C(=O)Nc1cc(C)c2c(=O)oc3ccccc3c2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F06 compound treatment 640.0 96.3 0.03 1480.0 772.0 0.59 0.4435 0.7466 3122146 ChemDiv3_008916 Cc1ccc(cc1)N2C(=O)C3C4OC(CNC(=S)NCc5ccccc5)(C=C4)C3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F07 compound treatment 640.0 96.3 0.03 760.0 52.4 0.04 0.0526 0.9967 3029128 ChemDiv3_008917 CN1CCN(CC1)c2ccccc2NC(=O)Cc3cn(C)c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F08 compound treatment 840.0 296.0 0.11 1720.0 1010.0 0.78 0.6239 0.7955 1580348 ChemDiv3_008918 Clc1ccc(cc1)C2(CCCC2)C(=O)OCn3nnc4ccccc4c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F09 compound treatment 880.0 336.0 0.12 1000.0 292.0 0.22 0.2431 0.9562 3029132 ChemDiv3_008919 CCOC(=O)N1CCN(CC1)C(=O)CSCC(=O)/N=c/2\sc3ccccc3n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F10 compound treatment 1760.0 1220.0 0.43 1000.0 292.0 0.22 0.4638 0.9537 3029134 ChemDiv3_008920 Cc1ccc(cc1)c2nn(c3ccc(C)cc3)c4c2cnc5c(F)cccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F11 compound treatment 440.0 -104.0 -0.04 800.0 92.4 0.07 0.0241 0.3021 3029137 ChemDiv3_008921 Cc1noc(C)c1S(=O)(=O)NC2CCCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F12 compound treatment 1040.0 496.0 0.18 1480.0 772.0 0.59 0.5438 0.8791 3029139 ChemDiv3_008922 CCSCC1COC(=N1)c2cccn2Cc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F13 compound treatment 1320.0 776.0 0.28 960.0 252.0 0.19 0.3317 0.9852 3029141 ChemDiv3_008923 CCN(c1ccccc1)S(=O)(=O)c2ccc3N(CCc3c2)C(=O)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F14 compound treatment 1560.0 1020.0 0.36 1640.0 932.0 0.72 0.7611 0.9496 3029212 ChemDiv3_008924 CCc1ccc(/C=C/2\C(=N)N3N=C(SC3=NC2=O)S(=O)(=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F15 compound treatment 400.0 -144.0 -0.05 3280.0 2570.0 1.97 1.3604 0.6886 3029215 ChemDiv3_008925 Cc1ccc(o1)c2nc3nc(C)cc(C)n3c2Nc4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F16 compound treatment 920.0 376.0 0.13 3600.0 2890.0 2.22 1.6646 0.7483 3029216 ChemDiv3_008926 Fc1cccc(NS(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F17 compound treatment 1680.0 1140.0 0.4 760.0 52.4 0.04 0.3135 0.7739 3029219 ChemDiv3_008927 COc1cc(cc(OC)c1OC)C(=O)NCc2nnc(SCC(=O)N3CCc4ccccc34)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F18 compound treatment 360.0 -184.0 -0.07 1480.0 772.0 0.59 0.3732 0.6256 3029220 ChemDiv3_008928 Cc1cccc(CCNS(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CCC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F19 compound treatment 640.0 96.3 0.03 2680.0 1970.0 1.51 1.0949 0.7229 3029222 ChemDiv3_008929 COc1ccc(cc1OC)C(=O)NCc2nnc(SCC(=O)Nc3cc(C)cc(C)c3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F20 compound treatment 920.0 376.0 0.13 3240.0 2530.0 1.94 1.4691 0.7539 1538082 ChemDiv3_008930 Cc1cccc(c1)n2c3ccccc3cc4c(=O)[nH]c(=O)nc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F21 compound treatment 1920.0 1380.0 0.49 3200.0 2490.0 1.91 1.6983 0.86 3029226 ChemDiv3_008931 COC(=O)CSc1nc([nH]c1c2ccc(C)cc2)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F22 compound treatment 640.0 96.3 0.03 1200.0 492.0 0.38 0.2915 0.7678 3122147 ChemDiv3_008932 Cc1cccc(CN2CCC(CNC(=O)c3cc4cc5ccc(C)cc5nc4o3)CC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F23 mock treatment 440.0 -104.0 -0.04 3160.0 2450.0 1.88 1.3053 0.6932 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 F24 mock treatment 680.0 136.0 0.05 6320.0 5610.0 4.31 3.0809 0.715 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G01 compound treatment 680.0 136.0 0.05 1240.0 532.0 0.41 0.3232 0.7853 3029231 ChemDiv3_008933 O=C(Nc1cccc(NC(=O)c2ccccc2)c1)C3COc4ccccc4O3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G02 compound treatment 2840.0 2300.0 0.81 400.0 -308.0 -0.24 0.409 0.4823 1328889 ChemDiv3_008934 Clc1c(CN2CCCC2)c(=O)oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G03 compound treatment 440.0 -104.0 -0.04 480.0 -228.0 -0.17 -0.1496 -0.8377 3029233 ChemDiv3_008935 Nc1nc(n[nH]1)c2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G04 compound treatment 720.0 176.0 0.06 3560.0 2850.0 2.19 1.5927 0.727 3122148 ChemDiv3_008936 Oc1c(NS(=O)(=O)c2ccc3CCCCc3c2)c(=O)oc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G05 compound treatment 760.0 216.0 0.08 600.0 -108.0 -0.08 -0.0042 -0.0369 3122149 ChemDiv3_008937 Fc1ccc(CNC(=O)CCc2nc3ccccc3[nH]2)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G06 compound treatment 320.0 -224.0 -0.08 440.0 -268.0 -0.21 -0.2014 -0.9144 3029646 ChemDiv3_008938 Cc1ccc2cc3cc(sc3nc2c1)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G07 compound treatment 800.0 256.0 0.09 2040.0 1330.0 1.02 0.7876 0.7669 3122150 ChemDiv3_008939 Clc1nc2ccc(cc2n3cnnc13)C(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G08 compound treatment 480.0 -63.8 -0.02 440.0 -268.0 -0.21 -0.1613 -0.7802 1751250 ChemDiv3_008940 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G09 compound treatment 360.0 -184.0 -0.07 360.0 -348.0 -0.27 -0.2348 -0.8547 3122151 ChemDiv3_008941 CC(CNC(=O)c1nnc(Cc2ccc(Cl)cc2)o1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G10 compound treatment 1960.0 1420.0 0.5 640.0 -67.6 -0.05 0.3186 0.6307 3028652 ChemDiv3_008942 COc1ccc2nc3sc(cc3cc2c1)C(=O)N(CC=C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G11 compound treatment 440.0 -104.0 -0.04 320.0 -388.0 -0.3 -0.2364 -0.7886 3122152 ChemDiv3_008943 CC(C)n1nnc(CC(=O)NN)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G12 compound treatment 1160.0 616.0 0.22 360.0 -348.0 -0.27 -0.0341 -0.0989 3122153 ChemDiv3_008944 CCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G13 compound treatment 680.0 136.0 0.05 440.0 -268.0 -0.21 -0.1111 -0.5264 1026727 ChemDiv3_008945 COc1nc2ccccc2nc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G14 compound treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 3122154 ChemDiv3_008946 CCC1=Nc2cc(ccc2Sc3ccc(C)cc13)C(=O)N(C)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G15 compound treatment 480.0 -63.8 -0.02 400.0 -308.0 -0.24 -0.183 -0.7713 3028659 ChemDiv3_008947 Fc1ccc(Cc2nnn[nH]2)c(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G16 compound treatment 2520.0 1980.0 0.7 400.0 -308.0 -0.24 0.3288 0.4444 3122155 ChemDiv3_008948 O=C(CN1CCN(Cc2ccccc2)C1=O)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G17 compound treatment 480.0 -63.8 -0.02 320.0 -388.0 -0.3 -0.2264 -0.7587 3028663 ChemDiv3_008949 Cc1ccc(Cc2nnn[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G18 compound treatment 600.0 56.3 0.02 800.0 92.4 0.07 0.0643 0.8721 3122156 ChemDiv3_008950 O=C(NCCc1ccccc1)/C=C/2\Sc3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G19 compound treatment 520.0 -23.8 -0.01 600.0 -108.0 -0.08 -0.0644 -0.7752 3028666 ChemDiv3_008951 Clc1cccc(c1)c2nnc(o2)C(=O)NCc3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G20 compound treatment 520.0 -23.8 -0.01 520.0 -188.0 -0.14 -0.1078 -0.7472 3122157 ChemDiv3_008952 CN1C(=O)/C(=C/c2ccc(cc2)C(=O)N3CCC(Cc4ccccc4)CC3)/Oc5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G21 compound treatment 320.0 -224.0 -0.08 920.0 212.0 0.16 0.0592 0.3263 3122158 ChemDiv3_008953 CC1CN(CCN1c2ccc(C)cc2)c3cnn(c4nc5ccccc5s4)c(=O)c3N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G22 compound treatment 320.0 -224.0 -0.08 1200.0 492.0 0.38 0.2112 0.5467 3028721 ChemDiv3_008954 CC1CC(C)CN(CCCNC(=O)c2ccc3S/C(=C\c4ccccc4F)/C(=O)N(C)c3c2)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G23 mock treatment 360.0 -184.0 -0.07 560.0 -148.0 -0.11 -0.1262 -0.9655 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 G24 mock treatment 560.0 16.3 0.01 840.0 132.0 0.1 0.076 0.746 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H01 compound treatment 720.0 176.0 0.06 1160.0 452.0 0.35 0.2898 0.8212 3122159 ChemDiv3_008955 Fc1ccccc1/C=C/2\Oc3ccccc3N(CC(=O)N4CCCC4)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H02 compound treatment 560.0 16.3 0.01 1080.0 372.0 0.29 0.2062 0.7212 3122160 ChemDiv3_008956 CCC(SC1=Nc2ccccc2C3=NC(C(=O)N31)c4ccccc4)C(=O)NCc5ccc(C)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H03 compound treatment 600.0 56.3 0.02 320.0 -388.0 -0.3 -0.1963 -0.6582 3028724 ChemDiv3_008957 FC(F)(F)c1ccc(/C=C\2/Sc3ccccc3N(CC(=O)N4CCc5ccccc5C4)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H04 compound treatment 560.0 16.3 0.01 440.0 -268.0 -0.21 -0.1412 -0.687 3122161 ChemDiv3_008958 CCc1ccc(CNC(=S)Nc2ccc3nc(cc(C)c3c2)N4CCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H05 compound treatment 440.0 -104.0 -0.04 320.0 -388.0 -0.3 -0.2364 -0.7886 3028730 ChemDiv3_008959 Cc1cc(NC(=O)C2CCCCC2)nc3c4ccccc4oc(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H06 compound treatment 360.0 -184.0 -0.07 880.0 172.0 0.13 0.0475 0.322 1209934 ChemDiv3_008960 O=C(OCn1nnc2ccccc2c1=O)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H07 compound treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 3122162 ChemDiv3_008961 COc1ccc(CNC(=O)Cc2cn(C)c3ccccc23)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H08 compound treatment 720.0 176.0 0.06 360.0 -348.0 -0.27 -0.1445 -0.5272 1398426 ChemDiv3_008962 COCC(=O)OCn1nnc2ccccc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H09 compound treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 3122346 ChemDiv3_008963 Cn1/c(=N/C(=O)CSCC(=O)N2CCCc3ccccc23)/sc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H10 compound treatment 720.0 176.0 0.06 360.0 -348.0 -0.27 -0.1445 -0.5272 3028735 ChemDiv3_008964 COc1cccc(c1)c2nn(c3ccccc3)c4c2cnc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H11 compound treatment 680.0 136.0 0.05 320.0 -388.0 -0.3 -0.1762 -0.5846 3122347 ChemDiv3_008965 CC1CCN(CC1)S(=O)(=O)c2c(C)noc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H12 compound treatment 480.0 -63.8 -0.02 480.0 -228.0 -0.17 -0.1395 -0.792 3028737 ChemDiv3_008966 CCC1COC(=N1)c2cccn2Cc3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H13 compound treatment 360.0 -184.0 -0.07 600.0 -108.0 -0.08 -0.1045 -0.9931 3028795 ChemDiv3_008967 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)Nc3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H14 compound treatment 880.0 336.0 0.12 1120.0 412.0 0.32 0.3082 0.911 3122348 ChemDiv3_008968 CC(C)CS(=O)(=O)C1=NN2C(=NC(=O)/C(=C/c3c(C)[nH]c4ccc(C)cc34)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H15 compound treatment 440.0 -104.0 -0.04 360.0 -348.0 -0.27 -0.2147 -0.7971 3028797 ChemDiv3_008969 CSc1ccc(cc1)c2nc3ncccn3c2Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H16 compound treatment 320.0 -224.0 -0.08 320.0 -388.0 -0.3 -0.2665 -0.8655 3122349 ChemDiv3_008970 CN(c1cccc(C)c1)S(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H17 compound treatment 2360.0 1820.0 0.64 2520.0 1810.0 1.39 1.4395 0.9388 3028798 ChemDiv3_008971 Fc1cccc(NC(=O)CSc2nnc(CNC(=O)COc3ccc(Cl)cc3)o2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H18 compound treatment 360.0 -184.0 -0.07 480.0 -228.0 -0.17 -0.1696 -0.9097 3122350 ChemDiv3_008972 O=C(C1CCC1)N2CCc3cc(ccc23)S(=O)(=O)NCCN4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H19 compound treatment 400.0 -144.0 -0.05 320.0 -388.0 -0.3 -0.2465 -0.8164 3122351 ChemDiv3_008973 COc1cccc(NC(=O)c2cn(C3CCCC3)c(=O)c4n(C)c5ccccc5c24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H20 compound treatment 320.0 -224.0 -0.08 600.0 -108.0 -0.08 -0.1145 -0.9998 1742555 ChemDiv3_008974 Cn1c(=O)nc2n(c3ccc(Cl)c(Cl)c3)c4ccccc4cc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H21 compound treatment 560.0 16.3 0.01 800.0 92.4 0.07 0.0542 0.762 3122352 ChemDiv3_008975 Cc1ccc(cc1)c2[nH]c(nc2SCC(=O)NCC3CCCO3)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H22 compound treatment 320.0 -224.0 -0.08 720.0 12.4 0.01 -0.0494 -0.6178 3028802 ChemDiv3_008976 Cc1ccc2cc3cc(oc3nc2c1)C(=O)NCC4(CCCC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H23 mock treatment 320.0 -224.0 -0.08 5760.0 5050.0 3.88 2.6866 0.6925 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 H24 mock treatment 360.0 -184.0 -0.07 1240.0 532.0 0.41 0.2429 0.5869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I01 compound treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 3122353 ChemDiv3_008977 O=C(c1n[nH]c2CCCCc12)n3ccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I02 compound treatment 320.0 -224.0 -0.08 600.0 -108.0 -0.08 -0.1145 -0.9998 3028804 ChemDiv3_008978 CCOC(=O)c1ncn(n1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I03 compound treatment 280.0 -264.0 -0.09 360.0 -348.0 -0.27 -0.2549 -0.9012 3122354 ChemDiv3_008979 CC1=NN(C(=O)C1)c2nc3ccccc3nc2Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I04 compound treatment 280.0 -264.0 -0.09 280.0 -428.0 -0.33 -0.2983 -0.8738 3028806 ChemDiv3_008980 OC(=O)CSc1nc2ccccc2n3cnnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I05 compound treatment 440.0 -104.0 -0.04 360.0 -348.0 -0.27 -0.2147 -0.7971 3122355 ChemDiv3_008981 O=C(CN1CC(CC1=O)c2ccccc2)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I06 compound treatment 360.0 -184.0 -0.07 360.0 -348.0 -0.27 -0.2348 -0.8547 3122356 ChemDiv3_008982 CCc1cccc(NC(=O)c2cc3cc4ccc(C)cc4nc3s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I07 compound treatment 2400.0 1860.0 0.66 360.0 -348.0 -0.27 0.2769 0.3898 3028808 ChemDiv3_008983 Brc1ccc(cc1)S(=O)(=O)Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I08 compound treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 3122357 ChemDiv3_008984 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCCC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I09 compound treatment 480.0 -63.8 -0.02 280.0 -428.0 -0.33 -0.2481 -0.754 3028810 ChemDiv3_008985 Clc1ccc(Cc2nnc(o2)C(=O)NC3CCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I10 compound treatment 800.0 256.0 0.09 360.0 -348.0 -0.27 -0.1244 -0.4413 3122358 ChemDiv3_008986 CCc1cccc(NC(=O)c2cc3cc4cc(OC)ccc4nc3s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I11 compound treatment 400.0 -144.0 -0.05 320.0 -388.0 -0.3 -0.2465 -0.8164 3122359 ChemDiv3_008987 CCOC(=O)c1nnc(Cc2ccc(F)cc2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I12 compound treatment 680.0 136.0 0.05 320.0 -388.0 -0.3 -0.1762 -0.5846 3028873 ChemDiv3_008988 CCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I13 compound treatment 760.0 216.0 0.08 440.0 -268.0 -0.21 -0.091 -0.4151 3122360 ChemDiv3_008989 COc1cc(Cc2nnc(o2)C(=O)NC3CCCCCC3)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I14 compound treatment 2000.0 1460.0 0.52 3000.0 2290.0 1.76 1.6097 0.8776 3122361 ChemDiv3_008990 CCC1=Nc2cc(ccc2Sc3ccc(Br)cc13)C(=O)NCCCN4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I15 compound treatment 560.0 16.3 0.01 360.0 -348.0 -0.27 -0.1846 -0.6917 3028877 ChemDiv3_008991 CCOC(=O)c1nnc(o1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I16 compound treatment 1240.0 696.0 0.25 1000.0 292.0 0.22 0.3334 0.9989 3122362 ChemDiv3_008992 COC(CNC(=O)/C=C/1\Sc2ccccc2N(Cc3ccccc3F)C1=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I17 compound treatment 400.0 -144.0 -0.05 400.0 -308.0 -0.24 -0.203 -0.8404 3028879 ChemDiv3_008993 COc1ccc(cc1)N2CCN(CCNC(=O)c3nnc(Cc4ccccc4Cl)o3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I18 compound treatment 280.0 -264.0 -0.09 360.0 -348.0 -0.27 -0.2549 -0.9012 3122363 ChemDiv3_008994 O=C(NCCCN1CCC(Cc2ccccc2)CC1)/C=C/3\Sc4ccccc4NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I19 compound treatment 280.0 -264.0 -0.09 280.0 -428.0 -0.33 -0.2983 -0.8738 3028881 ChemDiv3_008995 Cc1ccc(Cc2nnc(o2)C(=O)NCCC3=CCCCC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I20 compound treatment 480.0 -63.8 -0.02 320.0 -388.0 -0.3 -0.2264 -0.7587 3122364 ChemDiv3_008996 Fc1ccccc1CN2C(=O)/C(=C/c3ccc(cc3)C(=O)NCc4cccnc4)/Sc5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I21 compound treatment 280.0 -264.0 -0.09 280.0 -428.0 -0.33 -0.2983 -0.8738 3122365 ChemDiv3_008997 Cc1nnn(n1)C2(CC3CC4CC(C3)(C2)C(=O)N5CCCCCC5)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I22 compound treatment 280.0 -264.0 -0.09 280.0 -428.0 -0.33 -0.2983 -0.8738 3028883 ChemDiv3_008998 CC1CCN(CC1)C(=O)c2ccc3S/C(=C\c4cccc(C)c4)/C(=O)N(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I23 mock treatment 360.0 -184.0 -0.07 400.0 -308.0 -0.24 -0.2131 -0.8698 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 I24 mock treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J01 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122366 ChemDiv3_008999 CC1CCCC(NC(=O)CN2C(=O)/C(=C\c3ccccc3Cl)/Oc4ccccc24)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J02 compound treatment 280.0 -264.0 -0.09 360.0 -348.0 -0.27 -0.2549 -0.9012 3028885 ChemDiv3_009000 CCN(Cc1ccccc1)C(=O)CSC2=Nc3ccccc3C4=NC(C(=O)N42)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J03 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122367 ChemDiv3_009001 CN(Cc1ccco1)C(=O)CN2C(=O)/C(=C\c3ccc(cc3)C(F)(F)F)/Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J04 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122368 ChemDiv3_009002 Cc1cc(nc2ccc(NC(=S)NCCN3CCc4ccccc4C3)cc12)N5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J05 compound treatment 240.0 -304.0 -0.11 360.0 -348.0 -0.27 -0.2649 -0.9204 3028889 ChemDiv3_009003 Cc1cc(NC(=O)CCC2CCCC2)nc3c4ccccc4oc(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J06 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 3028815 ChemDiv3_009004 O=C(OCn1nnc2ccccc2c1=O)/C=C\c3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J07 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122369 ChemDiv3_009005 COC(=O)c1ccc2n(C)/c(=N/C(=O)CSC(=O)C)/sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J08 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3028817 ChemDiv3_009006 O=C(CCCc1ccccc1)OCn2nnc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J09 compound treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 3122370 ChemDiv3_009007 CCn1/c(=N/C(=O)CSCC(=O)Nc2cc(C)on2)/sc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J10 compound treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 3122371 ChemDiv3_009008 COc1ccc(cc1OC)c2nn(c3ccc(C)c(Cl)c3)c4c2cnc5ccc(F)cc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J11 compound treatment 560.0 16.3 0.01 2680.0 1970.0 1.51 1.0748 0.7098 3028822 ChemDiv3_009009 CC(NS(=O)(=O)c1c(C)noc1C)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J12 compound treatment 800.0 256.0 0.09 320.0 -388.0 -0.3 -0.1461 -0.4697 3122372 ChemDiv3_009010 CCC(C)C1COC(=N1)c2cccn2Cc3c(C)cc(C)cc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J13 compound treatment 480.0 -63.8 -0.02 240.0 -468.0 -0.36 -0.2698 -0.7502 3028824 ChemDiv3_009011 CCCCN(C)S(=O)(=O)c1ccc2N(CCc2c1)C(=O)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J14 compound treatment 4240.0 3700.0 1.31 2880.0 2170.0 1.67 2.1065 0.9929 3122373 ChemDiv3_009012 CC(C)CS(=O)(=O)C1=NN2C(=NC(=O)/C(=C/c3ccc(N(C)C)c(Br)c3)/C2=N)S1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J15 compound treatment 640.0 96.3 0.03 1000.0 292.0 0.22 0.1829 0.8054 3028829 ChemDiv3_009013 CCc1cccc(C)c1Nc2c(nc3ncccn23)c4ccccc4O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J16 compound treatment 400.0 -144.0 -0.05 440.0 -268.0 -0.21 -0.1813 -0.8566 3122560 ChemDiv3_009014 O=C(C1CC1)N2CCc3cc(ccc23)S(=O)(=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J17 compound treatment 720.0 176.0 0.06 280.0 -428.0 -0.33 -0.1879 -0.5623 3028893 ChemDiv3_009015 Fc1cccc(Cl)c1C(=O)NCc2nnc(SCC(=O)N3CCCC3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J18 compound treatment 560.0 16.3 0.01 400.0 -308.0 -0.24 -0.1629 -0.6896 3122561 ChemDiv3_009016 COc1ccc(N(C)S(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CCC4)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J19 compound treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 3028897 ChemDiv3_009017 COc1ccccc1CNC(=O)c2cn(C3CCCC3)c(=O)c4n(C)c5ccccc5c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J20 compound treatment 3640.0 3100.0 1.1 320.0 -388.0 -0.3 0.5663 0.4976 3122562 ChemDiv3_009018 Cc1ccc2cc3cc(oc3nc2c1)C(=O)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J21 compound treatment 560.0 16.3 0.01 280.0 -428.0 -0.33 -0.228 -0.6946 3122563 ChemDiv3_009019 CSc1ccc(cc1)c2nc(SCC(=O)NCc3ccco3)c([nH]2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J22 compound treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 3028901 ChemDiv3_009020 Clc1ccccc1CSc2nc3n(ncc3c(=O)[nH]2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J23 mock treatment 240.0 -304.0 -0.11 1720.0 1010.0 0.78 0.4734 0.6033 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 J24 mock treatment 280.0 -264.0 -0.09 800.0 92.4 0.07 -0.016 -0.1362 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K01 compound treatment 320.0 -224.0 -0.08 600.0 -108.0 -0.08 -0.1145 -0.9998 3028903 ChemDiv3_009021 O=C(c1cc(n[nH]1)C2CC2)n3ccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K02 compound treatment 440.0 -104.0 -0.04 400.0 -308.0 -0.24 -0.193 -0.8076 3122564 ChemDiv3_009022 CNc1c(NS(=O)(=O)c2ccc(C)cc2C)c(=O)oc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K03 compound treatment 1040.0 496.0 0.18 520.0 -188.0 -0.14 0.0226 0.0996 3122565 ChemDiv3_009023 O=C(CN1CC(CC1=O)c2ccccc2)NCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K04 compound treatment 880.0 336.0 0.12 360.0 -348.0 -0.27 -0.1043 -0.357 3028906 ChemDiv3_009024 C1Oc2ccc(cc2O1)c3nnn[nH]3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K05 compound treatment 360.0 -184.0 -0.07 2680.0 1970.0 1.51 1.0247 0.676 3029994 ChemDiv3_009025 Cc1cc(C)n(n1)c2nc3cc(C)ccc3nc2N4CCN(CC4)c5cccc(C)c5C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K06 compound treatment 520.0 -23.8 -0.01 240.0 -468.0 -0.36 -0.2598 -0.7235 3029995 ChemDiv3_009026 Cc1ccc2cc3cc(sc3nc2c1)C(=O)NCCN4CCN(CC4)c5cccc(Cl)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K07 compound treatment 360.0 -184.0 -0.07 360.0 -348.0 -0.27 -0.2348 -0.8547 3029996 ChemDiv3_009027 Cc1cc(C)c(c(C)c1)S(=O)(=O)Nc2ccc3[nH]c(=O)[nH]c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K08 compound treatment 320.0 -224.0 -0.08 1080.0 372.0 0.29 0.146 0.4922 3029997 ChemDiv3_009028 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCC4CCN(Cc5cccc(C)c5)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K09 compound treatment 360.0 -184.0 -0.07 360.0 -348.0 -0.27 -0.2348 -0.8547 3029998 ChemDiv3_009029 CC(C)CCNC(=O)c1nnc(Cc2ccc(Cl)cc2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K10 compound treatment 480.0 -63.8 -0.02 440.0 -268.0 -0.21 -0.1613 -0.7802 3029999 ChemDiv3_009030 CC1=Nc2cc(ccc2Sc3ccccc13)C(=O)NCc4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K11 compound treatment 440.0 -104.0 -0.04 360.0 -348.0 -0.27 -0.2147 -0.7971 3122566 ChemDiv3_009031 Fc1ccc(Cc2nnc(o2)C(=O)NCCc3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K12 compound treatment 720.0 176.0 0.06 360.0 -348.0 -0.27 -0.1445 -0.5272 3030000 ChemDiv3_009032 CCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)N4CCc5ccccc5C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K13 compound treatment 1440.0 896.0 0.32 2840.0 2130.0 1.64 1.3824 0.8289 3122567 ChemDiv3_009033 COc1cc(Cc2nnc(o2)C(=O)NCc3ccccc3)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K14 compound treatment 520.0 -23.8 -0.01 680.0 -27.6 -0.02 -0.0209 -0.9184 3122568 ChemDiv3_009034 CCC1=Nc2cc(ccc2Sc3ccc(Br)cc13)C(=O)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K15 compound treatment 4040.0 3500.0 1.24 480.0 -228.0 -0.17 0.7535 0.6016 3030001 ChemDiv3_009035 CNC(=O)c1nnc(o1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K16 compound treatment 800.0 256.0 0.09 400.0 -308.0 -0.24 -0.1027 -0.4059 3030002 ChemDiv3_009036 O=C(NCc1cccnc1)/C=C/2\Sc3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K17 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122569 ChemDiv3_009037 Cc1nnc2c(Nc3ccc4OCOc4c3)nc5ccccc5n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K18 compound treatment 560.0 16.3 0.01 280.0 -428.0 -0.33 -0.228 -0.6946 3122570 ChemDiv3_009038 O=C(/C=C/1\Sc2ccccc2NC1=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K19 compound treatment 320.0 -224.0 -0.08 440.0 -268.0 -0.21 -0.2014 -0.9144 3030003 ChemDiv3_009039 Cc1ccc(Cc2nnc(o2)C(=O)NCc3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K20 compound treatment 800.0 256.0 0.09 560.0 -148.0 -0.11 -0.0158 -0.109 3122571 ChemDiv3_009040 COC(CNC(=O)c1ccc(/C=C/2\Sc3ccccc3N(Cc4ccc(F)cc4)C2=O)cc1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K21 compound treatment 360.0 -184.0 -0.07 1360.0 652.0 0.5 0.3081 0.6099 3030004 ChemDiv3_009041 CCOC(=O)CSc1nc2ccccc2n3cnnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K22 compound treatment 840.0 296.0 0.11 560.0 -148.0 -0.11 -0.0058 -0.0376 3122572 ChemDiv3_009042 CC(C)NC(=O)c1ccc2S/C(=C\c3cccc(C)c3)/C(=O)N(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K23 mock treatment 520.0 -23.8 -0.01 360.0 -348.0 -0.27 -0.1946 -0.7291 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 K24 mock treatment 320.0 -224.0 -0.08 600.0 -108.0 -0.08 -0.1145 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L01 compound treatment 480.0 -63.8 -0.02 480.0 -228.0 -0.17 -0.1395 -0.792 3122573 ChemDiv3_009043 COc1cccc(/C=C\2/Oc3ccccc3N(CC(=O)NCC4CCCO4)C2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L02 compound treatment 440.0 -104.0 -0.04 600.0 -108.0 -0.08 -0.0844 -0.9337 3030005 ChemDiv3_009044 CN(C1CCCCC1)C(=O)CSC2=Nc3ccccc3C4=NC(C(=O)N42)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L03 compound treatment 320.0 -224.0 -0.08 440.0 -268.0 -0.21 -0.2014 -0.9144 3122574 ChemDiv3_009045 CSc1nc2NC(=C(C(C(C)C)n2n1)C(=O)Nc3ccccc3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L04 compound treatment 360.0 -184.0 -0.07 480.0 -228.0 -0.17 -0.1696 -0.9097 3030006 ChemDiv3_009046 Cc1cc(nc2ccc(NC(=S)NC3CCCC3)cc12)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L05 compound treatment 360.0 -184.0 -0.07 440.0 -268.0 -0.21 -0.1914 -0.8879 3122575 ChemDiv3_009047 COc1ccc(cc1)c2noc(CCC(=O)NCCN3CCN(CC3)c4ccccc4F)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L06 compound treatment 440.0 -104.0 -0.04 280.0 -428.0 -0.33 -0.2581 -0.7815 3122576 ChemDiv3_009048 O=C(CC1CCCCC1)OCn2nnc3ccccc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L07 compound treatment 440.0 -104.0 -0.04 400.0 -308.0 -0.24 -0.193 -0.8076 3030007 ChemDiv3_009049 CC(=O)SCC(=O)/N=c/1\sc2cc(F)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L08 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 3122577 ChemDiv3_009050 COc1cc(OC)c2c3n(nc(C)c3cnc2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L09 compound treatment 520.0 -23.8 -0.01 480.0 -228.0 -0.17 -0.1295 -0.7403 3030008 ChemDiv3_009051 CCn1/c(=N/C(=O)CSCC(=O)Nc2nc(cs2)c3ccccc3)/sc4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L10 compound treatment 480.0 -63.8 -0.02 1920.0 1210.0 0.93 0.6422 0.6897 3122578 ChemDiv3_009052 Fc1ccc(Cn2cccc2C3=NC(CO3)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L11 compound treatment 400.0 -144.0 -0.05 400.0 -308.0 -0.24 -0.203 -0.8404 1716980 ChemDiv3_009053 CC1Cc2ccccc2N1S(=O)(=O)c3c(C)noc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L12 compound treatment 520.0 -23.8 -0.01 720.0 12.4 0.01 8.0E-4 0.0614 3030009 ChemDiv3_009054 CCN(C(=O)Cn1cccc1C2=NC(CO2)c3ccccc3)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L13 compound treatment 240.0 -304.0 -0.11 440.0 -268.0 -0.21 -0.2215 -0.9546 3122579 ChemDiv3_009055 CCN(CC)S(=O)(=O)c1ccc2N(CCc2c1)C(=O)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L14 compound treatment 360.0 -184.0 -0.07 440.0 -268.0 -0.21 -0.1914 -0.8879 3122580 ChemDiv3_009056 CC1Cc2cc(ccc2N1C(=O)C)S(=O)(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L15 compound treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 3030010 ChemDiv3_009057 Cc1cc(C)n2c(Nc3cccc(c3)C(F)(F)F)c(nc2n1)c4ccc(O)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L16 compound treatment 840.0 296.0 0.11 440.0 -268.0 -0.21 -0.0709 -0.3075 3122581 ChemDiv3_009058 O=C(C1CC1)N2CCc3cc(ccc23)S(=O)(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L17 compound treatment 440.0 -104.0 -0.04 440.0 -268.0 -0.21 -0.1713 -0.8207 3030011 ChemDiv3_009059 Fc1ccc(NC(=O)CSc2nnc(CNC(=O)c3ccccc3F)o2)c(F)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L18 compound treatment 280.0 -264.0 -0.09 1560.0 852.0 0.65 0.3966 0.5999 3122582 ChemDiv3_009060 CSc1cccc(NC(=O)CCS(=O)(=O)c2ccc3N(CCc3c2)C(=O)C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L19 compound treatment 520.0 -23.8 -0.01 440.0 -268.0 -0.21 -0.1512 -0.7355 3122583 ChemDiv3_009061 COc1ccc(CCNC(=O)c2cn(C3CCCC3)c(=O)c4n(C)c5ccccc5c24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L20 compound treatment 400.0 -144.0 -0.05 760.0 52.4 0.04 -0.0076 -0.1171 3030012 ChemDiv3_009062 CCCCN(CC)C(=O)c1cc2cc3ccc(C)cc3nc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L21 compound treatment 1720.0 1180.0 0.42 600.0 -108.0 -0.08 0.2367 0.5563 3122584 ChemDiv3_009063 Fc1ccc(cc1)c2nc(SCC(=O)NC3CCCC3)c([nH]2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L22 compound treatment 400.0 -144.0 -0.05 440.0 -268.0 -0.21 -0.1813 -0.8566 3030013 ChemDiv3_009064 FC(F)(F)c1ccc(CSc2nc3n(ncc3c(=O)[nH]2)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L23 mock treatment 680.0 136.0 0.05 5520.0 4810.0 3.69 2.6466 0.7163 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 L24 mock treatment 600.0 56.3 0.02 480.0 -228.0 -0.17 -0.1094 -0.6223 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M01 compound treatment 760.0 216.0 0.08 1880.0 1170.0 0.9 0.6907 0.7646 3122585 ChemDiv3_009065 C(Cc1ccccc1)Nc2nc3ccccc3n4cnnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M02 compound treatment 560.0 16.3 0.01 760.0 52.4 0.04 0.0325 0.8002 3122586 ChemDiv3_009066 O=C(NCCc1ccccc1)c2cccc(Nc3nc4ccccc4n5nnnc35)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M03 compound treatment 480.0 -63.8 -0.02 400.0 -308.0 -0.24 -0.183 -0.7713 3030014 ChemDiv3_009067 CC(C)c1cc([nH]n1)C(=O)Nc2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M04 compound treatment 440.0 -104.0 -0.04 1880.0 1170.0 0.9 0.6104 0.6776 3030015 ChemDiv3_009068 CN1c2ccccc2Oc3nnc(cc13)N4CCN(CC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M05 compound treatment 440.0 -104.0 -0.04 840.0 132.0 0.1 0.0459 0.4242 3122769 ChemDiv3_009069 COc1ccc(Cc2nnc(o2)c3ccc(C)cc3)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M06 compound treatment 2000.0 1460.0 0.52 520.0 -188.0 -0.14 0.2635 0.4913 3122770 ChemDiv3_009070 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M07 compound treatment 800.0 256.0 0.09 560.0 -148.0 -0.11 -0.0158 -0.109 3030016 ChemDiv3_009071 O=C(CCc1nc2ccccc2[nH]1)N3CCN(CC3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M08 compound treatment 520.0 -23.8 -0.01 760.0 52.4 0.04 0.0225 0.5472 3122771 ChemDiv3_009072 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCCN4CCN(CC4)c5ccccc5F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M09 compound treatment 640.0 96.3 0.03 480.0 -228.0 -0.17 -0.0994 -0.5584 3122772 ChemDiv3_009073 Cc1cccc(C)c1NC(=O)C2NC(=O)CC2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M10 compound treatment 440.0 -104.0 -0.04 720.0 12.4 0.01 -0.0193 -0.5073 3030017 ChemDiv3_009074 CC1=Nc2cc(ccc2Sc3ccccc13)C(=O)NCc4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M11 compound treatment 920.0 376.0 0.13 840.0 132.0 0.1 0.1663 0.991 3122773 ChemDiv3_009075 COc1ccccc1CNC(=O)c2nnc(Cc3ccc(F)cc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M12 compound treatment 440.0 -104.0 -0.04 320.0 -388.0 -0.3 -0.2364 -0.7886 3030018 ChemDiv3_009076 CCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)N4CCC5(CC4)OCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M13 compound treatment 520.0 -23.8 -0.01 440.0 -268.0 -0.21 -0.1512 -0.7355 3122774 ChemDiv3_009077 Cc1cc(C)n(n1)c2nc3cc(Cl)c(Cl)cc3n4c(C)nnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M14 compound treatment 600.0 56.3 0.02 480.0 -228.0 -0.17 -0.1094 -0.6223 3122775 ChemDiv3_009078 CCC(C)NC(=O)CN1CCN(Cc2ccc(Cl)cc2)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M15 compound treatment 680.0 136.0 0.05 600.0 -108.0 -0.08 -0.0242 -0.2532 3030019 ChemDiv3_009079 COc1cc(Nc2cnn(c3nc4ccccc4s3)c(=O)c2Cl)cc(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M16 compound treatment 880.0 336.0 0.12 840.0 132.0 0.1 0.1562 0.9968 3122776 ChemDiv3_009080 CCC(C)NC(=O)/C=C/1\Sc2ccccc2NC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M17 compound treatment 480.0 -63.8 -0.02 600.0 -108.0 -0.08 -0.0744 -0.8687 3030020 ChemDiv3_009081 CCCOC(=O)c1ccc(Nc2nc3ccccc3n4c(C)nnc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M18 compound treatment 440.0 -104.0 -0.04 840.0 132.0 0.1 0.0459 0.4242 3122777 ChemDiv3_009082 Fc1ccccc1CN2C(=O)/C(=C/c3ccc(cc3)C(=O)NCc4ccco4)/Oc5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M19 compound treatment 440.0 -104.0 -0.04 1720.0 1010.0 0.78 0.5236 0.6729 3122778 ChemDiv3_009083 Cc1nnn(n1)C2(CC3CC4CC(C3)(C2)C(=O)NCc5ccccc5)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M20 compound treatment 640.0 96.3 0.03 1400.0 692.0 0.53 0.4 0.751 3030021 ChemDiv3_009084 CN1C(=O)/C(=C\c2ccccc2)/Sc3ccc(cc13)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M21 compound treatment 600.0 56.3 0.02 480.0 -228.0 -0.17 -0.1094 -0.6223 3122779 ChemDiv3_009085 Cc1cc(C)n(n1)c2nc3ccccc3nc2N4CCN(CC4)S(=O)(=O)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M22 compound treatment 480.0 -63.8 -0.02 400.0 -308.0 -0.24 -0.183 -0.7713 3030022 ChemDiv3_009086 CC(C)CCNC(=O)c1ccc2S/C(=C\c3cccc(C)c3)/C(=O)N(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M23 mock treatment 920.0 376.0 0.13 960.0 252.0 0.19 0.2314 0.9834 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 M24 mock treatment 840.0 296.0 0.11 1000.0 292.0 0.22 0.2331 0.9402 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N01 compound treatment 640.0 96.3 0.03 800.0 92.4 0.07 0.0743 0.9438 3122780 ChemDiv3_009087 Fc1ccccc1/C=C/2\Sc3ccccc3N(CC(=O)NCc4ccc5OCOc5c4)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N02 compound treatment 560.0 16.3 0.01 440.0 -268.0 -0.21 -0.1412 -0.687 3030023 ChemDiv3_009088 COC(=O)c1nnn(CC(=O)Nc2ccccc2)c1C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N03 compound treatment 320.0 -224.0 -0.08 480.0 -228.0 -0.17 -0.1797 -0.9363 3122781 ChemDiv3_009089 CC(C)CC1C(=C(C)Nc2nc(SCc3cccc(C)c3)nn12)C(=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N04 compound treatment 760.0 216.0 0.08 640.0 -67.6 -0.05 0.0176 0.1896 3122782 ChemDiv3_009090 CC1CC(C)CN(C1)C(=S)Nc2ccc3nc(cc(C)c3c2)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N05 compound treatment 480.0 -63.8 -0.02 360.0 -348.0 -0.27 -0.2047 -0.7643 3030024 ChemDiv3_009091 Cn1cc(CC(=O)NCCCN2CCOCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N06 compound treatment 400.0 -144.0 -0.05 520.0 -188.0 -0.14 -0.1379 -0.9026 1175426 ChemDiv3_009092 CCC(C(=O)OCn1nnc2ccccc2c1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N07 compound treatment 800.0 256.0 0.09 1640.0 932.0 0.72 0.5704 0.7906 3030025 ChemDiv3_009093 CC(=O)SCC(=O)/N=c/1\sc2ccccc2n1CC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N08 compound treatment 480.0 -63.8 -0.02 520.0 -188.0 -0.14 -0.1178 -0.8082 3122783 ChemDiv3_009094 c1ccc(cc1)c2nn(c3ccccc3)c4c2cnc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N09 compound treatment 680.0 136.0 0.05 680.0 -27.6 -0.02 0.0192 0.3639 3030026 ChemDiv3_009095 COC(=O)c1c(C)c(C)sc1NC(=O)/C=C/c2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N10 compound treatment 520.0 -23.8 -0.01 920.0 212.0 0.16 0.1094 0.6697 3122784 ChemDiv3_009096 Cc1ccc(Cn2cccc2C3=NC(Cc4ccccc4)CO3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N11 compound treatment 320.0 -224.0 -0.08 640.0 -67.6 -0.05 -0.0928 -0.9788 3030027 ChemDiv3_009097 Cc1noc(C)c1S(=O)(=O)Nc2cccc(C)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N12 compound treatment 640.0 96.3 0.03 520.0 -188.0 -0.14 -0.0777 -0.5249 3122785 ChemDiv3_009098 Cc1oc(nc1Cn2cccc2C3=NC(CO3)c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N13 compound treatment 600.0 56.3 0.02 280.0 -428.0 -0.33 -0.218 -0.6629 3030028 ChemDiv3_009099 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)NC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N14 compound treatment 480.0 -63.8 -0.02 480.0 -228.0 -0.17 -0.1395 -0.792 3122786 ChemDiv3_009100 CC1Cc2cc(ccc2N1C(=O)C)S(=O)(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N15 compound treatment 600.0 56.3 0.02 1640.0 932.0 0.72 0.5203 0.7265 3030081 ChemDiv3_009101 CC(C)C(=O)N1N=C(CC1c2ccccc2)c3ccc(NS(=O)(=O)C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N16 compound treatment 600.0 56.3 0.02 360.0 -348.0 -0.27 -0.1746 -0.6524 3030082 ChemDiv3_009102 CCOc1ccc(CCNS(=O)(=O)c2ccc3N(CCc3c2)C(=O)C4CC4)cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N17 compound treatment 480.0 -63.8 -0.02 640.0 -67.6 -0.05 -0.0527 -0.9307 3030083 ChemDiv3_009103 O=C(CSc1nnc(CNC(=O)c2cccs2)o1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N18 compound treatment 680.0 136.0 0.05 640.0 -67.6 -0.05 -0.0025 -0.0354 3030084 ChemDiv3_009104 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)CCC(=O)NCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N19 compound treatment 1080.0 536.0 0.19 480.0 -228.0 -0.17 0.011 0.0425 3030085 ChemDiv3_009105 Cn1c2ccccc2c3c(cn(C4CCCC4)c(=O)c13)C(=O)N5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N20 compound treatment 1280.0 736.0 0.26 400.0 -308.0 -0.24 0.0177 0.0503 3030086 ChemDiv3_009106 CCc1ccc(NC(=O)c2cc3cc4ccc(C)cc4nc3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N21 compound treatment 520.0 -23.8 -0.01 600.0 -108.0 -0.08 -0.0644 -0.7752 3122787 ChemDiv3_009107 COc1ccc(cc1)c2nc(SCC(=O)NC3CCCC3)c([nH]2)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N22 compound treatment 480.0 -63.8 -0.02 480.0 -228.0 -0.17 -0.1395 -0.792 3030087 ChemDiv3_009108 Clc1ccc(cc1)n2ncc3c(=O)[nH]c(SCC=C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N23 mock treatment 400.0 -144.0 -0.05 440.0 -268.0 -0.21 -0.1813 -0.8566 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 N24 mock treatment 680.0 136.0 0.05 560.0 -148.0 -0.11 -0.0459 -0.3729 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O01 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 1333689 ChemDiv3_009109 N(c1ccccc1)c2nc3ccccc3n4cnnc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O02 compound treatment 240.0 -304.0 -0.11 280.0 -428.0 -0.33 -0.3083 -0.8924 3030088 ChemDiv3_009110 O=c1oc2ccccc2c(NCc3ccc4OCOc4c3)c1CN5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O03 compound treatment 280.0 -264.0 -0.09 360.0 -348.0 -0.27 -0.2549 -0.9012 3122788 ChemDiv3_009111 Cc1cc(C)n(n1)c2nc3ccccc3nc2Nc4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O04 compound treatment 680.0 136.0 0.05 280.0 -428.0 -0.33 -0.1979 -0.5966 3122789 ChemDiv3_009112 CCOC(=O)N1CCN(Cc2nnc(o2)c3ccc4OCOc4c3)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O05 compound treatment 480.0 -63.8 -0.02 320.0 -388.0 -0.3 -0.2264 -0.7587 3030089 ChemDiv3_009113 CCOC(=O)C1CCN(CC1)C(=O)CCc2nc3ccccc3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O06 compound treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 3122790 ChemDiv3_009114 COc1ccc2cc3cc(sc3nc2c1)C(=O)NCC4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O07 compound treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 3030090 ChemDiv3_009115 CCc1nc2nc(C)cc(O)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O08 compound treatment 800.0 256.0 0.09 280.0 -428.0 -0.33 -0.1678 -0.4927 3122791 ChemDiv3_009116 COc1ccc2nc3sc(cc3cc2c1)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O09 compound treatment 280.0 -264.0 -0.09 200.0 -508.0 -0.39 -0.3417 -0.8527 3030091 ChemDiv3_009117 Cc1c(Cl)cccc1NC(=O)C2NC(=O)CC2c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O10 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122792 ChemDiv3_009118 CC(NC(=O)c1ccc2Sc3ccccc3C(=Nc2c1)C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O11 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 3030092 ChemDiv3_009119 CNC(=O)Cc1nnc(o1)c2ccc(C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O12 compound treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 3122793 ChemDiv3_009120 CCCC1=Nc2cc(ccc2Sc3ccccc13)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O13 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122794 ChemDiv3_009121 O=C(NCc1ccc2OCOc2c1)c3nnc(o3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O14 compound treatment 320.0 -224.0 -0.08 320.0 -388.0 -0.3 -0.2665 -0.8655 3030093 ChemDiv3_009122 Clc1ccc(CN2CCN(CC(=O)NCC3COc4ccccc4O3)C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O15 compound treatment 200.0 -344.0 -0.12 200.0 -508.0 -0.39 -0.3618 -0.886 3122970 ChemDiv3_009123 O=S(=O)(Cc1nnn[nH]1)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O16 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122971 ChemDiv3_009124 O=C(NCc1ccco1)/C=C/2\Sc3ccccc3NC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O17 compound treatment 360.0 -184.0 -0.07 320.0 -388.0 -0.3 -0.2565 -0.842 3030094 ChemDiv3_009125 CCCNc1nc2ccccc2n3c(C)nnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O18 compound treatment 440.0 -104.0 -0.04 240.0 -468.0 -0.36 -0.2799 -0.7755 3122972 ChemDiv3_009126 COC(CNC(=O)c1ccc(/C=C/2\Oc3ccccc3N(Cc4cccc(F)c4)C2=O)cc1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O19 compound treatment 400.0 -144.0 -0.05 200.0 -508.0 -0.39 -0.3116 -0.7929 3030095 ChemDiv3_009127 Cc1nnn(n1)C2(CC3CC4CC(C3)(C2)C(=O)Nc5cccc(C)c5)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O20 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 3122973 ChemDiv3_009128 CN1C(=O)/C(=C\c2ccccc2)/Sc3ccc(cc13)C(=O)NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O21 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3030096 ChemDiv3_009129 C(Sc1nc2ccccc2n3cnnc13)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O22 compound treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 3122974 ChemDiv3_009130 COc1ccc(/C=C/2\Sc3ccc(cc3N(C)C2=O)C(=O)N4CCOCC4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O23 mock treatment 280.0 -264.0 -0.09 280.0 -428.0 -0.33 -0.2983 -0.8738 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 O24 mock treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P01 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122975 ChemDiv3_009131 CCOC(=O)N1CCN(CC1)C(=O)CN2C(=O)/C(=C\c3ccc(C)cc3)/Sc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P02 compound treatment 720.0 176.0 0.06 320.0 -388.0 -0.3 -0.1662 -0.5466 3030097 ChemDiv3_009132 CCC(C(=O)Nc1cc(C)ccc1C)n2nnc(C(=O)O)c2C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P03 compound treatment 200.0 -344.0 -0.12 360.0 -348.0 -0.27 -0.2749 -0.937 3122976 ChemDiv3_009133 Cc1ccccc1C(=O)Nc2cc(C)c3c(=O)oc4ccccc4c3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P04 compound treatment 2600.0 2060.0 0.73 320.0 -388.0 -0.3 0.3054 0.3877 3030098 ChemDiv3_009134 CC(C)CCNC(=S)Nc1ccc2nc(cc(C)c2c1)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P05 compound treatment 440.0 -104.0 -0.04 280.0 -428.0 -0.33 -0.2581 -0.7815 3122977 ChemDiv3_009135 CCc1ccc(NC(=O)Cc2cn(C)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P06 compound treatment 2280.0 1740.0 0.62 360.0 -348.0 -0.27 0.2468 0.3677 3122978 ChemDiv3_009136 COc1cc(/C=C\C(=O)OCn2nnc3ccccc3c2=O)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P07 compound treatment 320.0 -224.0 -0.08 520.0 -188.0 -0.14 -0.158 -0.9606 3030099 ChemDiv3_009137 CCn1/c(=N/C(=O)CSCC(=O)NC2CCCCC2)/sc3cc(ccc13)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P08 compound treatment 320.0 -224.0 -0.08 360.0 -348.0 -0.27 -0.2448 -0.8794 3122979 ChemDiv3_009138 CCOC(=O)c1ccc2ncc3c(nn(c4ccccc4)c3c2c1)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P09 compound treatment 280.0 -264.0 -0.09 240.0 -468.0 -0.36 -0.32 -0.8626 3030100 ChemDiv3_009139 Cc1n[nH]c(C)c1S(=O)(=O)N2CCC3(CC2)OCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P10 compound treatment 400.0 -144.0 -0.05 280.0 -428.0 -0.33 -0.2682 -0.8073 3122980 ChemDiv3_009140 CSc1ccc(Cn2cccc2C3=NC(CO3)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P11 compound treatment 280.0 -264.0 -0.09 400.0 -308.0 -0.24 -0.2331 -0.9179 3030101 ChemDiv3_009141 COc1ccc(N(C)S(=O)(=O)c2c(C)noc2C)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P12 compound treatment 280.0 -264.0 -0.09 320.0 -388.0 -0.3 -0.2766 -0.8867 3122981 ChemDiv3_009142 CCc1ccc(/C=C/C2=CC(C)(C)NC(=S)N2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P13 compound treatment 280.0 -264.0 -0.09 360.0 -348.0 -0.27 -0.2549 -0.9012 3030102 ChemDiv3_009143 COc1ccc(cc1)c2nc3ncccn3c2Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P14 compound treatment 440.0 -104.0 -0.04 320.0 -388.0 -0.3 -0.2364 -0.7886 3122982 ChemDiv3_009144 CCC(=O)N1C(C)Cc2cc(ccc12)S(=O)(=O)NC3CCCCC3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P15 compound treatment 320.0 -224.0 -0.08 280.0 -428.0 -0.33 -0.2882 -0.8535 3122983 ChemDiv3_009145 CS(=O)(=O)Nc1cccc(c1)C2=NN(C(C2)c3ccccc3F)C(=O)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P16 compound treatment 240.0 -304.0 -0.11 240.0 -468.0 -0.36 -0.33 -0.8805 3030103 ChemDiv3_009146 O=C(C1CC1)N2CCc3cc(ccc23)S(=O)(=O)NCCCN4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P17 compound treatment 360.0 -184.0 -0.07 280.0 -428.0 -0.33 -0.2782 -0.8313 3122984 ChemDiv3_009147 O=C(CSc1nnc(CNC(=O)c2cccs2)o1)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P18 compound treatment 2560.0 2020.0 0.72 400.0 -308.0 -0.24 0.3388 0.4498 3030104 ChemDiv3_009148 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)CCC(=O)N(C)c3ccc(Br)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P19 compound treatment 320.0 -224.0 -0.08 400.0 -308.0 -0.24 -0.2231 -0.8956 3122985 ChemDiv3_009149 COc1ccc(cc1)N(C)C(=O)c2cn(C3CCCC3)c(=O)c4n(C)c5ccccc5c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P20 compound treatment 200.0 -344.0 -0.12 720.0 12.4 0.01 -0.0795 -0.6499 3122986 ChemDiv3_009150 Cc1ccc2cc3cc(oc3nc2c1)C(=O)NCCCN4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P21 compound treatment 1040.0 496.0 0.18 1480.0 772.0 0.59 0.5438 0.8791 3030105 ChemDiv3_009151 O=C(CSc1nc([nH]c1c2ccccc2)c3ccccc3)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P22 compound treatment 320.0 -224.0 -0.08 3600.0 2890.0 2.22 1.514 0.6814 3122987 ChemDiv3_009152 CCOC(=O)C(C)(C)Sc1nc2n(ncc2c(=O)[nH]1)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P23 mock treatment 240.0 -304.0 -0.11 2160.0 1450.0 1.12 0.7123 0.6358 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2026 P24 mock treatment 520.0 -23.8 -0.01 200.0 -508.0 -0.39 -0.2815 -0.7222 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A01 compound treatment 4920.0 4150.0 1.47 3640.0 2790.0 2.14 2.5552 0.9833 3030106 ChemDiv3_009153 Cc1ccc(cc1)n2ncc3c(=O)[nH]c(SCc4ccccc4)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A02 compound treatment 2560.0 1790.0 0.64 720.0 -131.0 -0.1 0.3781 0.5876 3122988 ChemDiv3_009154 COc1ccc(Nc2cc(C(=O)NC3CCCCC3)c4ccccc4n2)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A03 compound treatment 3000.0 2230.0 0.79 400.0 -451.0 -0.35 0.3147 0.3643 3122989 ChemDiv3_009155 CCS(=O)(=O)Nc1ccc(cc1)C2=NN(C(C2)c3ccccc3)S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A04 compound treatment 1400.0 631.0 0.22 400.0 -451.0 -0.35 -0.0866 -0.21 3030107 ChemDiv3_009156 Cc1ccccc1Nc2cc(C(=O)NCc3ccccc3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A05 compound treatment 240.0 -529.0 -0.19 480.0 -371.0 -0.29 -0.3342 -0.9794 3122990 ChemDiv3_009157 Cc1ccc(CCNC(=O)c2cccn3c(=O)c4c5CCCCc5sc4nc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A06 compound treatment 560.0 -209.0 -0.07 720.0 -131.0 -0.1 -0.1236 -0.9885 3030108 ChemDiv3_009158 CCc1ccc(NC(=O)N(Cc2c[nH]c3ccccc23)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A07 compound treatment 360.0 -409.0 -0.15 320.0 -531.0 -0.41 -0.3909 -0.9031 3122991 ChemDiv3_009159 COc1ccc2nc3oc(cc3cc2c1)C(=O)N4CCN(CC4)c5cccc(c5)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A08 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3030109 ChemDiv3_009160 CCC(C)N(Cc1cn(CC)c2ccccc12)C(=O)Nc3ccc(Cl)c(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A09 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3122992 ChemDiv3_009161 COc1ccc2cc3cc(oc3nc2c1)C(=O)NCCN(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A10 compound treatment 280.0 -489.0 -0.17 200.0 -651.0 -0.5 -0.4761 -0.8998 3122993 ChemDiv3_009162 O=C(NC1CCCCCC1)c2cccc(c2)N3CCCC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A11 compound treatment 1040.0 271.0 0.1 280.0 -571.0 -0.44 -0.2421 -0.5391 3030110 ChemDiv3_009163 CCc1cccc(NC(=O)c2cc3cc4ccc(OC)cc4nc3o2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A12 compound treatment 360.0 -409.0 -0.15 320.0 -531.0 -0.41 -0.3909 -0.9031 3122994 ChemDiv3_009164 CCOC(=O)N1CCC(CC1)N2CC3(OC4C=C3)C(C4C(=O)Nc5ccc(OCC)cc5)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A13 compound treatment 280.0 -489.0 -0.17 2440.0 1590.0 1.22 0.7399 0.6006 3030111 ChemDiv3_009165 CC(C)c1ccc(cc1)n2cccc2/C=C\3/C(=N)N4C=CSC4=NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A14 compound treatment 280.0 -489.0 -0.17 280.0 -571.0 -0.44 -0.4327 -0.9176 3122995 ChemDiv3_009166 CCOC(=O)N1CCC(CC1)c2cc(O)n3nc(cc3n2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A15 compound treatment 720.0 -48.8 -0.02 640.0 -211.0 -0.16 -0.1269 -0.7781 3122996 ChemDiv3_009167 CCCNC(=O)c1oc(=O)c2ccccc2c1c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A16 compound treatment 680.0 -88.8 -0.03 960.0 109.0 0.08 0.0368 0.4121 3030112 ChemDiv3_009168 Clc1ccccc1CN2C(Nc3ccc(cc3)S(=O)(=O)N4CCOCC4)c5ccccc5C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A17 compound treatment 480.0 -289.0 -0.1 360.0 -491.0 -0.38 -0.3391 -0.8677 3123175 ChemDiv3_009169 COc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)N3CC(C)CC(C)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A18 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3123176 ChemDiv3_009170 COC(=O)c1cc(NC2N(C(=O)c3ccccc23)c4ccccn4)cc(c1)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A19 compound treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 3030113 ChemDiv3_009171 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)NCCN3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A20 compound treatment 200.0 -569.0 -0.2 280.0 -571.0 -0.44 -0.4528 -0.9379 3123177 ChemDiv3_009172 CCOC(=O)CCc1c(C)nc2n(nc(C)c2c1C)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A21 compound treatment 200.0 -569.0 -0.2 280.0 -571.0 -0.44 -0.4528 -0.9379 3123178 ChemDiv3_009173 Fc1ccccc1NS(=O)(=O)c2ccc3[nH]cc(C(=O)N4CCOCC4)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A22 compound treatment 320.0 -449.0 -0.16 760.0 -91.3 -0.07 -0.1621 -0.932 3030114 ChemDiv3_009174 COc1ccc(c2nn(CCC(=O)O)c3nc(C)cc(C)c23)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A23 mock treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 A24 mock treatment 560.0 -209.0 -0.07 280.0 -571.0 -0.44 -0.3625 -0.815 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B01 compound treatment 360.0 -409.0 -0.15 360.0 -491.0 -0.38 -0.3692 -0.9138 3030115 ChemDiv3_009175 CC(C)C1N2C(OC1=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B02 compound treatment 280.0 -489.0 -0.17 440.0 -411.0 -0.32 -0.3459 -0.9602 3030173 ChemDiv3_009176 O=C(NCc1cccs1)c2cc3c(=O)[nH]c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B03 compound treatment 400.0 -369.0 -0.13 600.0 -251.0 -0.19 -0.2289 -0.9821 3030174 ChemDiv3_009177 COc1cc2[nH]c(=S)nc(NC3CCCCCC3)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B04 compound treatment 600.0 -169.0 -0.06 400.0 -451.0 -0.35 -0.2873 -0.8172 3030175 ChemDiv3_009178 COc1ccc(cc1)n2nc(C(=O)NCc3cc(OC)ccc3OC)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B05 compound treatment 320.0 -449.0 -0.16 3240.0 2390.0 1.83 1.1842 0.6433 3030176 ChemDiv3_009179 O=C(Cn1ncc2c(=O)oc3ccccc3c12)NCC4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B06 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3030177 ChemDiv3_009180 CCNC(=S)N(CCc1c(C)[nH]c2ccccc12)Cc3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B07 compound treatment 320.0 -449.0 -0.16 520.0 -331.0 -0.25 -0.2924 -0.9746 3030178 ChemDiv3_009181 O=C(NCc1cccs1)C2CCCN(C2)S(=O)(=O)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B08 compound treatment 280.0 -489.0 -0.17 200.0 -651.0 -0.5 -0.4761 -0.8998 3123179 ChemDiv3_009182 COc1ccc(cc1OC)c2nn(C)c3sc(cc23)C(=O)N(CC=C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B09 compound treatment 640.0 -129.0 -0.05 320.0 -531.0 -0.41 -0.3207 -0.7814 3123180 ChemDiv3_009183 CC1CN(CCN1c2ccc(C)cc2)C(=O)CN(c3ccc(C)cc3)S(=O)(=O)c4c(C)n[nH]c4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B10 compound treatment 360.0 -409.0 -0.15 360.0 -491.0 -0.38 -0.3692 -0.9138 3030179 ChemDiv3_009184 COc1ccc(CNC(=O)C2CCN(CC2)S(=O)(=O)c3c[nH]cn3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B11 compound treatment 480.0 -289.0 -0.1 320.0 -531.0 -0.41 -0.3608 -0.8581 3123181 ChemDiv3_009185 CC(=O)N1CCN=C1SCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B12 compound treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 3030180 ChemDiv3_009186 CN(Cc1ccccc1)C(=O)c2cnc3sccn3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B13 compound treatment 360.0 -409.0 -0.15 280.0 -571.0 -0.44 -0.4126 -0.8933 3123182 ChemDiv3_009187 Fc1ccccc1CSC2=NCCN2C(=O)C3c4ccccc4Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B14 compound treatment 360.0 -409.0 -0.15 560.0 -291.0 -0.22 -0.2606 -0.978 3030181 ChemDiv3_009188 Cn1c(=O)cc(SCC(=O)NC2CCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B15 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3123183 ChemDiv3_009189 CCCNS(=O)(=O)c1ccc2N(CCCc2c1)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B16 compound treatment 440.0 -329.0 -0.12 320.0 -531.0 -0.41 -0.3709 -0.8743 3123184 ChemDiv3_009190 CC(CCc1ccccc1)NC(=O)CSc2cc(=O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B17 compound treatment 1280.0 511.0 0.18 1480.0 629.0 0.48 0.4696 0.9106 3030182 ChemDiv3_009191 CSc1cccc(c1)N2C(=S)NC3C4CCCC42Oc5ccccc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B18 compound treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 3123185 ChemDiv3_009192 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)NC(CC(C)C)C(=O)Nc3cc(C)ccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B19 compound treatment 920.0 151.0 0.05 440.0 -411.0 -0.32 -0.1853 -0.5786 3123186 ChemDiv3_009193 CCCN1Cc2cccc(C(=O)N3CCN(CC3)c4ccccc4)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B20 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3030183 ChemDiv3_009194 CN(C)C(CNC(=O)Nc1cccc(Cl)c1)c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B21 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3123187 ChemDiv3_009195 O=C(N1CCN(CC1)C(=O)c2cccc3CN(C4CCCCC4)C(=O)c32)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B22 compound treatment 520.0 -249.0 -0.09 320.0 -531.0 -0.41 -0.3508 -0.8406 3030184 ChemDiv3_009196 Cn1c(=O)n(C)c2nc(CN3CCN(CC3)c4ccccc4)n(Cc5c(F)cccc5Cl)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B23 mock treatment 200.0 -569.0 -0.2 400.0 -451.0 -0.35 -0.3876 -0.9669 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 B24 mock treatment 320.0 -449.0 -0.16 1680.0 829.0 0.64 0.3373 0.5143 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C01 compound treatment 1920.0 1150.0 0.41 360.0 -491.0 -0.38 0.0221 0.0398 3123188 ChemDiv3_009197 CCOC(=O)N1CCN(CC1)C(=O)CSc2nc3n(ncc3c(=O)[nH]2)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C02 compound treatment 320.0 -449.0 -0.16 240.0 -611.0 -0.47 -0.4444 -0.8968 3123189 ChemDiv3_009198 CCOC(=O)N1CCN(CC1)C(=O)c2cc(Nc3ccc(OC)cc3OC)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C03 compound treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 3030185 ChemDiv3_009199 CCS(=O)(=O)Nc1cccc(c1)C2=NN(C(C2)c3ccccc3)S(=O)(=O)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C04 compound treatment 280.0 -489.0 -0.17 520.0 -331.0 -0.25 -0.3024 -0.9826 3123190 ChemDiv3_009200 Cc1ccc(Nc2cc(C(=O)NCCCN3CCOCC3)c4ccccc4n2)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C05 compound treatment 320.0 -449.0 -0.16 440.0 -411.0 -0.32 -0.3358 -0.9497 3030186 ChemDiv3_009201 CC1CCN(CC1)C(=O)c2cccn3c(=O)c4c5CCCCc5sc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C06 compound treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 3123191 ChemDiv3_009202 CCc1ccc(NC(=O)N(Cc2c[nH]c3ccccc23)C4CCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C07 compound treatment 200.0 -569.0 -0.2 400.0 -451.0 -0.35 -0.3876 -0.9669 3123192 ChemDiv3_009203 COc1ccc2nc3oc(cc3cc2c1)C(=O)N4CCC(CC4)N5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C08 compound treatment 320.0 -449.0 -0.16 320.0 -531.0 -0.41 -0.401 -0.9158 3030187 ChemDiv3_009204 CCOc1ccc(NC(=S)N(Cc2cn(CC)c3ccccc23)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C09 compound treatment 360.0 -409.0 -0.15 320.0 -531.0 -0.41 -0.3909 -0.9031 3123193 ChemDiv3_009205 CCCCN(C)C(=O)c1cc2cc3ccc(OC)cc3nc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C10 compound treatment 280.0 -489.0 -0.17 280.0 -571.0 -0.44 -0.4327 -0.9176 3030188 ChemDiv3_009206 O=C(NCc1ccco1)c2cccc(c2)N3CCCC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C11 compound treatment 320.0 -449.0 -0.16 320.0 -531.0 -0.41 -0.401 -0.9158 3123194 ChemDiv3_009207 COc1ccc2cc3cc(oc3nc2c1)C(=O)NCCN4CCN(CC4)c5ccccc5F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C12 compound treatment 2960.0 2190.0 0.78 400.0 -451.0 -0.35 0.3047 0.358 3123195 ChemDiv3_009208 O=C(NC1CCCCCC1)C2C3OC4(CN(Cc5cccnc5)C(=O)C24)C=C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C13 compound treatment 4360.0 3590.0 1.27 320.0 -531.0 -0.41 0.6124 0.4578 3030189 ChemDiv3_009209 CCc1cccc(c1)n2c(nc3n(ncc3c2=O)c4ccccc4Cl)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C14 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3123196 ChemDiv3_009210 CCOC(=O)N1CCC(CC1)N2C(O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C15 compound treatment 280.0 -489.0 -0.17 240.0 -611.0 -0.47 -0.4544 -0.9083 3030190 ChemDiv3_009211 CC(C)CN(CC(C)C)C(=O)c1oc(=O)c2ccccc2c1c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C16 compound treatment 280.0 -489.0 -0.17 440.0 -411.0 -0.32 -0.3459 -0.9602 3123197 ChemDiv3_009212 CCOC(=O)N1CCC(CC1)/N=C/c2ccc(OC(C)C)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C17 compound treatment 240.0 -529.0 -0.19 320.0 -531.0 -0.41 -0.421 -0.9379 3123198 ChemDiv3_009213 CC1CCC(CC1)NC(=O)c2ccc(CNS(=O)(=O)c3ccc(C)cc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C18 compound treatment 280.0 -489.0 -0.17 440.0 -411.0 -0.32 -0.3459 -0.9602 3030191 ChemDiv3_009214 O=C1N(C(Nc2ccc3OCCOc3c2)c4ccccc14)c5ccccn5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C19 compound treatment 360.0 -409.0 -0.15 280.0 -571.0 -0.44 -0.4126 -0.8933 3123199 ChemDiv3_009215 CCOC(=O)N1CCN(CC1)C(=O)c2ccc(CNS(=O)(=O)c3ccc(NC(=O)C)cc3)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C20 compound treatment 440.0 -329.0 -0.12 280.0 -571.0 -0.44 -0.3926 -0.8651 3030192 ChemDiv3_009216 Cc1ccccc1N2C(CNc3ccccc3)C(Oc4ccc(Cl)cc4)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C21 compound treatment 320.0 -449.0 -0.16 240.0 -611.0 -0.47 -0.4444 -0.8968 3123200 ChemDiv3_009217 CN(Cc1ccco1)C(=O)c2c[nH]c3ccc(cc3c2=O)S(=O)(=O)Nc4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C22 compound treatment 320.0 -449.0 -0.16 320.0 -531.0 -0.41 -0.401 -0.9158 3030193 ChemDiv3_009218 CC(=O)Nc1cc(C)nn1C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C23 mock treatment 400.0 -369.0 -0.13 320.0 -531.0 -0.41 -0.3809 -0.8893 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 C24 mock treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D01 compound treatment 880.0 111.0 0.04 320.0 -531.0 -0.41 -0.2605 -0.6357 3030194 ChemDiv3_009219 CNc1ncc(Br)nc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D02 compound treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 3123201 ChemDiv3_009220 Clc1ccc(CCNC(=O)c2cc3c(=O)[nH]c4ccccc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D03 compound treatment 240.0 -529.0 -0.19 400.0 -451.0 -0.35 -0.3776 -0.9585 3123379 ChemDiv3_009221 COc1ccc(Nc2nc(=S)[nH]c3cc(OC)c(OC)cc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D04 compound treatment 360.0 -409.0 -0.15 480.0 -371.0 -0.29 -0.3041 -0.9509 3030195 ChemDiv3_009222 Cc1ccc(cc1)n2nc(C(=O)N3CCCC3)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D05 compound treatment 480.0 -289.0 -0.1 320.0 -531.0 -0.41 -0.3608 -0.8581 3123380 ChemDiv3_009223 CCc1ccc(NC(=O)Cn2ncc3c(=O)oc4ccccc4c23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D06 compound treatment 280.0 -489.0 -0.17 280.0 -571.0 -0.44 -0.4327 -0.9176 3123381 ChemDiv3_009224 Cc1[nH]c2ccc(C)cc2c1CCN(Cc3ccco3)C(=S)Nc4cccc(C)c4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D07 compound treatment 200.0 -569.0 -0.2 320.0 -531.0 -0.41 -0.4311 -0.9473 3030196 ChemDiv3_009225 Cc1n[nH]c(C)c1S(=O)(=O)N2CCCC(C2)C(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D08 compound treatment 440.0 -329.0 -0.12 240.0 -611.0 -0.47 -0.4143 -0.8568 3123382 ChemDiv3_009226 COc1ccc(cc1OC)c2nn(C)c3sc(cc23)C(=O)NCC4(CCCC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D09 compound treatment 3320.0 2550.0 0.91 400.0 -451.0 -0.35 0.395 0.4076 3030197 ChemDiv3_009227 Cc1nn(C)c(C)c1S(=O)(=O)N2CCN(CC2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D10 compound treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 3123383 ChemDiv3_009228 CCOc1ccc(NC(=O)C2CCN(CC2)S(=O)(=O)c3c[nH]cn3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D11 compound treatment 320.0 -449.0 -0.16 240.0 -611.0 -0.47 -0.4444 -0.8968 3030198 ChemDiv3_009229 O=C(C1CC1)N2CCN=C2SCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D12 compound treatment 360.0 -409.0 -0.15 360.0 -491.0 -0.38 -0.3692 -0.9138 3123384 ChemDiv3_009230 CCN(C(=O)c1cnc2sccn2c1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D13 compound treatment 480.0 -289.0 -0.1 520.0 -331.0 -0.25 -0.2523 -0.9201 3030199 ChemDiv3_009231 CC1CCN(CC1)C(c2sc3nc(C)nn3c2O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D14 compound treatment 240.0 -529.0 -0.19 360.0 -491.0 -0.38 -0.3993 -0.948 3123385 ChemDiv3_009232 CN(C1CCCCC1)C(=O)CSc2cc(=O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D15 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3123386 ChemDiv3_009233 CCC(=O)N1CCCc2cc(ccc12)S(=O)(=O)N3CCN(CC3)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D16 compound treatment 480.0 -289.0 -0.1 480.0 -371.0 -0.29 -0.274 -0.9046 3030200 ChemDiv3_009234 Cn1c(=O)cc(SCC(=O)NCCCN2CCN(CC2)c3ccccc3F)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D17 compound treatment 360.0 -409.0 -0.15 240.0 -611.0 -0.47 -0.4344 -0.8843 3123387 ChemDiv3_009235 COCCN1C(=S)NC2C3CCCC31Oc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D18 compound treatment 240.0 -529.0 -0.19 320.0 -531.0 -0.41 -0.421 -0.9379 3123388 ChemDiv3_009236 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)NCCC(=O)Nc3ccc(Br)cc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D19 compound treatment 320.0 -449.0 -0.16 320.0 -531.0 -0.41 -0.401 -0.9158 3030201 ChemDiv3_009237 CCCN1Cc2cccc(C(=O)Nc3ccc(cc3)S(=O)(=O)N4CCCCCC4)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D20 compound treatment 280.0 -489.0 -0.17 280.0 -571.0 -0.44 -0.4327 -0.9176 3123389 ChemDiv3_009238 S=C(NCC(N1CCOCC1)c2cccnc2)Nc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D21 compound treatment 400.0 -369.0 -0.13 320.0 -531.0 -0.41 -0.3809 -0.8893 3123390 ChemDiv3_009239 CC(CCc1ccco1)NC(=O)c2cccc3CN(C4CCCCC4)C(=O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D22 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3030202 ChemDiv3_009240 Cn1c(=O)n(C)c2nc(CN3CCN(CC3)C(=O)c4ccco4)n(Cc5ccccc5F)c2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D23 mock treatment 2200.0 1430.0 0.51 360.0 -491.0 -0.38 0.0923 0.146 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 D24 mock treatment 240.0 -529.0 -0.19 240.0 -611.0 -0.47 -0.4645 -0.919 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E01 compound treatment 440.0 -329.0 -0.12 840.0 -11.3 -0.01 -0.0886 -0.7574 3123391 ChemDiv3_009241 Cc1ccc(cc1)n2ncc3c(=O)[nH]c(SCC(=O)N4CCCc5ccccc45)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E02 compound treatment 720.0 -48.8 -0.02 840.0 -11.3 -0.01 -0.0183 -0.9485 3030203 ChemDiv3_009242 COc1ccc(Nc2cc(C(=O)N3CCc4ccccc4C3)c5ccccc5n2)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E03 compound treatment 1720.0 951.0 0.34 2520.0 1670.0 1.28 1.1445 0.8639 3123392 ChemDiv3_009243 OC(=O)c1cccn2c(=O)c3c4CCCCc4sc3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E04 compound treatment 920.0 151.0 0.05 400.0 -451.0 -0.35 -0.207 -0.5905 3123393 ChemDiv3_009244 Cc1ccc(Nc2cc(C(=O)NCCC3=CCCCC3)c4ccccc4n2)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E05 compound treatment 680.0 -88.8 -0.03 640.0 -211.0 -0.16 -0.1369 -0.8289 3030204 ChemDiv3_009245 CC1CCCCN1CCNC(=O)c2cccn3c(=O)c4c5CCCCc5sc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E06 compound treatment 720.0 -48.8 -0.02 720.0 -131.0 -0.1 -0.0835 -0.8165 3123394 ChemDiv3_009246 CCOc1ccccc1NC(=S)N(Cc2c[nH]c3ccccc23)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E07 compound treatment 320.0 -449.0 -0.16 800.0 -51.3 -0.04 -0.1404 -0.8561 3123395 ChemDiv3_009247 CCOC(=O)N1CCC(CC1)NC(=O)c2cc3cc4cc(OC)ccc4nc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E08 compound treatment 3240.0 2470.0 0.88 360.0 -491.0 -0.38 0.3532 0.3701 3030205 ChemDiv3_009248 CCC(C)N(Cc1cn(CC)c2ccccc12)C(=S)Nc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E09 compound treatment 1800.0 1030.0 0.37 600.0 -251.0 -0.19 0.1223 0.2957 3123396 ChemDiv3_009249 COc1ccc2cc3cc(oc3nc2c1)C(=O)N4CCC5(CC4)OCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E10 compound treatment 2280.0 1510.0 0.54 920.0 68.8 0.05 0.4164 0.773 3030206 ChemDiv3_009250 COC(CNC(=O)c1cccc(c1)N2CCCC2=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E11 compound treatment 6680.0 5910.0 2.1 1160.0 309.0 0.24 1.6504 0.7821 3030264 ChemDiv3_009251 Clc1ccc2cc3cc(oc3nc2c1)C(=O)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E12 compound treatment 1200.0 431.0 0.15 520.0 -331.0 -0.25 -0.0716 -0.2414 3030265 ChemDiv3_009252 CCOC(=O)CN1CC2(OC3C=C2)C(C3C(=O)NCc4ccc(OC)cc4)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E13 compound treatment 1880.0 1110.0 0.39 600.0 -251.0 -0.19 0.1424 0.3244 3030266 ChemDiv3_009253 COc1cccc(c1)n2c(C)nc3n(ncc3c2=O)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E14 compound treatment 4560.0 3790.0 1.34 840.0 -11.3 -0.01 0.9449 0.7026 1033635 ChemDiv3_009254 Clc1ccc(cc1)N2C(=O)CCC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E15 compound treatment 4840.0 4070.0 1.44 1200.0 349.0 0.27 1.2106 0.8242 3030267 ChemDiv3_009255 CCCCN(C)C(=O)c1oc(=O)c2ccccc2c1c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E16 compound treatment 2960.0 2190.0 0.78 1360.0 509.0 0.39 0.8258 0.9493 3030268 ChemDiv3_009256 CCOc1ccc(NC(=O)/C=C/C(=O)NCc2ccc(OC)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E17 compound treatment 880.0 111.0 0.04 720.0 -131.0 -0.1 -0.0433 -0.4005 3030269 ChemDiv3_009257 Cc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)NCCN3CCN(CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E18 compound treatment 760.0 -8.75 0.0 1480.0 629.0 0.48 0.3391 0.7025 3123397 ChemDiv3_009258 CCOc1ccc(/N=C/C=N/c2ccc(OCC)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E19 compound treatment 1000.0 231.0 0.08 1160.0 309.0 0.24 0.2256 0.8995 3123398 ChemDiv3_009259 COc1cccc(NS(=O)(=O)c2ccc3[nH]cc(C(=O)N(C)Cc4ccccc4)c(=O)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E20 compound treatment 1880.0 1110.0 0.39 1520.0 669.0 0.51 0.6418 0.9915 1463342 ChemDiv3_009260 Cc1cc(C)c2c(=O)n([nH]c2n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E21 compound treatment 1400.0 631.0 0.22 480.0 -371.0 -0.29 -0.0432 -0.1192 3123399 ChemDiv3_009261 Cc1ccc(CNC(=O)c2c[nH]c3ccc(cc3c2=O)S(=O)(=O)Nc4ccc(C)cc4C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E22 compound treatment 760.0 -8.75 0.0 1000.0 149.0 0.11 0.0786 0.6876 3030270 ChemDiv3_009262 CCOC(=O)Cc1nc(OCC(=O)c2ccc(F)cc2)cs1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E23 mock treatment 920.0 151.0 0.05 1040.0 189.0 0.14 0.1404 0.9086 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 E24 mock treatment 1840.0 1070.0 0.38 2840.0 1990.0 1.53 1.3483 0.857 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F01 compound treatment 7680.0 6910.0 2.45 920.0 68.8 0.05 1.771 0.7222 3123400 ChemDiv3_009263 CCOc1ccc(cc1)N2C(Nc3ccccc3OC)c4ccccc4C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F02 compound treatment 1960.0 1190.0 0.42 1480.0 629.0 0.48 0.6401 0.9978 3030271 ChemDiv3_009264 O=C(NCC1(CCCC1)c2ccccc2)c3cc4c(=O)[nH]c5ccccc5c4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F03 compound treatment 5200.0 4430.0 1.57 2960.0 2110.0 1.62 2.2563 0.9999 3123401 ChemDiv3_009265 CCOc1ccc(NC(=O)c2ccc(cc2)N3C(=O)NC4CC3(C)Oc5ccccc45)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F04 compound treatment 7960.0 7190.0 2.55 920.0 68.8 0.05 1.8412 0.7216 3123402 ChemDiv3_009266 CCc1ccc(NC(=O)c2nn(c3ccc(C)cc3)c(=O)c4n(C)c5ccccc5c24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F05 compound treatment 5880.0 5110.0 1.81 640.0 -211.0 -0.16 1.1674 0.6413 3030272 ChemDiv3_009267 O=C(Cn1ncc2c(=O)oc3ccccc3c12)N4CCN(CC4)C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F06 compound treatment 1320.0 551.0 0.2 1320.0 469.0 0.36 0.3927 0.9589 3123403 ChemDiv3_009268 CC(C)CC(NS(=O)(=O)c1ccc2N(CCc2c1)C(=O)C)C(=O)NCc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F07 compound treatment 1480.0 711.0 0.25 560.0 -291.0 -0.22 0.0203 0.0602 3030273 ChemDiv3_009269 Cc1nn(C)c(C)c1S(=O)(=O)N2CCC(CC2)C(=O)NC3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F08 compound treatment 7240.0 6470.0 2.3 1040.0 189.0 0.14 1.7257 0.7502 3123404 ChemDiv3_009270 FC(F)(F)c1cc(NS(=O)(=O)c2c[nH]cn2)ccc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F09 compound treatment 1200.0 431.0 0.15 1000.0 149.0 0.11 0.1889 0.9896 3030274 ChemDiv3_009271 CCC(=O)N1CCN=C1SC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F10 compound treatment 1960.0 1190.0 0.42 2080.0 1230.0 0.94 0.9659 0.9344 3123405 ChemDiv3_009272 O=C(C1CCN(CC1)S(=O)(=O)c2c[nH]cn2)N(CCc3ccccc3)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F11 compound treatment 1040.0 271.0 0.1 760.0 -91.3 -0.07 0.0185 0.1555 3030275 ChemDiv3_009273 O=C(N1CCN=C1SCc2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F12 compound treatment 1080.0 311.0 0.11 560.0 -291.0 -0.22 -0.08 -0.3209 3120339 ChemDiv3_009274 Cc1cccc(NC(=O)c2cnc3sccn3c2=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F13 compound treatment 1360.0 591.0 0.21 1040.0 189.0 0.14 0.2508 0.9837 3030276 ChemDiv3_009275 CC1CCN(CCNC(=O)C2CCCN(C2)S(=O)(=O)c3cccc4nsnc34)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F14 compound treatment 1080.0 311.0 0.11 440.0 -411.0 -0.32 -0.1452 -0.434 3120340 ChemDiv3_009276 Cn1c(=O)cc(SCC(=O)N2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F15 compound treatment 1280.0 511.0 0.18 1760.0 909.0 0.7 0.6216 0.8623 3120341 ChemDiv3_009277 COc1ccc(CCNC(=O)CSc2nc3cc(OC)c(OC)cc3c4nc(C)nn24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F16 compound treatment 1360.0 591.0 0.21 1400.0 549.0 0.42 0.4462 0.9481 3030277 ChemDiv3_009278 Cn1c(=O)cc(SCC(=O)Nc2cccnc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F17 compound treatment 1240.0 471.0 0.17 600.0 -251.0 -0.19 -0.0182 -0.0712 3120342 ChemDiv3_009279 CCN1C(=S)NC2C3CCCC31Oc4ccc(C)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F18 compound treatment 520.0 -249.0 -0.09 3520.0 2670.0 2.05 1.3864 0.676 3120343 ChemDiv3_009280 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)NCCC(=O)Nc3ccc(OC(F)(F)F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F19 compound treatment 1600.0 831.0 0.29 520.0 -331.0 -0.25 0.0287 0.0737 3030278 ChemDiv3_009281 COCCN1Cc2cccc(C(=O)NC3CCCC3)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F20 compound treatment 1200.0 431.0 0.15 520.0 -331.0 -0.25 -0.0716 -0.2414 3120344 ChemDiv3_009282 S=C(NCCc1ccccc1)NCC(N2CCOCC2)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F21 compound treatment 2360.0 1590.0 0.56 760.0 -91.3 -0.07 0.3496 0.6146 3030279 ChemDiv3_009283 COc1ccc(CNC(=O)c2cccc3CN(C(=O)c32)c4ccc(OC)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F22 compound treatment 1880.0 1110.0 0.39 920.0 68.8 0.05 0.3161 0.7947 3120345 ChemDiv3_009284 CC1CC(C)CN(Cc2nc3n(C)c(=O)n(C)c(=O)c3n2CC(=O)N)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F23 mock treatment 2640.0 1870.0 0.66 2640.0 1790.0 1.37 1.4404 0.9444 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 F24 mock treatment 1240.0 471.0 0.17 1200.0 349.0 0.27 0.3075 0.9743 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G01 compound treatment 1040.0 271.0 0.1 2680.0 1830.0 1.4 1.0608 0.7538 3030280 ChemDiv3_009285 Cc1ccc(cc1)n2ncc3c(=O)[nH]c(SCC(=O)Nc4ccccc4C(F)(F)F)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G02 compound treatment 320.0 -449.0 -0.16 440.0 -411.0 -0.32 -0.3358 -0.9497 3120346 ChemDiv3_009286 CCc1ccccc1Nc2cc(C(=O)NCc3cccnc3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G03 compound treatment 1640.0 871.0 0.31 680.0 -171.0 -0.13 0.1256 0.3739 3120347 ChemDiv3_009287 CN(Cc1ccccc1)C(=O)c2cccn3c(=O)c4c5CCCCc5sc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G04 compound treatment 720.0 -48.8 -0.02 880.0 28.8 0.02 0.0034 0.1205 3030281 ChemDiv3_009288 Cc1cc(C)cc(Nc2cc(C(=O)NC3CCCC3)c4ccccc4n2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G05 compound treatment 1080.0 311.0 0.11 1360.0 509.0 0.39 0.3543 0.8728 3120348 ChemDiv3_009289 COc1ccc(Cl)cc1NC(=O)c2nnn(CC(=O)Nc3c(C)cccc3C)c2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G06 compound treatment 1160.0 391.0 0.14 880.0 28.8 0.02 0.1137 0.8094 3120349 ChemDiv3_009290 CC(C)N(Cc1c[nH]c2ccccc12)C(=S)Nc3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G07 compound treatment 520.0 -249.0 -0.09 640.0 -211.0 -0.16 -0.1771 -0.9591 3030282 ChemDiv3_009291 COc1ccc2nc3oc(cc3cc2c1)C(=O)NC4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G08 compound treatment 1080.0 311.0 0.11 1280.0 429.0 0.33 0.3108 0.8953 3120350 ChemDiv3_009292 O=C(NCc1ccccn1)c2ccc(cc2)N3CCCC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G09 compound treatment 800.0 31.3 0.01 560.0 -291.0 -0.22 -0.1503 -0.6712 3030283 ChemDiv3_009293 CCOC(=O)C1CCCN(C1)C(=O)c2cc3cc4ccc(OC)cc4nc3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G10 compound treatment 280.0 -489.0 -0.17 1400.0 549.0 0.42 0.1753 0.3848 3120351 ChemDiv3_009294 O=C(NCCc1ccccc1)c2cccc(c2)N3CCCC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G11 compound treatment 560.0 -209.0 -0.07 240.0 -611.0 -0.47 -0.3842 -0.8087 3120352 ChemDiv3_009295 Clc1cccc(NC(=O)c2cc3cc4ccc(Cl)cc4nc3o2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G12 compound treatment 1440.0 671.0 0.24 520.0 -331.0 -0.25 -0.0114 -0.0328 3030284 ChemDiv3_009296 CCOC(=O)CN1CC2(OC3C=C2)C(C3C(=O)Nc4ccc(CC)cc4)C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G13 compound treatment 400.0 -369.0 -0.13 360.0 -491.0 -0.38 -0.3592 -0.8998 3120353 ChemDiv3_009297 Cc1ccc(cc1)n2ncc3c(=O)n(c4ccc(F)c(Cl)c4)c(nc23)c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G14 compound treatment 280.0 -489.0 -0.17 1120.0 269.0 0.21 0.0233 0.0864 3120354 ChemDiv3_009298 Oc1cc(nn1c2ccccc2)C3CCN(CC3)C(=S)Nc4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G15 compound treatment 1040.0 271.0 0.1 480.0 -371.0 -0.29 -0.1335 -0.4438 3030285 ChemDiv3_009299 CCN(Cc1ccccc1)C(=O)c2oc(=O)c3ccccc3c2c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G16 compound treatment 680.0 -88.8 -0.03 1880.0 1030.0 0.79 0.5362 0.6784 3120355 ChemDiv3_009300 S=C(N1CCOCC1)/C(=C/N2CCOCC2)/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G17 compound treatment 640.0 -129.0 -0.05 320.0 -531.0 -0.41 -0.3207 -0.7814 3030286 ChemDiv3_009301 O=C(N1CCN(CC1)c2ccccn2)c3ccc(CNS(=O)(=O)c4ccccc4)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G18 compound treatment 3320.0 2550.0 0.91 840.0 -11.3 -0.01 0.6339 0.7003 3120356 ChemDiv3_009302 CCOc1ccc(/N=C/C2C(Oc3ccc(Cl)cc3)C(=O)N2c4ccc(OCC)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G19 compound treatment 600.0 -169.0 -0.06 400.0 -451.0 -0.35 -0.2873 -0.8172 3120357 ChemDiv3_009303 CCc1ccccc1NS(=O)(=O)c2ccc3[nH]cc(C(=O)NCC4CCCO4)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G20 compound treatment 7280.0 6510.0 2.31 1720.0 869.0 0.67 2.1049 0.8755 1876301 ChemDiv3_009304 Nc1sc2CCCCc2c1C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G21 compound treatment 1640.0 871.0 0.31 440.0 -411.0 -0.32 -0.0047 -0.0106 3120358 ChemDiv3_009305 Cc1cc(C)cc(NS(=O)(=O)c2ccc3[nH]cc(C(=O)NCCC4=CCCCC4)c(=O)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G22 compound treatment 320.0 -449.0 -0.16 1600.0 749.0 0.57 0.2939 0.4927 3030287 ChemDiv3_009306 COc1ccccc1c2cc(N)n(CCC#N)n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G23 mock treatment 1600.0 831.0 0.29 320.0 -531.0 -0.41 -0.0799 -0.1587 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 G24 mock treatment 1960.0 1190.0 0.42 480.0 -371.0 -0.29 0.0973 0.1909 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H01 compound treatment 1040.0 271.0 0.1 600.0 -251.0 -0.19 -0.0684 -0.3171 3030288 ChemDiv3_009307 CCc1ccc(NC2N(C(=O)c3ccccc23)c4ccccc4C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H02 compound treatment 360.0 -409.0 -0.15 480.0 -371.0 -0.29 -0.3041 -0.9509 3120359 ChemDiv3_009308 O=C(Nc1cccnc1)c2cc3c(=O)[nH]c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H03 compound treatment 600.0 -169.0 -0.06 520.0 -331.0 -0.25 -0.2222 -0.8503 3120360 ChemDiv3_009309 CC1(CC2NC(=O)N1c3ccc(cc3)C(=O)NCc4ccccc4)Oc5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H04 compound treatment 920.0 151.0 0.05 560.0 -291.0 -0.22 -0.1202 -0.5226 3030289 ChemDiv3_009310 Cc1ccc(cc1)n2nc(C(=O)NCCc3ccc(Cl)cc3)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H05 compound treatment 640.0 -129.0 -0.05 440.0 -411.0 -0.32 -0.2555 -0.8011 3120361 ChemDiv3_009311 CN(C(=O)Cn1ncc2c(=O)oc3ccccc3c12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H06 compound treatment 360.0 -409.0 -0.15 440.0 -411.0 -0.32 -0.3258 -0.9377 3030290 ChemDiv3_009312 CC(=O)N1CCc2cc(ccc12)S(=O)(=O)NCCC(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H07 compound treatment 440.0 -329.0 -0.12 2560.0 1710.0 1.31 0.8451 0.6417 3120362 ChemDiv3_009313 Cc1nn(C)c(C)c1S(=O)(=O)N2CCC(CC2)C(=O)NCc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H08 compound treatment 360.0 -409.0 -0.15 360.0 -491.0 -0.38 -0.3692 -0.9138 3030291 ChemDiv3_009314 CC1CCN(CC1)S(=O)(=O)c2c[nH]cn2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H09 compound treatment 480.0 -289.0 -0.1 520.0 -331.0 -0.25 -0.2523 -0.9201 3120363 ChemDiv3_009315 CSC1=NCCN1C(=O)C2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H10 compound treatment 280.0 -489.0 -0.17 400.0 -451.0 -0.35 -0.3676 -0.9488 3030292 ChemDiv3_009316 C(CSc1nnc2sc3ccccc3n12)Oc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H11 compound treatment 520.0 -249.0 -0.09 440.0 -411.0 -0.32 -0.2856 -0.8713 3120364 ChemDiv3_009317 CC(Oc1ccccc1)C(=O)N2CCN=C2SCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H12 compound treatment 720.0 -48.8 -0.02 440.0 -411.0 -0.32 -0.2355 -0.7447 3120365 ChemDiv3_009318 CCc1ccc(NC(=O)c2cnc3sccn3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H13 compound treatment 560.0 -209.0 -0.07 1240.0 389.0 0.3 0.1587 0.516 3030293 ChemDiv3_009319 CCC(=O)N1CCCc2cc(ccc12)S(=O)(=O)CCC(=O)Nc3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H14 compound treatment 800.0 31.3 0.01 320.0 -531.0 -0.41 -0.2806 -0.6876 3120366 ChemDiv3_009320 Cn1c(=O)cc(SCC(=O)N2CCN(CC2)c3cccc(Cl)c3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H15 compound treatment 280.0 -489.0 -0.17 440.0 -411.0 -0.32 -0.3459 -0.9602 3120538 ChemDiv3_009321 CCC(Sc1nc2cc(OC)c(OC)cc2c3nc(C)nn13)C(=O)NCc4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H16 compound treatment 440.0 -329.0 -0.12 400.0 -451.0 -0.35 -0.3274 -0.8958 3030294 ChemDiv3_009322 CCN1CCCC1CNC(=O)CSc2cc(=O)n(C)c3cc(Cl)ccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H17 compound treatment 640.0 -129.0 -0.05 360.0 -491.0 -0.38 -0.299 -0.787 3120539 ChemDiv3_009323 Fc1cccc(NC(=O)c2cccc3CN(Cc4cccnc4)C(=O)c32)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H18 compound treatment 2800.0 2030.0 0.72 680.0 -171.0 -0.13 0.4166 0.5687 3120540 ChemDiv3_009324 O=C(CCNS(=O)(=O)c1ccc2NC(=O)CCc2c1)NC3CCCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H19 compound treatment 600.0 -169.0 -0.06 560.0 -291.0 -0.22 -0.2004 -0.8659 3030295 ChemDiv3_009325 CCc1ccc(NC(=O)c2cccc3CN(CCOC)C(=O)c32)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H20 compound treatment 1040.0 271.0 0.1 640.0 -211.0 -0.16 -0.0466 -0.2473 3030332 ChemDiv3_009326 COc1cc(cc(OC)c1OC)C(=O)NCC(N2CCOCC2)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H21 compound treatment 1560.0 791.0 0.28 440.0 -411.0 -0.32 -0.0248 -0.0586 3030333 ChemDiv3_009327 COC(CNC(=O)c1cccc2CN(C(=O)c21)c3ccc(OC)cc3)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H22 compound treatment 720.0 -48.8 -0.02 680.0 -171.0 -0.13 -0.1052 -0.7933 3030334 ChemDiv3_009328 CC1CCCN(Cc2nc3n(C)c(=O)n(C)c(=O)c3n2CCc4ccccc4)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H23 mock treatment 800.0 31.3 0.01 1360.0 509.0 0.39 0.284 0.7269 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 H24 mock treatment 640.0 -129.0 -0.05 280.0 -571.0 -0.44 -0.3424 -0.7765 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I01 compound treatment 280.0 -489.0 -0.17 440.0 -411.0 -0.32 -0.3459 -0.9602 3030335 ChemDiv3_009329 COc1ccc(CCNC(=O)CSc2nc3n(ncc3c(=O)[nH]2)c4ccc(C)cc4)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I02 compound treatment 800.0 31.3 0.01 280.0 -571.0 -0.44 -0.3023 -0.689 3030336 ChemDiv3_009330 CCc1ccccc1Nc2cc(C(=O)NCC3COc4ccccc4O3)c5ccccc5n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I03 compound treatment 560.0 -209.0 -0.07 280.0 -571.0 -0.44 -0.3625 -0.815 3120541 ChemDiv3_009331 COc1ccc(CNC(=O)c2cccn3c(=O)c4c5CCCCc5sc4nc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I04 compound treatment 4680.0 3910.0 1.39 360.0 -491.0 -0.38 0.7144 0.4969 3030337 ChemDiv3_009332 CCC(C)NC(=O)c1cc(Nc2ccc(cc2)C(C)C)nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I05 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3120542 ChemDiv3_009333 CCc1ccccc1NC(=O)Cn2nnc(C(=O)NCc3ccccc3)c2N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I06 compound treatment 320.0 -449.0 -0.16 320.0 -531.0 -0.41 -0.401 -0.9158 3120543 ChemDiv3_009334 CCC(C)N(Cc1c[nH]c2ccccc12)C(=S)Nc3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I07 compound treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 3030338 ChemDiv3_009335 COc1ccc2cc3cc(oc3nc2c1)C(=O)Nc4ccc(Oc5ccccc5)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I08 compound treatment 320.0 -449.0 -0.16 400.0 -451.0 -0.35 -0.3575 -0.9378 3120544 ChemDiv3_009336 CC(C)NC(=O)c1ccc(cc1)N2CCCC2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I09 compound treatment 520.0 -249.0 -0.09 480.0 -371.0 -0.29 -0.2639 -0.8846 3030339 ChemDiv3_009337 COc1ccc2cc3cc(oc3nc2c1)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I10 compound treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 3120545 ChemDiv3_009338 Clc1ccc(cc1)N2C(c3cccs3)c4c(n[nH]c4C2=O)c5ccc(Br)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I11 compound treatment 440.0 -329.0 -0.12 280.0 -571.0 -0.44 -0.3926 -0.8651 3030340 ChemDiv3_009339 CC(C)NC(=O)c1cc2cc3ccc(Cl)cc3nc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I12 compound treatment 1080.0 311.0 0.11 360.0 -491.0 -0.38 -0.1886 -0.4799 3120546 ChemDiv3_009340 CC(C)c1ccc(NC(=O)C2C3OC4(CN(Cc5cccnc5)C(=O)C24)C=C3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I13 compound treatment 320.0 -449.0 -0.16 560.0 -291.0 -0.22 -0.2707 -0.9861 3120547 ChemDiv3_009341 Cc1cccc(CCNC(=O)C2CCN(CC2)S(=O)(=O)c3cccc4cccnc34)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I14 compound treatment 600.0 -169.0 -0.06 360.0 -491.0 -0.38 -0.309 -0.8092 3030341 ChemDiv3_009342 CCOC(=O)N1CCC(CC1)NC(=O)c2cc(ccc2CO)C(=O)NCc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I15 compound treatment 440.0 -329.0 -0.12 320.0 -531.0 -0.41 -0.3709 -0.8743 3120548 ChemDiv3_009343 Cc1ccc(cc1)c2c(oc(=O)c3ccccc23)C(=O)NCCc4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I16 compound treatment 280.0 -489.0 -0.17 880.0 28.8 0.02 -0.107 -0.6122 3030342 ChemDiv3_009344 Cc1c(cnc2cc(nn12)c3ccccc3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I17 compound treatment 400.0 -369.0 -0.13 320.0 -531.0 -0.41 -0.3809 -0.8893 3120549 ChemDiv3_009345 Brc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I18 compound treatment 360.0 -409.0 -0.15 760.0 -91.3 -0.07 -0.1521 -0.9443 3030343 ChemDiv3_009346 O=C1N(C(Nc2ccccc2)c3ccccc13)c4cccnc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I19 compound treatment 400.0 -369.0 -0.13 1520.0 669.0 0.51 0.2705 0.5106 3120550 ChemDiv3_009347 CCc1ccc(NS(=O)(=O)c2ccc3[nH]cc(C(=O)NC)c(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I20 compound treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 3120551 ChemDiv3_009348 Cc1ccccc1N2C(CNCCc3ccccc3)C(Oc4ccc(Cl)cc4)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I21 compound treatment 440.0 -329.0 -0.12 400.0 -451.0 -0.35 -0.3274 -0.8958 3030344 ChemDiv3_009349 CCN(CC)C(=O)c1c[nH]c2ccc(cc2c1=O)S(=O)(=O)Nc3cc(C)cc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I22 compound treatment 480.0 -289.0 -0.1 1240.0 389.0 0.3 0.1386 0.4393 3120552 ChemDiv3_009350 COc1ccccc1c2nn(CCC#N)c3nc(cc(C4CC4)c23)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I23 mock treatment 360.0 -409.0 -0.15 360.0 -491.0 -0.38 -0.3692 -0.9138 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 I24 mock treatment 280.0 -489.0 -0.17 240.0 -611.0 -0.47 -0.4544 -0.9083 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J01 compound treatment 240.0 -529.0 -0.19 320.0 -531.0 -0.41 -0.421 -0.9379 3030345 ChemDiv3_009351 O=C(NCc1ccccc1)c2cccc3CN(C4CCCCC4)C(=O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J02 compound treatment 400.0 -369.0 -0.13 320.0 -531.0 -0.41 -0.3809 -0.8893 3120553 ChemDiv3_009352 COc1ccc(cc1)n2nc(C(=O)NC3CCCC(C)C3C)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J03 compound treatment 280.0 -489.0 -0.17 560.0 -291.0 -0.22 -0.2807 -0.9921 3120554 ChemDiv3_009353 O=C(Cn1ncc2c(=O)oc3ccccc3c12)Nc4nc5ccccc5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J04 compound treatment 320.0 -449.0 -0.16 240.0 -611.0 -0.47 -0.4444 -0.8968 3030346 ChemDiv3_009354 CCOC(=O)N1CCC(CC1)NC(=O)c2nn(c3ccc(C)cc3)c(=O)c4n(C)c5ccccc5c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J05 compound treatment 280.0 -489.0 -0.17 960.0 109.0 0.08 -0.0636 -0.3303 3120555 ChemDiv3_009355 Fc1ccccc1N2CCN(CCCNC(=O)Cn3ncc4c(=O)oc5ccccc5c34)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J06 compound treatment 5360.0 4590.0 1.63 280.0 -571.0 -0.44 0.8416 0.4989 3120556 ChemDiv3_009356 COc1cccc(c1)c2nn(C)c3sc(cc23)C(=O)N4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J07 compound treatment 440.0 -329.0 -0.12 320.0 -531.0 -0.41 -0.3709 -0.8743 3030347 ChemDiv3_009357 Cc1nn(C)c(C)c1S(=O)(=O)N2CCC(CC2)C(=O)Nc3ccc(C)cc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J08 compound treatment 520.0 -249.0 -0.09 440.0 -411.0 -0.32 -0.2856 -0.8713 3120557 ChemDiv3_009358 CC1Cc2ccccc2N1S(=O)(=O)c3c[nH]cn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J09 compound treatment 3120.0 2350.0 0.83 600.0 -251.0 -0.19 0.4534 0.5296 3030348 ChemDiv3_009359 CSC1=NCCN1C(=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J10 compound treatment 360.0 -409.0 -0.15 320.0 -531.0 -0.41 -0.3909 -0.9031 3120558 ChemDiv3_009360 CCSc1nnc2[nH]c3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J11 compound treatment 320.0 -449.0 -0.16 1360.0 509.0 0.39 0.1636 0.3879 3030349 ChemDiv3_009361 O=C(Cc1ccccc1)N2CCN=C2SCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J12 compound treatment 640.0 -129.0 -0.05 320.0 -531.0 -0.41 -0.3207 -0.7814 3120559 ChemDiv3_009362 COc1ccc(CNC(=O)c2cnc3scc(C)n3c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J13 compound treatment 360.0 -409.0 -0.15 280.0 -571.0 -0.44 -0.4126 -0.8933 3030350 ChemDiv3_009363 CC(=O)N1CCCc2cc(ccc12)S(=O)(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J14 compound treatment 320.0 -449.0 -0.16 240.0 -611.0 -0.47 -0.4444 -0.8968 3120560 ChemDiv3_009364 Cn1c(=O)cc(SCC(=O)NCC2CCCO2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J15 compound treatment 720.0 -48.8 -0.02 200.0 -651.0 -0.5 -0.3658 -0.7311 3120561 ChemDiv3_009365 COc1cc2nc(SCC(=O)N(C)C3CCCCC3)n4nc(C)nc4c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J16 compound treatment 280.0 -489.0 -0.17 600.0 -251.0 -0.19 -0.259 -0.9986 3030351 ChemDiv3_009366 Cn1c(=O)cc(SCC(=O)NCCN2CCOCC2)c3ccc(Cl)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J17 compound treatment 280.0 -489.0 -0.17 240.0 -611.0 -0.47 -0.4544 -0.9083 3120562 ChemDiv3_009367 O=C(NCc1ccco1)c2cccc3CN(Cc4cccnc4)C(=O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J18 compound treatment 320.0 -449.0 -0.16 480.0 -371.0 -0.29 -0.3141 -0.9621 3120563 ChemDiv3_009368 Cc1ccc(Cl)cc1N2CCN(CC2)C(=O)CCNS(=O)(=O)c3ccc4NC(=O)CCc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J19 compound treatment 320.0 -449.0 -0.16 1280.0 429.0 0.33 0.1202 0.3287 3030352 ChemDiv3_009369 COCCN1Cc2cccc(C(=O)NC(C)C3(CC4CC5CC(C4)C3)C5)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J20 compound treatment 440.0 -329.0 -0.12 760.0 -91.3 -0.07 -0.132 -0.9703 3120564 ChemDiv3_009370 O=C(NCC(N1CCOCC1)c2cccnc2)c3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J21 compound treatment 400.0 -369.0 -0.13 1360.0 509.0 0.39 0.1837 0.4459 3030353 ChemDiv3_009371 O=C(N1CCCC1)c2cc3c(=O)[nH]c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J22 compound treatment 320.0 -449.0 -0.16 280.0 -571.0 -0.44 -0.4227 -0.9059 3120727 ChemDiv3_009372 OC1=C2C(Sc3ccccc3N=C2c4ccccc14)c5ccccc5F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J23 mock treatment 280.0 -489.0 -0.17 760.0 -91.3 -0.07 -0.1721 -0.9205 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 J24 mock treatment 400.0 -369.0 -0.13 1000.0 149.0 0.11 -0.0117 -0.0677 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K01 compound treatment 840.0 71.3 0.03 1360.0 509.0 0.39 0.2941 0.7513 3120728 ChemDiv3_009373 Cc1ccc(cc1C)n2ncc3c(=O)[nH]c(SCC=C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K02 compound treatment 1280.0 511.0 0.18 680.0 -171.0 -0.13 0.0353 0.1575 3030354 ChemDiv3_009374 CCc1ccccc1Nc2cc(C(=O)NCCN3CCCCCC3)c4ccccc4n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K03 compound treatment 1520.0 751.0 0.27 400.0 -451.0 -0.35 -0.0565 -0.1293 3120729 ChemDiv3_009375 CC1CCCCC1NC(=O)c2cccn3c(=O)c4c5CCCCc5sc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K04 compound treatment 600.0 -169.0 -0.06 240.0 -611.0 -0.47 -0.3742 -0.7909 3120730 ChemDiv3_009376 COc1ccc(CNC(=O)c2cc(Nc3ccccc3OC)nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K05 compound treatment 640.0 -129.0 -0.05 480.0 -371.0 -0.29 -0.2338 -0.8101 3030355 ChemDiv3_009377 COc1ccc2nc3oc(cc3cc2c1)C(=O)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K06 compound treatment 640.0 -129.0 -0.05 400.0 -451.0 -0.35 -0.2773 -0.7935 3120731 ChemDiv3_009378 CCOc1ccc(NC(=O)N(Cc2cn(C)c3ccccc23)C4CCCCC4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K07 compound treatment 840.0 71.3 0.03 400.0 -451.0 -0.35 -0.2271 -0.6538 3030356 ChemDiv3_009379 COc1ccc2cc3cc(oc3nc2c1)C(=O)N(C)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K08 compound treatment 1960.0 1190.0 0.42 680.0 -171.0 -0.13 0.2059 0.4651 3120732 ChemDiv3_009380 O=C(NCCCN1CCCC1=O)c2ccc(cc2)N3CCCC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K09 compound treatment 880.0 111.0 0.04 400.0 -451.0 -0.35 -0.2171 -0.6225 3120733 ChemDiv3_009381 COc1ccc2cc3cc(oc3nc2c1)C(=O)N(C)c4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K10 compound treatment 600.0 -169.0 -0.06 360.0 -491.0 -0.38 -0.309 -0.8092 3030357 ChemDiv3_009382 Cc1ccc(cc1)c2n[nH]c3C(=O)N(C(c23)c4ccccc4Cl)c5ccc(Cl)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K11 compound treatment 640.0 -129.0 -0.05 760.0 -91.3 -0.07 -0.0818 -0.9785 3120734 ChemDiv3_009383 CCN1CCN(CCCNC(=O)c2cc3cc4ccc(Cl)cc4nc3o2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K12 compound treatment 720.0 -48.8 -0.02 840.0 -11.3 -0.01 -0.0183 -0.9485 1500716 ChemDiv3_009384 CCCN1C(=O)c2ccc(cc2C1=O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K13 compound treatment 960.0 191.0 0.07 560.0 -291.0 -0.22 -0.1101 -0.4713 3120735 ChemDiv3_009385 CC1CCCCN1C(=O)c2oc(=O)c3ccccc3c2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K14 compound treatment 920.0 151.0 0.05 480.0 -371.0 -0.29 -0.1636 -0.5641 3120736 ChemDiv3_009386 CC(C)(C)OC(=O)N1CCC(CC1)c2cc(O)n3ncc(C(=O)Nc4ccc(F)c(Cl)c4)c3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K15 compound treatment 760.0 -8.75 0.0 880.0 28.8 0.02 0.0134 0.6017 1332995 ChemDiv3_009387 Cc1ccc(cc1)c2c(oc(=O)c3ccccc23)C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K16 compound treatment 1000.0 231.0 0.08 400.0 -451.0 -0.35 -0.187 -0.5251 3120737 ChemDiv3_009388 COc1ccc(CNC(=O)c2ccc3C(=O)N(Cc4ccco4)C(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K17 compound treatment 640.0 -129.0 -0.05 680.0 -171.0 -0.13 -0.1253 -0.9 3030358 ChemDiv3_009389 Brc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K18 compound treatment 1000.0 231.0 0.08 400.0 -451.0 -0.35 -0.187 -0.5251 3120738 ChemDiv3_009390 Cc1ccccc1/N=C/C=N/c2ccccc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K19 compound treatment 440.0 -329.0 -0.12 920.0 68.8 0.05 -0.0451 -0.3527 3030359 ChemDiv3_009391 CCCN(CCC)C(=O)c1c[nH]c2ccc(cc2c1=O)S(=O)(=O)Nc3ccc(CC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K20 compound treatment 760.0 -8.75 0.0 640.0 -211.0 -0.16 -0.1169 -0.7205 3120739 ChemDiv3_009392 CCOC(=O)CCc1c(C)nc2ccc(Br)cn2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K21 compound treatment 1080.0 311.0 0.11 440.0 -411.0 -0.32 -0.1452 -0.434 3120740 ChemDiv3_009393 COc1ccc(Nc2cc(C(=O)NCc3ccco3)c4ccccc4n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K22 compound treatment 8080.0 7310.0 2.59 600.0 -251.0 -0.19 1.6976 0.6527 3030360 ChemDiv3_009394 Brc1cnc(nc1)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K23 mock treatment 720.0 -48.8 -0.02 1160.0 309.0 0.24 0.1554 0.6538 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 K24 mock treatment 1000.0 231.0 0.08 480.0 -371.0 -0.29 -0.1435 -0.4839 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L01 compound treatment 1040.0 271.0 0.1 600.0 -251.0 -0.19 -0.0684 -0.3171 3120741 ChemDiv3_009395 O=C(NCCc1ccccc1)c2cc(c(s2)N3CCOCC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L02 compound treatment 1080.0 311.0 0.11 400.0 -451.0 -0.35 -0.1669 -0.459 3030361 ChemDiv3_009396 COc1ccc(cc1)n2nc(C(=O)NCC3CCCO3)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L03 compound treatment 520.0 -249.0 -0.09 440.0 -411.0 -0.32 -0.2856 -0.8713 3120742 ChemDiv3_009397 Clc1cccc(NC(=O)Cn2ncc3c(=O)oc4ccccc4c23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L04 compound treatment 760.0 -8.75 0.0 400.0 -451.0 -0.35 -0.2472 -0.7134 3120743 ChemDiv3_009398 CC(CCc1ccccc1)NC(=O)c2nn(c3ccc(C)cc3)c(=O)c4n(C)c5ccccc5c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L05 compound treatment 520.0 -249.0 -0.09 840.0 -11.3 -0.01 -0.0685 -0.7726 3030362 ChemDiv3_009399 Cn1c(cc2c(=O)oc3ccccc3c12)C(=O)Nc4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L06 compound treatment 600.0 -169.0 -0.06 480.0 -371.0 -0.29 -0.2439 -0.8374 3120744 ChemDiv3_009400 COc1cccc(c1)c2nn(C)c3sc(cc23)C(=O)N4CCCCC4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L07 compound treatment 1040.0 271.0 0.1 320.0 -531.0 -0.41 -0.2204 -0.5258 3120745 ChemDiv3_009401 Cc1ccc(cc1)N(CC(=O)NCc2cccs2)S(=O)(=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L08 compound treatment 400.0 -369.0 -0.13 400.0 -451.0 -0.35 -0.3375 -0.9113 3030393 ChemDiv3_009402 Cc1cccc(CCNS(=O)(=O)c2c[nH]cn2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L09 compound treatment 520.0 -249.0 -0.09 400.0 -451.0 -0.35 -0.3074 -0.8598 3120746 ChemDiv3_009403 CSC1=NCCN1C(=O)COc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L10 compound treatment 1320.0 551.0 0.2 400.0 -451.0 -0.35 -0.1067 -0.2682 3030394 ChemDiv3_009404 CCSc1nnc2n(CC)c3ccccc3n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L11 compound treatment 360.0 -409.0 -0.15 520.0 -331.0 -0.25 -0.2824 -0.9645 3120747 ChemDiv3_009405 Fc1cccc(Cl)c1CSC2=NCCN2C(=O)c3ccc(cc3)S(=O)(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L12 compound treatment 600.0 -169.0 -0.06 440.0 -411.0 -0.32 -0.2656 -0.8265 3030395 ChemDiv3_009406 CN(C(=O)c1cnc2scc(C)n2c1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L13 compound treatment 1040.0 271.0 0.1 520.0 -331.0 -0.25 -0.1118 -0.4111 3120748 ChemDiv3_009407 CCCN(CCC)S(=O)(=O)c1ccc2N(CCCc2c1)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L14 compound treatment 720.0 -48.8 -0.02 1000.0 149.0 0.11 0.0685 0.5933 3120749 ChemDiv3_009408 Cn1c(=O)cc(SCC(=O)NCc2cccnc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L15 compound treatment 560.0 -209.0 -0.07 400.0 -451.0 -0.35 -0.2973 -0.8393 3030396 ChemDiv3_009409 COc1cc2nc(SCc3ccc(C)cc3)n4nc(nc4c2cc1OC)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L16 compound treatment 1160.0 391.0 0.14 560.0 -291.0 -0.22 -0.06 -0.2279 3120750 ChemDiv3_009410 CCN(CC)C(=O)CSc1cc(=O)n(C)c2cc(Cl)ccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L17 compound treatment 880.0 111.0 0.04 1960.0 1110.0 0.85 0.6298 0.7391 3120751 ChemDiv3_009411 CCOC(=O)c1ccc(NC(=O)c2cccc3CN(Cc4cccnc4)C(=O)c32)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L18 compound treatment 720.0 -48.8 -0.02 280.0 -571.0 -0.44 -0.3223 -0.7344 3030397 ChemDiv3_009412 COc1ccccc1N2CCN(CC2)C(=O)CCNS(=O)(=O)c3ccc4NC(=O)CCc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L19 compound treatment 480.0 -289.0 -0.1 680.0 -171.0 -0.13 -0.1654 -0.9924 3120752 ChemDiv3_009413 COCCN1Cc2cccc(C(=O)Nc3ccc4c(C)cc(=O)oc4c3)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L20 compound treatment 560.0 -209.0 -0.07 560.0 -291.0 -0.22 -0.2105 -0.8936 3030398 ChemDiv3_009414 O=C(NCC(N1CCOCC1)c2cccnc2)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L21 compound treatment 4520.0 3750.0 1.33 720.0 -131.0 -0.1 0.8697 0.6517 3120753 ChemDiv3_009415 O=C(NCC1CCCO1)c2cc3c(=O)[nH]c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L22 compound treatment 960.0 191.0 0.07 1040.0 189.0 0.14 0.1504 0.9402 3120754 ChemDiv3_009416 OC1=C2C(Sc3ccccc3N=C2c4ccccc14)c5ccsc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L23 mock treatment 600.0 -169.0 -0.06 640.0 -211.0 -0.16 -0.157 -0.9082 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 L24 mock treatment 640.0 -129.0 -0.05 880.0 28.8 0.02 -0.0167 -0.329 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M01 compound treatment 960.0 191.0 0.07 1840.0 989.0 0.76 0.5847 0.7672 3030399 ChemDiv3_009417 CCOC(=O)C(CC)Sc1nc2n(ncc2c(=O)[nH]1)c3ccc(C)c(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M02 compound treatment 4040.0 3270.0 1.16 680.0 -171.0 -0.13 0.7276 0.623 3120933 ChemDiv3_009418 CCc1ccc(Nc2cc(C(=O)NCC(OC)OC)c3ccccc3n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M03 compound treatment 360.0 -409.0 -0.15 1040.0 189.0 0.14 -1.0E-4 -3.0E-4 3120934 ChemDiv3_009419 CC(C)CCNC(=O)c1cccn2c(=O)c3c4CCCCc4sc3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M04 compound treatment 760.0 -8.75 0.0 840.0 -11.3 -0.01 -0.0083 -0.9046 3030400 ChemDiv3_009420 COc1ccccc1Nc2cc(C(=O)NCCN3CCC(Cc4ccccc4)CC3)c5ccccc5n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M05 compound treatment 1400.0 631.0 0.22 560.0 -291.0 -0.22 2.0E-4 7.0E-4 3120935 ChemDiv3_009421 CCC(C)NC(=O)c1cc2cc3cc(OC)ccc3nc2o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M06 compound treatment 560.0 -209.0 -0.07 440.0 -411.0 -0.32 -0.2756 -0.8499 3120936 ChemDiv3_009422 CC(C)N(Cc1cn(C)c2ccccc12)C(=S)Nc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M07 compound treatment 760.0 -8.75 0.0 480.0 -371.0 -0.29 -0.2037 -0.7148 3030401 ChemDiv3_009423 COc1ccc2cc3cc(oc3nc2c1)C(=O)NC4CCCC(C)C4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M08 compound treatment 880.0 111.0 0.04 720.0 -131.0 -0.1 -0.0433 -0.4005 3120937 ChemDiv3_009424 CC1CCCC(NC(=O)c2ccc(cc2)N3CCCC3=O)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M09 compound treatment 800.0 31.3 0.01 440.0 -411.0 -0.32 -0.2154 -0.6819 3120938 ChemDiv3_009425 CCCN(C(=O)c1cc2cc3ccc(OC)cc3nc2o1)c4ccc(CC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M10 compound treatment 680.0 -88.8 -0.03 480.0 -371.0 -0.29 -0.2238 -0.7805 3030402 ChemDiv3_009426 Cc1n[nH]c2C(=O)N(C(c12)c3ccc(C)cc3)c4ccc(C)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M11 compound treatment 11720.0 11000.0 3.88 6800.0 5950.0 4.57 5.9764 0.9968 3120939 ChemDiv3_009427 N=C/1N2N=CSC2=NC(=O)\C1=C\c3cccn3c4ccc5ccccc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M12 compound treatment 1120.0 351.0 0.12 640.0 -211.0 -0.16 -0.0266 -0.1299 3030403 ChemDiv3_009428 CCOC(=O)N1CCC(CC1)c2nc3ccccc3[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M13 compound treatment 880.0 111.0 0.04 440.0 -411.0 -0.32 -0.1953 -0.6139 3120940 ChemDiv3_009429 CCCNC(=O)c1oc(=O)c2ccccc2c1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M14 compound treatment 2160.0 1390.0 0.49 560.0 -291.0 -0.22 0.1909 0.3523 3030404 ChemDiv3_009430 CCOC(=O)N1CCC(CC1)N2Cc3cccc(C(=O)O)c3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M15 compound treatment 720.0 -48.8 -0.02 720.0 -131.0 -0.1 -0.0835 -0.8165 3120941 ChemDiv3_009431 CCOc1ccc(CN2C(=O)c3ccccc3Sc4ccc(cc24)C(=O)N5CCOCC5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M16 compound treatment 8120.0 7350.0 2.61 1080.0 229.0 0.18 1.9682 0.753 3030405 ChemDiv3_009432 OC1N(C(=O)c2ccccc12)c3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M17 compound treatment 920.0 151.0 0.05 1160.0 309.0 0.24 0.2055 0.8458 3120942 ChemDiv3_009433 CC1CCCC(NC(=O)c2ccc(CNS(=O)(=O)c3ccc(NC(=O)C)cc3)cc2)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M18 compound treatment 320.0 -449.0 -0.16 720.0 -131.0 -0.1 -0.1838 -0.9757 3030406 ChemDiv3_009434 CCOC(=O)CCn1nc(cc1N)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M19 compound treatment 600.0 -169.0 -0.06 920.0 68.8 0.05 -0.005 -0.0628 3120943 ChemDiv3_009435 CCc1ccc(NS(=O)(=O)c2ccc3[nH]cc(C(=O)N4CCCC4)c(=O)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M20 compound treatment 1200.0 431.0 0.15 720.0 -131.0 -0.1 0.0369 0.2016 3030407 ChemDiv3_009436 CCOC(=O)CCc1c(C)nc2ccc(C)cn2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M21 compound treatment 2360.0 1590.0 0.56 800.0 -51.3 -0.04 0.3713 0.6562 3120944 ChemDiv3_009437 COc1ccc(Nc2cc(C(=O)NCCc3ccccc3)c4ccccc4n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M22 compound treatment 680.0 -88.8 -0.03 840.0 -11.3 -0.01 -0.0284 -0.869 3030408 ChemDiv3_009438 OC(=O)c1cnc(nc1)N2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M23 mock treatment 600.0 -169.0 -0.06 960.0 109.0 0.08 0.0167 0.1626 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 M24 mock treatment 640.0 -129.0 -0.05 1840.0 989.0 0.76 0.5045 0.6634 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N01 compound treatment 600.0 -169.0 -0.06 240.0 -611.0 -0.47 -0.3742 -0.7909 3120945 ChemDiv3_009439 CCc1cccc(NC(=O)c2cccc3CN(CC4CCCO4)C(=O)c32)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N02 compound treatment 560.0 -209.0 -0.07 800.0 -51.3 -0.04 -0.0802 -0.9562 3030409 ChemDiv3_009440 CCN(CC)C(=O)c1nn(c2ccc(OC)cc2)c(=O)c3n(C)c4ccccc4c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N03 compound treatment 400.0 -369.0 -0.13 560.0 -291.0 -0.22 -0.2506 -0.9674 3120946 ChemDiv3_009441 O=C(Cn1ncc2c(=O)oc3ccccc3c12)N4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N04 compound treatment 800.0 31.3 0.01 720.0 -131.0 -0.1 -0.0634 -0.6255 3120947 ChemDiv3_009442 Cc1[nH]c2ccc(F)cc2c1CCN(Cc3ccco3)C(=S)NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N05 compound treatment 1520.0 751.0 0.27 360.0 -491.0 -0.38 -0.0782 -0.1694 3030410 ChemDiv3_009443 Cc1ccc(NC(=O)c2cc3c(=O)oc4ccccc4c3n2C)cc1F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N06 compound treatment 1720.0 951.0 0.34 880.0 28.8 0.02 0.2542 0.7518 3120948 ChemDiv3_009444 COc1cccc(c1)c2nn(C)c3sc(cc23)C(=O)N4CCN(CC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N07 compound treatment 1080.0 311.0 0.11 560.0 -291.0 -0.22 -0.08 -0.3209 3030411 ChemDiv3_009445 COc1ccc2nc(NC(=O)CN(c3ccc(C)cc3)S(=O)(=O)c4c(C)noc4C)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N08 compound treatment 560.0 -209.0 -0.07 720.0 -131.0 -0.1 -0.1236 -0.9885 3120949 ChemDiv3_009446 Clc1ccc(CNS(=O)(=O)c2c[nH]cn2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N09 compound treatment 800.0 31.3 0.01 600.0 -251.0 -0.19 -0.1286 -0.6654 3030412 ChemDiv3_009447 CSC1=NCCN1C(=O)Cc2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N10 compound treatment 520.0 -249.0 -0.09 760.0 -91.3 -0.07 -0.1119 -0.9935 3120950 ChemDiv3_009448 C(Cn1c2nnc(SCc3ccccc3)n2c4ccccc14)Oc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N11 compound treatment 800.0 31.3 0.01 760.0 -91.3 -0.07 -0.0417 -0.5879 3120951 ChemDiv3_009449 Cc1ccc(C)c(CSC2=NCCN2C(=O)COc3ccccc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N12 compound treatment 840.0 71.3 0.03 680.0 -171.0 -0.13 -0.0751 -0.5609 3030413 ChemDiv3_009450 CC1Cc2ccccc2N1C(=O)c3cnc4scc(C)n4c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N13 compound treatment 800.0 31.3 0.01 1000.0 149.0 0.11 0.0886 0.7721 3029946 ChemDiv3_009451 CCc1ccc(NS(=O)(=O)c2ccc3N(CCCc3c2)C(=O)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N14 compound treatment 520.0 -249.0 -0.09 1280.0 429.0 0.33 0.1704 0.4999 3029947 ChemDiv3_009452 Cn1c(=O)cc(SCC(=O)N(CC=C)c2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N15 compound treatment 960.0 191.0 0.07 520.0 -331.0 -0.25 -0.1318 -0.5009 3029948 ChemDiv3_009453 COc1cc2nc(SCc3ccc(F)cc3)n4nc(nc4c2cc1OC)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N16 compound treatment 960.0 191.0 0.07 800.0 -51.3 -0.04 0.0202 0.257 3029949 ChemDiv3_009454 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)NC(CC(C)C)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N17 compound treatment 2520.0 1750.0 0.62 760.0 -91.3 -0.07 0.3898 0.6234 3029950 ChemDiv3_009455 CCc1cccc(C)c1NC(=O)c2cccc3CN(Cc4cccnc4)C(=O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N18 compound treatment 840.0 71.3 0.03 600.0 -251.0 -0.19 -0.1185 -0.6092 3120952 ChemDiv3_009456 Cc1ccc(NC(=O)CCNS(=O)(=O)c2ccc3NC(=O)CCc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N19 compound treatment 800.0 31.3 0.01 1800.0 949.0 0.73 0.5229 0.7178 3029951 ChemDiv3_009457 O=C(NC1CCCCCC1)c2cccc3CN(C4CCCCC4)C(=O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N20 compound treatment 1120.0 351.0 0.12 680.0 -171.0 -0.13 -0.0049 -0.0268 3120953 ChemDiv3_009458 CN(C)C(CNS(=O)(=O)c1ccc(F)cc1)c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N21 compound treatment 600.0 -169.0 -0.06 560.0 -291.0 -0.22 -0.2004 -0.8659 3029952 ChemDiv3_009459 COC(=O)CNC(=O)c1cc2c(=O)[nH]c3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N22 compound treatment 1280.0 511.0 0.18 480.0 -371.0 -0.29 -0.0733 -0.217 3120954 ChemDiv3_009460 COc1cc(ccc1OC(=O)C)C2Sc3ccccc3N=C4C2=C(O)c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N23 mock treatment 560.0 -209.0 -0.07 1040.0 189.0 0.14 0.0501 0.3079 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 N24 mock treatment 720.0 -48.8 -0.02 560.0 -291.0 -0.22 -0.1703 -0.7595 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O01 compound treatment 320.0 -449.0 -0.16 240.0 -611.0 -0.47 -0.4444 -0.8968 3029953 ChemDiv3_009461 CS(=O)(=O)Nc1ccc(cc1)C2=NN(C(C2)c3ccccc3F)S(=O)(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O02 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3120955 ChemDiv3_009462 CCc1ccc(Nc2cc(C(=O)NCc3cccs3)c4ccccc4n2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O03 compound treatment 2400.0 1630.0 0.58 280.0 -571.0 -0.44 0.0991 0.1365 3120956 ChemDiv3_009463 CC(C)NC(=O)c1cccn2c(=O)c3c4CCCCc4sc3nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O04 compound treatment 480.0 -289.0 -0.1 280.0 -571.0 -0.44 -0.3825 -0.8494 3029954 ChemDiv3_009464 COc1ccccc1Nc2cc(C(=O)N3CCN(Cc4ccccc4)CC3)c5ccccc5n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O05 compound treatment 240.0 -529.0 -0.19 280.0 -571.0 -0.44 -0.4427 -0.9282 3120957 ChemDiv3_009465 COc1ccc2nc3oc(cc3cc2c1)C(=O)Nc4ccc(cc4)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O06 compound treatment 520.0 -249.0 -0.09 240.0 -611.0 -0.47 -0.3942 -0.8256 3120958 ChemDiv3_009466 CCn1cc(CN(C2CCCCC2)C(=O)Nc3cccc(OC)c3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O07 compound treatment 3120.0 2350.0 0.83 320.0 -531.0 -0.41 0.3014 0.3246 3029957 ChemDiv3_009467 COc1ccc2cc3cc(oc3nc2c1)C(=O)NCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O08 compound treatment 4520.0 3750.0 1.33 360.0 -491.0 -0.38 0.6743 0.4875 3029958 ChemDiv3_009468 O=C(N1CCCC1)c2ccc(cc2)N3CCCC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O09 compound treatment 2240.0 1470.0 0.52 240.0 -611.0 -0.47 0.0372 0.053 3120959 ChemDiv3_009469 COc1ccc2cc3cc(oc3nc2c1)C(=O)N(C)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O10 compound treatment 360.0 -409.0 -0.15 320.0 -531.0 -0.41 -0.3909 -0.9031 3120960 ChemDiv3_009470 Cc1ccc(cc1)c2n[nH]c3C(=O)NC(c23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O11 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3029959 ChemDiv3_009471 Brc1ccc(cc1)n2cccc2/C=C\3/C(=N)N4C=CSC4=NC3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O12 compound treatment 320.0 -449.0 -0.16 360.0 -491.0 -0.38 -0.3792 -0.9264 3121144 ChemDiv3_009472 CCOC(=O)N1CCC(CC1)N2C(=O)c3ccc(cc3C2=O)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O13 compound treatment 520.0 -249.0 -0.09 400.0 -451.0 -0.35 -0.3074 -0.8598 1213585 ChemDiv3_009473 NS(=O)(=O)c1ccc(CCNC(=O)c2oc(=O)c3ccccc3c2c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O14 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3029961 ChemDiv3_009474 Oc1cc(nc2c(cnn12)C(=O)Nc3ccc(Cl)cc3)C4CCNCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O15 compound treatment 400.0 -369.0 -0.13 200.0 -651.0 -0.5 -0.446 -0.8631 3121145 ChemDiv3_009475 Cc1cc(C)c(c(C)c1)S(=O)(=O)NCc2ccc(cc2)C(=O)NCCc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O16 compound treatment 400.0 -369.0 -0.13 320.0 -531.0 -0.41 -0.3809 -0.8893 3029962 ChemDiv3_009476 O=C1N(C(Nc2ccc(cc2)S(=O)(=O)N3CCCCC3)c4ccccc14)c5ccccn5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O17 compound treatment 3160.0 2390.0 0.85 280.0 -571.0 -0.44 0.2897 0.3034 3121146 ChemDiv3_009477 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)C(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O18 compound treatment 400.0 -369.0 -0.13 360.0 -491.0 -0.38 -0.3592 -0.8998 3029964 ChemDiv3_009478 Cc1ccccc1N2C(CNC(C)(C)C)C(Oc3ccc(Cl)cc3)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O19 compound treatment 1600.0 831.0 0.29 320.0 -531.0 -0.41 -0.0799 -0.1587 3121147 ChemDiv3_009479 Fc1ccccc1NS(=O)(=O)c2ccc3[nH]cc(C(=O)NC4CCCC4)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O20 compound treatment 280.0 -489.0 -0.17 320.0 -531.0 -0.41 -0.411 -0.9274 3121148 ChemDiv3_009480 CC(=O)N(CCc1ccccc1)CC2C(Oc3ccc(Cl)cc3)C(=O)N2c4ccccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O21 compound treatment 280.0 -489.0 -0.17 360.0 -491.0 -0.38 -0.3893 -0.9378 3029967 ChemDiv3_009481 CCOC(=O)C1CCCN(C1)C(=O)c2cc(Nc3ccc(OC)cc3)nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O22 compound treatment 320.0 -449.0 -0.16 640.0 -211.0 -0.16 -0.2272 -1.0 3121149 ChemDiv3_009482 O=C1OCC2=C1C(NC(=O)N2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O23 mock treatment 640.0 -129.0 -0.05 320.0 -531.0 -0.41 -0.3207 -0.7814 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 O24 mock treatment 400.0 -369.0 -0.13 480.0 -371.0 -0.29 -0.294 -0.9376 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P01 compound treatment 360.0 -409.0 -0.15 320.0 -531.0 -0.41 -0.3909 -0.9031 3029804 ChemDiv3_009483 COc1cc2[nH]c(=S)nc(NCCC(C)C)c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P02 compound treatment 2520.0 1750.0 0.62 320.0 -531.0 -0.41 0.1509 0.203 3029806 ChemDiv3_009484 COc1ccc(cc1)n2nc(C(=O)N(C)c3ccccc3)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P03 compound treatment 4360.0 3590.0 1.27 400.0 -451.0 -0.35 0.6559 0.4968 3029808 ChemDiv3_009485 CN(C)CCNC(=O)Cn1ncc2c(=O)oc3ccccc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P04 compound treatment 600.0 -169.0 -0.06 840.0 -11.3 -0.01 -0.0484 -0.8008 3029811 ChemDiv3_009486 COc1ccc(OC)c(NC(=S)N(CCc2c(C)[nH]c3ccc(F)cc23)Cc4ccco4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P05 compound treatment 520.0 -249.0 -0.09 2360.0 1510.0 1.16 0.7566 0.6513 3029812 ChemDiv3_009487 CCc1cccc(NC(=O)C2CCCN(C2)S(=O)(=O)c3cccnc3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P06 compound treatment 5320.0 4550.0 1.61 1600.0 749.0 0.57 1.5481 0.9033 3029815 ChemDiv3_009488 COc1cccc(c1)c2nn(C)c3sc(cc23)C(=O)N4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P07 compound treatment 520.0 -249.0 -0.09 2160.0 1310.0 1.0 0.6481 0.6425 3121150 ChemDiv3_009489 Cc1noc(C)c1S(=O)(=O)N(CC(=O)N2CCCCCC2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P08 compound treatment 1160.0 391.0 0.14 440.0 -411.0 -0.32 -0.1251 -0.3628 3121151 ChemDiv3_009490 O=C(C1CCN(CC1)S(=O)(=O)c2c[nH]cn2)N3CCn4c3nc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P09 compound treatment 1200.0 431.0 0.15 280.0 -571.0 -0.44 -0.2019 -0.4348 3029819 ChemDiv3_009491 CCN(CC)S(=O)(=O)c1ccc(cc1)C(=O)N2CCN=C2SC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P10 compound treatment 2480.0 1710.0 0.61 280.0 -571.0 -0.44 0.1191 0.1591 3029874 ChemDiv3_009492 CCSc1nnc2n(c3ccccc3)c4ccccc4n12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P11 compound treatment 360.0 -409.0 -0.15 360.0 -491.0 -0.38 -0.3692 -0.9138 3029876 ChemDiv3_009493 Cc1ccc(C)c(CSC2=NCCN2C(=O)c3ccc(cc3)S(=O)(=O)N4CCOCC4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P12 compound treatment 1280.0 511.0 0.18 400.0 -451.0 -0.35 -0.1167 -0.2985 3029878 ChemDiv3_009494 COc1cc2NC(=S)N3C(=O)C(CCC(=O)NCCc4ccc(Cl)cc4)N=C3c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P13 compound treatment 360.0 -409.0 -0.15 280.0 -571.0 -0.44 -0.4126 -0.8933 3029881 ChemDiv3_009495 CC(=O)N1CCCc2cc(ccc12)S(=O)(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P14 compound treatment 320.0 -449.0 -0.16 320.0 -531.0 -0.41 -0.401 -0.9158 3029882 ChemDiv3_009496 Cc1ccc(NC(=O)CSc2cc(=O)n(C)c3ccccc23)nc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P15 compound treatment 520.0 -249.0 -0.09 240.0 -611.0 -0.47 -0.3942 -0.8256 3029884 ChemDiv3_009497 COc1cc2nc(SCC(=O)N)n3nc(CCn4c(C)nc5ccccc45)nc3c2cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P16 compound treatment 3440.0 2670.0 0.95 240.0 -611.0 -0.47 0.3382 0.3199 3121152 ChemDiv3_009498 CCC(=O)N1CCc2cc(ccc12)S(=O)(=O)NC(CC(C)C)C(=O)N3CCC(C)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P17 compound treatment 6240.0 5470.0 1.94 280.0 -571.0 -0.44 1.0623 0.5339 3029886 ChemDiv3_009499 CCOc1ccccc1NC(=O)c2cccc3CN(Cc4cccnc4)C(=O)c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P18 compound treatment 360.0 -409.0 -0.15 280.0 -571.0 -0.44 -0.4126 -0.8933 3121153 ChemDiv3_009500 CN(C)C(CNC(=S)Nc1ccccc1)c2cccnc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P19 compound treatment 360.0 -409.0 -0.15 480.0 -371.0 -0.29 -0.3041 -0.9509 3121154 ChemDiv3_009501 CCc1ccc(NC(=O)c2cccc3CN(C4CCCCC4)C(=O)c32)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P20 compound treatment 320.0 -449.0 -0.16 2920.0 2070.0 1.59 1.0105 0.6331 3029889 ChemDiv3_009502 CC(=O)Nc1ccc(OCCOc2ccc(/C=C\3/C(=N)N4C=CSC4=NC3=O)cc2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P21 compound treatment 280.0 -489.0 -0.17 560.0 -291.0 -0.22 -0.2807 -0.9921 3121155 ChemDiv3_009503 CC1CC(C)CN(CCCNC(=O)c2cc3c(=O)[nH]c4ccccc4c3s2)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P22 compound treatment 680.0 -88.8 -0.03 1520.0 669.0 0.51 0.3408 0.6625 3121156 ChemDiv3_009504 O=C(C(NS(=O)(=O)c1cccc2nsnc12)c3ccccc3)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P23 mock treatment 360.0 -409.0 -0.15 2120.0 1270.0 0.97 0.5862 0.5953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2027 P24 mock treatment 240.0 -529.0 -0.19 360.0 -491.0 -0.38 -0.3993 -0.948 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A01 compound treatment 480.0 -331.0 -0.12 3320.0 2420.0 1.86 1.2299 0.661 3029892 ChemDiv3_009505 CC1CCN(CC1)C(=O)CN(C)S(=O)(=O)c2cccc3nsnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A02 compound treatment 3280.0 2470.0 0.88 640.0 -261.0 -0.2 0.4774 0.5314 3029893 ChemDiv3_009506 Cc1cc(C)c2sc(nc2c1)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A03 compound treatment 320.0 -491.0 -0.17 4200.0 3300.0 2.53 1.6675 0.6569 3121157 ChemDiv3_009507 COc1ccc(OC)c(c1)C2N(Cc3ccc(C)cc3)CCCN2Cc4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A04 compound treatment 440.0 -371.0 -0.13 1680.0 779.0 0.6 0.3296 0.5384 3029896 ChemDiv3_009508 N=C/1N2C=CSC2=NC(=O)\C1=C/c3ccc(SC4CCCCC4)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A05 compound treatment 640.0 -171.0 -0.06 1080.0 179.0 0.14 0.0541 0.3603 3121158 ChemDiv3_009509 CC1CN(CC(C)O1)C(=O)CCn2c(=O)oc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A06 compound treatment 400.0 -411.0 -0.15 520.0 -381.0 -0.29 -0.3101 -0.9483 3121159 ChemDiv3_009510 O=C(CSc1c2CCCc2nc3ccccc13)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A07 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3029899 ChemDiv3_009511 CC(C)NC(=O)CCn1c(=O)sc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A08 compound treatment 400.0 -411.0 -0.15 600.0 -301.0 -0.23 -0.2667 -0.9753 3029968 ChemDiv3_009512 COc1ccc(cc1)n2c(Cc3cc(=O)[nH]c(=O)[nH]3)nnc2SCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A09 compound treatment 320.0 -491.0 -0.17 800.0 -101.0 -0.08 -0.1782 -0.9338 3029970 ChemDiv3_009513 CC(C1Sc2ccccc2N(Cc3ccc(F)cc3)C1=O)C(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A10 compound treatment 320.0 -491.0 -0.17 520.0 -381.0 -0.29 -0.3302 -0.9693 3029973 ChemDiv3_009514 CCc1ccc(cc1)n2c(nc3ccccc3c2=O)N(C)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A11 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3029974 ChemDiv3_009515 Cn1c(cc2c(=O)[nH]c3ccccc3c12)C(=O)N4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A12 compound treatment 280.0 -531.0 -0.19 240.0 -661.0 -0.51 -0.4922 -0.909 3029975 ChemDiv3_009516 CC1CCC(CC1)NS(=O)(=O)c2ccc3n(C)c(=O)c(=O)n(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A13 compound treatment 320.0 -491.0 -0.17 400.0 -501.0 -0.38 -0.3953 -0.9358 3121160 ChemDiv3_009517 CC1CCN(CCCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A14 compound treatment 1280.0 469.0 0.17 800.0 -101.0 -0.08 0.0626 0.3411 3029978 ChemDiv3_009518 CCCCN(C)S(=O)(=O)c1ccc2n(C)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A15 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3121161 ChemDiv3_009519 O=C(CSc1c2CCCCc2nc3ccccc13)NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A16 compound treatment 480.0 -331.0 -0.12 240.0 -661.0 -0.51 -0.4421 -0.8484 3029981 ChemDiv3_009520 COc1ccc(cc1)N(C)S(=O)(=O)c2ccc3n(C)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A17 compound treatment 240.0 -571.0 -0.2 240.0 -661.0 -0.51 -0.5023 -0.9189 3121162 ChemDiv3_009521 CC1CCCN(C1)c2c3CCCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A18 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3029984 ChemDiv3_009522 CN(C1CCCCC1)S(=O)(=O)c2ccc3n(C)cc(C(=O)NCCN4CCCC4)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A19 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3121163 ChemDiv3_009523 CC1(C)CC(=O)c2sc(Nc3nc4c(F)cccc4s3)nc2C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A20 compound treatment 360.0 -451.0 -0.16 320.0 -581.0 -0.45 -0.4287 -0.9043 3121164 ChemDiv3_009524 CCn1cc(C(=O)N2CCCCC2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A21 compound treatment 280.0 -531.0 -0.19 320.0 -581.0 -0.45 -0.4488 -0.9265 3029987 ChemDiv3_009525 Fc1ccc(Nc2nc3ccc(F)cc3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A22 compound treatment 640.0 -171.0 -0.06 360.0 -541.0 -0.42 -0.3368 -0.802 3121165 ChemDiv3_009526 CCN(CC)S(=O)(=O)c1ccc2n(CC=C)cc(C(=O)NC3CCCC3)c(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A23 mock treatment 400.0 -411.0 -0.15 400.0 -501.0 -0.38 -0.3753 -0.9119 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 A24 mock treatment 360.0 -451.0 -0.16 2600.0 1700.0 1.3 0.809 0.6157 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B01 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3029990 ChemDiv3_009527 Cc1ccc(cc1)S(=O)(=O)Cc2ccc(o2)C(=O)N3CCC4(CC3)OCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B02 compound treatment 520.0 -291.0 -0.1 280.0 -621.0 -0.48 -0.4103 -0.8408 3029992 ChemDiv3_009528 CC(C)NC(=O)c1cc(C)nn1c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B03 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3030151 ChemDiv3_009529 CCN(CC)C(=O)c1ccc(CS(=O)(=O)c2ccccc2C)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B04 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3030154 ChemDiv3_009530 CC1=C(C(=O)Nc2ccccc2Br)C3(CCCCC3)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B05 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3030157 ChemDiv3_009531 Clc1cccc(Cl)c1S(=O)(=O)Cc2ccc(o2)C(=O)N3CCN(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B06 compound treatment 320.0 -491.0 -0.17 320.0 -581.0 -0.45 -0.4388 -0.9159 3030158 ChemDiv3_009532 CCCN(CCC)C(=O)C1=C(C)C(=O)OC21CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B07 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3030161 ChemDiv3_009533 Cc1oc(nc1CN2CCC(CC2)C(=O)NCc3ccc(Cl)cc3)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B08 compound treatment 1240.0 429.0 0.15 320.0 -581.0 -0.45 -0.208 -0.4412 3030163 ChemDiv3_009534 COc1ccc(CCNc2cc(C)nc3c(c(C)nn23)c4ccc(OC)c(OC)c4)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B09 compound treatment 280.0 -531.0 -0.19 320.0 -581.0 -0.45 -0.4488 -0.9265 3121166 ChemDiv3_009535 Cc1oc(nc1CSCC(=O)NC2CCCC2)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B10 compound treatment 360.0 -451.0 -0.16 280.0 -621.0 -0.48 -0.4504 -0.8954 3030165 ChemDiv3_009536 Cc1c(sc2nc(cn12)c3ccccc3)C(=O)N4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B11 compound treatment 920.0 109.0 0.04 1480.0 579.0 0.44 0.3415 0.7656 3121167 ChemDiv3_009537 Cc1oc(nc1CSCC(=O)NC2CC2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B12 compound treatment 200.0 -611.0 -0.22 280.0 -621.0 -0.48 -0.4906 -0.9364 3030168 ChemDiv3_009538 Cc1cc2cc(CNC(=O)C3CCCCC3)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B13 compound treatment 560.0 -251.0 -0.09 280.0 -621.0 -0.48 -0.4003 -0.825 3121168 ChemDiv3_009539 Cc1oc(nc1CS(=O)CC(=O)NCc2ccccn2)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B14 compound treatment 400.0 -411.0 -0.15 240.0 -661.0 -0.51 -0.4621 -0.8749 3121169 ChemDiv3_009540 Cc1cc2cc(CNC(=O)Cc3cccc(C)c3)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B15 compound treatment 320.0 -491.0 -0.17 240.0 -661.0 -0.51 -0.4822 -0.8984 3030241 ChemDiv3_009541 COc1ccc(cc1OC)c2nc(CS(=O)CC(=O)NC(C)c3ccccc3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B16 compound treatment 240.0 -571.0 -0.2 360.0 -541.0 -0.42 -0.4371 -0.9455 3030245 ChemDiv3_009542 Cc1cc2cc(CNC(=O)C(C)(C)Oc3ccc(Cl)cc3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B17 compound treatment 440.0 -371.0 -0.13 400.0 -501.0 -0.38 -0.3652 -0.898 3030246 ChemDiv3_009543 Cc1oc(nc1CS(=O)(=O)CC(=O)NCc2ccc3OCOc3c2)c4ccccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B18 compound treatment 280.0 -531.0 -0.19 320.0 -581.0 -0.45 -0.4488 -0.9265 3030247 ChemDiv3_009544 Fc1ccc(cc1F)C(=O)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B19 compound treatment 520.0 -291.0 -0.1 320.0 -581.0 -0.45 -0.3886 -0.8484 3030251 ChemDiv3_009545 CCN1C(=O)c2ccccc2S(=O)c3ccc(cc13)C(=O)NCC(OC)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B20 compound treatment 400.0 -411.0 -0.15 1320.0 419.0 0.32 0.1242 0.3517 3030252 ChemDiv3_009546 O=C1N(Cc2ccc3[nH]c4CCCCc4c3c2)C(=O)c5ccccc15 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B21 compound treatment 400.0 -411.0 -0.15 3360.0 2460.0 1.89 1.2316 0.6505 3121348 ChemDiv3_009547 CN(C)CCNC(=O)c1ccc2c(c1)N(Cc3ccc(F)cc3)C(=O)c4ccccc4S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B22 compound treatment 360.0 -451.0 -0.16 280.0 -621.0 -0.48 -0.4504 -0.8954 3030257 ChemDiv3_009548 Cc1cc2cc(CNC(=S)Nc3ccccc3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B23 mock treatment 240.0 -571.0 -0.2 240.0 -661.0 -0.51 -0.5023 -0.9189 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 B24 mock treatment 200.0 -611.0 -0.22 840.0 -61.3 -0.05 -0.1866 -0.8409 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C01 compound treatment 160.0 -651.0 -0.23 320.0 -581.0 -0.45 -0.4789 -0.953 3121349 ChemDiv3_009549 O=C(C(Cc1ccccc1)NS(=O)(=O)c2cccc3nsnc23)N4CCC5(CC4)OCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C02 compound treatment 360.0 -451.0 -0.16 320.0 -581.0 -0.45 -0.4287 -0.9043 3030261 ChemDiv3_009550 COc1ccc(C)c2sc(nc12)N3CCN(CC3)c4nc5c(OC)ccc(C)c5s4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C03 compound treatment 360.0 -451.0 -0.16 280.0 -621.0 -0.48 -0.4504 -0.8954 3121350 ChemDiv3_009551 Cc1ccc(cc1)n2c(=O)n(Cc3ccccc3F)c4cc(ccc4c2=O)C(=O)NCc5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C04 compound treatment 280.0 -531.0 -0.19 3480.0 2580.0 1.98 1.2666 0.6369 3030646 ChemDiv3_009552 Cn1nc(c2ccc(Cl)cc2)c3cc(sc13)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C05 compound treatment 320.0 -491.0 -0.17 440.0 -461.0 -0.35 -0.3736 -0.9467 3121351 ChemDiv3_009553 CC(C)NC(=O)CCn1c(=O)oc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C06 compound treatment 320.0 -491.0 -0.17 320.0 -581.0 -0.45 -0.4388 -0.9159 3121352 ChemDiv3_009554 Clc1ccc2nc3CCCCc3c(SCC(=O)NCCN4CCOCC4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C07 compound treatment 520.0 -291.0 -0.1 360.0 -541.0 -0.42 -0.3669 -0.8568 3030650 ChemDiv3_009555 O=C(CCn1c(=O)sc2ccccc12)NCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C08 compound treatment 1120.0 309.0 0.11 320.0 -581.0 -0.45 -0.2381 -0.5182 3121353 ChemDiv3_009556 CC(C)Sc1nnc(Cc2cc(=O)[nH]c(=O)[nH]2)n1c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C09 compound treatment 480.0 -331.0 -0.12 400.0 -501.0 -0.38 -0.3552 -0.8828 3121354 ChemDiv3_009557 CC(C1Sc2ccccc2N(Cc3cc(C)ccc3C)C1=O)C(=O)NCCc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C10 compound treatment 320.0 -491.0 -0.17 400.0 -501.0 -0.38 -0.3953 -0.9358 3030655 ChemDiv3_009558 CCc1ccc(cc1)n2c(nc3ccccc3c2=O)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C11 compound treatment 320.0 -491.0 -0.17 320.0 -581.0 -0.45 -0.4388 -0.9159 3030656 ChemDiv3_009559 Cn1c(cc2c(=O)[nH]c3ccccc3c12)C(=O)N4CCN(CC4)c5ccccc5F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C12 compound treatment 360.0 -451.0 -0.16 440.0 -461.0 -0.35 -0.3636 -0.9356 3121355 ChemDiv3_009560 CC1Cc2ccccc2N1S(=O)(=O)c3ccc4n(C)c(=O)c(=O)n(C)c4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C13 compound treatment 360.0 -451.0 -0.16 360.0 -541.0 -0.42 -0.407 -0.914 3121356 ChemDiv3_009561 Cn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C14 compound treatment 280.0 -531.0 -0.19 280.0 -621.0 -0.48 -0.4705 -0.9175 3030662 ChemDiv3_009562 CC1CCC(CC1)NS(=O)(=O)c2ccc3n(C)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C15 compound treatment 240.0 -571.0 -0.2 600.0 -301.0 -0.23 -0.3068 -0.9978 3121357 ChemDiv3_009563 CCC(C)NC(=O)CSc1c2CCCCc2nc3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C16 compound treatment 280.0 -531.0 -0.19 400.0 -501.0 -0.38 -0.4054 -0.946 3121358 ChemDiv3_009564 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NCCN3CCC(Cc4ccccc4)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C17 compound treatment 240.0 -571.0 -0.2 320.0 -581.0 -0.45 -0.4588 -0.9362 3030711 ChemDiv3_009565 CCc1ccc(Nc2c3CCCCc3nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C18 compound treatment 400.0 -411.0 -0.15 240.0 -661.0 -0.51 -0.4621 -0.8749 3121359 ChemDiv3_009566 CC1CCN(CC1)S(=O)(=O)c2ccc3n(C)cc(C(=O)N(C)Cc4ccccc4)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C19 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3030714 ChemDiv3_009567 Fc1cccc2sc(NCc3ccccc3)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C20 compound treatment 160.0 -651.0 -0.23 320.0 -581.0 -0.45 -0.4789 -0.953 3121360 ChemDiv3_009568 CCn1cc(C(=O)NCc2ccccc2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C21 compound treatment 280.0 -531.0 -0.19 360.0 -541.0 -0.42 -0.4271 -0.936 3030717 ChemDiv3_009569 Fc1ccc2nc(Nc3nnc(o3)c4ccco4)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C22 compound treatment 280.0 -531.0 -0.19 280.0 -621.0 -0.48 -0.4705 -0.9175 3121361 ChemDiv3_009570 CCN(CC)S(=O)(=O)c1ccc2n(CC=C)cc(C(=O)NCCN3CCCCCC3)c(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C23 mock treatment 280.0 -531.0 -0.19 280.0 -621.0 -0.48 -0.4705 -0.9175 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 C24 mock treatment 360.0 -451.0 -0.16 360.0 -541.0 -0.42 -0.407 -0.914 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D01 compound treatment 280.0 -531.0 -0.19 400.0 -501.0 -0.38 -0.4054 -0.946 3030721 ChemDiv3_009571 CC(C)CCNC(=O)c1ccc(CS(=O)(=O)c2ccc(Br)cc2)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D02 compound treatment 360.0 -451.0 -0.16 3320.0 2420.0 1.86 1.1998 0.6438 3121362 ChemDiv3_009572 CCCNC(=O)c1cc(C)nn1c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D03 compound treatment 280.0 -531.0 -0.19 400.0 -501.0 -0.38 -0.4054 -0.946 3030724 ChemDiv3_009573 Cc1ccccc1S(=O)(=O)Cc2ccc(o2)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D04 compound treatment 360.0 -451.0 -0.16 480.0 -421.0 -0.32 -0.3419 -0.9474 3121363 ChemDiv3_009574 CC1=C(C(=O)NCc2ccco2)C3(CCCCC3)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D05 compound treatment 280.0 -531.0 -0.19 320.0 -581.0 -0.45 -0.4488 -0.9265 3121364 ChemDiv3_009575 Clc1cccc(Cl)c1S(=O)(=O)Cc2ccc(o2)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D06 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3029682 ChemDiv3_009576 CC1=C(C(=O)N2CCCCC2)C3(CCCCC3)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D07 compound treatment 560.0 -251.0 -0.09 280.0 -621.0 -0.48 -0.4003 -0.825 3121365 ChemDiv3_009577 Cc1oc(nc1CN2CCC(CC2)C(=O)NCCCN3CCCC3)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D08 compound treatment 400.0 -411.0 -0.15 480.0 -421.0 -0.32 -0.3318 -0.9353 3121366 ChemDiv3_009578 COc1ccc(cc1OC)c2c(C)nn3c(cc(C)nc23)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D09 compound treatment 280.0 -531.0 -0.19 280.0 -621.0 -0.48 -0.4705 -0.9175 3029686 ChemDiv3_009579 CSc1ccc(cc1)c2nc(CSCC(=O)N3CCCC3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D10 compound treatment 240.0 -571.0 -0.2 240.0 -661.0 -0.51 -0.5023 -0.9189 3029687 ChemDiv3_009580 CNC(=O)c1sc2nc(cn2c1C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D11 compound treatment 360.0 -451.0 -0.16 520.0 -381.0 -0.29 -0.3202 -0.9597 3121367 ChemDiv3_009581 Cc1oc(nc1CSCC(=O)N2CCC3(CC2)OCCO3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D12 compound treatment 320.0 -491.0 -0.17 480.0 -421.0 -0.32 -0.3519 -0.9579 3121368 ChemDiv3_009582 Cc1cc2cc(CNC(=O)C3(CC4CC5CC(C4)C3)C5)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D13 compound treatment 200.0 -611.0 -0.22 480.0 -421.0 -0.32 -0.382 -0.9811 3029691 ChemDiv3_009583 Cc1oc(nc1CS(=O)CC(=O)NC2CCCCCC2)c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D14 compound treatment 240.0 -571.0 -0.2 320.0 -581.0 -0.45 -0.4588 -0.9362 3121369 ChemDiv3_009584 Cc1cc2cc(CNC(=O)Cc3cccc4ccccc34)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D15 compound treatment 440.0 -371.0 -0.13 320.0 -581.0 -0.45 -0.4087 -0.8783 3121370 ChemDiv3_009585 CN(Cc1ccccc1)C(=O)CS(=O)Cc2nc(oc2C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D16 compound treatment 320.0 -491.0 -0.17 480.0 -421.0 -0.32 -0.3519 -0.9579 3029749 ChemDiv3_009586 Cc1cc2cc(CNC(=O)COc3ccc4ccccc4c3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D17 compound treatment 360.0 -451.0 -0.16 320.0 -581.0 -0.45 -0.4287 -0.9043 3121371 ChemDiv3_009587 COC(CNC(=O)c1ccc2S(=O)c3ccccc3C(=O)N(Cc4ccccc4F)c2c1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D18 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3029751 ChemDiv3_009588 FC(F)(F)c1ccc(cc1)C(=O)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D19 compound treatment 240.0 -571.0 -0.2 360.0 -541.0 -0.42 -0.4371 -0.9455 3121372 ChemDiv3_009589 CCN1C(=O)c2ccccc2S(=O)(=O)c3ccc(cc13)C(=O)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D20 compound treatment 320.0 -491.0 -0.17 240.0 -661.0 -0.51 -0.4822 -0.8984 3029753 ChemDiv3_009590 Cc1cc2cc(CNS(=O)(=O)c3ccccc3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D21 compound treatment 360.0 -451.0 -0.16 1440.0 539.0 0.41 0.1793 0.4042 3121373 ChemDiv3_009591 CN(C)CCNC(=O)c1ccc2c(c1)N(Cc3cc(C)ccc3C)C(=O)c4ccccc4S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D22 compound treatment 320.0 -491.0 -0.17 320.0 -581.0 -0.45 -0.4388 -0.9159 3029756 ChemDiv3_009592 CNC(=S)NCc1ccc2[nH]c3CCCCc3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D23 mock treatment 400.0 -411.0 -0.15 280.0 -621.0 -0.48 -0.4404 -0.883 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 D24 mock treatment 320.0 -491.0 -0.17 400.0 -501.0 -0.38 -0.3953 -0.9358 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E01 compound treatment 1680.0 869.0 0.31 4040.0 3140.0 2.41 1.9218 0.7911 3121547 ChemDiv3_009593 CC1CC(C)CN(C1)C(=O)C(Cc2ccccc2)NS(=O)(=O)c3cccc4nsnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E02 compound treatment 1920.0 1110.0 0.39 1680.0 779.0 0.6 0.7009 0.9794 3029759 ChemDiv3_009594 C1Oc2cc3nc(sc3cc2O1)N4CCc5ccccc5C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E03 compound treatment 880.0 68.8 0.02 760.0 -141.0 -0.11 -0.0594 -0.5347 3121548 ChemDiv3_009595 Cc1cc(N)nn1C(=O)Cn2c(=O)n(CC=C)c(=O)c3ccc(cc23)C(=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E04 compound treatment 2840.0 2030.0 0.72 1640.0 739.0 0.57 0.9099 0.993 3029762 ChemDiv3_009596 CCCCN(CC)C(=O)c1cc2c(nn(C)c2s1)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E05 compound treatment 1600.0 789.0 0.28 840.0 -61.3 -0.05 0.1646 0.5801 3121549 ChemDiv3_009597 CC1CC(CC(C)(C)C1)NC(=O)CCn2c(=O)oc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E06 compound treatment 1640.0 829.0 0.29 520.0 -381.0 -0.29 9.0E-4 0.0022 3029765 ChemDiv3_009598 Clc1ccc2nc3CCCCc3c(SCC(=O)NCc4ccccn4)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E07 compound treatment 760.0 -51.3 -0.02 2640.0 1740.0 1.33 0.931 0.6974 3029822 ChemDiv3_009599 O=C(CCn1c(=O)sc2ccccc12)NCCCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E08 compound treatment 880.0 68.8 0.02 440.0 -461.0 -0.35 -0.2331 -0.6568 3121550 ChemDiv3_009600 Fc1ccc(cc1)n2c(Cc3cc(=O)[nH]c(=O)[nH]3)nnc2SCc4c(F)cccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E09 compound treatment 560.0 -251.0 -0.09 520.0 -381.0 -0.29 -0.27 -0.8824 3029825 ChemDiv3_009601 CC(C1Sc2ccccc2N(Cc3cc(C)ccc3C)C1=O)C(=O)NCc4ccc5OCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E10 compound treatment 1040.0 229.0 0.08 840.0 -61.3 -0.05 0.0241 0.2573 3121551 ChemDiv3_009602 CC1CN(CCN1c2cccc(C)c2)c3nc4ccccc4c(=O)n3Cc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E11 compound treatment 880.0 68.8 0.02 400.0 -501.0 -0.38 -0.2549 -0.661 3121552 ChemDiv3_009603 CCc1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E12 compound treatment 1280.0 469.0 0.17 680.0 -221.0 -0.17 -0.0025 -0.0106 3029830 ChemDiv3_009604 CN(c1cccc(C)c1)S(=O)(=O)c2ccc3n(C)c(=O)c(=O)n(C)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E13 compound treatment 640.0 -171.0 -0.06 360.0 -541.0 -0.42 -0.3368 -0.802 3121553 ChemDiv3_009605 Cn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCC4(CCCC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E14 compound treatment 400.0 -411.0 -0.15 920.0 18.8 0.01 -0.093 -0.6343 3029832 ChemDiv3_009606 CCN(Cc1ccccc1)S(=O)(=O)c2ccc3n(C)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E15 compound treatment 840.0 28.8 0.01 1840.0 939.0 0.72 0.5168 0.717 3121554 ChemDiv3_009607 CN(C1CCCCC1)C(=O)CSc2c3CCCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E16 compound treatment 520.0 -291.0 -0.1 360.0 -541.0 -0.42 -0.3669 -0.8568 3029836 ChemDiv3_009608 CN(C)S(=O)(=O)c1ccc2n(C)cc(C(=O)NCc3ccccc3)c(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E17 compound treatment 1440.0 629.0 0.22 1520.0 619.0 0.48 0.4936 0.9406 3121555 ChemDiv3_009609 CCc1ccc(cc1)C2CC(=O)N3CN(CSC3=C2C#N)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E18 compound treatment 600.0 -211.0 -0.07 5680.0 4780.0 3.67 2.5412 0.6925 3121556 ChemDiv3_009610 CC(C)CCNC(=O)c1cn(C)c2ccc(cc2c1=O)S(=O)(=O)N3CCC(C)CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E19 compound treatment 1000.0 189.0 0.07 1520.0 619.0 0.48 0.3832 0.7989 3029840 ChemDiv3_009611 CC(C)c1ccc2nc(Nc3nc4ccc(NC(=O)C)cc4s3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E20 compound treatment 440.0 -371.0 -0.13 640.0 -261.0 -0.2 -0.2349 -0.9792 3121557 ChemDiv3_009612 CCn1cc(C(=O)NCC(OC)OC)c(=O)c2cc(ccc12)S(=O)(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E21 compound treatment 560.0 -251.0 -0.09 1600.0 699.0 0.54 0.3163 0.5816 3029900 ChemDiv3_009613 C1Oc2cc3nc(Nc4nccs4)sc3cc2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E22 compound treatment 520.0 -291.0 -0.1 6760.0 5860.0 4.5 3.1074 0.6907 3121558 ChemDiv3_009614 O=C(N1CCN(CC1)c2ccccc2)c3ccc(CS(=O)c4ccccc4)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E23 mock treatment 680.0 -131.0 -0.05 1160.0 259.0 0.2 0.1075 0.5271 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 E24 mock treatment 840.0 28.8 0.01 2200.0 1300.0 1.0 0.7122 0.7143 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F01 compound treatment 1160.0 349.0 0.12 1240.0 339.0 0.26 0.2714 0.9423 3121559 ChemDiv3_009615 CC(CCc1ccccc1)NC(=O)c2ccc(CS(=O)(=O)c3ccc(Br)cc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F02 compound treatment 1520.0 709.0 0.25 1400.0 499.0 0.38 0.4485 0.9792 3029905 ChemDiv3_009616 COC(CNC(=O)c1cc(C)nn1c2ccccc2)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F03 compound treatment 1000.0 189.0 0.07 1560.0 659.0 0.51 0.405 0.7938 3121560 ChemDiv3_009617 CC(NC(=O)c1ccc(CS(=O)(=O)c2ccccc2C)o1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F04 compound treatment 2800.0 1990.0 0.71 1000.0 98.8 0.08 0.5525 0.7786 3029908 ChemDiv3_009618 CC(C)NC(=O)C1=C(C)C(=O)OC21CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F05 compound treatment 760.0 -51.3 -0.02 2800.0 1900.0 1.46 1.0179 0.6982 3121561 ChemDiv3_009619 COc1ccc(cc1OC)c2nc(CN3CCC(CC3)C(=O)NC(C)C)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F06 compound treatment 720.0 -91.3 -0.03 1080.0 179.0 0.14 0.0741 0.5259 3029911 ChemDiv3_009620 CC1=C(C(=O)N(CC2CCCO2)CC3CCC=CC3)C4(CCCCC4)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F07 compound treatment 1040.0 229.0 0.08 1000.0 98.8 0.08 0.111 0.9994 3121562 ChemDiv3_009621 COc1ccc(CCNC(=O)C2CCN(Cc3nc(oc3C)c4ccccc4F)CC2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F08 compound treatment 9080.0 8270.0 2.93 600.0 -301.0 -0.23 1.9106 0.6493 3121563 ChemDiv3_009622 Cc1nn2c(cc(C)nc2c1c3ccc(Cl)cc3)N4CCC(CC4)C(=O)Nc5cccnc5Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F09 compound treatment 640.0 -171.0 -0.06 1840.0 939.0 0.72 0.4667 0.6452 3029916 ChemDiv3_009623 CCc1ccc(cc1)c2nc(CSCC(=O)N3CCc4ccccc34)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F10 compound treatment 1160.0 349.0 0.12 2960.0 2060.0 1.58 1.2051 0.7601 3121564 ChemDiv3_009624 CN(C1CCCCC1)C(=O)c2sc3nc(cn3c2C)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F11 compound treatment 520.0 -291.0 -0.1 1640.0 739.0 0.57 0.328 0.5689 3029919 ChemDiv3_009625 CC1CCCCC1N(C)C2CCN(CCNC(=O)/C=C/c3ccccc3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F12 compound treatment 920.0 109.0 0.04 1120.0 219.0 0.17 0.146 0.8475 3121565 ChemDiv3_009626 CCOc1ccccc1C(=O)NCc2ccc3[nH]c(C)cc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F13 compound treatment 1240.0 429.0 0.15 2920.0 2020.0 1.55 1.2034 0.7728 3121566 ChemDiv3_009627 Cc1oc(nc1CS(=O)CC(=O)NCc2cccs2)c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F14 compound treatment 560.0 -251.0 -0.09 3000.0 2100.0 1.61 1.0763 0.667 3030556 ChemDiv3_009628 Cc1cc2cc(CNC(=O)C3CCCCC3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F15 compound treatment 1400.0 589.0 0.21 1480.0 579.0 0.44 0.4619 0.9407 3121567 ChemDiv3_009629 CCN1CCN(CC1)C(=O)CS(=O)Cc2nc(oc2C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F16 compound treatment 640.0 -171.0 -0.06 6600.0 5700.0 4.38 3.0507 0.6972 3121568 ChemDiv3_009630 Cc1cc2cc(CNC(=O)Cc3cccc4ccccc34)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F17 compound treatment 680.0 -131.0 -0.05 1000.0 98.8 0.08 0.0207 0.2325 3030560 ChemDiv3_009631 Fc1ccc(CN2C(=O)c3ccccc3S(=O)c4ccc(cc24)C(=O)NCCc5ccccc5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F18 compound treatment 1760.0 949.0 0.34 1880.0 979.0 0.75 0.7693 0.9344 3121569 ChemDiv3_009632 COc1cc(/C=C\C(=O)NCc2ccc3[nH]c4CCCCc4c3c2)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F19 compound treatment 880.0 68.8 0.02 1360.0 459.0 0.35 0.2663 0.7543 3030600 ChemDiv3_009633 CCN1C(=O)c2ccccc2S(=O)(=O)c3ccc(cc13)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F20 compound treatment 2600.0 1790.0 0.63 1960.0 1060.0 0.81 1.0234 0.9925 3121570 ChemDiv3_009634 O=S(=O)(NCc1ccc2[nH]c3CCCCc3c2c1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F21 compound treatment 600.0 -211.0 -0.07 1080.0 179.0 0.14 0.044 0.2817 3121571 ChemDiv3_009635 O=C(N1CCCCC1)c2ccc3c(c2)N(Cc4ccccc4)C(=O)c5ccccc5S3(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F22 compound treatment 6880.0 6070.0 2.15 1280.0 379.0 0.29 1.7279 0.7954 3030607 ChemDiv3_009636 S=C(NCc1ccc2[nH]c3CCCCc3c2c1)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F23 mock treatment 840.0 28.8 0.01 1720.0 819.0 0.63 0.4517 0.7185 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 F24 mock treatment 2760.0 1950.0 0.69 1760.0 859.0 0.66 0.955 0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G01 compound treatment 240.0 -571.0 -0.2 600.0 -301.0 -0.23 -0.3068 -0.9978 3121572 ChemDiv3_009637 O=C(NCc1cccs1)C(NS(=O)(=O)c2cccc3nsnc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G02 compound treatment 1040.0 229.0 0.08 2280.0 1380.0 1.06 0.8058 0.7591 3030611 ChemDiv3_009638 C1COc2cc3sc(nc3cc2O1)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G03 compound treatment 1720.0 909.0 0.32 1440.0 539.0 0.41 0.5204 0.9924 3121747 ChemDiv3_009639 C=CCn1c(=O)n(Cc2ccccc2C#N)c3cc(ccc3c1=O)C(=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G04 compound treatment 1280.0 469.0 0.17 3840.0 2940.0 2.26 1.7129 0.7572 3030665 ChemDiv3_009640 CN(C(=O)c1cc2c(nn(C)c2s1)c3ccc(Cl)cc3)c4cc(Cl)ccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G05 compound treatment 440.0 -371.0 -0.13 2440.0 1540.0 1.18 0.7422 0.6244 1628704 ChemDiv3_009641 O=C(CCn1c(=O)oc2ccccc12)NCCC3=CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G06 compound treatment 1280.0 469.0 0.17 640.0 -261.0 -0.2 -0.0242 -0.093 3121748 ChemDiv3_009642 CCN(CC)C(=O)CSc1c2CCCCc2nc3ccc(Cl)cc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G07 compound treatment 480.0 -331.0 -0.12 440.0 -461.0 -0.35 -0.3335 -0.8938 3030670 ChemDiv3_009643 CCN(C(=O)CCn1c(=O)sc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G08 compound treatment 760.0 -51.3 -0.02 720.0 -181.0 -0.14 -0.1112 -0.7928 3121749 ChemDiv3_009644 Clc1ccc(cc1)n2c(Cc3cc(=O)[nH]c(=O)[nH]3)nnc2SCC(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G09 compound treatment 1280.0 469.0 0.17 640.0 -261.0 -0.2 -0.0242 -0.093 3121750 ChemDiv3_009645 CCC(Sc1nc2sc(C(=O)OC)c(C)c2c(=O)n1N)C(=O)Nc3cccc(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G10 compound treatment 1440.0 629.0 0.22 1120.0 219.0 0.17 0.2765 0.9902 3030674 ChemDiv3_009646 CCOC(=O)c1cn(CC(=O)Nc2ccccc2)nn1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G11 compound treatment 640.0 -171.0 -0.06 440.0 -461.0 -0.35 -0.2934 -0.8165 3121751 ChemDiv3_009647 Cn1c(cc2c(=O)[nH]c3ccccc3c12)C(=O)NCCCN4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G12 compound treatment 680.0 -131.0 -0.05 840.0 -61.3 -0.05 -0.0662 -1.0 3030677 ChemDiv3_009648 CCc1ccc(NC(=O)CN(c2ccc3OCOc3c2)S(=O)(=O)c4c(C)noc4C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G13 compound treatment 3800.0 2990.0 1.06 440.0 -461.0 -0.35 0.4993 0.4467 3121752 ChemDiv3_009649 CN(CCNC(=O)c1cc2c(=O)n(C)c3ccccc3c2s1)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G14 compound treatment 1400.0 589.0 0.21 1920.0 1020.0 0.78 0.7007 0.8656 1173384 ChemDiv3_009650 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G15 compound treatment 360.0 -451.0 -0.16 480.0 -421.0 -0.32 -0.3419 -0.9474 3121753 ChemDiv3_009651 CC1CCN(CC1)C(=O)CSc2c3CCCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G16 compound treatment 3320.0 2510.0 0.89 1680.0 779.0 0.6 1.0521 0.9813 3121754 ChemDiv3_009652 CCCN(CCC)C(=O)c1cn(C)c2ccc(cc2c1=O)S(=O)(=O)N(CC)CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G17 compound treatment 360.0 -451.0 -0.16 880.0 -21.3 -0.02 -0.1247 -0.7752 3030731 ChemDiv3_009653 CN1CSC2=C(C#N)C(CC(=O)N2C1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G18 compound treatment 1120.0 309.0 0.11 1120.0 219.0 0.17 0.1962 0.9786 3121755 ChemDiv3_009654 CCn1cc(C(=O)N2CCCC2)c(=O)c3cc(ccc13)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G19 compound treatment 1800.0 989.0 0.35 1600.0 699.0 0.54 0.6273 0.9788 3030735 ChemDiv3_009655 CC(C)c1ccc2nc(Nc3nc4ccc(cc4s3)S(=O)(=O)C)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G20 compound treatment 1280.0 469.0 0.17 440.0 -461.0 -0.35 -0.1328 -0.3395 3121756 ChemDiv3_009656 CCn1cc(C(=O)NC2CCCC2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G21 compound treatment 320.0 -491.0 -0.17 600.0 -301.0 -0.23 -0.2868 -0.9903 3030738 ChemDiv3_009657 COc1cccc2sc(nc12)N3CCc4ccccc4C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G22 compound treatment 1920.0 1110.0 0.39 1400.0 499.0 0.38 0.5489 0.9999 3121757 ChemDiv3_009658 O=C(NCc1ccccc1)c2ccc(CS(=O)c3ccccc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G23 mock treatment 1760.0 949.0 0.34 1240.0 339.0 0.26 0.4219 0.9919 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 G24 mock treatment 360.0 -451.0 -0.16 1080.0 179.0 0.14 -0.0162 -0.0766 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H01 compound treatment 480.0 -331.0 -0.12 640.0 -261.0 -0.2 -0.2249 -0.9676 3121758 ChemDiv3_009659 Brc1ccc(cc1)S(=O)(=O)Cc2ccc(o2)C(=O)NCCN3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H02 compound treatment 480.0 -331.0 -0.12 640.0 -261.0 -0.2 -0.2249 -0.9676 3029701 ChemDiv3_009660 CC(C)c1ccc(NC(=O)c2cc(C)nn2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H03 compound treatment 480.0 -331.0 -0.12 760.0 -141.0 -0.11 -0.1598 -0.9992 3121759 ChemDiv3_009661 COc1ccccc1S(=O)(=O)Cc2ccc(o2)C(=O)NC3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H04 compound treatment 1280.0 469.0 0.17 640.0 -261.0 -0.2 -0.0242 -0.093 3029705 ChemDiv3_009662 CCCNC(=O)C1=C(C)C(=O)OC21CCCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H05 compound treatment 5600.0 4790.0 1.7 560.0 -341.0 -0.26 1.016 0.5911 3121760 ChemDiv3_009663 Cc1oc(nc1CN2CCC(CC2)C(=O)NC3CCCC3)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H06 compound treatment 520.0 -291.0 -0.1 720.0 -181.0 -0.14 -0.1715 -0.9893 3029709 ChemDiv3_009664 COC(CNc1cc(C)nc2c(c(C)nn12)c3ccccc3OC)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H07 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3121761 ChemDiv3_009665 Cc1oc(nc1CN2CCCC(C2)C(=O)NCCc3ccc(C)cc3)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H08 compound treatment 400.0 -411.0 -0.15 1200.0 299.0 0.23 0.059 0.2171 3029714 ChemDiv3_009666 Cc1nn2c(cc(C)nc2c1c3ccc(Cl)cc3)N4CCC(CC4)C(=O)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H09 compound treatment 480.0 -331.0 -0.12 640.0 -261.0 -0.2 -0.2249 -0.9676 3029766 ChemDiv3_009667 CCc1ccc(cc1)c2nc(CSCC(=O)N3CCc4ccccc4C3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H10 compound treatment 560.0 -251.0 -0.09 1640.0 739.0 0.57 0.338 0.5888 3121762 ChemDiv3_009668 CC1CCN(CC1)C(=O)c2sc3nc(cn3c2C)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H11 compound treatment 2400.0 1590.0 0.56 4400.0 3500.0 2.69 2.2979 0.8372 3121763 ChemDiv3_009669 CC1CCCCC1N(C)C2CCN(CCCNC(=O)/C=C/c3cccc(c3)C(F)(F)F)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H12 compound treatment 2080.0 1270.0 0.45 600.0 -301.0 -0.23 0.1547 0.3058 3029773 ChemDiv3_009670 CCOc1cc(cc(OCC)c1OCC)C(=O)NCc2ccc3[nH]c(C)cc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H13 compound treatment 840.0 28.8 0.01 680.0 -221.0 -0.17 -0.1129 -0.6635 3121764 ChemDiv3_009671 Cc1oc(nc1CS(=O)CC(=O)NCCC2=CCCCC2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H14 compound treatment 440.0 -371.0 -0.13 640.0 -261.0 -0.2 -0.2349 -0.9792 3029778 ChemDiv3_009672 Cc1cc2cc(CNC(=O)CCC3CCCCC3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H15 compound treatment 440.0 -371.0 -0.13 480.0 -421.0 -0.32 -0.3218 -0.9216 3121765 ChemDiv3_009673 CCOC(=O)N1CCC(CC1)NC(=O)CS(=O)(=O)Cc2nc(oc2C)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H16 compound treatment 640.0 -171.0 -0.06 600.0 -301.0 -0.23 -0.2065 -0.8636 3029780 ChemDiv3_009674 O=C(CCC1CCCC1)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H17 compound treatment 2240.0 1430.0 0.51 440.0 -461.0 -0.35 0.108 0.1747 3121766 ChemDiv3_009675 Cc1ccc(C)c(CN2C(=O)c3ccccc3S(=O)c4ccc(cc24)C(=O)N5CCCCCC5)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H18 compound treatment 880.0 68.8 0.02 480.0 -421.0 -0.32 -0.2114 -0.6519 3029842 ChemDiv3_009676 Clc1ccc(OCC(=O)NCc2ccc3[nH]c4CCCCc4c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H19 compound treatment 400.0 -411.0 -0.15 560.0 -341.0 -0.26 -0.2884 -0.9618 3029843 ChemDiv3_009677 CCN1C(=O)c2ccccc2S(=O)(=O)c3ccc(cc13)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H20 compound treatment 400.0 -411.0 -0.15 680.0 -221.0 -0.17 -0.2233 -0.9971 3121767 ChemDiv3_009678 Cc1cc2cc(CNC(=S)NCc3ccccc3)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H21 compound treatment 1600.0 789.0 0.28 800.0 -101.0 -0.08 0.1429 0.492 3121768 ChemDiv3_009679 Fc1ccc(CN2C(=O)CS(=O)c3ccc(cc23)C(=O)Nc4ccccc4Br)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H22 compound treatment 440.0 -371.0 -0.13 800.0 -101.0 -0.08 -0.1481 -0.9684 3029851 ChemDiv3_009680 Cc1cc2cc(CNC(=O)Nc3cccc(Cl)c3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H23 mock treatment 400.0 -411.0 -0.15 1640.0 739.0 0.57 0.2979 0.5087 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 H24 mock treatment 440.0 -371.0 -0.13 400.0 -501.0 -0.38 -0.3652 -0.898 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I01 compound treatment 360.0 -451.0 -0.16 280.0 -621.0 -0.48 -0.4504 -0.8954 3121769 ChemDiv3_009681 O=C(NCc1ccccc1)C(Cc2ccccc2)NS(=O)(=O)c3cccc4nsnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I02 compound treatment 2360.0 1550.0 0.55 320.0 -581.0 -0.45 0.073 0.1031 3029855 ChemDiv3_009682 COc1ccc(cc1Cl)n2nc(C(=O)Nc3cc(C)on3)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I03 compound treatment 280.0 -531.0 -0.19 280.0 -621.0 -0.48 -0.4705 -0.9175 3121770 ChemDiv3_009683 Cc1ccccc1Cn2c(=O)n(Cc3ccco3)c(=O)c4ccc(cc24)C(=O)NC5CCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I04 compound treatment 360.0 -451.0 -0.16 200.0 -701.0 -0.54 -0.4939 -0.8793 3121771 ChemDiv3_009684 CCN(C(=O)c1cc2c(nn(C)c2s1)c3ccc(Cl)cc3)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I05 compound treatment 1000.0 189.0 0.07 440.0 -461.0 -0.35 -0.203 -0.5634 3029925 ChemDiv3_009685 COc1ccc(CCNC(=O)CCn2c(=O)oc3ccccc23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I06 compound treatment 440.0 -371.0 -0.13 320.0 -581.0 -0.45 -0.4087 -0.8783 3121772 ChemDiv3_009686 Cc1cccc(CCNC(=O)CSc2c3CCCCc3nc4ccc(Cl)cc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I07 compound treatment 280.0 -531.0 -0.19 480.0 -421.0 -0.32 -0.3619 -0.967 3029930 ChemDiv3_009687 CCc1ccccc1NC(=O)CCn2c(=O)sc3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I08 compound treatment 360.0 -451.0 -0.16 320.0 -581.0 -0.45 -0.4287 -0.9043 3121957 ChemDiv3_009688 O=C(N(CN1CCCC1=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I09 compound treatment 640.0 -171.0 -0.06 520.0 -381.0 -0.29 -0.2499 -0.8361 3029932 ChemDiv3_009689 COC(=O)c1sc2nc(SCC(=O)N(C)c3ccccc3)n(N)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I10 compound treatment 640.0 -171.0 -0.06 320.0 -581.0 -0.45 -0.3585 -0.796 3121958 ChemDiv3_009690 CC1Cc2ccccc2N1C(=O)C3CCN(CC3)S(=O)(=O)c4c(C)noc4/C=C/c5ccco5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I11 compound treatment 1080.0 269.0 0.1 1480.0 579.0 0.44 0.3816 0.8397 3121959 ChemDiv3_009691 COc1ccc(Br)cc1CNC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I12 compound treatment 360.0 -451.0 -0.16 5640.0 4740.0 3.64 2.4593 0.6753 3029937 ChemDiv3_009692 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N(CC=C)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I13 compound treatment 1000.0 189.0 0.07 1520.0 619.0 0.48 0.3832 0.7989 3121960 ChemDiv3_009693 Cc1cccc(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I14 compound treatment 5120.0 4310.0 1.53 2240.0 1340.0 1.03 1.8076 0.9814 3029940 ChemDiv3_009694 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N3CC(=O)N(CCc4ccccc4)C(=O)C3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I15 compound treatment 360.0 -451.0 -0.16 280.0 -621.0 -0.48 -0.4504 -0.8954 3031103 ChemDiv3_009695 O=C(CSc1c2CCCCc2nc3ccccc13)N4CCCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I16 compound treatment 520.0 -291.0 -0.1 720.0 -181.0 -0.14 -0.1715 -0.9893 3031104 ChemDiv3_009696 Cn1cc(C(=O)N2CCCC2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I17 compound treatment 560.0 -251.0 -0.09 4280.0 3380.0 2.59 1.7712 0.6824 3031105 ChemDiv3_009697 O=C1CC(C(=C2SCN(Cc3ccccc3)CN12)C#N)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I18 compound treatment 5960.0 5150.0 1.83 640.0 -261.0 -0.2 1.1497 0.6257 3031106 ChemDiv3_009698 CCn1cc(C(=O)N2CCN(C)CC2)c(=O)c3cc(ccc13)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I19 compound treatment 480.0 -331.0 -0.12 320.0 -581.0 -0.45 -0.3986 -0.8639 3031107 ChemDiv3_009699 CCOC(=O)c1sc(Nc2nc3ccc(OC)cc3s2)cc1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I20 compound treatment 840.0 28.8 0.01 720.0 -181.0 -0.14 -0.0912 -0.6535 3031108 ChemDiv3_009700 CCn1cc(C(=O)NCCC(C)C)c(=O)c2cc(ccc12)S(=O)(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I21 compound treatment 320.0 -491.0 -0.17 360.0 -541.0 -0.42 -0.417 -0.9256 3031109 ChemDiv3_009701 COc1cccc2sc(nc12)N(C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I22 compound treatment 320.0 -491.0 -0.17 480.0 -421.0 -0.32 -0.3519 -0.9579 3121961 ChemDiv3_009702 COC(CNC(=O)c1ccc(CS(=O)c2ccccc2)o1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I23 mock treatment 280.0 -531.0 -0.19 560.0 -341.0 -0.26 -0.3185 -0.9869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 I24 mock treatment 720.0 -91.3 -0.03 320.0 -581.0 -0.45 -0.3384 -0.7564 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J01 compound treatment 280.0 -531.0 -0.19 240.0 -661.0 -0.51 -0.4922 -0.909 3121962 ChemDiv3_009703 COc1ccc(cc1)S(=O)(=O)Cc2ccc(o2)C(=O)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J02 compound treatment 200.0 -611.0 -0.22 320.0 -581.0 -0.45 -0.4689 -0.945 3031110 ChemDiv3_009704 Cc1cc(C(=O)NCCCN2CCN(CC2)c3ccccc3F)n(n1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J03 compound treatment 360.0 -451.0 -0.16 560.0 -341.0 -0.26 -0.2984 -0.9721 3121963 ChemDiv3_009705 COc1ccccc1S(=O)(=O)Cc2ccc(o2)C(=O)NC(C)c3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J04 compound treatment 480.0 -331.0 -0.12 320.0 -581.0 -0.45 -0.3986 -0.8639 3031111 ChemDiv3_009706 CCc1cccc(NC(=O)C2=C(C)C(=O)OC32CCCCC3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J05 compound treatment 360.0 -451.0 -0.16 2880.0 1980.0 1.52 0.961 0.6291 3121964 ChemDiv3_009707 COC(CNC(=O)C1CCN(Cc2nc(oc2C)c3ccc(Cl)cc3)CC1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J06 compound treatment 280.0 -531.0 -0.19 520.0 -381.0 -0.29 -0.3402 -0.9773 3121965 ChemDiv3_009708 COc1ccccc1c2c(C)nn3c(NCCCN4CCCC4=O)cc(C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J07 compound treatment 200.0 -611.0 -0.22 1320.0 419.0 0.32 0.074 0.1908 3121966 ChemDiv3_009709 Cc1oc(nc1CN2CCCC(C2)C(=O)NC3CCCc4ccccc34)c5cccc(Cl)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J08 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3031112 ChemDiv3_009710 O=C(NC1CCCCC1)C2N(CCCN3CCCC3=O)C(=O)Cn4cccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J09 compound treatment 200.0 -611.0 -0.22 1000.0 98.8 0.08 -0.0997 -0.4341 3121967 ChemDiv3_009711 CCc1ccc(cc1)c2nc(CSCC(=O)NCc3ccccc3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J10 compound treatment 1520.0 709.0 0.25 360.0 -541.0 -0.42 -0.116 -0.2389 3031113 ChemDiv3_009712 CCOC(=O)C1CCCN(C1)C(=O)c2sc3nc(cn3c2C)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J11 compound treatment 720.0 -91.3 -0.03 480.0 -421.0 -0.32 -0.2516 -0.774 3121968 ChemDiv3_009713 CC1CCCCC1N(C)C2CCN(CCCNC(=O)/C=C/c3ccccc3Cl)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J12 compound treatment 360.0 -451.0 -0.16 5200.0 4300.0 3.3 2.2204 0.672 3031114 ChemDiv3_009714 Cc1cc2cc(CNC(=O)c3ccccc3C(F)(F)F)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J13 compound treatment 640.0 -171.0 -0.06 4080.0 3180.0 2.44 1.6827 0.6893 3121969 ChemDiv3_009715 CC1CCCCN1CCNC(=O)CS(=O)Cc2nc(oc2C)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J14 compound treatment 560.0 -251.0 -0.09 520.0 -381.0 -0.29 -0.27 -0.8824 3121970 ChemDiv3_009716 Cc1cc2cc(CNC(=O)C3(CC4CC5CC(C4)C3)C5)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J15 compound treatment 440.0 -371.0 -0.13 320.0 -581.0 -0.45 -0.4087 -0.8783 3031115 ChemDiv3_009717 Cc1oc(nc1CS(=O)(=O)CC(=O)NCC2CCCO2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J16 compound treatment 360.0 -451.0 -0.16 480.0 -421.0 -0.32 -0.3419 -0.9474 3121971 ChemDiv3_009718 Cc1ccc(cc1C)C(=O)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J17 compound treatment 3680.0 2870.0 1.02 400.0 -501.0 -0.38 0.4475 0.4113 3121972 ChemDiv3_009719 COC(CNC(=O)c1ccc2S(=O)c3ccccc3C(=O)N(Cc4cc(C)ccc4C)c2c1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J18 compound treatment 1080.0 269.0 0.1 320.0 -581.0 -0.45 -0.2481 -0.5438 3031116 ChemDiv3_009720 COc1ccc(CC(=O)NCc2ccc3[nH]c4CCCCc4c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J19 compound treatment 2240.0 1430.0 0.51 400.0 -501.0 -0.38 0.0863 0.1356 3121973 ChemDiv3_009721 CCN1C(=O)c2ccccc2S(=O)(=O)c3ccc(cc13)C(=O)NCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J20 compound treatment 400.0 -411.0 -0.15 280.0 -621.0 -0.48 -0.4404 -0.883 3031117 ChemDiv3_009722 Cc1cc2cc(CNC(=S)Nc3cccc(C)c3C)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J21 compound treatment 400.0 -411.0 -0.15 360.0 -541.0 -0.42 -0.397 -0.9014 3121974 ChemDiv3_009723 CCOc1ccc(OCC)c(NC(=O)c2ccc3S(=O)CC(=O)N(Cc4ccccc4)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J22 compound treatment 440.0 -371.0 -0.13 960.0 58.8 0.05 -0.0612 -0.4399 3031118 ChemDiv3_009724 O=C(NCc1ccc2[nH]c3CCCCc3c2c1)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J23 mock treatment 240.0 -571.0 -0.2 280.0 -621.0 -0.48 -0.4805 -0.9273 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 J24 mock treatment 720.0 -91.3 -0.03 280.0 -621.0 -0.48 -0.3601 -0.7534 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K01 compound treatment 480.0 -331.0 -0.12 1840.0 939.0 0.72 0.4265 0.5841 3121975 ChemDiv3_009725 CC1=CC2=NC(=O)/C(=C\c3ccco3)/C(=N)N2O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K02 compound treatment 440.0 -371.0 -0.13 600.0 -301.0 -0.23 -0.2567 -0.9644 3121976 ChemDiv3_009726 COc1ccc(cc1Cl)n2nc(C(=O)NCc3ccc(C)cc3)c4c5ccccc5n(C)c4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K03 compound treatment 1360.0 549.0 0.19 1280.0 379.0 0.29 0.3433 0.981 3031119 ChemDiv3_009727 Cc1ccccc1Cn2c(=O)n(Cc3ccco3)c(=O)c4ccc(cc24)C(=O)NCCc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K04 compound treatment 800.0 -11.3 0.0 760.0 -141.0 -0.11 -0.0795 -0.7326 3121977 ChemDiv3_009728 COc1ccccc1NC(=O)CSc2c3CCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K05 compound treatment 320.0 -491.0 -0.17 1120.0 219.0 0.17 -0.0045 -0.0185 3031120 ChemDiv3_009729 CN(C(=O)CCn1c(=O)oc2ccccc12)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K06 compound treatment 440.0 -371.0 -0.13 5720.0 4820.0 3.7 2.5228 0.6815 3121978 ChemDiv3_009730 Clc1cccc(c1)N2CCN(CC2)c3c4CCCc4nc5ccc(Cl)cc35 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K07 compound treatment 360.0 -451.0 -0.16 920.0 18.8 0.01 -0.103 -0.6409 3121979 ChemDiv3_009731 N=c1oc2c3CCCN4CCCc(cc2cc1C(=O)Nc5ccc(C#N)cc5)c43 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K08 compound treatment 480.0 -331.0 -0.12 520.0 -381.0 -0.29 -0.2901 -0.9196 3031121 ChemDiv3_009732 COc1ccccc1N(CN2CCCC2=O)C(=O)COc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K09 compound treatment 400.0 -411.0 -0.15 7160.0 6260.0 4.8 3.2945 0.6853 3121980 ChemDiv3_009733 CCOC(=O)c1sc2nc(SCC(=O)Nc3ccc(OCC)cc3)n(N)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K10 compound treatment 600.0 -211.0 -0.07 480.0 -421.0 -0.32 -0.2817 -0.8485 3031122 ChemDiv3_009734 Cc1noc(/C=C/c2ccco2)c1S(=O)(=O)N3CCC(CC3)C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K11 compound treatment 480.0 -331.0 -0.12 440.0 -461.0 -0.35 -0.3335 -0.8938 3121981 ChemDiv3_009735 Cn1c(=O)c2cc(sc2c3ccccc13)C(=O)Nc4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K12 compound treatment 3080.0 2270.0 0.8 440.0 -461.0 -0.35 0.3187 0.3625 3031123 ChemDiv3_009736 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K13 compound treatment 560.0 -251.0 -0.09 2320.0 1420.0 1.09 0.7072 0.6471 3121982 ChemDiv3_009737 CCOC(=O)N1CCC(CC1)NC(=O)c2cc3c(nn(C)c3s2)c4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K14 compound treatment 880.0 68.8 0.02 480.0 -421.0 -0.32 -0.2114 -0.6519 3031124 ChemDiv3_009738 Cc1cccc(NS(=O)(=O)c2ccc3n(C)c(=O)oc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K15 compound treatment 1640.0 829.0 0.29 680.0 -221.0 -0.17 0.0878 0.2585 3122163 ChemDiv3_009739 O=C(CSc1c2CCCCc2nc3ccccc13)NCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K16 compound treatment 400.0 -411.0 -0.15 760.0 -141.0 -0.11 -0.1798 -0.9893 3122164 ChemDiv3_009740 Cn1cc(C(=O)NCCc2ccccc2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K17 compound treatment 2160.0 1350.0 0.48 480.0 -421.0 -0.32 0.1096 0.1899 3031125 ChemDiv3_009741 COc1ccccc1C2CC(=O)N3CN(CSC3=C2C#N)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K18 compound treatment 480.0 -331.0 -0.12 440.0 -461.0 -0.35 -0.3335 -0.8938 3122165 ChemDiv3_009742 CCn1cc(C(=O)NCc2ccccc2Cl)c(=O)c3cc(ccc13)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K19 compound treatment 3680.0 2870.0 1.02 640.0 -261.0 -0.2 0.5778 0.557 1618758 ChemDiv3_009743 COc1ccc2nc(Nc3ccccc3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K20 compound treatment 2240.0 1430.0 0.51 800.0 -101.0 -0.08 0.3034 0.5917 3122166 ChemDiv3_009744 CCC(C)NC(=O)c1cn(CC)c2ccc(cc2c1=O)S(=O)(=O)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K21 compound treatment 560.0 -251.0 -0.09 800.0 -101.0 -0.08 -0.118 -0.9977 3031126 ChemDiv3_009745 Clc1cccc2sc(nc12)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K22 compound treatment 1000.0 189.0 0.07 520.0 -381.0 -0.29 -0.1596 -0.5316 3122167 ChemDiv3_009746 O=C(NCCCN1CCCC1)c2ccc(CS(=O)c3ccccc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K23 mock treatment 880.0 68.8 0.02 600.0 -301.0 -0.23 -0.1463 -0.6291 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 K24 mock treatment 760.0 -51.3 -0.02 440.0 -461.0 -0.35 -0.2632 -0.7424 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L01 compound treatment 2000.0 1190.0 0.42 440.0 -461.0 -0.35 0.0478 0.0868 3031127 ChemDiv3_009747 CCOC(=O)N1CCC(CC1)NC(=O)c2ccc(CS(=O)(=O)c3ccc(OC)cc3)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L02 compound treatment 440.0 -371.0 -0.13 600.0 -301.0 -0.23 -0.2567 -0.9644 3122168 ChemDiv3_009748 CCOc1ccc(CCNC(=O)C2=C(C)C(=O)OC32CCC(C)CC3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L03 compound treatment 480.0 -331.0 -0.12 960.0 58.8 0.05 -0.0512 -0.4068 3122169 ChemDiv3_009749 FC(F)(F)c1cccc(c1)S(=O)(=O)Cc2ccc(o2)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L04 compound treatment 560.0 -251.0 -0.09 440.0 -461.0 -0.35 -0.3134 -0.8583 3031128 ChemDiv3_009750 CC1=C(C(=O)Nc2ccc(C)cc2)C3(CCCCC3)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L05 compound treatment 440.0 -371.0 -0.13 560.0 -341.0 -0.26 -0.2784 -0.9494 3122170 ChemDiv3_009751 CC(CCc1ccccc1)NC(=O)C2CCN(Cc3nc(oc3C)c4ccc(Cl)cc4)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L06 compound treatment 360.0 -451.0 -0.16 720.0 -181.0 -0.14 -0.2116 -0.9976 3031129 ChemDiv3_009752 CCCN(CCC)CCNc1cc(C)nc2c(c(C)nn12)c3ccccc3OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L07 compound treatment 440.0 -371.0 -0.13 520.0 -381.0 -0.29 -0.3001 -0.935 3122171 ChemDiv3_009753 CCOC(=O)N1CCC(CC1)NC(=O)C2CCCN(Cc3nc(oc3C)c4cccc(C)c4)C2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L08 compound treatment 240.0 -571.0 -0.2 680.0 -221.0 -0.17 -0.2634 -0.9961 3031130 ChemDiv3_009754 CCCN(CCC)C(=O)c1sc2nc(cn2c1C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L09 compound treatment 1880.0 1070.0 0.38 3240.0 2340.0 1.8 1.5377 0.8379 3122172 ChemDiv3_009755 CCc1ccc(cc1)c2nc(CSCC(=O)NC3CC3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L10 compound treatment 320.0 -491.0 -0.17 800.0 -101.0 -0.08 -0.1782 -0.9338 3122173 ChemDiv3_009756 COc1ccc(cc1)c2cn3c(C)c(sc3n2)C(=O)N4CCN(CC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L11 compound treatment 320.0 -491.0 -0.17 1120.0 219.0 0.17 -0.0045 -0.0185 3031131 ChemDiv3_009757 CN(C1CCCC1)C2CCN(CC2)C(=O)CNC(=O)/C=C/c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L12 compound treatment 360.0 -451.0 -0.16 880.0 -21.3 -0.02 -0.1247 -0.7752 3122174 ChemDiv3_009758 Cc1cc2cc(CNC(=O)c3ccc4ccccc4c3)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L13 compound treatment 3440.0 2630.0 0.93 520.0 -381.0 -0.29 0.4524 0.4629 3122175 ChemDiv3_009759 Cc1oc(nc1CS(=O)CC(=O)N2CCC3(CC2)OCCO3)c4ccccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L14 compound treatment 480.0 -331.0 -0.12 2760.0 1860.0 1.43 0.9259 0.6467 3031132 ChemDiv3_009760 Cc1cc2cc(CNC(=O)c3ccc(C)cc3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L15 compound treatment 3200.0 2390.0 0.85 1280.0 379.0 0.29 0.8048 0.8983 3122176 ChemDiv3_009761 COc1cccc(c1)c2nc(CS(=O)(=O)CC(=O)Nc3ccccc3C)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L16 compound treatment 440.0 -371.0 -0.13 560.0 -341.0 -0.26 -0.2784 -0.9494 3031133 ChemDiv3_009762 COc1ccccc1C(=O)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L17 compound treatment 880.0 68.8 0.02 680.0 -221.0 -0.17 -0.1029 -0.5994 3122177 ChemDiv3_009763 CCN1C(=O)c2ccccc2S(=O)c3ccc(cc13)C(=O)N(C)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L18 compound treatment 320.0 -491.0 -0.17 680.0 -221.0 -0.17 -0.2433 -0.9999 3031134 ChemDiv3_009764 Clc1ccc(CC(=O)NCc2ccc3[nH]c4CCCCc4c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L19 compound treatment 1480.0 669.0 0.24 760.0 -141.0 -0.11 0.0911 0.3491 3122178 ChemDiv3_009765 CCCN(CCC)C(=O)c1ccc2c(c1)N(Cc3ccccc3F)C(=O)c4ccccc4S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L20 compound treatment 640.0 -171.0 -0.06 680.0 -221.0 -0.17 -0.1631 -0.9039 3031135 ChemDiv3_009766 COc1ccc(OC)c(NC(=S)NCc2ccc3[nH]c(C)cc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L21 compound treatment 760.0 -51.3 -0.02 6040.0 5140.0 3.95 2.7768 0.7038 3122179 ChemDiv3_009767 O=C(N1CCCCC1)c2ccc3S(=O)CC(=O)N(Cc4ccccc4)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L22 compound treatment 600.0 -211.0 -0.07 720.0 -181.0 -0.14 -0.1514 -0.9578 3122180 ChemDiv3_009768 Cn1c(=O)cc(OCC(=O)NCCC2=CCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L23 mock treatment 360.0 -451.0 -0.16 520.0 -381.0 -0.29 -0.3202 -0.9597 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 L24 mock treatment 640.0 -171.0 -0.06 800.0 -101.0 -0.08 -0.0979 -0.9926 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M01 compound treatment 1360.0 549.0 0.19 2000.0 1100.0 0.84 0.7341 0.848 3031281 ChemDiv3_009769 COc1cccc(CN2CCN(Cc3ccc(F)cc3)C2c4ccc(SC)cc4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M02 compound treatment 1600.0 789.0 0.28 1160.0 259.0 0.2 0.3383 0.9859 3031282 ChemDiv3_009770 CCc1ccc(Nc2c3CCCc3nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M03 compound treatment 440.0 -371.0 -0.13 400.0 -501.0 -0.38 -0.3652 -0.898 3031284 ChemDiv3_009771 CC(C)CN(CC(C)C)C(=O)CCn1c(=O)oc2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M04 compound treatment 800.0 -11.3 0.0 1480.0 579.0 0.44 0.3114 0.7007 3031285 ChemDiv3_009772 Clc1cccc(NC(=O)CSc2c3CCCc3nc4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M05 compound treatment 840.0 28.8 0.01 360.0 -541.0 -0.42 -0.2866 -0.6895 3031287 ChemDiv3_009773 CC1Cc2ccccc2N1C(=O)CCn3c(=O)oc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M06 compound treatment 400.0 -411.0 -0.15 520.0 -381.0 -0.29 -0.3101 -0.9483 3031288 ChemDiv3_009774 NC(=O)CSc1nnc(Cc2cc(=O)[nH]c(=O)[nH]2)n1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M07 compound treatment 1160.0 349.0 0.12 5600.0 4700.0 3.61 2.6382 0.7309 3122181 ChemDiv3_009775 CC(C1Sc2ccccc2N(Cc3cccc(Cl)c3)C1=O)C(=O)NC4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M08 compound treatment 440.0 -371.0 -0.13 960.0 58.8 0.05 -0.0612 -0.4399 3031290 ChemDiv3_009776 CC1CC(C)CN(C1)c2nc3ccccc3c(=O)n2c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M09 compound treatment 920.0 109.0 0.04 880.0 -21.3 -0.02 0.0157 0.3759 3122182 ChemDiv3_009777 Cn1c(=O)c2cc(sc2c3ccc(Cl)cc13)C(=O)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M10 compound treatment 1080.0 269.0 0.1 1720.0 819.0 0.63 0.5119 0.8051 3031292 ChemDiv3_009778 CCCNS(=O)(=O)c1ccc2n(C)c(=O)c(=O)n(C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M11 compound treatment 800.0 -11.3 0.0 880.0 -21.3 -0.02 -0.0144 -0.8549 3122183 ChemDiv3_009779 Cn1c(=O)c2cc(sc2c3ccccc13)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M12 compound treatment 560.0 -251.0 -0.09 720.0 -181.0 -0.14 -0.1614 -0.9768 3031294 ChemDiv3_009780 COC(CN(C)S(=O)(=O)c1ccc2n(C)c(=O)oc2c1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M13 compound treatment 1000.0 189.0 0.07 600.0 -301.0 -0.23 -0.1162 -0.4826 3122184 ChemDiv3_009781 Cn1nc(c2ccccc2F)c3cc(sc13)C(=O)NCCCN4CCN(CC4)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M14 compound treatment 360.0 -451.0 -0.16 560.0 -341.0 -0.26 -0.2984 -0.9721 3122185 ChemDiv3_009782 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NCCCN3CCN(CC3)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M15 compound treatment 680.0 -131.0 -0.05 1400.0 499.0 0.38 0.2378 0.6166 3031297 ChemDiv3_009783 CCc1ccc(NC(=O)CSc2c3CCCCc3nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M16 compound treatment 600.0 -211.0 -0.07 680.0 -221.0 -0.17 -0.1731 -0.9324 3122186 ChemDiv3_009784 Cn1cc(C(=O)NCc2cccs2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M17 compound treatment 760.0 -51.3 -0.02 720.0 -181.0 -0.14 -0.1112 -0.7928 3031298 ChemDiv3_009785 COc1cccc2sc(Nc3sc4CCCCc4c3C(=O)N)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M18 compound treatment 400.0 -411.0 -0.15 680.0 -221.0 -0.17 -0.2233 -0.9971 3122187 ChemDiv3_009786 CCn1cc(C(=O)NC2CCCCCC2)c(=O)c3cc(ccc13)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M19 compound treatment 1280.0 469.0 0.17 800.0 -101.0 -0.08 0.0626 0.3411 3031358 ChemDiv3_009787 COc1ccc2nc(Nc3nnc(o3)c4ccccc4)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M20 compound treatment 560.0 -251.0 -0.09 840.0 -61.3 -0.05 -0.0963 -0.9554 3031359 ChemDiv3_009788 CCn1cc(C(=O)NCCc2ccccc2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCC(C)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M21 compound treatment 440.0 -371.0 -0.13 480.0 -421.0 -0.32 -0.3218 -0.9216 1644633 ChemDiv3_009789 CCOc1ccc2nc(sc2c1)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M22 compound treatment 1840.0 1030.0 0.36 720.0 -181.0 -0.14 0.1597 0.4088 3031361 ChemDiv3_009790 Clc1ccc(cc1)S(=O)Cc2ccc(o2)C(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M23 mock treatment 480.0 -331.0 -0.12 960.0 58.8 0.05 -0.0512 -0.4068 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 M24 mock treatment 1600.0 789.0 0.28 640.0 -261.0 -0.2 0.056 0.1628 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N01 compound treatment 1000.0 189.0 0.07 600.0 -301.0 -0.23 -0.1162 -0.4826 3031362 ChemDiv3_009791 Cc1ccccc1S(=O)(=O)Cc2ccc(o2)C(=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N02 compound treatment 1440.0 629.0 0.22 560.0 -341.0 -0.26 -0.0275 -0.08 3031364 ChemDiv3_009792 CC1CCC2(CC1)OC(=O)C(=C2C(=O)N(C)Cc3ccccc3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N03 compound treatment 600.0 -211.0 -0.07 600.0 -301.0 -0.23 -0.2165 -0.8906 3031365 ChemDiv3_009793 FC(F)(F)c1cccc(c1)S(=O)(=O)Cc2ccc(o2)C(=O)NCc3ccc4OCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N04 compound treatment 560.0 -251.0 -0.09 440.0 -461.0 -0.35 -0.3134 -0.8583 3122188 ChemDiv3_009794 CC1=C(C(=O)NC2CCCCC2)C3(CCCCC3)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N05 compound treatment 760.0 -51.3 -0.02 480.0 -421.0 -0.32 -0.2415 -0.7457 3122374 ChemDiv3_009795 Cc1oc(nc1CN2CCC(CC2)C(=O)NCc3ccco3)c4ccccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N06 compound treatment 320.0 -491.0 -0.17 760.0 -141.0 -0.11 -0.1999 -0.9739 3031367 ChemDiv3_009796 COc1ccccc1c2c(C)nn3c(NCCN4CCCCC4C)cc(C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N07 compound treatment 640.0 -171.0 -0.06 640.0 -261.0 -0.2 -0.1848 -0.8817 3122375 ChemDiv3_009797 COc1ccc(cc1OC)c2nc(CSCC(=O)N(C)Cc3ccccc3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N08 compound treatment 440.0 -371.0 -0.13 320.0 -581.0 -0.45 -0.4087 -0.8783 3122376 ChemDiv3_009798 CCC1CCCCN1C(=O)c2sc3nc(cn3c2C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N09 compound treatment 1200.0 389.0 0.14 440.0 -461.0 -0.35 -0.1529 -0.4023 3031371 ChemDiv3_009799 CCc1ccc(cc1)c2nc(CSCC(=O)NCCc3ccccc3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N10 compound treatment 400.0 -411.0 -0.15 720.0 -181.0 -0.14 -0.2016 -0.9997 3122377 ChemDiv3_009800 COc1ccc(cc1)c2cn3c(C)c(sc3n2)C(=O)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N11 compound treatment 440.0 -371.0 -0.13 800.0 -101.0 -0.08 -0.1481 -0.9684 3031373 ChemDiv3_009801 COc1ccc(cc1)c2nc(CS(=O)CC(=O)N3CCCC3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N12 compound treatment 600.0 -211.0 -0.07 600.0 -301.0 -0.23 -0.2165 -0.8906 3122378 ChemDiv3_009802 Cc1cc2cc(CNC(=O)/C=C\c3ccccc3)ccc2[nH]1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N13 compound treatment 880.0 68.8 0.02 960.0 58.8 0.05 0.0491 0.9583 3031374 ChemDiv3_009803 CC(C)NC(=O)CS(=O)Cc1nc(oc1C)c2ccccc2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N14 compound treatment 400.0 -411.0 -0.15 680.0 -221.0 -0.17 -0.2233 -0.9971 3122379 ChemDiv3_009804 Cc1cc2cc(CNC(=O)/C=C\c3ccc4OCOc4c3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N15 compound treatment 680.0 -131.0 -0.05 560.0 -341.0 -0.26 -0.2182 -0.8199 3122380 ChemDiv3_009805 COc1cccc(c1)c2nc(CS(=O)(=O)CC(=O)NCCc3ccccc3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N16 compound treatment 520.0 -291.0 -0.1 480.0 -421.0 -0.32 -0.3017 -0.8888 3031376 ChemDiv3_009806 COc1cccc(c1)C(=O)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N17 compound treatment 680.0 -131.0 -0.05 960.0 58.8 0.05 -0.001 -0.0159 3122381 ChemDiv3_009807 CCCCN(C)C(=O)c1ccc2S(=O)c3ccccc3C(=O)N(CC)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N18 compound treatment 680.0 -131.0 -0.05 720.0 -181.0 -0.14 -0.1313 -0.8949 3031378 ChemDiv3_009808 Cc1cccc(CC(=O)NCc2ccc3[nH]c4CCCCc4c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N19 compound treatment 640.0 -171.0 -0.06 1120.0 219.0 0.17 0.0758 0.4244 3122382 ChemDiv3_009809 CC(C)NC(=O)c1ccc2c(c1)N(Cc3ccccc3F)C(=O)c4ccccc4S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N20 compound treatment 760.0 -51.3 -0.02 1200.0 299.0 0.23 0.1493 0.649 3122383 ChemDiv3_009810 Cc1cc2cc(CNC(=S)NC(C)(C)C)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N21 compound treatment 600.0 -211.0 -0.07 480.0 -421.0 -0.32 -0.2817 -0.8485 3031380 ChemDiv3_009811 COc1ccc(NC(=O)c2cc(C)nn2c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N22 compound treatment 480.0 -331.0 -0.12 1800.0 899.0 0.69 0.4048 0.5784 3122384 ChemDiv3_009812 Cn1c(=O)cc(OCC(=O)N2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N23 mock treatment 3640.0 2830.0 1.0 1080.0 179.0 0.14 0.8066 0.7964 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 N24 mock treatment 320.0 -491.0 -0.17 960.0 58.8 0.05 -0.0913 -0.5074 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O01 compound treatment 400.0 -411.0 -0.15 280.0 -621.0 -0.48 -0.4404 -0.883 3122385 ChemDiv3_009813 COc1ccc(OC)c(c1)C2N(Cc3ccccc3C)CCN2Cc4ccccc4F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O02 compound treatment 3080.0 2270.0 0.8 200.0 -701.0 -0.54 0.1884 0.1946 3031382 ChemDiv3_009814 O=C/1NN(C(=O)\C1=C\c2ccc(SC3CCCCC3)o2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O03 compound treatment 400.0 -411.0 -0.15 440.0 -461.0 -0.35 -0.3536 -0.9232 3122386 ChemDiv3_009815 O=C(CCn1c(=O)oc2ccccc12)N3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O04 compound treatment 360.0 -451.0 -0.16 280.0 -621.0 -0.48 -0.4504 -0.8954 3031385 ChemDiv3_009816 CN(Cc1ccccc1)C(=O)CSc2c3CCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O05 compound treatment 400.0 -411.0 -0.15 400.0 -501.0 -0.38 -0.3753 -0.9119 3031415 ChemDiv3_009817 CCc1ccc(NC(=O)CCn2c(=O)oc3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O06 compound treatment 360.0 -451.0 -0.16 5680.0 4780.0 3.67 2.481 0.6756 3031417 ChemDiv3_009818 CCSc1nnc(Cc2cc(=O)[nH]c(=O)[nH]2)n1c3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O07 compound treatment 240.0 -571.0 -0.2 440.0 -461.0 -0.35 -0.3937 -0.9649 3031418 ChemDiv3_009819 CC(C1Sc2ccccc2N(Cc3cccc(Cl)c3)C1=O)C(=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O08 compound treatment 400.0 -411.0 -0.15 280.0 -621.0 -0.48 -0.4404 -0.883 3031420 ChemDiv3_009820 CCCCN(C)c1nc2ccccc2c(=O)n1c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O09 compound treatment 280.0 -531.0 -0.19 400.0 -501.0 -0.38 -0.4054 -0.946 3031422 ChemDiv3_009821 Cn1c(=O)c2cc(sc2c3ccc(Cl)cc13)C(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O10 compound treatment 360.0 -451.0 -0.16 320.0 -581.0 -0.45 -0.4287 -0.9043 3031424 ChemDiv3_009822 CSc1cccc(NS(=O)(=O)c2ccc3n(C)c(=O)c(=O)n(C)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O11 compound treatment 400.0 -411.0 -0.15 360.0 -541.0 -0.42 -0.397 -0.9014 3122387 ChemDiv3_009823 CCc1ccc(NC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O12 compound treatment 320.0 -491.0 -0.17 320.0 -581.0 -0.45 -0.4388 -0.9159 3031425 ChemDiv3_009824 CCCNS(=O)(=O)c1ccc2n(C)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O13 compound treatment 200.0 -611.0 -0.22 320.0 -581.0 -0.45 -0.4689 -0.945 3122388 ChemDiv3_009825 O=C(CSc1c2CCCCc2nc3ccccc13)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O14 compound treatment 280.0 -531.0 -0.19 320.0 -581.0 -0.45 -0.4488 -0.9265 3031427 ChemDiv3_009826 CCN(c1ccc(C)c(C)c1)S(=O)(=O)c2ccc3n(C)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O15 compound treatment 360.0 -451.0 -0.16 360.0 -541.0 -0.42 -0.407 -0.914 3122389 ChemDiv3_009827 COc1cccc(c1)C(=O)Nc2c3CCCCc3nc4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O16 compound treatment 360.0 -451.0 -0.16 320.0 -581.0 -0.45 -0.4287 -0.9043 3031429 ChemDiv3_009828 Cn1cc(C(=O)NC2CCCCCC2)c(=O)c3cc(ccc13)S(=O)(=O)N4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O17 compound treatment 400.0 -411.0 -0.15 200.0 -701.0 -0.54 -0.4838 -0.8674 3122390 ChemDiv3_009829 COc1cccc2sc(NCc3ccccc3)nc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O18 compound treatment 320.0 -491.0 -0.17 320.0 -581.0 -0.45 -0.4388 -0.9159 3122391 ChemDiv3_009830 CCn1cc(C(=O)NCCc2ccccc2)c(=O)c3cc(ccc13)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O19 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3031431 ChemDiv3_009831 Fc1ccc2nc(Nc3nc4ccc(F)cc4s3)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O20 compound treatment 280.0 -531.0 -0.19 240.0 -661.0 -0.51 -0.4922 -0.909 3122392 ChemDiv3_009832 CCn1cc(C(=O)N2CC(C)CC(C)C2)c(=O)c3cc(ccc13)S(=O)(=O)N4CC(C)CC(C)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O21 compound treatment 280.0 -531.0 -0.19 280.0 -621.0 -0.48 -0.4705 -0.9175 3031433 ChemDiv3_009833 Brc1ccc2nc(sc2c1)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O22 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3122393 ChemDiv3_009834 Cc1ccccc1S(=O)Cc2ccc(o2)C(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O23 mock treatment 440.0 -371.0 -0.13 2280.0 1380.0 1.06 0.6553 0.6144 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 O24 mock treatment 240.0 -571.0 -0.2 280.0 -621.0 -0.48 -0.4805 -0.9273 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P01 compound treatment 3840.0 3030.0 1.07 280.0 -621.0 -0.48 0.4225 0.3594 3031434 ChemDiv3_009835 COC(CN(C)C(=O)c1ccc(CS(=O)(=O)c2ccccc2C)o1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P02 compound treatment 600.0 -211.0 -0.07 320.0 -581.0 -0.45 -0.3685 -0.8145 3122394 ChemDiv3_009836 CC1CCC2(CC1)OC(=O)C(=C2C(=O)N(C)C3CCCCC3)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P03 compound treatment 1280.0 469.0 0.17 280.0 -621.0 -0.48 -0.2197 -0.4349 3031435 ChemDiv3_009837 CC(C)CCNC(=O)c1ccc(CS(=O)(=O)c2cccc(c2)C(F)(F)F)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P04 compound treatment 560.0 -251.0 -0.09 280.0 -621.0 -0.48 -0.4003 -0.825 3122395 ChemDiv3_009838 CC1=C(C(=O)NCCCN2CCN(CC2)c3cc(Cl)ccc3C)C4(CCCCC4)OC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P05 compound treatment 400.0 -411.0 -0.15 280.0 -621.0 -0.48 -0.4404 -0.883 3122396 ChemDiv3_009839 CCc1ccc(cc1)c2nc(CN3CCC(CC3)C(=O)NC4CC4)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P06 compound treatment 680.0 -131.0 -0.05 440.0 -461.0 -0.35 -0.2833 -0.7933 3031438 ChemDiv3_009840 COc1ccc(cc1OC)c2c(C)nn3c(NCCC4=CCCCC4)cc(C)nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P07 compound treatment 240.0 -571.0 -0.2 360.0 -541.0 -0.42 -0.4371 -0.9455 3122397 ChemDiv3_009841 Cc1oc(nc1CSCC(=O)N2CCCC2)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P08 compound treatment 280.0 -531.0 -0.19 360.0 -541.0 -0.42 -0.4271 -0.936 3031441 ChemDiv3_009842 Cc1c(sc2nc(cn12)c3ccccc3)C(=O)N4CCC5(CC4)OCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P09 compound treatment 440.0 -371.0 -0.13 1840.0 939.0 0.72 0.4165 0.5685 3122398 ChemDiv3_009843 Cc1oc(nc1CSCC(=O)N2CCCC2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P10 compound treatment 800.0 -11.3 0.0 2200.0 1300.0 1.0 0.7022 0.7043 3122399 ChemDiv3_009844 COc1ccc(cc1)c2cn3c(C)c(sc3n2)C(=O)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P11 compound treatment 440.0 -371.0 -0.13 1800.0 899.0 0.69 0.3948 0.562 3031443 ChemDiv3_009845 COc1ccc(cc1)c2nc(CS(=O)CC(=O)NCC3CCCO3)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P12 compound treatment 480.0 -331.0 -0.12 240.0 -661.0 -0.51 -0.4421 -0.8484 3122400 ChemDiv3_009846 CCOc1ccc(CC(=O)NCc2ccc3[nH]c(C)cc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P13 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3122401 ChemDiv3_009847 Cc1oc(nc1CS(=O)CC(=O)NC2CC2)c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P14 compound treatment 400.0 -411.0 -0.15 360.0 -541.0 -0.42 -0.397 -0.9014 3031445 ChemDiv3_009848 COc1cc(/C=C\C(=O)NCc2ccc3n(C)c(C)cc3c2)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P15 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3031483 ChemDiv3_009849 COc1cccc(c1)c2nc(CS(=O)(=O)CC(=O)NC3CCCC(C)C3C)c(C)o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P16 compound treatment 320.0 -491.0 -0.17 280.0 -621.0 -0.48 -0.4605 -0.9068 3031484 ChemDiv3_009850 CCOc1ccc(cc1)C(=O)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P17 compound treatment 360.0 -451.0 -0.16 400.0 -501.0 -0.38 -0.3853 -0.9245 3031485 ChemDiv3_009851 CCN1C(=O)c2ccccc2S(=O)c3ccc(cc13)C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P18 compound treatment 360.0 -451.0 -0.16 440.0 -461.0 -0.35 -0.3636 -0.9356 3031486 ChemDiv3_009852 O=C(Cc1cccs1)NCc2ccc3[nH]c4CCCCc4c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P19 compound treatment 2440.0 1630.0 0.58 440.0 -461.0 -0.35 0.1582 0.2334 3031488 ChemDiv3_009853 CN(CCC#N)C(=O)c1ccc2c(c1)N(Cc3ccc(F)cc3)C(=O)c4ccccc4S2(=O)=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P20 compound treatment 280.0 -531.0 -0.19 200.0 -701.0 -0.54 -0.5139 -0.901 3122587 ChemDiv3_009854 Cc1cc2cc(CNC(=S)NCCc3ccccc3)ccc2n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P21 compound treatment 200.0 -611.0 -0.22 640.0 -261.0 -0.2 -0.2951 -0.9992 3031490 ChemDiv3_009855 Cc1cc(C(=O)Nc2cc(C)ccc2C)n(n1)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P22 compound treatment 360.0 -451.0 -0.16 1240.0 339.0 0.26 0.0707 0.2315 3122588 ChemDiv3_009856 CN1CCN(CC1)C(=O)COc2cc(=O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P23 mock treatment 3600.0 2790.0 0.99 1800.0 899.0 0.69 1.1874 0.9845 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2028 P24 mock treatment 400.0 -411.0 -0.15 440.0 -461.0 -0.35 -0.3536 -0.9232 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A01 compound treatment 9120.0 8130.0 2.89 240.0 -425.0 -0.33 1.8098 0.6233 3031492 ChemDiv3_009857 COc1ccc(CCNC(=O)COc2cc(=O)n(C)c3ccccc23)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A02 compound treatment 2320.0 1330.0 0.47 960.0 295.0 0.23 0.495 0.9433 3122589 ChemDiv3_009858 CCN(CC)C(=O)CSc1cc(=O)n(CC)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A03 compound treatment 3440.0 2450.0 0.87 400.0 -265.0 -0.2 0.4719 0.528 3122590 ChemDiv3_009859 CCc1ccc(CNC(=O)COc2cc(=O)n(C)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A04 compound treatment 8960.0 7970.0 2.83 240.0 -425.0 -0.33 1.7697 0.6215 3031494 ChemDiv3_009860 CCn1c(=O)cc(SCC(=O)NCCN2CCN(Cc3ccccc3)CC2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A05 compound treatment 720.0 -266.0 -0.09 280.0 -385.0 -0.3 -0.2755 -0.889 3122591 ChemDiv3_009861 CCOc1ccc(cc1)N(CC)C(=O)COc2cc(=O)n(CC)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A06 compound treatment 360.0 -626.0 -0.22 320.0 -345.0 -0.26 -0.3441 -0.9962 3031496 ChemDiv3_009862 O=C(c1ccccc1)c2cn(Cc3ccccc3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A07 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3122592 ChemDiv3_009863 CCc1ccccc1NC(=O)CCCOc2cc(=O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A08 compound treatment 320.0 -666.0 -0.24 360.0 -305.0 -0.23 -0.3324 -1.0 3122593 ChemDiv3_009864 Fc1ccc(cc1)c2cc(COCC(=O)N3CCOCC3)no2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A09 compound treatment 400.0 -586.0 -0.21 320.0 -345.0 -0.26 -0.3341 -0.9929 3031498 ChemDiv3_009865 CC(C)C(NS(=O)(=O)c1cccc2nsnc12)C(=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A10 compound treatment 200.0 -786.0 -0.28 320.0 -345.0 -0.26 -0.3842 -0.9996 3122594 ChemDiv3_009866 COc1ccc(cc1)c2cc3C(=O)CC(C)(C)Cc3n2Cc4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A11 compound treatment 400.0 -586.0 -0.21 280.0 -385.0 -0.3 -0.3558 -0.9853 3122595 ChemDiv3_009867 CCCNC(=O)C1CCC(CNS(=O)(=O)c2cccc3nsnc23)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A12 compound treatment 280.0 -706.0 -0.25 1000.0 335.0 0.26 0.005 0.0138 3031501 ChemDiv3_009868 CCc1ccc(NC(=O)c2cc(C)n[nH]2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A13 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3122596 ChemDiv3_009869 O=C(NC1CCN(Cc2ccccc2)CC1)[C@H](Cc3ccccc3)N4Cc5ccccc5C4=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A14 compound treatment 520.0 -466.0 -0.17 240.0 -425.0 -0.33 -0.3474 -0.9506 3031503 ChemDiv3_009870 CCCSc1nnc(c2c[nH]c3ccccc23)n1CC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A15 compound treatment 280.0 -706.0 -0.25 360.0 -305.0 -0.23 -0.3425 -0.9994 3122597 ChemDiv3_009871 COc1ccccc1NC(=O)[C@H](Cc2ccccc2)N3Cc4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A16 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3031505 ChemDiv3_009872 CN(Cc1ccccc1)C(=O)c2cc3c(Cl)nc4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A17 compound treatment 160.0 -826.0 -0.29 280.0 -385.0 -0.3 -0.416 -1.0 3122598 ChemDiv3_009873 Cc1nc2cc(nn2c(C)c1CCC(=O)N3CCc4ccccc34)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A18 compound treatment 440.0 -546.0 -0.19 360.0 -305.0 -0.23 -0.3023 -0.9957 3031507 ChemDiv3_009874 Clc1ccc(CNC(=O)c2cc3c(Cl)nc4ccccc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A19 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3122599 ChemDiv3_009875 Cc1nc2ncnn2c(C)c1CCC(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A20 compound treatment 280.0 -706.0 -0.25 400.0 -265.0 -0.2 -0.3208 -0.9946 3122600 ChemDiv3_009876 CCOC(=O)N1CCN(CC1)C(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A21 compound treatment 240.0 -746.0 -0.26 280.0 -385.0 -0.3 -0.3959 -0.9985 3031509 ChemDiv3_009877 CCCNC(=O)CCc1c(C)nc2n(C)c(=O)n(C)c(=O)c2c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A22 compound treatment 4520.0 3530.0 1.25 280.0 -385.0 -0.3 0.6777 0.5262 3031546 ChemDiv3_009878 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)NCC4(CCCC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A23 mock treatment 600.0 -386.0 -0.14 240.0 -425.0 -0.33 -0.3273 -0.9259 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 A24 mock treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B01 compound treatment 520.0 -466.0 -0.17 320.0 -345.0 -0.26 -0.304 -0.9744 3031547 ChemDiv3_009879 CCc1ccc(NC(=O)c2cc3c(=O)n(CC)c4ccccc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B02 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3031548 ChemDiv3_009880 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)Nc3cccc(CC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B03 compound treatment 360.0 -626.0 -0.22 3160.0 2500.0 1.92 1.1976 0.6209 3031550 ChemDiv3_009881 CCCN(CCC)C(=O)c1cc2c(=O)n(CC)c3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B04 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3031552 ChemDiv3_009882 O=C(/C=C/c1ccco1)N2CCn3c(C2)nc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B05 compound treatment 440.0 -546.0 -0.19 1480.0 815.0 0.63 0.3057 0.4664 3031554 ChemDiv3_009883 CCN1CCCC1CNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B06 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3122601 ChemDiv3_009884 Fc1ccc(CN2CCCN(C2)C(=O)c3oc(=O)c4ccccc4c3c5ccccc5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B07 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3031557 ChemDiv3_009885 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)NCCN4CCN(Cc5ccccc5)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B08 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3122602 ChemDiv3_009886 COc1ccc(cc1)C(=O)NC(C)C(N2CCOCC2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B09 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 3031559 ChemDiv3_009887 COc1ccc2cc3c(N)nn(C(=O)c4ccncc4)c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B10 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3122603 ChemDiv3_009888 CCN1CCN(CC1)C(C(C)NS(=O)(=O)c2ccc(C)cc2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B11 compound treatment 240.0 -746.0 -0.26 240.0 -425.0 -0.33 -0.4176 -0.9947 3122604 ChemDiv3_009889 CC1CCN(CC1)C(=O)C(Cc2ccccc2)NS(=O)(=O)c3ccc4n(C)c(=O)n(C)c(=O)c4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B12 compound treatment 240.0 -746.0 -0.26 360.0 -305.0 -0.23 -0.3525 -0.9981 3031560 ChemDiv3_009890 Cn1c(=O)n(C)c2nc(nc(SCc3cccc(c3)C(F)(F)F)c2c1=O)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B13 compound treatment 320.0 -666.0 -0.24 240.0 -425.0 -0.33 -0.3976 -0.9876 3122605 ChemDiv3_009891 COc1cccc(NC(=O)c2ccc3c(SCC(=O)O)c4CCCCc4nc3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B14 compound treatment 240.0 -746.0 -0.26 280.0 -385.0 -0.3 -0.3959 -0.9985 3031562 ChemDiv3_009892 CC(N1C(Nc2ccc(F)cc2)c3ccccc3C1=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B15 compound treatment 320.0 -666.0 -0.24 400.0 -265.0 -0.2 -0.3107 -0.9971 3122606 ChemDiv3_009893 Clc1c2CCCCc2nc3cc(ccc13)C(=O)N4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B16 compound treatment 320.0 -666.0 -0.24 480.0 -185.0 -0.14 -0.2673 -0.97 3031563 ChemDiv3_009894 Cc1nc2c(C)cccn2c1C(Nc3ccc(F)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B17 compound treatment 280.0 -706.0 -0.25 2200.0 1540.0 1.18 0.6564 0.5447 3122607 ChemDiv3_009895 Clc1ccc(CCNC(=O)c2ccc3c(Cl)c4CCCCc4nc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B18 compound treatment 600.0 -386.0 -0.14 680.0 15.5 0.01 -0.0885 -0.6433 3122608 ChemDiv3_009896 COc1ccc(CN2CNc3c(C2)c(C)nn3c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B19 compound treatment 1880.0 894.0 0.32 400.0 -265.0 -0.2 0.0806 0.2141 3031564 ChemDiv3_009897 CC1CCCCN1CCNC(=O)c2ccc3c(Cl)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B20 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3122609 ChemDiv3_009898 CCOC(=O)N1CCC(=CC1)c2c(C)[nH]c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B21 compound treatment 4360.0 3370.0 1.2 320.0 -345.0 -0.26 0.6593 0.5379 3031566 ChemDiv3_009899 Brc1ccc(NC(=O)CSC2=NS(=O)(=O)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B22 compound treatment 400.0 -586.0 -0.21 400.0 -265.0 -0.2 -0.2907 -0.9999 3122610 ChemDiv3_009900 Cc1ccc2[nH]c3C(CCCc3c2c1)Nc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B23 mock treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 B24 mock treatment 2160.0 1170.0 0.42 280.0 -385.0 -0.3 0.0857 0.1679 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C01 compound treatment 520.0 -466.0 -0.17 200.0 -465.0 -0.36 -0.3691 -0.939 3122611 ChemDiv3_009901 Cn1c(=O)cc(OCC(=O)NCC2COc3ccccc3O2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C02 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3031569 ChemDiv3_009902 CCn1c(=O)cc(SCC(=O)N2CCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C03 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3122612 ChemDiv3_009903 CC(NC(=O)COc1cc(=O)n(C)c2ccccc12)c3ccc4OCCOc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C04 compound treatment 320.0 -666.0 -0.24 360.0 -305.0 -0.23 -0.3324 -1.0 3031572 ChemDiv3_009904 CCn1c(=O)cc(SCC(=O)Nc2cccnc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C05 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3122613 ChemDiv3_009905 CCn1c(=O)cc(OCC(=O)N(C)c2ccccc2F)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C06 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 3122614 ChemDiv3_009906 Cc1cccc(Cn2cc(C(=O)c3ccc(C)c(C)c3)c(=O)c4cc5OCOc5cc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C07 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3031574 ChemDiv3_009907 COc1cccc(CNC(=O)CCCOc2cc(=O)n(C)c3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C08 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3031614 ChemDiv3_009908 CC(C)CC(NS(=O)(=O)c1ccc2nc(C)sc2c1)C(=O)NC3CCCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C09 compound treatment 360.0 -626.0 -0.22 520.0 -145.0 -0.11 -0.2355 -0.9485 3031615 ChemDiv3_009909 O=C(C1CCCN1S(=O)(=O)c2cccc3nsnc23)N4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C10 compound treatment 400.0 -586.0 -0.21 280.0 -385.0 -0.3 -0.3558 -0.9853 3031616 ChemDiv3_009910 FC(F)(F)c1cccc(c1)N2CCN(CC2)C(=O)c3cc(n[nH]3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C11 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3031618 ChemDiv3_009911 CC(C)c1ccc(NC(=O)C2CCC(CNS(=O)(=O)c3cccc4nsnc34)CC2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C12 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 3031619 ChemDiv3_009912 CC1CC(C)CN(C1)C(=O)c2cc(C)n[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C13 compound treatment 360.0 -626.0 -0.22 440.0 -225.0 -0.17 -0.279 -0.9921 3031620 ChemDiv3_009913 Cc1cccc(CCNC(=O)[C@H](Cc2ccccc2)N3Cc4ccccc4C3=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C14 compound treatment 240.0 -746.0 -0.26 320.0 -345.0 -0.26 -0.3742 -1.0 3122795 ChemDiv3_009914 CCn1c(SCC(=O)N2CCCC2)nnc1c3c[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C15 compound treatment 240.0 -746.0 -0.26 360.0 -305.0 -0.23 -0.3525 -0.9981 3122796 ChemDiv3_009915 CCOc1ccc(NC(=O)[C@H](C(C)CC)N2Cc3ccccc3C2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C16 compound treatment 360.0 -626.0 -0.22 240.0 -425.0 -0.33 -0.3875 -0.9826 3031622 ChemDiv3_009916 Clc1nc2ccccc2c3sc(cc13)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C17 compound treatment 400.0 -586.0 -0.21 320.0 -345.0 -0.26 -0.3341 -0.9929 3122797 ChemDiv3_009917 Cc1nc2cc(nn2c(C)c1CCC(=O)Nc3ccc4OCCOc4c3)c5cccc(F)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C18 compound treatment 240.0 -746.0 -0.26 400.0 -265.0 -0.2 -0.3308 -0.9914 3031624 ChemDiv3_009918 CC(C)CN(CC(C)C)C(=O)c1cc2c(Cl)nc3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C19 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 3122798 ChemDiv3_009919 Cc1nc2nc(C)c(CCC(=O)NCCC3=CCCCC3)c(C)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C20 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3031626 ChemDiv3_009920 CCOc1ccc(NC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C21 compound treatment 520.0 -466.0 -0.17 240.0 -425.0 -0.33 -0.3474 -0.9506 3122799 ChemDiv3_009921 CCOC(=O)N1CCN(CC1)C(=O)C(CC(C)C)NS(=O)(=O)c2ccc3n(C)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C22 compound treatment 280.0 -706.0 -0.25 360.0 -305.0 -0.23 -0.3425 -0.9994 3031629 ChemDiv3_009922 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C23 mock treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 C24 mock treatment 320.0 -666.0 -0.24 200.0 -465.0 -0.36 -0.4193 -0.98 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D01 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3122800 ChemDiv3_009923 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D02 compound treatment 360.0 -626.0 -0.22 240.0 -425.0 -0.33 -0.3875 -0.9826 3122801 ChemDiv3_009924 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N3C(C)Cc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D03 compound treatment 240.0 -746.0 -0.26 400.0 -265.0 -0.2 -0.3308 -0.9914 3031631 ChemDiv3_009925 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N(C)CCC#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D04 compound treatment 400.0 -586.0 -0.21 400.0 -265.0 -0.2 -0.2907 -0.9999 3031633 ChemDiv3_009926 O=S(=O)(Cc1ccccc1)N2CCn3c(C2)nc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D05 compound treatment 320.0 -666.0 -0.24 360.0 -305.0 -0.23 -0.3324 -1.0 3122802 ChemDiv3_009927 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)N4CCN(CC4)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D06 compound treatment 360.0 -626.0 -0.22 400.0 -265.0 -0.2 -0.3007 -0.999 3122803 ChemDiv3_009928 CN(C(=O)c1oc(=O)c2ccccc2c1c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D07 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3031635 ChemDiv3_009929 Cc1ccc(CCNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D08 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 3122804 ChemDiv3_009930 CC(NC(=O)c1ccc(F)cc1)C(N2CCN(C)CC2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D09 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3031636 ChemDiv3_009931 COc1ccc2cc3c(N)nn(C(=O)Cc4c(F)cccc4Cl)c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D10 compound treatment 360.0 -626.0 -0.22 320.0 -345.0 -0.26 -0.3441 -0.9962 3122805 ChemDiv3_009932 COc1ccccc1N2CCN(CC2)C(C(C)NS(=O)(=O)c3ccc(F)cc3)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D11 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 3122806 ChemDiv3_009933 Cc1ccccc1NC(=O)C(NS(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D12 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3031638 ChemDiv3_009934 COc1ccc(cc1)C(=O)CSc2nc(nc3n(C)c(=O)n(C)c(=O)c23)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D13 compound treatment 400.0 -586.0 -0.21 360.0 -305.0 -0.23 -0.3124 -0.9983 3122807 ChemDiv3_009935 CC1CCN(CC1)C(=O)c2ccc3c(SCC(=O)O)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D14 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3031640 ChemDiv3_009936 Cc1csc(NC2N(Cc3ccccc3)C(=O)c4ccccc24)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D15 compound treatment 320.0 -666.0 -0.24 440.0 -225.0 -0.17 -0.289 -0.988 3122808 ChemDiv3_009937 CC1CCN(CC1)C(=O)c2ccc3c(Cl)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D16 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3031642 ChemDiv3_009938 COC(=O)c1cc(cc(c1)C(=O)OC)N2Cc3nccnc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D17 compound treatment 320.0 -666.0 -0.24 360.0 -305.0 -0.23 -0.3324 -1.0 3031677 ChemDiv3_009939 CCN(Cc1ccccc1)C(=O)c2ccc3c(Cl)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D18 compound treatment 240.0 -746.0 -0.26 400.0 -265.0 -0.2 -0.3308 -0.9914 3031679 ChemDiv3_009940 COC(=O)c1cnn2CN(Cc3ccccc3)CNc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D19 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3031680 ChemDiv3_009941 CC(C)N(Cc1nc(no1)c2ccccc2)C(=O)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D20 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3031682 ChemDiv3_009942 Cc1[nH]c2ccccc2c1C3=CCNCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D21 compound treatment 240.0 -746.0 -0.26 360.0 -305.0 -0.23 -0.3525 -0.9981 3031683 ChemDiv3_009943 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D22 compound treatment 200.0 -786.0 -0.28 400.0 -265.0 -0.2 -0.3408 -0.9878 3031685 ChemDiv3_009944 Cc1ccc2[nH]c3C(CCCc3c2c1)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D23 mock treatment 240.0 -746.0 -0.26 960.0 295.0 0.23 -0.0268 -0.0768 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 D24 mock treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E01 compound treatment 280.0 -706.0 -0.25 1760.0 1100.0 0.84 0.4175 0.4758 3031686 ChemDiv3_009945 Cn1c(=O)cc(OCC(=O)NCCCN2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E02 compound treatment 360.0 -626.0 -0.22 880.0 215.0 0.17 -0.0401 -0.1448 3122809 ChemDiv3_009946 CCn1c(=O)cc(SCC(=O)NCCCN2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E03 compound treatment 2120.0 1130.0 0.4 2520.0 1860.0 1.42 1.2917 0.8726 3031687 ChemDiv3_009947 CCC(C)NC(=O)CSc1cc(=O)n(C)c2ccc(Cl)cc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E04 compound treatment 560.0 -426.0 -0.15 600.0 -64.5 -0.05 -0.1419 -0.8921 3122810 ChemDiv3_009948 Cc1ccc(cc1)S(=O)(=O)c2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E05 compound treatment 1000.0 13.8 0.0 1880.0 1220.0 0.93 0.6633 0.7108 3031689 ChemDiv3_009949 CCn1c(=O)cc(OCC(=O)NCCCN2CCCC2=O)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E06 compound treatment 360.0 -626.0 -0.22 920.0 255.0 0.2 -0.0184 -0.0621 3122811 ChemDiv3_009950 Clc1ccc(CNC(=O)c2cc3CSCc3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E07 compound treatment 960.0 -26.3 -0.01 1400.0 735.0 0.56 0.3927 0.6954 3122812 ChemDiv3_009951 O=C(NC1CCCCCCC1)C2CCCN(C2)S(=O)(=O)c3c[nH]cn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E08 compound treatment 1840.0 854.0 0.3 1280.0 615.0 0.47 0.5483 0.9769 3031692 ChemDiv3_009952 O=S(=O)(c1ccccc1)c/2cc3ccccc3o\c2=N/c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E09 compound treatment 680.0 -306.0 -0.11 1160.0 495.0 0.38 0.1922 0.4857 3122813 ChemDiv3_009953 Cc1ccc(C)c(c1)N2CCN(CC2)C(=O)C3CCCN3S(=O)(=O)c4cccc5nsnc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E10 compound treatment 520.0 -466.0 -0.17 240.0 -425.0 -0.33 -0.3474 -0.9506 3031693 ChemDiv3_009954 O=C(N1CCCCC1)c2cc(n[nH]2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E11 compound treatment 2440.0 1450.0 0.52 600.0 -64.5 -0.05 0.3296 0.6363 3122814 ChemDiv3_009955 CN(CC(=O)NCc1ccccc1)S(=O)(=O)c2ccc3NC(=O)CCc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E12 compound treatment 1720.0 734.0 0.26 1240.0 575.0 0.44 0.4965 0.9682 3122815 ChemDiv3_009956 Cc1ccc(C)c(c1)N2CCN(CC2)C(=O)C3CCN(CC3)c4ccc(nn4)N5CCOCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E13 compound treatment 1200.0 214.0 0.08 640.0 -24.5 -0.02 0.0403 0.5159 3031696 ChemDiv3_009957 CCC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)NCc3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E14 compound treatment 1600.0 614.0 0.22 560.0 -105.0 -0.08 0.0972 0.419 3122816 ChemDiv3_009958 CCn1c(SCC(=O)N2CCCc3ccccc23)nnc1c4c[nH]c5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E15 compound treatment 520.0 -466.0 -0.17 4800.0 4140.0 3.17 2.128 0.6694 3031698 ChemDiv3_009959 COc1ccc(NC(=O)[C@H](CCS(=O)(=O)C)N2Cc3ccccc3C2=O)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E16 compound treatment 1680.0 694.0 0.25 2360.0 1700.0 1.3 1.0944 0.8262 3122817 ChemDiv3_009960 CN(C)CCNC(=O)c1cc2c(Cl)nc3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E17 compound treatment 3240.0 2250.0 0.8 4000.0 3340.0 2.56 2.376 0.8857 3122818 ChemDiv3_009961 COc1ccc(cc1)N2Cc3cccc(C(=O)Nc4cccc(OC)c4)c3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E18 compound treatment 440.0 -546.0 -0.19 1800.0 1140.0 0.87 0.4794 0.5368 3031701 ChemDiv3_009962 Clc1nc2ccccc2c3sc(cc13)C(=O)NCCc4ccsc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E19 compound treatment 480.0 -506.0 -0.18 1320.0 655.0 0.5 0.2288 0.4283 3122819 ChemDiv3_009963 CC(NC(=O)CCc1c(C)nc2n(nc(C)c2c1C)c3ccc(C)cc3)c4ccc5OCCOc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E20 compound treatment 1720.0 734.0 0.26 1240.0 575.0 0.44 0.4965 0.9682 3031703 ChemDiv3_009964 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)N4CCN(Cc5ccccc5)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E21 compound treatment 2760.0 1770.0 0.63 5280.0 4620.0 3.54 2.9505 0.8198 3122820 ChemDiv3_009965 CC(C)CC(NS(=O)(=O)c1ccc2n(C)c(=O)oc2c1)C(=O)Nc3cccc(C)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E22 compound treatment 560.0 -426.0 -0.15 3800.0 3140.0 2.41 1.5952 0.6614 3031705 ChemDiv3_009966 COC(CNC(=O)c1cc2c(=O)n(C)c3ccccc3c2n1C)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E23 mock treatment 720.0 -266.0 -0.09 1840.0 1180.0 0.9 0.5713 0.6297 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 E24 mock treatment 760.0 -226.0 -0.08 840.0 175.0 0.13 0.0385 0.2456 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F01 compound treatment 2000.0 1010.0 0.36 3000.0 2340.0 1.79 1.5221 0.8324 3122821 ChemDiv3_009967 CCOc1ccccc1N(C)C(=O)c2cc3c(=O)n(CC)c4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F02 compound treatment 4560.0 3570.0 1.27 1440.0 775.0 0.6 1.3174 0.9406 3031758 ChemDiv3_009968 CCCCN(Cc1ccccc1)S(=O)(=O)c2ccc3n(CC(=O)OCC)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F03 compound treatment 1200.0 214.0 0.08 2480.0 1820.0 1.39 1.0392 0.7445 3031760 ChemDiv3_009969 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N(C)CC(OC)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F04 compound treatment 1000.0 13.8 0.0 1280.0 615.0 0.47 0.3376 0.7144 3031762 ChemDiv3_009970 O=C(Nc1ccccc1)N2CCn3c(C2)nc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F05 compound treatment 800.0 -186.0 -0.07 1280.0 615.0 0.47 0.2874 0.6024 3031763 ChemDiv3_009971 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F06 compound treatment 2520.0 1530.0 0.54 2520.0 1860.0 1.42 1.392 0.9129 3031765 ChemDiv3_009972 CC(C)CCN(Cc1ccco1)C(=O)c2oc(=O)c3ccccc3c2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F07 compound treatment 640.0 -346.0 -0.12 1360.0 695.0 0.53 0.2907 0.5306 3031766 ChemDiv3_009973 CC(C)CN(CC(C)C)C(=O)c1cc2c(=O)oc3ccc(C)cc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F08 compound treatment 1320.0 334.0 0.12 1280.0 615.0 0.47 0.4178 0.8578 3122997 ChemDiv3_009974 CCN1CCN(CC1)C(C(C)NC(=O)C(C)C)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F09 compound treatment 1160.0 174.0 0.06 2160.0 1500.0 1.15 0.8554 0.744 3031768 ChemDiv3_009975 COc1ccc2cc3c(N)nn(C(=O)CCn4c(=S)oc5ccccc45)c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F10 compound treatment 800.0 -186.0 -0.07 1200.0 535.0 0.41 0.244 0.5859 3122998 ChemDiv3_009976 Cc1nc(SCc2ccc(cc2)C(F)(F)F)c3c(=O)n(C)c(=O)n(C)c3n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F11 compound treatment 880.0 -106.0 -0.04 3520.0 2860.0 2.19 1.5235 0.6948 3122999 ChemDiv3_009977 CN(CC(=O)NC1CCCC1)S(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F12 compound treatment 840.0 -146.0 -0.05 1640.0 975.0 0.75 0.4929 0.6565 3031771 ChemDiv3_009978 Cn1c(=O)n(C)c2nc(nc(SCC(=O)N3CCCc4ccccc34)c2c1=O)c5cccs5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F13 compound treatment 840.0 -146.0 -0.05 2240.0 1580.0 1.21 0.8186 0.6762 3123000 ChemDiv3_009979 COc1ccccc1CNC(=O)c2ccc3c(SCC(=O)O)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F14 compound treatment 2160.0 1170.0 0.42 1880.0 1220.0 0.93 0.9543 0.9339 1211662 ChemDiv3_009980 OC(=O)c1nccnc1C(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F15 compound treatment 960.0 -26.3 -0.01 960.0 295.0 0.23 0.1538 0.6775 3123001 ChemDiv3_009981 Clc1c2CCCCc2nc3cc(ccc13)C(=O)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F16 compound treatment 2480.0 1490.0 0.53 1120.0 455.0 0.35 0.622 0.9796 3031773 ChemDiv3_009982 CCN1Cc2cccc(C(=O)O)c2C1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F17 compound treatment 960.0 -26.3 -0.01 960.0 295.0 0.23 0.1538 0.6775 3123002 ChemDiv3_009983 Cc1cccc(CN2CCC(CNC(=O)c3ccc4c(Cl)c5CCCCc5nc4c3)CC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F18 compound treatment 880.0 -106.0 -0.04 800.0 135.0 0.1 0.0469 0.4239 3031776 ChemDiv3_009984 O=C(NCCc1ccccc1)c2cc3ccccn3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F19 compound treatment 1040.0 53.8 0.02 520.0 -145.0 -0.11 -0.065 -0.5771 3123003 ChemDiv3_009985 COc1ccc(CC(=O)N(Cc2nc(no2)c3ccc(Cl)cc3)C(C)C)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F20 compound treatment 1760.0 774.0 0.27 4640.0 3980.0 3.05 2.3522 0.7676 3031778 ChemDiv3_009986 Cc1ccc(cc1)c2cc(N)[nH]n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F21 compound treatment 760.0 -226.0 -0.08 1080.0 415.0 0.32 0.1688 0.5132 3123004 ChemDiv3_009987 CCCN(CCC)S(=O)(=O)c1ccc2n(CC(=O)OCC)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F22 compound treatment 2480.0 1490.0 0.53 4680.0 4020.0 3.08 2.5545 0.8167 3031780 ChemDiv3_009988 Cc1ccnc(c1)N2C(Nc3ccc(Br)c(C)c3)c4ccccc4C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F23 mock treatment 4600.0 3610.0 1.28 1840.0 1180.0 0.9 1.5446 0.9852 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 F24 mock treatment 3120.0 2130.0 0.76 1200.0 535.0 0.41 0.8259 0.9589 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G01 compound treatment 2440.0 1450.0 0.52 480.0 -185.0 -0.14 0.2645 0.4946 3123005 ChemDiv3_009989 CCOc1ccccc1N(C)C(=O)COc2cc(=O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G02 compound treatment 440.0 -546.0 -0.19 520.0 -145.0 -0.11 -0.2155 -0.965 3123006 ChemDiv3_009990 CCn1c(=O)cc(SCC(=O)N(CC=C)c2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G03 compound treatment 680.0 -306.0 -0.11 1080.0 415.0 0.32 0.1487 0.4414 3031782 ChemDiv3_009991 CCn1c(=O)cc(OCC(=O)Nc2cccc(OC)c2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G04 compound treatment 1120.0 134.0 0.05 1280.0 615.0 0.47 0.3677 0.7742 3123007 ChemDiv3_009992 Fc1ccc(cc1)S(=O)(=O)c2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G05 compound treatment 400.0 -586.0 -0.21 560.0 -105.0 -0.08 -0.2038 -0.9142 3031783 ChemDiv3_009993 CCn1c(=O)cc(OCC(=O)NC2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G06 compound treatment 7040.0 6050.0 2.15 3640.0 2980.0 2.28 3.1338 0.9995 3123008 ChemDiv3_009994 CC(C)CCNC(=O)c1cc2CSCc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G07 compound treatment 1080.0 93.8 0.03 1920.0 1260.0 0.96 0.7051 0.7311 3123009 ChemDiv3_009995 COc1ccc(cc1)N2CCN(CCCNC(=O)C3CCCN(C3)S(=O)(=O)c4c[nH]cn4)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G08 compound treatment 1160.0 174.0 0.06 1160.0 495.0 0.38 0.3126 0.8111 3031842 ChemDiv3_009996 COc1ccc2cc(/c(=N/c3ccc4OCCOc4c3)/oc2c1)S(=O)(=O)c5ccc(C)c(C)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G09 compound treatment 440.0 -546.0 -0.19 1600.0 935.0 0.72 0.3708 0.4985 3031844 ChemDiv3_009997 O=C(NCCc1ccccc1)C2CCCN2S(=O)(=O)c3cccc4nsnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G10 compound treatment 600.0 -386.0 -0.14 1720.0 1060.0 0.81 0.4761 0.5793 3031846 ChemDiv3_009998 CC1CCCC(C)N1C(=O)c2cc(n[nH]2)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G11 compound treatment 1160.0 174.0 0.06 1600.0 935.0 0.72 0.5514 0.765 3031848 ChemDiv3_009999 Cc1ccc(CNC(=O)[C@H](N2Cc3ccccc3C2=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G12 compound treatment 680.0 -306.0 -0.11 440.0 -225.0 -0.17 -0.1987 -0.9752 3031849 ChemDiv3_010000 COc1ccc(CCNC(=O)C2CCN(CC2)c3ccc(nn3)N4CCOCC4)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G13 compound treatment 280.0 -706.0 -0.25 520.0 -145.0 -0.11 -0.2556 -0.9329 3123010 ChemDiv3_010001 CCC(C)[C@H](N1Cc2ccccc2C1=O)C(=O)NCc3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G14 compound treatment 520.0 -466.0 -0.17 1320.0 655.0 0.5 0.2389 0.451 3031851 ChemDiv3_010002 CCn1c(SCC(=O)NCCc2ccccc2)nnc1c3c[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G15 compound treatment 1000.0 13.8 0.0 1320.0 655.0 0.5 0.3593 0.7139 3123011 ChemDiv3_010003 CCCNC(=O)CCc1c(C)nc2cc(nn2c1C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G16 compound treatment 2800.0 1810.0 0.64 1200.0 535.0 0.41 0.7457 0.9766 3031853 ChemDiv3_010004 CCCCN(C)C(=O)c1cc2c(Cl)nc3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G17 compound treatment 5920.0 4930.0 1.75 480.0 -185.0 -0.14 1.1374 0.6478 3123012 ChemDiv3_010005 COc1ccc(cc1)N2Cc3cccc(C(=O)NCCc4cccc(C)c4)c3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G18 compound treatment 400.0 -586.0 -0.21 960.0 295.0 0.23 0.0133 0.0434 3123013 ChemDiv3_010006 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G19 compound treatment 560.0 -426.0 -0.15 320.0 -345.0 -0.26 -0.2939 -0.9648 3031856 ChemDiv3_010007 COc1ccc(CNC(=O)C2C(Oc3ccc(Cl)cc3Cl)C(=O)N2c4cccc(C)c4C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G20 compound treatment 440.0 -546.0 -0.19 1920.0 1260.0 0.96 0.5445 0.5539 3123014 ChemDiv3_010008 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)N4CCN(CC4)c5ccccn5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G21 compound treatment 1840.0 854.0 0.3 1000.0 335.0 0.26 0.3963 0.9967 3123015 ChemDiv3_010009 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NC(Cc3ccccc3)C(=O)NCc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G22 compound treatment 7840.0 6850.0 2.43 720.0 55.5 0.04 1.7493 0.7194 3031859 ChemDiv3_010010 CN1CCN(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G23 mock treatment 1120.0 134.0 0.05 720.0 55.5 0.04 0.0637 0.9986 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 G24 mock treatment 2920.0 1930.0 0.69 320.0 -345.0 -0.26 0.298 0.4054 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H01 compound treatment 640.0 -346.0 -0.12 1560.0 895.0 0.69 0.3993 0.5717 3123016 ChemDiv3_010011 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N(C)c4cc(Cl)ccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H02 compound treatment 2160.0 1170.0 0.42 400.0 -265.0 -0.2 0.1508 0.3256 3031861 ChemDiv3_010012 Fc1ccc(CSc2nc3c4ccccc4sc3c(=O)n2CCC(=O)NCC5CCCO5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H03 compound treatment 640.0 -346.0 -0.12 480.0 -185.0 -0.14 -0.187 -0.9975 3123017 ChemDiv3_010013 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCC(OC)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H04 compound treatment 680.0 -306.0 -0.11 2200.0 1540.0 1.18 0.7567 0.6392 3031863 ChemDiv3_010014 CC(=O)OCC(=O)c1ccc2ccn(C(=O)C)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H05 compound treatment 640.0 -346.0 -0.12 1720.0 1060.0 0.81 0.4861 0.5931 3123018 ChemDiv3_010015 CCc1ccc(NC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H06 compound treatment 1960.0 974.0 0.35 400.0 -265.0 -0.2 0.1007 0.2512 3123019 ChemDiv3_010016 CCOC(=O)N1CCN(CC(O)c2ccc3NCCc3c2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H07 compound treatment 1600.0 614.0 0.22 1360.0 695.0 0.53 0.5315 0.9218 3031866 ChemDiv3_010017 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)Nc4ccc5c(C)cc(=O)oc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H08 compound treatment 3480.0 2490.0 0.88 2720.0 2060.0 1.58 1.7414 0.9626 3123020 ChemDiv3_010018 CCC(=O)NC(C)C(N1CCN(CC1)c2ccccc2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H09 compound treatment 920.0 -66.3 -0.02 480.0 -185.0 -0.14 -0.1168 -0.8133 3031868 ChemDiv3_010019 Cc1ccc(NC(=O)Cn2nnc(c2N)S(=O)(=O)c3ccc(cc3)C(C)(C)C)c(C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H10 compound treatment 680.0 -306.0 -0.11 880.0 215.0 0.17 0.0402 0.2029 3123021 ChemDiv3_010020 COC(=O)CSc1nc(C)nc2n(C)c(=O)n(C)c(=O)c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H11 compound treatment 3440.0 2450.0 0.87 680.0 15.5 0.01 0.6239 0.7167 3123022 ChemDiv3_010021 CN(CC(=O)Nc1ccc(F)cc1F)S(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H12 compound treatment 1160.0 174.0 0.06 360.0 -305.0 -0.23 -0.1217 -0.5035 3031923 ChemDiv3_010022 COC(=O)c1ccc(CSc2nc(nc3n(C)c(=O)n(C)c(=O)c23)c4cccs4)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H13 compound treatment 600.0 -386.0 -0.14 2880.0 2220.0 1.7 1.1058 0.648 3031924 ChemDiv3_010023 OC(=O)CSc1c2CCCCc2nc3cc(ccc13)C(=O)NCc4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H14 compound treatment 4560.0 3570.0 1.27 480.0 -185.0 -0.14 0.7963 0.6242 3031926 ChemDiv3_010024 O=C(N1CCOCC1)c2ccc3C(=O)N(Cc4ccco4)C(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H15 compound treatment 720.0 -266.0 -0.09 1040.0 375.0 0.29 0.137 0.4518 3031927 ChemDiv3_010025 CC(C)NC(=O)c1ccc2c(Cl)c3CCCCc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H16 compound treatment 520.0 -466.0 -0.17 400.0 -265.0 -0.2 -0.2606 -0.9948 3031928 ChemDiv3_010026 COc1cc(OC)c(NC2N(Cc3cccs3)C(=O)c4cccnc24)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H17 compound treatment 960.0 -26.3 -0.01 760.0 95.5 0.07 0.0452 0.6124 3031930 ChemDiv3_010027 Clc1c2CCCCc2nc3cc(ccc13)C(=O)NCCN4CCN(Cc5ccccc5)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H18 compound treatment 1800.0 814.0 0.29 520.0 -145.0 -0.11 0.1257 0.4064 3123023 ChemDiv3_010028 CC(C)NC(=S)N1CCN(CC1)c2ccc(nn2)N3CCOCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H19 compound treatment 8200.0 7210.0 2.56 1200.0 535.0 0.41 2.1002 0.8103 3031931 ChemDiv3_010029 CC(C)N(Cc1nc(no1)c2ccccc2)C(=O)CCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H20 compound treatment 1200.0 214.0 0.08 1280.0 615.0 0.47 0.3877 0.8102 3123024 ChemDiv3_010030 COC(=O)c1c(N)onc1c2ccc(Br)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H21 compound treatment 360.0 -626.0 -0.22 3000.0 2340.0 1.79 1.1107 0.6148 3031933 ChemDiv3_010031 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N(C)CCC#N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H22 compound treatment 840.0 -146.0 -0.05 400.0 -265.0 -0.2 -0.1803 -0.8601 3123202 ChemDiv3_010032 COc1cc(NC2N(C(=O)c3ccccc23)c4cc(C)ccn4)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H23 mock treatment 520.0 -466.0 -0.17 280.0 -385.0 -0.3 -0.3257 -0.9625 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 H24 mock treatment 320.0 -666.0 -0.24 640.0 -24.5 -0.02 -0.1804 -0.761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I01 compound treatment 240.0 -746.0 -0.26 320.0 -345.0 -0.26 -0.3742 -1.0 3123203 ChemDiv3_010033 CCCN(C(=O)COc1cc(=O)n(C)c2ccccc12)c3ccccc3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I02 compound treatment 320.0 -666.0 -0.24 2360.0 1700.0 1.3 0.7533 0.5694 3031936 ChemDiv3_010034 CCn1c(=O)cc(SCC(=O)NCc2cccs2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I03 compound treatment 400.0 -586.0 -0.21 440.0 -225.0 -0.17 -0.2689 -0.9956 3123204 ChemDiv3_010035 CCn1c(=O)cc(OCC(=O)N2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I04 compound treatment 440.0 -546.0 -0.19 280.0 -385.0 -0.3 -0.3458 -0.9792 3031938 ChemDiv3_010036 COc1ccc2oc(=O)c(cc2c1)S(=O)(=O)c3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I05 compound treatment 240.0 -746.0 -0.26 520.0 -145.0 -0.11 -0.2656 -0.9255 3123205 ChemDiv3_010037 CCOc1ccc(CNC(=O)COc2cc(=O)n(CC)c3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I06 compound treatment 240.0 -746.0 -0.26 280.0 -385.0 -0.3 -0.3959 -0.9985 3031940 ChemDiv3_010038 CCC1CCCCN1CCCNC(=O)c2cc3CSCc3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I07 compound treatment 1640.0 654.0 0.23 480.0 -185.0 -0.14 0.0638 0.2349 3123206 ChemDiv3_010039 Fc1ccccc1N2CCN(CCNC(=O)C3CCCN(C3)S(=O)(=O)c4c[nH]cn4)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I08 compound treatment 360.0 -626.0 -0.22 280.0 -385.0 -0.3 -0.3658 -0.9902 1469954 ChemDiv3_010040 NCCC1(CC2CC3C1)CC(C2)(C3)C(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I09 compound treatment 1120.0 134.0 0.05 1200.0 535.0 0.41 0.3242 0.7835 3123207 ChemDiv3_010041 CC1Cc2ccccc2N1C(=O)C3CCCN3S(=O)(=O)c4cccc5nsnc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I10 compound treatment 2000.0 1010.0 0.36 320.0 -345.0 -0.26 0.0673 0.1507 3031944 ChemDiv3_010042 COc1ccc(cc1)c2cc([nH]n2)C(=O)N3CCC4(CC3)OCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I11 compound treatment 560.0 -426.0 -0.15 440.0 -225.0 -0.17 -0.2288 -0.9979 3123208 ChemDiv3_010043 O=C(NCCc1ccccc1)[C@H](N2Cc3ccccc3C2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I12 compound treatment 400.0 -586.0 -0.21 320.0 -345.0 -0.26 -0.3341 -0.9929 3031945 ChemDiv3_010044 Cn1c(SCC(=O)NCc2ccco2)nnc1c3c[nH]c4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I13 compound treatment 1720.0 734.0 0.26 440.0 -225.0 -0.17 0.0622 0.1992 3123209 ChemDiv3_010045 O=C(NC1CCCC1)[C@H](CSCc2ccccc2)N3Cc4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I14 compound treatment 360.0 -626.0 -0.22 400.0 -265.0 -0.2 -0.3007 -0.999 3031947 ChemDiv3_010046 CCSc1nnc(c2c[nH]c3ccccc23)n1CCOC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I15 compound treatment 360.0 -626.0 -0.22 320.0 -345.0 -0.26 -0.3441 -0.9962 3123210 ChemDiv3_010047 Cc1nc2cc(nn2c(C)c1CCC(=O)N3CCCC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I16 compound treatment 320.0 -666.0 -0.24 280.0 -385.0 -0.3 -0.3759 -0.9939 3123211 ChemDiv3_010048 Clc1nc2ccccc2c3sc(cc13)C(=O)N4CCC5(CC4)OCCO5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I17 compound treatment 400.0 -586.0 -0.21 480.0 -185.0 -0.14 -0.2472 -0.9825 3031949 ChemDiv3_010049 COc1ccc(c2cc3nc(C)c(CCC(=O)NCc4ccc5OCOc5c4)c(C)n3n2)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I18 compound treatment 400.0 -586.0 -0.21 3200.0 2540.0 1.95 1.2294 0.628 3123212 ChemDiv3_010050 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)Nc4cnc5ccccc5c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I19 compound treatment 400.0 -586.0 -0.21 800.0 135.0 0.1 -0.0735 -0.3161 3030807 ChemDiv3_010051 Cc1nn(c2ccc(C)c(C)c2)c3nc(C)c(CCC(=O)NCC4CCN(C4)C5CCCC5)c(C)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I20 compound treatment 360.0 -626.0 -0.22 840.0 175.0 0.13 -0.0618 -0.238 3030808 ChemDiv3_010052 CC1CCN(CCCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I21 compound treatment 400.0 -586.0 -0.21 480.0 -185.0 -0.14 -0.2472 -0.9825 3030810 ChemDiv3_010053 COc1ccc(NC(=O)C(NS(=O)(=O)c2ccc3n(C)c(=O)oc3c2)C(C)C)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I22 compound treatment 320.0 -666.0 -0.24 1000.0 335.0 0.26 0.015 0.0429 3030811 ChemDiv3_010054 CCC(C)NC(=O)c1cc2c(=O)n(CC)c3ccccc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I23 mock treatment 840.0 -146.0 -0.05 360.0 -305.0 -0.23 -0.202 -0.8435 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 I24 mock treatment 240.0 -746.0 -0.26 320.0 -345.0 -0.26 -0.3742 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J01 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3030813 ChemDiv3_010055 CCN(C(=O)c1cc2c(=O)n(CC)c3ccccc3c2s1)c4ccc(CC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J02 compound treatment 240.0 -746.0 -0.26 280.0 -385.0 -0.3 -0.3959 -0.9985 3123213 ChemDiv3_010056 FC(F)(F)c1nc2ccccc2n(CC(=O)N3CCc4ccccc34)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J03 compound treatment 360.0 -626.0 -0.22 480.0 -185.0 -0.14 -0.2573 -0.9764 3030815 ChemDiv3_010057 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N(Cc4ccccc4)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J04 compound treatment 400.0 -586.0 -0.21 400.0 -265.0 -0.2 -0.2907 -0.9999 3123214 ChemDiv3_010058 O=C(CCn1c(=S)oc2ccccc12)N3CCn4c(C3)nc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J05 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3123215 ChemDiv3_010059 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J06 compound treatment 480.0 -506.0 -0.18 240.0 -425.0 -0.33 -0.3574 -0.9606 3030817 ChemDiv3_010060 CCOC(=O)N1CCN(CC(O)c2ccc3N(CCc3c2)C(=O)C)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J07 compound treatment 520.0 -466.0 -0.17 240.0 -425.0 -0.33 -0.3474 -0.9506 3123216 ChemDiv3_010061 CC1CCCCN1CCNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J08 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3123217 ChemDiv3_010062 CC(NC(=O)c1ccncc1)C(N2CCN(Cc3ccccc3)CC2)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J09 compound treatment 360.0 -626.0 -0.22 440.0 -225.0 -0.17 -0.279 -0.9921 3030820 ChemDiv3_010063 CCCN1C(O)c2ccc(cc2C1=O)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J10 compound treatment 400.0 -586.0 -0.21 280.0 -385.0 -0.3 -0.3558 -0.9853 3123218 ChemDiv3_010064 COc1ccc(cc1)c2nc(SCC(=O)N)c3c(=O)n(C)c(=O)n(C)c3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J11 compound treatment 360.0 -626.0 -0.22 480.0 -185.0 -0.14 -0.2573 -0.9764 3030822 ChemDiv3_010065 CCOC(=O)N1CCN(CC1)C(=O)CN(C)S(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J12 compound treatment 160.0 -826.0 -0.29 160.0 -505.0 -0.39 -0.4811 -0.9905 3123219 ChemDiv3_010066 Cc1[nH]c(nc1C(=O)O)c2ccc3OCOc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J13 compound treatment 2800.0 1810.0 0.64 360.0 -305.0 -0.23 0.2897 0.4231 3123220 ChemDiv3_010067 COc1ccc(CCNC(=O)c2ccc3c(SCC(=O)O)c4CCCCc4nc3c2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J14 compound treatment 520.0 -466.0 -0.17 320.0 -345.0 -0.26 -0.304 -0.9744 3030825 ChemDiv3_010068 O=C1N(Cc2ccccc2)Cc3ccncc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J15 compound treatment 360.0 -626.0 -0.22 320.0 -345.0 -0.26 -0.3441 -0.9962 3030826 ChemDiv3_010069 Clc1c2CCCCc2nc3cc(ccc13)C(=O)NCC4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J16 compound treatment 320.0 -666.0 -0.24 720.0 55.5 0.04 -0.137 -0.5705 3123221 ChemDiv3_010070 OCc1nccnc1C(=O)Nc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J17 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3123222 ChemDiv3_010071 Clc1ccccc1CNC(=O)c2ccc3c(Cl)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J18 compound treatment 680.0 -306.0 -0.11 400.0 -265.0 -0.2 -0.2204 -0.957 3030830 ChemDiv3_010072 Clc1ccc(nn1)N2CCN(CC2)C(=O)c3cc4ccccn4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J19 compound treatment 360.0 -626.0 -0.22 480.0 -185.0 -0.14 -0.2573 -0.9764 3123223 ChemDiv3_010073 CC(C)N(Cc1nc(no1)c2ccc(C)cc2)C(=O)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J20 compound treatment 360.0 -626.0 -0.22 1080.0 415.0 0.32 0.0685 0.1761 1113344 ChemDiv3_010074 Clc1ccc(cc1)N2C(=O)c3ccccc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J21 compound treatment 320.0 -666.0 -0.24 1040.0 375.0 0.29 0.0367 0.0985 3123224 ChemDiv3_010075 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J22 compound treatment 440.0 -546.0 -0.19 320.0 -345.0 -0.26 -0.324 -0.9883 3030833 ChemDiv3_010076 COc1ccc(Cn2c(CCC(=O)NCc3ccccc3)nc4cccnc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J23 mock treatment 400.0 -586.0 -0.21 320.0 -345.0 -0.26 -0.3341 -0.9929 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 J24 mock treatment 440.0 -546.0 -0.19 600.0 -64.5 -0.05 -0.172 -0.8602 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K01 compound treatment 440.0 -546.0 -0.19 520.0 -145.0 -0.11 -0.2155 -0.965 3123225 ChemDiv3_010077 Cn1c(=O)cc(OCC(=O)NC2CCN(Cc3ccccc3)CC2)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K02 compound treatment 720.0 -266.0 -0.09 440.0 -225.0 -0.17 -0.1887 -0.9599 3030888 ChemDiv3_010078 CCn1c(=O)cc(SCC(=O)NC2CCCc3ccccc23)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K03 compound treatment 640.0 -346.0 -0.12 480.0 -185.0 -0.14 -0.187 -0.9975 3030889 ChemDiv3_010079 CCn1c(=O)cc(OCC(=O)N2CCCCC2C)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K04 compound treatment 1120.0 134.0 0.05 5760.0 5100.0 3.91 2.7997 0.7156 3030890 ChemDiv3_010080 COc1cccc2cc(c(=O)oc12)S(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K05 compound treatment 520.0 -466.0 -0.17 600.0 -64.5 -0.05 -0.152 -0.8802 3030892 ChemDiv3_010081 Cn1c(=O)cc(OCCCC(=O)NC2CCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K06 compound treatment 440.0 -546.0 -0.19 1080.0 415.0 0.32 0.0885 0.2372 3030893 ChemDiv3_010082 Fc1ccc(cc1)c2cc(COCC(=O)Nc3ccc(F)cc3F)no2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K07 compound treatment 6520.0 5530.0 1.96 520.0 -145.0 -0.11 1.3097 0.6661 3030895 ChemDiv3_010083 CC(C)C(NS(=O)(=O)c1cccc2nsnc12)C(=O)N3CCN(C(C)C3)c4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K08 compound treatment 560.0 -426.0 -0.15 480.0 -185.0 -0.14 -0.2071 -0.9995 3123226 ChemDiv3_010084 O=C1CCCN1CC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K09 compound treatment 640.0 -346.0 -0.12 1160.0 495.0 0.38 0.1821 0.4556 3030897 ChemDiv3_010085 CC(=O)Nc1ccc(NC(=O)C2CCCN2S(=O)(=O)c3cccc4nsnc34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K10 compound treatment 520.0 -466.0 -0.17 400.0 -265.0 -0.2 -0.2606 -0.9948 3123227 ChemDiv3_010086 COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)c3cc(n[nH]3)c4ccccc4OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K11 compound treatment 680.0 -306.0 -0.11 1440.0 775.0 0.6 0.3442 0.5687 3123228 ChemDiv3_010087 O=C([C@H](N1Cc2ccccc2C1=O)c3ccccc3)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K12 compound treatment 960.0 -26.3 -0.01 480.0 -185.0 -0.14 -0.1068 -0.752 3030900 ChemDiv3_010088 Cc1cccc(CSc2nnc(c3c[nH]c4ccccc34)n2C)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K13 compound treatment 3160.0 2170.0 0.77 960.0 295.0 0.23 0.7057 0.8779 3123229 ChemDiv3_010089 COc1ccccc1NC(=O)[C@H](CSCc2ccccc2)N3Cc4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K14 compound treatment 6920.0 5930.0 2.1 480.0 -185.0 -0.14 1.3883 0.658 3030901 ChemDiv3_010090 CCSc1nnc(c2c[nH]c3ccccc23)n1c4cccc(OC)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K15 compound treatment 3920.0 2930.0 1.04 520.0 -145.0 -0.11 0.6575 0.6282 3123406 ChemDiv3_010091 CCOC(=O)N1CCC(CC1)NC(=O)CCc2c(C)nc3c(c(C)nn3c2C)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K16 compound treatment 880.0 -106.0 -0.04 680.0 15.5 0.01 -0.0182 -0.4617 3030904 ChemDiv3_010092 Clc1nc2ccccc2c3sc(cc13)C(=O)NCCCN4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K17 compound treatment 1440.0 454.0 0.16 4520.0 3860.0 2.96 2.2068 0.7445 3123407 ChemDiv3_010093 COc1ccc(c2cc3nc(C)c(CCC(=O)NC(C)c4cccs4)c(C)n3n2)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K18 compound treatment 1160.0 174.0 0.06 480.0 -185.0 -0.14 -0.0566 -0.3663 3123408 ChemDiv3_010094 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K19 compound treatment 560.0 -426.0 -0.15 1480.0 815.0 0.63 0.3358 0.5213 3030907 ChemDiv3_010095 Cc1nn(c2ccccc2)c3nc(cc(C)c13)C(=O)NN4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K20 compound treatment 840.0 -146.0 -0.05 400.0 -265.0 -0.2 -0.1803 -0.8601 3123409 ChemDiv3_010096 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)NCCc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K21 compound treatment 800.0 -186.0 -0.07 680.0 15.5 0.01 -0.0383 -0.5707 3030909 ChemDiv3_010097 Cc1ccc(C)c(c1)N2CCN(CC2)S(=O)(=O)c3ccc4N(CCc4c3)C(=O)CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K22 compound treatment 1360.0 374.0 0.13 400.0 -265.0 -0.2 -0.0498 -0.2055 3123410 ChemDiv3_010098 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCC4CCCO4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K23 mock treatment 760.0 -226.0 -0.08 440.0 -225.0 -0.17 -0.1786 -0.9395 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 K24 mock treatment 2400.0 1410.0 0.5 1400.0 735.0 0.56 0.7539 0.9983 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L01 compound treatment 1680.0 694.0 0.25 760.0 95.5 0.07 0.2259 0.8795 3123411 ChemDiv3_010099 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N(C)c4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L02 compound treatment 560.0 -426.0 -0.15 400.0 -265.0 -0.2 -0.2505 -0.9895 3030911 ChemDiv3_010100 FC(F)(F)c1nc2ccccc2n(CC(=O)N3CCc4ccccc4C3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L03 compound treatment 920.0 -66.3 -0.02 2040.0 1380.0 1.06 0.7301 0.6912 3123412 ChemDiv3_010101 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N(C)Cc4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L04 compound treatment 320.0 -666.0 -0.24 4960.0 4300.0 3.3 2.1647 0.6547 3030913 ChemDiv3_010102 CC(=O)OCC(=O)c1ccc2N(CCc2c1)C(=O)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L05 compound treatment 800.0 -186.0 -0.07 480.0 -185.0 -0.14 -0.1469 -0.9397 3123413 ChemDiv3_010103 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)N(CC=C)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L06 compound treatment 320.0 -666.0 -0.24 4800.0 4140.0 3.17 2.0779 0.6527 3030974 ChemDiv3_010104 CC1CCCCN1S(=O)(=O)c2ccc3n(C)c(=O)oc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L07 compound treatment 1480.0 494.0 0.18 360.0 -305.0 -0.23 -0.0415 -0.1419 3123414 ChemDiv3_010105 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)N(Cc4ccco4)C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L08 compound treatment 800.0 -186.0 -0.07 600.0 -64.5 -0.05 -0.0817 -0.9899 3123415 ChemDiv3_010106 COc1ccc(cc1OC)C(=O)NC(C)C(N2CCN(CC2)c3ccccc3F)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L09 compound treatment 480.0 -506.0 -0.18 720.0 55.5 0.04 -0.0969 -0.5248 3030976 ChemDiv3_010107 CCCN1C(O)c2ccc(cc2C1=O)C(=O)NCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L10 compound treatment 600.0 -386.0 -0.14 520.0 -145.0 -0.11 -0.1753 -0.9945 3123416 ChemDiv3_010108 CCOC(=O)C(C)Sc1nc(nc2n(C)c(=O)n(C)c(=O)c12)c3ccc(OC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L11 compound treatment 560.0 -426.0 -0.15 560.0 -105.0 -0.08 -0.1637 -0.9561 3030977 ChemDiv3_010109 CN(CC(=O)NCc1ccccc1)S(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L12 compound treatment 600.0 -386.0 -0.14 360.0 -305.0 -0.23 -0.2622 -0.9676 3123417 ChemDiv3_010110 O=C1N(Cc2ccccc2)C(Nc3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L13 compound treatment 920.0 -66.3 -0.02 520.0 -145.0 -0.11 -0.0951 -0.8383 3123418 ChemDiv3_010111 OC(=O)CSc1c2CCCCc2nc3cc(ccc13)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L14 compound treatment 3840.0 2850.0 1.01 600.0 -64.5 -0.05 0.6808 0.6717 3030979 ChemDiv3_010112 Cc1cc(NC2N(C3CCCCC3)C(=O)c4cccnc24)ccc1Br 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L15 compound treatment 480.0 -506.0 -0.18 3600.0 2940.0 2.25 1.4666 0.6487 3123419 ChemDiv3_010113 Clc1c2CCCCc2nc3cc(ccc13)C(=O)NCCCN4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L16 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3030982 ChemDiv3_010114 CCc1ccc(cc1)N2C(=O)c3ccncc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L17 compound treatment 760.0 -226.0 -0.08 1200.0 535.0 0.41 0.2339 0.5585 3123420 ChemDiv3_010115 CCCN(CCC)C(=O)c1ccc2c(Cl)c3CCCCc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L18 compound treatment 5240.0 4250.0 1.51 600.0 -64.5 -0.05 1.032 0.6835 3030984 ChemDiv3_010116 Cc1cccc(c1)C(=O)N2CCN(CC2)c3ccc(nn3)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L19 compound treatment 920.0 -66.3 -0.02 480.0 -185.0 -0.14 -0.1168 -0.8133 3123421 ChemDiv3_010117 CC(C)N(Cc1nc(no1)c2ccccc2)C(=O)C(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L20 compound treatment 1640.0 654.0 0.23 1320.0 655.0 0.5 0.5198 0.9381 3123422 ChemDiv3_010118 COc1ccc(NC2N(C(=O)c3ccccc23)c4ccc(Cl)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L21 compound treatment 1200.0 214.0 0.08 1680.0 1020.0 0.78 0.6049 0.7722 3030986 ChemDiv3_010119 CCCNS(=O)(=O)c1ccc2n(CC(=O)OCC)c(=O)oc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L22 compound treatment 480.0 -506.0 -0.18 4440.0 3780.0 2.9 1.9226 0.662 3123423 ChemDiv3_010120 Cc1[nH]c2ccccc2c1C3=CCN(CC3)S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L23 mock treatment 360.0 -626.0 -0.22 520.0 -145.0 -0.11 -0.2355 -0.9485 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 L24 mock treatment 680.0 -306.0 -0.11 1400.0 735.0 0.56 0.3224 0.5608 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M01 compound treatment 920.0 -66.3 -0.02 320.0 -345.0 -0.26 -0.2036 -0.7669 3030988 ChemDiv3_010121 CCc1cccc(NC(=O)COc2cc(=O)n(C)c3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M02 compound treatment 560.0 -426.0 -0.15 1640.0 975.0 0.75 0.4226 0.5532 3123424 ChemDiv3_010122 CCn1c(=O)cc(SCC(=O)NCC2(CCCC2)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M03 compound treatment 15440.0 14500.0 5.13 600.0 -64.5 -0.05 3.5906 0.7002 3030991 ChemDiv3_010123 CCn1c(=O)cc(OCC(=O)NCCCN2CCOCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M04 compound treatment 920.0 -66.3 -0.02 480.0 -185.0 -0.14 -0.1168 -0.8133 3123425 ChemDiv3_010124 COc1ccc(OC)c(c1)S(=O)(=O)c2cc3ccccc3oc2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M05 compound treatment 1040.0 53.8 0.02 280.0 -385.0 -0.3 -0.1953 -0.6601 3123426 ChemDiv3_010125 Cn1c(=O)cc(OCCCC(=O)N2CCCCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M06 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3031061 ChemDiv3_010126 Fc1ccc(cc1)c2cc(COCC(=O)NCC3CCCO3)no2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M07 compound treatment 920.0 -66.3 -0.02 680.0 15.5 0.01 -0.0082 -0.3118 3031062 ChemDiv3_010127 CC(C)C(NS(=O)(=O)c1cccc2nsnc12)C(=O)Nc3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M08 compound treatment 760.0 -226.0 -0.08 440.0 -225.0 -0.17 -0.1786 -0.9395 3031063 ChemDiv3_010128 O=C1CCCN1CCC2(CC3CC4CC(C3)C2)C4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M09 compound treatment 760.0 -226.0 -0.08 760.0 95.5 0.07 -0.0049 -0.0453 3031064 ChemDiv3_010129 CCCN(C(=O)C1CCCN1S(=O)(=O)c2cccc3nsnc23)c4ccc(cc4)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M10 compound treatment 920.0 -66.3 -0.02 720.0 55.5 0.04 0.0135 0.2775 3031066 ChemDiv3_010130 COc1cccc(c1)c2cc([nH]n2)C(=O)NC3CC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M11 compound treatment 600.0 -386.0 -0.14 640.0 -24.5 -0.02 -0.1102 -0.7968 3031067 ChemDiv3_010131 Fc1cccc(NC(=O)[C@H](Cc2ccccc2)N3Cc4ccccc4C3=O)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M12 compound treatment 680.0 -306.0 -0.11 1000.0 335.0 0.26 0.1053 0.3767 3123427 ChemDiv3_010132 COC(=O)c1ccc(CSc2nnc(c3c[nH]c4ccccc34)n2C)o1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M13 compound treatment 840.0 -146.0 -0.05 840.0 175.0 0.13 0.0586 0.4058 3031069 ChemDiv3_010133 Fc1ccc(CNC(=O)[C@H](CSCc2ccccc2)N3Cc4ccccc4C3=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M14 compound treatment 560.0 -426.0 -0.15 920.0 255.0 0.2 0.0318 0.1283 3123428 ChemDiv3_010134 COC(=O)C(C)Sc1nnc(c2c[nH]c3ccccc23)n1c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M15 compound treatment 1880.0 894.0 0.32 3680.0 3020.0 2.32 1.8612 0.7965 3123429 ChemDiv3_010135 CN(C(=O)CCc1c(C)nc2c(c(C)nn2c1C)c3ccc(F)cc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M16 compound treatment 640.0 -346.0 -0.12 920.0 255.0 0.2 0.0518 0.224 3031072 ChemDiv3_010136 CN(C(=O)c1cc2c(Cl)nc3ccccc3c2s1)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M17 compound treatment 1080.0 93.8 0.03 440.0 -225.0 -0.17 -0.0984 -0.5603 3123430 ChemDiv3_010137 COc1ccc(c2cc3nc(C)c(CCC(=O)Nc4ccccc4C(=O)N)c(C)n3n2)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M18 compound treatment 760.0 -226.0 -0.08 1400.0 735.0 0.56 0.3425 0.6006 3031073 ChemDiv3_010138 CCN1CCCC1CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M19 compound treatment 960.0 -26.3 -0.01 840.0 175.0 0.13 0.0887 0.6567 3123431 ChemDiv3_010139 CCOC(=O)C1=C(CN2CCc3ccccc23)NC(=O)NC1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M20 compound treatment 920.0 -66.3 -0.02 800.0 135.0 0.1 0.0569 0.5339 3031076 ChemDiv3_010140 Cn1c(cc2c(=O)n(C)c3ccccc3c12)C(=O)NC4CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M21 compound treatment 1160.0 174.0 0.06 520.0 -145.0 -0.11 -0.0349 -0.2747 3123432 ChemDiv3_010141 COc1ccccc1NS(=O)(=O)c2ccc3N(CCc3c2)C(=O)CCC(=O)O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M22 compound treatment 1080.0 93.8 0.03 1720.0 1060.0 0.81 0.5965 0.7355 3120367 ChemDiv3_010142 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCCN(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M23 mock treatment 520.0 -466.0 -0.17 1040.0 375.0 0.29 0.0869 0.2614 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 M24 mock treatment 840.0 -146.0 -0.05 4400.0 3740.0 2.87 1.9912 0.6942 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N01 compound treatment 400.0 -586.0 -0.21 800.0 135.0 0.1 -0.0735 -0.3161 3031078 ChemDiv3_010143 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N02 compound treatment 2360.0 1370.0 0.49 760.0 95.5 0.07 0.3964 0.8044 3120368 ChemDiv3_010144 FC(F)(F)c1nc2ccccc2n(CC(=O)NCc3ccccc3)c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N03 compound treatment 2160.0 1170.0 0.42 400.0 -265.0 -0.2 0.1508 0.3256 3031080 ChemDiv3_010145 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NCCc4ccsc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N04 compound treatment 9360.0 8370.0 2.97 2280.0 1620.0 1.24 2.9775 0.925 3030865 ChemDiv3_010146 S=C(NCc1ccccc1)N2CCn3c(C2)nc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N05 compound treatment 4760.0 3770.0 1.34 400.0 -265.0 -0.2 0.803 0.5931 3030868 ChemDiv3_010147 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)NCc4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N06 compound treatment 680.0 -306.0 -0.11 400.0 -265.0 -0.2 -0.2204 -0.957 3030932 ChemDiv3_010148 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NCc3ccco3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N07 compound treatment 440.0 -546.0 -0.19 560.0 -105.0 -0.08 -0.1938 -0.9238 3030934 ChemDiv3_010149 CCCCN(Cc1ccco1)C(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N08 compound treatment 680.0 -306.0 -0.11 480.0 -185.0 -0.14 -0.177 -0.9914 3030937 ChemDiv3_010150 COc1ccc(cc1)N2CCN(CC2)C(C(C)NC(=O)c3ccccc3OC)c4cccs4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N09 compound treatment 640.0 -346.0 -0.12 400.0 -265.0 -0.2 -0.2304 -0.971 3030939 ChemDiv3_010151 CC1CCCN(C1)C(=O)C(Cc2ccccc2)NS(=O)(=O)c3ccc4NC(=O)CCc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N10 compound treatment 600.0 -386.0 -0.14 720.0 55.5 0.04 -0.0668 -0.4653 3030941 ChemDiv3_010152 CCOC(=O)C(C)(C)Sc1nc(nc2n(C)c(=O)n(C)c(=O)c12)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N11 compound treatment 720.0 -266.0 -0.09 480.0 -185.0 -0.14 -0.167 -0.9806 3030943 ChemDiv3_010153 OC(=O)CSc1c2CCCCc2nc3cc(ccc13)C(=O)Nc4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N12 compound treatment 560.0 -426.0 -0.15 440.0 -225.0 -0.17 -0.2288 -0.9979 3120369 ChemDiv3_010154 CCN(CC)S(=O)(=O)c1ccc(NC2N(Cc3ccccc3)C(=O)c4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N13 compound treatment 720.0 -266.0 -0.09 1160.0 495.0 0.38 0.2022 0.5159 3120370 ChemDiv3_010155 Clc1c2CCCCc2nc3cc(ccc13)C(=O)NC4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N14 compound treatment 440.0 -546.0 -0.19 800.0 135.0 0.1 -0.0635 -0.2886 1681444 ChemDiv3_010156 Cc1ccc(NC(=O)c2nccnc2C(=O)O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N15 compound treatment 600.0 -386.0 -0.14 1320.0 655.0 0.5 0.2589 0.4965 3120371 ChemDiv3_010157 CN(C(=O)c1ccc2c(Cl)c3CCCCc3nc2c1)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N16 compound treatment 720.0 -266.0 -0.09 520.0 -145.0 -0.11 -0.1452 -0.9968 1027433 ChemDiv3_010158 OC(=O)c1ccnc(Cl)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N17 compound treatment 640.0 -346.0 -0.12 1040.0 375.0 0.29 0.117 0.3733 3030950 ChemDiv3_010159 COC(CNC(=O)c1ccc2c(Cl)c3CCCCc3nc2c1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N18 compound treatment 560.0 -426.0 -0.15 1280.0 615.0 0.47 0.2272 0.4579 3120372 ChemDiv3_010160 CC1CCN(CC1)c2cc(C)c3c(O)cccc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N19 compound treatment 800.0 -186.0 -0.07 840.0 175.0 0.13 0.0485 0.3235 3031012 ChemDiv3_010161 CC(C)N(Cc1nc(no1)c2cccc(C)c2)C(=O)/C=C/c3ccccc3Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N20 compound treatment 640.0 -346.0 -0.12 1120.0 455.0 0.35 0.1604 0.4328 3031014 ChemDiv3_010162 CCOC(=O)c1ccc(NC2CCCc3c2[nH]c4ccc(C)cc34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N21 compound treatment 1440.0 454.0 0.16 4040.0 3380.0 2.59 1.9462 0.7496 3031016 ChemDiv3_010163 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NCC3CCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N22 compound treatment 2320.0 1330.0 0.47 520.0 -145.0 -0.11 0.2561 0.527 3031018 ChemDiv3_010164 CCn1c(C)c(C2=CCN(CC2)S(=O)(=O)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N23 mock treatment 1760.0 774.0 0.27 1480.0 815.0 0.63 0.6368 0.9315 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 N24 mock treatment 1640.0 654.0 0.23 840.0 175.0 0.13 0.2593 0.9666 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O01 compound treatment 280.0 -706.0 -0.25 240.0 -425.0 -0.33 -0.4076 -0.9916 3031020 ChemDiv3_010165 CC(CCc1ccccc1)NC(=O)COc2cc(=O)n(C)c3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O02 compound treatment 2800.0 1810.0 0.64 320.0 -345.0 -0.26 0.2679 0.3852 3031023 ChemDiv3_010166 CCn1c(=O)cc(SCC(=O)NC2CCCC2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O03 compound treatment 480.0 -506.0 -0.18 400.0 -265.0 -0.2 -0.2706 -0.9981 3120373 ChemDiv3_010167 CCN(CC)C(=O)COc1cc(=O)n(CC)c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O04 compound treatment 480.0 -506.0 -0.18 360.0 -305.0 -0.23 -0.2923 -0.9915 3120374 ChemDiv3_010168 CCN(CC)c1ccc2cc(c(=O)oc2c1)S(=O)(=O)c3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O05 compound treatment 520.0 -466.0 -0.17 320.0 -345.0 -0.26 -0.304 -0.9744 3031029 ChemDiv3_010169 Cn1c(=O)cc(OCCCC(=O)NCC2(CCCC2)c3ccccc3)c4ccccc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O06 compound treatment 480.0 -506.0 -0.18 320.0 -345.0 -0.26 -0.314 -0.9822 3120375 ChemDiv3_010170 Fc1ccc(cc1)c2cc(COCC(=O)NCc3cccs3)no2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O07 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3120376 ChemDiv3_010171 CC(C)C(NS(=O)(=O)c1cccc2nsnc12)C(=O)NC3CCCC(C)C3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O08 compound treatment 440.0 -546.0 -0.19 320.0 -345.0 -0.26 -0.324 -0.9883 3031033 ChemDiv3_010172 Cc1ccc(cc1)c2cc3C(=O)CC(C)(C)Cc3n2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O09 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3120377 ChemDiv3_010173 CN(Cc1ccco1)C(=O)C2CCCN2S(=O)(=O)c3cccc4nsnc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O10 compound treatment 360.0 -626.0 -0.22 560.0 -105.0 -0.08 -0.2138 -0.9053 3031082 ChemDiv3_010174 COc1cccc(c1)c2cc([nH]n2)C(=O)N3CCN(CC3)c4cc(C)ccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O11 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3031084 ChemDiv3_010175 O=C([C@H](Cc1ccccc1)N2Cc3ccccc3C2=O)N4CCN(CC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O12 compound treatment 280.0 -706.0 -0.25 320.0 -345.0 -0.26 -0.3642 -0.9996 3031086 ChemDiv3_010176 CCC(Sc1nnc(c2c[nH]c3ccccc23)n1C)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O13 compound treatment 200.0 -786.0 -0.28 320.0 -345.0 -0.26 -0.3842 -0.9996 3031088 ChemDiv3_010177 O=C(NCc1ccco1)[C@H](Cc2ccccc2)N3Cc4ccccc4C3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O14 compound treatment 240.0 -746.0 -0.26 280.0 -385.0 -0.3 -0.3959 -0.9985 3031089 ChemDiv3_010178 CN(C1CCCCC1)C(=O)c2cc3c(Cl)nc4ccccc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O15 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3031092 ChemDiv3_010179 COc1ccc(NC(=O)CCc2c(C)nc3cc(nn3c2C)c4ccc(Cl)cc4)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O16 compound treatment 360.0 -626.0 -0.22 320.0 -345.0 -0.26 -0.3441 -0.9962 3120378 ChemDiv3_010180 Clc1nc2ccccc2c3sc(cc13)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O17 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3031095 ChemDiv3_010181 CN(C(=O)CCc1c(C)nc2ncnn2c1C)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O18 compound treatment 280.0 -706.0 -0.25 360.0 -305.0 -0.23 -0.3425 -0.9994 3120379 ChemDiv3_010182 COc1ccc(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O19 compound treatment 600.0 -386.0 -0.14 440.0 -225.0 -0.17 -0.2188 -0.9935 3031097 ChemDiv3_010183 CCOC(=O)C1=C(CNc2cccnc2)NC(=O)NC1c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O20 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3120380 ChemDiv3_010184 Cc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O21 compound treatment 280.0 -706.0 -0.25 480.0 -185.0 -0.14 -0.2773 -0.9636 3120381 ChemDiv3_010185 CCn1c(=O)cc(SCC(=O)N(C)Cc2ccccc2)c3ccccc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O22 compound treatment 520.0 -466.0 -0.17 320.0 -345.0 -0.26 -0.304 -0.9744 3031100 ChemDiv3_010186 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)N4CCN(Cc5ccccc5)CC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O23 mock treatment 400.0 -586.0 -0.21 200.0 -465.0 -0.36 -0.3992 -0.967 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 O24 mock treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P01 compound treatment 4840.0 3850.0 1.37 440.0 -225.0 -0.17 0.8448 0.6131 3120382 ChemDiv3_010187 CCn1c(=O)c2cc(sc2c3ccccc13)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P02 compound treatment 440.0 -546.0 -0.19 440.0 -225.0 -0.17 -0.2589 -0.9983 3120383 ChemDiv3_010188 O=S(=O)(N1CCn2c(C1)nc3ccccc23)c4ccc(cc4)C5CCCCC5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P03 compound treatment 360.0 -626.0 -0.22 360.0 -305.0 -0.23 -0.3224 -0.9997 3031256 ChemDiv3_010189 CC(C)NC(=O)c1cc2c(=O)oc3ccc(C)cc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P04 compound treatment 280.0 -706.0 -0.25 440.0 -225.0 -0.17 -0.299 -0.9833 3031258 ChemDiv3_010190 CC1CCC(CC1)NC(=O)c2oc(=O)c3ccccc3c2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P05 compound treatment 5720.0 4730.0 1.68 320.0 -345.0 -0.26 1.0004 0.5885 3031260 ChemDiv3_010191 Cc1ccc2oc(=O)c3cc(sc3c2c1)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P06 compound treatment 320.0 -666.0 -0.24 360.0 -305.0 -0.23 -0.3324 -1.0 3031261 ChemDiv3_010192 CCC(=O)NC(C)C(N1CCOCC1)c2cccs2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P07 compound treatment 320.0 -666.0 -0.24 320.0 -345.0 -0.26 -0.3541 -0.9984 3031263 ChemDiv3_010193 CCOc1ccc(CCNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P08 compound treatment 400.0 -586.0 -0.21 360.0 -305.0 -0.23 -0.3124 -0.9983 3031266 ChemDiv3_010194 CC(NS(=O)(=O)c1ccc(Cl)cc1)C(N2CCN(C)CC2)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P09 compound treatment 4400.0 3410.0 1.21 360.0 -305.0 -0.23 0.691 0.5603 3120384 ChemDiv3_010195 CCc1cccc(NC(=O)C(Cc2ccccc2)NS(=O)(=O)c3ccc4NC(=O)CCc4c3)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P10 compound treatment 1920.0 934.0 0.33 360.0 -305.0 -0.23 0.0689 0.17 3031270 ChemDiv3_010196 CC1CCN(CC1)C(=O)CSc2nc(nc3n(C)c(=O)n(C)c(=O)c23)c4ccco4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P11 compound treatment 400.0 -586.0 -0.21 400.0 -265.0 -0.2 -0.2907 -0.9999 3120385 ChemDiv3_010197 OC(=O)CSc1c2CCCCc2nc3cc(ccc13)C(=O)Nc4ccc(F)c(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P12 compound treatment 280.0 -706.0 -0.25 280.0 -385.0 -0.3 -0.3859 -0.9967 3031337 ChemDiv3_010198 Clc1cccc(c1)C(=O)OC2N(Cc3ccccc3)C(=O)c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P13 compound treatment 400.0 -586.0 -0.21 280.0 -385.0 -0.3 -0.3558 -0.9853 3031339 ChemDiv3_010199 CN(C1CCCCC1)C(=O)c2ccc3c(Cl)c4CCCCc4nc3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P14 compound treatment 240.0 -746.0 -0.26 280.0 -385.0 -0.3 -0.3959 -0.9985 3031340 ChemDiv3_010200 OC(=O)[C@H](Cc1ccccc1)N2C(=O)c3ccncc3C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P15 compound treatment 6160.0 5170.0 1.84 320.0 -345.0 -0.26 1.1108 0.599 3031342 ChemDiv3_010201 CC(C)CCNC(=O)c1ccc2c(Cl)c3CCCCc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P16 compound treatment 400.0 -586.0 -0.21 240.0 -425.0 -0.33 -0.3775 -0.9765 3031345 ChemDiv3_010202 COc1ccc(CNC(=O)OCc2nccnc2C(=O)Nc3ccc(Br)cn3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P17 compound treatment 4920.0 3930.0 1.4 240.0 -425.0 -0.33 0.7563 0.5278 3031346 ChemDiv3_010203 Clc1c2CCCCc2nc3cc(ccc13)C(=O)N4CCC(=CC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P18 compound treatment 4960.0 3970.0 1.41 320.0 -345.0 -0.26 0.8098 0.5646 3031348 ChemDiv3_010204 CN(Cc1ccccc1)c2cc(C)c3ccc(O)cc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P19 compound treatment 1840.0 854.0 0.3 360.0 -305.0 -0.23 0.0488 0.1277 3120386 ChemDiv3_010205 Cc1cccc(NC(=O)CSC2=NS(=O)(=O)c3ccccc23)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P20 compound treatment 2400.0 1410.0 0.5 1400.0 735.0 0.56 0.7539 0.9983 3120387 ChemDiv3_010206 CCOC(=O)c1ccc(NC2CCCc3c2n(C)c4ccc(C)cc34)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P21 compound treatment 280.0 -706.0 -0.25 2120.0 1460.0 1.12 0.613 0.5353 3031355 ChemDiv3_010207 CCOC(=O)Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NCc3cccc(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P22 compound treatment 680.0 -306.0 -0.11 520.0 -145.0 -0.11 -0.1553 -0.9999 3120388 ChemDiv3_010208 Cc1[nH]c2ccccc2c1C3=CCN(CC3)S(=O)(=O)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P23 mock treatment 960.0 -26.3 -0.01 480.0 -185.0 -0.14 -0.1068 -0.752 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2029 P24 mock treatment 360.0 -626.0 -0.22 320.0 -345.0 -0.26 -0.3441 -0.9962 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A01 compound treatment 240.0 -1040.0 -0.37 1720.0 1040.0 0.8 0.3035 0.3445 3031756 ChemDiv3_010209 COc1ccc(Cl)cc1NC(=O)c2cnn(c2C3CCNCC3)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A02 compound treatment 280.0 -1000.0 -0.36 3720.0 3040.0 2.33 1.3993 0.5924 3120389 ChemDiv3_010210 Cc1ccc(Cl)cc1N2CCN(CCCNC(=O)c3cc4c(C)nc5ccccc5c4o3)CC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A03 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3031821 ChemDiv3_010211 Cc1cccc(NC(=O)c2cnn(c2C3CCN(CC3)C(=O)OC(C)(C)C)c4ccc(F)cc4)c1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A04 compound treatment 280.0 -1000.0 -0.36 440.0 -239.0 -0.18 -0.3813 -0.9523 3120390 ChemDiv3_010212 COc1ccc(cc1)C2SC[C@@H]3N2C(=S)N(C3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A05 compound treatment 520.0 -764.0 -0.27 2440.0 1760.0 1.35 0.7646 0.5544 3031824 ChemDiv3_010213 O=C(CCc1nc2cccnc2n1c3ccccc3)NCCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A06 compound treatment 280.0 -1000.0 -0.36 8640.0 7960.0 6.11 4.0701 0.6648 3120391 ChemDiv3_010214 COC(=O)c1cc(=O)n(C2CCCCC2)/c(=N/C3CCCCC3)/s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A07 compound treatment 280.0 -1000.0 -0.36 480.0 -199.0 -0.15 -0.3596 -0.9284 3031828 ChemDiv3_010215 COC(CN(C)C(=O)c1cc2c(Cl)nc3ccc(C)cc3c2s1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A08 compound treatment 6080.0 4800.0 1.7 360.0 -319.0 -0.24 1.0301 0.5993 3120392 ChemDiv3_010216 Fc1ccc(cc1)C2SC[C@@H]3N2C(=O)N(C3=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A09 compound treatment 2800.0 1520.0 0.54 480.0 -199.0 -0.15 0.2725 0.4874 3120393 ChemDiv3_010217 CN(C(=O)CSc1c2CCCCc2nc3cc(Cl)ccc13)c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A10 compound treatment 1160.0 -124.0 -0.04 400.0 -279.0 -0.21 -0.1823 -0.8348 3031834 ChemDiv3_010218 FC(F)(F)c1ccccc1C(=O)Nc2cccc(c2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A11 compound treatment 360.0 -924.0 -0.33 360.0 -319.0 -0.24 -0.4047 -0.9896 3120394 ChemDiv3_010219 Cc1ccc2oc(=O)c3cnn(CC(=O)NCC4(CCCC4)c5ccccc5)c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A12 compound treatment 320.0 -964.0 -0.34 440.0 -239.0 -0.18 -0.3713 -0.9572 3031837 ChemDiv3_010220 O=C(Nc1ccc(cc1)c2cn3cccnc3n2)/C=C\c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A13 compound treatment 280.0 -1000.0 -0.36 480.0 -199.0 -0.15 -0.3596 -0.9284 3120565 ChemDiv3_010221 CC(C)CNc1cc(Cl)c2noc3-c4ccccc4C(=O)c1c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A14 compound treatment 240.0 -1040.0 -0.37 280.0 -399.0 -0.31 -0.4782 -0.9955 3031840 ChemDiv3_010222 C(c1ccccc1)n2cc3c(nnc3c4ccccc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A15 compound treatment 400.0 -884.0 -0.31 400.0 -279.0 -0.21 -0.3729 -0.9826 3120566 ChemDiv3_010223 CC1(OC(=O)C[n+]2ccccc21)/C(=N/c3ccc(Cl)cc3)/C(=O)Nc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A16 compound treatment 320.0 -964.0 -0.34 400.0 -279.0 -0.21 -0.393 -0.9745 3120567 ChemDiv3_010224 Cc1ccc2nc(NC(=O)C3CCCN(C3)S(=O)(=O)c4ccc5n(C)c(=O)oc5c4)sc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A17 compound treatment 240.0 -1040.0 -0.37 240.0 -439.0 -0.34 -0.4999 -0.9989 3031907 ChemDiv3_010225 Cc1cc(on1)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A18 compound treatment 240.0 -1040.0 -0.37 400.0 -279.0 -0.21 -0.4131 -0.966 3031909 ChemDiv3_010226 COc1ccc(cc1)C2=NOC(C2)C(=O)N3CCCCC3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A19 compound treatment 280.0 -1000.0 -0.36 520.0 -159.0 -0.12 -0.3379 -0.8979 3120568 ChemDiv3_010227 Cc1noc(C(=O)N2CCN(CC2)c3cc(Cl)ccc3C)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A20 compound treatment 240.0 -1040.0 -0.37 4640.0 3960.0 3.04 1.8887 0.6165 3120569 ChemDiv3_010228 COc1ccccc1C2=NOC(C2)C(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A21 compound treatment 360.0 -924.0 -0.33 3040.0 2360.0 1.81 1.0502 0.5701 3031914 ChemDiv3_010229 CCN(C(=O)c1cc2c(C)nc3ccccc3c2o1)c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A22 compound treatment 320.0 -964.0 -0.34 520.0 -159.0 -0.12 -0.3279 -0.9034 3120570 ChemDiv3_010230 CC(C)NC(=O)C1CC(=NO1)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A23 mock treatment 280.0 -1000.0 -0.36 400.0 -279.0 -0.21 -0.403 -0.9703 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 A24 mock treatment 320.0 -964.0 -0.34 320.0 -359.0 -0.28 -0.4364 -0.9942 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B01 compound treatment 280.0 -1000.0 -0.36 400.0 -279.0 -0.21 -0.403 -0.9703 3031918 ChemDiv3_010231 COc1cc(Br)cc2cc3c(=O)n(nc3oc12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B02 compound treatment 360.0 -924.0 -0.33 1120.0 441.0 0.34 0.0079 0.0167 3120571 ChemDiv3_010232 CCOC(=O)c1ccccc1NC(=O)CSc2nnc(Cc3cccn3C)n2c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B03 compound treatment 240.0 -1040.0 -0.37 880.0 201.0 0.15 -0.1525 -0.3801 3120572 ChemDiv3_010233 CCC(C(=O)OC)n1cnc2n(Cc3ccccc3F)nnc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B04 compound treatment 400.0 -884.0 -0.31 2920.0 2240.0 1.72 0.9951 0.5689 3030788 ChemDiv3_010234 C1CCN(C1)c2nc3c(nnn3c4ccccc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B05 compound treatment 240.0 -1040.0 -0.37 1520.0 841.0 0.65 0.1949 0.2618 3120573 ChemDiv3_010235 CCC(C(=O)OC)n1cnc2n(nnc2c1=O)c3cccc(Cl)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B06 compound treatment 320.0 -964.0 -0.34 440.0 -239.0 -0.18 -0.3713 -0.9572 3120574 ChemDiv3_010236 Fc1ccc(Cn2cc(c(=O)c3cc(F)ccc23)S(=O)(=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B07 compound treatment 3520.0 2240.0 0.79 360.0 -319.0 -0.24 0.388 0.4674 3030792 ChemDiv3_010237 COc1ccc(CCC(=O)Nc2n[nH]c3nc4cc(OC)ccc4cc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B08 compound treatment 640.0 -644.0 -0.23 920.0 241.0 0.19 -0.0304 -0.1035 3120575 ChemDiv3_010238 Cc1nc2c3ccccc3n4c(CCCC(=O)NCCc5ccc(Cl)cc5)nnc4n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B09 compound treatment 5120.0 3840.0 1.36 320.0 -359.0 -0.28 0.7676 0.5529 3120576 ChemDiv3_010239 CN(CCNC(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1)Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B10 compound treatment 1160.0 -124.0 -0.04 240.0 -439.0 -0.34 -0.2692 -0.7926 3030798 ChemDiv3_010240 CCOCC(=O)Nc1c(oc2ccccc12)C(=O)Nc3cccc(OC)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B11 compound treatment 400.0 -884.0 -0.31 880.0 201.0 0.15 -0.1124 -0.3214 3030799 ChemDiv3_010241 Cc1ncoc1C(=O)NCc2ccc(Cl)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B12 compound treatment 4200.0 2920.0 1.03 400.0 -279.0 -0.21 0.5803 0.5493 3120577 ChemDiv3_010242 CCc1ccc(NC(=O)c2cnn3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B13 compound treatment 240.0 -1040.0 -0.37 400.0 -279.0 -0.21 -0.4131 -0.966 3120578 ChemDiv3_010243 CCCSc1nnc(Cn2c(=O)sc3ccccc23)n1CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B14 compound treatment 360.0 -924.0 -0.33 240.0 -439.0 -0.34 -0.4698 -0.9999 3030805 ChemDiv3_010244 O=C(NCCc1ccsc1)c2cnn3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B15 compound treatment 360.0 -924.0 -0.33 1640.0 961.0 0.74 0.2902 0.3593 3120579 ChemDiv3_010245 COc1ccc(cc1)c2cc(N)n(n2)S(=O)(=O)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B16 compound treatment 320.0 -964.0 -0.34 400.0 -279.0 -0.21 -0.393 -0.9745 3030869 ChemDiv3_010246 CCOC(=O)N1CCc2c(C1)sc3n(CC(=O)NC(C)CC)c(=O)n(Cc4ccccc4)c(=O)c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B17 compound treatment 480.0 -804.0 -0.29 480.0 -199.0 -0.15 -0.3094 -0.957 3120580 ChemDiv3_010247 OC(=O)CSc1c2CCCc2nc3cc(ccc13)C(=O)NCC4COc5ccccc5O4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B18 compound treatment 240.0 -1040.0 -0.37 240.0 -439.0 -0.34 -0.4999 -0.9989 3030873 ChemDiv3_010248 CC(C)NC(=O)Cn1nc(Cc2ccncc2)c3ccccc3c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B19 compound treatment 280.0 -1000.0 -0.36 680.0 1.38 0.0 -0.251 -0.705 3120581 ChemDiv3_010249 COc1ccc2[nH]c3c(=O)n(CCCCC(=O)NCc4ccccc4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B20 compound treatment 360.0 -924.0 -0.33 2760.0 2080.0 1.6 0.8982 0.5506 3120582 ChemDiv3_010250 CCOC(=O)N1CCC(CC1)NC(=O)Cn2nc(Cc3cccnc3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B21 compound treatment 240.0 -1040.0 -0.37 1600.0 921.0 0.71 0.2384 0.2985 3030877 ChemDiv3_010251 Cn1cccc1Cc2nnc(SCC(=O)Nc3ccccc3C(F)(F)F)n2CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B22 compound treatment 480.0 -804.0 -0.29 320.0 -359.0 -0.28 -0.3963 -0.9998 3120583 ChemDiv3_010252 O=C(NCc1ccccc1)c2ccc3SCCN(Cc4ccccc4)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B23 mock treatment 560.0 -724.0 -0.26 280.0 -399.0 -0.31 -0.3979 -0.9962 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 B24 mock treatment 320.0 -964.0 -0.34 240.0 -439.0 -0.34 -0.4799 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C01 compound treatment 400.0 -884.0 -0.31 6840.0 6160.0 4.73 3.1231 0.6588 3030880 ChemDiv3_010253 Nc1cccnc1NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C02 compound treatment 320.0 -964.0 -0.34 400.0 -279.0 -0.21 -0.393 -0.9745 3120584 ChemDiv3_010254 Fc1ccc(Cn2c(=O)cc([nH]c2=O)N3CCc4ccccc4C3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C03 compound treatment 360.0 -924.0 -0.33 2640.0 1960.0 1.51 0.833 0.5406 3030886 ChemDiv3_010255 CCOC(=O)N1CCC(CC1)c2nc(C)sc2C(=O)NCc3ccc(Cl)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C04 compound treatment 360.0 -924.0 -0.33 320.0 -359.0 -0.28 -0.4264 -0.9962 3030954 ChemDiv3_010256 COC(=O)c1cc(=O)n(C)/c(=N/c2ccc(F)cc2)/s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C05 compound treatment 280.0 -1000.0 -0.36 3920.0 3240.0 2.49 1.5078 0.5998 3120585 ChemDiv3_010257 O=C(CCc1nc2cccnc2n1c3ccccc3)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C06 compound treatment 320.0 -964.0 -0.34 240.0 -439.0 -0.34 -0.4799 -1.0 3030958 ChemDiv3_010258 C=CCN1C(CC(=O)Nc2ccccc2)C(=O)N(C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C07 compound treatment 320.0 -964.0 -0.34 320.0 -359.0 -0.28 -0.4364 -0.9942 3120586 ChemDiv3_010259 CN1CC(=O)N=C1NC(=O)c2cc3c(Cl)nc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C08 compound treatment 280.0 -1000.0 -0.36 280.0 -399.0 -0.31 -0.4682 -0.9972 3120587 ChemDiv3_010260 COC(=O)c1ccc(NC(=O)CC2N(C3CCCC3)C(=O)N(C2=O)c4ccc(F)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C09 compound treatment 440.0 -844.0 -0.3 280.0 -399.0 -0.31 -0.428 -0.9999 3030965 ChemDiv3_010261 COc1ccc(CCNC(=O)CSc2c3CCCCc3nc4cc(Cl)ccc24)c(OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C10 compound treatment 360.0 -924.0 -0.33 320.0 -359.0 -0.28 -0.4264 -0.9962 3120588 ChemDiv3_010262 O=C(CSCc1ccccc1)Nc2cccc(c2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C11 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3120589 ChemDiv3_010263 Cc1ccc2oc(=O)c3cnn(CC(=O)NCCN4CCN(Cc5ccccc5)CC4)c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C12 compound treatment 360.0 -924.0 -0.33 360.0 -319.0 -0.24 -0.4047 -0.9896 3030968 ChemDiv3_010264 O=C(Cc1ccccc1)Nc2ccc(cc2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C13 compound treatment 200.0 -1080.0 -0.38 360.0 -319.0 -0.24 -0.4448 -0.9762 3120590 ChemDiv3_010265 CC(C)Nc1cc(Br)c2noc3-c4ccccc4C(=O)c1c32 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C14 compound treatment 240.0 -1040.0 -0.37 400.0 -279.0 -0.21 -0.4131 -0.966 3120591 ChemDiv3_010266 CC(C)C(NS(=O)(=O)c1ccc2nc(C)sc2c1)C(=O)N3CCn4c3nc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C15 compound treatment 2880.0 1600.0 0.57 320.0 -359.0 -0.28 0.2057 0.3267 3031039 ChemDiv3_010267 O=C(Nc1ccccc1)C2N(C(=O)C[n+]3ccccc23)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C16 compound treatment 2320.0 1040.0 0.37 320.0 -359.0 -0.28 0.0653 0.1421 3120755 ChemDiv3_010268 Cn1c(=O)n(C)c2ccc(cc2c1=O)S(=O)(=O)NCCC(=O)NC3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C17 compound treatment 440.0 -844.0 -0.3 360.0 -319.0 -0.24 -0.3846 -0.995 3031045 ChemDiv3_010269 Cc1cc(on1)C(=O)NCc2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C18 compound treatment 400.0 -884.0 -0.31 280.0 -399.0 -0.31 -0.4381 -0.9999 3120756 ChemDiv3_010270 COc1ccc(cc1)C2=NOC(C2)C(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C19 compound treatment 1560.0 276.0 0.1 320.0 -359.0 -0.28 -0.1254 -0.429 3120757 ChemDiv3_010271 CC(C)c1ccc(cc1)N(CC(=O)N2CCCC2)S(=O)(=O)c3c(C)nn(C)c3C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C20 compound treatment 2880.0 1600.0 0.57 360.0 -319.0 -0.24 0.2274 0.3687 3031051 ChemDiv3_010272 Fc1ccc(cc1)C2=NOC(C2)C(=O)Nc3cccnc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C21 compound treatment 7040.0 5760.0 2.04 400.0 -279.0 -0.21 1.2927 0.6296 3032301 ChemDiv3_010273 CCOc1ccc(CCNC(=O)c2cc3c(C)nc4ccccc4c3o2)cc1OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C22 compound treatment 9040.0 7760.0 2.75 280.0 -399.0 -0.31 1.7292 0.6246 3032302 ChemDiv3_010274 Fc1ccccc1C2=NOC(C2)C(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C23 mock treatment 5800.0 4520.0 1.6 240.0 -439.0 -0.34 0.8948 0.5465 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 C24 mock treatment 3520.0 2240.0 0.79 320.0 -359.0 -0.28 0.3663 0.4362 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D01 compound treatment 400.0 -884.0 -0.31 440.0 -239.0 -0.18 -0.3512 -0.9673 3032303 ChemDiv3_010275 CCOC(=O)C1=C(CS(=O)(=O)c2ccccc2)NC(=O)NC1c3ccc(SC)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D02 compound treatment 240.0 -1040.0 -0.37 800.0 121.0 0.09 -0.1959 -0.5131 3032304 ChemDiv3_010276 Cc1nnc(NC(=O)CSc2nnc(Cc3cccn3C)n2c4ccc(F)cc4)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D03 compound treatment 440.0 -844.0 -0.3 560.0 -119.0 -0.09 -0.276 -0.8823 3032305 ChemDiv3_010277 Clc1ccc(Cn2nnc3c(=O)n(CC(=O)N4CCCc5ccccc45)cnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D04 compound treatment 240.0 -1040.0 -0.37 440.0 -239.0 -0.18 -0.3914 -0.9473 3120758 ChemDiv3_010278 NS(=O)(=O)c1ccc(CCNc2nc3c(nnn3c4ccccc24)c5ccc(Cl)cc5)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D05 compound treatment 5080.0 3800.0 1.35 360.0 -319.0 -0.24 0.7793 0.5694 3032306 ChemDiv3_010279 Clc1cccc(c1)n2nnc3c(=O)n(CC(=O)OCc4ccccc4)cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D06 compound treatment 440.0 -844.0 -0.3 320.0 -359.0 -0.28 -0.4063 -0.9991 3032307 ChemDiv3_010280 CSc1nc(nc2Oc3ccccc3Cc12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D07 compound treatment 400.0 -884.0 -0.31 320.0 -359.0 -0.28 -0.4164 -0.9979 3120759 ChemDiv3_010281 Clc1c2CCCc2nc3cc(ccc13)C(=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D08 compound treatment 280.0 -1000.0 -0.36 440.0 -239.0 -0.18 -0.3813 -0.9523 3120760 ChemDiv3_010282 Cc1nc2c3ccccc3n4c(CCCC(=O)NCc5ccc(C)cc5)nnc4n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D09 compound treatment 440.0 -844.0 -0.3 240.0 -439.0 -0.34 -0.4498 -0.9983 3032308 ChemDiv3_010283 CC1CCCCC1NC(=O)Cn2ncc3c(=O)oc4ccccc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D10 compound treatment 400.0 -884.0 -0.31 240.0 -439.0 -0.34 -0.4598 -0.9994 3120761 ChemDiv3_010284 COc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D11 compound treatment 360.0 -924.0 -0.33 400.0 -279.0 -0.21 -0.383 -0.9786 3032309 ChemDiv3_010285 Cc1ncoc1C(=O)NCCC(c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D12 compound treatment 400.0 -884.0 -0.31 440.0 -239.0 -0.18 -0.3512 -0.9673 3120762 ChemDiv3_010286 CCOC(=O)N1CCN(CC1)C(=O)c2cnn3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D13 compound treatment 240.0 -1040.0 -0.37 240.0 -439.0 -0.34 -0.4999 -0.9989 3120763 ChemDiv3_010287 CSc1nnc(Cn2c(=O)sc3ccccc23)n1c4ccccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D14 compound treatment 560.0 -724.0 -0.26 320.0 -359.0 -0.28 -0.3762 -0.9994 3032310 ChemDiv3_010288 O=C(NCC1CCN(C1)C2CCCC2)c3cnn4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D15 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3120764 ChemDiv3_010289 CCOC(=O)N1CCC(CC1)Nc2nc3ccccc3nc2NS(=O)(=O)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D16 compound treatment 240.0 -1040.0 -0.37 280.0 -399.0 -0.31 -0.4782 -0.9955 3032311 ChemDiv3_010290 Cc1nc2c3ccccc3n(CC(=O)c4ccc(Br)cc4)c(=O)n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D17 compound treatment 1920.0 636.0 0.23 440.0 -239.0 -0.18 0.0301 0.1034 3120765 ChemDiv3_010291 CC1CC(C)CN(CCCNC(=O)c2ccc3c(SCC(=O)O)c4CCCc4nc3c2)C1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D18 compound treatment 1840.0 556.0 0.2 440.0 -239.0 -0.18 0.01 0.0371 3120766 ChemDiv3_010292 CN(C(=O)Cn1nc(Cc2ccncc2)c3ccccc3c1=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D19 compound treatment 1200.0 -83.8 -0.03 280.0 -399.0 -0.31 -0.2374 -0.7721 3032312 ChemDiv3_010293 COc1ccc2[nH]c3c(=O)n(CC(=O)NCCc4ccc(OC)c(OC)c4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D20 compound treatment 480.0 -804.0 -0.29 240.0 -439.0 -0.34 -0.4397 -0.9966 3120767 ChemDiv3_010294 CN(Cc1ccccc1)C(=O)C2CCCN2S(=O)(=O)c3ccc4n(C)c(=O)c(=O)n(C)c4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D21 compound treatment 600.0 -684.0 -0.24 240.0 -439.0 -0.34 -0.4096 -0.987 3120768 ChemDiv3_010295 Cn1cccc1Cc2nnc(SCC(=O)NC3CCCCC3)n2CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D22 compound treatment 3960.0 2680.0 0.95 280.0 -399.0 -0.31 0.4549 0.4561 3032313 ChemDiv3_010296 O=C(NC1CC1)c2ccc3SCCN(Cc4ccccc4)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D23 mock treatment 1840.0 556.0 0.2 280.0 -399.0 -0.31 -0.0769 -0.2111 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 D24 mock treatment 360.0 -924.0 -0.33 360.0 -319.0 -0.24 -0.4047 -0.9896 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E01 compound treatment 440.0 -844.0 -0.3 960.0 281.0 0.22 -0.0589 -0.1596 3120769 ChemDiv3_010297 Cc1cc(C)c2c(nn3c(C)c(CCC(=O)O)c(C)nc23)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E02 compound treatment 480.0 -804.0 -0.29 1240.0 561.0 0.43 0.1031 0.1996 3032314 ChemDiv3_010298 CC1CN(CC(C)O1)c2cc(=O)n(c3ccc(Cl)cc3)c(=O)[nH]2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E03 compound treatment 480.0 -804.0 -0.29 840.0 161.0 0.12 -0.114 -0.3667 3120770 ChemDiv3_010299 CCOC(=O)c1cnn(c1C2CCN(CC2)C(=O)OC(C)(C)C)c3ccc(cc3)C(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E04 compound treatment 2000.0 716.0 0.25 480.0 -199.0 -0.15 0.0718 0.2424 3120771 ChemDiv3_010300 COc1ccc(NC(=O)CC2N(C(C)C)C(=O)N(C2=O)c3ccccc3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E05 compound treatment 2400.0 1120.0 0.4 4920.0 4240.0 3.26 2.5825 0.7873 3032315 ChemDiv3_010301 O=C(CCc1nc2cccnc2n1c3ccccc3)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E06 compound treatment 2240.0 956.0 0.34 3560.0 2880.0 2.21 1.8041 0.8061 3120772 ChemDiv3_010302 CCOC(=O)c1ccc(NC(=O)CC2N(Cc3cccs3)C(=O)N(C2=O)c4ccc(F)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E07 compound treatment 4360.0 3080.0 1.09 1360.0 681.0 0.52 1.1415 0.9433 3032316 ChemDiv3_010303 COc1cc2CCN(C(C)c2cc1OC)C(=O)c3cc4c(Cl)nc5ccc(C)cc5c4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E08 compound treatment 2360.0 1080.0 0.38 3200.0 2520.0 1.94 1.6387 0.8306 3120773 ChemDiv3_010304 CCOc1ccc(cc1)c2cc(CCCC(=O)Nc3ccc(CC)cc3)no2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E09 compound treatment 1720.0 436.0 0.15 880.0 201.0 0.15 0.2188 1.0 3032317 ChemDiv3_010305 CN(Cc1ccccc1)C(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E10 compound treatment 960.0 -324.0 -0.11 600.0 -78.6 -0.06 -0.1239 -0.9549 3120774 ChemDiv3_010306 Cc1ccc(cc1NC(=O)CC(C)(C)C)c2cn3cccnc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E11 compound treatment 2600.0 1320.0 0.47 2400.0 1720.0 1.32 1.2646 0.9023 3120775 ChemDiv3_010307 Cc1ccc2oc(=O)c3cnn(CC(=O)Nc4cccnc4)c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E12 compound treatment 1200.0 -83.8 -0.03 4000.0 3320.0 2.55 1.782 0.6988 3032318 ChemDiv3_010308 Cc1c(nc2ncccn12)c3cccc(NC(=O)C(C)(C)Oc4ccc(Cl)cc4)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E13 compound treatment 400.0 -884.0 -0.31 2480.0 1800.0 1.38 0.7562 0.5333 3120776 ChemDiv3_010309 CC(C)CNc1cc(NCCO)c2C(=O)c3ccccc3-c4onc1c42 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E14 compound treatment 600.0 -684.0 -0.24 480.0 -199.0 -0.15 -0.2793 -0.975 3120777 ChemDiv3_010310 COc1ccc(CNC(=O)C(NS(=O)(=O)c2ccc3nc(C)sc3c2)C(C)C)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E15 compound treatment 1920.0 636.0 0.23 1080.0 401.0 0.31 0.3775 0.9883 3032319 ChemDiv3_010311 Cc1cccc(C)c1/N=C/2\Oc3ccccc3NC2(C)c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E16 compound treatment 1680.0 396.0 0.14 3720.0 3040.0 2.33 1.7504 0.7483 3120778 ChemDiv3_010312 CC1CCCN(C1)C(=O)CCNS(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E17 compound treatment 680.0 -604.0 -0.21 1560.0 881.0 0.68 0.327 0.4608 3032320 ChemDiv3_010313 Cc1cc(on1)C(=O)NC(C)(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E18 compound treatment 4480.0 3200.0 1.13 1400.0 721.0 0.55 1.1934 0.9457 3032321 ChemDiv3_010314 COc1ccc(cc1)C2=NOC(C2)C(=O)N3CCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E19 compound treatment 2000.0 716.0 0.25 680.0 1.38 0.0 0.1804 0.71 3120779 ChemDiv3_010315 O=C(Nc1ccc(Cc2ccncc2)cc1)c3cc4ccccn4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E20 compound treatment 6120.0 4840.0 1.72 1080.0 401.0 0.31 1.431 0.821 3120780 ChemDiv3_010316 Fc1ccc(cc1)C2=NOC(C2)C(=O)NCC3CCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E21 compound treatment 960.0 -324.0 -0.11 760.0 81.4 0.06 -0.037 -0.2833 3032322 ChemDiv3_010317 CCc1ccc(CNC(=O)c2cc3c(C)nc4ccccc4c3o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E22 compound treatment 1800.0 516.0 0.18 480.0 -199.0 -0.15 0.0217 0.091 3120781 ChemDiv3_010318 CN(C(=O)C1CC(=NO1)c2ccccc2F)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E23 mock treatment 1560.0 276.0 0.1 480.0 -199.0 -0.15 -0.0385 -0.2126 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 E24 mock treatment 1480.0 196.0 0.07 2840.0 2160.0 1.66 1.2226 0.7361 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F01 compound treatment 1640.0 356.0 0.13 1360.0 681.0 0.52 0.4593 0.8534 3120961 ChemDiv3_010319 CCc1ccc(NC(=O)Cn2cc(c(=O)c3ccccc23)S(=O)(=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F02 compound treatment 2000.0 716.0 0.25 1760.0 1080.0 0.83 0.7667 0.8831 3032323 ChemDiv3_010320 CCSc1nnc(NC(=O)CSc2nnc(Cc3cccn3C)n2c4ccc(F)cc4)s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F03 compound treatment 960.0 -324.0 -0.11 4120.0 3440.0 2.64 1.787 0.6757 3120962 ChemDiv3_010321 Clc1ccc(Cn2nnc3c(=O)n(CC(=O)NC4CCCCC4)cnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F04 compound treatment 2200.0 916.0 0.33 840.0 161.0 0.12 0.3174 0.9126 3032324 ChemDiv3_010322 CC(=O)NCCNc1nc2c(nnn2c3ccccc13)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F05 compound treatment 3360.0 2080.0 0.74 2080.0 1400.0 1.08 1.2816 0.9829 3120963 ChemDiv3_010323 COc1cccc(c1)n2nnc3c(=O)n(CC(=O)c4ccc(Cl)cc4)cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F06 compound treatment 1360.0 76.3 0.03 1360.0 681.0 0.52 0.389 0.7427 3120964 ChemDiv3_010324 O=C(CSc1nc(nc2Oc3ccccc3Cc12)c4ccccc4)Nc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F07 compound treatment 1840.0 556.0 0.2 1240.0 561.0 0.43 0.4443 0.9373 3032325 ChemDiv3_010325 CCN(CC)S(=O)(=O)c1ccc(Nc2c3CCCCc3nc4ccccc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F08 compound treatment 5880.0 4600.0 1.63 2520.0 1840.0 1.41 2.1525 0.9975 3120965 ChemDiv3_010326 OC(=O)CCCc1nnc2n3nc(nc3c4ccccc4n12)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F09 compound treatment 6520.0 5240.0 1.86 1760.0 1080.0 0.83 1.9005 0.9341 3120966 ChemDiv3_010327 CC(C)N(C1CCCCC1)C(=O)Cn2ncc3c(=O)oc4ccccc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F10 compound treatment 6400.0 5120.0 1.81 3720.0 3040.0 2.33 2.9344 0.9922 3032326 ChemDiv3_010328 Cc1cccc(OCC(=O)Nc2c(oc3ccccc23)C(=O)Nc4cccc(F)c4)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F11 compound treatment 1440.0 156.0 0.06 2680.0 2000.0 1.54 1.1257 0.7321 3120967 ChemDiv3_010329 Cc1ncoc1C(=O)Nc2ccccc2F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F12 compound treatment 880.0 -404.0 -0.14 6040.0 5360.0 4.12 2.8092 0.6821 3032327 ChemDiv3_010330 O=C(N1CCc2ccccc12)c3cnn4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F13 compound treatment 760.0 -524.0 -0.19 3040.0 2360.0 1.81 1.1505 0.6313 3120968 ChemDiv3_010331 Clc1cccc(c1)n2c(Cn3c(=O)sc4ccccc34)nnc2SCc5ccccn5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F14 compound treatment 760.0 -524.0 -0.19 4040.0 3360.0 2.58 1.6934 0.6545 3120969 ChemDiv3_010332 CCOC(=O)c1cnn(CCOC(=O)c2ccccc2F)c1NC(=O)c3ccccc3F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F15 compound treatment 1440.0 156.0 0.06 4080.0 3400.0 2.61 1.8857 0.722 3032328 ChemDiv3_010333 CCC(C)NC(=O)c1ccc2c(Cl)c3CCCc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F16 compound treatment 1040.0 -244.0 -0.09 1440.0 761.0 0.58 0.3522 0.596 3120970 ChemDiv3_010334 COc1ccccc1NC(=O)Cn2c(=O)n3nc(C)nc3c4ccccc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F17 compound treatment 4480.0 3200.0 1.13 2040.0 1360.0 1.05 1.5408 0.9992 3032329 ChemDiv3_010335 CCN(C(=O)c1ccc2c(SCC(=O)O)c3CCCc3nc2c1)c4cc(Cl)ccc4OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F18 compound treatment 5040.0 3760.0 1.33 1960.0 1280.0 0.98 1.6378 0.9889 3120971 ChemDiv3_010336 COC(CNC(=O)Cn1nc(Cc2ccncc2)c3ccccc3c1=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F19 compound treatment 2560.0 1280.0 0.45 6400.0 5720.0 4.39 3.426 0.7759 3120972 ChemDiv3_010337 COc1ccc2[nH]c3c(=O)n(CC(=O)NC4CCCCCC4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F20 compound treatment 2280.0 996.0 0.35 2960.0 2280.0 1.75 1.4884 0.833 3032330 ChemDiv3_010338 CN(C)/C=C/c1onc(C)c1S(=O)(=O)N2CCCC(C2)C(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F21 compound treatment 1920.0 636.0 0.23 2760.0 2080.0 1.6 1.2895 0.7991 3120973 ChemDiv3_010339 Cn1cccc1Cc2nnc(SCC(=O)NCc3ccco3)n2CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F22 compound treatment 5120.0 3840.0 1.36 3120.0 2440.0 1.87 2.2876 0.9876 3032331 ChemDiv3_010340 CC(C)CCNC(=O)c1ccc2SCCN(Cc3ccccc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F23 mock treatment 2120.0 836.0 0.3 760.0 81.4 0.06 0.2539 0.8377 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 F24 mock treatment 960.0 -324.0 -0.11 3840.0 3160.0 2.43 1.635 0.6729 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G01 compound treatment 240.0 -1040.0 -0.37 520.0 -159.0 -0.12 -0.3479 -0.8926 3120974 ChemDiv3_010341 CN(Cc1ccccc1)C(=O)CCc2nc3cccnc3n2Cc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G02 compound treatment 480.0 -804.0 -0.29 520.0 -159.0 -0.12 -0.2877 -0.928 3120975 ChemDiv3_010342 Clc1ccc(cc1)n2c(=O)cc([nH]c2=O)N3CCN(CC3)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G03 compound treatment 1440.0 156.0 0.06 1440.0 761.0 0.58 0.4525 0.7707 3032332 ChemDiv3_010343 NCc1ccc2cc[nH]c(=O)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G04 compound treatment 800.0 -484.0 -0.17 1200.0 521.0 0.4 0.1617 0.3713 3120976 ChemDiv3_010344 CCNC(=O)CC1N(CCOC)C(=O)N(C1=O)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G05 compound treatment 760.0 -524.0 -0.19 1280.0 601.0 0.46 0.1951 0.392 3032333 ChemDiv3_010345 O=C(CCc1nc2cccnc2n1c3ccccc3)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G06 compound treatment 5240.0 3960.0 1.4 680.0 1.38 0.0 0.9931 0.7076 3120977 ChemDiv3_010346 COC(=O)c1cc(=O)n(CCc2ccccc2)/c(=N/CCc3ccccc3)/s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G07 compound treatment 520.0 -764.0 -0.27 1000.0 321.0 0.25 -0.0171 -0.0467 3032334 ChemDiv3_010347 CN1CCN(CCNC(=O)c2cc3c(Cl)nc4ccc(C)cc4c3s2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G08 compound treatment 2920.0 1640.0 0.58 2520.0 1840.0 1.41 1.4101 0.9227 3032480 ChemDiv3_010348 CCOc1ccc(cc1)c2cc(CCCC(=O)NCCc3ccccc3)no2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G09 compound treatment 2400.0 1120.0 0.4 640.0 -38.6 -0.03 0.259 0.6523 3032481 ChemDiv3_010349 CC1CCCCN1C(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G10 compound treatment 5960.0 4680.0 1.66 360.0 -319.0 -0.24 1.0 0.5964 3032483 ChemDiv3_010350 CCCC(CCC)C(=O)Nc1cc(ccc1C)c2cn3cccnc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G11 compound treatment 1040.0 -244.0 -0.09 680.0 1.38 0.0 -0.0604 -0.6984 3032484 ChemDiv3_010351 CCCN(CCC)C(=O)Cn1ncc2c(=O)oc3ccc(C)cc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G12 compound treatment 1120.0 -164.0 -0.06 640.0 -38.6 -0.03 -0.062 -0.9513 3032486 ChemDiv3_010352 Clc1ccc(NC(=O)Nc2cccc(c2)c3cn4cccnc4n3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G13 compound treatment 1240.0 -43.8 -0.02 840.0 161.0 0.12 0.0766 0.6137 3032542 ChemDiv3_010353 CN1C(C(=O)Nc2ccccc2)c3cccc[n+]3CC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G14 compound treatment 840.0 -444.0 -0.16 480.0 -199.0 -0.15 -0.2191 -0.9999 3032543 ChemDiv3_010354 CC(C)C(NS(=O)(=O)c1ccc2nc(C)sc2c1)C(=O)Nc3nc4ccc(Cl)cc4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G15 compound treatment 720.0 -564.0 -0.2 480.0 -199.0 -0.15 -0.2492 -0.991 3032545 ChemDiv3_010355 C/C(=C\C(=N\c1ccccc1O)\c2ccccn2)/c3ccccn3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G16 compound treatment 560.0 -724.0 -0.26 480.0 -199.0 -0.15 -0.2894 -0.969 3032546 ChemDiv3_010356 Cc1ccnc(NC(=O)CCNS(=O)(=O)c2ccc3n(C)c(=O)n(C)c(=O)c3c2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G17 compound treatment 1760.0 476.0 0.17 480.0 -199.0 -0.15 0.0116 0.0512 3032549 ChemDiv3_010357 COc1ccc(CCNC(=O)c2cc(C)no2)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G18 compound treatment 6320.0 5040.0 1.79 1040.0 361.0 0.28 1.4595 0.8072 3032550 ChemDiv3_010358 CCCNC(=O)C1CC(=NO1)c2ccc(OC)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G19 compound treatment 520.0 -764.0 -0.27 480.0 -199.0 -0.15 -0.2994 -0.963 3032552 ChemDiv3_010359 Clc1ccccc1CNC(=O)c2cc3ccccn3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G20 compound treatment 560.0 -724.0 -0.26 1600.0 921.0 0.71 0.3186 0.4234 3120978 ChemDiv3_010360 CC1CCCC(C)N1C(=O)C2CC(=NO2)c3ccc(F)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G21 compound treatment 880.0 -404.0 -0.14 5200.0 4520.0 3.47 2.3532 0.6774 3032553 ChemDiv3_010361 Cc1nc2ccccc2c3oc(cc13)C(=O)NC4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G22 compound treatment 920.0 -364.0 -0.13 2240.0 1560.0 1.2 0.7564 0.6274 3120979 ChemDiv3_010362 Fc1ccccc1C2=NOC(C2)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G23 mock treatment 1360.0 76.3 0.03 1200.0 521.0 0.4 0.3022 0.7532 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 G24 mock treatment 1120.0 -164.0 -0.06 720.0 41.4 0.03 -0.0186 -0.2811 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H01 compound treatment 1400.0 116.0 0.04 520.0 -159.0 -0.12 -0.0569 -0.4429 3120980 ChemDiv3_010363 Cc1ccc(Cn2nnc3c(=O)n(CC(=O)N)cnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H02 compound treatment 2320.0 1040.0 0.37 400.0 -279.0 -0.21 0.1087 0.2555 3032556 ChemDiv3_010364 CCc1nn2c(=O)cc(COc3ccc(/C=C\4/C(=N)N5C=CSC5=NC4=O)cc3OC)nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H03 compound treatment 2320.0 1040.0 0.37 800.0 121.0 0.09 0.3258 0.8592 3120981 ChemDiv3_010365 COC(=O)Cn1cnc2n(Cc3ccc(Cl)cc3)nnc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H04 compound treatment 960.0 -324.0 -0.11 1840.0 1160.0 0.89 0.5493 0.611 3120982 ChemDiv3_010366 CNc1nc2c(nnn2c3ccccc13)c4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H05 compound treatment 600.0 -684.0 -0.24 1440.0 761.0 0.58 0.2418 0.3821 3032558 ChemDiv3_010367 COc1ccc(cc1)n2nnc3c(=O)n(Cc4cccc(c4)C(F)(F)F)cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H06 compound treatment 520.0 -764.0 -0.27 400.0 -279.0 -0.21 -0.3428 -0.9932 3120983 ChemDiv3_010368 CCOc1cccc2Cc3c(SCC(=O)N(CC)CC)nc(nc3Oc12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H07 compound treatment 720.0 -564.0 -0.2 760.0 81.4 0.06 -0.0972 -0.4641 3032561 ChemDiv3_010369 Cc1ccc2cc3c(N)nn(C(=O)c4ccccc4F)c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H08 compound treatment 480.0 -804.0 -0.29 2680.0 2000.0 1.54 0.8849 0.5662 3120984 ChemDiv3_010370 O=C(NCc1ccccc1)c2cccc(NC3=NC4CS(=O)(=O)CC4S3)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H09 compound treatment 520.0 -764.0 -0.27 640.0 -38.6 -0.03 -0.2125 -0.7798 3120985 ChemDiv3_010371 COC(CNC(=O)Cn1ncc2c(=O)oc3ccccc3c12)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H10 compound treatment 8840.0 7560.0 2.68 5640.0 4960.0 3.81 4.5888 0.9852 3032563 ChemDiv3_010372 Fc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H11 compound treatment 600.0 -684.0 -0.24 2800.0 2120.0 1.63 0.9801 0.5952 3120986 ChemDiv3_010373 Cc1ncoc1C(=O)Nc2ccccc2C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H12 compound treatment 4280.0 3000.0 1.06 520.0 -159.0 -0.12 0.6655 0.622 3032565 ChemDiv3_010374 O=C(N1CCCc2ccccc12)c3cnn4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H13 compound treatment 360.0 -924.0 -0.33 520.0 -159.0 -0.12 -0.3178 -0.9091 3120987 ChemDiv3_010375 CCOC(=O)C(C)Sc1nnc(Cn2c(=O)sc3ccccc23)n1c4cccc(Cl)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H14 compound treatment 960.0 -324.0 -0.11 5320.0 4640.0 3.56 2.4384 0.684 3120988 ChemDiv3_010376 CCOC(=O)c1cnn(CCOC(=O)c2ccc(C)cc2)c1NC(=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H15 compound treatment 640.0 -644.0 -0.23 440.0 -239.0 -0.18 -0.291 -0.994 3032567 ChemDiv3_010377 CCc1ccc(NC(=O)c2ccc3c(Cl)c4CCCc4nc3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H16 compound treatment 600.0 -684.0 -0.24 1400.0 721.0 0.55 0.2201 0.364 3121170 ChemDiv3_010378 Brc1ccc(cc1)C(=O)Cn2c(=O)n3nc(nc3c4ccccc24)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H17 compound treatment 720.0 -564.0 -0.2 1320.0 641.0 0.49 0.2068 0.3891 3032569 ChemDiv3_010379 CC(C)CCNC(=O)c1ccc2c(SCC(=O)O)c3CCCc3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H18 compound treatment 760.0 -524.0 -0.19 280.0 -399.0 -0.31 -0.3478 -0.9714 3121171 ChemDiv3_010380 O=C(Cn1nc(Cc2cccnc2)c3ccccc3c1=O)Nc4ccc(Oc5ccccc5)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H19 compound treatment 400.0 -884.0 -0.31 560.0 -119.0 -0.09 -0.2861 -0.8763 3121172 ChemDiv3_010381 COc1ccc2[nH]c3c(=O)n(CC(=O)N(C)Cc4ccccc4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H20 compound treatment 1040.0 -244.0 -0.09 400.0 -279.0 -0.21 -0.2124 -0.9206 3032571 ChemDiv3_010382 CCC(C)NC(=O)C1CCCN(C1)S(=O)(=O)c2cccc3cccnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H21 compound treatment 400.0 -884.0 -0.31 1480.0 801.0 0.62 0.2134 0.309 3032607 ChemDiv3_010383 Cc1ccc(cc1)n2c(Cc3cccn3C)nnc2SCC(=O)N4CCN(CC4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H22 compound treatment 2440.0 1160.0 0.41 920.0 241.0 0.19 0.4211 0.9355 3032608 ChemDiv3_010384 O=C(NCCc1ccccc1)c2ccc3SCCN(Cc4ccccc4)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H23 mock treatment 600.0 -684.0 -0.24 920.0 241.0 0.19 -0.0405 -0.1326 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 H24 mock treatment 5440.0 4160.0 1.47 600.0 -78.6 -0.06 0.9999 0.6776 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I01 compound treatment 880.0 -404.0 -0.14 320.0 -359.0 -0.28 -0.296 -0.9536 3032609 ChemDiv3_010385 O=C(CCc1nc2cccnc2n1Cc3ccccc3)N4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I02 compound treatment 2720.0 1440.0 0.51 2400.0 1720.0 1.32 1.2947 0.9141 3032611 ChemDiv3_010386 Brc1ccc(cc1)n2c(=O)cc(NCc3ccco3)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I03 compound treatment 2360.0 1080.0 0.38 400.0 -279.0 -0.21 0.1187 0.2713 1060194 ChemDiv3_010387 Cc1cccc(c1)C(=O)NN 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I04 compound treatment 320.0 -964.0 -0.34 520.0 -159.0 -0.12 -0.3279 -0.9034 3032613 ChemDiv3_010388 COC(=O)c1ccc(/N=c/2\sc(cc(=O)n2Cc3ccccc3)C(=O)OC)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I05 compound treatment 320.0 -964.0 -0.34 1240.0 561.0 0.43 0.063 0.1145 3032614 ChemDiv3_010389 CN(Cc1ccccc1)C(=O)CCc2nc3cccnc3n2c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I06 compound treatment 360.0 -924.0 -0.33 320.0 -359.0 -0.28 -0.4264 -0.9962 3121173 ChemDiv3_010390 Cc1ccc(cc1)N2C(=O)C(CC(=O)Nc3ccccc3)N(Cc4ccc5OCOc5c4)C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I07 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3032616 ChemDiv3_010391 CN(C)CCN(Cc1ccco1)C(=O)c2cc3c(Cl)nc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I08 compound treatment 440.0 -844.0 -0.3 440.0 -239.0 -0.18 -0.3412 -0.9722 3121174 ChemDiv3_010392 COc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(nn3)N4CCOCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I09 compound treatment 400.0 -884.0 -0.31 280.0 -399.0 -0.31 -0.4381 -0.9999 3032618 ChemDiv3_010393 CC(C)NC(=O)Cn1ncc2c(=O)oc3ccc(C)cc3c12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I10 compound treatment 520.0 -764.0 -0.27 440.0 -239.0 -0.18 -0.3211 -0.9818 3121175 ChemDiv3_010394 Cc1ccc(cc1NC(=O)c2ccccc2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I11 compound treatment 680.0 -604.0 -0.21 280.0 -399.0 -0.31 -0.3678 -0.9848 3121176 ChemDiv3_010395 Cc1cc2ccccc2n1C(=O)Cn3ncc4c(=O)oc5ccc(C)cc5c34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I12 compound treatment 360.0 -924.0 -0.33 360.0 -319.0 -0.24 -0.4047 -0.9896 3032620 ChemDiv3_010396 Cc1ccc(cc1NC(=O)Nc2ccccc2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I13 compound treatment 360.0 -924.0 -0.33 920.0 241.0 0.19 -0.1007 -0.2674 3121177 ChemDiv3_010397 CN1C(C(=O)Nc2c(C)cccc2C)c3cccc[n+]3CC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I14 compound treatment 1320.0 36.3 0.01 280.0 -399.0 -0.31 -0.2073 -0.6768 3032623 ChemDiv3_010398 CC(C)C(NS(=O)(=O)c1ccc2nc(C)sc2c1)C(=O)Nc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I15 compound treatment 960.0 -324.0 -0.11 200.0 -479.0 -0.37 -0.341 -0.8859 3121178 ChemDiv3_010399 Cc1ccccc1NC(=O)C2N(Cc3ccc4OCOc4c3)C(=O)C[n+]5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I16 compound treatment 680.0 -604.0 -0.21 480.0 -199.0 -0.15 -0.2593 -0.9861 3121179 ChemDiv3_010400 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)N3CCC(CC3)C(=O)NCCc4ccc(Cl)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I17 compound treatment 400.0 -884.0 -0.31 440.0 -239.0 -0.18 -0.3512 -0.9673 3032627 ChemDiv3_010401 Cc1cc(on1)C(=O)Nc2sc3CCCCc3c2C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I18 compound treatment 320.0 -964.0 -0.34 400.0 -279.0 -0.21 -0.393 -0.9745 3121180 ChemDiv3_010402 COc1ccc(cc1)C2=NOC(C2)C(=O)NC(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I19 compound treatment 280.0 -1000.0 -0.36 3480.0 2800.0 2.15 1.269 0.5821 3032629 ChemDiv3_010403 O=C(N1CCC2(CC1)OCCO2)c3cc4ccccn4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I20 compound treatment 400.0 -884.0 -0.31 760.0 81.4 0.06 -0.1775 -0.5553 3121181 ChemDiv3_010404 Fc1ccc(cc1)C2=NOC(C2)C(=O)NCc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I21 compound treatment 320.0 -964.0 -0.34 4320.0 3640.0 2.8 1.735 0.616 3032631 ChemDiv3_010405 COC(CN(C)C(=O)c1cc2c(C)nc3ccccc3c2o1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I22 compound treatment 400.0 -884.0 -0.31 680.0 1.38 0.0 -0.2209 -0.7047 3121182 ChemDiv3_010406 COc1ccc(OC)c(c1)C2=NOC(C2)C(=O)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I23 mock treatment 2440.0 1160.0 0.41 760.0 81.4 0.06 0.3342 0.8055 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 I24 mock treatment 360.0 -924.0 -0.33 640.0 -38.6 -0.03 -0.2527 -0.7679 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J01 compound treatment 960.0 -324.0 -0.11 320.0 -359.0 -0.28 -0.2759 -0.9248 3032633 ChemDiv3_010407 Cc1ccc(Cn2nnc3c(=O)n(Cc4cccc(C)c4)cnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J02 compound treatment 360.0 -924.0 -0.33 320.0 -359.0 -0.28 -0.4264 -0.9962 3032666 ChemDiv3_010408 CC(N1C(=O)NC(=O)/C(=C/c2coc3ccccc3c2=O)/C1=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J03 compound treatment 360.0 -924.0 -0.33 360.0 -319.0 -0.24 -0.4047 -0.9896 3032667 ChemDiv3_010409 CCOC(=O)Cn1cnc2n(nnc2c1=O)c3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J04 compound treatment 320.0 -964.0 -0.34 1000.0 321.0 0.25 -0.0673 -0.1596 3032669 ChemDiv3_010410 COc1ccccc1CNc2nc3c(nnn3c4ccccc24)c5cccc(C)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J05 compound treatment 360.0 -924.0 -0.33 200.0 -479.0 -0.37 -0.4915 -0.9984 3032670 ChemDiv3_010411 CNC(=S)NCCc1c(C)[nH]c2ccccc12 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J06 compound treatment 600.0 -684.0 -0.24 240.0 -439.0 -0.34 -0.4096 -0.987 3032671 ChemDiv3_010412 COC(=O)CSc1nc(nc2Oc3ccc(Br)cc3Cc12)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J07 compound treatment 1200.0 -83.8 -0.03 1520.0 841.0 0.65 0.4357 0.6739 3032673 ChemDiv3_010413 COc1ccc2nc3[nH]nc(NC(=O)Cc4ccccc4OC)c3cc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J08 compound treatment 360.0 -924.0 -0.33 520.0 -159.0 -0.12 -0.3178 -0.9091 3121183 ChemDiv3_010414 O=C(Cc1ccc(NC2=NC3CS(=O)(=O)CC3S2)cc1)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J09 compound treatment 320.0 -964.0 -0.34 320.0 -359.0 -0.28 -0.4364 -0.9942 3032676 ChemDiv3_010415 O=C(Cn1nc(Cc2ccncc2)c3ccccc3c1=O)NCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J10 compound treatment 840.0 -444.0 -0.16 240.0 -439.0 -0.34 -0.3494 -0.94 3121184 ChemDiv3_010416 Cc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J11 compound treatment 400.0 -884.0 -0.31 320.0 -359.0 -0.28 -0.4164 -0.9979 3032678 ChemDiv3_010417 Cc1ncoc1C(=O)Nc2ccc(cc2)C(=O)N 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J12 compound treatment 280.0 -1000.0 -0.36 400.0 -279.0 -0.21 -0.403 -0.9703 3121185 ChemDiv3_010418 CSc1cccc(NC(=O)c2cnn3ccccc23)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J13 compound treatment 320.0 -964.0 -0.34 1360.0 681.0 0.52 0.1281 0.2051 3121186 ChemDiv3_010419 OC(=O)CSc1nnc(Cn2c(=O)sc3ccccc23)n1c4cccc(c4)C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J14 compound treatment 360.0 -924.0 -0.33 320.0 -359.0 -0.28 -0.4264 -0.9962 3032680 ChemDiv3_010420 CCOC(=O)c1cnn(CCOC(=O)c2cccs2)c1NC(=O)c3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J15 compound treatment 6400.0 5120.0 1.81 1000.0 321.0 0.25 1.4578 0.7959 3121187 ChemDiv3_010421 CN(C(=O)c1ccc2c(Cl)c3CCCc3nc2c1)c4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J16 compound treatment 3400.0 2120.0 0.75 320.0 -359.0 -0.28 0.3362 0.4204 3032682 ChemDiv3_010422 Cc1cc(C)n(CCc2nc3c4ccccc4n(Cc5ccc(Cl)cc5)c(=O)n3n2)n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J17 compound treatment 3400.0 2120.0 0.75 520.0 -159.0 -0.12 0.4447 0.5848 3121188 ChemDiv3_010423 COc1ccc2[nH]c3c(=O)n(Cc4ccc(cc4)C(=O)NCc5cccnc5)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J18 compound treatment 560.0 -724.0 -0.26 440.0 -239.0 -0.18 -0.3111 -0.9863 3121189 ChemDiv3_010424 CN(C1CCCCC1)C(=O)Cn2nc(Cc3cccnc3)c4ccccc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J19 compound treatment 240.0 -1040.0 -0.37 880.0 201.0 0.15 -0.1525 -0.3801 3032684 ChemDiv3_010425 COc1ccc2[nH]c3c(=O)n(CC(=O)N4CCN(CC4)c5ccc(F)cc5)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J20 compound treatment 720.0 -564.0 -0.2 1040.0 361.0 0.28 0.0548 0.1601 3121190 ChemDiv3_010426 O=C(C1CCCN(C1)S(=O)(=O)c2cccc3cccnc23)N4CCc5ccccc45 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J21 compound treatment 400.0 -884.0 -0.31 4760.0 4080.0 3.13 1.9939 0.6332 3032686 ChemDiv3_010427 CCOC(=O)N1CCN(CC1)C(=O)CSc2nnc(Cc3cccn3C)n2c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J22 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3121191 ChemDiv3_010428 CCC(C)NC(=O)c1ccc2SCCN(Cc3ccc(C)cc3)c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J23 mock treatment 480.0 -804.0 -0.29 480.0 -199.0 -0.15 -0.3094 -0.957 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 J24 mock treatment 400.0 -884.0 -0.31 280.0 -399.0 -0.31 -0.4381 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K01 compound treatment 480.0 -804.0 -0.29 1880.0 1200.0 0.92 0.4506 0.4667 3121192 ChemDiv3_010429 COc1ccc(NC(=O)c2cnn(c2C3CCNCC3)c4ccc(C)c(C)c4)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K02 compound treatment 400.0 -884.0 -0.31 760.0 81.4 0.06 -0.1775 -0.5553 3032689 ChemDiv3_010430 Brc1ccc(cc1)n2c(=O)cc(Nc3ccc4OCOc4c3)[nH]c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K03 compound treatment 3480.0 2200.0 0.78 2760.0 2080.0 1.6 1.6808 0.9455 3121193 ChemDiv3_010431 CCCn1c(CCC(=O)Nc2ccccc2)nc3cccnc13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K04 compound treatment 840.0 -444.0 -0.16 400.0 -279.0 -0.21 -0.2626 -0.9886 3032692 ChemDiv3_010432 CCn/1c(=O)cc(s\c1=N/c2ccc(F)c(F)c2)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K05 compound treatment 1040.0 -244.0 -0.09 360.0 -319.0 -0.24 -0.2341 -0.9023 3121194 ChemDiv3_010433 CCc1ccc(NC(=O)CCc2nc3cccnc3n2c4ccccc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K06 compound treatment 1480.0 196.0 0.07 320.0 -359.0 -0.28 -0.1455 -0.5122 3121195 ChemDiv3_010434 O=C(CC1N(C2CCCCC2)C(=O)N(C1=O)c3ccccc3)Nc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K07 compound treatment 840.0 -444.0 -0.16 600.0 -78.6 -0.06 -0.154 -0.9134 3032694 ChemDiv3_010435 CC(CCc1ccco1)NC(=O)c2cc3c(Cl)nc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K08 compound treatment 520.0 -764.0 -0.27 560.0 -119.0 -0.09 -0.256 -0.8955 3032733 ChemDiv3_010436 CCC(=O)Nc1cccc(c1)c2cn3cccnc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K09 compound treatment 640.0 -644.0 -0.23 440.0 -239.0 -0.18 -0.291 -0.994 3032735 ChemDiv3_010437 Cc1ccc2oc(=O)c3cnn(CC(=O)N4CCCCC4)c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K10 compound treatment 440.0 -844.0 -0.3 400.0 -279.0 -0.21 -0.3629 -0.9864 3032736 ChemDiv3_010438 COc1ccc(cc1NC(=O)C(C)C)c2cn3cccnc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K11 compound treatment 400.0 -884.0 -0.31 440.0 -239.0 -0.18 -0.3512 -0.9673 3032738 ChemDiv3_010439 COc1ccccc1Nc2c3CCCCc3nc4ccc(NC(=O)Cc5cccs5)cc24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K12 compound treatment 760.0 -524.0 -0.19 440.0 -239.0 -0.18 -0.2609 -1.0 3032739 ChemDiv3_010440 Clc1ccc(CSc2ccc(C=C3C(=O)NC(=O)NC3=O)o2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K13 compound treatment 320.0 -964.0 -0.34 320.0 -359.0 -0.28 -0.4364 -0.9942 3032741 ChemDiv3_010441 CCCN1C(C(=O)Nc2ccccc2C)c3cccc[n+]3CC1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K14 compound treatment 440.0 -844.0 -0.3 480.0 -199.0 -0.15 -0.3195 -0.951 3121196 ChemDiv3_010442 COc1cccc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c4cc(OC)ccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K15 compound treatment 560.0 -724.0 -0.26 800.0 121.0 0.09 -0.1157 -0.4234 3032743 ChemDiv3_010443 Cc1cc(on1)C(=O)Nc2cccc(Cl)c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K16 compound treatment 1280.0 -3.75 0.0 4600.0 3920.0 3.01 2.1278 0.7068 3121374 ChemDiv3_010444 CCSc1nc2NC3=C(C(c4cccs4)n2n1)C(=O)CCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K17 compound treatment 440.0 -844.0 -0.3 960.0 281.0 0.22 -0.0589 -0.1596 3032744 ChemDiv3_010445 Cc1noc(C(=O)N2CCCc3ccccc23)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K18 compound treatment 480.0 -804.0 -0.29 320.0 -359.0 -0.28 -0.3963 -0.9998 3121375 ChemDiv3_010446 COc1ccc(NC(=O)C2CC(=NO2)c3cccc(OC)c3)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K19 compound treatment 2160.0 876.0 0.31 2200.0 1520.0 1.17 1.0457 0.8652 3032746 ChemDiv3_010447 CC1CCN(CC1)C(=O)c2cc3c(C)nc4ccccc4c3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K20 compound treatment 720.0 -564.0 -0.2 6720.0 6040.0 4.64 3.1382 0.676 3121376 ChemDiv3_010448 Fc1ccc(cc1)C2=NOC(C2)C(=O)N3CCCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K21 compound treatment 480.0 -804.0 -0.29 5880.0 5200.0 3.99 2.622 0.6549 3032749 ChemDiv3_010449 COC(CNC(=O)c1cc2c(C)nc3ccccc3c2o1)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K22 compound treatment 1200.0 -83.8 -0.03 1280.0 601.0 0.46 0.3055 0.6602 3121377 ChemDiv3_010450 COc1ccc(OC)c(c1)C2=NOC(C2)C(=O)N(C)C3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K23 mock treatment 640.0 -644.0 -0.23 1200.0 521.0 0.4 0.1216 0.2638 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 K24 mock treatment 1880.0 596.0 0.21 440.0 -239.0 -0.18 0.02 0.0716 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L01 compound treatment 1080.0 -204.0 -0.07 1240.0 561.0 0.43 0.2536 0.5804 3121378 ChemDiv3_010451 Cc1ccc(Cn2nnc3c(=O)n(Cc4ccc(cc4)C(F)(F)F)cnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L02 compound treatment 1000.0 -284.0 -0.1 400.0 -279.0 -0.21 -0.2224 -0.9409 3032752 ChemDiv3_010452 O=C/1NN(C(=O)\C1=C\c2coc3ccccc3c2=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L03 compound treatment 8040.0 6760.0 2.4 3560.0 2880.0 2.21 3.2589 0.9992 3121379 ChemDiv3_010453 Clc1cccc(c1)n2nnc3c(=O)n(CC(=O)N4CCCc5ccccc45)cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L04 compound treatment 640.0 -644.0 -0.23 360.0 -319.0 -0.24 -0.3344 -0.9994 3032754 ChemDiv3_010454 Brc1ccc(NC(=O)Cn2c(=O)c3ccccc3n4nncc24)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L05 compound treatment 1280.0 -3.75 0.0 400.0 -279.0 -0.21 -0.1522 -0.7115 3121380 ChemDiv3_010455 COc1ccc2cc3c(NC(=O)Cc4cccc(c4)C(F)(F)F)n[nH]c3nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L06 compound treatment 960.0 -324.0 -0.11 400.0 -279.0 -0.21 -0.2325 -0.9575 3032757 ChemDiv3_010456 COc1ccc(cc1)c2nc(SCC(=O)N)c3Cc4ccccc4Oc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L07 compound treatment 760.0 -524.0 -0.19 680.0 1.38 0.0 -0.1306 -0.7031 3121381 ChemDiv3_010457 CC(C)CCNC(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L08 compound treatment 520.0 -764.0 -0.27 920.0 241.0 0.19 -0.0605 -0.1845 3032801 ChemDiv3_010458 COc1ccccc1NC(=O)c2oc3ccccc3c2NC(=O)CSCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L09 compound treatment 440.0 -844.0 -0.3 560.0 -119.0 -0.09 -0.276 -0.8823 3032759 ChemDiv3_010459 O=C(NCc1ccccc1)c2cc3CSc4ccccc4-c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L10 compound treatment 520.0 -764.0 -0.27 400.0 -279.0 -0.21 -0.3428 -0.9932 1477644 ChemDiv3_010460 CCOC(=O)c1oc2ccccc2c1NC(=O)c3ccc(cc3)S(=O)(=O)N(C)C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L11 compound treatment 480.0 -804.0 -0.29 480.0 -199.0 -0.15 -0.3094 -0.957 3032761 ChemDiv3_010461 CCSc1nnc(Cn2c(=O)sc3ccccc23)n1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L12 compound treatment 440.0 -844.0 -0.3 4880.0 4200.0 3.23 2.0691 0.6387 3121382 ChemDiv3_010462 OC(C1CCN(CC1)C(=O)c2cnn3ccccc23)(c4ccccc4)c5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L13 compound treatment 1000.0 -284.0 -0.1 1680.0 1000.0 0.77 0.4724 0.6093 3121383 ChemDiv3_010463 COc1ccc2[nH]c3c(=O)n(CCCC(=O)N4CCCC4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L14 compound treatment 480.0 -804.0 -0.29 400.0 -279.0 -0.21 -0.3529 -0.99 3032802 ChemDiv3_010464 CCCCn1c(CN2CCN(CC)CC2)nc3n(C)c(=O)[nH]c(=O)c13 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L15 compound treatment 520.0 -764.0 -0.27 440.0 -239.0 -0.18 -0.3211 -0.9818 3032803 ChemDiv3_010465 COc1cc(NC(=O)c2ccc3c(SCC(=O)O)c4CCCc4nc3c2)cc(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L16 compound treatment 440.0 -844.0 -0.3 360.0 -319.0 -0.24 -0.3846 -0.995 3032804 ChemDiv3_010466 CCN(C(=O)Cn1c(=O)n2nc(CCn3nc(C)cc3C)nc2c4ccccc14)c5cccc(C)c5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L17 compound treatment 720.0 -564.0 -0.2 400.0 -279.0 -0.21 -0.2927 -0.9994 3032806 ChemDiv3_010467 COc1ccc2[nH]c3c(=O)n(Cc4ccc(cc4)C(=O)NC5CC5)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L18 compound treatment 5080.0 3800.0 1.35 680.0 1.38 0.0 0.953 0.7077 3032807 ChemDiv3_010468 O=C(Cn1nc(Cc2cccnc2)c3ccccc3c1=O)N4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L19 compound treatment 560.0 -724.0 -0.26 440.0 -239.0 -0.18 -0.3111 -0.9863 3121384 ChemDiv3_010469 Cn1cccc1Cc2nnc(SCC(=O)N3CCCCC3)n2CCc4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L20 compound treatment 520.0 -764.0 -0.27 2360.0 1680.0 1.29 0.7212 0.5468 3121385 ChemDiv3_010470 Cn1c(=O)oc2cc(ccc12)S(=O)(=O)NCCC(=O)Nc3cccc(F)c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L21 compound treatment 1080.0 -204.0 -0.07 7560.0 6880.0 5.28 3.6845 0.6974 3032810 ChemDiv3_010471 Cn1cccc1Cc2nnc(SCC(=O)N3CCCc4ccccc34)n2c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L22 compound treatment 1000.0 -284.0 -0.1 560.0 -119.0 -0.09 -0.1356 -0.9988 3121386 ChemDiv3_010472 Cc1ccc(CN2CCSc3ccc(cc23)C(=O)Nc4ccc(F)cc4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L23 mock treatment 1000.0 -284.0 -0.1 6760.0 6080.0 4.67 3.2302 0.6917 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 L24 mock treatment 280.0 -1000.0 -0.36 600.0 -78.6 -0.06 -0.2945 -0.8153 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M01 compound treatment 1360.0 76.3 0.03 760.0 81.4 0.06 0.0633 0.9298 3032813 ChemDiv3_010473 CCOC(=O)N1CCC(CC1)c2nc3ccccn3c2C(=O)OCC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M02 compound treatment 360.0 -924.0 -0.33 680.0 1.38 0.0 -0.231 -0.7048 3121387 ChemDiv3_010474 Cc1ccc(cc1)n2c(=O)cc([nH]c2=O)N3CCc4ccccc34 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M03 compound treatment 1320.0 36.3 0.01 800.0 121.0 0.09 0.075 0.7971 3121388 ChemDiv3_010475 CCCn1c(CCC(=O)N2CCc3ccccc3C2)nc4cccnc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M04 compound treatment 960.0 -324.0 -0.11 920.0 241.0 0.19 0.0498 0.2285 3032815 ChemDiv3_010476 COC(=O)c1cc(=O)n(c2ccccc2)/c(=N/c3ccccc3)/s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M05 compound treatment 1800.0 516.0 0.18 1440.0 761.0 0.58 0.5428 0.8862 3121389 ChemDiv3_010477 COc1ccc(Cl)cc1NC(=O)c2cc3c(Cl)nc4ccc(C)cc4c3s2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M06 compound treatment 720.0 -564.0 -0.2 840.0 161.0 0.12 -0.0538 -0.2287 3032816 ChemDiv3_010478 CCNC(=O)CC1N(Cc2ccc(OC)cc2)C(=O)N(C1=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M07 compound treatment 880.0 -404.0 -0.14 560.0 -119.0 -0.09 -0.1657 -0.9761 3121390 ChemDiv3_010479 Clc1ccc2c(SCC(=O)N3CCCCCC3)c4CCCCc4nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M08 compound treatment 1040.0 -244.0 -0.09 440.0 -239.0 -0.18 -0.1907 -0.9413 3121391 ChemDiv3_010480 O=C(Nc1cccc(c1)c2cn3cccnc3n2)C4CCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M09 compound treatment 600.0 -684.0 -0.24 1160.0 481.0 0.37 0.0898 0.2032 3032819 ChemDiv3_010481 CC1CCN(CCCNC(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c23)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M10 compound treatment 1760.0 476.0 0.17 520.0 -159.0 -0.12 0.0334 0.1602 3121392 ChemDiv3_010482 O=C(CCC1CCCCC1)Nc2ccc(cc2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M11 compound treatment 3760.0 2480.0 0.88 720.0 41.4 0.03 0.6436 0.7322 3121393 ChemDiv3_010483 COc1ccc(Nc2c3CCCCc3nc4ccc(NC(=O)C5CC5)cc24)cc1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M12 compound treatment 960.0 -324.0 -0.11 1120.0 441.0 0.34 0.1584 0.4427 3032821 ChemDiv3_010484 CN1C(=O)/C(=C/c2ccc(SCc3ccccc3)o2)/SC1=S 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M13 compound treatment 680.0 -604.0 -0.21 1560.0 881.0 0.68 0.327 0.4608 3121394 ChemDiv3_010485 COc1ccc(cc1)N2C(C(=O)Nc3c(C)cccc3C)c4cccc[n+]4C2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M14 compound treatment 640.0 -644.0 -0.23 560.0 -119.0 -0.09 -0.2259 -0.9187 3032823 ChemDiv3_010486 COc1ccc(NC(=O)C2CCCN(C2)S(=O)(=O)c3ccc4n(C)c(=O)oc4c3)cc1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M15 compound treatment 1000.0 -284.0 -0.1 2800.0 2120.0 1.63 1.0804 0.6621 3121395 ChemDiv3_010487 CCc1ccc(NC(=O)c2cc(C)no2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M16 compound treatment 440.0 -844.0 -0.3 440.0 -239.0 -0.18 -0.3412 -0.9722 3121396 ChemDiv3_010488 COc1ccc(cc1)C2=NOC(C2)C(=O)Nc3ccc(C)cc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M17 compound treatment 1480.0 196.0 0.07 1800.0 1120.0 0.86 0.658 0.7618 3032826 ChemDiv3_010489 CCC(C)NC(=O)c1onc(C)c1Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M18 compound treatment 2720.0 1440.0 0.51 720.0 41.4 0.03 0.3827 0.7497 3121397 ChemDiv3_010490 COc1cccc(c1)C2=NOC(C2)C(=O)NCC3CCCO3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M19 compound treatment 920.0 -364.0 -0.13 3160.0 2480.0 1.91 1.2558 0.6577 3032828 ChemDiv3_010491 CCOC(=O)C1CCCN(C1)C(=O)c2cc3c(C)nc4ccccc4c3o2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M20 compound treatment 4200.0 2920.0 1.03 520.0 -159.0 -0.12 0.6454 0.6196 3032867 ChemDiv3_010492 Fc1ccc(cc1)C2=NOC(C2)C(=O)N3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M21 compound treatment 7240.0 5960.0 2.11 560.0 -119.0 -0.09 1.4297 0.676 3032869 ChemDiv3_010493 CN1CCN(CCNC(=O)c2cc3c(C)nc4ccccc4c3o2)CC1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M22 compound treatment 1080.0 -204.0 -0.07 840.0 161.0 0.12 0.0365 0.2544 3032870 ChemDiv3_010494 COc1ccc(OC)c(c1)C2=NOC(C2)C(=O)NCC=C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M23 mock treatment 640.0 -644.0 -0.23 640.0 -38.6 -0.03 -0.1824 -0.7923 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 M24 mock treatment 1840.0 556.0 0.2 1200.0 521.0 0.4 0.4226 0.9469 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N01 compound treatment 5800.0 4520.0 1.6 1000.0 321.0 0.25 1.3073 0.8065 3032871 ChemDiv3_010495 CCOC(=O)C(C)n1cnc2n(Cc3ccc(C)cc3)nnc2c1=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N02 compound treatment 1160.0 -124.0 -0.04 1360.0 681.0 0.52 0.3389 0.6455 3032873 ChemDiv3_010496 N=C/1N2N=CSC2=NC(=O)\C1=C\c3coc4ccccc4c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N03 compound treatment 800.0 -484.0 -0.17 320.0 -359.0 -0.28 -0.316 -0.9741 3032874 ChemDiv3_010497 Clc1cccc(c1)n2nnc3c(=O)n(CC(=O)NC4CCCCC4)cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N04 compound treatment 960.0 -324.0 -0.11 400.0 -279.0 -0.21 -0.2325 -0.9575 3121398 ChemDiv3_010498 COc1ccc2n(Cc3ccccc3)cc(c(=O)c2c1)S(=O)(=O)c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N05 compound treatment 1560.0 276.0 0.1 480.0 -199.0 -0.15 -0.0385 -0.2126 3032876 ChemDiv3_010499 Clc1c2CCCc2nc3cc(ccc13)C(=O)NCCC4=CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N06 compound treatment 360.0 -924.0 -0.33 1120.0 441.0 0.34 0.0079 0.0167 3121399 ChemDiv3_010500 Cc1nc2c3ccccc3n4c(CCCC(=O)O)nnc4n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N07 compound treatment 760.0 -524.0 -0.19 440.0 -239.0 -0.18 -0.2609 -1.0 3121400 ChemDiv3_010501 Cc1cccc(CN2CCC(CNC(=O)c3cc4c(=O)[nH]c5ccc(C)cc5c4s3)CC2)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N08 compound treatment 1240.0 -43.8 -0.02 920.0 241.0 0.19 0.1201 0.6456 3032878 ChemDiv3_010502 COc1ccccc1NC(=O)c2oc3ccccc3c2NC(=O)Cc4cccc(C)c4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N09 compound treatment 800.0 -484.0 -0.17 2360.0 1680.0 1.29 0.7914 0.6078 3121573 ChemDiv3_010503 COc1ccc2[nH]c3c(=O)n(CCC(=O)NCCc4ccc(OC)c(OC)c4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N10 compound treatment 720.0 -564.0 -0.2 880.0 201.0 0.15 -0.0321 -0.127 3032880 ChemDiv3_010504 COc1ccccc1NC(=O)Cn2c(=O)n(Cc3ccccn3)c(=O)c4sc5ccccc5c24 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N11 compound treatment 720.0 -564.0 -0.2 480.0 -199.0 -0.15 -0.2492 -0.991 3121574 ChemDiv3_010505 Cn1c(Cn2c(=O)sc3ccccc23)nnc1SCC(=O)NCc4ccccc4Cl 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N12 compound treatment 1000.0 -284.0 -0.1 360.0 -319.0 -0.24 -0.2441 -0.923 3032882 ChemDiv3_010506 Cc1ccccc1NC(=O)c2cnn3ccccc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N13 compound treatment 680.0 -604.0 -0.21 560.0 -119.0 -0.09 -0.2158 -0.9274 3121575 ChemDiv3_010507 Nc1cc(nn1S(=O)(=O)c2ccccc2)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N14 compound treatment 960.0 -324.0 -0.11 560.0 -119.0 -0.09 -0.1456 -0.9934 3121576 ChemDiv3_010508 CC(C)Cn1c(CN(Cc2ccccc2)Cc3ccccc3)nc4n(C)c(=O)[nH]c(=O)c14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N15 compound treatment 720.0 -564.0 -0.2 640.0 -38.6 -0.03 -0.1624 -0.8032 3032884 ChemDiv3_010509 CC1CCCC(NC(=O)c2ccc3c(SCC(=O)O)c4CCCc4nc3c2)C1C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N16 compound treatment 1120.0 -164.0 -0.06 440.0 -239.0 -0.18 -0.1706 -0.8878 3121577 ChemDiv3_010510 Clc1cccc(Nc2nnc(Cc3cccnc3)c4ccccc24)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N17 compound treatment 800.0 -484.0 -0.17 520.0 -159.0 -0.12 -0.2075 -0.9859 3121578 ChemDiv3_010511 COc1ccc2[nH]c3c(=O)n(Cc4ccc(cc4)C(=O)NCCc5ccc(C)cc5)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N18 compound treatment 600.0 -684.0 -0.24 1040.0 361.0 0.28 0.0247 0.0669 3032885 ChemDiv3_010512 CC1CN(CCN1c2ccc(C)cc2)C(=O)Cn3nc(Cc4cccnc4)c5ccccc5c3=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N19 compound treatment 680.0 -604.0 -0.21 720.0 41.4 0.03 -0.129 -0.5957 3121579 ChemDiv3_010513 Cn1cccc1Cc2nnc(SCC(=O)N3CCc4ccccc34)n2CCc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N20 compound treatment 1200.0 -83.8 -0.03 400.0 -279.0 -0.21 -0.1723 -0.7977 3032887 ChemDiv3_010514 CCn1c(=O)c(=O)n(CC)c2cc(ccc12)S(=O)(=O)NC3CCCCC3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N21 compound treatment 1480.0 196.0 0.07 840.0 161.0 0.12 0.1368 0.9628 3121580 ChemDiv3_010515 Cn1cccc1Cc2nnc(SCC(=O)Nc3ccc4OCOc4c3)n2c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N22 compound treatment 1440.0 156.0 0.06 760.0 81.4 0.06 0.0834 0.9982 3121581 ChemDiv3_010516 CCOc1ccc(NC(=O)c2ccc3SCCN(Cc4ccc(C)cc4)c3c2)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N23 mock treatment 480.0 -804.0 -0.29 720.0 41.4 0.03 -0.1792 -0.6245 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 N24 mock treatment 520.0 -764.0 -0.27 1520.0 841.0 0.65 0.2652 0.3786 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O01 compound treatment 360.0 -924.0 -0.33 280.0 -399.0 -0.31 -0.4481 -0.9994 3032891 ChemDiv3_010517 CCOC(=O)c1cn2nc(cc2nc1C3CCN(CC3)C(=O)OC(C)(C)C)c4ccc(OC)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O02 compound treatment 280.0 -1000.0 -0.36 280.0 -399.0 -0.31 -0.4682 -0.9972 3121582 ChemDiv3_010518 CCc1ccc2[nH]cc(c(=O)c2c1)S(=O)(=O)c3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O03 compound treatment 320.0 -964.0 -0.34 360.0 -319.0 -0.24 -0.4147 -0.9865 3032894 ChemDiv3_010519 CCCn1c(CCC(=O)N2CCc3ccccc23)nc4cccnc14 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O04 compound treatment 400.0 -884.0 -0.31 280.0 -399.0 -0.31 -0.4381 -0.9999 3121583 ChemDiv3_010520 CC/N=c/1\sc(cc(=O)n1CC)C(=O)OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O05 compound treatment 280.0 -1000.0 -0.36 240.0 -439.0 -0.34 -0.4899 -0.9996 3032940 ChemDiv3_010521 COc1cccc(c1)N2CCN(CC2)C(=O)c3cc4c(Cl)nc5ccc(C)cc5c4s3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O06 compound treatment 320.0 -964.0 -0.34 440.0 -239.0 -0.18 -0.3713 -0.9572 3032941 ChemDiv3_010522 CCc1ccc(NC(=O)CC2N(C3CC3)C(=O)N(C2=O)c4cccc(C)c4)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O07 compound treatment 360.0 -924.0 -0.33 560.0 -119.0 -0.09 -0.2961 -0.8706 3032943 ChemDiv3_010523 Clc1ccc2c(SCC(=O)NCCCN3CCCCCC3)c4CCCCc4nc2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O08 compound treatment 2240.0 956.0 0.34 280.0 -399.0 -0.31 0.0235 0.0514 3032944 ChemDiv3_010524 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2)c3cn4cccnc4n3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O09 compound treatment 2680.0 1400.0 0.5 360.0 -319.0 -0.24 0.1773 0.3209 3032946 ChemDiv3_010525 CCOC(=O)N1CCC(CC1)NC(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O10 compound treatment 400.0 -884.0 -0.31 360.0 -319.0 -0.24 -0.3946 -0.9925 3032947 ChemDiv3_010526 COCC(=O)Nc1ccc(cc1)c2cn3cccnc3n2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O11 compound treatment 360.0 -924.0 -0.33 240.0 -439.0 -0.34 -0.4698 -0.9999 3121584 ChemDiv3_010527 Brc1cc(N2CCCCC2)c3C(=O)c4ccccc4-c5onc1c53 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O12 compound treatment 320.0 -964.0 -0.34 480.0 -199.0 -0.15 -0.3496 -0.9338 3032949 ChemDiv3_010528 N=C/1N2C=CSC2=NC(=O)\C1=C/c3ccc(SCc4ccccc4)o3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O13 compound treatment 320.0 -964.0 -0.34 440.0 -239.0 -0.18 -0.3713 -0.9572 3121585 ChemDiv3_010529 C/C(=C\C(=N\c1ccc2OCOc2c1)\c3ccccn3)/c4ccccn4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O14 compound treatment 280.0 -1000.0 -0.36 400.0 -279.0 -0.21 -0.403 -0.9703 3121586 ChemDiv3_010530 CN1CC(=O)N=C1NC(=O)C2CCCN(C2)S(=O)(=O)c3ccc4n(C)c(=O)oc4c3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O15 compound treatment 320.0 -964.0 -0.34 240.0 -439.0 -0.34 -0.4799 -1.0 3032951 ChemDiv3_010531 Cc1cc(on1)C(=O)NC2CCCC2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O16 compound treatment 320.0 -964.0 -0.34 400.0 -279.0 -0.21 -0.393 -0.9745 3032952 ChemDiv3_010532 COc1ccc(cc1)C2=NOC(C2)C(=O)N(C)Cc3ccccc3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O17 compound treatment 400.0 -884.0 -0.31 280.0 -399.0 -0.31 -0.4381 -0.9999 3121587 ChemDiv3_010533 CN(C(=O)c1onc(C)c1Cl)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O18 compound treatment 320.0 -964.0 -0.34 280.0 -399.0 -0.31 -0.4581 -0.9985 3121588 ChemDiv3_010534 COc1ccccc1C2=NOC(C2)C(=O)Nc3ccccc3C(F)(F)F 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O19 compound treatment 320.0 -964.0 -0.34 480.0 -199.0 -0.15 -0.3496 -0.9338 3032955 ChemDiv3_010535 CN(C(=O)c1cc2c(C)nc3ccccc3c2o1)c4cc(Cl)ccc4C 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O20 compound treatment 320.0 -964.0 -0.34 320.0 -359.0 -0.28 -0.4364 -0.9942 3121589 ChemDiv3_010536 CCCNC(=O)C1CC(=NO1)c2ccc(F)cc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O21 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3121590 ChemDiv3_010537 CN(CCNC(=O)c1cc2c(C)nc3ccccc3c2o1)C4CCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O22 compound treatment 480.0 -804.0 -0.29 320.0 -359.0 -0.28 -0.3963 -0.9998 3032958 ChemDiv3_010538 Clc1ccc(cc1)n2nc3oc4ccccc4cc3c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O23 mock treatment 400.0 -884.0 -0.31 4720.0 4040.0 3.1 1.9722 0.6324 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 O24 mock treatment 640.0 -644.0 -0.23 560.0 -119.0 -0.09 -0.2259 -0.9187 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P01 compound treatment 320.0 -964.0 -0.34 200.0 -479.0 -0.37 -0.5016 -0.9994 3032960 ChemDiv3_010539 Fc1ccc(Cn2nnc3c(=O)n(Cc4ccc(F)cc4)cnc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P02 compound treatment 1760.0 476.0 0.17 240.0 -439.0 -0.34 -0.1186 -0.3149 3121591 ChemDiv3_010540 Cc1nn2c(=O)cc(CSc3nc4ccccc4[nH]3)nc2s1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P03 compound treatment 240.0 -1040.0 -0.37 320.0 -359.0 -0.28 -0.4565 -0.9894 3121592 ChemDiv3_010541 Clc1cccc(c1)n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P04 compound treatment 440.0 -844.0 -0.3 280.0 -399.0 -0.31 -0.428 -0.9999 3032964 ChemDiv3_010542 Cc1ccc(cc1)S(=O)(=O)c2cn(Cc3cccc(Cl)c3)c4cc5OCOc5cc4c2=O 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P05 compound treatment 6360.0 5080.0 1.8 360.0 -319.0 -0.24 1.1004 0.6055 3121593 ChemDiv3_010543 CCCC1CCC(CC1)C(=O)n2nc(N)c3cc4ccc(OC)cc4nc23 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P06 compound treatment 600.0 -684.0 -0.24 360.0 -319.0 -0.24 -0.3445 -1.0 3121594 ChemDiv3_010544 Cc1nc2c3ccccc3n4c(CCCC(=O)NC5CCCCC5)nnc4n2n1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P07 compound treatment 560.0 -724.0 -0.26 360.0 -319.0 -0.24 -0.3545 -0.9997 3033016 ChemDiv3_010545 Cc1ccc2[nH]c(=O)c3cc(sc3c2c1)C(=O)NCCCN4CCN(CC4)c5ccc(F)cc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P08 compound treatment 400.0 -884.0 -0.31 360.0 -319.0 -0.24 -0.3946 -0.9925 3033019 ChemDiv3_010546 COc1cccc(OCC(=O)Nc2c(oc3ccccc23)C(=O)Nc4ccccc4OC)c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P09 compound treatment 520.0 -764.0 -0.27 320.0 -359.0 -0.28 -0.3863 -1.0 3033021 ChemDiv3_010547 COc1ccc2[nH]c3c(=O)n(CCC(=O)NC4CCCCCC4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P10 compound treatment 3000.0 1720.0 0.61 240.0 -439.0 -0.34 0.1924 0.2765 3033023 ChemDiv3_010548 Clc1ccc(CNC(=O)c2cnn3ccccc23)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P11 compound treatment 400.0 -884.0 -0.31 320.0 -359.0 -0.28 -0.4164 -0.9979 3033025 ChemDiv3_010549 CCCSc1nnc(Cn2c(=O)sc3ccccc23)n1c4ccccc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P12 compound treatment 680.0 -604.0 -0.21 320.0 -359.0 -0.28 -0.3461 -0.9923 3033026 ChemDiv3_010550 COc1ccc(CCNC(=O)c2cnn3ccccc23)c(OC)c1OC 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P13 compound treatment 400.0 -884.0 -0.31 200.0 -479.0 -0.37 -0.4815 -0.9969 3033028 ChemDiv3_010551 CCS(=O)(=O)n1nc(cc1N)c2ccccc2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P14 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3121595 ChemDiv3_010552 CC1CN(Cc2nc3n(C)c(=O)[nH]c(=O)c3n2Cc4ccc(C)cc4)CC(C)O1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P15 compound treatment 360.0 -924.0 -0.33 240.0 -439.0 -0.34 -0.4698 -0.9999 3121596 ChemDiv3_010553 OC(=O)CSc1c2CCCc2nc3cc(ccc13)C(=O)NC4CCCCCC4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P16 compound treatment 280.0 -1000.0 -0.36 320.0 -359.0 -0.28 -0.4465 -0.9919 3033031 ChemDiv3_010554 C(c1ccncc1)c2nnc(N3CCC4(CC3)OCCO4)c5ccccc25 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P17 compound treatment 320.0 -964.0 -0.34 200.0 -479.0 -0.37 -0.5016 -0.9994 3121597 ChemDiv3_010555 COc1ccc2[nH]c3c(=O)n(CCCCC(=O)Nc4ccccc4)c(=S)[nH]c3c2c1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P18 compound treatment 440.0 -844.0 -0.3 200.0 -479.0 -0.37 -0.4715 -0.9948 3033033 ChemDiv3_010556 Clc1ccc(CCNC(=O)Cn2nc(Cc3cccnc3)c4ccccc4c2=O)cc1 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P19 compound treatment 360.0 -924.0 -0.33 240.0 -439.0 -0.34 -0.4698 -0.9999 3121598 ChemDiv3_010557 Cn1cccc1Cc2nnc(SCC(=O)Nc3ccc4OCCOc4c3)n2CCc5ccccc5 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P20 compound treatment 360.0 -924.0 -0.33 320.0 -359.0 -0.28 -0.4264 -0.9962 3033036 ChemDiv3_010558 CCn1c(=O)c(=O)n(CC)c2cc(ccc12)S(=O)(=O)NCc3cccs3 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P21 compound treatment 560.0 -724.0 -0.26 320.0 -359.0 -0.28 -0.3762 -0.9994 3121599 ChemDiv3_010559 Cn1cccc1Cc2nnc(SCC(=O)Nc3ccccc3C(F)(F)F)n2c4ccc(F)cc4 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P22 compound treatment 320.0 -964.0 -0.34 360.0 -319.0 -0.24 -0.4147 -0.9865 3121773 ChemDiv3_010560 CCN1CCN(CC1)C(=O)c2ccc3SCCN(Cc4ccc(C)cc4)c3c2 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P23 mock treatment 1160.0 -124.0 -0.04 320.0 -359.0 -0.28 -0.2257 -0.8096 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.2030 P24 mock treatment 280.0 -1000.0 -0.36 360.0 -319.0 -0.24 -0.4248 -0.9832 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A01 mock treatment 520.0 -926.0 -0.33 200.0 -492.0 -0.38 -0.4996 -0.9976 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A02 mock treatment 200.0 -1250.0 -0.44 280.0 -412.0 -0.32 -0.5364 -0.9866 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A03 mock treatment 320.0 -1130.0 -0.4 320.0 -372.0 -0.29 -0.4846 -0.9866 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A04 mock treatment 360.0 -1090.0 -0.39 240.0 -452.0 -0.35 -0.518 -0.9987 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A05 mock treatment 760.0 -686.0 -0.24 2880.0 2190.0 1.68 1.0155 0.5984 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A06 mock treatment 400.0 -1050.0 -0.37 520.0 -172.0 -0.13 -0.356 -0.9036 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A07 mock treatment 4120.0 2670.0 0.95 680.0 -12.4 -0.01 0.664 0.7 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A08 mock treatment 1120.0 -326.0 -0.12 200.0 -492.0 -0.38 -0.3491 -0.883 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A09 mock treatment 240.0 -1210.0 -0.43 4200.0 3510.0 2.69 1.6016 0.5874 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A10 mock treatment 440.0 -1010.0 -0.36 280.0 -412.0 -0.32 -0.4762 -0.9982 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A11 mock treatment 600.0 -846.0 -0.3 280.0 -412.0 -0.32 -0.4361 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A12 mock treatment 480.0 -966.0 -0.34 280.0 -412.0 -0.32 -0.4662 -0.9992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A13 mock treatment 520.0 -926.0 -0.33 5600.0 4910.0 3.77 2.4318 0.643 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A14 mock treatment 440.0 -1010.0 -0.36 800.0 108.0 0.08 -0.194 -0.5295 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A15 mock treatment 680.0 -766.0 -0.27 2520.0 1830.0 1.4 0.8 0.5598 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A16 mock treatment 480.0 -966.0 -0.34 1560.0 868.0 0.67 0.2286 0.3053 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A17 mock treatment 400.0 -1050.0 -0.37 280.0 -412.0 -0.32 -0.4863 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A18 mock treatment 4120.0 2670.0 0.95 400.0 -292.0 -0.22 0.512 0.5253 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A19 mock treatment 560.0 -886.0 -0.31 280.0 -412.0 -0.32 -0.4461 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A20 mock treatment 2640.0 1190.0 0.42 1560.0 868.0 0.67 0.7705 0.9761 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A21 mock treatment 4680.0 3230.0 1.15 2040.0 1350.0 1.03 1.5428 0.9987 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A22 mock treatment 2920.0 1470.0 0.52 280.0 -412.0 -0.32 0.1458 0.2386 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A23 mock treatment 560.0 -886.0 -0.31 240.0 -452.0 -0.35 -0.4679 -0.9988 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base A24 mock treatment 6240.0 4790.0 1.7 160.0 -532.0 -0.41 0.9135 0.5223 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B01 mock treatment 920.0 -526.0 -0.19 440.0 -252.0 -0.19 -0.269 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B02 mock treatment 160.0 -1290.0 -0.46 240.0 -452.0 -0.35 -0.5682 -0.9909 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B03 mock treatment 200.0 -1250.0 -0.44 240.0 -452.0 -0.35 -0.5582 -0.9929 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B04 mock treatment 560.0 -886.0 -0.31 1920.0 1230.0 0.94 0.4441 0.4471 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B05 mock treatment 400.0 -1050.0 -0.37 400.0 -292.0 -0.22 -0.4211 -0.971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B06 mock treatment 3800.0 2350.0 0.84 280.0 -412.0 -0.32 0.3666 0.4105 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B07 mock treatment 3680.0 2230.0 0.79 2640.0 1950.0 1.5 1.6176 0.9559 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B08 mock treatment 360.0 -1090.0 -0.39 480.0 -212.0 -0.16 -0.3877 -0.9268 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B09 mock treatment 920.0 -526.0 -0.19 560.0 -132.0 -0.1 -0.2038 -0.9592 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B10 mock treatment 200.0 -1250.0 -0.44 400.0 -292.0 -0.22 -0.4713 -0.9507 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B11 mock treatment 240.0 -1210.0 -0.43 1040.0 348.0 0.27 -0.1138 -0.2258 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B12 mock treatment 240.0 -1210.0 -0.43 800.0 108.0 0.08 -0.2441 -0.5603 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B13 mock treatment 280.0 -1170.0 -0.41 3240.0 2550.0 1.96 1.0905 0.5455 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B14 mock treatment 800.0 -646.0 -0.23 520.0 -172.0 -0.13 -0.2557 -0.966 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B15 mock treatment 320.0 -1130.0 -0.4 560.0 -132.0 -0.1 -0.3543 -0.8597 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B16 mock treatment 560.0 -886.0 -0.31 1480.0 788.0 0.6 0.2053 0.3012 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B17 mock treatment 3640.0 2190.0 0.78 200.0 -492.0 -0.38 0.283 0.3271 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B18 mock treatment 6560.0 5110.0 1.81 640.0 -52.4 -0.04 1.2543 0.6913 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B19 mock treatment 4360.0 2910.0 1.03 920.0 228.0 0.17 0.8545 0.8151 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B20 mock treatment 720.0 -726.0 -0.26 520.0 -172.0 -0.13 -0.2757 -0.9521 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B21 mock treatment 360.0 -1090.0 -0.39 4440.0 3750.0 2.88 1.762 0.607 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B22 mock treatment 560.0 -886.0 -0.31 1120.0 428.0 0.33 0.0099 0.0217 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B23 mock treatment 400.0 -1050.0 -0.37 960.0 268.0 0.21 -0.1171 -0.2762 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base B24 mock treatment 560.0 -886.0 -0.31 240.0 -452.0 -0.35 -0.4679 -0.9988 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C01 mock treatment 680.0 -766.0 -0.27 280.0 -412.0 -0.32 -0.416 -0.9971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C02 mock treatment 240.0 -1210.0 -0.43 240.0 -452.0 -0.35 -0.5481 -0.9946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C03 mock treatment 360.0 -1090.0 -0.39 280.0 -412.0 -0.32 -0.4963 -0.9953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C04 mock treatment 1000.0 -446.0 -0.16 320.0 -372.0 -0.29 -0.3141 -0.9611 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C05 mock treatment 360.0 -1090.0 -0.39 240.0 -452.0 -0.35 -0.518 -0.9987 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C06 mock treatment 480.0 -966.0 -0.34 280.0 -412.0 -0.32 -0.4662 -0.9992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C07 mock treatment 880.0 -566.0 -0.2 240.0 -452.0 -0.35 -0.3876 -0.9661 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C08 mock treatment 320.0 -1130.0 -0.4 280.0 -412.0 -0.32 -0.5063 -0.9934 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C09 mock treatment 400.0 -1050.0 -0.37 200.0 -492.0 -0.38 -0.5297 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C10 mock treatment 400.0 -1050.0 -0.37 240.0 -452.0 -0.35 -0.508 -0.9995 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C11 mock treatment 360.0 -1090.0 -0.39 400.0 -292.0 -0.22 -0.4312 -0.967 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C12 mock treatment 320.0 -1130.0 -0.4 280.0 -412.0 -0.32 -0.5063 -0.9934 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C13 mock treatment 320.0 -1130.0 -0.4 240.0 -452.0 -0.35 -0.5281 -0.9976 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C14 mock treatment 280.0 -1170.0 -0.41 280.0 -412.0 -0.32 -0.5164 -0.9913 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C15 mock treatment 320.0 -1130.0 -0.4 640.0 -52.4 -0.04 -0.3109 -0.7744 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C16 mock treatment 400.0 -1050.0 -0.37 280.0 -412.0 -0.32 -0.4863 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C17 mock treatment 480.0 -966.0 -0.34 320.0 -372.0 -0.29 -0.4445 -0.9959 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C18 mock treatment 2480.0 1030.0 0.37 520.0 -172.0 -0.13 0.1658 0.4251 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C19 mock treatment 360.0 -1090.0 -0.39 320.0 -372.0 -0.29 -0.4746 -0.9892 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C20 mock treatment 1200.0 -246.0 -0.09 3600.0 2910.0 2.23 1.5167 0.6789 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C21 mock treatment 960.0 -486.0 -0.17 4240.0 3550.0 2.72 1.8039 0.661 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C22 mock treatment 400.0 -1050.0 -0.37 4200.0 3510.0 2.69 1.6417 0.604 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C23 mock treatment 3680.0 2230.0 0.79 320.0 -372.0 -0.29 0.3582 0.4252 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base C24 mock treatment 240.0 -1210.0 -0.43 320.0 -372.0 -0.29 -0.5047 -0.9808 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D01 mock treatment 240.0 -1210.0 -0.43 200.0 -492.0 -0.38 -0.5698 -0.9981 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D02 mock treatment 1960.0 514.0 0.18 200.0 -492.0 -0.38 -0.1384 -0.3297 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D03 mock treatment 400.0 -1050.0 -0.37 320.0 -372.0 -0.29 -0.4646 -0.9917 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D04 mock treatment 2240.0 794.0 0.28 400.0 -292.0 -0.22 0.0404 0.1122 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D05 mock treatment 320.0 -1130.0 -0.4 200.0 -492.0 -0.38 -0.5498 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D06 mock treatment 400.0 -1050.0 -0.37 280.0 -412.0 -0.32 -0.4863 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D07 mock treatment 280.0 -1170.0 -0.41 1400.0 708.0 0.54 0.0916 0.1342 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D08 mock treatment 320.0 -1130.0 -0.4 280.0 -412.0 -0.32 -0.5063 -0.9934 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D09 mock treatment 280.0 -1170.0 -0.41 200.0 -492.0 -0.38 -0.5598 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D10 mock treatment 440.0 -1010.0 -0.36 200.0 -492.0 -0.38 -0.5197 -0.9996 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D11 mock treatment 200.0 -1250.0 -0.44 280.0 -412.0 -0.32 -0.5364 -0.9866 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D12 mock treatment 240.0 -1210.0 -0.43 240.0 -452.0 -0.35 -0.5481 -0.9946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D13 mock treatment 360.0 -1090.0 -0.39 200.0 -492.0 -0.38 -0.5397 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D14 mock treatment 240.0 -1210.0 -0.43 240.0 -452.0 -0.35 -0.5481 -0.9946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D15 mock treatment 280.0 -1170.0 -0.41 200.0 -492.0 -0.38 -0.5598 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D16 mock treatment 320.0 -1130.0 -0.4 280.0 -412.0 -0.32 -0.5063 -0.9934 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D17 mock treatment 3360.0 1910.0 0.68 200.0 -492.0 -0.38 0.2128 0.2738 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D18 mock treatment 3240.0 1790.0 0.64 200.0 -492.0 -0.38 0.1827 0.2468 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D19 mock treatment 2600.0 1150.0 0.41 200.0 -492.0 -0.38 0.0221 0.0398 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D20 mock treatment 6600.0 5150.0 1.83 1920.0 1230.0 0.94 1.9592 0.9525 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D21 mock treatment 6160.0 4710.0 1.67 240.0 -452.0 -0.35 0.9369 0.5485 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D22 mock treatment 400.0 -1050.0 -0.37 320.0 -372.0 -0.29 -0.4646 -0.9917 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D23 mock treatment 3240.0 1790.0 0.64 1000.0 308.0 0.24 0.617 0.9089 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base D24 mock treatment 440.0 -1010.0 -0.36 3440.0 2750.0 2.11 1.2392 0.5792 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E01 mock treatment 320.0 -1130.0 -0.4 600.0 -92.4 -0.07 -0.3326 -0.8199 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E02 mock treatment 4880.0 3430.0 1.22 1040.0 348.0 0.27 1.0501 0.842 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E03 mock treatment 5080.0 3630.0 1.29 2160.0 1470.0 1.13 1.7082 0.9977 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E04 mock treatment 3560.0 2110.0 0.75 320.0 -372.0 -0.29 0.3281 0.4088 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E05 mock treatment 1200.0 -246.0 -0.09 480.0 -212.0 -0.16 -0.177 -0.9571 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E06 mock treatment 1400.0 -46.0 -0.02 1640.0 948.0 0.73 0.5029 0.6911 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E07 mock treatment 2080.0 634.0 0.22 2160.0 1470.0 1.13 0.9557 0.8318 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E08 mock treatment 1080.0 -366.0 -0.13 1680.0 988.0 0.76 0.4443 0.5776 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E09 mock treatment 2640.0 1190.0 0.42 1440.0 748.0 0.57 0.7053 0.9888 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E10 mock treatment 4000.0 2550.0 0.91 320.0 -372.0 -0.29 0.4385 0.4615 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E11 mock treatment 1400.0 -46.0 -0.02 320.0 -372.0 -0.29 -0.2137 -0.7463 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E12 mock treatment 640.0 -806.0 -0.29 720.0 27.6 0.02 -0.1872 -0.653 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E13 mock treatment 1920.0 474.0 0.17 400.0 -292.0 -0.22 -0.0399 -0.1421 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E14 mock treatment 800.0 -646.0 -0.23 1920.0 1230.0 0.94 0.5043 0.52 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E15 mock treatment 920.0 -526.0 -0.19 2760.0 2070.0 1.59 0.9905 0.6197 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E16 mock treatment 2640.0 1190.0 0.42 2480.0 1790.0 1.37 1.2699 0.8842 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E17 mock treatment 2200.0 754.0 0.27 5000.0 4310.0 3.31 2.5275 0.7618 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E18 mock treatment 760.0 -686.0 -0.24 320.0 -372.0 -0.29 -0.3743 -0.9968 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E19 mock treatment 640.0 -806.0 -0.29 1640.0 948.0 0.73 0.3122 0.3994 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E20 mock treatment 880.0 -566.0 -0.2 360.0 -332.0 -0.26 -0.3224 -0.993 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E21 mock treatment 1680.0 234.0 0.08 1120.0 428.0 0.33 0.2908 0.8589 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E22 mock treatment 2760.0 1310.0 0.47 1800.0 1110.0 0.85 0.9309 0.96 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E23 mock treatment 3760.0 2310.0 0.82 360.0 -332.0 -0.26 0.4 0.4653 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base E24 mock treatment 960.0 -486.0 -0.17 1040.0 348.0 0.27 0.0668 0.2102 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F01 mock treatment 1680.0 234.0 0.08 240.0 -452.0 -0.35 -0.1869 -0.5234 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F02 mock treatment 1080.0 -366.0 -0.13 2400.0 1710.0 1.31 0.8352 0.634 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F03 mock treatment 600.0 -846.0 -0.3 1120.0 428.0 0.33 0.0199 0.0447 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F04 mock treatment 480.0 -966.0 -0.34 2640.0 1950.0 1.5 0.8149 0.5313 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F05 mock treatment 960.0 -486.0 -0.17 2680.0 1990.0 1.53 0.9571 0.6232 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F06 mock treatment 1040.0 -406.0 -0.14 160.0 -532.0 -0.41 -0.3909 -0.9019 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F07 mock treatment 2560.0 1110.0 0.4 440.0 -252.0 -0.19 0.1424 0.3235 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F08 mock treatment 360.0 -1090.0 -0.39 1840.0 1150.0 0.88 0.3505 0.3646 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F09 mock treatment 1720.0 274.0 0.1 200.0 -492.0 -0.38 -0.1986 -0.5088 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F10 mock treatment 2600.0 1150.0 0.41 1560.0 868.0 0.67 0.7604 0.9727 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F11 mock treatment 400.0 -1050.0 -0.37 840.0 148.0 0.11 -0.1823 -0.4698 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F12 mock treatment 320.0 -1130.0 -0.4 1400.0 708.0 0.54 0.1017 0.1508 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F13 mock treatment 1000.0 -446.0 -0.16 880.0 188.0 0.14 -0.0101 -0.047 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F14 mock treatment 720.0 -726.0 -0.26 760.0 67.6 0.05 -0.1454 -0.5535 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F15 mock treatment 760.0 -686.0 -0.24 1760.0 1070.0 0.82 0.4075 0.4766 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F16 mock treatment 680.0 -766.0 -0.27 920.0 228.0 0.17 -0.0686 -0.2124 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F17 mock treatment 960.0 -486.0 -0.17 320.0 -372.0 -0.29 -0.3241 -0.9707 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F18 mock treatment 880.0 -566.0 -0.2 280.0 -412.0 -0.32 -0.3659 -0.9759 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F19 mock treatment 2720.0 1270.0 0.45 1920.0 1230.0 0.94 0.986 0.9433 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F20 mock treatment 3720.0 2270.0 0.81 880.0 188.0 0.14 0.6722 0.8204 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F21 mock treatment 2600.0 1150.0 0.41 400.0 -292.0 -0.22 0.1307 0.28 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F22 mock treatment 1480.0 34.0 0.01 2200.0 1510.0 1.16 0.8269 0.7144 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F23 mock treatment 1400.0 -46.0 -0.02 520.0 -172.0 -0.13 -0.1051 -0.7884 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base F24 mock treatment 520.0 -926.0 -0.33 280.0 -412.0 -0.32 -0.4562 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G01 mock treatment 320.0 -1130.0 -0.4 320.0 -372.0 -0.29 -0.4846 -0.9866 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G02 mock treatment 4040.0 2590.0 0.92 440.0 -252.0 -0.19 0.5136 0.5462 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G03 mock treatment 400.0 -1050.0 -0.37 480.0 -212.0 -0.16 -0.3777 -0.9318 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G04 mock treatment 480.0 -966.0 -0.34 360.0 -332.0 -0.26 -0.4228 -0.9895 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G05 mock treatment 2600.0 1150.0 0.41 1440.0 748.0 0.57 0.6953 0.9863 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G06 mock treatment 920.0 -526.0 -0.19 1120.0 428.0 0.33 0.1002 0.2653 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G07 mock treatment 1360.0 -86.0 -0.03 840.0 148.0 0.11 0.0585 0.4988 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G08 mock treatment 840.0 -606.0 -0.21 1920.0 1230.0 0.94 0.5144 0.5321 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G09 mock treatment 3080.0 1630.0 0.58 440.0 -252.0 -0.19 0.2728 0.4464 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G10 mock treatment 5120.0 3670.0 1.3 320.0 -372.0 -0.29 0.7194 0.5392 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G11 mock treatment 680.0 -766.0 -0.27 1400.0 708.0 0.54 0.192 0.316 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G12 mock treatment 1960.0 514.0 0.18 5520.0 4830.0 3.71 2.7496 0.741 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G13 mock treatment 1880.0 434.0 0.15 560.0 -132.0 -0.1 0.037 0.2004 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G14 mock treatment 520.0 -926.0 -0.33 360.0 -332.0 -0.26 -0.4127 -0.9922 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G15 mock treatment 1240.0 -206.0 -0.07 2000.0 1310.0 1.0 0.6581 0.6539 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G16 mock treatment 680.0 -766.0 -0.27 800.0 108.0 0.08 -0.1338 -0.4709 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G17 mock treatment 2200.0 754.0 0.27 440.0 -252.0 -0.19 0.0521 0.1577 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G18 mock treatment 600.0 -846.0 -0.3 840.0 148.0 0.11 -0.1321 -0.4118 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G19 mock treatment 1320.0 -126.0 -0.04 480.0 -212.0 -0.16 -0.1469 -0.8689 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G20 mock treatment 1280.0 -166.0 -0.06 600.0 -92.4 -0.07 -0.0918 -0.9957 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G21 mock treatment 4160.0 2710.0 0.96 5480.0 4790.0 3.68 3.2798 0.8632 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G22 mock treatment 6080.0 4630.0 1.64 360.0 -332.0 -0.26 0.9819 0.5903 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G23 mock treatment 3680.0 2230.0 0.79 2800.0 2110.0 1.62 1.7045 0.9461 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base G24 mock treatment 360.0 -1090.0 -0.39 680.0 -12.4 -0.01 -0.2792 -0.7244 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H01 mock treatment 320.0 -1130.0 -0.4 4400.0 3710.0 2.85 1.7302 0.602 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H02 mock treatment 800.0 -646.0 -0.23 760.0 67.6 0.05 -0.1254 -0.5335 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H03 mock treatment 4840.0 3390.0 1.2 1040.0 348.0 0.27 1.04 0.8434 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H04 mock treatment 800.0 -646.0 -0.23 480.0 -212.0 -0.16 -0.2774 -0.9861 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H05 mock treatment 5000.0 3550.0 1.26 1480.0 788.0 0.6 1.319 0.9433 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H06 mock treatment 520.0 -926.0 -0.33 2880.0 2190.0 1.68 0.9553 0.5582 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H07 mock treatment 1240.0 -206.0 -0.07 720.0 27.6 0.02 -0.0367 -0.4824 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H08 mock treatment 640.0 -806.0 -0.29 1160.0 468.0 0.36 0.0516 0.1125 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H09 mock treatment 2320.0 874.0 0.31 760.0 67.6 0.05 0.2559 0.8141 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H10 mock treatment 600.0 -846.0 -0.3 440.0 -252.0 -0.19 -0.3493 -0.9776 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H11 mock treatment 720.0 -726.0 -0.26 440.0 -252.0 -0.19 -0.3191 -0.9902 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H12 mock treatment 680.0 -766.0 -0.27 640.0 -52.4 -0.04 -0.2206 -0.8031 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H13 mock treatment 440.0 -1010.0 -0.36 1600.0 908.0 0.7 0.2403 0.307 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H14 mock treatment 1080.0 -366.0 -0.13 520.0 -172.0 -0.13 -0.1854 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H15 mock treatment 1760.0 314.0 0.11 280.0 -412.0 -0.32 -0.1451 -0.4324 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H16 mock treatment 400.0 -1050.0 -0.37 2720.0 2030.0 1.56 0.8383 0.5239 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H17 mock treatment 2120.0 674.0 0.24 560.0 -132.0 -0.1 0.0972 0.374 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H18 mock treatment 480.0 -966.0 -0.34 440.0 -252.0 -0.19 -0.3794 -0.9636 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H19 mock treatment 600.0 -846.0 -0.3 320.0 -372.0 -0.29 -0.4144 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H20 mock treatment 640.0 -806.0 -0.29 560.0 -132.0 -0.1 -0.2741 -0.9031 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H21 mock treatment 960.0 -486.0 -0.17 2000.0 1310.0 1.0 0.5879 0.5772 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H22 mock treatment 4360.0 2910.0 1.03 760.0 67.6 0.05 0.7676 0.7417 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H23 mock treatment 760.0 -686.0 -0.24 360.0 -332.0 -0.26 -0.3525 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base H24 mock treatment 5160.0 3710.0 1.32 4160.0 3470.0 2.66 2.814 0.9474 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I01 mock treatment 2080.0 634.0 0.22 320.0 -372.0 -0.29 -0.0431 -0.1186 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I02 mock treatment 1280.0 -166.0 -0.06 360.0 -332.0 -0.26 -0.2221 -0.848 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I03 mock treatment 1000.0 -446.0 -0.16 320.0 -372.0 -0.29 -0.3141 -0.9611 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I04 mock treatment 560.0 -886.0 -0.31 280.0 -412.0 -0.32 -0.4461 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I05 mock treatment 520.0 -926.0 -0.33 840.0 148.0 0.11 -0.1522 -0.4379 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I06 mock treatment 560.0 -886.0 -0.31 4360.0 3670.0 2.82 1.7687 0.6243 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I07 mock treatment 1440.0 -6.04 0.0 4680.0 3990.0 3.06 2.1632 0.7066 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I08 mock treatment 440.0 -1010.0 -0.36 680.0 -12.4 -0.01 -0.2591 -0.7257 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I09 mock treatment 320.0 -1130.0 -0.4 280.0 -412.0 -0.32 -0.5063 -0.9934 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I10 mock treatment 480.0 -966.0 -0.34 320.0 -372.0 -0.29 -0.4445 -0.9959 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I11 mock treatment 400.0 -1050.0 -0.37 280.0 -412.0 -0.32 -0.4863 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I12 mock treatment 480.0 -966.0 -0.34 1040.0 348.0 0.27 -0.0536 -0.1235 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I13 mock treatment 360.0 -1090.0 -0.39 320.0 -372.0 -0.29 -0.4746 -0.9892 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I14 mock treatment 360.0 -1090.0 -0.39 4440.0 3750.0 2.88 1.762 0.607 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I15 mock treatment 840.0 -606.0 -0.21 400.0 -292.0 -0.22 -0.3108 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I16 mock treatment 440.0 -1010.0 -0.36 280.0 -412.0 -0.32 -0.4762 -0.9982 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I17 mock treatment 1160.0 -286.0 -0.1 600.0 -92.4 -0.07 -0.1219 -0.9847 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I18 mock treatment 400.0 -1050.0 -0.37 400.0 -292.0 -0.22 -0.4211 -0.971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I19 mock treatment 360.0 -1090.0 -0.39 4040.0 3350.0 2.57 1.5448 0.5945 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I20 mock treatment 320.0 -1130.0 -0.4 5640.0 4950.0 3.8 2.4034 0.6293 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I21 mock treatment 960.0 -486.0 -0.17 200.0 -492.0 -0.38 -0.3892 -0.9368 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I22 mock treatment 3560.0 2110.0 0.75 1000.0 308.0 0.24 0.6972 0.8868 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I23 mock treatment 360.0 -1090.0 -0.39 320.0 -372.0 -0.29 -0.4746 -0.9892 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base I24 mock treatment 360.0 -1090.0 -0.39 4720.0 4030.0 3.09 1.914 0.6143 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J01 mock treatment 7600.0 6150.0 2.18 320.0 -372.0 -0.29 1.3415 0.6093 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J02 mock treatment 4160.0 2710.0 0.96 240.0 -452.0 -0.35 0.4352 0.4252 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J03 mock treatment 400.0 -1050.0 -0.37 440.0 -252.0 -0.19 -0.3994 -0.9541 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J04 mock treatment 3480.0 2030.0 0.72 320.0 -372.0 -0.29 0.308 0.3969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J05 mock treatment 1080.0 -366.0 -0.13 3280.0 2590.0 1.99 1.3129 0.6595 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J06 mock treatment 1720.0 274.0 0.1 320.0 -372.0 -0.29 -0.1334 -0.4419 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J07 mock treatment 280.0 -1170.0 -0.41 360.0 -332.0 -0.26 -0.4729 -0.9731 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J08 mock treatment 5280.0 3830.0 1.36 680.0 -12.4 -0.01 0.955 0.7021 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J09 mock treatment 680.0 -766.0 -0.27 200.0 -492.0 -0.38 -0.4595 -0.9869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J10 mock treatment 7000.0 5550.0 1.97 800.0 108.0 0.08 1.4516 0.7361 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J11 mock treatment 360.0 -1090.0 -0.39 760.0 67.6 0.05 -0.2357 -0.6064 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J12 mock treatment 360.0 -1090.0 -0.39 120.0 -572.0 -0.44 -0.5832 -0.9978 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J13 mock treatment 320.0 -1130.0 -0.4 160.0 -532.0 -0.41 -0.5715 -0.9999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J14 mock treatment 280.0 -1170.0 -0.41 240.0 -452.0 -0.35 -0.5381 -0.9962 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J15 mock treatment 280.0 -1170.0 -0.41 600.0 -92.4 -0.07 -0.3427 -0.8165 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J16 mock treatment 320.0 -1130.0 -0.4 600.0 -92.4 -0.07 -0.3326 -0.8199 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J17 mock treatment 400.0 -1050.0 -0.37 280.0 -412.0 -0.32 -0.4863 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J18 mock treatment 320.0 -1130.0 -0.4 360.0 -332.0 -0.26 -0.4629 -0.9766 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J19 mock treatment 320.0 -1130.0 -0.4 400.0 -292.0 -0.22 -0.4412 -0.9629 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J20 mock treatment 280.0 -1170.0 -0.41 360.0 -332.0 -0.26 -0.4729 -0.9731 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J21 mock treatment 240.0 -1210.0 -0.43 240.0 -452.0 -0.35 -0.5481 -0.9946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J22 mock treatment 1040.0 -406.0 -0.14 240.0 -452.0 -0.35 -0.3475 -0.924 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J23 mock treatment 6160.0 4710.0 1.67 1840.0 1150.0 0.88 1.8054 0.9552 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base J24 mock treatment 1040.0 -406.0 -0.14 680.0 -12.4 -0.01 -0.1086 -0.7523 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K01 mock treatment 8360.0 6910.0 2.45 680.0 -12.4 -0.01 1.7276 0.7044 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K02 mock treatment 1000.0 -446.0 -0.16 1520.0 828.0 0.64 0.3374 0.5153 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K03 mock treatment 680.0 -766.0 -0.27 640.0 -52.4 -0.04 -0.2206 -0.8031 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K04 mock treatment 2640.0 1190.0 0.42 440.0 -252.0 -0.19 0.1625 0.3488 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K05 mock treatment 680.0 -766.0 -0.27 2560.0 1870.0 1.43 0.8217 0.5631 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K06 mock treatment 880.0 -566.0 -0.2 240.0 -452.0 -0.35 -0.3876 -0.9661 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K07 mock treatment 400.0 -1050.0 -0.37 320.0 -372.0 -0.29 -0.4646 -0.9917 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K08 mock treatment 1040.0 -406.0 -0.14 400.0 -292.0 -0.22 -0.2606 -0.977 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K09 mock treatment 1600.0 154.0 0.05 320.0 -372.0 -0.29 -0.1636 -0.5619 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K10 mock treatment 3960.0 2510.0 0.89 360.0 -332.0 -0.26 0.4502 0.4853 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K11 mock treatment 760.0 -686.0 -0.24 720.0 27.6 0.02 -0.1571 -0.6432 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K12 mock treatment 640.0 -806.0 -0.29 280.0 -412.0 -0.32 -0.4261 -0.9987 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K13 mock treatment 720.0 -726.0 -0.26 400.0 -292.0 -0.22 -0.3409 -0.9977 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K14 mock treatment 840.0 -606.0 -0.21 280.0 -412.0 -0.32 -0.3759 -0.9822 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K15 mock treatment 520.0 -926.0 -0.33 400.0 -292.0 -0.22 -0.391 -0.9828 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K16 mock treatment 520.0 -926.0 -0.33 400.0 -292.0 -0.22 -0.391 -0.9828 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K17 mock treatment 960.0 -486.0 -0.17 320.0 -372.0 -0.29 -0.3241 -0.9707 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K18 mock treatment 360.0 -1090.0 -0.39 360.0 -332.0 -0.26 -0.4529 -0.98 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K19 mock treatment 560.0 -886.0 -0.31 880.0 188.0 0.14 -0.1204 -0.3483 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K20 mock treatment 560.0 -886.0 -0.31 400.0 -292.0 -0.22 -0.381 -0.9864 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K21 mock treatment 680.0 -766.0 -0.27 200.0 -492.0 -0.38 -0.4595 -0.9869 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K22 mock treatment 720.0 -726.0 -0.26 360.0 -332.0 -0.26 -0.3626 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K23 mock treatment 680.0 -766.0 -0.27 2840.0 2150.0 1.65 0.9737 0.5827 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base K24 mock treatment 1120.0 -326.0 -0.12 1520.0 828.0 0.64 0.3675 0.569 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L01 mock treatment 640.0 -806.0 -0.29 600.0 -92.4 -0.07 -0.2524 -0.8566 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L02 mock treatment 680.0 -766.0 -0.27 320.0 -372.0 -0.29 -0.3943 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L03 mock treatment 280.0 -1170.0 -0.41 480.0 -212.0 -0.16 -0.4078 -0.9172 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L04 mock treatment 560.0 -886.0 -0.31 560.0 -132.0 -0.1 -0.2941 -0.8904 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L05 mock treatment 1240.0 -206.0 -0.07 1600.0 908.0 0.7 0.441 0.6295 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L06 mock treatment 640.0 -806.0 -0.29 440.0 -252.0 -0.19 -0.3392 -0.982 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L07 mock treatment 440.0 -1010.0 -0.36 360.0 -332.0 -0.26 -0.4328 -0.9865 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L08 mock treatment 7600.0 6150.0 2.18 320.0 -372.0 -0.29 1.3415 0.6093 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L09 mock treatment 520.0 -926.0 -0.33 360.0 -332.0 -0.26 -0.4127 -0.9922 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L10 mock treatment 600.0 -846.0 -0.3 320.0 -372.0 -0.29 -0.4144 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L11 mock treatment 4360.0 2910.0 1.03 600.0 -92.4 -0.07 0.6808 0.657 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L12 mock treatment 320.0 -1130.0 -0.4 1120.0 428.0 0.33 -0.0503 -0.0974 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L13 mock treatment 240.0 -1210.0 -0.43 320.0 -372.0 -0.29 -0.5047 -0.9808 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L14 mock treatment 400.0 -1050.0 -0.37 280.0 -412.0 -0.32 -0.4863 -0.9969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L15 mock treatment 440.0 -1010.0 -0.36 280.0 -412.0 -0.32 -0.4762 -0.9982 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L16 mock treatment 160.0 -1290.0 -0.46 400.0 -292.0 -0.22 -0.4813 -0.9467 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L17 mock treatment 400.0 -1050.0 -0.37 2160.0 1470.0 1.13 0.5343 0.4504 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L18 mock treatment 400.0 -1050.0 -0.37 440.0 -252.0 -0.19 -0.3994 -0.9541 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L19 mock treatment 440.0 -1010.0 -0.36 280.0 -412.0 -0.32 -0.4762 -0.9982 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L20 mock treatment 240.0 -1210.0 -0.43 1320.0 628.0 0.48 0.0382 0.0592 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L21 mock treatment 320.0 -1130.0 -0.4 360.0 -332.0 -0.26 -0.4629 -0.9766 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L22 mock treatment 680.0 -766.0 -0.27 1000.0 308.0 0.24 -0.0252 -0.0699 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L23 mock treatment 360.0 -1090.0 -0.39 440.0 -252.0 -0.19 -0.4095 -0.9494 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base L24 mock treatment 480.0 -966.0 -0.34 1160.0 468.0 0.36 0.0115 0.0232 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M01 mock treatment 2680.0 1230.0 0.44 6440.0 5750.0 4.41 3.4297 0.7735 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M02 mock treatment 600.0 -846.0 -0.3 320.0 -372.0 -0.29 -0.4144 -0.9997 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M03 mock treatment 1520.0 74.0 0.03 280.0 -412.0 -0.32 -0.2053 -0.6463 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M04 mock treatment 320.0 -1130.0 -0.4 680.0 -12.4 -0.01 -0.2892 -0.7238 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M05 mock treatment 640.0 -806.0 -0.29 800.0 108.0 0.08 -0.1438 -0.4831 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M06 mock treatment 3080.0 1630.0 0.58 240.0 -452.0 -0.35 0.1643 0.2431 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M07 mock treatment 400.0 -1050.0 -0.37 560.0 -132.0 -0.1 -0.3343 -0.8688 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M08 mock treatment 2360.0 914.0 0.32 4960.0 4270.0 3.28 2.546 0.7733 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M09 mock treatment 1920.0 474.0 0.17 1320.0 628.0 0.48 0.4596 0.9006 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M10 mock treatment 1440.0 -6.04 0.0 320.0 -372.0 -0.29 -0.2037 -0.7124 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M11 mock treatment 1080.0 -366.0 -0.13 1360.0 668.0 0.51 0.2706 0.5118 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M12 mock treatment 1920.0 474.0 0.17 1040.0 348.0 0.27 0.3076 0.9752 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M13 mock treatment 400.0 -1050.0 -0.37 720.0 27.6 0.02 -0.2474 -0.6657 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M14 mock treatment 1120.0 -326.0 -0.12 800.0 108.0 0.08 -0.0234 -0.1645 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M15 mock treatment 1280.0 -166.0 -0.06 2440.0 1750.0 1.34 0.907 0.6754 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M16 mock treatment 440.0 -1010.0 -0.36 360.0 -332.0 -0.26 -0.4328 -0.9865 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M17 mock treatment 3120.0 1670.0 0.59 1280.0 588.0 0.45 0.7389 0.9908 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M18 mock treatment 480.0 -966.0 -0.34 400.0 -292.0 -0.22 -0.4011 -0.979 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M19 mock treatment 4080.0 2630.0 0.93 1000.0 308.0 0.24 0.8277 0.8588 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M20 mock treatment 440.0 -1010.0 -0.36 1960.0 1270.0 0.97 0.4358 0.4204 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M21 mock treatment 3880.0 2430.0 0.86 240.0 -452.0 -0.35 0.3649 0.3921 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M22 mock treatment 280.0 -1170.0 -0.41 200.0 -492.0 -0.38 -0.5598 -0.999 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M23 mock treatment 320.0 -1130.0 -0.4 600.0 -92.4 -0.07 -0.3326 -0.8199 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base M24 mock treatment 1160.0 -286.0 -0.1 440.0 -252.0 -0.19 -0.2088 -0.9544 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N01 mock treatment 920.0 -526.0 -0.19 320.0 -372.0 -0.29 -0.3341 -0.9786 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N02 mock treatment 400.0 -1050.0 -0.37 400.0 -292.0 -0.22 -0.4211 -0.971 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N03 mock treatment 320.0 -1130.0 -0.4 640.0 -52.4 -0.04 -0.3109 -0.7744 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N04 mock treatment 920.0 -526.0 -0.19 1760.0 1070.0 0.82 0.4476 0.5325 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N05 mock treatment 320.0 -1130.0 -0.4 600.0 -92.4 -0.07 -0.3326 -0.8199 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N06 mock treatment 480.0 -966.0 -0.34 240.0 -452.0 -0.35 -0.4879 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N07 mock treatment 520.0 -926.0 -0.33 960.0 268.0 0.21 -0.087 -0.2246 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N08 mock treatment 400.0 -1050.0 -0.37 1160.0 468.0 0.36 -0.0086 -0.0166 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N09 mock treatment 840.0 -606.0 -0.21 880.0 188.0 0.14 -0.0502 -0.194 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N10 mock treatment 360.0 -1090.0 -0.39 2600.0 1910.0 1.46 0.7631 0.5039 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N11 mock treatment 1480.0 34.0 0.01 400.0 -292.0 -0.22 -0.1502 -0.6682 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N12 mock treatment 760.0 -686.0 -0.24 400.0 -292.0 -0.22 -0.3308 -0.9992 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N13 mock treatment 200.0 -1250.0 -0.44 840.0 148.0 0.11 -0.2324 -0.5094 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N14 mock treatment 320.0 -1130.0 -0.4 2480.0 1790.0 1.37 0.6879 0.4813 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N15 mock treatment 320.0 -1130.0 -0.4 320.0 -372.0 -0.29 -0.4846 -0.9866 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N16 mock treatment 1720.0 274.0 0.1 120.0 -572.0 -0.44 -0.242 -0.5377 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N17 mock treatment 400.0 -1050.0 -0.37 160.0 -532.0 -0.41 -0.5514 -0.9988 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N18 mock treatment 240.0 -1210.0 -0.43 280.0 -412.0 -0.32 -0.5264 -0.989 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N19 mock treatment 840.0 -606.0 -0.21 200.0 -492.0 -0.38 -0.4193 -0.9642 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N20 mock treatment 600.0 -846.0 -0.3 240.0 -452.0 -0.35 -0.4578 -0.9974 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N21 mock treatment 720.0 -726.0 -0.26 280.0 -412.0 -0.32 -0.406 -0.9948 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N22 mock treatment 360.0 -1090.0 -0.39 1040.0 348.0 0.27 -0.0837 -0.1787 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N23 mock treatment 3120.0 1670.0 0.59 440.0 -252.0 -0.19 0.2829 0.4529 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base N24 mock treatment 480.0 -966.0 -0.34 360.0 -332.0 -0.26 -0.4228 -0.9895 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O01 mock treatment 240.0 -1210.0 -0.43 240.0 -452.0 -0.35 -0.5481 -0.9946 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O02 mock treatment 5800.0 4350.0 1.54 360.0 -332.0 -0.26 0.9117 0.5824 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O03 mock treatment 5480.0 4030.0 1.43 360.0 -332.0 -0.26 0.8314 0.572 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O04 mock treatment 1080.0 -366.0 -0.13 440.0 -252.0 -0.19 -0.2288 -0.981 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O05 mock treatment 3960.0 2510.0 0.89 400.0 -292.0 -0.22 0.4719 0.5131 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O06 mock treatment 5520.0 4070.0 1.45 240.0 -452.0 -0.35 0.7763 0.5223 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O07 mock treatment 720.0 -726.0 -0.26 640.0 -52.4 -0.04 -0.2106 -0.8078 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O08 mock treatment 4520.0 3070.0 1.09 280.0 -412.0 -0.32 0.5472 0.4819 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O09 mock treatment 2360.0 914.0 0.32 280.0 -412.0 -0.32 0.0054 0.0119 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O10 mock treatment 1000.0 -446.0 -0.16 160.0 -532.0 -0.41 -0.4009 -0.9147 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O11 mock treatment 360.0 -1090.0 -0.39 240.0 -452.0 -0.35 -0.518 -0.9987 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O12 mock treatment 2320.0 874.0 0.31 320.0 -372.0 -0.29 0.0171 0.0404 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O13 mock treatment 2160.0 714.0 0.25 240.0 -452.0 -0.35 -0.0665 -0.1547 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O14 mock treatment 2120.0 674.0 0.24 360.0 -332.0 -0.26 -0.0114 -0.0326 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O15 mock treatment 2360.0 914.0 0.32 280.0 -412.0 -0.32 0.0054 0.0119 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O16 mock treatment 2520.0 1070.0 0.38 240.0 -452.0 -0.35 0.0238 0.0462 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O17 mock treatment 2000.0 554.0 0.2 200.0 -492.0 -0.38 -0.1284 -0.3013 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O18 mock treatment 2280.0 834.0 0.3 240.0 -452.0 -0.35 -0.0364 -0.0798 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O19 mock treatment 1920.0 474.0 0.17 360.0 -332.0 -0.26 -0.0616 -0.2015 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O20 mock treatment 2200.0 754.0 0.27 280.0 -412.0 -0.32 -0.0348 -0.0839 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O21 mock treatment 2080.0 634.0 0.22 240.0 -452.0 -0.35 -0.0866 -0.2092 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O22 mock treatment 520.0 -926.0 -0.33 280.0 -412.0 -0.32 -0.4562 -0.9998 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O23 mock treatment 2160.0 714.0 0.25 200.0 -492.0 -0.38 -0.0882 -0.1939 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base O24 mock treatment 1840.0 394.0 0.14 160.0 -532.0 -0.41 -0.1902 -0.4403 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P01 mock treatment 1080.0 -366.0 -0.13 960.0 268.0 0.21 0.0534 0.2199 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P02 mock treatment 6440.0 4990.0 1.77 200.0 -492.0 -0.38 0.9854 0.544 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P03 mock treatment 6240.0 4790.0 1.7 1160.0 468.0 0.36 1.4564 0.8379 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P04 mock treatment 520.0 -926.0 -0.33 3920.0 3230.0 2.48 1.5198 0.608 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P05 mock treatment 6480.0 5030.0 1.79 240.0 -452.0 -0.35 1.0171 0.5591 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P06 mock treatment 2520.0 1070.0 0.38 200.0 -492.0 -0.38 0.0021 0.0039 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P07 mock treatment 1760.0 314.0 0.11 360.0 -332.0 -0.26 -0.1017 -0.3652 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P08 mock treatment 1240.0 -206.0 -0.07 240.0 -452.0 -0.35 -0.2973 -0.8376 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P09 mock treatment 3240.0 1790.0 0.64 160.0 -532.0 -0.41 0.161 0.2128 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P10 mock treatment 720.0 -726.0 -0.26 240.0 -452.0 -0.35 -0.4277 -0.9892 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P11 mock treatment 320.0 -1130.0 -0.4 240.0 -452.0 -0.35 -0.5281 -0.9976 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P12 mock treatment 360.0 -1090.0 -0.39 200.0 -492.0 -0.38 -0.5397 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P13 mock treatment 2320.0 874.0 0.31 280.0 -412.0 -0.32 -0.0047 -0.0105 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P14 mock treatment 2160.0 714.0 0.25 320.0 -372.0 -0.29 -0.0231 -0.0604 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P15 mock treatment 1960.0 514.0 0.18 240.0 -452.0 -0.35 -0.1167 -0.2974 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P16 mock treatment 1920.0 474.0 0.17 240.0 -452.0 -0.35 -0.1267 -0.3284 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P17 mock treatment 2320.0 874.0 0.31 240.0 -452.0 -0.35 -0.0264 -0.0566 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P18 mock treatment 2800.0 1350.0 0.48 200.0 -492.0 -0.38 0.0723 0.1183 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P19 mock treatment 360.0 -1090.0 -0.39 280.0 -412.0 -0.32 -0.4963 -0.9953 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P20 mock treatment 1840.0 394.0 0.14 240.0 -452.0 -0.35 -0.1468 -0.392 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P21 mock treatment 280.0 -1170.0 -0.41 160.0 -532.0 -0.41 -0.5815 -1.0 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P22 mock treatment 2040.0 594.0 0.21 280.0 -412.0 -0.32 -0.0749 -0.1969 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P23 mock treatment 2000.0 554.0 0.2 200.0 -492.0 -0.38 -0.1284 -0.3013 1096.0004 KinaseGlo(1096.0004) GALKActivityAssay 1096.0004.Base P24 mock treatment 520.0 -926.0 -0.33 280.0 -412.0 -0.32 -0.4562 -0.9998