ASSAY_ID ASSAY PROJECT PLATE WELL WELL_TYPE RAW_VALUE_A BSUB_VALUE_A Z_SCORE_A RAW_VALUE_B BSUB_VALUE_B Z_SCORE_B COMPOSITE_Z REPRODUCIBILITY CHEMBANK_ID VIRTUAL_ID SMILES 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A01 compound treatment 1311880.0 36200.0 0.61 1278000.0 84300.0 1.52 1.5013 0.9187 1965040 CMLD1_000001 CCCC=C(CCC)[C@@H](NC(=O)c1ccccc1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A02 compound treatment 1295800.0 20100.0 0.34 1268880.0 75100.0 1.35 1.1949 0.8567 1965041 CMLD1_000002 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(O)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A03 compound treatment 1130440.0 -145000.0 -2.43 1145080.0 -48700.0 -0.88 -2.3391 -0.9051 1965042 CMLD1_000003 CCCC=C(CCC)[C@@H](NC(=O)c1cccs1)c2ccc(cc2)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A04 compound treatment 849760.0 -426000.0 -7.13 952000.0 -242000.0 -4.36 -8.1202 -0.9721 1965043 CMLD1_000004 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@H]3[C@H](CC(=O)C(=O)N4CCCC4)C(=O)C=C3CN1C(=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A05 compound treatment 1301520.0 25800.0 0.43 1263720.0 70000.0 1.26 1.1968 0.8981 1965044 CMLD1_000005 CCCC=C(CCC)[C@@H](NC(=O)c1ccc(cc1)C(F)(F)F)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A06 compound treatment 1325800.0 50100.0 0.84 1275680.0 81900.0 1.48 1.6365 0.964 1965045 CMLD1_000006 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7c[nH]c8ccc(OC)cc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A07 compound treatment 1341920.0 66200.0 1.11 1263280.0 69500.0 1.25 1.6693 0.9981 1965046 CMLD1_000007 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1ccc(cc1)c2ccccc2)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A08 compound treatment 1293520.0 17800.0 0.3 1261400.0 67700.0 1.22 1.0726 0.8548 1965047 CMLD1_000008 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(F)c(F)c(F)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A09 compound treatment 1337880.0 62200.0 1.04 1255200.0 61500.0 1.11 1.5185 0.9995 1965048 CMLD1_000009 CCCCC=C[C@@H](NC(=O)Oc1cccc(c1)C(F)(F)F)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A10 compound treatment 1260680.0 -15000.0 -0.25 1220120.0 26400.0 0.48 0.1581 0.294 1965049 CMLD1_000010 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6c[nH]c7ccc(OC)cc67 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A11 compound treatment 1342920.0 67200.0 1.12 1244080.0 50300.0 0.91 1.4365 0.9943 1965050 CMLD1_000011 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NC(=O)c3cccs3)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A12 compound treatment 1261800.0 -13900.0 -0.23 1240320.0 46600.0 0.84 0.4287 0.4923 1965051 CMLD1_000012 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)o6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A13 compound treatment 1290840.0 15100.0 0.25 1253200.0 59500.0 1.07 0.9364 0.8508 1965052 CMLD1_000013 CCCC=C(CCC)[C@@H](NC(=O)OCC(C)C)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A14 compound treatment 1225040.0 -50700.0 -0.85 1201680.0 7930.0 0.14 -0.4986 -0.5797 1965053 CMLD1_000014 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccc(OC)c(Br)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A15 compound treatment 1317120.0 41400.0 0.69 1234880.0 41100.0 0.74 1.014 0.9994 1965054 CMLD1_000015 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccco2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A16 compound treatment 1288560.0 12800.0 0.21 1231160.0 37400.0 0.67 0.6286 0.8885 1965055 CMLD1_000016 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cccc7ccccc67 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A17 compound treatment 1039160.0 -237000.0 -3.96 1152560.0 -41200.0 -0.74 -3.3239 -0.8253 1965056 CMLD1_000017 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)C(C)(C)C)c2ccc(cc2)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A18 compound treatment 1183120.0 -92600.0 -1.55 1179760.0 -14000.0 -0.25 -1.2739 -0.8114 1965057 CMLD1_000018 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)c(F)c6F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A19 compound treatment 1262680.0 -13000.0 -0.22 1220880.0 27100.0 0.49 0.1914 0.3576 1965058 CMLD1_000019 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccs2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A20 compound treatment 1337680.0 62000.0 1.04 1232240.0 38500.0 0.69 1.2237 0.9809 1965059 CMLD1_000020 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(OC)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A21 compound treatment 1299640.0 23900.0 0.4 1202360.0 8610.0 0.16 0.3928 0.9149 1965060 CMLD1_000021 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NC(=O)Cc3ccccc3)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A22 mock treatment 1286440.0 10700.0 0.18 1210440.0 16700.0 0.3 0.3396 0.9695 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A23 mock treatment 1246440.0 -29300.0 -0.49 1198680.0 4930.0 0.09 -0.2836 -0.5695 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 A24 mock treatment 1258640.0 -17100.0 -0.29 1205160.0 11400.0 0.21 -0.0566 -0.1609 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B01 compound treatment 1285000.0 9280.0 0.16 1269800.0 76100.0 1.37 1.0788 0.7823 1965061 CMLD1_000022 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(O)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B02 compound treatment 1371920.0 96200.0 1.61 1301160.0 107000.0 1.94 2.5069 0.9958 1965062 CMLD1_000023 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCN7CNCC7=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B03 compound treatment 1383760.0 108000.0 1.81 1296080.0 102000.0 1.84 2.5822 1.0 1965063 CMLD1_000024 COCCn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccccc5)C(=O)OC)Cc21)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B04 compound treatment 1383880.0 108000.0 1.81 1288640.0 94900.0 1.71 2.4889 0.9996 1965064 CMLD1_000025 CCOC(=O)N(CC[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)C4(CC(=C)c5ccccc5)CC4)S(=O)(=O)c6ccc(C)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B05 compound treatment 1353560.0 77800.0 1.3 1272840.0 79100.0 1.43 1.9288 0.999 1965065 CMLD1_000026 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccccn7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B06 compound treatment 1385920.0 110000.0 1.84 1300640.0 107000.0 1.93 2.6659 0.9998 1965066 CMLD1_000027 CC(NP(=O)(c1ccccc1)c2ccccc2)C3(CC(=C)c4ccccc4)CC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B07 compound treatment 1389120.0 113000.0 1.9 1257440.0 63700.0 1.15 2.1534 0.971 1965067 CMLD1_000028 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccccn7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B08 compound treatment 1391520.0 116000.0 1.94 1270000.0 76300.0 1.37 2.3418 0.9858 1965068 CMLD1_000029 COC(=O)C1(C)NCC2=C(C)C(=O)C(C)C2=C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B09 compound treatment 1335360.0 59600.0 1.0 1255280.0 61500.0 1.11 1.4897 0.9986 1965069 CMLD1_000030 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCF 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B10 compound treatment 1323040.0 47300.0 0.79 1249800.0 56100.0 1.01 1.2741 0.9928 1965070 CMLD1_000031 COC(=O)C1(Cc2ccccc2)NCC3=C(C(C)C)C(=O)C(C)C3=C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B11 compound treatment 1346280.0 70600.0 1.18 1253560.0 59800.0 1.08 1.597 0.999 1965071 CMLD1_000032 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(cc6)S(=O)(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B12 compound treatment 1221920.0 -53800.0 -0.9 1200680.0 6930.0 0.12 -0.5482 -0.6032 1965072 CMLD1_000033 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1CCc5ccc(Cl)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B13 compound treatment 1335680.0 60000.0 1.0 1249160.0 55400.0 1.0 1.4155 1.0 1965073 CMLD1_000034 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CC7CC7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B14 compound treatment 1343360.0 67600.0 1.13 1250440.0 56700.0 1.02 1.5227 0.9987 1965074 CMLD1_000035 COc1ccc(COC2OC[C@]3(C)[C@@H]4[C@H]2CCC5C(CO)C(CO)[C@@H](C)C(=C54)CN3C(=O)OC(C)(C)C)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B15 compound treatment 1310280.0 34600.0 0.58 1241280.0 47500.0 0.86 1.0146 0.9817 1965075 CMLD1_000036 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(C)n(C)n6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B16 compound treatment 1292680.0 17000.0 0.28 1249200.0 55500.0 1.0 0.9072 0.8734 1965076 CMLD1_000037 CC1(C)C(=O)C(=C2CN3C(=O)N(CCc4ccccc4)C(=O)C3(Cc5ccc(F)cc5)C=C21)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B17 compound treatment 1315800.0 40100.0 0.67 1235440.0 41700.0 0.75 1.0055 0.9984 1965077 CMLD1_000038 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B18 compound treatment 1318560.0 42800.0 0.72 1240040.0 46300.0 0.83 1.0968 0.9972 1965078 CMLD1_000039 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccccn7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B19 compound treatment 1317320.0 41600.0 0.7 1207280.0 13500.0 0.24 0.6647 0.9011 1965079 CMLD1_000040 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5C[C@H](O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B20 compound treatment 1306680.0 31000.0 0.52 1211520.0 17800.0 0.32 0.5928 0.9733 1965080 CMLD1_000041 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6c(O)c(C)cnc6CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B21 compound treatment 1268920.0 -6800.0 -0.11 1190680.0 -3070.0 -0.06 -0.1195 -0.945 1965081 CMLD1_000042 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCN7CNCC7=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B22 mock treatment 1295000.0 19300.0 0.32 1219240.0 25500.0 0.46 0.553 0.9851 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B23 mock treatment 1274880.0 -836.0 -0.01 1182240.0 -11500.0 -0.21 -0.1565 -0.7531 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 B24 mock treatment 1291600.0 15900.0 0.27 1208160.0 14400.0 0.26 0.3716 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C01 compound treatment 1358920.0 83200.0 1.39 1285480.0 91700.0 1.65 2.1533 0.9964 1965082 CMLD1_000043 CCCC=C(CCC)[C@@H](NS(=O)(=O)CC1(CCC2CC1=O)C2(C)C)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C02 compound treatment 255320.0 -1020000.0 -17.08 383320.0 -810000.0 -14.6 -22.3993 -0.997 1965083 CMLD1_000044 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(C)o7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C03 compound treatment 1304840.0 29100.0 0.49 1269360.0 75600.0 1.36 1.308 0.904 1965084 CMLD1_000045 CCCC=C(CCC)[C@@H](NC(=O)CCc1ccccc1)c2ccc(cc2)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C04 compound treatment 1347000.0 71300.0 1.19 1270560.0 76800.0 1.38 1.8221 0.9973 1965085 CMLD1_000046 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C05 compound treatment 1344680.0 69000.0 1.15 1270920.0 77200.0 1.39 1.7993 0.9957 1965086 CMLD1_000047 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1ccc(Cl)cc1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C06 compound treatment 1363120.0 87400.0 1.46 1279080.0 85300.0 1.54 2.1214 0.9997 1965087 CMLD1_000048 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@H]3[C@H](CC(=O)C(=O)N(C)C)C(=O)C=C3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C07 compound treatment 1309000.0 33300.0 0.56 1247640.0 53900.0 0.97 1.0805 0.9652 1965088 CMLD1_000049 CCCCC=C[C@@H](NC(=O)CCc1ccccc1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C08 compound treatment 1327960.0 52200.0 0.87 1262280.0 68500.0 1.23 1.4913 0.9857 1965089 CMLD1_000050 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6c(C)onc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C09 compound treatment 1301720.0 26000.0 0.44 1248960.0 55200.0 0.99 1.0111 0.9312 1965090 CMLD1_000051 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)c2ccc(cc2)c3ccccc3)c4cccc(Cl)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C10 compound treatment 1308160.0 32400.0 0.54 1256320.0 62600.0 1.13 1.1811 0.9439 1965091 CMLD1_000052 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccsc6Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C11 compound treatment 1320280.0 44600.0 0.75 1255840.0 62100.0 1.12 1.3184 0.9806 1965092 CMLD1_000053 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NC(=O)c3ccccc3)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C12 compound treatment 1268760.0 -6960.0 -0.12 1242840.0 49100.0 0.88 0.5432 0.6088 1965093 CMLD1_000054 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5C[C@H](O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C13 compound treatment 1327200.0 51500.0 0.86 1221640.0 27900.0 0.5 0.9646 0.9671 1965094 CMLD1_000055 CCCCC=C[C@@H](NC(=O)c1ccccc1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C14 compound treatment 1263320.0 -12400.0 -0.21 1207000.0 13300.0 0.24 0.0222 0.0701 1965095 CMLD1_000056 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cc(F)cc8COCOc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C15 compound treatment 1296720.0 21000.0 0.35 1235400.0 41700.0 0.75 0.7792 0.9403 1965096 CMLD1_000057 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccc(cc2)c3ccccc3)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C16 compound treatment 1304520.0 28800.0 0.48 1241040.0 47300.0 0.85 0.9434 0.9636 1965097 CMLD1_000058 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cccc8ccccc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C17 compound treatment 1315600.0 39900.0 0.67 1258160.0 64400.0 1.16 1.2926 0.9655 1965098 CMLD1_000059 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NS(=O)(=O)c3cccc4cccnc34)c5ccc(cc5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C18 compound treatment 1268120.0 -7600.0 -0.13 1244080.0 50300.0 0.91 0.5514 0.6021 1965099 CMLD1_000060 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccc(O)c(OC)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C19 compound treatment 1300160.0 24400.0 0.41 1213600.0 19900.0 0.36 0.5422 0.9978 1965100 CMLD1_000061 CC(C)(C)C(=O)N[C@@H](c1ccc(Cl)cc1)[C@]2(C)C[C@H]2C3CCCCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C20 compound treatment 1310680.0 35000.0 0.59 1208120.0 14400.0 0.26 0.5969 0.9328 1965101 CMLD1_000062 CCCCC=C[C@@H](NC(=O)OCC#C)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C21 compound treatment 1294040.0 18300.0 0.31 1208560.0 14800.0 0.27 0.4056 0.9976 1965060 CMLD1_000063 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NC(=O)Cc3ccccc3)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C22 mock treatment 1283560.0 7840.0 0.13 1199680.0 5930.0 0.11 0.1684 0.9948 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C23 mock treatment 1276800.0 1080.0 0.02 1199200.0 5450.0 0.1 0.0823 0.8237 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 C24 mock treatment 1291160.0 15400.0 0.26 1213360.0 19600.0 0.35 0.4326 0.9882 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D01 compound treatment 1398920.0 123000.0 2.06 1295680.0 102000.0 1.84 2.7565 0.9983 1965102 CMLD1_000064 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccccn6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D02 compound treatment 1431720.0 156000.0 2.61 1315560.0 122000.0 2.19 3.3979 0.9963 1965103 CMLD1_000065 COCCn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(F)cc5)C(=O)OC)Cc21)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D03 compound treatment 1368600.0 92900.0 1.55 1276760.0 83000.0 1.5 2.1567 0.9998 1965104 CMLD1_000066 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(OC)c(OC)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D04 compound treatment 1403920.0 128000.0 2.15 1295640.0 102000.0 1.84 2.8152 0.997 1965105 CMLD1_000067 CCCC[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)C4(CC(=C)c5ccccc5)CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D05 compound treatment 1324160.0 48400.0 0.81 1266600.0 72900.0 1.31 1.5014 0.9732 1965106 CMLD1_000068 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7nc8ccccc8[nH]7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D06 compound treatment 1387320.0 112000.0 1.87 1285800.0 92100.0 1.66 2.4934 0.9982 1965107 CMLD1_000069 CC(=O)N1CC2(CC2)CC1c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D07 compound treatment 843760.0 -432000.0 -7.23 1011720.0 -182000.0 -3.28 -7.4304 -0.9361 1965108 CMLD1_000070 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccc(O)c(O)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D08 compound treatment 1353480.0 77800.0 1.3 1269640.0 75900.0 1.37 1.8871 0.9997 1965109 CMLD1_000071 COC(=O)C1(C)NCC2=C(C(=O)C(C)C2=C1)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D09 compound treatment 1323800.0 48100.0 0.8 1245040.0 51300.0 0.92 1.2225 0.9976 1965110 CMLD1_000072 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCn7cc(nc7C)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D10 compound treatment 1354680.0 79000.0 1.32 1276200.0 82500.0 1.49 1.9849 0.9983 1965111 CMLD1_000073 COC(=O)C1(Cc2ccccc2)NCC3=C(C(=O)C(C)C3=C1)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D11 compound treatment 1350160.0 74400.0 1.25 1249840.0 56100.0 1.01 1.5956 0.9946 1965112 CMLD1_000074 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccccn6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D12 compound treatment 851200.0 -425000.0 -7.1 991440.0 -202000.0 -3.64 -7.6007 -0.9519 1965113 CMLD1_000075 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1Cc5ccco5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D13 compound treatment 1309080.0 33400.0 0.56 1223400.0 29700.0 0.53 0.7726 0.9998 1965057 CMLD1_000076 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)c(F)c6F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D14 compound treatment 1273200.0 -2520.0 -0.04 1243800.0 50100.0 0.9 0.6079 0.6734 1965114 CMLD1_000077 C[C@@H]1C(CO)C(CO)C2CC[C@H]3C(OCc4ccc(F)cc4C(F)(F)F)OC[C@]5(C)[C@H]3C2=C1CN5C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D15 compound treatment 1308560.0 32800.0 0.55 1232880.0 39100.0 0.71 0.8872 0.9924 1965115 CMLD1_000078 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(C)n(C)n6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D16 compound treatment 1303920.0 28200.0 0.47 1244480.0 50700.0 0.91 0.9801 0.9527 1965116 CMLD1_000079 CC(=C1[C@H]2C(=C(C1=O)c3ccccc3)CN4C(=O)N(CCc5ccccc5)C(=O)[C@]24Cc6ccc(F)cc6)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D17 compound treatment 1271640.0 -4080.0 -0.07 1205600.0 11900.0 0.21 0.1028 0.4585 1965117 CMLD1_000080 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCSCCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D18 compound treatment 1316400.0 40700.0 0.68 1248880.0 55100.0 0.99 1.1838 0.983 1965118 CMLD1_000081 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(cc7)S(=O)(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D19 compound treatment 1314520.0 38800.0 0.65 1205480.0 11700.0 0.21 0.6087 0.8913 1965119 CMLD1_000082 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cc(C)n(C)n7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D20 compound treatment 1281680.0 5960.0 0.1 1209520.0 15800.0 0.28 0.2715 0.9014 1965120 CMLD1_000083 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(C)n(C)n6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D21 compound treatment 1283840.0 8120.0 0.14 1196000.0 2250.0 0.04 0.1249 0.8799 1965121 CMLD1_000084 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCF 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D22 mock treatment 1280200.0 4480.0 0.08 1207320.0 13600.0 0.24 0.226 0.8834 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D23 mock treatment 1282760.0 7040.0 0.12 1195800.0 2050.0 0.04 0.1095 0.8865 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 D24 mock treatment 1280480.0 4760.0 0.08 1205680.0 11900.0 0.22 0.2084 0.9088 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E01 compound treatment 1374520.0 98800.0 1.65 1296720.0 103000.0 1.86 2.4811 0.9983 1965122 CMLD1_000085 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1cccc2cccnc12)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E02 compound treatment 1367400.0 91700.0 1.53 1284680.0 90900.0 1.64 2.2434 0.9995 1965123 CMLD1_000086 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)c(F)c6F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E03 compound treatment 1379760.0 104000.0 1.74 1276480.0 82700.0 1.49 2.2852 0.997 1965124 CMLD1_000087 CCCC=C(CCC)[C@@H](NC(=O)c1ccc(cc1)C(F)(F)F)c2ccc(cc2)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E04 compound treatment 1348040.0 72300.0 1.21 1294520.0 101000.0 1.82 2.1397 0.9806 1965125 CMLD1_000088 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E05 compound treatment 1390480.0 115000.0 1.92 1300560.0 107000.0 1.92 2.7188 1.0 1965126 CMLD1_000089 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1ccc(cc1)C(F)(F)F)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E06 compound treatment 1336800.0 61100.0 1.02 1271880.0 78100.0 1.41 1.7183 0.9876 1965127 CMLD1_000090 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(OC)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E07 compound treatment 1349080.0 73400.0 1.23 1263920.0 70200.0 1.26 1.7622 0.9999 1965128 CMLD1_000091 CCCCC=C[C@@H](NC(=O)C(C)(C)C)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E08 compound treatment 1340640.0 64900.0 1.09 1241080.0 47300.0 0.85 1.3713 0.9928 1965129 CMLD1_000092 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCCNc7ncc(cc7Cl)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E09 compound treatment 1318600.0 42900.0 0.72 1256120.0 62400.0 1.12 1.3021 0.9765 1965130 CMLD1_000093 CCCC=C(CCC)[C@@H](NC(=O)c1ccc(cc1)C(=O)OC)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E10 compound treatment 1306440.0 30700.0 0.51 1243880.0 50100.0 0.9 1.0023 0.9643 1965131 CMLD1_000094 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(OC(F)(F)F)cc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E11 compound treatment 1370520.0 94800.0 1.59 1256040.0 62300.0 1.12 1.9155 0.9856 1965060 CMLD1_000095 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NC(=O)Cc3ccccc3)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E12 compound treatment 1326200.0 50500.0 0.84 1263640.0 69900.0 1.26 1.4878 0.9811 1965132 CMLD1_000096 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccccn6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E13 compound treatment 1292360.0 16600.0 0.28 1216600.0 22900.0 0.41 0.4881 0.9819 1965133 CMLD1_000097 CCCCC=C[C@@H](NC(=O)OCc1ccccc1Cl)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E14 compound treatment 1331480.0 55800.0 0.93 1271880.0 78100.0 1.41 1.6553 0.9801 1965134 CMLD1_000098 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E15 compound treatment 1333080.0 57400.0 0.96 1234960.0 41200.0 0.74 1.2039 0.9919 1965135 CMLD1_000099 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccs2)c3ccc(cc3)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E16 compound treatment 1434400.0 159000.0 2.66 1418320.0 225000.0 4.05 4.7388 0.9791 1965136 CMLD1_000100 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cccc7ccccc67 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E17 compound treatment 1300320.0 24600.0 0.41 1227560.0 33800.0 0.61 0.7219 0.9818 1965137 CMLD1_000101 CC(=CC1CCCCC1)[C@@H](NC(=O)c2cccnc2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E18 compound treatment 1314720.0 39000.0 0.65 1225000.0 31300.0 0.56 0.8597 0.9973 1965138 CMLD1_000102 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(OC(F)(F)F)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E19 compound treatment 1306680.0 31000.0 0.52 1190200.0 -3550.0 -0.06 0.3212 0.6153 1965139 CMLD1_000103 C[C@]1(C[C@H]1C2CCCCC2)[C@@H](NC(=O)c3ccc(cc3)c4ccccc4)c5ccc(Cl)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E20 compound treatment 1328560.0 52800.0 0.88 1227200.0 33500.0 0.6 1.0515 0.9825 1965140 CMLD1_000104 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccsc6Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E21 compound treatment 1320960.0 45200.0 0.76 1217720.0 24000.0 0.43 0.8408 0.9646 1965141 CMLD1_000105 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)c2ccccc2)c3cccc(Cl)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E22 mock treatment 1298040.0 22300.0 0.37 1216240.0 22500.0 0.41 0.5507 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E23 mock treatment 1289920.0 14200.0 0.24 1205360.0 11600.0 0.21 0.316 0.998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 E24 mock treatment 1308680.0 33000.0 0.55 1224520.0 30800.0 0.55 0.7821 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F01 compound treatment 1398360.0 123000.0 2.05 1287040.0 93300.0 1.68 2.6398 0.9951 1965142 CMLD1_000106 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCN6CCOCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F02 compound treatment 1398280.0 123000.0 2.05 1294800.0 101000.0 1.82 2.7378 0.9982 1965143 CMLD1_000107 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cc(F)cc8COCOc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F03 compound treatment 1395680.0 120000.0 2.01 1298120.0 104000.0 1.88 2.7493 0.9995 1965144 CMLD1_000108 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(OC)c(OC)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F04 compound treatment 1393800.0 118000.0 1.98 1287120.0 93400.0 1.68 2.5869 0.9968 1965145 CMLD1_000109 CCCC[C@H]1C[C@@H]1[C@H](NP(=O)(c2ccccc2)c3ccccc3)C4(CC(=C)c5cccc(OC)c5)CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F05 compound treatment 1365520.0 89800.0 1.5 1260200.0 66500.0 1.2 1.9093 0.9937 1965146 CMLD1_000110 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccccn7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F06 compound treatment 1388440.0 113000.0 1.89 1279240.0 85500.0 1.54 2.4231 0.9949 1965147 CMLD1_000111 CC1N(CC(O)(CC21CC2)c3ccccc3)P(=O)(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F07 compound treatment 1381840.0 106000.0 1.78 1277080.0 83300.0 1.5 2.3175 0.9965 1965148 CMLD1_000112 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(nc6)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F08 compound treatment 1383520.0 108000.0 1.8 1275000.0 81300.0 1.46 2.3108 0.9946 1965149 CMLD1_000113 CCCCCC1=C2CNC(C)(C=C2C(C)C1=O)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F09 compound treatment 1371680.0 96000.0 1.61 1262720.0 69000.0 1.24 2.0143 0.992 1965150 CMLD1_000114 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7c(O)c(C)cnc7CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F10 compound treatment 1279440.0 3720.0 0.06 1223480.0 29700.0 0.54 0.4229 0.7841 1965151 CMLD1_000115 CCCCCC1=C2CNC(Cc3ccccc3)(C=C2C(C)C1=O)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F11 compound treatment 1348200.0 72500.0 1.21 1248880.0 55100.0 0.99 1.5601 0.9951 1965152 CMLD1_000116 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccccn6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F12 compound treatment 1278360.0 2640.0 0.04 1196160.0 2410.0 0.04 0.062 1.0 1965153 CMLD1_000117 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F13 compound treatment 1303040.0 27300.0 0.46 1287880.0 94100.0 1.7 1.5226 0.8668 1965154 CMLD1_000118 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(Cl)c(c6)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F14 compound treatment 1352040.0 76300.0 1.28 1250000.0 56300.0 1.01 1.6198 0.9934 1965155 CMLD1_000119 C[C@@H]1C(COC(=O)C)C(COC(=O)C)C2CC[C@H]3C(OCc4ccc(F)cc4C(F)(F)F)OC[C@]5(C)[C@H]3C2=C1CN5C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F15 compound treatment 1300080.0 24400.0 0.41 1252720.0 59000.0 1.06 1.0396 0.9135 1965156 CMLD1_000120 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(O)c(OC)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F16 compound treatment 1318320.0 42600.0 0.71 1251200.0 57500.0 1.04 1.2361 0.9834 1965157 CMLD1_000121 CC1(C)C(=O)C(=C2CN3C(=O)N(CCc4ccccc4)C(=O)C3(Cc5ccc(cc5)C(F)(F)F)C=C21)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F17 compound treatment 1275480.0 -236.0 0.0 1244480.0 50700.0 0.91 0.6436 0.704 1965158 CMLD1_000122 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCSCCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F18 compound treatment 1327440.0 51700.0 0.87 1225320.0 31600.0 0.57 1.0143 0.9793 1965150 CMLD1_000123 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7c(O)c(C)cnc7CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F19 compound treatment 1314720.0 39000.0 0.65 1196760.0 3010.0 0.05 0.4999 0.7633 1965159 CMLD1_000124 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCSCCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F20 compound treatment 1321440.0 45700.0 0.77 1221720.0 28000.0 0.5 0.8975 0.9795 1965160 CMLD1_000125 COC(=O)Cn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(F)cc5)C(=O)OC)Cc21)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F21 compound treatment 855240.0 -420000.0 -7.04 994760.0 -199000.0 -3.59 -7.5106 -0.9511 1965161 CMLD1_000126 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccc(O)c(O)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F22 mock treatment 1294040.0 18300.0 0.31 1200240.0 6490.0 0.12 0.2996 0.9127 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F23 mock treatment 1278160.0 2440.0 0.04 1190000.0 -3750.0 -0.07 -0.0188 -0.2382 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 F24 mock treatment 1310600.0 34900.0 0.58 1210200.0 16500.0 0.3 0.6224 0.9506 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G01 compound treatment 1400280.0 125000.0 2.08 1300880.0 107000.0 1.93 2.8389 0.9993 1965162 CMLD1_000127 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1ccc(Cl)cc1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G02 compound treatment 1386400.0 111000.0 1.85 1290160.0 96400.0 1.74 2.5381 0.9995 1965163 CMLD1_000128 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCCNc7ncc(cc7Cl)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G03 compound treatment 1374600.0 98900.0 1.65 1265520.0 71800.0 1.29 2.0845 0.9926 1965164 CMLD1_000129 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1ccccc1)c2ccc(cc2)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G04 compound treatment 1398120.0 122000.0 2.05 1332840.0 139000.0 2.51 3.2205 0.995 1965165 CMLD1_000130 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@H]3C(=C)C(=O)C=C3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G05 compound treatment 1359960.0 84200.0 1.41 1280360.0 86600.0 1.56 2.1003 0.9987 1965166 CMLD1_000131 CCCC=C(CCC)[C@@H](NS(=O)(=O)CC)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G06 compound treatment 1360560.0 84800.0 1.42 1286520.0 92800.0 1.67 2.1859 0.9967 1965167 CMLD1_000132 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@H]3[C@H](CC(=O)C(=O)N4CCCC4)C(=O)C[C@H]3CN1C(=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G07 compound treatment 1363400.0 87700.0 1.47 1270080.0 76300.0 1.38 2.0101 0.9995 1965168 CMLD1_000133 CCCCC=C[C@@H](NC(=O)c1ccc(cc1)c2ccccc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G08 compound treatment 1349160.0 73400.0 1.23 1286040.0 92300.0 1.66 2.0449 0.9889 1965169 CMLD1_000134 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7c[nH]c8ccccc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G09 compound treatment 1350880.0 75200.0 1.26 1265400.0 71700.0 1.29 1.8023 0.9999 1965170 CMLD1_000135 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccco2)c3ccccc3C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G10 compound treatment 1347160.0 71400.0 1.2 1280480.0 86700.0 1.56 1.9504 0.9913 1965171 CMLD1_000136 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cc(F)c(F)c(F)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G11 compound treatment 1288240.0 12500.0 0.21 1254560.0 60800.0 1.1 0.923 0.8274 1965172 CMLD1_000137 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G12 compound treatment 1300400.0 24700.0 0.41 1252280.0 58500.0 1.05 1.0378 0.9163 1965173 CMLD1_000138 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(Cl)c(c6)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G13 compound treatment 1370520.0 94800.0 1.59 1257720.0 64000.0 1.15 1.9369 0.9877 1965174 CMLD1_000139 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccco2)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G14 compound treatment 1333120.0 57400.0 0.96 1256560.0 62800.0 1.13 1.4795 0.9967 1965175 CMLD1_000140 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6c(O)c(C)cnc6CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G15 compound treatment 1214400.0 -61300.0 -1.03 1216320.0 22600.0 0.41 -0.438 -0.3968 1965176 CMLD1_000141 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G16 compound treatment 907320.0 -368000.0 -6.16 937160.0 -257000.0 -4.62 -7.6282 -0.9899 1965177 CMLD1_000142 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(nc7)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G17 compound treatment 1309960.0 34200.0 0.57 1259720.0 66000.0 1.19 1.2457 0.944 1965178 CMLD1_000143 CC(=CC1CCCCC1)[C@@H](NC(=O)c2ccc(cc2)C(F)(F)F)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G18 compound treatment 1345760.0 70000.0 1.17 1237320.0 43600.0 0.79 1.384 0.981 1965179 CMLD1_000144 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(OC(F)(F)F)cc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G19 compound treatment 1329840.0 54100.0 0.91 1246600.0 52900.0 0.95 1.3138 0.9997 1965180 CMLD1_000145 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccccc3C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G20 compound treatment 1307520.0 31800.0 0.53 1213360.0 19600.0 0.35 0.6262 0.9802 1965181 CMLD1_000146 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccc(OC)c(Br)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G21 compound treatment 1295600.0 19900.0 0.33 1222040.0 28300.0 0.51 0.5958 0.9786 1965182 CMLD1_000147 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@H]3[C@H](CC(=O)C(=O)N4CCCC4)C(=O)C[C@H]3CN1C(=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G22 mock treatment 1324920.0 49200.0 0.82 1244680.0 50900.0 0.92 1.2311 0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G23 mock treatment 1292840.0 17100.0 0.29 1204600.0 10900.0 0.2 0.3409 0.9827 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 G24 mock treatment 1300520.0 24800.0 0.42 1228280.0 34500.0 0.62 0.7335 0.9806 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H01 compound treatment 1401560.0 126000.0 2.11 1312400.0 119000.0 2.14 3.0008 1.0 1965183 CMLD1_000148 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccccn6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H02 compound treatment 1428200.0 152000.0 2.55 1298920.0 105000.0 1.89 3.1443 0.9893 1965184 CMLD1_000149 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(nc7)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H03 compound treatment 1387240.0 112000.0 1.87 1276680.0 82900.0 1.49 2.3763 0.9939 1965185 CMLD1_000150 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccccn7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H04 compound treatment 1363920.0 88200.0 1.48 1296560.0 103000.0 1.85 2.3536 0.9937 1965186 CMLD1_000151 CCCC[C@H]1C[C@@H]1[C@@H]2N(C[C@](O)(CC32CC3)c4ccccc4)P(=O)(c5ccccc5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H05 compound treatment 1338080.0 62400.0 1.04 1255880.0 62100.0 1.12 1.5296 0.9994 1965187 CMLD1_000152 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7nc8ccccc8[nH]7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H06 compound treatment 1403800.0 128000.0 2.14 1266280.0 72500.0 1.31 2.4397 0.9718 1965147 CMLD1_000153 CC1N(CC(O)(CC21CC2)c3ccccc3)P(=O)(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H07 compound treatment 1392960.0 117000.0 1.96 1280560.0 86800.0 1.56 2.4934 0.9937 1965188 CMLD1_000154 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7c(O)c(C)cnc7CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H08 compound treatment 1394680.0 119000.0 1.99 1260720.0 67000.0 1.21 2.261 0.9712 1965189 CMLD1_000155 CCCC1(NCC2=C(C)C(=O)C(C)C2=C1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H09 compound treatment 1382600.0 107000.0 1.79 1266040.0 72300.0 1.3 2.1858 0.9879 1965190 CMLD1_000156 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C[C@H](O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H10 compound treatment 1373120.0 97400.0 1.63 1258400.0 64700.0 1.16 1.9763 0.9864 1965191 CMLD1_000157 COC(=O)C1(CC(C)C)NCC2=C(C)C(=O)C(C)C2=C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H11 compound treatment 1378400.0 103000.0 1.72 1258800.0 65100.0 1.17 2.0439 0.9826 1965192 CMLD1_000158 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H12 compound treatment 1342960.0 67200.0 1.13 1251960.0 58200.0 1.05 1.5374 0.9994 1965193 CMLD1_000159 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H13 compound treatment 1334320.0 58600.0 0.98 1241680.0 47900.0 0.86 1.3042 0.998 1965194 CMLD1_000160 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(cc7)S(=O)(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H14 compound treatment 1361000.0 85300.0 1.43 1260000.0 66300.0 1.19 1.8533 0.9961 1965195 CMLD1_000161 C[C@@H]1C2COC(=O)OCC2C3CC[C@H]4C(OCc5ccc(F)cc5C(F)(F)F)OC[C@]6(C)[C@H]4C3=C1CN6C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H15 compound treatment 1156240.0 -119000.0 -2.0 1094280.0 -99500.0 -1.79 -2.681 -0.9985 1965196 CMLD1_000162 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(C)o7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H16 compound treatment 1274800.0 -916.0 -0.02 1222800.0 29100.0 0.52 0.3593 0.6861 1965197 CMLD1_000163 CC(=C1[C@H]2C(=C(C1=O)c3ccccc3)CN4C(=O)N(CCc5ccccc5)C(=O)[C@]24Cc6ccc(cc6)C(F)(F)F)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H17 compound treatment 1331960.0 56200.0 0.94 1233840.0 40100.0 0.72 1.1763 0.9915 1965198 CMLD1_000164 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5[nH]c(cc35)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H18 compound treatment 1347520.0 71800.0 1.2 1233160.0 39400.0 0.71 1.3518 0.9685 1965199 CMLD1_000165 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CC7CC7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H19 compound treatment 1319000.0 43300.0 0.72 1212040.0 18300.0 0.33 0.7453 0.9365 1965200 CMLD1_000166 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H20 compound treatment 1287400.0 11700.0 0.2 1187880.0 -5870.0 -0.11 0.0635 0.2858 1965201 CMLD1_000167 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCSCCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H21 compound treatment 1292000.0 16300.0 0.27 1222080.0 28300.0 0.51 0.5537 0.9568 1965202 CMLD1_000168 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccc(O)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H22 mock treatment 1300280.0 24600.0 0.41 1196600.0 2850.0 0.05 0.327 0.7894 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H23 mock treatment 1278960.0 3240.0 0.05 1206760.0 13000.0 0.23 0.2042 0.8484 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 H24 mock treatment 1279920.0 4200.0 0.07 1192240.0 -1510.0 -0.03 0.0306 0.4054 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I01 compound treatment 1375920.0 100000.0 1.68 1322160.0 128000.0 2.31 2.8217 0.9875 1965203 CMLD1_000169 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1cccc(c1)C(F)(F)F)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I02 compound treatment 1374960.0 99200.0 1.66 1290840.0 97100.0 1.75 2.4114 0.9997 1965204 CMLD1_000170 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6nc7ccccc7[nH]6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I03 compound treatment 1403960.0 128000.0 2.15 1282000.0 88300.0 1.59 2.6419 0.9891 1965205 CMLD1_000171 CCCC=C(CCC)[C@@H](NP(=O)(c1ccccc1)c2ccccc2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I04 compound treatment 1352200.0 76500.0 1.28 1282320.0 88600.0 1.6 2.0335 0.994 1965206 CMLD1_000172 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(OC(F)(F)F)cc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I05 compound treatment 1392800.0 117000.0 1.96 1293880.0 100000.0 1.8 2.6612 0.9992 1965207 CMLD1_000173 CCCC=C(CCC)[C@@H](NC(=O)c1ccco1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I06 compound treatment 1278080.0 2360.0 0.04 1250440.0 56700.0 1.02 0.7503 0.7339 1965208 CMLD1_000174 COCCn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(OC)cc5)C(=O)OC)Cc21)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I07 compound treatment 1304720.0 29000.0 0.49 1247160.0 53400.0 0.96 1.0237 0.9498 1965209 CMLD1_000175 CCCCC=C[C@@H](NC(=O)c1ccc(cc1)C(F)(F)F)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I08 compound treatment 1333040.0 57300.0 0.96 1280080.0 86300.0 1.56 1.7782 0.973 1965210 CMLD1_000176 COC(=O)Cn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(OC)cc5)C(=O)OC)Cc21)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I09 compound treatment 1338400.0 62700.0 1.05 1269560.0 75800.0 1.37 1.7076 0.9915 1965211 CMLD1_000177 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccc(Cl)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I10 compound treatment 1355840.0 80100.0 1.34 1248920.0 55200.0 0.99 1.651 0.9892 1965212 CMLD1_000178 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(Cl)c(c6)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I11 compound treatment 1301880.0 26200.0 0.44 1244560.0 50800.0 0.92 0.957 0.943 1965213 CMLD1_000179 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)Cc2ccccc2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I12 compound treatment 1316560.0 40800.0 0.68 1265760.0 72000.0 1.3 1.4008 0.9552 1965214 CMLD1_000180 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cccc8ccccc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I13 compound treatment 1326880.0 51200.0 0.86 1239720.0 46000.0 0.83 1.1911 0.9999 1965215 CMLD1_000181 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I14 compound treatment 1313520.0 37800.0 0.63 1259480.0 65700.0 1.18 1.2848 0.9569 1965216 CMLD1_000182 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@H]3[C@H](CC(=O)C(=O)N(C)C)C(=O)C[C@H]3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I15 compound treatment 1352440.0 76700.0 1.28 1251920.0 58200.0 1.05 1.649 0.9949 1965217 CMLD1_000183 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccs2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I16 compound treatment 1318520.0 42800.0 0.72 1255040.0 61300.0 1.1 1.2874 0.978 1965218 CMLD1_000184 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(OC)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I17 compound treatment 1345160.0 69400.0 1.16 1247520.0 53800.0 0.97 1.5068 0.9959 1965219 CMLD1_000185 COC(=O)c1ccc(cc1)[C@H](NC(=O)c2ccccc2)[C@]3(C)C[C@H]3C4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I18 compound treatment 1350680.0 75000.0 1.25 1249440.0 55700.0 1.0 1.5966 0.9939 1965220 CMLD1_000186 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(OC(F)(F)F)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I19 compound treatment 1362760.0 87000.0 1.46 1249960.0 56200.0 1.01 1.7462 0.9842 1965221 CMLD1_000187 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccs2)c3ccccc3C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I20 compound treatment 1306280.0 30600.0 0.51 1218560.0 24800.0 0.45 0.6778 0.9978 1965222 CMLD1_000188 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(nc6)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I21 compound treatment 1286160.0 10400.0 0.17 1198480.0 4730.0 0.09 0.1839 0.9456 1965223 CMLD1_000189 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CC6CC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I22 mock treatment 1303120.0 27400.0 0.46 1204160.0 10400.0 0.19 0.457 0.9222 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I23 mock treatment 1289880.0 14200.0 0.24 1204040.0 10300.0 0.19 0.2988 0.9926 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 I24 mock treatment 1289000.0 13300.0 0.22 1197960.0 4210.0 0.08 0.2109 0.8977 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J01 compound treatment 1429120.0 153000.0 2.57 1298680.0 105000.0 1.89 3.1521 0.9887 1965224 CMLD1_000190 COC(=O)Cn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccccc5)C(=O)OC)Cc21)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J02 compound treatment 571440.0 -704000.0 -11.79 793040.0 -401000.0 -7.22 -13.4388 -0.9723 1965225 CMLD1_000191 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(C)o7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J03 compound treatment 1388000.0 112000.0 1.88 1274480.0 80700.0 1.45 2.3572 0.992 1965226 CMLD1_000192 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(nc7)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J04 compound treatment 1385640.0 110000.0 1.84 1307560.0 114000.0 2.05 2.7507 0.9985 1965227 CMLD1_000193 CCCC[C@H]1C[C@@H]1[C@@H]2N([C@@](CO)(CC32CC3)c4ccccc4)P(=O)(c5ccccc5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J05 compound treatment 1346240.0 70500.0 1.18 1268960.0 75200.0 1.36 1.7928 0.9976 1965228 CMLD1_000194 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccsc7Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J06 compound treatment 1380600.0 105000.0 1.76 1287880.0 94100.0 1.7 2.4404 0.9999 1965229 CMLD1_000195 OC1(CN(CC2(CC2)C1)P(=O)(c3ccccc3)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J07 compound treatment 1389000.0 113000.0 1.9 1266880.0 73100.0 1.32 2.2722 0.9842 1965230 CMLD1_000196 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5[nH]c(cc35)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J08 compound treatment 1351920.0 76200.0 1.28 1270480.0 76700.0 1.38 1.8793 0.9992 1965231 CMLD1_000197 CCCC1(NCC2=C(C(C)C)C(=O)C(C)C2=C1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J09 compound treatment 1346080.0 70400.0 1.18 1286200.0 92500.0 1.67 2.0105 0.9856 1965232 CMLD1_000198 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J10 compound treatment 1327600.0 51900.0 0.87 1276160.0 82400.0 1.48 1.6639 0.9673 1965233 CMLD1_000199 COC(=O)C1(CC(C)C)NCC2=C(C(C)C)C(=O)C(C)C2=C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J11 compound treatment 1371520.0 95800.0 1.6 1270600.0 76900.0 1.38 2.1128 0.9973 1965234 CMLD1_000200 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J12 compound treatment 1287800.0 12100.0 0.2 1226920.0 33200.0 0.6 0.5656 0.8964 1965235 CMLD1_000201 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1Cc5cccc(Cl)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J13 compound treatment 1268200.0 -7520.0 -0.13 1273080.0 79300.0 1.43 0.9218 0.6424 1965236 CMLD1_000202 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(cc7)S(=O)(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J14 compound treatment 1331080.0 55400.0 0.93 1234200.0 40500.0 0.73 1.1705 0.9929 1965237 CMLD1_000203 CC[C@@H]1C(COC(=O)C)C(COC(=O)C)C2CC[C@H]3C(OCc4ccc(F)cc4C(F)(F)F)OC[C@]5(C)[C@H]3C2=C1CN5C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J15 compound treatment 1313240.0 37500.0 0.63 1228440.0 34700.0 0.63 0.886 1.0 1965238 CMLD1_000204 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J16 compound treatment 1268640.0 -7080.0 -0.12 1206400.0 12700.0 0.23 0.0775 0.3016 1965239 CMLD1_000205 CC(=C1[C@H]2C(=C(C1=O)c3ccccc3)CN4C(=O)N(CCc5ccccc5)C(=O)[C@]24C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J17 compound treatment 1332480.0 56800.0 0.95 1230720.0 37000.0 0.67 1.1428 0.9849 1965240 CMLD1_000206 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCSCCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J18 compound treatment 1333720.0 58000.0 0.97 1217120.0 23400.0 0.42 0.9842 0.9301 1965241 CMLD1_000207 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCn6cc(nc6C)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J19 compound treatment 1290960.0 15200.0 0.26 1215520.0 21800.0 0.39 0.4578 0.9783 1965242 CMLD1_000208 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccccn7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J20 compound treatment 1283280.0 7560.0 0.13 1190880.0 -2870.0 -0.05 0.053 0.3877 1965243 CMLD1_000209 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J21 compound treatment 1290000.0 14300.0 0.24 1197360.0 3610.0 0.07 0.2151 0.8681 1965244 CMLD1_000210 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccc(O)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J22 mock treatment 1301480.0 25800.0 0.43 1213000.0 19300.0 0.35 0.5502 0.9942 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J23 mock treatment 1290760.0 15000.0 0.25 1187040.0 -6710.0 -0.12 0.0926 0.3316 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 J24 mock treatment 1287480.0 11800.0 0.2 1178600.0 -15100.0 -0.27 -0.0538 -0.1597 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K01 compound treatment 1398160.0 122000.0 2.05 1280240.0 86500.0 1.56 2.5508 0.9909 1965245 CMLD1_000211 CCCC=C(CCC)[C@@H](NP(=O)(c1ccccc1)c2ccccc2)c3ccc(cc3)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K02 compound treatment 1374360.0 98600.0 1.65 1291280.0 97500.0 1.76 2.4099 0.9995 1965246 CMLD1_000212 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7c[nH]c8cc(F)ccc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K03 compound treatment 1351840.0 76100.0 1.27 1285040.0 91300.0 1.64 2.0639 0.992 1965247 CMLD1_000213 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1cccc2cccnc12)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K04 compound treatment 1330560.0 54800.0 0.92 1282360.0 88600.0 1.6 1.7779 0.9654 1965248 CMLD1_000214 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(F)c(F)c(F)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K05 compound treatment 1344440.0 68700.0 1.15 1279680.0 85900.0 1.55 1.908 0.9893 1965249 CMLD1_000215 CCCC=C(CCC)[C@@H](NC(=O)C(C)(C)C)c1ccc(cc1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K06 compound treatment 1367040.0 91300.0 1.53 1294640.0 101000.0 1.82 2.3661 0.9963 1965250 CMLD1_000216 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(F)c(F)c(F)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K07 compound treatment 1336000.0 60300.0 1.01 1273280.0 79500.0 1.43 1.7266 0.9852 1965251 CMLD1_000217 CCCCC=C[C@@H](NC(=O)c1ccc(cc1)C(=O)OC)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K08 compound treatment 1302760.0 27000.0 0.45 1261600.0 67900.0 1.22 1.1845 0.9086 1965252 CMLD1_000218 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6c[nH]c7ccc(O)cc67 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K09 compound treatment 1329280.0 53600.0 0.9 1264520.0 70800.0 1.28 1.5355 0.9851 1965253 CMLD1_000219 CCCC=C(CCC)[C@@H](NC(=O)Cc1ccccc1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K10 compound treatment 1310040.0 34300.0 0.57 1254480.0 60700.0 1.09 1.1799 0.9547 1965254 CMLD1_000220 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(Cl)c(c7)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K11 compound treatment 1320200.0 44500.0 0.74 1244200.0 50500.0 0.91 1.1692 0.9951 1965255 CMLD1_000221 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccco2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K12 compound treatment 1327560.0 51800.0 0.87 1247280.0 53500.0 0.96 1.2955 0.9986 1965256 CMLD1_000222 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7c[nH]c8ccc(OC)cc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K13 compound treatment 1271720.0 -4000.0 -0.07 1257960.0 64200.0 1.16 0.7708 0.6651 1965257 CMLD1_000223 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccco2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K14 compound treatment 1331360.0 55600.0 0.93 1265280.0 71500.0 1.29 1.5698 0.9873 1965258 CMLD1_000224 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(nc6)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K15 compound treatment 1249400.0 -26300.0 -0.44 1222600.0 28900.0 0.52 0.0562 0.0825 1965259 CMLD1_000225 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccnc2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K16 compound treatment 1311640.0 35900.0 0.6 1232840.0 39100.0 0.7 0.9232 0.9969 1965260 CMLD1_000226 COC(=O)Cn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(OC)cc5)C(=O)OC)Cc21)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K17 compound treatment 1336400.0 60700.0 1.02 1242800.0 49100.0 0.88 1.343 0.9976 1965261 CMLD1_000227 COC(=O)c1ccc(cc1)[C@H](NC(=O)c2ccco2)[C@]3(C)C[C@H]3C4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K18 compound treatment 1288480.0 12800.0 0.21 1246800.0 53100.0 0.96 0.827 0.8443 1965262 CMLD1_000228 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cc(F)cc8COCOc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K19 compound treatment 1273400.0 -2320.0 -0.04 1210280.0 16500.0 0.3 0.1832 0.61 1965263 CMLD1_000229 CCCC[C@@H]1C[C@H]1[C@@H](NP(=O)(c2ccccc2)c3ccccc3)c4ccc(Cl)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K20 compound treatment 602520.0 -673000.0 -11.27 838720.0 -355000.0 -6.4 -12.4891 -0.964 1965264 CMLD1_000230 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(C)c(F)c7F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K21 compound treatment 1283720.0 8000.0 0.13 1224200.0 30500.0 0.55 0.4827 0.8546 1965265 CMLD1_000231 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)o6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K22 mock treatment 1318920.0 43200.0 0.72 1229520.0 35800.0 0.64 0.967 0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K23 mock treatment 1275880.0 164.0 0.0 1199000.0 5250.0 0.09 0.0689 0.7273 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 K24 mock treatment 1242480.0 -33200.0 -0.56 1189920.0 -3830.0 -0.07 -0.442 -0.7887 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L01 compound treatment 1387200.0 111000.0 1.87 1280040.0 86300.0 1.55 2.4186 0.9959 1965266 CMLD1_000232 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCN7CNCC7=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L02 compound treatment 1394280.0 119000.0 1.98 1258080.0 64300.0 1.16 2.2226 0.9672 1965267 CMLD1_000233 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L03 compound treatment 1349920.0 74200.0 1.24 1262480.0 68700.0 1.24 1.7537 1.0 1965268 CMLD1_000234 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(O)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L04 compound treatment 1370680.0 95000.0 1.59 1274240.0 80500.0 1.45 2.1492 0.999 1965269 CMLD1_000235 CCCC[C@H]1C[C@@H]1[C@@H]2N([C@@H](CC32CC3)c4cccc(OC)c4)C(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L05 compound treatment 1351760.0 76000.0 1.27 1273160.0 79400.0 1.43 1.9116 0.9983 1965270 CMLD1_000236 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7cc8ccccc8[nH]7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L06 compound treatment 1386000.0 110000.0 1.85 1263360.0 69600.0 1.25 2.1919 0.9823 1965271 CMLD1_000237 C=C(CC1(CNP(=O)(c2ccccc2)c3ccccc3)CC1)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L07 compound treatment 1361200.0 85500.0 1.43 1239520.0 45800.0 0.82 1.5947 0.9658 1965272 CMLD1_000238 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L08 compound treatment 1310160.0 34400.0 0.58 1248680.0 54900.0 0.99 1.1074 0.9669 1965273 CMLD1_000239 CCCC1(NCC2=C(C(=O)C(C)C2=C1)c3ccccc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L09 compound treatment 1331960.0 56200.0 0.94 1268960.0 75200.0 1.36 1.6238 0.9841 1965274 CMLD1_000240 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(O)c(OC)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L10 compound treatment 1291360.0 15600.0 0.26 1220840.0 27100.0 0.49 0.5303 0.9573 1965275 CMLD1_000241 COC(=O)C1(CC(C)C)NCC2=C(C(=O)C(C)C2=C1)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L11 compound treatment 1315640.0 39900.0 0.67 1237000.0 43300.0 0.78 1.0235 0.9971 1965276 CMLD1_000242 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCF 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L12 compound treatment 1220720.0 -55000.0 -0.92 1154600.0 -39100.0 -0.71 -1.1495 -0.9914 1965277 CMLD1_000243 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1Cc5cc(F)cc(F)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L13 compound treatment 1260280.0 -15400.0 -0.26 1229320.0 35600.0 0.64 0.2706 0.3915 1965278 CMLD1_000244 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L14 compound treatment 1243440.0 -32300.0 -0.54 1208160.0 14400.0 0.26 -0.1983 -0.3308 1965279 CMLD1_000245 CC[C@@H]1C2COC(=O)OCC2C3CC[C@H]4C(OCc5ccc(F)cc5C(F)(F)F)OC[C@]6(C)[C@H]4C3=C1CN6C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L15 compound treatment 1337720.0 62000.0 1.04 1231560.0 37800.0 0.68 1.2155 0.9792 1965280 CMLD1_000246 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C[C@H](O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L16 compound treatment 1291640.0 15900.0 0.27 1214320.0 20600.0 0.37 0.4506 0.9869 1965281 CMLD1_000247 CC(=C1[C@H]2C(=C(C1=O)c3ccccc3)CN4C(=O)N(CCc5ccccc5)C(=O)[C@]24Cc6ccccc6)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L17 compound treatment 1329640.0 53900.0 0.9 1232400.0 38700.0 0.7 1.1306 0.9918 1965282 CMLD1_000248 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCSC(=N)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L18 compound treatment 1369200.0 93500.0 1.56 1236920.0 43200.0 0.78 1.6563 0.948 1965079 CMLD1_000249 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5C[C@H](O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L19 compound treatment 1286240.0 10500.0 0.18 1213640.0 19900.0 0.36 0.378 0.9465 1965283 CMLD1_000250 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7c[nH]c8cc(F)ccc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L20 compound treatment 1286840.0 11100.0 0.19 1199280.0 5530.0 0.1 0.2021 0.9572 1965284 CMLD1_000251 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(cc6)S(=O)(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L21 compound treatment 1305040.0 29300.0 0.49 1197440.0 3690.0 0.07 0.3941 0.7957 1965285 CMLD1_000252 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCN6CNCC6=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L22 mock treatment 1301160.0 25400.0 0.43 1191720.0 -2030.0 -0.04 0.2753 0.6441 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L23 mock treatment 1262240.0 -13500.0 -0.23 1174760.0 -19000.0 -0.34 -0.4013 -0.9796 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 L24 mock treatment 1265920.0 -9800.0 -0.16 1195160.0 1410.0 0.03 -0.0979 -0.5901 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M01 compound treatment 1361160.0 85400.0 1.43 1289800.0 96100.0 1.73 2.2348 0.9955 1965286 CMLD1_000253 CCCC=C(CCC)[C@@H](NC(=O)c1cccs1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M02 compound treatment 1264480.0 -11200.0 -0.19 1269000.0 75300.0 1.36 0.8258 0.6033 1965287 CMLD1_000254 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@H]3[C@H](CC(=O)C(=O)N4CCCC4)C(=O)C=C3CN1C(=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M03 compound treatment 1376920.0 101000.0 1.69 1306360.0 113000.0 2.03 2.6323 0.996 1965288 CMLD1_000255 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1ccc(cc1)C(F)(F)F)c2ccc(cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M04 compound treatment 1343280.0 67600.0 1.13 1291920.0 98200.0 1.77 2.0502 0.9766 1965289 CMLD1_000256 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7c(C)onc7c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M05 compound treatment 1354160.0 78400.0 1.31 1272320.0 78600.0 1.42 1.9293 0.9993 1965290 CMLD1_000257 CCCC=C(CCC)[C@@H](NC(=O)c1ccc(cc1)c2ccccc2)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M06 compound treatment 1325520.0 49800.0 0.83 1285960.0 92200.0 1.66 1.7642 0.9491 1965090 CMLD1_000258 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)c2ccc(cc2)c3ccccc3)c4cccc(Cl)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M07 compound treatment 1369680.0 94000.0 1.57 1277880.0 84100.0 1.52 2.1838 0.9998 1965291 CMLD1_000259 CCCCC=C[C@@H](NC(=O)c1ccco1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M08 compound treatment 1311160.0 35400.0 0.59 1258400.0 64700.0 1.16 1.2431 0.951 1965292 CMLD1_000260 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@H]3[C@H](CC(=O)C(=O)N(C)C)C(=O)C=C3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M09 compound treatment 1193000.0 -82700.0 -1.38 1210560.0 16800.0 0.3 -0.7646 -0.5396 1965293 CMLD1_000261 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)OCc2ccccc2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M10 compound treatment 1281920.0 6200.0 0.1 1233440.0 39700.0 0.72 0.5791 0.8014 1965294 CMLD1_000262 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCCNc6ccc(cc6Cl)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M11 compound treatment 1323200.0 47500.0 0.79 1222480.0 28700.0 0.52 0.928 0.9785 1965295 CMLD1_000263 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2cccnc2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M12 compound treatment 1269440.0 -6280.0 -0.11 1219440.0 25700.0 0.46 0.2531 0.5331 1965296 CMLD1_000264 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccc(OC)c(Br)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M13 compound treatment 1257920.0 -17800.0 -0.3 1213680.0 19900.0 0.36 0.0434 0.093 1965297 CMLD1_000265 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M14 compound treatment 1299480.0 23800.0 0.4 1232920.0 39200.0 0.71 0.7803 0.9632 1965298 CMLD1_000266 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccsc6Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M15 compound treatment 1298160.0 22400.0 0.38 1222560.0 28800.0 0.52 0.6327 0.9874 1965299 CMLD1_000267 CCCC[C@@H]1C[C@H]1[C@@H](NS(=O)(=O)c2cccc3cccnc23)c4ccc(cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M16 compound treatment 1290840.0 15100.0 0.25 1224320.0 30600.0 0.55 0.5685 0.9377 1965300 CMLD1_000268 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6ccc(O)c(O)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M17 compound treatment 1273440.0 -2280.0 -0.04 1210760.0 17000.0 0.31 0.1898 0.6145 1965301 CMLD1_000269 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NS(=O)(=O)c2cccc3cccnc23)c4ccc(Cl)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M18 compound treatment 1297480.0 21800.0 0.36 1217320.0 23600.0 0.42 0.5579 0.9971 1965302 CMLD1_000270 COC(=O)[C@@]1(Cc2ccccc2)[C@H]3[C@H](CC(=O)C(=O)N(C)C)C(=O)C[C@H]3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M19 compound treatment 1300160.0 24400.0 0.41 1211520.0 17800.0 0.32 0.5157 0.9927 1965303 CMLD1_000271 CCCC=C(CCC)[C@@H](NC(=O)Oc1ccc(F)cc1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M20 compound treatment 1280360.0 4640.0 0.08 1196360.0 2610.0 0.05 0.0883 0.9712 1965304 CMLD1_000272 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)c(F)c6F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M21 mock treatment 1258160.0 -17600.0 -0.29 1190040.0 -3710.0 -0.07 -0.255 -0.8462 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M22 mock treatment 1284320.0 8600.0 0.14 1187400.0 -6350.0 -0.11 0.021 0.1141 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M23 mock treatment 1266360.0 -9360.0 -0.16 1190320.0 -3430.0 -0.06 -0.1544 -0.9171 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 M24 mock treatment 1260320.0 -15400.0 -0.26 1179320.0 -14400.0 -0.26 -0.366 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N01 compound treatment 1419120.0 143000.0 2.4 1281520.0 87800.0 1.58 2.8152 0.9795 1965305 CMLD1_000273 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCN6CNCC6=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N02 compound treatment 1350920.0 75200.0 1.26 1260760.0 67000.0 1.21 1.7437 0.9998 1965306 CMLD1_000274 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N03 compound treatment 357880.0 -918000.0 -15.36 595360.0 -598000.0 -10.78 -18.4843 -0.985 1965307 CMLD1_000275 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(C)o6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N04 compound treatment 1289080.0 13400.0 0.22 1248280.0 54500.0 0.98 0.8529 0.8464 1965308 CMLD1_000276 COC(=O)c1ccc(C#CC(NP(=O)(c2ccccc2)c3ccccc3)c4ccccc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N05 compound treatment 1335280.0 59600.0 1.0 1251440.0 57700.0 1.04 1.4399 0.9998 1965309 CMLD1_000277 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(C)c(F)c7F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N06 compound treatment 1337560.0 61800.0 1.03 1240920.0 47200.0 0.85 1.3328 0.9952 1965310 CMLD1_000278 O=P(NCC1(CC2(CO2)c3ccccc3)CC1)(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N07 compound treatment 1367280.0 91600.0 1.53 1253280.0 59500.0 1.07 1.842 0.9848 1965311 CMLD1_000279 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5C[C@H](O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N08 compound treatment 1294840.0 19100.0 0.32 1210760.0 17000.0 0.31 0.4431 0.9998 1965312 CMLD1_000280 CCCCCC1=C2CNC(CCC)(C=C2C(C)C1=O)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N09 compound treatment 1336240.0 60500.0 1.01 1225640.0 31900.0 0.57 1.1225 0.964 1965313 CMLD1_000281 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCN7CCOCC7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N10 compound treatment 1269800.0 -5920.0 -0.1 1194360.0 615.0 0.01 -0.0622 -0.6241 1965314 CMLD1_000282 CCCCCC1=C2CNC(CC(C)C)(C=C2C(C)C1=O)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N11 compound treatment 1316880.0 41200.0 0.69 1215840.0 22100.0 0.4 0.7686 0.966 1965315 CMLD1_000283 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cc(C)n(C)n7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N12 compound treatment 1258240.0 -17500.0 -0.29 1211600.0 17900.0 0.32 0.0207 0.0475 1965316 CMLD1_000284 COC1OC[C@]2(C)[C@@H]3[C@H]1CCC4C(CO)C(CO)[C@@H](C)C(=C43)CN2C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N13 compound treatment 1303080.0 27400.0 0.46 1220080.0 26300.0 0.47 0.6593 0.9998 1965317 CMLD1_000285 COC(=O)Cn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccccc5)C(=O)OC)Cc21)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N14 compound treatment 1281120.0 5400.0 0.09 1212520.0 18800.0 0.34 0.3031 0.8657 1965318 CMLD1_000286 CC[C@@H]1C(COC)C(COC)C2CC[C@H]3C(OCc4ccc(F)cc4C(F)(F)F)OC[C@]5(C)[C@H]3C2=C1CN5C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N15 compound treatment 1291800.0 16100.0 0.27 1208560.0 14800.0 0.27 0.3791 1.0 1965319 CMLD1_000287 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6c(O)c(C)cnc6CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N16 compound treatment 1286600.0 10900.0 0.18 1202840.0 9090.0 0.16 0.2447 0.9986 1965320 CMLD1_000288 CC1(C)C(=O)C(=C2CN3C(=O)N(CCc4ccccc4)C(=O)C3(Cc5ccccc5)C=C21)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N17 compound treatment 1270800.0 -4920.0 -0.08 1204640.0 10900.0 0.2 0.0806 0.3788 1965321 CMLD1_000289 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5[nH]c(cc35)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N18 compound treatment 1275360.0 -356.0 -0.01 1193000.0 -745.0 -0.01 -0.0137 -0.9332 1965322 CMLD1_000290 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5[nH]c(cc35)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N19 compound treatment 1188280.0 -87400.0 -1.46 1172360.0 -21400.0 -0.39 -1.3071 -0.8639 1965323 CMLD1_000291 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7c[nH]c8ccc(O)cc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N20 compound treatment 1243400.0 -32300.0 -0.54 1171680.0 -22100.0 -0.4 -0.6635 -0.9885 1965324 CMLD1_000292 COCCn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(F)cc5)C(=O)OC)Cc21)C(=O)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N21 mock treatment 1235280.0 -40400.0 -0.68 1174600.0 -19100.0 -0.34 -0.7224 -0.9511 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N22 mock treatment 1271560.0 -4160.0 -0.07 1180360.0 -13400.0 -0.24 -0.2197 -0.8754 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N23 mock treatment 1239840.0 -35900.0 -0.6 1141760.0 -52000.0 -0.94 -1.0868 -0.9769 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 N24 mock treatment 1259160.0 -16600.0 -0.28 1181080.0 -12700.0 -0.23 -0.3573 -0.9954 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O01 compound treatment 1376920.0 101000.0 1.69 1283680.0 89900.0 1.62 2.3433 0.9998 1965325 CMLD1_000293 CCCC=C(CCC)[C@@H](NC(=O)OCC(C)C)c1ccc(cc1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O02 compound treatment 1252920.0 -22800.0 -0.38 1280880.0 87100.0 1.57 0.8404 0.5201 1965326 CMLD1_000294 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O03 compound treatment 1309120.0 33400.0 0.56 1256440.0 62700.0 1.13 1.194 0.9474 1965327 CMLD1_000295 CCCC=C(CCC)[C@@H](NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O04 compound treatment 1308600.0 32900.0 0.55 1247920.0 54200.0 0.98 1.0793 0.9632 1965268 CMLD1_000296 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(O)c(OC)c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O05 compound treatment 1304640.0 28900.0 0.48 1238840.0 45100.0 0.81 0.9168 0.9694 1965328 CMLD1_000297 CCCC=C(CCC)[C@@H](NS(=O)(=O)c1cccs1)c2ccc(cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O06 compound treatment 1313960.0 38200.0 0.64 1260680.0 66900.0 1.21 1.3053 0.9561 1965329 CMLD1_000298 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7cccc8ccccc78 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O07 compound treatment 1281920.0 6200.0 0.1 1264040.0 70300.0 1.27 0.969 0.7625 1965330 CMLD1_000299 CCCCC=C[C@@H](NC(=O)c1cccs1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O08 compound treatment 1308840.0 33100.0 0.55 1237360.0 43600.0 0.79 0.9476 0.9854 1965331 CMLD1_000300 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCF 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O09 compound treatment 1294600.0 18900.0 0.32 1248040.0 54300.0 0.98 0.9152 0.8902 1965332 CMLD1_000301 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccc(cc2)C(F)(F)F)c3ccc(cc3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O10 compound treatment 1242320.0 -33400.0 -0.56 1203320.0 9570.0 0.17 -0.2732 -0.4671 1965333 CMLD1_000302 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@H]3[C@H](CC(=O)C(=O)N(C)C)C(=O)C[C@H]3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O11 compound treatment 1265720.0 -10000.0 -0.17 1206320.0 12600.0 0.23 0.0419 0.1488 1965334 CMLD1_000303 CCCC=C(CCC)[C@@H](NC(=O)c1ccccc1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O12 compound treatment 1243560.0 -32200.0 -0.54 1216840.0 23100.0 0.42 -0.0863 -0.1268 1965335 CMLD1_000304 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCc7ccc(OC)c(Br)c7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O13 compound treatment 1306240.0 30500.0 0.51 1214400.0 20700.0 0.37 0.6243 0.9879 1965336 CMLD1_000305 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)Cc2ccccc2)c3ccc(cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O14 compound treatment 1221280.0 -54400.0 -0.91 1183280.0 -10500.0 -0.19 -0.7775 -0.8358 1965337 CMLD1_000306 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccsc7Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O15 compound treatment 1278160.0 2440.0 0.04 1213960.0 20200.0 0.36 0.2865 0.7816 1965338 CMLD1_000307 CCCC[C@@H]1C[C@H]1[C@@H](NC(=O)c2ccccc2)c3ccc(cc3)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O16 compound treatment 1221520.0 -54200.0 -0.91 1195040.0 1290.0 0.02 -0.6248 -0.6887 1965339 CMLD1_000308 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6nc7ccccc7[nH]6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O17 compound treatment 1250120.0 -25600.0 -0.43 1193160.0 -585.0 -0.01 -0.3103 -0.7243 1965340 CMLD1_000309 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)c2ccco2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O18 compound treatment 1228560.0 -47200.0 -0.79 1192640.0 -1110.0 -0.02 -0.5721 -0.7247 1965341 CMLD1_000310 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCSCCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O19 compound treatment 1159200.0 -117000.0 -1.95 1129360.0 -64400.0 -1.16 -2.199 -0.9692 1965342 CMLD1_000311 CCC[C@@H]1C[C@@]1(CCC)[C@@H](NC(=O)c2cccs2)c3ccc(Cl)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O20 compound treatment 290080.0 -986000.0 -16.49 462680.0 -731000.0 -13.17 -20.977 -0.9938 1965343 CMLD1_000312 COC(=O)[C@@]1(Cc2ccccc2)[C@H]3[C@H](CC(=O)C(=O)N(C)C)C(=O)C=C3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O21 mock treatment 1234920.0 -40800.0 -0.68 1146080.0 -47700.0 -0.86 -1.09 -0.9935 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O22 mock treatment 1237520.0 -38200.0 -0.64 1174600.0 -19100.0 -0.34 -0.6959 -0.9581 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O23 mock treatment 1230880.0 -44800.0 -0.75 1149400.0 -44300.0 -0.8 -1.0955 -0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 O24 mock treatment 1233400.0 -42300.0 -0.71 1185000.0 -8750.0 -0.16 -0.6121 -0.8438 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P01 compound treatment 1361760.0 86000.0 1.44 1251120.0 57400.0 1.03 1.7491 0.9868 1965344 CMLD1_000313 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6ccc(cc6)S(=O)(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P02 compound treatment 1314280.0 38600.0 0.65 1253440.0 59700.0 1.08 1.2168 0.9701 1965345 CMLD1_000314 COC(=O)Cn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(F)cc5)C(=O)OC)Cc21)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P03 compound treatment 1116280.0 -159000.0 -2.67 1120680.0 -73100.0 -1.32 -2.8175 -0.947 1965346 CMLD1_000315 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCc6c[nH]c7ccc(O)cc67 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P04 compound treatment 1011000.0 -265000.0 -4.43 970600.0 -223000.0 -4.02 -5.9753 -0.9988 1965347 CMLD1_000316 COC(=O)c1ccc(cc1)C23CC3(C2)C(NP(=O)(c4ccccc4)c5ccccc5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P05 compound treatment 1262760.0 -13000.0 -0.22 1218840.0 25100.0 0.45 0.1664 0.3318 1965348 CMLD1_000317 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7ccc(Cl)c(c7)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P06 compound treatment 1280560.0 4840.0 0.08 1208680.0 14900.0 0.27 0.2476 0.881 1965349 CMLD1_000318 COCC1[C@@H](C)C2=C3C(CC[C@H]4C(OCc5ccc(F)cc5C(F)(F)F)OC[C@](C)([C@H]43)N(C2)C(=O)OC(C)(C)C)C1COC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P07 compound treatment 1313040.0 37300.0 0.62 1224600.0 30900.0 0.56 0.8347 0.9983 1965350 CMLD1_000319 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5Cc7c(O)c(C)cnc7CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P08 compound treatment 1254800.0 -20900.0 -0.35 1204360.0 10600.0 0.19 -0.1123 -0.2815 1965351 CMLD1_000320 COC(=O)C1(Cc2ccccc2)NCC3=C(C)C(=O)C(C)C3=C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P09 compound treatment 1311800.0 36100.0 0.6 1230200.0 36500.0 0.66 0.8914 0.9991 1965352 CMLD1_000321 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N6CCCC6)n5CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P10 compound treatment 1204680.0 -71000.0 -1.19 1167680.0 -26100.0 -0.47 -1.1727 -0.9175 1965353 CMLD1_000322 CCCc1cc2C3C(CN(C(=O)c4ccccc4)C3(C)C(=O)OC)C(C)c2n1Cc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P11 compound treatment 1286840.0 11100.0 0.19 1217800.0 24100.0 0.43 0.4381 0.9288 1965354 CMLD1_000323 COCCn1c(cc2[C@H]3[C@H](CN(C(=O)c4ccccc4)[C@@]3(Cc5ccc(OC)cc5)C(=O)OC)Cc21)C(=O)N6CCCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P12 compound treatment 1286320.0 10600.0 0.18 1196440.0 2690.0 0.05 0.1598 0.8686 1965355 CMLD1_000324 CC[C@@H]1C(CO)C(CO)C2CC[C@H]3C(OC)OC[C@]4(C)[C@H]3C2=C1CN4C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P13 compound treatment 1275440.0 -276.0 0.0 1205880.0 12100.0 0.22 0.1513 0.692 1965356 CMLD1_000325 COC(=O)[C@@]1(Cc2ccc(OC)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6c(O)c(C)cnc6OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P14 compound treatment 1240440.0 -35300.0 -0.59 1187000.0 -6750.0 -0.12 -0.5034 -0.8352 1965357 CMLD1_000326 COCC1[C@@H](C)C2=C3C(CC[C@H]4C(OCc5ccc(OC)cc5)OC[C@](C)([C@H]43)N(C2)C(=O)OC(C)(C)C)C1COC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P15 compound treatment 1279320.0 3600.0 0.06 1185400.0 -8350.0 -0.15 -0.0637 -0.3931 1965358 CMLD1_000327 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCn6cc(nc6C)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P16 compound treatment 1226320.0 -49400.0 -0.83 1182800.0 -10900.0 -0.2 -0.724 -0.8519 1965359 CMLD1_000328 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6cc(F)cc7COCOc67 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P17 compound treatment 170320.0 -1110000.0 -18.5 213240.0 -981000.0 -17.67 -25.572 -0.9997 1965360 CMLD1_000329 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@H]3C(=C)C(=O)C=C3CN1C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P18 compound treatment 1238920.0 -36800.0 -0.62 1174280.0 -19500.0 -0.35 -0.6834 -0.9644 1965361 CMLD1_000330 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P19 compound treatment 1168240.0 -107000.0 -1.8 1154280.0 -39500.0 -0.71 -1.7746 -0.9176 1965362 CMLD1_000331 COC(=O)[C@@]1(Cc2ccccc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5Cc6nc7ccccc7[nH]6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P20 compound treatment 1220680.0 -55000.0 -0.92 1159320.0 -34400.0 -0.62 -1.0898 -0.9815 1965363 CMLD1_000332 COC(=O)[C@@]1(Cc2ccc(F)cc2)[C@@H]3[C@H](CN1C(=O)c4ccccc4)Cc5c3cc(C(=O)N(C)C)n5CCF 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P21 mock treatment 1233760.0 -42000.0 -0.7 1164560.0 -29200.0 -0.53 -0.8683 -0.9899 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P22 mock treatment 1257640.0 -18100.0 -0.3 1155760.0 -38000.0 -0.68 -0.6978 -0.9326 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P23 mock treatment 1242640.0 -33100.0 -0.55 1164080.0 -29700.0 -0.53 -0.7693 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1462 P24 mock treatment 1258320.0 -17400.0 -0.29 1180840.0 -12900.0 -0.23 -0.3703 -0.9938 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A01 compound treatment 1288320.0 81300.0 1.36 1268400.0 74500.0 1.34 1.9108 1.0 2065621 ICCB6_000001 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccccc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A02 compound treatment 1300160.0 93100.0 1.56 1286200.0 92300.0 1.66 2.2777 0.9995 2065622 ICCB6_000002 OCCCCCCCCCc1ccc(C=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A03 compound treatment 1300640.0 93600.0 1.57 1289040.0 95100.0 1.71 2.3195 0.999 2065623 ICCB6_000003 CC1(C)OC(=O)C=C(CC(O)c2ccccc2)O1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A04 compound treatment 1182920.0 -24100.0 -0.4 1176960.0 -17000.0 -0.31 -0.5014 -0.9906 2065624 ICCB6_000004 CO[C@H]1O[C@H](CO)[C@@H](OCc2ccccc2)[C@H](OCc3ccccc3)[C@@H]1OCCCc4ccc(C=O)o4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A05 compound treatment 1237520.0 30500.0 0.51 1229600.0 35700.0 0.64 0.8153 0.9934 2065625 ICCB6_000005 Clc1ccccc1C(CC(=O)c2ccccc2)C(=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A06 compound treatment 1161480.0 -45600.0 -0.76 1144200.0 -49700.0 -0.9 -1.1724 -0.9968 2065626 ICCB6_000006 OCCCCCCCCCCc1ccc(C=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A07 compound treatment 1247240.0 40200.0 0.67 1257480.0 63600.0 1.15 1.2856 0.9679 2065627 ICCB6_000007 CCOC(=O)CC1[C@@H]2[C@@H](NCc3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A08 compound treatment 1116800.0 -90200.0 -1.51 1124920.0 -69000.0 -1.24 -1.9468 -0.9953 2065628 ICCB6_000008 OC[C@H](COCCCc1ccc(C=O)o1)OCc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A09 compound treatment 1256200.0 49200.0 0.82 1244840.0 50900.0 0.92 1.2305 0.9985 2065629 ICCB6_000009 CCOC(=O)CC1[C@@H]2[C@@H](NCc3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C(C)C)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A10 compound treatment 1219920.0 12900.0 0.22 1213760.0 19800.0 0.36 0.4053 0.9707 2065630 ICCB6_000010 OCCOCCCc1ccc(C=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A11 compound treatment 1253160.0 46100.0 0.77 1237400.0 43500.0 0.78 1.0998 1.0 2065631 ICCB6_000011 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](Cc5ccccc5)N1C(=O)Cc6ccc(OC)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A12 compound treatment 1191800.0 -15200.0 -0.25 1178200.0 -15700.0 -0.28 -0.3805 -0.9986 2065632 ICCB6_000012 OCc1ccc(CCc2ccc(C=O)o2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A13 compound treatment 1248040.0 41000.0 0.69 1247360.0 53400.0 0.96 1.1661 0.9862 2065633 ICCB6_000013 CCOC(=O)CC(C#N)(C(=O)OCC)c1nsc2ccccc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A14 compound treatment 1227160.0 20100.0 0.34 1215720.0 21800.0 0.39 0.5159 0.9971 2065634 ICCB6_000014 OCCOCCOCCCc1ccc(C=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A15 compound treatment 1212520.0 5490.0 0.09 1205600.0 11700.0 0.21 0.2138 0.9309 ICCB6_000015 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A16 compound treatment 1223600.0 16600.0 0.28 1196240.0 2320.0 0.04 0.2256 0.8046 2065635 ICCB6_000016 OCC1CC2CCN1CC2CCc3ccc(C=O)o3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A17 compound treatment 1238400.0 31400.0 0.52 1225840.0 31900.0 0.58 0.7779 0.999 1952805 ICCB6_000017 CC(C)(C)[Si](C)(C)OCCNC(=O)c1cc(cc2c(coc12)C(O)(c3ccccc3)c4ccccc4)c5cc(I)cc(I)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A18 compound treatment 1137200.0 -69800.0 -1.17 1133040.0 -60900.0 -1.1 -1.6019 -0.9995 2065636 ICCB6_000018 OCCCCNC(=O)OCCCc1ccc(C=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A19 compound treatment 1186400.0 -20600.0 -0.35 1194720.0 800.0 0.01 -0.2339 -0.677 1952839 ICCB6_000019 Oc1ccccc1C#CC#Cc2ccccc2O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A20 compound treatment 1209880.0 2850.0 0.05 1199160.0 5240.0 0.09 0.1005 0.9499 2065637 ICCB6_000020 OCCCCc1ccc(C=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A21 compound treatment 1213160.0 6130.0 0.1 1206880.0 13000.0 0.23 0.2376 0.9318 1952635 ICCB6_000021 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCC(c3ccccc3)c4ccccc4)O2)O1)OC(=O)NCc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A22 compound treatment 1005960.0 -201000.0 -3.36 998240.0 -196000.0 -3.53 -4.8723 -0.9997 2065638 ICCB6_000022 OCCCCCCc1ccc(/C=C/COC(=O)Nc2ccccc2)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A23 mock treatment 1202760.0 -4270.0 -0.07 1201920.0 8000.0 0.14 0.0514 0.3193 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 A24 mock treatment 1215800.0 8770.0 0.15 1202160.0 8240.0 0.15 0.2087 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B01 compound treatment 1295800.0 88800.0 1.49 1287800.0 93900.0 1.69 2.2464 0.9979 2065621 ICCB6_000023 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccccc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B02 compound treatment 1270480.0 63400.0 1.06 1276320.0 82400.0 1.48 1.8006 0.9865 2065639 ICCB6_000024 OB1OC(COCc2ccccc2)CC=C1C(=C)CCCc3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B03 compound treatment 1297240.0 90200.0 1.51 1283720.0 89800.0 1.62 2.2115 0.9994 2065640 ICCB6_000025 CC1(C)OC(=O)C=C(CC(O)C2CCCCC2)O1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B04 compound treatment 1265880.0 58800.0 0.98 1266840.0 72900.0 1.31 1.6254 0.9899 2065641 ICCB6_000026 CC(C)C(=C)C1=CCC(COCc2ccccc2)OB1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B05 compound treatment 1263400.0 56400.0 0.94 1270080.0 76200.0 1.37 1.6373 0.9833 2065642 ICCB6_000027 C[Si](C)(C(NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B06 compound treatment 1281080.0 74000.0 1.24 1284640.0 90700.0 1.63 2.032 0.9907 2065643 ICCB6_000028 CCCC(=C)C1=CCC(COCc2ccccc2)OB1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B07 compound treatment 1265720.0 58700.0 0.98 1249000.0 55100.0 0.99 1.3962 1.0 2065644 ICCB6_000029 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B08 compound treatment 1284080.0 77000.0 1.29 1268560.0 74600.0 1.34 1.8626 0.9998 2065645 ICCB6_000030 O[C@@H]([C@H](Oc1ccccc1)C=C)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B09 compound treatment 1251160.0 44100.0 0.74 1236680.0 42800.0 0.77 1.0669 0.9998 2065646 ICCB6_000031 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](C(C)C)N1C(=O)Cc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B10 compound treatment 1276760.0 69700.0 1.17 1255400.0 61500.0 1.11 1.6084 0.9997 2065647 ICCB6_000032 O[C@H](COCc1ccccc1)[C@H](Oc2ccccc2)C=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B11 compound treatment 1263160.0 56100.0 0.94 1250720.0 56800.0 1.02 1.3878 0.9991 2065648 ICCB6_000033 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](Cc4ccccc4)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B12 compound treatment 1263400.0 56400.0 0.94 1257320.0 63400.0 1.14 1.4747 0.9955 2065649 ICCB6_000034 CC(C)C(=C)C(=O)CCC(COCc1ccccc1)OC(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B13 compound treatment 1266560.0 59500.0 1.0 1246480.0 52600.0 0.95 1.374 0.9997 2065650 ICCB6_000035 [O-][N+](=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B14 compound treatment 1237760.0 30700.0 0.51 1235840.0 41900.0 0.76 0.8977 0.9824 2065651 ICCB6_000036 CCCC(=C=CC[C@@H](OC(=O)Nc1ccc(Br)cc1)c2ccccc2)CCOC(=O)Nc3ccc(Br)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B15 compound treatment 1223120.0 16100.0 0.27 1215920.0 22000.0 0.4 0.4707 0.9822 1952458 ICCB6_000037 Fc1ccc(cc1Br)[C@@H]2C3=C(C[C@@H]4C2=CCn5n4c(=O)n(c6ccccc6)c5=O)C(=O)OC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B16 compound treatment 1177640.0 -29400.0 -0.49 1157200.0 -36700.0 -0.66 -0.8156 -0.9893 2065652 ICCB6_000038 CC(C)C(=C=CC[C@H](COCc1ccccc1)OC(=O)c2ccc(Br)cc2)CCOC(=O)c3ccc(Br)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B17 compound treatment 1219400.0 12400.0 0.21 1197840.0 3920.0 0.07 0.1963 0.8976 1952808 ICCB6_000039 CCCCCc1cc2ccccc2o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B18 compound treatment 1239960.0 32900.0 0.55 1241880.0 48000.0 0.86 1.0007 0.9764 2065653 ICCB6_000040 CC1(C)OC[C@@H](C=C)[C@H](CCc2ccccc2)O1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B19 compound treatment 1194920.0 -12100.0 -0.2 1184680.0 -9240.0 -0.17 -0.261 -0.9952 1952842 ICCB6_000041 COC(=O)Cc1cc(cc(I)c1O)c2cc(F)cc(I)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B20 compound treatment 1209280.0 2250.0 0.04 1197680.0 3760.0 0.07 0.0745 0.9615 2065654 ICCB6_000042 CCC[C@@]1(CCO[Si](c2ccccc2)(c3ccccc3)C(C)(C)C)O[C@@H](Cc4ccccc4)CC=C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B21 compound treatment 1189600.0 -17400.0 -0.29 1193520.0 -400.0 -0.01 -0.2114 -0.7244 1952636 ICCB6_000043 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCCc3ccc(Cl)cc3)O2)O1)OC(=O)NCc4ccc5OCOc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B22 compound treatment 1185920.0 -21100.0 -0.35 1170320.0 -23600.0 -0.43 -0.5505 -0.9958 3056822 ICCB6_000044 CC(C)[Si](OC[C@H]1OB(O)C[C@@H]2[C@H]3[C@@H](CC(=C12)C)C(=O)c4ccccc4C3=O)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B23 mock treatment 1194840.0 -12200.0 -0.2 1186640.0 -7280.0 -0.13 -0.237 -0.9772 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 B24 mock treatment 1208520.0 1490.0 0.02 1219600.0 25700.0 0.46 0.3448 0.7441 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C01 compound treatment 1307040.0 100000.0 1.67 1285960.0 92000.0 1.66 2.356 1.0 2065655 ICCB6_000045 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccc(C)cc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C02 compound treatment 1213480.0 6450.0 0.11 1208600.0 14700.0 0.26 0.2633 0.9218 2065656 ICCB6_000046 C[C@@H]([C@H](O)c1ccc(CCCCCCO)o1)C(=O)N2[C@@H](C)[C@H](OC2=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C03 compound treatment 1234480.0 27400.0 0.46 1234600.0 40700.0 0.73 0.8431 0.9747 2065657 ICCB6_000047 COC(=O)c1cn2c(c1C(=O)OC)c(=O)n(C)c3ccccc32 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C04 compound treatment 1209440.0 2410.0 0.04 1206600.0 12700.0 0.23 0.19 0.8192 2065658 ICCB6_000048 C[C@@H]([C@H](O)c1ccc(CCCCCCO)o1)C(=O)N2[C@H](COC2=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C05 compound treatment 1278840.0 71800.0 1.2 1253920.0 60000.0 1.08 1.6141 0.9986 2065659 ICCB6_000049 C[Si](C)(C(NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3Cl)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C06 compound treatment 1193360.0 -13700.0 -0.23 1201000.0 7080.0 0.13 -0.0716 -0.2732 2065660 ICCB6_000050 CC(C)[C@H]1COC(=O)N1C(=O)[C@@H](C)[C@H](O)c2ccc(CCCCCCO)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C07 compound treatment 1243200.0 36200.0 0.61 1242720.0 48800.0 0.88 1.0497 0.9834 2065661 ICCB6_000051 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](C)N1C(=O)CCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C08 compound treatment 1222480.0 15400.0 0.26 1195720.0 1800.0 0.03 0.2057 0.7896 2065662 ICCB6_000052 CC(C)[C@@H]1N(C(=O)[C@@H](C)[C@H](O)c2ccc(CCCCCCO)o2)C(=O)OC1(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C09 compound treatment 1251680.0 44600.0 0.75 1242320.0 48400.0 0.87 1.145 0.997 2065663 ICCB6_000053 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](CC(C)C)N1C(=O)Cc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C10 compound treatment 998960.0 -208000.0 -3.48 943200.0 -251000.0 -4.52 -5.6563 -0.9917 2065664 ICCB6_000054 COC(=O)[C@H](Cc1ccccc1)NC(=O)OC/C=C/c2ccc(CCCCCCO)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C11 compound treatment 1233480.0 26400.0 0.44 1229760.0 35800.0 0.65 0.7696 0.983 2065665 ICCB6_000055 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](Cc4ccccc4)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C12 compound treatment 929120.0 -278000.0 -4.65 870960.0 -323000.0 -5.82 -7.4031 -0.9938 2065666 ICCB6_000056 CCc1cccc(NC(=O)OC/C=C/c2ccc(CCCCCCO)o2)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C13 compound treatment 1253360.0 46300.0 0.78 1241480.0 47600.0 0.86 1.1541 0.9988 1065064 ICCB6_000057 [O-][N+](=O)c1ccc(CBr)c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C14 compound treatment 895320.0 -312000.0 -5.22 888200.0 -306000.0 -5.51 -7.5834 -0.9996 2065667 ICCB6_000058 OCCCCCCc1ccc(/C=C/COC(=O)Nc2ccc(Oc3ccccc3)cc2)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C15 compound treatment 1161120.0 -45900.0 -0.77 1111080.0 -82800.0 -1.49 -1.5987 -0.9523 1952482 ICCB6_000059 Fc1ccc(cc1Br)[C@H]2C3=CC[C@H]4[C@@H]([C@@H]3C[C@@]5(C#N)C(=O)C(=C(Cl)C(=O)[C@@]25C#N)Cl)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C16 compound treatment 776960.0 -430000.0 -7.2 814040.0 -380000.0 -6.84 -9.9288 -0.9997 2065668 ICCB6_000060 COc1cccc(C)c1NC(=O)OC/C=C/c2ccc(CCCCCCO)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C17 compound treatment 1241880.0 34800.0 0.58 1229800.0 35900.0 0.65 0.8695 0.9987 1952809 ICCB6_000061 CC(=O)Oc1ccccc1C#Cc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C18 compound treatment 781680.0 -425000.0 -7.12 881040.0 -313000.0 -5.64 -9.0193 -0.9933 2065669 ICCB6_000062 OCCCCCCc1ccc(/C=C/COC(=O)Nc2ccc(C#N)cc2)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C19 compound treatment 1200280.0 -6750.0 -0.11 1173480.0 -20400.0 -0.37 -0.3403 -0.8834 1952773 ICCB6_000063 CCCNC(=O)c1cc(cc2c3C(=O)OC4(CCCC4)c3oc12)c5cc(F)cc(F)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C20 compound treatment 825720.0 -381000.0 -6.38 902720.0 -291000.0 -5.25 -8.222 -0.9953 2065670 ICCB6_000064 CCOC(=O)CNC(=O)OC/C=C/c1ccc(CCCCCCO)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C21 compound treatment 1165360.0 -41700.0 -0.7 1156680.0 -37200.0 -0.67 -0.9675 -0.9998 1952585 ICCB6_000065 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)CC[C@@H]2C[C@H](C[C@@]3(CCC[C@H](COC(=O)NCCCN4CCCC4=O)O3)O2)OC(=O)NCc5cccc6ccccc56 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C22 compound treatment 876600.0 -330000.0 -5.53 896240.0 -298000.0 -5.36 -7.7025 -0.9999 2065671 ICCB6_000066 OCCCCCCc1ccc(/C=C/COC(=O)Nc2ccccc2F)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C23 mock treatment 1195920.0 -11100.0 -0.19 1181880.0 -12000.0 -0.22 -0.2849 -0.9971 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 C24 mock treatment 1211560.0 4530.0 0.08 1212440.0 18500.0 0.33 0.2895 0.8462 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D01 compound treatment 1319080.0 112000.0 1.88 1289160.0 95200.0 1.72 2.5393 0.999 2065672 ICCB6_000067 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccc(Cl)cc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D02 compound treatment 1336680.0 130000.0 2.17 1317880.0 124000.0 2.23 3.1134 0.9999 2065673 ICCB6_000068 CC(C)[Si](OC[C@@H]1CC=C(C)B(O)O1)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D03 compound treatment 1287160.0 80100.0 1.34 1276560.0 82600.0 1.49 2.001 0.9986 2065674 ICCB6_000069 CCOC(=O)C1[C@H](CCc2ccccc2)O[C@H](CCc3ccccc3)CC1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D04 compound treatment 1297680.0 90600.0 1.52 1282200.0 88300.0 1.59 2.1974 0.9997 2065675 ICCB6_000070 CC(C)[Si](OC[C@H]1OB(O)CC=C1)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D05 compound treatment 1300160.0 93100.0 1.56 1279520.0 85600.0 1.54 2.1926 1.0 2065676 ICCB6_000071 C[Si](C)(C(N[Si](=O)(=O)c1ccccc1)c2ccccc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D06 compound treatment 1310160.0 103000.0 1.73 1260120.0 66200.0 1.19 2.0637 0.9837 2065677 ICCB6_000072 CC(C)[Si](OCC(O)C1=C(C)C[C@@H]2[C@H]([C@H]1CO)C(=O)N(Cc3ccccc3)C2=O)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D07 compound treatment 1283120.0 76100.0 1.27 1240040.0 46100.0 0.83 1.4879 0.9786 2065678 ICCB6_000073 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D08 compound treatment 1278680.0 71600.0 1.2 1254560.0 60600.0 1.09 1.6204 0.9989 2065679 ICCB6_000074 CC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D09 compound treatment 1267120.0 60100.0 1.01 1234240.0 40300.0 0.73 1.2247 0.9873 2065680 ICCB6_000075 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](CC(C)C)N1C(=O)CCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D10 compound treatment 1264840.0 57800.0 0.97 1235560.0 41600.0 0.75 1.2146 0.9921 2065681 ICCB6_000076 CC1=C2[C@H](OB(O)C[C@@H]2[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D11 compound treatment 1260240.0 53200.0 0.89 1269920.0 76000.0 1.37 1.5979 0.9783 2065682 ICCB6_000077 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](Cc5ccccc5)N1C(=O)Cc6ccc(OC)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D12 compound treatment 1250960.0 43900.0 0.74 1228440.0 34500.0 0.62 0.9596 0.9965 2065683 ICCB6_000078 CC(C)[Si](OCC(O)/C(=C\CO)/C)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D13 compound treatment 1269680.0 62600.0 1.05 1225480.0 31600.0 0.57 1.1434 0.9587 1952278 ICCB6_000079 COC(=O)c1nc(oc1C)C(NC(=O)CCc2cn(CC=C)c3ccccc23)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D14 compound treatment 1242240.0 35200.0 0.59 1224680.0 30800.0 0.55 0.8085 0.9995 2065684 ICCB6_000080 CC(C)[Si](OCC(O)/C=C\CO)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D15 compound treatment 1226440.0 19400.0 0.32 1213400.0 19500.0 0.35 0.4778 0.9993 2065685 ICCB6_000081 CCOCOc1cc(O)c(C(=O)/C=C/c2ccccc2)c(OCOCC)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D16 compound treatment 1258160.0 51100.0 0.86 1231480.0 37600.0 0.68 1.0835 0.9933 2065686 ICCB6_000082 CC(C)[Si](OC[C@@H](O)[C@@]1(C)OC(C)(C)OC1CO)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D17 compound treatment 1179240.0 -27800.0 -0.47 1167200.0 -26700.0 -0.48 -0.6693 -0.9999 1952811 ICCB6_000083 CC(C)(C)[Si](C)(C)Oc1ccc(C#C)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D18 compound treatment 1235760.0 28700.0 0.48 1207960.0 14000.0 0.25 0.5188 0.955 2065687 ICCB6_000084 CC(C)[Si](OC[C@@H](O)[C@H]1OC(C)(C)OC1CO)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D19 compound treatment 1216880.0 9850.0 0.16 1198440.0 4520.0 0.08 0.1741 0.9472 1952780 ICCB6_000085 COc1cccc(c1)c2c(oc3ccccc23)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D20 compound treatment 1209840.0 2810.0 0.05 1209360.0 15400.0 0.28 0.2299 0.815 2065688 ICCB6_000086 CC1(C)OC(CO)[C@H](O1)[C@H](O)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D21 compound treatment 1212320.0 5290.0 0.09 1184560.0 -9360.0 -0.17 -0.0567 -0.2975 1952670 ICCB6_000087 COCCNC(=O)OC[C@H]1CCC[C@@]2(C[C@@H](C[C@@H](CCC(=O)N[C@@H](C)C(=O)OC)O2)OC(=O)NCCc3ccc(F)cc3)O1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D22 compound treatment 1208800.0 1770.0 0.03 1195440.0 1520.0 0.03 0.0403 0.9992 2065689 ICCB6_000088 C/C(=C/CO)/[C@H](O)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D23 mock treatment 1194640.0 -12400.0 -0.21 1181880.0 -12000.0 -0.22 -0.3 -0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 D24 mock treatment 1215840.0 8810.0 0.15 1204360.0 10400.0 0.19 0.2372 0.9927 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E01 compound treatment 1289120.0 82100.0 1.37 1285840.0 91900.0 1.66 2.1424 0.9957 2065690 ICCB6_000089 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccc(Cl)c(Cl)c4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E02 compound treatment 740560.0 -466000.0 -7.81 750160.0 -444000.0 -8.0 -11.1733 -0.9999 2065691 ICCB6_000090 COc1ccc(NC(=O)OC/C=C/c2ccc(CCCCCCO)o2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E03 compound treatment 1303440.0 96400.0 1.61 1267280.0 73400.0 1.32 2.0754 0.9951 2065692 ICCB6_000091 CCOC(=O)C1[C@@H](O[C@@H](CC1=O)c2ccccc2)C3CCCCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E04 compound treatment 1241240.0 34200.0 0.57 1219880.0 26000.0 0.47 0.7355 0.995 2065693 ICCB6_000092 COc1cccc(c1)c2cc(oc2CCCCCCO)[C@@H](O)[C@H](C)C(=O)N3[C@@H](Cc4ccccc4)COC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E05 compound treatment 1302640.0 95600.0 1.6 1282840.0 88900.0 1.6 2.2642 1.0 2065694 ICCB6_000093 COc1ccc(cc1)C(NP(=O)(c2ccccc2)c3ccccc3)[Si](C)(C)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E06 compound treatment 1288200.0 81200.0 1.36 1235960.0 42000.0 0.76 1.4961 0.962 2065695 ICCB6_000094 CC(=O)OC/C=C/c1ccc(CCCCCCO)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E07 compound treatment 1275080.0 68000.0 1.14 1249240.0 55300.0 1.0 1.51 0.9978 2065696 ICCB6_000095 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](C)N1C(=O)Cc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E08 compound treatment 1086720.0 -120000.0 -2.01 909080.0 -285000.0 -5.13 -5.0525 -0.9165 2065697 ICCB6_000096 CCOC(=O)c1cccc(NC(=O)OC/C=C/c2ccc(CCCCCCO)o2)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E09 compound treatment 1272320.0 65300.0 1.09 1248800.0 54900.0 0.99 1.4717 0.9988 2065698 ICCB6_000097 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](CC(C)C)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E10 compound treatment 1138360.0 -68700.0 -1.15 1013120.0 -181000.0 -3.26 -3.116 -0.9021 2065699 ICCB6_000098 CCCCOC(=O)c1ccc(NC(=O)OC/C=C/c2ccc(CCCCCCO)o2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E11 compound treatment 1276680.0 69600.0 1.17 1244480.0 50600.0 0.91 1.4683 0.9926 1952474 ICCB6_000099 OCCCCCNC(CCO)Cc1ccc2ccccc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E12 compound treatment 886840.0 -320000.0 -5.36 890360.0 -304000.0 -5.47 -7.6562 -0.9999 2065700 ICCB6_000100 COC(=O)[C@@H](NC(=O)OC/C=C/c1ccc(CCCCCCO)o1)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E13 compound treatment 1249840.0 42800.0 0.72 1224880.0 31000.0 0.56 0.901 0.9923 1952280 ICCB6_000101 COC(=O)c1nc2oc1CC/C=C/Cn3cc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2C(C)C)c4ccccc34 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E14 compound treatment 982640.0 -224000.0 -3.76 812960.0 -381000.0 -6.86 -7.5087 -0.9597 2065701 ICCB6_000102 COc1cccc(Cl)c1NC(=O)OC/C=C/c2ccc(CCCCCCO)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E15 compound treatment 1012720.0 -194000.0 -3.25 931080.0 -263000.0 -4.74 -5.6479 -0.9832 1952487 ICCB6_000103 Fc1ccc(cc1Br)[C@H]2C3=CCn4n(C3C[C@@]5(C#N)C(=O)C(=C(Cl)C(=O)[C@@]25C#N)Cl)c(=O)n(c6ccccc6)c4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E16 compound treatment 1275120.0 68100.0 1.14 1222080.0 28200.0 0.51 1.1645 0.9336 2065702 ICCB6_000104 C[C@@H]([C@H](O)c1cc(c(CCCCCCO)o1)c2ccccc2)C(=O)N3[C@@H](Cc4ccccc4)COC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E17 compound treatment 1202640.0 -4390.0 -0.07 1138680.0 -55200.0 -1.0 -0.7557 -0.7573 1952813 ICCB6_000105 OCCCC#Cc1cc(O)cc(Cl)c1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E18 compound treatment 1214000.0 6970.0 0.12 1176480.0 -17400.0 -0.31 -0.1397 -0.4169 2065703 ICCB6_000106 COc1cccc(c1)c2cc(oc2CCCCCCO)[C@@H](OC(=O)C)[C@H](C)C(=O)N3[C@@H](Cc4ccccc4)COC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E19 compound treatment 1243120.0 36100.0 0.6 1215000.0 21100.0 0.38 0.6956 0.975 3107406 ICCB6_000107 COC(=O)/C=C/c1cc(OC)c2oc(c(C)c2c1)c3ccccc3.c1ccsc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E20 compound treatment 1209320.0 2290.0 0.04 1190080.0 -3840.0 -0.07 -0.0218 -0.2762 2065704 ICCB6_000108 C[C@@H]([C@H](OC(=O)C)c1cc(c(CCCCCCO)o1)c2ccccc2)C(=O)N3[C@@H](Cc4ccccc4)COC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E21 compound treatment 1214400.0 7370.0 0.12 1190720.0 -3200.0 -0.06 0.0464 0.3411 ICCB6_000109 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E22 compound treatment 1174120.0 -32900.0 -0.55 1140200.0 -53700.0 -0.97 -1.0738 -0.9643 2065705 ICCB6_000110 C[C@@H]([C@H](O)c1cc(c(CCCCCCO)o1)c2cccc(C)c2)C(=O)N3[C@@H](Cc4ccccc4)COC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E23 mock treatment 1221480.0 14400.0 0.24 1196600.0 2680.0 0.05 0.2051 0.8319 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 E24 mock treatment 1230920.0 23900.0 0.4 1212320.0 18400.0 0.33 0.5171 0.9957 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F01 compound treatment 1317360.0 110000.0 1.85 1297480.0 104000.0 1.87 2.6249 1.0 2065706 ICCB6_000111 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccc(OC)cc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F02 compound treatment 1292120.0 85100.0 1.42 1268080.0 74200.0 1.34 1.9517 0.9995 2065707 ICCB6_000112 CC(C)[Si](OC[C@@H](O)C(C=C)C(O)c1ccccc1)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F03 compound treatment 1305840.0 98800.0 1.65 1276640.0 82700.0 1.49 2.2231 0.9987 1009686 ICCB6_000113 O=C(CC(C(=O)c1ccccc1)c2ccccc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F04 compound treatment 1296280.0 89200.0 1.49 1282600.0 88700.0 1.6 2.1859 0.9994 2065708 ICCB6_000114 OC/C=C\C(O)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F05 compound treatment 1313360.0 106000.0 1.78 1312720.0 119000.0 2.14 2.7717 0.9958 2065709 ICCB6_000115 CCCCCCCCNC(=O)CC[C@H]1O[C@H](O[C@H]2O[C@H](CCC(=O)NCCCCCCCC)[C@@H](O)[C@H](O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F06 compound treatment 1284680.0 77600.0 1.3 1266440.0 72500.0 1.31 1.8427 1.0 2065710 ICCB6_000116 CC1=C([C@H](O)C(C)(C)C)[C@H](CO)[C@H]2[C@@H](C1)C(=O)N(Cc3ccccc3)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F07 compound treatment 1255320.0 48300.0 0.81 1258120.0 64200.0 1.16 1.3893 0.9846 2065711 ICCB6_000117 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F08 compound treatment 1276760.0 69700.0 1.17 1272320.0 78400.0 1.41 1.8239 0.9955 2065712 ICCB6_000118 CC1=C([C@H](O)c2ccccc2)[C@H](CO)[C@H]3[C@@H](C1)C(=O)N(Cc4ccccc4)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F09 compound treatment 1273280.0 66200.0 1.11 1243840.0 49900.0 0.9 1.4199 0.9946 2065713 ICCB6_000119 CCOC(=O)CC1[C@@H]2[C@@H](NCc3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](CC(C)C)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F10 compound treatment 1261520.0 54500.0 0.91 1264920.0 71000.0 1.28 1.5493 0.9862 2065714 ICCB6_000120 C[C@@H](O)C1=CC[C@@H]2[C@H]([C@H]1CO)C(=O)N(Cc3ccccc3)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F11 compound treatment 1270880.0 63800.0 1.07 1223840.0 29900.0 0.54 1.1367 0.9498 1952476 ICCB6_000121 OCCCCCN(Cc1ccccc1Br)[C@@H](COCc2c(Br)sc3ccc(Cl)cc23)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F12 compound treatment 1291560.0 84500.0 1.41 1268760.0 74800.0 1.35 1.9537 0.9997 2065715 ICCB6_000122 OC[C@@H]1[C@H]2[C@@H](CC=C1CO)C(=O)N(Cc3ccccc3)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F13 compound treatment 1271320.0 64300.0 1.08 1248400.0 54500.0 0.98 1.4548 0.999 1952282 ICCB6_000123 COC(=O)c1nc2oc1CC/C=C/CNC(=O)O[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NC2C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F14 compound treatment 1265080.0 58000.0 0.97 1239160.0 45200.0 0.82 1.2633 0.9962 2065716 ICCB6_000124 CC1=C(CO)[C@H](CO)[C@H]2[C@@H](C1)C(=O)N(Cc3ccccc3)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F15 compound treatment 1052840.0 -154000.0 -2.58 860440.0 -333000.0 -6.01 -6.0731 -0.9288 1952488 ICCB6_000125 Fc1ccc(cc1Br)[C@H]2C3=CCC4=C(C3CC5=C2C(=O)C(=CC5=O)I)C(=O)C(=CC4=O)I 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F16 compound treatment 1251280.0 44200.0 0.74 1238360.0 44400.0 0.8 1.0898 0.9992 2065717 ICCB6_000126 C/C(=C/CO)/C(O)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F17 compound treatment 1229000.0 22000.0 0.37 1196840.0 2920.0 0.05 0.2972 0.8001 1952814 ICCB6_000127 CC(=O)Cc1c(Cl)cc(cc1I)C(=O)NCCO[Si](C)(C)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F18 compound treatment 1239920.0 32900.0 0.55 1212480.0 18600.0 0.33 0.6256 0.9715 2065718 ICCB6_000128 CC(C)[Si](OCC1OB(O)CC=C1C)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F19 compound treatment 1224640.0 17600.0 0.29 1209280.0 15400.0 0.28 0.4041 0.9995 1952785 ICCB6_000129 CCc1cc(OC)c2oc(c(C(=O)c3ccccc3)c2c1)c4ccc(Oc5ccccc5)c(OC)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F20 compound treatment 1110560.0 -96500.0 -1.61 1061200.0 -133000.0 -2.39 -2.8324 -0.9817 2065719 ICCB6_000130 OB1CC=C(C(O1)c2ccccc2)C(=C)COCc3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F21 compound treatment 1211640.0 4610.0 0.08 1192040.0 -1880.0 -0.03 0.0306 0.3631 3107360 ICCB6_000131 Cc1ccc(cc1)S(=O)(=O)O.Cc1cc(=O)oc2ccccc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F22 compound treatment 1138200.0 -68800.0 -1.15 1078800.0 -115000.0 -2.07 -2.2811 -0.9615 2065720 ICCB6_000132 OC/C=C(\C(O)c1ccccc1)/C(=C)COCc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F23 mock treatment 1187920.0 -19100.0 -0.32 1177520.0 -16400.0 -0.3 -0.4351 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 F24 mock treatment 1239240.0 32200.0 0.54 1220840.0 26900.0 0.49 0.7241 0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G01 compound treatment 1325120.0 118000.0 1.98 1300080.0 106000.0 1.91 2.7498 0.9999 2065721 ICCB6_000133 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4cccs4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G02 compound treatment 1320600.0 114000.0 1.9 1293360.0 99400.0 1.79 2.6107 0.9996 3057351 ICCB6_000134 CC(C)C[C@H](CI)C(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G03 compound treatment 1303880.0 96800.0 1.62 1278600.0 84700.0 1.53 2.2249 0.9995 2065722 ICCB6_000135 Clc1ccc(cc1)C(NP(=O)(c2ccccc2)c3ccccc3)C(=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G04 compound treatment 1317760.0 111000.0 1.85 1313560.0 120000.0 2.16 2.8345 0.9972 3057353 ICCB6_000136 CC(C)(C)OC[C@@H](O)[C@H]1O[C@H](NO)C2OC(C)(C)OC12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G05 compound treatment 1319920.0 113000.0 1.89 1299160.0 105000.0 1.9 2.6766 1.0 2065723 ICCB6_000137 CCCCCCCNCC(=O)NC[C@H]1O[C@H](O[C@H]2O[C@H](CNC(=O)CCNCCCCCC)[C@@H](O)[C@H](O)[C@H]2O)[C@H](O)[C@@H](O)[C@@H]1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G06 compound treatment 1286560.0 79500.0 1.33 1279760.0 85800.0 1.55 2.0347 0.9972 2065724 ICCB6_000138 CC(C)[Si](C)(C)Oc1cccc2C(C=C)N(C=Cc12)C(=O)c3ccccc3Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G07 compound treatment 1266000.0 59000.0 0.99 1264960.0 71000.0 1.28 1.6028 0.9917 2065725 ICCB6_000139 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G08 compound treatment 1279880.0 72800.0 1.22 1262520.0 68600.0 1.24 1.736 1.0 2065726 ICCB6_000140 CC(C)(C)[Si](C)(C)OCC1=CC(C#C)N(C=C1)C(=O)c2ccccc2Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G09 compound treatment 1278320.0 71300.0 1.19 1247760.0 53800.0 0.97 1.5295 0.9947 2065727 ICCB6_000141 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](CC(C)C)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G10 compound treatment 1281680.0 74600.0 1.25 1268120.0 74200.0 1.34 1.8286 0.9994 3057357 ICCB6_000142 OC(=O)c1[se]c2ccccc2c1Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G11 compound treatment 1237680.0 30600.0 0.51 1220600.0 26700.0 0.48 0.7026 0.9995 1952478 ICCB6_000143 OCCCCCN(Cc1ccccc1Br)[C@@H](COCc2ccc3ccccc3c2Br)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G12 compound treatment 1181880.0 -25200.0 -0.42 1144680.0 -49200.0 -0.89 -0.9249 -0.9419 3057359 ICCB6_000144 CC(C)(C)[Si](C)(C)OCC1=CC(C=C)N(C=C1)C(=O)c2[se]c3ccccc3c2Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G13 compound treatment 1267640.0 60600.0 1.01 1245880.0 52000.0 0.94 1.3792 0.9992 1952284 ICCB6_000145 COC(=O)c1nc2oc1CC/C=C/CNC(=O)O[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]2C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G14 compound treatment 1265640.0 58600.0 0.98 1245280.0 51400.0 0.93 1.3479 0.9996 2065728 ICCB6_000146 CCCCCC1C=C(CO[Si](C)(C)C(C)(C)C)C=CN1C(=O)c2ccccc2Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G15 compound treatment 1256080.0 49000.0 0.82 1221320.0 27400.0 0.49 0.9295 0.9704 2065729 ICCB6_000147 CCOCOc1cc(OCOCC)c2C(=O)CC(Oc2c1)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G16 compound treatment 1264520.0 57500.0 0.96 1223000.0 29100.0 0.52 1.0508 0.9592 2065730 ICCB6_000148 CC(C)(C)[Si](C)(C)Oc1cccc2C(C=C)N(C=Cc12)C(=O)c3ccccc3Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G17 compound treatment 1238680.0 31600.0 0.53 1221760.0 27800.0 0.5 0.7292 0.9996 1952760 ICCB6_000149 CC(C)(C)[Si](C)(C)OCCNC(=O)c1cc(c2cc(F)cc(F)c2)c3oc4c(C(=O)OC4(c5ccccc5)c6ccccc6)c3c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G18 compound treatment 1255960.0 48900.0 0.82 1230160.0 36200.0 0.65 1.0407 0.9937 2065731 ICCB6_000150 CC(=O)N[C@@H](CI)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G19 compound treatment 1229280.0 22200.0 0.37 1211280.0 17400.0 0.31 0.4844 0.9962 1952788 ICCB6_000151 CCc1cc(OC)c2oc(c(C(=O)c3ccc(OC)cc3)c2c1)c4ccc(Oc5ccccc5)c(OC)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G20 compound treatment 1207800.0 769.0 0.01 1193920.0 0.0 0.0 0.0091 0.7071 2065732 ICCB6_000152 COc1cc2CCN(Cc3ccccc3Br)C(C=C)c2cc1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G21 compound treatment 1239800.0 32800.0 0.55 1202640.0 8720.0 0.16 0.4989 0.8745 1952728 ICCB6_000153 Cc1ccc2oc(=O)cc(c3cccs3)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G22 compound treatment 1238920.0 31900.0 0.53 1211880.0 18000.0 0.32 0.6062 0.9713 2065733 ICCB6_000154 CN1C(=O)C2C(C1=O)C3(C4C(C5C=C(CCCO[Si](C)(C)C(C)(C)C)CC2N53)C(=O)N(C)C4=O)C(=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G23 mock treatment 1223560.0 16500.0 0.28 1204680.0 10800.0 0.19 0.3327 0.9849 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 G24 mock treatment 1218240.0 11200.0 0.19 1205360.0 11400.0 0.21 0.2784 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H01 compound treatment 1317480.0 110000.0 1.85 1302680.0 109000.0 1.96 2.6926 0.9996 2065734 ICCB6_000155 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccccc4Cl)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H02 compound treatment 1299280.0 92200.0 1.54 1267480.0 73600.0 1.33 2.0288 0.9971 2065735 ICCB6_000156 CC(=C)C1=CCB(O)OC1c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H03 compound treatment 1285880.0 78800.0 1.32 1286600.0 92700.0 1.67 2.1138 0.9932 2065736 ICCB6_000157 CC(C(NP(=O)(c1ccccc1)c2ccccc2)c3ccccc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H04 compound treatment 1285040.0 78000.0 1.31 1257520.0 63600.0 1.15 1.7334 0.9979 2065737 ICCB6_000158 CN1C(=O)[C@@H]2CC(=C([C@H](O)c3ccccc3)[C@H](CO)[C@@H]2C1=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H05 compound treatment 1286400.0 79400.0 1.33 1268200.0 74300.0 1.34 1.8855 1.0 2065738 ICCB6_000159 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)CN1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H06 compound treatment 1316440.0 109000.0 1.83 1277160.0 83200.0 1.5 2.3551 0.9951 2065739 ICCB6_000160 CC(=C)/C(=C/CO)/C(O)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H07 compound treatment 1300400.0 93400.0 1.56 1239000.0 45100.0 0.81 1.6792 0.9535 2065740 ICCB6_000161 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](C)N1C(=O)Cc4ccc(OC)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H08 compound treatment 1279480.0 72400.0 1.21 1258800.0 64900.0 1.17 1.6839 0.9998 2065741 ICCB6_000162 CC1=NC(C)(C)[C@@H]2CCC(=C)C1C2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H09 compound treatment 1277280.0 70200.0 1.18 1244760.0 50800.0 0.92 1.479 0.9924 2065742 ICCB6_000163 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](CC(C)C)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H10 compound treatment 1285600.0 78600.0 1.31 1257720.0 63800.0 1.15 1.7425 0.9978 2065743 ICCB6_000164 C[C@H]1NC(C)(C)C2CCC(=C)[C@H]1C2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H11 compound treatment 1252000.0 45000.0 0.75 1267560.0 73600.0 1.33 1.4703 0.9639 1952534 ICCB6_000165 C[C@H](N)C(Oc1ccccc1Br)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H12 compound treatment 1260720.0 53700.0 0.9 1264160.0 70200.0 1.27 1.5302 0.9859 2065744 ICCB6_000166 C[C@@H]1[C@@H]2CC(CCC2=C)C(C)(C)N1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H13 compound treatment 1262280.0 55200.0 0.92 1223040.0 29100.0 0.52 1.0248 0.964 1952286 ICCB6_000167 COC(=O)c1nc(oc1CCC=C)C(NC(=O)[C@H](Cc2cn(CC=C)cn2)NC(=O)OCc3ccccc3)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H14 compound treatment 1273880.0 66800.0 1.12 1241120.0 47200.0 0.85 1.3924 0.9908 2065745 ICCB6_000168 CC(C)C[C@H]1NC(C)(C)C2CCC(=C)[C@H]1C2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H15 compound treatment 1239120.0 32100.0 0.54 1225880.0 32000.0 0.58 0.7869 0.9994 1952677 ICCB6_000169 CCCCCCC#Cc1c(C(CC(=O)C)c2ccccc2)c(=O)oc3ccccc13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H16 compound treatment 1250240.0 43200.0 0.72 1223080.0 29200.0 0.53 0.8828 0.9877 2065746 ICCB6_000170 CC(C)C[C@@H]1[C@@H]2CC(CCC2=C)C(C)(C)N1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H17 compound treatment 1221280.0 14200.0 0.24 1205920.0 12000.0 0.22 0.3215 0.9988 1952821 ICCB6_000171 CC(C)(C)[Si](C)(C)COCNC(=O)C1CC2C3C(OC2C(Cl)C1)C4(CCCC4)OC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H18 compound treatment 1239400.0 32400.0 0.54 1231560.0 37600.0 0.68 0.8626 0.9938 2065747 ICCB6_000172 COc1cc(C[C@H]2NC(C)(C)C3CCC(=C)[C@H]2C3)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H19 compound treatment 1197720.0 -9310.0 -0.16 1205800.0 11900.0 0.21 0.0412 0.1555 1952600 ICCB6_000173 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCc3ccccc3)O2)O1)OC(=O)NCc4cccc5ccccc45 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H20 compound treatment 1204880.0 -2150.0 -0.04 1180480.0 -13400.0 -0.24 -0.1967 -0.8034 2065748 ICCB6_000174 COc1cc(C[C@@H]2[C@@H]3CC(CCC3=C)C(C)(C)N2C)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H21 compound treatment 1217840.0 10800.0 0.18 1196120.0 2200.0 0.04 0.1559 0.8421 1952730 ICCB6_000175 O=c1cc(Cc2ccccc2)c3ccccc3o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H22 compound treatment 1191960.0 -15100.0 -0.25 1158720.0 -35200.0 -0.63 -0.6268 -0.9184 2065749 ICCB6_000176 CC1(C)N=C(/C=C/2\C(=O)Nc3ccccc23)[C@@H]4CC1CCC4=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H23 mock treatment 1201640.0 -5390.0 -0.09 1185680.0 -8240.0 -0.15 -0.1688 -0.9715 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 H24 mock treatment 1208480.0 1450.0 0.02 1191360.0 -2560.0 -0.05 -0.0155 -0.2969 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I01 compound treatment 1314520.0 107000.0 1.8 1286080.0 92200.0 1.66 2.4461 0.9992 2065750 ICCB6_000177 COC(=O)[C@@H]1[C@H](N([C@H](c2ccccc2)[C@@]13C(=O)N(Cc4ccccc4)c5ccccc53)c6ccccc6)C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I02 compound treatment 1269320.0 62300.0 1.04 1248120.0 54200.0 0.98 1.4276 0.9995 2065751 ICCB6_000178 CC(C)(C)[Si](C)(C)OCCCC1=CC2C3C(C(=O)N(Cc4ccccc4)C3=O)C5(C6C(C(C1)N25)C(=O)N(Cc7ccccc7)C6=O)C(=O)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I03 compound treatment 1308520.0 101000.0 1.7 1287160.0 93200.0 1.68 2.3888 1.0 2065752 ICCB6_000179 CCOC(=O)[C@H]1N(C(C(=C1C(=O)OC)C(=O)OC)c2ccc(Cl)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I04 compound treatment 1310640.0 104000.0 1.73 1288320.0 94400.0 1.7 2.4287 1.0 2065753 ICCB6_000180 COc1cc(CN[C@@H](C)[C@H](Oc2ccccc2Br)c3ccccc3)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I05 compound treatment 1319120.0 112000.0 1.88 1306280.0 112000.0 2.02 2.7578 0.9993 2065754 ICCB6_000181 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)CN1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I06 compound treatment 1312040.0 105000.0 1.76 1287040.0 93100.0 1.68 2.4289 0.9997 2065755 ICCB6_000182 COc1cc(CN[C@H]([C@H](O)c2ccccc2)c3ccccc3)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I07 compound treatment 1281440.0 74400.0 1.25 1227720.0 33800.0 0.61 1.3111 0.9459 2065756 ICCB6_000183 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I08 compound treatment 1289360.0 82300.0 1.38 1287560.0 93600.0 1.69 2.1672 0.9949 2065757 ICCB6_000184 COc1cc(CN(Cc2ccccc2Br)[C@H]([C@H](O)c3ccccc3)c4ccccc4)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I09 compound treatment 1282640.0 75600.0 1.27 1266440.0 72500.0 1.31 1.8186 0.9999 2065758 ICCB6_000185 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](CC(C)C)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I10 compound treatment 1289720.0 82700.0 1.38 1270120.0 76200.0 1.37 1.9493 1.0 2065759 ICCB6_000186 COc1cc(CN(Cc2ccccc2Br)[C@H](C)C(Oc3ccccc3Br)c4ccccc4)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I11 compound treatment 1262800.0 55800.0 0.93 1244080.0 50200.0 0.9 1.299 0.9999 1952544 ICCB6_000187 O=C1Nc2ccccc2[C@@]31[C@@H](C#N)C4N([C@H]3c5ccccc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I12 compound treatment 1230040.0 23000.0 0.39 1227480.0 33600.0 0.6 0.6998 0.9763 2065760 ICCB6_000188 COc1cc(CN(Cc2ccccc2Br)[C@H](C(Oc3ccccc3Br)c4ccccc4)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I13 compound treatment 1263320.0 56300.0 0.94 1244120.0 50200.0 0.9 1.3056 0.9998 1952288 ICCB6_000189 COC(=O)c1nc2oc1CC/C=C/Cn3cnc(C[C@H](NC(=O)OCc4ccccc4)C(=O)NC2C(C)C)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I14 compound treatment 1263720.0 56700.0 0.95 1246920.0 53000.0 0.95 1.346 1.0 2065761 ICCB6_000190 C[C@@H](C(Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])c2ccccc2)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I15 compound treatment 1262480.0 55400.0 0.93 1234280.0 40400.0 0.73 1.1703 0.9927 1952679 ICCB6_000191 Clc1ccc2oc(=O)cc(Sc3ccccc3)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I16 compound treatment 1267440.0 60400.0 1.01 1236400.0 42500.0 0.77 1.256 0.9906 2065762 ICCB6_000192 C[C@H](C(Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])c2ccccc2)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I17 compound treatment 1223000.0 16000.0 0.27 1205640.0 11700.0 0.21 0.3383 0.9932 1952823 ICCB6_000193 C#Cc1ccccc1Oc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I18 compound treatment 1257840.0 50800.0 0.85 1234760.0 40800.0 0.74 1.1215 0.9974 2065763 ICCB6_000194 C[C@H](C(Oc1ccc(cc1)[N+](=O)[O-])c2ccccc2)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I19 compound treatment 1206320.0 -711.0 -0.01 1158760.0 -35200.0 -0.63 -0.4564 -0.7203 1952601 ICCB6_000195 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCCOc3ccccc3)O2)O1)OC(=O)NCc4cccc5ccccc45 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I20 compound treatment 1227320.0 20300.0 0.34 1202680.0 8760.0 0.16 0.3517 0.9393 2065764 ICCB6_000196 C[C@H]([C@@H](Oc1ccccc1Br)c2ccccc2)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I21 compound treatment 1219400.0 12400.0 0.21 1203560.0 9640.0 0.17 0.2692 0.9962 1952746 ICCB6_000197 Cc1ccc(cc1)c2cc(=O)oc3ccccc23 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I22 compound treatment 1216920.0 9890.0 0.17 1203080.0 9160.0 0.17 0.2337 1.0 2065765 ICCB6_000198 C[C@@H]([C@@H](Oc1ccccc1Br)c2ccccc2)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I23 mock treatment 1210280.0 3250.0 0.05 1198320.0 4400.0 0.08 0.0945 0.9831 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 I24 mock treatment 1197920.0 -9110.0 -0.15 1184040.0 -9880.0 -0.18 -0.2337 -0.997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J01 compound treatment 1168560.0 -38500.0 -0.64 1116440.0 -77500.0 -1.4 -1.4423 -0.9382 2065766 ICCB6_000199 COC(=O)C1=CN([C@H](c2ccccc2)[C@]31C(=O)N(Cc4ccccc4)c5ccccc53)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J02 compound treatment 1301800.0 94800.0 1.59 1277400.0 83500.0 1.5 2.185 0.9996 2065767 ICCB6_000200 CC1(C)N[C@H](CC2C(=O)Nc3ccccc23)[C@@H]4CC1CCC4=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J03 compound treatment 1309360.0 102000.0 1.71 1289080.0 95200.0 1.71 2.4232 1.0 2065768 ICCB6_000201 CCOC(=O)[C@H]1N(C(C(=C1C(=O)OC)C(=O)OC)c2ccc(Br)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J04 compound treatment 1297720.0 90700.0 1.52 1267400.0 73500.0 1.32 2.0093 0.9977 2065769 ICCB6_000202 CN1[C@H](CC2C(=O)Nc3ccccc23)[C@@H]4CC(CCC4=C)C1(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J05 compound treatment 1288160.0 81100.0 1.36 1261560.0 67600.0 1.22 1.8217 0.9985 2065770 ICCB6_000203 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)CN1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J06 compound treatment 1301560.0 94500.0 1.58 1280680.0 86800.0 1.56 2.2239 1.0 2065771 ICCB6_000204 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)OCC=C)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J07 compound treatment 1281440.0 74400.0 1.25 1249720.0 55800.0 1.01 1.5914 0.9944 2065772 ICCB6_000205 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C(C)C)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J08 compound treatment 1272080.0 65000.0 1.09 1242040.0 48100.0 0.87 1.3828 0.9936 2065773 ICCB6_000206 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)OCC=C)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J09 compound treatment 1285360.0 78300.0 1.31 1246800.0 52900.0 0.95 1.6006 0.9877 2065774 ICCB6_000207 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](CC(C)C)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J10 compound treatment 1286600.0 79600.0 1.33 1262440.0 68500.0 1.23 1.8145 0.9993 2065775 ICCB6_000208 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)OCC=C)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J11 compound treatment 1275240.0 68200.0 1.14 1259520.0 65600.0 1.18 1.6429 0.9998 2065776 ICCB6_000209 Cc1ccc(SC2(CC(=O)N(Cc3ccccc3)C2c4ccccc4I)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J12 compound treatment 1275440.0 68400.0 1.14 1221720.0 27800.0 0.5 1.1637 0.9313 2065777 ICCB6_000210 OCCOc1cccc(c1)[C@@H]2N3[C@H]([C@H](C(=O)OCC=C)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J13 compound treatment 1188200.0 -18800.0 -0.32 1150520.0 -43400.0 -0.78 -0.7758 -0.9202 1952295 ICCB6_000211 COC(=O)c1nc(oc1CC(=O)CCl)C(NC(=O)NC(=O)OC(C)(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J14 compound treatment 850240.0 -357000.0 -5.97 905840.0 -288000.0 -5.19 -7.8921 -0.9976 2065778 ICCB6_000212 OCc1ccc(o1)[C@@H]2N3[C@H]([C@H](C(=O)OCC=C)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J15 compound treatment 1260920.0 53900.0 0.9 1226760.0 32800.0 0.59 1.0561 0.9791 1952690 ICCB6_000213 COC(=O)CC(C(=O)OC)c1ccccc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J16 compound treatment 1253040.0 46000.0 0.77 1228240.0 34300.0 0.62 0.9817 0.9941 2065779 ICCB6_000214 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCC(C(=O)OC)C(=O)OC)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J17 compound treatment 1255120.0 48100.0 0.8 1237400.0 43500.0 0.78 1.123 0.9999 1952825 ICCB6_000215 CCCC(C)(O)C#Cc1cc(cc(C(=O)NCCO[Si](C)(C)C(C)(C)C)c1OC(=O)C)c2cc(F)cc(F)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J18 compound treatment 1215240.0 8210.0 0.14 1162320.0 -31600.0 -0.57 -0.3055 -0.5215 2065780 ICCB6_000216 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J19 compound treatment 1193200.0 -13800.0 -0.23 1146160.0 -47800.0 -0.86 -0.7721 -0.8665 1952605 ICCB6_000217 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCCC(C)C)O2)O1)OC(=O)NCc3cccc4ccccc34 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J20 compound treatment 1214120.0 7090.0 0.12 1187680.0 -6240.0 -0.11 0.0044 0.0268 2065781 ICCB6_000218 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J21 compound treatment 1195360.0 -11700.0 -0.2 1173600.0 -20300.0 -0.37 -0.397 -0.9567 3005760 ICCB6_000219 CCOP(=O)(O)OCC.Cc1cc(=O)oc2ccc(Cl)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J22 compound treatment 1196000.0 -11000.0 -0.18 1179680.0 -14200.0 -0.26 -0.312 -0.987 2065782 ICCB6_000220 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCNC(=O)N)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J23 mock treatment 1204640.0 -2390.0 -0.04 1193200.0 -720.0 -0.01 -0.0375 -0.8907 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 J24 mock treatment 1219840.0 12800.0 0.21 1199240.0 5320.0 0.1 0.2193 0.9342 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K01 compound treatment 1319320.0 112000.0 1.88 1276560.0 82600.0 1.49 2.3816 0.9934 2065783 ICCB6_000221 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccccc4)C(=O)N(C)c5ccccc52 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K02 compound treatment 1308400.0 101000.0 1.7 1293320.0 99400.0 1.79 2.4659 0.9996 2065784 ICCB6_000222 CC(Oc1ccccc1Br)[C@H](N(C)C)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K03 compound treatment 1287280.0 80200.0 1.34 1251200.0 57300.0 1.03 1.6793 0.9915 2065785 ICCB6_000223 COC(=O)C(C(c1ccc(OC)cc1)[Si](C)(C)c2ccccc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K04 compound treatment 1296440.0 89400.0 1.5 1281240.0 87300.0 1.57 2.1704 0.9997 2065786 ICCB6_000224 C[C@H](C(Oc1ccccc1[N+](=O)[O-])c2ccccc2)N(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K05 compound treatment 1277360.0 70300.0 1.18 1268840.0 74900.0 1.35 1.7867 0.9977 2065787 ICCB6_000225 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)CN1C(=O)Cc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K06 compound treatment 1280480.0 73400.0 1.23 1278680.0 84800.0 1.53 1.949 0.9942 2065788 ICCB6_000226 COc1cc(/C=C/C=O)ccc1O[Si](C(C)C)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K07 compound treatment 1275080.0 68000.0 1.14 1260520.0 66600.0 1.2 1.6537 0.9997 2065789 ICCB6_000227 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](C(C)C)N1C(=O)CCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K08 compound treatment 1074640.0 -132000.0 -2.22 1034240.0 -160000.0 -2.88 -3.6009 -0.9917 2065790 ICCB6_000228 COc1cc(/C=C/CN[C@H](C)[C@@H](O)c2ccccc2)ccc1O[Si](C(C)C)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K09 compound treatment 1268240.0 61200.0 1.02 1253880.0 60000.0 1.08 1.4882 0.9996 2065791 ICCB6_000229 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](CC(C)C)N1C(=O)Cc4ccc(OC)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K10 compound treatment 1281640.0 74600.0 1.25 1260960.0 67000.0 1.21 1.7369 0.9999 2065792 ICCB6_000230 CC(C)[Si](OCC1CCC=CC1)(C(C)C)C(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K11 compound treatment 959680.0 -247000.0 -4.14 917200.0 -277000.0 -4.99 -6.4524 -0.9957 1034979 ICCB6_000231 c1c(cn2ccccc12)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K12 compound treatment 1272040.0 65000.0 1.09 1253400.0 59500.0 1.07 1.527 1.0 2065793 ICCB6_000232 CC1(C)COC(=O)C1OC(=O)C2CC3CCC2C=C3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K13 compound treatment 1260800.0 53800.0 0.9 1249400.0 55500.0 1.0 1.3431 0.9986 1952379 ICCB6_000233 CC(C)[Si](OCc1ccc(C=O)o1)(C(C)C)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K14 compound treatment 1263360.0 56300.0 0.94 1243160.0 49200.0 0.89 1.2939 0.9995 2065794 ICCB6_000234 OCC1CC2CCC1C=C2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K15 compound treatment 805280.0 -402000.0 -6.72 721360.0 -473000.0 -8.51 -10.7744 -0.9932 1952707 ICCB6_000235 CCCCSc1cc(=O)oc2cc(OC)ccc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K16 compound treatment 718440.0 -489000.0 -8.18 602720.0 -591000.0 -10.65 -13.3135 -0.9915 2065795 ICCB6_000236 Ic1ccc2NC(=O)/C(=C/C(=O)OCC=C)/c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K17 compound treatment 1160600.0 -46400.0 -0.78 1123000.0 -70900.0 -1.28 -1.453 -0.9716 1952828 ICCB6_000237 CCc1cc(OC)c(O)c(C#CC(O)c2ccccc2)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K18 compound treatment 1250920.0 43900.0 0.73 1215800.0 21900.0 0.39 0.7981 0.9574 2065796 ICCB6_000238 C=CCOC(=O)[C@H]1[C@H]2N([C@@H](c3cccnc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K19 compound treatment 1249000.0 42000.0 0.7 1232320.0 38400.0 0.69 0.9858 1.0 1952608 ICCB6_000239 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCCc3ccccc3OC)O2)O1)OC(=O)NCc4cccc5ccccc45 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K20 compound treatment 1106120.0 -101000.0 -1.69 1025520.0 -168000.0 -3.03 -3.3395 -0.9617 2065797 ICCB6_000240 C=CCOC(=O)[C@H]1[C@H]2N([C@@H](c3ccco3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K21 compound treatment 1229000.0 22000.0 0.37 1207720.0 13800.0 0.25 0.4358 0.9819 3005761 ICCB6_000241 Cc1ccc(cc1)S(=O)(=O)O.Cc1cc(=O)oc2ccc(Cl)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K22 compound treatment 959040.0 -248000.0 -4.15 691120.0 -503000.0 -9.06 -9.3402 -0.9374 2065798 ICCB6_000242 Ic1ccc2NC(=O)/C(=C/C#N)/c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K23 mock treatment 1214320.0 7290.0 0.12 1189280.0 -4640.0 -0.08 0.0271 0.1835 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 K24 mock treatment 1198920.0 -8110.0 -0.14 1172200.0 -21700.0 -0.39 -0.3727 -0.8998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L01 compound treatment 1299640.0 92600.0 1.55 1271920.0 78000.0 1.41 2.0896 0.9988 2065799 ICCB6_000243 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccccc4)C(=O)N(C(=O)C)c5ccccc52 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L02 compound treatment 1289720.0 82700.0 1.38 1269680.0 75800.0 1.36 1.9437 1.0 2065800 ICCB6_000244 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#Cc6ccccc6F)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L03 compound treatment 1270840.0 63800.0 1.07 1257880.0 64000.0 1.15 1.5699 0.9993 2065801 ICCB6_000245 COC(=O)C(C(c1ccco1)[Si](C)(C)c2ccccc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L04 compound treatment 1279800.0 72800.0 1.22 1254280.0 60400.0 1.09 1.6301 0.9984 2065802 ICCB6_000246 CCCCC[C@H](O)C#Cc1ccc2NC(=O)[C@@]3([C@H](C4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N(C)OC)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L05 compound treatment 1296880.0 89800.0 1.5 1272320.0 78400.0 1.41 2.062 0.9995 2065803 ICCB6_000247 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)CN1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L06 compound treatment 1245520.0 38500.0 0.64 1237760.0 43800.0 0.79 1.014 0.9949 2065804 ICCB6_000248 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCN(C)[C@H](C)Cc6ccccc6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L07 compound treatment 1253040.0 46000.0 0.77 1249080.0 55200.0 0.99 1.2472 0.992 2065805 ICCB6_000249 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C(C)C)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L08 compound treatment 1261720.0 54700.0 0.92 1243680.0 49800.0 0.9 1.2811 0.9999 2065806 ICCB6_000250 OCCOc1ccc(cc1)C2N3[C@@H]([C@@H](C(=O)OCC=C)[C@]24C(=O)Nc5ccc(Br)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L09 compound treatment 1285000.0 78000.0 1.3 1251400.0 57500.0 1.04 1.6549 0.9935 2065807 ICCB6_000251 CCOC(=O)CC1[C@@H]2[C@@H](NCc3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](Cc5ccccc5)N1C(=O)CCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L10 compound treatment 1256640.0 49600.0 0.83 1227000.0 33100.0 0.6 1.0085 0.9868 2065808 ICCB6_000252 CON(C)C(=O)[C@H]1[C@H]2N(C(c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(I)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L11 compound treatment 1257640.0 50600.0 0.85 1249840.0 55900.0 1.01 1.3113 0.9963 2065809 ICCB6_000253 COC(=O)Cc1cn[nH]c1C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L12 compound treatment 1251280.0 44200.0 0.74 1250120.0 56200.0 1.01 1.2396 0.9882 2065810 ICCB6_000254 CCOC(=O)[C@H]1[C@H]2N(C(c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(Br)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L13 compound treatment 1181320.0 -25700.0 -0.43 1166680.0 -27200.0 -0.49 -0.6513 -0.9978 1952411 ICCB6_000255 CC(C)[Si](OCc1ccc(o1)[C@@H](O)[C@H](C)C(=O)N2[C@@H](C)[C@H](OC2=O)c3ccccc3)(C(C)C)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L14 compound treatment 1237880.0 30800.0 0.52 1237240.0 43300.0 0.78 0.9169 0.9799 2065811 ICCB6_000256 OCCOc1ccc(cc1)C2N3[C@H]([C@H](C(=O)OCC=C)[C@@]24C(=O)Nc5ccc(Br)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L15 compound treatment 1245360.0 38300.0 0.64 1218320.0 24400.0 0.44 0.7644 0.983 1952793 ICCB6_000257 FC(F)(F)c1ccc(cc1)C(=O)Oc2ccccc2C#Cc3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L16 compound treatment 1229440.0 22400.0 0.38 1201800.0 7880.0 0.14 0.3656 0.9117 2065812 ICCB6_000258 CON(C)C(=O)[C@H]1C2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L17 compound treatment 1238440.0 31400.0 0.53 1216280.0 22400.0 0.4 0.6565 0.9914 1952829 ICCB6_000259 O=C(/C(=C\c1ccccc1)/c2cccc(c2)S(=O)=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L18 compound treatment 1250240.0 43200.0 0.72 1229200.0 35300.0 0.64 0.9608 0.9979 2065813 ICCB6_000260 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)OCC=C)[C@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L19 compound treatment 1232600.0 25600.0 0.43 1214840.0 20900.0 0.38 0.5691 0.998 1952582 ICCB6_000261 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)CC[C@@H]2C[C@H](C[C@@]3(CCC[C@H](COC(=O)NCCOC)O3)O2)OC(=O)NCc4cccc5ccccc45 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L20 compound treatment 1206800.0 -231.0 0.0 1207360.0 13400.0 0.24 0.1685 0.6957 2065814 ICCB6_000262 CON(C)C(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccc(Br)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L21 compound treatment 1217400.0 10400.0 0.17 1190440.0 -3480.0 -0.06 0.0784 0.4247 1952748 ICCB6_000263 O=Cc1cccc(c1)c2cc(=O)oc3ccccc23 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L22 compound treatment 1174240.0 -32800.0 -0.55 1164480.0 -29400.0 -0.53 -0.7631 -0.9999 2065815 ICCB6_000264 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCC6CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L23 mock treatment 1199400.0 -7630.0 -0.13 1187000.0 -6920.0 -0.12 -0.1785 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 L24 mock treatment 1202800.0 -4230.0 -0.07 1179680.0 -14200.0 -0.26 -0.2315 -0.8697 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M01 compound treatment 1293840.0 86800.0 1.45 1272720.0 78800.0 1.42 2.0311 0.9999 2065816 ICCB6_000265 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccccc3)c4ccccc4)C(=O)N(C(=O)C)c5ccc(Cl)cc52 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M02 compound treatment 1289440.0 82400.0 1.38 1269160.0 75200.0 1.36 1.9337 1.0 2065817 ICCB6_000266 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C#N)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M03 compound treatment 1311960.0 105000.0 1.76 1296760.0 103000.0 1.85 2.5518 0.9996 2065818 ICCB6_000267 COc1ccc(cc1)C(CC(=O)c2ccccc2)[Si](C)(C)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M04 compound treatment 949520.0 -258000.0 -4.31 902480.0 -291000.0 -5.25 -6.7601 -0.9952 2065819 ICCB6_000268 OCc1ccc(o1)[C@@H]2N3[C@H]([C@H](C#N)[C@@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M05 compound treatment 1275200.0 68200.0 1.14 1247160.0 53200.0 0.96 1.4849 0.9963 2065820 ICCB6_000269 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)CN1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M06 compound treatment 1000280.0 -207000.0 -3.46 1048880.0 -145000.0 -2.61 -4.2943 -0.9904 2065821 ICCB6_000270 COC(=O)/C=C\1/C(=O)Nc2ccc(I)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M07 compound treatment 1288880.0 81800.0 1.37 1264760.0 70800.0 1.28 1.871 0.9994 2065822 ICCB6_000271 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C(C)C)N1C(=O)Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M08 compound treatment 1236840.0 29800.0 0.5 1215400.0 21500.0 0.39 0.6264 0.9921 2065823 ICCB6_000272 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCC4)[C@]25C(=O)Nc6ccc(I)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M09 compound treatment 1279880.0 72800.0 1.22 1252200.0 58300.0 1.05 1.6045 0.9972 2065824 ICCB6_000273 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](Cc4ccccc4)N1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M10 compound treatment 1239800.0 32800.0 0.55 1226600.0 32700.0 0.59 0.8041 0.9994 2065825 ICCB6_000274 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCc4ccccc4)[C@]25C(=O)Nc6ccc(I)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M11 compound treatment 1272320.0 65300.0 1.09 1286560.0 92600.0 1.67 1.9528 0.9789 2065826 ICCB6_000275 CC(C(=O)O)c1ccccc1C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M12 compound treatment 1219520.0 12500.0 0.21 1216720.0 22800.0 0.41 0.4383 0.9509 2065827 ICCB6_000276 OCCNC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccc(I)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M13 compound treatment 1207600.0 569.0 0.01 1203840.0 9920.0 0.18 0.1331 0.7437 1952416 ICCB6_000277 Clc1c(Cl)c(Cl)c(OCc2ccccc2)c(Cl)c1Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M14 compound treatment 1228400.0 21400.0 0.36 1212280.0 18400.0 0.33 0.4868 0.9992 2065828 ICCB6_000278 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M15 compound treatment 1226320.0 19300.0 0.32 1203600.0 9680.0 0.17 0.3516 0.9582 1952795 ICCB6_000279 COC(=O)/C=C/c1cc(OC)cc(C#Cc2ccc(Oc3ccccc3)c(OC)c2)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M16 compound treatment 1221520.0 14500.0 0.24 1197040.0 3120.0 0.06 0.2112 0.8485 2065829 ICCB6_000280 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)C(C(OC3=O)c5ccccc5)c6ccccc6)C(=O)N(C)OC)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M17 compound treatment 1234560.0 27500.0 0.46 1216520.0 22600.0 0.41 0.6137 0.9981 1952832 ICCB6_000281 CCc1cc(OC)c(O)c(C#CC(C)(O)C=C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M18 compound treatment 1215480.0 8450.0 0.14 1194400.0 480.0 0.01 0.1061 0.749 3176523 ICCB6_000282 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)N(C(=O)OCC(C)C)c5ccc(C#CC6(O)CCCCCC6)cc54)C(C(OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M19 compound treatment 1200640.0 -6390.0 -0.11 1191880.0 -2040.0 -0.04 -0.1016 -0.8985 1952627 ICCB6_000283 CCOC(=O)[C@H](CC(C)C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCCC(C)C)O2)O1)OC(=O)NCc3ccc4OCOc4c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M20 compound treatment 1208240.0 1210.0 0.02 1194760.0 840.0 0.02 0.025 0.9898 3056713 ICCB6_000284 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)N(C(=O)N[C@@H](C(C)C)C(=O)OC)c5ccc(C#CC6(O)CCCCCC6)cc54)C(C(OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M21 compound treatment 1195920.0 -11100.0 -0.19 1185000.0 -8920.0 -0.16 -0.2451 -0.9974 1107217 ICCB6_000285 Cc1cccnc1I 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M22 compound treatment 1175600.0 -31400.0 -0.53 1171640.0 -22300.0 -0.4 -0.6558 -0.9911 3176524 ICCB6_000286 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)N(C(=O)N[C@H](C)c5ccccc5)c6ccc(C#CC7(O)CCCCCC7)cc64)C(C(OC2=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M23 mock treatment 1208640.0 1610.0 0.03 1193120.0 -800.0 -0.01 0.0088 0.2896 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 M24 mock treatment 1219040.0 12000.0 0.2 1211960.0 18000.0 0.33 0.3719 0.9733 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N01 compound treatment 1305520.0 98500.0 1.65 1281080.0 87200.0 1.57 2.2759 0.9997 2065830 ICCB6_000287 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3ccc(Cl)cc3)c4ccccc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N02 compound treatment 1263680.0 56600.0 0.95 1245320.0 51400.0 0.93 1.3252 0.9999 2065831 ICCB6_000288 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCN(C)Cc6ccccc6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N03 compound treatment 1253360.0 46300.0 0.78 1253560.0 59600.0 1.07 1.308 0.9872 2065832 ICCB6_000289 C[Si](C)(F)C(CC(=O)c1ccccc1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N04 compound treatment 1252520.0 45500.0 0.76 1212520.0 18600.0 0.34 0.7752 0.9321 2065833 ICCB6_000290 CCCCOc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N(C)OC)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N05 compound treatment 1258200.0 51200.0 0.86 1247920.0 54000.0 0.97 1.2934 0.998 2065834 ICCB6_000291 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)CN1C(=O)CCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N06 compound treatment 1228800.0 21800.0 0.36 1218000.0 24100.0 0.43 0.5644 0.9962 2065835 ICCB6_000292 CC1(C)N[C@H](Cc2c[nH]c3ccccc23)[C@@H]4CC1CCC4=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N07 compound treatment 1249840.0 42800.0 0.72 1247920.0 54000.0 0.97 1.1945 0.9887 2065836 ICCB6_000293 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)[C@H](C(C)C)N1C(=O)Cc4ccc(OC)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N08 compound treatment 1238040.0 31000.0 0.52 1223560.0 29600.0 0.53 0.7445 0.9999 2065837 ICCB6_000294 CN1[C@H](Cc2c[nH]c3ccccc23)[C@@H]4CC(CCC4=C)C1(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N09 compound treatment 1246760.0 39700.0 0.66 1232160.0 38200.0 0.69 0.9573 0.9998 2065838 ICCB6_000295 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](Cc5ccccc5)N1C(=O)CCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N10 compound treatment 1237480.0 30400.0 0.51 1238880.0 45000.0 0.81 0.9331 0.975 2065839 ICCB6_000296 Cc1ccc(cc1)S(=O)(=O)N[C@H]2CC3CCC2(C)C3(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N11 compound treatment 1244560.0 37500.0 0.63 1236440.0 42500.0 0.77 0.9858 0.9951 2065840 ICCB6_000297 CCOC(=O)CC(CC(=O)OCC)(C(=O)OCC)c1cccnc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N12 compound treatment 1170600.0 -36400.0 -0.61 1176160.0 -17800.0 -0.32 -0.6574 -0.9547 2065841 ICCB6_000298 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CCC6CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N13 compound treatment 1083320.0 -124000.0 -2.07 1075240.0 -119000.0 -2.14 -2.9759 -0.9999 1952445 ICCB6_000299 Clc1ccc2oc(nc2c1)c3ccc(NC(=O)c4ccc(CNC(=O)OCc5ccccc5)cc4)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N14 compound treatment 1208760.0 1730.0 0.03 1195240.0 1320.0 0.02 0.0373 0.9953 2065842 ICCB6_000300 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N15 compound treatment 1240400.0 33400.0 0.56 1211600.0 17700.0 0.32 0.6201 0.9646 1952801 ICCB6_000301 Oc1ccccc1C#Cc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N16 compound treatment 1034800.0 -172000.0 -2.88 1130400.0 -63500.0 -1.14 -2.8473 -0.9181 2065843 ICCB6_000302 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N17 compound treatment 1204520.0 -2510.0 -0.04 1192640.0 -1280.0 -0.02 -0.046 -0.9601 1952836 ICCB6_000303 CC(=O)c1ccc2oc(cc2c1)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N18 compound treatment 1191800.0 -15200.0 -0.25 1177840.0 -16100.0 -0.29 -0.3851 -0.998 2065844 ICCB6_000304 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N19 compound treatment 1203480.0 -3550.0 -0.06 1193200.0 -720.0 -0.01 -0.0512 -0.8416 1952631 ICCB6_000305 CCOC(=O)[C@H](CC(C)C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCc3cccc(c3)C(F)(F)F)O2)O1)OC(=O)NCc4ccc5OCOc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N20 compound treatment 1132320.0 -74700.0 -1.25 1125840.0 -68100.0 -1.23 -1.7514 -1.0 2065845 ICCB6_000306 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N21 compound treatment 1172160.0 -34900.0 -0.58 1166360.0 -27600.0 -0.5 -0.7638 -0.9968 3005761 ICCB6_000307 Cc1ccc(cc1)S(=O)(=O)O.Cc1cc(=O)oc2ccc(Cl)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N22 compound treatment 1111480.0 -95600.0 -1.6 1127160.0 -66800.0 -1.2 -1.9812 -0.9902 2065846 ICCB6_000308 CN(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)Cc8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N23 mock treatment 1183560.0 -23500.0 -0.39 1171840.0 -22100.0 -0.4 -0.559 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 N24 mock treatment 1201880.0 -5150.0 -0.09 1189360.0 -4560.0 -0.08 -0.1191 -0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O01 compound treatment 1314840.0 108000.0 1.8 1293160.0 99200.0 1.79 2.54 1.0 2065847 ICCB6_000309 CCOC(=O)[C@@H]1[C@@H](C(=O)OC)[C@@]2([C@H](N1c3cccc(F)c3)c4ccccc4)C(=O)N(Cc5ccccc5)c6ccccc62 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O02 compound treatment 1267960.0 60900.0 1.02 1235240.0 41300.0 0.74 1.2474 0.9881 3176588 ICCB6_000310 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)N(C(=O)NCc5ccc(Cl)c(Cl)c5)c6ccc(C#CC7(O)CCCCCC7)cc64)C(C(OC2=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O03 compound treatment 1272520.0 65500.0 1.1 1256120.0 62200.0 1.12 1.5674 0.9999 2065848 ICCB6_000311 Cc1ccc(cc1)c2c(cc(c3ccccc3)n2c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O04 compound treatment 1282080.0 75000.0 1.26 1251240.0 57300.0 1.03 1.6183 0.9953 3176589 ICCB6_000312 CON(C)C(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)N(C(=O)OCc5ccc(cc5)[N+](=O)[O-])c6ccc(C#CC7(O)CCCCCC7)cc64)C(C(OC2=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O05 compound treatment 1287280.0 80200.0 1.34 1266200.0 72300.0 1.3 1.8704 0.9999 2065849 ICCB6_000313 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)CN1C(=O)CCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O06 compound treatment 1247040.0 40000.0 0.67 1233720.0 39800.0 0.72 0.9805 0.9994 2065850 ICCB6_000314 COc1cc(C[C@@H]2[C@@H]3CC(CCC3=C)C(C)(C)N2N=Nc4ccc(Br)cc4)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O07 compound treatment 1235920.0 28900.0 0.48 1213840.0 19900.0 0.36 0.5956 0.9892 2065851 ICCB6_000315 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C(C)C)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O08 compound treatment 1261200.0 54200.0 0.91 1248960.0 55000.0 0.99 1.3422 0.999 2065852 ICCB6_000316 COc1cc(C[C@@H]2[C@@H]3CC(CCC3=C)C(C)(C)N2N=Nc4ccc(cc4)[N+](=O)[O-])cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O09 compound treatment 1268640.0 61600.0 1.03 1246400.0 52500.0 0.95 1.3976 0.9991 2065853 ICCB6_000317 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccc(OC)c(OC)c3)c4cc(OCCCO)ccc4N2C(=O)[C@H](Cc5ccccc5)N1C(=O)Cc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O10 compound treatment 1206360.0 -671.0 -0.01 1204360.0 10400.0 0.19 0.1251 0.6637 2065854 ICCB6_000318 CC(C)C[C@@H]1[C@@H]2CC(CCC2=C)C(C)(C)N1N=Nc3ccc(Br)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O11 compound treatment 1246360.0 39300.0 0.66 1221720.0 27800.0 0.5 0.8196 0.9909 2065855 ICCB6_000319 CCOC(=O)CC(C(=O)OCC)c1cccnc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O12 compound treatment 1231400.0 24400.0 0.41 1215640.0 21700.0 0.39 0.5651 0.9998 2065856 ICCB6_000320 CC(C)C[C@@H]1[C@@H]2CC(CCC2=C)C(C)(C)N1N=Nc3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O13 compound treatment 1209160.0 2130.0 0.04 1207680.0 13800.0 0.25 0.2005 0.8005 1952450 ICCB6_000321 CCOC(=O)C(O)C(O)c1ccc(CO[Si](C(C)C)(C(C)C)c2ccccc2)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O14 compound treatment 1202200.0 -4830.0 -0.08 1178320.0 -15600.0 -0.28 -0.2559 -0.875 2065857 ICCB6_000322 C[C@@H]1[C@@H]2CC(CCC2=C)C(C)(C)N1N=Nc3ccc(Br)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O15 compound treatment 1189400.0 -17600.0 -0.3 1178960.0 -15000.0 -0.27 -0.3992 -0.999 1952761 ICCB6_000323 COc1ccc(cc1)C(=C2C(=O)Oc3ccccc23)c4ccc(OC)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O16 compound treatment 1184800.0 -22200.0 -0.37 1183240.0 -10700.0 -0.19 -0.3991 -0.9529 2065858 ICCB6_000324 C[C@@H]1[C@@H]2CC(CCC2=C)C(C)(C)N1N=Nc3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O17 compound treatment 1186440.0 -20600.0 -0.34 1167480.0 -26400.0 -0.48 -0.5805 -0.9874 1952837 ICCB6_000325 COCCNC(=O)c1ccc(c(C#CC(C)(O)CC(C)C)c1O)c2cc(F)cc(F)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O18 compound treatment 576200.0 -631000.0 -10.56 700200.0 -494000.0 -8.9 -13.7547 -0.9964 2065859 ICCB6_000326 CO[C@H]1O[C@@H]2COC(O[C@H]2[C@H](OC(=O)/C=C/C=C/C)[C@H]1OC(=O)/C=C/C=C/C)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O19 compound treatment 1191360.0 -15700.0 -0.26 1178680.0 -15200.0 -0.27 -0.3796 -0.9997 1952633 ICCB6_000327 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCc3ccccc3)O2)O1)OC(=O)NCc4ccc5OCOc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O20 compound treatment 1185320.0 -21700.0 -0.36 1174240.0 -19700.0 -0.35 -0.5076 -0.9999 2065860 ICCB6_000328 CC(C)(C)[Si](C)(C)O[C@@H]1[C@@H](COC(c2ccccc2)(c3ccccc3)c4ccccc4)O[C@H](CC=C)[C@H](O[Si](C)(C)C(C)(C)C)[C@H]1N=[N+]=[N-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O21 compound treatment 1183840.0 -23200.0 -0.39 1180760.0 -13200.0 -0.24 -0.4421 -0.9721 1952755 ICCB6_000329 C=C(c1ccccc1)c2cc(=O)oc3ccccc23 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O22 compound treatment 1180240.0 -26800.0 -0.45 1175480.0 -18400.0 -0.33 -0.552 -0.9891 2065861 ICCB6_000330 C[C@H]1[C@H](OC(=O)N1C(=O)[C@@H](CC=C)C(C)(C)C)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O23 mock treatment 1175440.0 -31600.0 -0.53 1172640.0 -21300.0 -0.38 -0.6449 -0.9876 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 O24 mock treatment 1207960.0 929.0 0.02 1193320.0 -600.0 -0.01 0.0033 0.1767 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P01 compound treatment 1278680.0 71600.0 1.2 1261760.0 67800.0 1.22 1.7121 1.0 2065862 ICCB6_000331 CC1(C)OCC2=C(CC(CCc3ccccc3)OC2CCc4ccccc4)O1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P02 compound treatment 1243400.0 36400.0 0.61 1221720.0 27800.0 0.5 0.7845 0.9953 2065863 ICCB6_000332 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(I)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P03 compound treatment 1251920.0 44900.0 0.75 1225880.0 32000.0 0.58 0.9383 0.9914 2065864 ICCB6_000333 C1CCC(CC1)c2c(cc(c3ccccc3)n2c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P04 compound treatment 1180720.0 -26300.0 -0.44 1177640.0 -16300.0 -0.29 -0.5188 -0.9805 2065865 ICCB6_000334 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P05 compound treatment 1238600.0 31600.0 0.53 1229400.0 35500.0 0.64 0.8256 0.9955 2065866 ICCB6_000335 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)C(C)C)c3cc(OCCCO)ccc3N2C(=O)CN1C(=O)Cc4ccc(OC)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P06 compound treatment 1139000.0 -68000.0 -1.14 1118560.0 -75400.0 -1.36 -1.7651 -0.9962 2065867 ICCB6_000336 CCCCOc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P07 compound treatment 1248640.0 41600.0 0.7 1232120.0 38200.0 0.69 0.979 1.0 2065868 ICCB6_000337 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](C(C)C)N1C(=O)Cc5ccc(OC)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P08 compound treatment 1009720.0 -197000.0 -3.3 1000760.0 -193000.0 -3.48 -4.7957 -0.9997 2065869 ICCB6_000338 C[C@H](Cc1ccccc1)N(C)CC#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P09 compound treatment 1254360.0 47300.0 0.79 1240960.0 47000.0 0.85 1.1593 0.9994 2065870 ICCB6_000339 CCOC(=O)CC1[C@@H]2[C@@H](NC(=O)c3ccccc3)c4cc(OCCCO)ccc4N2C(=O)[C@H](Cc5ccccc5)N1C(=O)Cc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P10 compound treatment 1177480.0 -29600.0 -0.49 1169920.0 -24000.0 -0.43 -0.6554 -0.9978 2065871 ICCB6_000340 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P11 compound treatment 1013600.0 -193000.0 -3.24 1003800.0 -190000.0 -3.43 -4.711 -0.9996 2065872 ICCB6_000341 CCOC(=O)/C(=C/1\NSc2ccccc12)/C#N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P12 compound treatment 1088680.0 -118000.0 -1.98 1091360.0 -103000.0 -1.85 -2.7071 -0.9994 2065873 ICCB6_000342 CCOC(OCC)C#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P13 compound treatment 1225160.0 18100.0 0.3 1212560.0 18600.0 0.34 0.452 0.9987 2065874 ICCB6_000343 COC(=O)C(C(=O)OC)c1ccc(cc1I)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P14 compound treatment 733320.0 -474000.0 -7.93 837720.0 -356000.0 -6.42 -10.1435 -0.9945 2065875 ICCB6_000344 Brc1ccc2NC(=O)/C(=C/C(=O)OCC=C)/c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P15 compound treatment 227120.0 -980000.0 -16.4 241680.0 -952000.0 -17.16 -23.727 -0.9997 1952804 ICCB6_000345 COc1cc(CO[Si](C)(C)C(C)(C)C)cc(C#CC2(O)CCCCC2)c1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P16 compound treatment 1147480.0 -59600.0 -1.0 1128280.0 -65600.0 -1.18 -1.5409 -0.9964 2065876 ICCB6_000346 CCOC(=O)/C=C\1/C(=O)Nc2ccc(Br)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P17 compound treatment 1170200.0 -36800.0 -0.62 1151400.0 -42500.0 -0.77 -0.9775 -0.9942 1952838 ICCB6_000347 COc1cc(CO[Si](C)(C)C(C)(C)C)cc(C#CC2(O)CCC3C2CC4Cc5cc(O)ccc5C43)c1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P18 compound treatment 1164400.0 -42600.0 -0.71 1157440.0 -36500.0 -0.66 -0.9692 -0.9992 2065877 ICCB6_000348 O=C(/C=C\1/C(=O)Nc2ccccc12)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P19 compound treatment 1182880.0 -24200.0 -0.4 1165560.0 -28400.0 -0.51 -0.6471 -0.9933 1952634 ICCB6_000349 COC(=O)[C@H](C)NC(=O)CC[C@@H]1C[C@H](C[C@@]2(CCC[C@H](COC(=O)NCCOc3ccccc3)O2)O1)OC(=O)NCc4ccc5OCOc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P20 compound treatment 1162120.0 -44900.0 -0.75 1163680.0 -30200.0 -0.54 -0.9167 -0.9875 2065878 ICCB6_000350 CON(C)C(=O)/C=C\1/C(=O)Nc2ccc(Br)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P21 compound treatment 1180320.0 -26700.0 -0.45 1167960.0 -26000.0 -0.47 -0.6468 -0.9997 1952770 ICCB6_000351 O=C/1Oc2ccccc2C\C1=C(/c3ccccc3)\c4ccc5ccccc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P22 compound treatment 1159840.0 -47200.0 -0.79 1151200.0 -42700.0 -0.77 -1.1027 -0.9999 2065879 ICCB6_000352 CON(C)C(=O)/C=C\1/C(=O)Nc2ccc(I)cc12 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P23 mock treatment 1194880.0 -12200.0 -0.2 1183560.0 -10400.0 -0.19 -0.2758 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.1463 P24 mock treatment 1214120.0 7090.0 0.12 1201440.0 7520.0 0.14 0.1797 0.9978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A01 mock treatment 1288040.0 51900.0 0.87 1273720.0 40500.0 0.73 1.1304 0.9963 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A02 mock treatment 1287880.0 51700.0 0.87 1276640.0 43400.0 0.78 1.1657 0.9987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A03 compound treatment 1157200.0 -78900.0 -1.32 1138960.0 -94200.0 -1.7 -2.1347 -0.9923 3000673 BCB01_000001 COc1cc(NN2C3C(C=CC2C(O)c4ccccc4)C(=O)N(C3=O)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A04 compound treatment 1240040.0 3900.0 0.07 1243080.0 9880.0 0.18 0.172 0.9072 3000674 BCB01_000002 CC(C)C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A05 compound treatment 1233760.0 -2380.0 -0.04 1213040.0 -20200.0 -0.36 -0.285 -0.78 3000675 BCB01_000003 COc1cc(NN2C3C(C=CC2C(O)c4ccc(I)cc4)C(=O)N(C3=O)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A06 compound treatment 1252640.0 16500.0 0.28 1257800.0 24600.0 0.44 0.5087 0.974 3000676 BCB01_000004 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5cccc(O)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A07 compound treatment 1236360.0 219.0 0.0 1241600.0 8400.0 0.15 0.1096 0.724 3093034 BCB01_000005 COc1cc(NN2C3C(C=CC2C(O)c4ccc(cc4)N(C)C)C(=O)N(C3=O)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A08 compound treatment 1216680.0 -19500.0 -0.33 1225280.0 -7920.0 -0.14 -0.3312 -0.9314 3000677 BCB01_000006 OB(O)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A09 compound treatment 1197000.0 -39100.0 -0.66 1209040.0 -24200.0 -0.44 -0.7709 -0.9803 3093035 BCB01_000007 COc1cc(NN2C3C(C=CC2C(O)c4cc(OC)c(OC)c(OC)c4)C(=O)N(C3=O)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A10 compound treatment 1224920.0 -11200.0 -0.19 1219080.0 -14100.0 -0.25 -0.3126 -0.9888 3000678 BCB01_000008 OC(C1CCC=CC1)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A11 compound treatment 1221360.0 -14800.0 -0.25 1211640.0 -21600.0 -0.39 -0.4496 -0.9763 3093104 BCB01_000009 COc1cc(NN2C3C(C=CC2C(O)C4CCCCC4)C(=O)N(C3=O)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A12 compound treatment 1244200.0 8060.0 0.13 1245520.0 12300.0 0.22 0.2523 0.9715 3093105 BCB01_000010 CC(=O)n1cc(C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A13 compound treatment 1124320.0 -112000.0 -1.87 1140080.0 -93100.0 -1.68 -2.5095 -0.9985 3000679 BCB01_000011 COc1cc(NN2C3C(C=CC2C(O)c4ccco4)C(=O)N(C3=O)c5ccccc5)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A14 compound treatment 1229200.0 -6940.0 -0.12 1227840.0 -5360.0 -0.1 -0.1504 -0.9958 3093106 BCB01_000012 CCCCC(CC)C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A15 compound treatment 1149000.0 -87100.0 -1.46 1160680.0 -72500.0 -1.31 -1.955 -0.9985 3093107 BCB01_000013 CCCCCCCCCC(O)C1C=CC2C(N1Nc3cc(OC)c(OC)c(OC)c3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A16 compound treatment 1204760.0 -31400.0 -0.53 1209440.0 -23800.0 -0.43 -0.674 -0.9949 3000680 BCB01_000014 CC(C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A17 compound treatment 1167200.0 -68900.0 -1.15 1164400.0 -68800.0 -1.24 -1.6923 -0.9994 3093108 BCB01_000015 COc1cc(NN2C3C(C=CC2C(O)c4ccccc4)C(=O)N(C)C3=O)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A18 compound treatment 1190480.0 -45700.0 -0.76 1179560.0 -53600.0 -0.97 -1.2237 -0.9932 3093109 BCB01_000016 CC(CC(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(C)o5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A19 compound treatment 1186440.0 -49700.0 -0.83 1202640.0 -30600.0 -0.55 -0.9774 -0.9799 3000681 BCB01_000017 COc1cc(NN2C3C(C=CC2C(O)c4ccc(I)cc4)C(=O)N(C)C3=O)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A20 compound treatment 1199360.0 -36800.0 -0.62 1204440.0 -28800.0 -0.52 -0.8016 -0.9963 3093110 BCB01_000018 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5cccs5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A21 compound treatment 1191840.0 -44300.0 -0.74 1194560.0 -38600.0 -0.7 -1.0165 -0.9995 3000682 BCB01_000019 OC(C1CCCCC1)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A22 compound treatment 1186000.0 -50100.0 -0.84 1181200.0 -52000.0 -0.94 -1.2558 -0.9985 3093111 BCB01_000020 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(C#N)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A23 mock treatment 1202840.0 -33300.0 -0.56 1199600.0 -33600.0 -0.61 -0.8221 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 A24 mock treatment 1193360.0 -42800.0 -0.72 1185960.0 -47200.0 -0.85 -1.108 -0.9963 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B01 mock treatment 1290040.0 53900.0 0.9 1284440.0 51200.0 0.92 1.2906 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B02 mock treatment 1284960.0 48800.0 0.82 1279760.0 46600.0 0.84 1.1709 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B03 compound treatment 1173920.0 -62200.0 -1.04 1172920.0 -60300.0 -1.09 -1.5042 -0.9998 3093112 BCB01_000021 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccccn4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B04 compound treatment 1217040.0 -19100.0 -0.32 1226120.0 -7080.0 -0.13 -0.3162 -0.9188 3000683 BCB01_000022 CN(C)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B05 compound treatment 1238560.0 2420.0 0.04 1240400.0 7200.0 0.13 0.1204 0.8856 3093113 BCB01_000023 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccc(cc4)C(C)C)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B06 compound treatment 1232600.0 -3540.0 -0.06 1233880.0 682.0 0.01 -0.0332 -0.5488 3093114 BCB01_000024 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B07 compound treatment 1233640.0 -2500.0 -0.04 1241080.0 7880.0 0.14 0.0708 0.4784 3000684 BCB01_000025 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B08 compound treatment 1247840.0 11700.0 0.2 1244640.0 11400.0 0.21 0.2842 0.9997 3093115 BCB01_000026 CC(=O)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B09 compound treatment 1188280.0 -47900.0 -0.8 1189440.0 -43800.0 -0.79 -1.1238 -1.0 3093116 BCB01_000027 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4c(F)cccc4Cl)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B10 compound treatment 1224800.0 -11300.0 -0.19 1218280.0 -14900.0 -0.27 -0.3243 -0.9855 3000685 BCB01_000028 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccc(s5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B11 compound treatment 1225640.0 -10500.0 -0.18 1227480.0 -5720.0 -0.1 -0.1971 -0.9676 3093117 BCB01_000029 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4c(C)cc(C)cc4C)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B12 compound treatment 1230200.0 -5940.0 -0.1 1240440.0 7240.0 0.13 0.022 0.1339 3093118 BCB01_000030 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B13 compound treatment 1222960.0 -13200.0 -0.22 1224800.0 -8400.0 -0.15 -0.263 -0.9831 3000686 BCB01_000031 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccccc4C)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B14 compound treatment 1219960.0 -16200.0 -0.27 1208000.0 -25200.0 -0.45 -0.5125 -0.9695 3093119 BCB01_000032 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccco4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B15 compound treatment 1206000.0 -30100.0 -0.5 1199960.0 -33200.0 -0.6 -0.7801 -0.9964 3093120 BCB01_000033 CC(C)c1ccc(NN2C3C(C=CC2C(O)C(c4ccccc4)c5ccccc5)C(=O)N(C3=O)c6ccccc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B16 compound treatment 1181560.0 -54600.0 -0.91 1181200.0 -52000.0 -0.94 -1.3083 -0.9999 3000687 BCB01_000034 CCCCC(O)C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B17 compound treatment 1196760.0 -39400.0 -0.66 1194520.0 -38700.0 -0.7 -0.9588 -0.9996 3000688 BCB01_000035 C/C=C/C(O)C1C=CC2C(N1Nc3ccc(cc3)C(C)C)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B18 compound treatment 1201000.0 -35100.0 -0.59 1200240.0 -33000.0 -0.59 -0.8357 -1.0 3093121 BCB01_000036 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B19 compound treatment 1153840.0 -82300.0 -1.38 1185840.0 -47400.0 -0.85 -1.5772 -0.9735 3093122 BCB01_000037 CCC(CC)C(O)C1C=CC2C(N1Nc3ccc(cc3)C(C)C)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B20 compound treatment 1180080.0 -56100.0 -0.94 1182000.0 -51200.0 -0.92 -1.3156 -1.0 3093123 BCB01_000038 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc(F)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B21 compound treatment 1162240.0 -73900.0 -1.24 1166120.0 -67100.0 -1.21 -1.7291 -0.9999 3000689 BCB01_000039 CC(C)C(O)C1C=CC2C(N1Nc3ccc(cc3)C(C)C)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B22 compound treatment 1154240.0 -81900.0 -1.37 1158160.0 -75000.0 -1.35 -1.9251 -1.0 3093124 BCB01_000040 COc1ccc(C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O)c5ccccc15 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B23 mock treatment 1179760.0 -56400.0 -0.94 1177680.0 -55500.0 -1.0 -1.3745 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 B24 mock treatment 1211200.0 -24900.0 -0.42 1186960.0 -46200.0 -0.83 -0.8842 -0.9489 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C01 mock treatment 1280640.0 44500.0 0.74 1274120.0 40900.0 0.74 1.0479 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C02 mock treatment 1283600.0 47500.0 0.79 1271520.0 38300.0 0.69 1.0498 0.9976 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C03 compound treatment 1240680.0 4540.0 0.08 1246920.0 13700.0 0.25 0.2285 0.8836 3000690 BCB01_000041 COc1cc(NN2C3C(C=CC2C(O)c4cc(OC)c(OC)c(OC)c4)C(=O)N(C)C3=O)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C04 compound treatment 1258240.0 22100.0 0.37 1249200.0 16000.0 0.29 0.4654 0.9924 3093125 BCB01_000042 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C05 compound treatment 1216800.0 -19300.0 -0.32 1209800.0 -23400.0 -0.42 -0.527 -0.9915 3093282 BCB01_000043 COc1cc(NN2C3C(C=CC2C(O)C4CCCCC4)C(=O)N(C)C3=O)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C06 compound treatment 1260840.0 24700.0 0.41 1248400.0 15200.0 0.27 0.4859 0.98 3000691 BCB01_000044 CC1(C)[C@H]2C[C@@H]1C=C(C2)C(O)C3C=CC4C(N3Nc5ccccc5)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C07 compound treatment 1197480.0 -38700.0 -0.65 1185160.0 -48000.0 -0.87 -1.0695 -0.9897 3093194 BCB01_000045 COc1cc(NN2C3C(C=CC2C(O)C4CCC(CC4)C(=C)C)C(=O)N(C)C3=O)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C08 compound treatment 1247920.0 11800.0 0.2 1245520.0 12300.0 0.22 0.2964 0.9982 3093195 BCB01_000046 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(Br)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C09 compound treatment 1229120.0 -7020.0 -0.12 1220200.0 -13000.0 -0.23 -0.2487 -0.9491 3000692 BCB01_000047 COc1cc(NN2C3C(C=CC2C(O)c4ccco4)C(=O)N(C)C3=O)cc(OC)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C10 compound treatment 1240160.0 4020.0 0.07 1230600.0 -2600.0 -0.05 0.0145 0.1764 3093196 BCB01_000048 CC(=CCC/C(=C/C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)/C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C11 compound treatment 1188800.0 -47300.0 -0.79 1212920.0 -20300.0 -0.37 -0.8185 -0.9382 3093197 BCB01_000049 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3cc(OC)c(OC)c(OC)c3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C12 compound treatment 1235040.0 -1100.0 -0.02 1227360.0 -5840.0 -0.11 -0.0874 -0.8185 3000693 BCB01_000050 OC(CCc1ccccc1)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C13 compound treatment 1206560.0 -29600.0 -0.5 1235960.0 2760.0 0.05 -0.3148 -0.6328 3093198 BCB01_000051 CN1C(=O)C2C=CC(C(O)c3ccccc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C14 compound treatment 1230080.0 -6060.0 -0.1 1228160.0 -5040.0 -0.09 -0.1359 -0.9985 3000694 BCB01_000052 CN1C(=O)C2C=CC(C(O)c3ccccc3)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C15 compound treatment 1215960.0 -20200.0 -0.34 1218120.0 -15100.0 -0.27 -0.4309 -0.9942 3093199 BCB01_000053 CN1C(=O)C2C=CC(C(O)c3ccc(I)cc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C16 compound treatment 1188240.0 -47900.0 -0.8 1195240.0 -38000.0 -0.68 -1.0504 -0.9969 3093200 BCB01_000054 CN1C(=O)C2C=CC(C(O)c3ccc(I)cc3)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C17 compound treatment 1216040.0 -20100.0 -0.34 1210280.0 -22900.0 -0.41 -0.5298 -0.9948 3000695 BCB01_000055 CN1C(=O)C2C=CC(C(O)c3ccc(cc3)[N+](=O)[O-])N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C18 compound treatment 1211800.0 -24300.0 -0.41 1203880.0 -29300.0 -0.53 -0.6615 -0.9918 3093201 BCB01_000056 CN1C(=O)C2C=CC(C(O)c3ccc(cc3)[N+](=O)[O-])N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C19 compound treatment 1182000.0 -54100.0 -0.91 1191440.0 -41800.0 -0.75 -1.1727 -0.9957 3093202 BCB01_000057 COc1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C20 compound treatment 1194800.0 -41300.0 -0.69 1186480.0 -46700.0 -0.84 -1.0844 -0.9953 3000696 BCB01_000058 COc1ccc(cc1)C(O)C2C=CC3C(N2N4CCCCC4)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C21 compound treatment 1175200.0 -60900.0 -1.02 1182840.0 -50400.0 -0.91 -1.3627 -0.9983 3093203 BCB01_000059 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C22 compound treatment 1166280.0 -69900.0 -1.17 1165440.0 -67800.0 -1.22 -1.6899 -0.9998 3093204 BCB01_000060 CN1C(=O)C2C=CC(C(O)C#Cc3ccccc3)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C23 mock treatment 1187240.0 -48900.0 -0.82 1192080.0 -41100.0 -0.74 -1.1025 -0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 C24 mock treatment 1201400.0 -34700.0 -0.58 1193920.0 -39300.0 -0.71 -0.9115 -0.9952 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D01 mock treatment 1301480.0 65300.0 1.09 1298320.0 65100.0 1.17 1.6028 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D02 mock treatment 1297080.0 60900.0 1.02 1281680.0 48500.0 0.87 1.3388 0.997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D03 compound treatment 1201600.0 -34500.0 -0.58 1200640.0 -32600.0 -0.59 -0.8235 -1.0 3000697 BCB01_000061 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4cccc(O)c4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D04 compound treatment 1269960.0 33800.0 0.57 1258240.0 25000.0 0.45 0.7192 0.9937 3093205 BCB01_000062 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D05 compound treatment 1003840.0 -232000.0 -3.89 965120.0 -268000.0 -4.83 -6.1642 -0.9942 3093206 BCB01_000063 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccc(cc4)B(O)O)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D06 compound treatment 1243920.0 7780.0 0.13 1244600.0 11400.0 0.21 0.2373 0.9758 3000698 BCB01_000064 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccccn4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D07 compound treatment 1240680.0 4540.0 0.08 1246280.0 13100.0 0.24 0.2204 0.8899 3093207 BCB01_000065 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4cn(C(=O)C)c5ccccc45)C(=O)N(C3=O)c6ccccc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D08 compound treatment 1258480.0 22300.0 0.37 1247360.0 14200.0 0.26 0.4448 0.9827 3000792 BCB01_000066 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D09 compound treatment 1246520.0 10400.0 0.17 1240960.0 7760.0 0.14 0.2217 0.9942 3000794 BCB01_000067 CC(C)c1ccc(NN2C3C(C=CC2C(O)C(C)c4ccccc4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D10 compound treatment 1238000.0 1860.0 0.03 1245000.0 11800.0 0.21 0.1724 0.802 3000796 BCB01_000068 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D11 compound treatment 1210360.0 -25800.0 -0.43 1215680.0 -17500.0 -0.32 -0.5283 -0.9882 3000797 BCB01_000069 CC(C)c1ccc(NN2C3C(C=CC2C(O)CC(C)c4ccc(C)o4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D12 compound treatment 1238800.0 2660.0 0.04 1248880.0 15700.0 0.28 0.2313 0.8085 3093208 BCB01_000070 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4c(F)cccc4Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D13 compound treatment 1198360.0 -37800.0 -0.63 1198160.0 -35000.0 -0.63 -0.8935 -1.0 3093209 BCB01_000071 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4cccs4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D14 compound treatment 1216520.0 -19600.0 -0.33 1228760.0 -4440.0 -0.08 -0.2887 -0.8543 3000798 BCB01_000072 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc(s4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D15 compound treatment 1195360.0 -40800.0 -0.68 1195800.0 -37400.0 -0.67 -0.959 -1.0 3093210 BCB01_000073 CC(C)c1ccc(NN2C3C(C=CC2C(O)Cc4ccccc4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D16 compound treatment 1176520.0 -59600.0 -1.0 1178960.0 -54200.0 -0.98 -1.3965 -0.9999 3000800 BCB01_000074 Cn1cccc1C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D17 compound treatment 1197720.0 -38400.0 -0.64 1192480.0 -40700.0 -0.73 -0.9734 -0.9978 3093211 BCB01_000075 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D18 compound treatment 1187280.0 -48900.0 -0.82 1166400.0 -66800.0 -1.2 -1.4292 -0.9823 3000876 BCB01_000076 Cc1cc(C)c(C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O)c(C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D19 compound treatment 1158400.0 -77700.0 -1.3 1170040.0 -63200.0 -1.14 -1.7246 -0.9978 3000877 BCB01_000077 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccc5OCOc5c4)C(=O)N(C3=O)c6ccccc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D20 compound treatment 1182960.0 -53200.0 -0.89 1197480.0 -35700.0 -0.64 -1.0843 -0.9873 3000878 BCB01_000078 Cc1ccccc1C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D21 compound treatment 1153480.0 -82700.0 -1.38 1171080.0 -62100.0 -1.12 -1.7695 -0.9945 3000880 BCB01_000079 CC(C)c1ccc(NN2C3C(C=CC2C(O)C4=C[C@H]5C[C@@H](C4)C5(C)C)C(=O)N(C3=O)c6ccccc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D22 compound treatment 1097960.0 -138000.0 -2.31 1095200.0 -138000.0 -2.49 -3.3932 -0.9993 3093212 BCB01_000080 OC(/C=C/c1ccc(cc1)[N+](=O)[O-])C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D23 mock treatment 1185520.0 -50600.0 -0.85 1187920.0 -45300.0 -0.82 -1.1759 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 D24 mock treatment 1179280.0 -56900.0 -0.95 1185400.0 -47800.0 -0.86 -1.2818 -0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E01 mock treatment 1283400.0 47300.0 0.79 1285920.0 52700.0 0.95 1.2309 0.9959 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E02 mock treatment 1272200.0 36100.0 0.6 1274160.0 41000.0 0.74 0.9485 0.995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E03 compound treatment 1192320.0 -43800.0 -0.73 1178680.0 -54500.0 -0.98 -1.2131 -0.9896 3000882 BCB01_000081 CN1C(=O)C2C=CC(C(O)C#Cc3ccccc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E04 compound treatment 1251600.0 15500.0 0.26 1257280.0 24100.0 0.43 0.4897 0.9695 3093213 BCB01_000082 CN1C(=O)C2C=CC(C(O)C3CCCCC3)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E05 compound treatment 1265960.0 29800.0 0.5 1243560.0 10400.0 0.19 0.4849 0.91 3093214 BCB01_000083 CN1C(=O)C2C=CC(C(O)C3=CC[C@H](CC3)C(=C)C)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E06 compound treatment 1250960.0 14800.0 0.25 1246400.0 13200.0 0.24 0.3435 0.9998 3000884 BCB01_000084 CN1C(=O)C2C=CC(C(O)C3CCC(CC3)C(=C)C)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E07 compound treatment 1235120.0 -1020.0 -0.02 1235760.0 2560.0 0.05 0.0206 0.4177 3093215 BCB01_000085 CN1C(=O)C2C=CC(C(O)c3ccco3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E08 compound treatment 1255880.0 19700.0 0.33 1250360.0 17200.0 0.31 0.4522 0.9995 3093216 BCB01_000086 CCCCC(O)C1C=CC2C(N1N3CCCCC3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E09 compound treatment 1241040.0 4900.0 0.08 1241200.0 8000.0 0.14 0.1599 0.9642 3000885 BCB01_000087 CCCCC(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E10 compound treatment 1224280.0 -11900.0 -0.2 1226640.0 -6560.0 -0.12 -0.2239 -0.9693 3093283 BCB01_000088 CCCCCCCCCCC(O)C1C=CC2C(N1N3CCCCC3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E11 compound treatment 1221520.0 -14600.0 -0.24 1221720.0 -11500.0 -0.21 -0.3192 -0.9965 3093284 BCB01_000089 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E12 compound treatment 1233920.0 -2220.0 -0.04 1236960.0 3760.0 0.07 0.0216 0.28 3000886 BCB01_000090 CN1C(=O)C2C=CC(C(O)c3ccc(F)cc3)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E13 compound treatment 1225440.0 -10700.0 -0.18 1234360.0 1160.0 0.02 -0.1118 -0.6202 3093285 BCB01_000091 CN1C(=O)C2C=CC(C(O)c3ccc(F)cc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E14 compound treatment 1234720.0 -1420.0 -0.02 1224360.0 -8840.0 -0.16 -0.1294 -0.8038 3093286 BCB01_000092 COc1ccc(C(O)C2C=CC3C(N2N4CCCCC4)C(=O)N(C)C3=O)c5ccccc15 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E15 compound treatment 1200200.0 -35900.0 -0.6 1203080.0 -30100.0 -0.54 -0.809 -0.9987 3000889 BCB01_000093 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E16 compound treatment 1235360.0 -781.0 -0.01 1222880.0 -10300.0 -0.19 -0.1407 -0.755 3093287 BCB01_000094 COc1cc(Br)cc(C(O)C2C=CC3C(N2N4CCCCC4)C(=O)N(C)C3=O)c1OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E17 compound treatment 1212960.0 -23200.0 -0.39 1214720.0 -18500.0 -0.33 -0.5097 -0.9971 3093288 BCB01_000095 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccccc5)C(=O)N(C)C4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E18 compound treatment 1219160.0 -17000.0 -0.28 1219040.0 -14200.0 -0.26 -0.3813 -0.9985 3000890 BCB01_000096 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3N5CCCCC5)C(=O)N(C)C4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E19 compound treatment 1185000.0 -51100.0 -0.86 1192480.0 -40700.0 -0.73 -1.1239 -0.9971 3093289 BCB01_000097 CN1C(=O)C2C=CC(C(O)c3ccccn3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E20 compound treatment 1196080.0 -40100.0 -0.67 1199280.0 -33900.0 -0.61 -0.9062 -0.9989 3093290 BCB01_000098 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2N4CCCCC4)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E21 compound treatment 1184040.0 -52100.0 -0.87 1187080.0 -46100.0 -0.83 -1.2041 -0.9997 3000891 BCB01_000099 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E22 compound treatment 1171080.0 -65100.0 -1.09 1177800.0 -55400.0 -1.0 -1.4756 -0.9991 3093291 BCB01_000100 CN1C(=O)C2C=CC(C(O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E23 mock treatment 1171120.0 -65000.0 -1.09 1188560.0 -44600.0 -0.8 -1.3381 -0.9889 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 E24 mock treatment 1192280.0 -43900.0 -0.73 1188840.0 -44400.0 -0.8 -1.0841 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F01 mock treatment 1278800.0 42700.0 0.71 1275280.0 42100.0 0.76 1.0409 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F02 mock treatment 1278480.0 42300.0 0.71 1269840.0 36600.0 0.66 0.9678 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F03 compound treatment 1260080.0 23900.0 0.4 1244720.0 11500.0 0.21 0.4301 0.9532 3093292 BCB01_000101 CC(C)c1ccc(NN2C3C(C=CC2C(O)/C=C(\C)/CCC=C(C)C)C(=O)N(C3=O)c4ccccc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F04 compound treatment 1256920.0 20800.0 0.35 1232040.0 -1160.0 -0.02 0.2311 0.6635 3000892 BCB01_000102 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3Nc5ccc(Cl)cc5Cl)C(=O)NC4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F05 compound treatment 1254720.0 18600.0 0.31 1233200.0 1.94 0.0 0.2199 0.7072 3093293 BCB01_000103 CN1C(=O)C2C=CC(C(O)c3ccccc3)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F06 compound treatment 1242680.0 6540.0 0.11 1232600.0 -598.0 -0.01 0.0698 0.6344 3000894 BCB01_000104 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4cccc5ccccc45 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F07 compound treatment 1260120.0 24000.0 0.4 1258600.0 25400.0 0.46 0.6074 0.9979 3093294 BCB01_000105 CN1C(=O)C2C=CC(C(O)c3ccc(I)cc3)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F08 compound treatment 1235040.0 -1100.0 -0.02 1221840.0 -11400.0 -0.2 -0.1577 -0.7677 3093295 BCB01_000106 C/C=C/C(O)C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F09 compound treatment 1241720.0 5580.0 0.09 1245680.0 12500.0 0.22 0.225 0.9242 3000896 BCB01_000107 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2NC(=O)OC(C)(C)C)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F10 compound treatment 1214720.0 -21400.0 -0.36 1211240.0 -22000.0 -0.4 -0.5332 -0.9988 3093296 BCB01_000108 CCC(CC)C(O)C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F11 compound treatment 1237760.0 1620.0 0.03 1226360.0 -6840.0 -0.12 -0.068 -0.5387 3093297 BCB01_000109 CN1C(=O)C2C=CC(C(O)c3ccc(cc3)C(=O)C)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F12 compound treatment 1235640.0 -501.0 -0.01 1226680.0 -6520.0 -0.12 -0.089 -0.7557 3000898 BCB01_000110 CC(C)C(O)C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F13 compound treatment 1199080.0 -37100.0 -0.62 1163120.0 -70100.0 -1.26 -1.3313 -0.9464 3000979 BCB01_000111 CCCCCCCCCCC(O)C1C=CC2C(N1NC(=O)OC(C)(C)C)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F14 compound treatment 1221360.0 -14800.0 -0.25 1226600.0 -6600.0 -0.12 -0.259 -0.9436 3000980 BCB01_000112 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4cccc(O)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F15 compound treatment 1222520.0 -13600.0 -0.23 1206040.0 -27200.0 -0.49 -0.5072 -0.9396 3000981 BCB01_000113 CN1C(=O)C2C=CC(C(O)c3ccc(F)cc3)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F16 compound treatment 1215920.0 -20200.0 -0.34 1202560.0 -30600.0 -0.55 -0.6296 -0.9724 3000982 BCB01_000114 OB(O)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F17 compound treatment 1188520.0 -47600.0 -0.8 1206760.0 -26400.0 -0.48 -0.9003 -0.9697 3000984 BCB01_000115 COc1ccc(C(O)C2C=CC3C(N2NC(=O)OC(C)(C)C)C(=O)N(C)C3=O)c4ccccc14 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F18 compound treatment 1207880.0 -28300.0 -0.47 1200880.0 -32300.0 -0.58 -0.7462 -0.9947 3093298 BCB01_000116 Cc1cc(C)c(C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5)c(C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F19 compound treatment 1179200.0 -56900.0 -0.95 1207880.0 -25300.0 -0.46 -0.9963 -0.9431 3093299 BCB01_000117 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2NC(=O)OC(C)(C)C)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F20 compound treatment 1182280.0 -53900.0 -0.9 1173440.0 -59800.0 -1.08 -1.3987 -0.9961 3000987 BCB01_000118 CC(=O)N1CC(C(O)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O)c5ccccc15 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F21 compound treatment 1175520.0 -60600.0 -1.01 1181240.0 -52000.0 -0.94 -1.3793 -0.9992 3093300 BCB01_000119 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F22 compound treatment 1168840.0 -67300.0 -1.13 1166720.0 -66500.0 -1.2 -1.6433 -0.9995 3093301 BCB01_000120 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4cccs4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F23 mock treatment 1165240.0 -70900.0 -1.19 1174760.0 -58400.0 -1.05 -1.5835 -0.9982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 F24 mock treatment 1184360.0 -51800.0 -0.87 1176520.0 -56700.0 -1.02 -1.3348 -0.9967 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G01 mock treatment 1290920.0 54800.0 0.92 1297120.0 63900.0 1.15 1.4626 0.9936 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G02 mock treatment 1292040.0 55900.0 0.94 1290280.0 57100.0 1.03 1.3887 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G03 compound treatment 1259960.0 23800.0 0.4 1272840.0 39600.0 0.71 0.7869 0.9621 3000990 BCB01_000121 CN1C(=O)C2C=CC(C(O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G04 compound treatment 1291720.0 55600.0 0.93 1281680.0 48500.0 0.87 1.2753 0.9995 3093302 BCB01_000122 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccc(F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G05 compound treatment 1270880.0 34700.0 0.58 1245280.0 12100.0 0.22 0.565 0.9102 3093303 BCB01_000123 CN1C(=O)C2C=CC(C(O)c3c(F)cccc3Cl)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G06 compound treatment 1277920.0 41800.0 0.7 1266200.0 33000.0 0.59 0.9148 0.9968 3000991 BCB01_000124 CN1C(=O)C2C=CC(C(O)c3c(C)cc(C)cc3C)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G07 compound treatment 1236800.0 659.0 0.01 1245920.0 12700.0 0.23 0.1699 0.7403 3093304 BCB01_000125 CN1C(=O)C2C=CC(C(O)c3ccc(s3)c4ccccc4)N(Nc5ccccc5)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G08 compound treatment 1253320.0 17200.0 0.29 1256280.0 23100.0 0.42 0.4973 0.9837 3000992 BCB01_000126 CN1C(=O)C2C=CC(C(O)c3ccccc3C)N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G09 compound treatment 1251880.0 15700.0 0.26 1263160.0 30000.0 0.54 0.568 0.9456 3093373 BCB01_000127 CN1C(=O)C2C=CC(C(O)c3c(C)cc(C)cc3C)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G10 compound treatment 1170240.0 -65900.0 -1.1 1154160.0 -79000.0 -1.42 -1.7868 -0.992 3093374 BCB01_000128 CN1C(=O)C2C=CC(C(O)/C=C/c3ccc(cc3)[N+](=O)[O-])N(C2C1=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G11 compound treatment 1239120.0 2980.0 0.05 1253320.0 20100.0 0.36 0.2916 0.7968 3000993 BCB01_000129 CN1C(=O)C2C=CC(C(O)c3ccccc3C)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G12 compound treatment 1204760.0 -31400.0 -0.53 1195760.0 -37400.0 -0.67 -0.8483 -0.9923 3093375 BCB01_000130 CN1C(=O)C2C=CC(C(O)c3cccc4ccccc34)N(C2C1=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G13 compound treatment 1197440.0 -38700.0 -0.65 1189000.0 -44200.0 -0.8 -1.021 -0.9947 3093376 BCB01_000131 CN1C(=O)C2C=CC(C(O)/C=C/c3ccc(cc3)[N+](=O)[O-])N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G14 compound treatment 1236400.0 259.0 0.0 1197560.0 -35600.0 -0.64 -0.451 -0.7023 3000994 BCB01_000132 C/C=C/C(O)C1C=CC2C(N1N3CCCCC3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G15 compound treatment 1227560.0 -8580.0 -0.14 1240160.0 6960.0 0.13 -0.0128 -0.0674 3093377 BCB01_000133 CN1C(=O)C2C=CC(C(O)C(c3ccccc3)c4ccccc4)N(Nc5ccccc5)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G16 compound treatment 1224760.0 -11400.0 -0.19 1227800.0 -5400.0 -0.1 -0.2034 -0.9513 3000995 BCB01_000134 CCC(CC)C(O)C1C=CC2C(N1N3CCCCC3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G17 compound treatment 1226520.0 -9620.0 -0.16 1238800.0 5600.0 0.1 -0.0425 -0.2235 3093378 BCB01_000135 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccco5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G18 compound treatment 1218160.0 -18000.0 -0.3 1196040.0 -37200.0 -0.67 -0.6862 -0.9348 3000996 BCB01_000136 CC(C)C(O)C1C=CC2C(N1N3CCCCC3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G19 compound treatment 1214320.0 -21800.0 -0.37 1218560.0 -14600.0 -0.26 -0.4447 -0.9872 3093379 BCB01_000137 CCC(CC)C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G20 compound treatment 1187280.0 -48900.0 -0.82 1184760.0 -48400.0 -0.87 -1.1953 -0.9995 3093380 BCB01_000138 CN(C)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G21 compound treatment 1191760.0 -44400.0 -0.74 1198480.0 -34700.0 -0.63 -0.9675 -0.9964 3000997 BCB01_000139 CC(C)C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G22 compound treatment 1164280.0 -71900.0 -1.2 1160960.0 -72200.0 -1.3 -1.7707 -0.9992 3093381 BCB01_000140 COc1ccc(C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G23 mock treatment 1187560.0 -48600.0 -0.81 1198480.0 -34700.0 -0.63 -1.0172 -0.9916 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 G24 mock treatment 1191320.0 -44800.0 -0.75 1190480.0 -42700.0 -0.77 -1.0746 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H01 mock treatment 1294960.0 58800.0 0.98 1302520.0 69300.0 1.25 1.5792 0.9931 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H02 mock treatment 1288080.0 51900.0 0.87 1274200.0 41000.0 0.74 1.137 0.9967 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H03 compound treatment 1269440.0 33300.0 0.56 1261160.0 28000.0 0.5 0.7503 0.9987 3000998 BCB01_000141 CN1C(=O)C2C=CC(C(O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H04 compound treatment 1272680.0 36500.0 0.61 1276280.0 43100.0 0.78 0.9812 0.993 3093382 BCB01_000142 OC(Cc1ccccc1)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H05 compound treatment 1264600.0 28500.0 0.48 1260320.0 27100.0 0.49 0.6823 0.9999 3093383 BCB01_000143 CN1C(=O)C2C=CC(C(O)c3c(F)cccc3Cl)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H06 compound treatment 1259640.0 23500.0 0.39 1234400.0 1200.0 0.02 0.2934 0.7449 3000999 BCB01_000144 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc(C#N)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H07 compound treatment 1263080.0 26900.0 0.45 1257320.0 24100.0 0.43 0.6261 0.9998 3093384 BCB01_000145 CN1C(=O)C2C=CC(C(O)c3ccc(s3)c4ccccc4)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H08 compound treatment 1226520.0 -9620.0 -0.16 1233600.0 402.0 0.01 -0.1087 -0.6746 3093385 BCB01_000146 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc5OCOc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H09 compound treatment 1229080.0 -7060.0 -0.12 1235680.0 2480.0 0.04 -0.0519 -0.4111 3001000 BCB01_000147 CN1C(=O)C2C=CC(C(O)C(c3ccccc3)c4ccccc4)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H10 compound treatment 1252360.0 16200.0 0.27 1230320.0 -2880.0 -0.05 0.1553 0.5619 3001068 BCB01_000148 CC1(C)[C@H]2CC1C=C(C2)C(O)C3C=CC4C(N3Nc5ccc(Cl)cc5Cl)C(=O)NC4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H11 compound treatment 1246160.0 10000.0 0.17 1240880.0 7680.0 0.14 0.2164 0.9955 3001069 BCB01_000149 CN1C(=O)C2C=CC(C(O)c3cccc4ccccc34)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H12 compound treatment 1255320.0 19200.0 0.32 1244320.0 11100.0 0.2 0.3686 0.9743 3001070 BCB01_000150 OC(CCc1ccccc1)C2C=CC3C(N2Nc4ccc(Cl)cc4Cl)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H13 compound treatment 1196720.0 -39400.0 -0.66 1219160.0 -14000.0 -0.25 -0.6453 -0.9134 3001072 BCB01_000151 C/C=C/C(O)C1C=CC2C(N1NC(=O)OC(C)(C)C)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H14 compound treatment 1191720.0 -44400.0 -0.74 1204680.0 -28500.0 -0.51 -0.889 -0.9837 3093386 BCB01_000152 CC(=CCC/C(=C/C(O)C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)/C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H15 compound treatment 1195520.0 -40600.0 -0.68 1215200.0 -18000.0 -0.32 -0.71 -0.9427 3001073 BCB01_000153 CN1C(=O)C2C=CC(C(O)C3CCC=CC3)N(NC(=O)OC(C)(C)C)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H16 compound treatment 1197480.0 -38700.0 -0.65 1207760.0 -25400.0 -0.46 -0.7816 -0.9857 3093387 BCB01_000154 Cc1ccccc1C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H17 compound treatment 1196720.0 -39400.0 -0.66 1194040.0 -39200.0 -0.71 -0.9653 -0.9994 3093388 BCB01_000155 COC(=O)c1ccc(o1)C(O)C2C=CC3C(N2NC(=O)OC(C)(C)C)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H18 compound treatment 1214440.0 -21700.0 -0.36 1193800.0 -39400.0 -0.71 -0.7587 -0.9516 3001076 BCB01_000156 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(I)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H19 compound treatment 1190840.0 -45300.0 -0.76 1201920.0 -31300.0 -0.56 -0.9345 -0.9893 3093389 BCB01_000157 CC(C(O)C1C=CC2C(N1NC(=O)OC(C)(C)C)C(=O)N(C)C2=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H20 compound treatment 1170680.0 -65500.0 -1.1 1178160.0 -55000.0 -0.99 -1.4758 -0.9988 3093390 BCB01_000158 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H21 compound treatment 1169640.0 -66500.0 -1.11 1192960.0 -40200.0 -0.72 -1.2996 -0.9784 3001078 BCB01_000159 CC(CC(O)C1C=CC2C(N1NC(=O)OC(C)(C)C)C(=O)N(C)C2=O)c3ccc(C)o3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H22 compound treatment 1158760.0 -77400.0 -1.29 1148840.0 -84400.0 -1.52 -1.9904 -0.9968 3093391 BCB01_000160 COc1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H23 mock treatment 1168680.0 -67500.0 -1.13 1180360.0 -52800.0 -0.95 -1.4714 -0.9964 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 H24 mock treatment 1174600.0 -61500.0 -1.03 1186120.0 -47100.0 -0.85 -1.328 -0.9954 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I01 mock treatment 1303680.0 67500.0 1.13 1307440.0 74200.0 1.34 1.745 0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I02 mock treatment 1287080.0 50900.0 0.85 1284680.0 51500.0 0.93 1.2587 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I03 compound treatment 1271400.0 35300.0 0.59 1278200.0 45000.0 0.81 0.9906 0.9878 3001079 BCB01_000161 CN1C(=O)C2C=CC(C(O)c3cccc(O)c3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I04 compound treatment 1276000.0 39900.0 0.67 1258880.0 25700.0 0.46 0.7988 0.984 3093392 BCB01_000162 CN1C(=O)C2C=CC(C(O)C3CCCCC3)N(Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I05 compound treatment 1273360.0 37200.0 0.62 1266480.0 33300.0 0.6 0.8644 0.9998 3093393 BCB01_000163 CN1C(=O)C2C=CC(C(O)C3CCC=CC3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I06 compound treatment 1267200.0 31100.0 0.52 1244440.0 11200.0 0.2 0.5107 0.9156 3001081 BCB01_000164 CN1C(=O)C2C=CC(C(O)C3=CC[C@H](CC3)C(=C)C)N(Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I07 compound treatment 1244560.0 8420.0 0.14 1254920.0 21700.0 0.39 0.3764 0.9048 3093394 BCB01_000165 CN1C(=O)C2C=CC(C(O)c3cn(C(=O)C)c4ccccc34)N(Nc5ccccc5)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I08 compound treatment 1249760.0 13600.0 0.23 1266160.0 33000.0 0.59 0.5811 0.9135 3093395 BCB01_000166 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I09 compound treatment 1261440.0 25300.0 0.42 1252600.0 19400.0 0.35 0.5465 0.9955 3001082 BCB01_000167 CCCCC(CC)C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I10 compound treatment 1244040.0 7900.0 0.13 1233280.0 81.9 0.0 0.0945 0.715 3093464 BCB01_000168 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccc(cc5[N+](=O)[O-])[N+](=O)[O-])C(=O)N(C)C4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I11 compound treatment 1250840.0 14700.0 0.25 1235680.0 2480.0 0.04 0.2056 0.8222 3001083 BCB01_000169 CC(C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I12 compound treatment 1268400.0 32300.0 0.54 1256520.0 23300.0 0.42 0.6788 0.9923 3093465 BCB01_000170 CN1C(=O)C2C=CC(C(O)c3cccn3C)N(Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I13 compound treatment 1245520.0 9380.0 0.16 1242240.0 9040.0 0.16 0.2262 0.9998 3093466 BCB01_000171 CC(CC(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C)C2=O)c4ccc(C)o4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I14 compound treatment 1244240.0 8100.0 0.14 1237240.0 4040.0 0.07 0.1473 0.9576 3001084 BCB01_000172 CN1C(=O)C2C=CC(C(O)c3ccccc3C)N(Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I15 compound treatment 1235160.0 -981.0 -0.02 1234000.0 802.0 0.01 -0.0014 -0.0636 3093467 BCB01_000173 CN1C(=O)C2C=CC(C(O)c3cccs3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I16 compound treatment 1210520.0 -25600.0 -0.43 1222200.0 -11000.0 -0.2 -0.4433 -0.9385 3093468 BCB01_000174 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I17 compound treatment 1207240.0 -28900.0 -0.48 1221440.0 -11800.0 -0.21 -0.4918 -0.9314 3001085 BCB01_000175 CN1C(=O)C2C=CC(C(O)Cc3ccccc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I18 compound treatment 1216120.0 -20000.0 -0.34 1218880.0 -14300.0 -0.26 -0.4193 -0.9917 3093469 BCB01_000176 C/C=C/C(O)C1C=CC2C(N1Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I19 compound treatment 1220520.0 -15600.0 -0.26 1233640.0 442.0 0.01 -0.1792 -0.6853 3001086 BCB01_000177 CN1C(=O)C2C=CC(C(O)C3=C[C@H]4C[C@@H](C3)C4(C)C)N(Nc5ccccc5)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I20 compound treatment 1202440.0 -33700.0 -0.56 1195400.0 -37800.0 -0.68 -0.8803 -0.9956 3093470 BCB01_000178 CN1C(=O)C2C=CC(C(O)C3=C[C@H]4C[C@@H](C3)C4(C)C)N(Nc5ccc(cc5[N+](=O)[O-])[N+](=O)[O-])C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I21 compound treatment 1181680.0 -54500.0 -0.91 1196840.0 -36400.0 -0.66 -1.1076 -0.9869 3001087 BCB01_000179 CN1C(=O)C2C=CC(C(O)c3ccc(Br)cc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I22 compound treatment 1182880.0 -53300.0 -0.89 1200040.0 -33200.0 -0.6 -1.0527 -0.9811 3093471 BCB01_000180 CN1C(=O)C2C=CC(C(O)COCc3ccccc3)N(Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I23 mock treatment 1160080.0 -76100.0 -1.27 1191480.0 -41700.0 -0.75 -1.4315 -0.9684 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 I24 mock treatment 1192920.0 -43200.0 -0.72 1175800.0 -57400.0 -1.03 -1.2427 -0.9847 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J01 mock treatment 1294840.0 58700.0 0.98 1299680.0 66500.0 1.2 1.5416 0.9951 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J02 mock treatment 1300560.0 64400.0 1.08 1291760.0 58600.0 1.06 1.5084 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J03 compound treatment 1275560.0 39400.0 0.66 1266000.0 32800.0 0.59 0.8843 0.9985 3093472 BCB01_000181 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J04 compound treatment 1211480.0 -24700.0 -0.41 1188120.0 -45100.0 -0.81 -0.8661 -0.9507 3001088 BCB01_000182 CN(C)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J05 compound treatment 1258040.0 21900.0 0.37 1262160.0 29000.0 0.52 0.6281 0.9851 3093473 BCB01_000183 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccc(I)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J06 compound treatment 1226920.0 -9220.0 -0.15 1234240.0 1040.0 0.02 -0.0958 -0.6165 3093474 BCB01_000184 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J07 compound treatment 1272760.0 36600.0 0.61 1265360.0 32200.0 0.58 0.8431 0.9996 3001089 BCB01_000185 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J08 compound treatment 1229840.0 -6300.0 -0.11 1221480.0 -11700.0 -0.21 -0.2238 -0.9485 3001153 BCB01_000186 OC(C1CCCCC1)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J09 compound treatment 1265200.0 29100.0 0.49 1258640.0 25400.0 0.46 0.668 0.9996 3001154 BCB01_000187 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J10 compound treatment 1223480.0 -12700.0 -0.21 1218880.0 -14300.0 -0.26 -0.3322 -0.9952 3001156 BCB01_000188 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J11 compound treatment 1247160.0 11000.0 0.18 1245080.0 11900.0 0.21 0.2818 0.9972 3001157 BCB01_000189 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J12 compound treatment 1183120.0 -53000.0 -0.89 1170680.0 -62500.0 -1.13 -1.4239 -0.993 3093475 BCB01_000190 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccco4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J13 compound treatment 1230600.0 -5540.0 -0.09 1235720.0 2520.0 0.05 -0.0334 -0.3238 3093476 BCB01_000191 CC(=O)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J14 compound treatment 1222280.0 -13900.0 -0.23 1214160.0 -19000.0 -0.34 -0.4066 -0.9819 3001159 BCB01_000192 CCCCC(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J15 compound treatment 1215920.0 -20200.0 -0.34 1221040.0 -12200.0 -0.22 -0.3942 -0.9778 3093477 BCB01_000193 OC(C1CCCCC1)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J16 compound treatment 1214720.0 -21400.0 -0.36 1193080.0 -40100.0 -0.72 -0.7646 -0.9476 3001160 BCB01_000194 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J17 compound treatment 1219320.0 -16800.0 -0.28 1229160.0 -4040.0 -0.07 -0.2505 -0.8616 3093478 BCB01_000195 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J18 compound treatment 1190160.0 -46000.0 -0.77 1208760.0 -24400.0 -0.44 -0.8554 -0.9649 3093479 BCB01_000196 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(F)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J19 compound treatment 1203560.0 -32600.0 -0.55 1206960.0 -26200.0 -0.47 -0.7198 -0.9975 3001161 BCB01_000197 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccco5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J20 compound treatment 1170560.0 -65600.0 -1.1 1179760.0 -53400.0 -0.96 -1.4568 -0.9979 3093480 BCB01_000198 COc1ccc(C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O)c5ccccc15 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J21 compound treatment 1157120.0 -79000.0 -1.32 1193120.0 -40100.0 -0.72 -1.4457 -0.9595 3093481 BCB01_000199 CCCCC(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J22 compound treatment 1182560.0 -53600.0 -0.9 1175840.0 -57400.0 -1.03 -1.3648 -0.9975 3001163 BCB01_000200 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J23 mock treatment 1174000.0 -62100.0 -1.04 1200760.0 -32400.0 -0.58 -1.1486 -0.9629 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 J24 mock treatment 1160000.0 -76100.0 -1.27 1174600.0 -58600.0 -1.06 -1.6475 -0.9956 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K01 mock treatment 1292600.0 56500.0 0.94 1281440.0 48200.0 0.87 1.2827 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K02 mock treatment 1291840.0 55700.0 0.93 1281760.0 48600.0 0.87 1.2778 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K03 compound treatment 1275400.0 39300.0 0.66 1273840.0 40600.0 0.73 0.9823 0.9985 3093482 BCB01_000201 CN1C(=O)C2C=CC(C(O)COCc3ccccc3)N(Nc4ccccc4)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K04 compound treatment 1283360.0 47200.0 0.79 1273680.0 40500.0 0.73 1.0745 0.9992 3001164 BCB01_000202 CN1C(=O)C2C=CC(C(O)c3ccccc3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K05 compound treatment 1247040.0 10900.0 0.18 1234840.0 1640.0 0.03 0.1499 0.8112 3093483 BCB01_000203 CN1C(=O)C2C=CC(C(O)/C=C(\C)/CCC=C(C)C)N(Nc3ccccc3)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K06 compound treatment 1268520.0 32400.0 0.54 1273680.0 40500.0 0.73 0.8989 0.9893 3093484 BCB01_000204 CN1C(=O)C2C=CC(C(O)c3ccc(I)cc3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K07 compound treatment 1267120.0 31000.0 0.52 1271600.0 38400.0 0.69 0.8558 0.9899 3000112 BCB01_000205 CN1C(=O)C2C=CC(C(O)C(C)(C)C)N(Nc3ccccc3)C2C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K08 compound treatment 1249520.0 13400.0 0.22 1246040.0 12800.0 0.23 0.3219 0.9999 3000114 BCB01_000206 COc1ccc(cc1)C(O)C2C=CC3C(N2N(c4ccccc4)c5ccccc5)C(=O)N(C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K09 compound treatment 1244760.0 8620.0 0.14 1244560.0 11400.0 0.2 0.2467 0.9853 3000115 BCB01_000207 CCCCC(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K10 compound treatment 1236360.0 219.0 0.0 1243600.0 10400.0 0.19 0.1351 0.7208 3000116 BCB01_000208 CN1C(=O)C2C=CC(C(O)C3CCCCC3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K11 compound treatment 1230360.0 -5780.0 -0.1 1230560.0 -2640.0 -0.05 -0.102 -0.9465 3000118 BCB01_000209 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(I)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K12 compound treatment 1236400.0 259.0 0.0 1232640.0 -558.0 -0.01 -0.004 -0.3694 3093485 BCB01_000210 CCCCC(O)C1C=CC2C(N1N(c3ccccc3)c4ccccc4)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K13 compound treatment 1208760.0 -27400.0 -0.46 1236320.0 3120.0 0.06 -0.2842 -0.6157 3093645 BCB01_000211 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K14 compound treatment 1241200.0 5060.0 0.08 1232360.0 -838.0 -0.02 0.0492 0.572 3000120 BCB01_000212 CN1C(=O)C2C=CC(C(O)c3ccc(F)cc3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K15 compound treatment 1219560.0 -16600.0 -0.28 1234280.0 1080.0 0.02 -0.1824 -0.6558 3093555 BCB01_000213 COc1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K16 compound treatment 1233360.0 -2780.0 -0.05 1228640.0 -4560.0 -0.08 -0.091 -0.9638 3093556 BCB01_000214 COc1ccc(C(O)C2C=CC3C(N2N(c4ccccc4)c5ccccc5)C(=O)N(C)C3=O)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K17 compound treatment 1227720.0 -8420.0 -0.14 1227640.0 -5560.0 -0.1 -0.1705 -0.986 3000122 BCB01_000215 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K18 compound treatment 1233400.0 -2740.0 -0.05 1235040.0 1840.0 0.03 -0.009 -0.1584 3093557 BCB01_000216 CN1C(=O)C2C=CC(C(O)c3ccccn3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K19 compound treatment 1183040.0 -53100.0 -0.89 1209200.0 -24000.0 -0.43 -0.9341 -0.9452 3000123 BCB01_000217 OC(C#Cc1ccccc1)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K20 compound treatment 1224480.0 -11700.0 -0.2 1214480.0 -18700.0 -0.34 -0.3765 -0.9662 3093558 BCB01_000218 CN1C(=O)C2C=CC(C(O)c3ccc(s3)c4ccccc4)N(C2C1=O)N(c5ccccc5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K21 compound treatment 1185320.0 -50800.0 -0.85 1182760.0 -50400.0 -0.91 -1.244 -0.9995 3093559 BCB01_000219 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K22 compound treatment 1207400.0 -28700.0 -0.48 1212120.0 -21100.0 -0.38 -0.6086 -0.9932 3000124 BCB01_000220 CN1C(=O)C2C=CC(C(O)c3ccccc3C)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K23 mock treatment 1182640.0 -53500.0 -0.9 1195760.0 -37400.0 -0.67 -1.11 -0.9903 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 K24 mock treatment 1173160.0 -63000.0 -1.05 1185840.0 -47400.0 -0.85 -1.3486 -0.9945 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L01 mock treatment 1280960.0 44800.0 0.75 1297120.0 63900.0 1.15 1.3447 0.9784 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L02 mock treatment 1280160.0 44000.0 0.74 1271280.0 38100.0 0.69 1.006 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L03 compound treatment 1267600.0 31500.0 0.53 1256960.0 23800.0 0.43 0.675 0.9947 3093560 BCB01_000221 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L04 compound treatment 1245520.0 9380.0 0.16 1243360.0 10200.0 0.18 0.2404 0.9971 3093561 BCB01_000222 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccccn5)C(=O)NC4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L05 compound treatment 1263600.0 27500.0 0.46 1258440.0 25200.0 0.45 0.6465 1.0 3000127 BCB01_000223 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccc(F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L06 compound treatment 1244360.0 8220.0 0.14 1245160.0 12000.0 0.22 0.2497 0.9765 3093562 BCB01_000224 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L07 compound treatment 1199760.0 -36400.0 -0.61 1205280.0 -27900.0 -0.5 -0.7862 -0.9955 3093563 BCB01_000225 COc1ccc(C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L08 compound treatment 1226920.0 -9220.0 -0.15 1243320.0 10100.0 0.18 0.0198 0.0831 3000128 BCB01_000226 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L09 compound treatment 1247200.0 11100.0 0.19 1245640.0 12400.0 0.22 0.2894 0.9955 3093564 BCB01_000227 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L10 compound treatment 1222440.0 -13700.0 -0.23 1230680.0 -2520.0 -0.05 -0.1942 -0.8309 3000129 BCB01_000228 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4c(F)cccc4Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L11 compound treatment 1238920.0 2780.0 0.05 1245400.0 12200.0 0.22 0.1883 0.8381 3093565 BCB01_000229 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccc(C#N)cc5)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L12 compound treatment 1189280.0 -46900.0 -0.78 1209200.0 -24000.0 -0.43 -0.8602 -0.9606 3093566 BCB01_000230 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(s4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L13 compound treatment 1210840.0 -25300.0 -0.42 1215960.0 -17200.0 -0.31 -0.519 -0.9884 3000131 BCB01_000231 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L14 compound treatment 1181320.0 -54800.0 -0.92 1173320.0 -59900.0 -1.08 -1.4116 -0.9967 3093567 BCB01_000232 Cn1cccc1C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L15 compound treatment 1219080.0 -17100.0 -0.29 1208720.0 -24500.0 -0.44 -0.5137 -0.9778 3093568 BCB01_000233 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L16 compound treatment 1175440.0 -60700.0 -1.02 1167160.0 -66000.0 -1.19 -1.5596 -0.9969 3000133 BCB01_000234 Cc1cc(C)c(C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O)c(C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L17 compound treatment 1205160.0 -31000.0 -0.52 1209320.0 -23900.0 -0.43 -0.6708 -0.9957 3093569 BCB01_000235 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5c(F)cccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L18 compound treatment 1207080.0 -29100.0 -0.49 1198000.0 -35200.0 -0.63 -0.7923 -0.9914 3000205 BCB01_000236 Cc1ccccc1C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L19 compound treatment 1202520.0 -33600.0 -0.56 1205520.0 -27700.0 -0.5 -0.7505 -0.9982 3000206 BCB01_000237 Cc1cc(C)c(C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5)c(C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L20 compound treatment 1193520.0 -42600.0 -0.71 1188760.0 -44400.0 -0.8 -1.0705 -0.9983 3000207 BCB01_000238 OC(/C=C/c1ccc(cc1)[N+](=O)[O-])C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L21 compound treatment 1177920.0 -58200.0 -0.97 1182960.0 -50200.0 -0.91 -1.329 -0.9993 3000208 BCB01_000239 Cc1ccccc1C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L22 compound treatment 1159840.0 -76300.0 -1.28 1143840.0 -89400.0 -1.61 -2.0413 -0.9934 3093570 BCB01_000240 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3Nc5ccccn5)C(=O)NC4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L23 mock treatment 1172800.0 -63300.0 -1.06 1166120.0 -67100.0 -1.21 -1.6041 -0.9979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 L24 mock treatment 1183400.0 -52700.0 -0.88 1187880.0 -45300.0 -0.82 -1.2014 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M01 mock treatment 1283080.0 46900.0 0.79 1287120.0 53900.0 0.97 1.2424 0.9944 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M02 mock treatment 1295640.0 59500.0 1.0 1292120.0 58900.0 1.06 1.4547 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M03 compound treatment 1280400.0 44300.0 0.74 1275280.0 42100.0 0.76 1.0598 0.9999 3000209 BCB01_000241 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccco5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M04 compound treatment 1289280.0 53100.0 0.89 1290440.0 57200.0 1.03 1.3581 0.9973 3093571 BCB01_000242 C/C=C/C(O)C1C=CC2C(N1N(c3ccccc3)c4ccccc4)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M05 compound treatment 1253840.0 17700.0 0.3 1251160.0 18000.0 0.32 0.4383 0.999 3093572 BCB01_000243 CCCCC(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M06 compound treatment 1257000.0 20900.0 0.35 1271440.0 38200.0 0.69 0.734 0.9503 3000211 BCB01_000244 CC(C)C(O)C1C=CC2C(N1N(c3ccccc3)c4ccccc4)C(=O)N(C)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M07 compound treatment 1240720.0 4580.0 0.08 1262040.0 28800.0 0.52 0.4216 0.8027 3093573 BCB01_000245 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M08 compound treatment 1254040.0 17900.0 0.3 1258080.0 24900.0 0.45 0.5288 0.9808 3093574 BCB01_000246 CN1C(=O)C2C=CC(C(O)C3CCC=CC3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M09 compound treatment 1239920.0 3780.0 0.06 1242600.0 9400.0 0.17 0.1645 0.9098 3000213 BCB01_000247 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M10 compound treatment 1229720.0 -6420.0 -0.11 1220560.0 -12600.0 -0.23 -0.237 -0.9413 3093575 BCB01_000248 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccccc5F)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M11 compound treatment 1200000.0 -36100.0 -0.6 1219880.0 -13300.0 -0.24 -0.5973 -0.918 3000215 BCB01_000249 COc1ccc(C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M12 compound treatment 1206000.0 -30100.0 -0.5 1239800.0 6600.0 0.12 -0.2726 -0.5259 3093576 BCB01_000250 CC(C(O)C1C=CC2C(N1N(c3ccccc3)c4ccccc4)C(=O)N(C)C2=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M13 compound treatment 1215840.0 -20300.0 -0.34 1234080.0 882.0 0.02 -0.229 -0.6733 3093646 BCB01_000251 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M14 compound treatment 1216200.0 -19900.0 -0.33 1197000.0 -36200.0 -0.65 -0.6971 -0.9516 3000219 BCB01_000252 CN1C(=O)C2C=CC(C(O)c3cccs3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M15 compound treatment 1209280.0 -26900.0 -0.45 1225640.0 -7560.0 -0.14 -0.4141 -0.8817 3093647 BCB01_000253 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccccc5)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M16 compound treatment 1214080.0 -22100.0 -0.37 1222520.0 -10700.0 -0.19 -0.3971 -0.9538 3000221 BCB01_000254 CN1C(=O)C2C=CC(C(O)Cc3ccccc3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M17 compound treatment 1195480.0 -40700.0 -0.68 1186240.0 -47000.0 -0.85 -1.0794 -0.9942 3093648 BCB01_000255 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccccn5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M18 compound treatment 1218200.0 -17900.0 -0.3 1211040.0 -22200.0 -0.4 -0.4946 -0.9901 3093649 BCB01_000256 CN1C(=O)C2C=CC(C(O)c3ccc(Br)cc3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M19 compound treatment 1175080.0 -61100.0 -1.02 1199640.0 -33600.0 -0.6 -1.1501 -0.9686 3000223 BCB01_000257 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M20 compound treatment 1181240.0 -54900.0 -0.92 1201200.0 -32000.0 -0.58 -1.0573 -0.9748 3093650 BCB01_000258 CN1C(=O)C2C=CC(C(O)COCc3ccccc3)N(C2C1=O)N(c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M21 compound treatment 1160120.0 -76000.0 -1.27 1188160.0 -45000.0 -0.81 -1.4734 -0.9764 3093651 BCB01_000259 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M22 compound treatment 1147640.0 -88500.0 -1.48 1155160.0 -78000.0 -1.41 -2.0415 -0.9997 3000225 BCB01_000260 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccccc4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M23 mock treatment 1161120.0 -75000.0 -1.26 1181720.0 -51500.0 -0.93 -1.5436 -0.9889 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 M24 mock treatment 1154480.0 -81700.0 -1.37 1175120.0 -58100.0 -1.05 -1.7062 -0.9913 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N01 mock treatment 1276400.0 40300.0 0.67 1284920.0 51700.0 0.93 1.1353 0.9873 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N02 mock treatment 1281960.0 45800.0 0.77 1272840.0 39600.0 0.71 1.0472 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N03 compound treatment 1255440.0 19300.0 0.32 1256320.0 23100.0 0.42 0.5229 0.9921 3093652 BCB01_000261 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3Nc5ccc(C#N)cc5)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N04 compound treatment 1233480.0 -2660.0 -0.04 1246280.0 13100.0 0.24 0.1352 0.5635 3093653 BCB01_000262 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4cccc5ccccc45 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N05 compound treatment 1249640.0 13500.0 0.23 1260880.0 27700.0 0.5 0.5124 0.9359 3000227 BCB01_000263 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5cccc6ccccc56 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N06 compound treatment 1231440.0 -4700.0 -0.08 1234200.0 1000.0 0.02 -0.0429 -0.531 3093654 BCB01_000264 C/C=C/C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N07 compound treatment 1229520.0 -6620.0 -0.11 1234720.0 1520.0 0.03 -0.059 -0.5165 3093655 BCB01_000265 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5c(F)cccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N08 compound treatment 1232600.0 -3540.0 -0.06 1230280.0 -2920.0 -0.05 -0.0791 -0.9982 3000229 BCB01_000266 CCC(CC)C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N09 compound treatment 1218560.0 -17600.0 -0.29 1228320.0 -4880.0 -0.09 -0.2702 -0.8799 3093656 BCB01_000267 CCC(CC)C(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N10 compound treatment 1223880.0 -12300.0 -0.21 1216160.0 -17000.0 -0.31 -0.3622 -0.9808 3000231 BCB01_000268 CC(C)C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N11 compound treatment 1198760.0 -37400.0 -0.63 1224360.0 -8840.0 -0.16 -0.5549 -0.8597 3093657 BCB01_000269 CC(C)C(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N12 compound treatment 1188040.0 -48100.0 -0.8 1189320.0 -43900.0 -0.79 -1.1282 -1.0 3000297 BCB01_000270 OC(C1CCC=CC1)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N13 compound treatment 1174440.0 -61700.0 -1.03 1192880.0 -40300.0 -0.73 -1.2438 -0.9852 3000298 BCB01_000271 OB(O)c1ccc(cc1)C(O)C2C=CC3CN(C(=O)C3N2Nc4ccc(C#N)cc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N14 compound treatment 1170320.0 -65800.0 -1.1 1188000.0 -45200.0 -0.81 -1.3547 -0.989 3000299 BCB01_000272 CC(=O)n1cc(C(O)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O)c5ccccc15 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N15 compound treatment 1193080.0 -43100.0 -0.72 1206320.0 -26900.0 -0.48 -0.852 -0.9813 3093658 BCB01_000273 OC(C1CCC=CC1)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N16 compound treatment 1169600.0 -66500.0 -1.11 1173360.0 -59800.0 -1.08 -1.5497 -0.9999 3093659 BCB01_000274 CCCCC(CC)C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N17 compound treatment 1187600.0 -48500.0 -0.81 1200960.0 -32200.0 -0.58 -0.9851 -0.9865 3000301 BCB01_000275 CC(=O)n1cc(C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N18 compound treatment 1172440.0 -63700.0 -1.07 1163520.0 -69700.0 -1.26 -1.6415 -0.9967 3093660 BCB01_000276 CC(C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N19 compound treatment 1171120.0 -65000.0 -1.09 1190040.0 -43200.0 -0.78 -1.3192 -0.9864 3093661 BCB01_000277 COC(=O)c1ccc(o1)C(O)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N20 compound treatment 1152320.0 -83800.0 -1.4 1139360.0 -93800.0 -1.69 -2.1874 -0.9957 3000302 BCB01_000278 CC(CC(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(C)o4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N21 compound treatment 1151440.0 -84700.0 -1.42 1161560.0 -71600.0 -1.29 -1.915 -0.9989 3093662 BCB01_000279 CCCCC(CC)C(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N22 compound treatment 1158960.0 -77200.0 -1.29 1173360.0 -59800.0 -1.08 -1.6756 -0.996 3093663 BCB01_000280 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4cccs4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N23 mock treatment 1171720.0 -64400.0 -1.08 1173840.0 -59400.0 -1.07 -1.5185 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 N24 mock treatment 1175080.0 -61100.0 -1.02 1181320.0 -51900.0 -0.93 -1.3835 -0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O01 mock treatment 1284920.0 48800.0 0.82 1283000.0 49800.0 0.9 1.2117 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O02 mock treatment 1302720.0 66600.0 1.11 1281960.0 48800.0 0.88 1.4091 0.9931 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O03 compound treatment 1258160.0 22000.0 0.37 1246400.0 13200.0 0.24 0.4287 0.9776 3000303 BCB01_000281 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5c(F)cccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O04 compound treatment 1203000.0 -33100.0 -0.55 1189960.0 -43200.0 -0.78 -0.943 -0.9861 3093664 BCB01_000282 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccc(cc4)N(C)C)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O05 compound treatment 1251040.0 14900.0 0.25 1234400.0 1200.0 0.02 0.1916 0.7656 3093665 BCB01_000283 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5ccc(s5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O06 compound treatment 1228720.0 -7420.0 -0.12 1214760.0 -18400.0 -0.33 -0.3227 -0.9099 3000304 BCB01_000284 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccccn5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O07 compound treatment 1223560.0 -12600.0 -0.21 1198640.0 -34600.0 -0.62 -0.5891 -0.8963 3093666 BCB01_000285 Cn1cccc1C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O08 compound treatment 1193160.0 -43000.0 -0.72 1162800.0 -70400.0 -1.27 -1.4055 -0.9639 3093667 BCB01_000286 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccc(cc4)C(=O)C)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O09 compound treatment 1210800.0 -25300.0 -0.42 1210920.0 -22300.0 -0.4 -0.5837 -0.9996 3000307 BCB01_000287 Cc1cc(C)c(C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5)c(C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O10 compound treatment 1183840.0 -52300.0 -0.88 1174800.0 -58400.0 -1.05 -1.3629 -0.9958 3093736 BCB01_000288 CC(C)c1ccc(NN2C3C(C=CC2C(O)C4CCCCC4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O11 compound treatment 1200520.0 -35600.0 -0.6 1202080.0 -31100.0 -0.56 -0.818 -0.9995 3000308 BCB01_000289 Cc1ccccc1C(O)C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O12 compound treatment 1183200.0 -52900.0 -0.89 1181360.0 -51800.0 -0.93 -1.2869 -0.9997 3093737 BCB01_000290 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccco4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O13 compound treatment 1163600.0 -72500.0 -1.21 1171400.0 -61800.0 -1.11 -1.6457 -0.9991 3093738 BCB01_000291 OC(/C=C/c1ccc(cc1)[N+](=O)[O-])C2C=CC3C(N2Nc4ccccc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O14 compound treatment 1180520.0 -55600.0 -0.93 1170120.0 -63100.0 -1.14 -1.4618 -0.9951 3000310 BCB01_000292 CCCCC(O)C1C=CC2C(N1Nc3ccc(cc3)C(C)C)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O15 compound treatment 1197160.0 -39000.0 -0.65 1187120.0 -46100.0 -0.83 -1.0483 -0.9929 3093739 BCB01_000293 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3Nc5ccccc5)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O16 compound treatment 1151560.0 -84600.0 -1.42 1153680.0 -79500.0 -1.43 -2.0139 -1.0 3000311 BCB01_000294 CC(C)c1ccc(NN2C3C(C=CC2C(O)c4ccc(F)cc4)C(=O)N(C3=O)c5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O17 compound treatment 1185040.0 -51100.0 -0.86 1197880.0 -35300.0 -0.64 -1.0546 -0.9894 3093740 BCB01_000295 OC(C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4)c5cccc6ccccc56 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O18 compound treatment 1167120.0 -69000.0 -1.16 1167640.0 -65600.0 -1.18 -1.6519 -0.9999 3093741 BCB01_000296 COc1ccc(C(O)C2C=CC3C(N2Nc4ccc(cc4)C(C)C)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O19 compound treatment 1139000.0 -97100.0 -1.63 1149400.0 -83800.0 -1.51 -2.2171 -0.9993 3000313 BCB01_000297 C/C=C/C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O20 compound treatment 1160440.0 -75700.0 -1.27 1169320.0 -63900.0 -1.15 -1.7096 -0.9989 3093742 BCB01_000298 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2Nc4ccc(cc4)C(C)C)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O21 compound treatment 1144800.0 -91300.0 -1.53 1168560.0 -64600.0 -1.16 -1.9043 -0.991 3000315 BCB01_000299 CCC(CC)C(O)C1C=CC2C(N1Nc3ccccc3)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O22 compound treatment 1157400.0 -78700.0 -1.32 1152440.0 -80800.0 -1.46 -1.9606 -0.9988 3093743 BCB01_000300 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccc(cc5)C(C)C)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O23 mock treatment 1137960.0 -98200.0 -1.64 1149840.0 -83400.0 -1.5 -2.2238 -0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 O24 mock treatment 1167880.0 -68300.0 -1.14 1180120.0 -53100.0 -0.96 -1.484 -0.9961 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P01 mock treatment 1270200.0 34100.0 0.57 1270520.0 37300.0 0.67 0.8785 0.9966 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P02 mock treatment 1261440.0 25300.0 0.42 1257520.0 24300.0 0.44 0.6092 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P03 compound treatment 1221440.0 -14700.0 -0.25 1213600.0 -19600.0 -0.35 -0.4236 -0.9844 3000135 BCB01_000301 CC(C(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P04 compound treatment 1216240.0 -19900.0 -0.33 1210640.0 -22600.0 -0.41 -0.5229 -0.9951 3000137 BCB01_000302 OC(Cc1ccccc1)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P05 compound treatment 1194880.0 -41300.0 -0.69 1193600.0 -39600.0 -0.71 -0.9927 -0.9999 3000138 BCB01_000303 CC(CC(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccc(C)o5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P06 compound treatment 1184080.0 -52100.0 -0.87 1183680.0 -49500.0 -0.89 -1.2469 -0.9999 3000139 BCB01_000304 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(C#N)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P07 compound treatment 1210240.0 -25900.0 -0.43 1211000.0 -22200.0 -0.4 -0.5893 -0.9992 3093744 BCB01_000305 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5cccs5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P08 compound treatment 1208920.0 -27200.0 -0.46 1202320.0 -30900.0 -0.56 -0.7155 -0.9951 3000141 BCB01_000306 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc5OCOc5c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P09 compound treatment 1219560.0 -16600.0 -0.28 1208040.0 -25200.0 -0.45 -0.5167 -0.9723 3093745 BCB01_000307 OC(C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)c5ccc(Br)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P10 compound treatment 1182400.0 -53700.0 -0.9 1163760.0 -69400.0 -1.25 -1.5206 -0.9869 3093746 BCB01_000308 OC(C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)c4ccc(Br)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P11 compound treatment 1195480.0 -40700.0 -0.68 1194040.0 -39200.0 -0.71 -0.98 -0.9998 3000143 BCB01_000309 OC(CCc1ccccc1)C2C=CC3C(N2Nc4ccc(C#N)cc4)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P12 compound treatment 1195120.0 -41000.0 -0.69 1182920.0 -50300.0 -0.91 -1.126 -0.9906 3093747 BCB01_000310 OC(CCc1ccccc1)C2C=CC3C(N2Nc4ccccn4)C(=O)NC3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P13 compound treatment 1177760.0 -58400.0 -0.98 1184160.0 -49000.0 -0.88 -1.3156 -0.9987 3093748 BCB01_000311 CC(=CCC/C=C(\C)/C(O)C1C=CC2C(N1Nc3ccc(C#N)cc3)C(=O)N(C2=O)c4ccccc4)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P14 compound treatment 1194920.0 -41200.0 -0.69 1179560.0 -53600.0 -0.97 -1.1711 -0.9863 3000145 BCB01_000312 CC(=CCC/C(=C/C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O)/C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P15 compound treatment 1176320.0 -59800.0 -1.0 1175720.0 -57500.0 -1.04 -1.4401 -0.9999 3093749 BCB01_000313 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P16 compound treatment 1179040.0 -57100.0 -0.96 1175600.0 -57600.0 -1.04 -1.4095 -0.9992 3093750 BCB01_000314 OCC(O)C(O)C1C=CC2C(N1Nc3ccccn3)C(=O)NC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P17 compound treatment 1186200.0 -49900.0 -0.84 1175560.0 -57600.0 -1.04 -1.3253 -0.9942 3000147 BCB01_000315 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc(I)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P18 compound treatment 1181240.0 -54900.0 -0.92 1162360.0 -70800.0 -1.28 -1.5521 -0.987 3093751 BCB01_000316 OC(C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P19 compound treatment 1155520.0 -80600.0 -1.35 1165960.0 -67200.0 -1.21 -1.8106 -0.9986 3093752 BCB01_000317 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P20 compound treatment 1175480.0 -60700.0 -1.02 1159440.0 -73800.0 -1.33 -1.6575 -0.9912 3000149 BCB01_000318 CN(C)c1ccc(cc1)C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P21 compound treatment 1132360.0 -104000.0 -1.74 1146080.0 -87100.0 -1.57 -2.3379 -0.9987 3093752 BCB01_000319 OC(C1C=CC2C(N1Nc3ccc(Cl)cc3Cl)C(=O)NC2=O)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P22 compound treatment 1141880.0 -94300.0 -1.58 1150440.0 -82800.0 -1.49 -2.1697 -0.9996 3093753 BCB01_000320 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P23 mock treatment 1158280.0 -77900.0 -1.3 1172960.0 -60200.0 -1.09 -1.6888 -0.9959 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2000 P24 mock treatment 1173360.0 -62800.0 -1.05 1174080.0 -59100.0 -1.07 -1.4961 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A01 compound treatment 1225360.0 38600.0 0.65 1223160.0 33500.0 0.6 0.8831 0.9994 3000745 BCB02_000001 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5cccc(O)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A02 compound treatment 1271120.0 84300.0 1.41 1275160.0 85500.0 1.54 2.0871 0.999 3000746 BCB02_000002 CC(C)OC(=O)C1=CCC(O1)c2cccc(Cl)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A03 compound treatment 1250720.0 63900.0 1.07 1250920.0 61300.0 1.1 1.5369 0.9999 3000747 BCB02_000003 OC(C1CCCCC1)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A04 compound treatment 1257120.0 70300.0 1.18 1257480.0 67800.0 1.22 1.6962 0.9998 3000748 BCB02_000004 CCOC(=O)C1=CCC(O1)c2cccc(Cl)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A05 compound treatment 1249040.0 62200.0 1.04 1263160.0 73500.0 1.32 1.6729 0.9929 3000749 BCB02_000005 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A06 compound treatment 1262880.0 76100.0 1.27 1255840.0 66200.0 1.19 1.7434 0.9995 3000750 BCB02_000006 COC(=O)C1=CCC(O1)c2cccc(Cl)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A07 compound treatment 1238600.0 51800.0 0.87 1257440.0 67800.0 1.22 1.4765 0.9859 3093754 BCB02_000007 CCCCC(O)C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A08 compound treatment 1170000.0 -16800.0 -0.28 1163480.0 -26200.0 -0.47 -0.5323 -0.9695 2065163 BCB02_000008 CCOC(=O)/C=C/c1ccccc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A09 compound treatment 1224800.0 38000.0 0.64 1224400.0 34700.0 0.63 0.8923 1.0 3093755 BCB02_000009 CCCCCCCCCCC(O)C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A10 compound treatment 1219600.0 32800.0 0.55 1214240.0 24600.0 0.44 0.7013 0.9944 3000752 BCB02_000010 CCOC(=O)/C=C/c1cc(F)ccc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A11 compound treatment 1234880.0 48100.0 0.8 1242160.0 52500.0 0.95 1.2378 0.9968 3093756 BCB02_000011 OC(C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5ccc(F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A12 compound treatment 1231720.0 44900.0 0.75 1256560.0 66900.0 1.21 1.3839 0.9742 3000753 BCB02_000012 CCOC(=O)/C=C/c1cc(ccc1O)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A13 compound treatment 1225400.0 38600.0 0.65 1233000.0 43300.0 0.78 1.009 0.9955 3093757 BCB02_000013 COc1ccc(C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A14 compound treatment 474440.0 -712000.0 -11.92 469320.0 -720000.0 -12.98 -17.6066 -0.9991 3000754 BCB02_000014 CCOC(=O)/C=C/c1cccc(OC)c1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A15 compound treatment 1206040.0 19200.0 0.32 1222560.0 32900.0 0.59 0.6469 0.9588 3093824 BCB02_000015 COc1cc(OC)c(cc1Br)C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A16 compound treatment 810240.0 -377000.0 -6.3 814200.0 -375000.0 -6.76 -9.2392 -0.9994 3000755 BCB02_000016 CCOC(=O)/C=C/c1cccc(C)c1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A17 mock treatment 1199960.0 13200.0 0.22 1203360.0 13700.0 0.25 0.3303 0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A18 mock treatment 1211880.0 25100.0 0.42 1220560.0 30900.0 0.56 0.6905 0.9903 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A19 mock treatment 1199560.0 12800.0 0.21 1214880.0 25200.0 0.45 0.4723 0.9406 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A20 mock treatment 1196520.0 9720.0 0.16 1210080.0 20400.0 0.37 0.3752 0.9326 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A21 mock treatment 1180280.0 -6520.0 -0.11 1195120.0 5470.0 0.1 -0.0076 -0.0514 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A22 mock treatment 1192880.0 6080.0 0.1 1203880.0 14200.0 0.26 0.2531 0.918 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A23 mock treatment 1186160.0 -643.0 -0.01 1181640.0 -8010.0 -0.14 -0.1097 -0.7577 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 A24 mock treatment 1190920.0 4120.0 0.07 1204680.0 15000.0 0.27 0.2401 0.8596 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B01 compound treatment 1258560.0 71800.0 1.2 1262000.0 72300.0 1.3 1.7708 0.9992 3093825 BCB02_000017 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3n5cnnc5)C(=O)N(Cc6ccccc6)C4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B02 compound treatment 1263920.0 77100.0 1.29 1256880.0 67200.0 1.21 1.769 0.9995 3000756 BCB02_000018 CCOC(=O)C1=CCC(N(CCN2CC(=CCC2c3cc4ccccc4[nH]3)C(=O)OCC)C1)c5cc6ccccc6[nH]5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B03 compound treatment 1248800.0 62000.0 1.04 1247040.0 57400.0 1.03 1.4647 1.0 3093826 BCB02_000019 OC(C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B04 compound treatment 1260240.0 73400.0 1.23 1247040.0 57400.0 1.03 1.6001 0.9963 3000757 BCB02_000020 CC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B05 compound treatment 1264280.0 77500.0 1.3 1256840.0 67200.0 1.21 1.7727 0.9994 3093827 BCB02_000021 OC(C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5ccc(s5)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B06 compound treatment 1262240.0 75400.0 1.26 1267080.0 77400.0 1.39 1.8791 0.9988 3093828 BCB02_000022 Cc1ccc(cc1)[C@@H]2C[C@@H](Sc3ccccc3)[C@@H](CN2S(=O)(=O)c4ccc(C)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B07 compound treatment 1240880.0 54100.0 0.9 1258600.0 68900.0 1.24 1.5183 0.9879 3000758 BCB02_000023 CC(C(O)C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B08 compound treatment 1271520.0 84700.0 1.42 1240040.0 50400.0 0.91 1.6444 0.9768 3093829 BCB02_000024 Cc1ccc(cc1)C2CC=C(CN2S(=O)(=O)c3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B09 compound treatment 1215920.0 29100.0 0.49 1224240.0 34600.0 0.62 0.7852 0.9926 3000759 BCB02_000025 CC(CC(O)C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5ccc(C)o5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B10 compound treatment 1240720.0 53900.0 0.9 1259000.0 69300.0 1.25 1.5215 0.9872 3093830 BCB02_000026 Cc1ccc(cc1)S(=O)(=O)N2CC(=CCC2c3ccccc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B11 compound treatment 1227760.0 41000.0 0.69 1223920.0 34300.0 0.62 0.9212 0.9986 3093831 BCB02_000027 OC(Cc1ccccc1)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B12 compound treatment 1237360.0 50600.0 0.85 1246800.0 57100.0 1.03 1.3263 0.9952 3000760 BCB02_000028 Cc1ccc(cc1)[C@@H]2CC=C([C@@H](N2S(=O)(=O)c3ccc(C)cc3)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B13 compound treatment 1215800.0 29000.0 0.49 1211200.0 21500.0 0.39 0.6176 0.9939 3093832 BCB02_000029 OC(C1CCCCC1)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B14 compound treatment 1212600.0 25800.0 0.43 1231440.0 41800.0 0.75 0.8376 0.9652 3093833 BCB02_000030 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](CC=C([C@@H]2c3ccccc3)C(=O)O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B15 compound treatment 1196920.0 10100.0 0.17 1192640.0 2990.0 0.05 0.1578 0.8881 3000761 BCB02_000031 CC(=C)[C@H]1CCC(=CC1)C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B16 compound treatment 1207640.0 20800.0 0.35 1221600.0 31900.0 0.58 0.6536 0.9712 3093834 BCB02_000032 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](CC=C([C@@H]2c3ccccc3)C(=O)O)c4ccc(C#N)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B17 mock treatment 1186200.0 -603.0 -0.01 1206560.0 16900.0 0.3 0.2082 0.6833 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B18 mock treatment 1200600.0 13800.0 0.23 1215560.0 25900.0 0.47 0.4933 0.9473 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B19 mock treatment 1177960.0 -8840.0 -0.15 1195160.0 5510.0 0.1 -0.0345 -0.1936 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B20 mock treatment 1181840.0 -4960.0 -0.08 1192240.0 2590.0 0.05 -0.0258 -0.2708 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B21 mock treatment 1164720.0 -22100.0 -0.37 1183160.0 -6490.0 -0.12 -0.344 -0.8876 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B22 mock treatment 1176480.0 -10300.0 -0.17 1197680.0 8030.0 0.14 -0.0199 -0.0884 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B23 mock treatment 1159880.0 -26900.0 -0.45 1168760.0 -20900.0 -0.38 -0.5848 -0.996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 B24 mock treatment 1176360.0 -10400.0 -0.17 1194880.0 5230.0 0.09 -0.057 -0.2871 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C01 compound treatment 1244120.0 57300.0 0.96 1241720.0 52100.0 0.94 1.3416 0.9999 3093835 BCB02_000033 CC(=O)n1cc(C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C02 compound treatment 1254320.0 67500.0 1.13 1245120.0 55500.0 1.0 1.5056 0.9981 3000762 BCB02_000034 CCOC(=O)/C=C/c1ccccc1OC(=O)C#CC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C03 compound treatment 1243280.0 56500.0 0.95 1246080.0 56400.0 1.02 1.3872 0.9993 3000763 BCB02_000035 Cc1ccccc1C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C04 compound treatment 1251920.0 65100.0 1.09 1233000.0 43300.0 0.78 1.3228 0.9867 3093836 BCB02_000036 CCOC(=O)[C@H]1CC=C2[C@@H]1c3ccccc3OC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C05 compound treatment 1227400.0 40600.0 0.68 1220360.0 30700.0 0.55 0.8716 0.9948 3093837 BCB02_000037 OC(/C=C/c1ccc(cc1)[N+](=O)[O-])C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C06 compound treatment 1240680.0 53900.0 0.9 1213080.0 23400.0 0.42 0.936 0.9402 3000764 BCB02_000038 CCOC(=O)[C@H]1CC=C2[C@@H]1c3cc(Br)ccc3OC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C07 compound treatment 1231840.0 45000.0 0.75 1226720.0 37100.0 0.67 1.0051 0.9982 3093838 BCB02_000039 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3n5cnnc5)C(=O)N(Cc6ccccc6)C4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C08 compound treatment 1179480.0 -7320.0 -0.12 1165840.0 -23800.0 -0.43 -0.39 -0.8741 3000765 BCB02_000040 CCOC(=O)/C=C/c1cc(Br)ccc1OC(=O)C#CC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C09 compound treatment 1229320.0 42500.0 0.71 1233400.0 43700.0 0.79 1.0604 0.9987 3093839 BCB02_000041 OC(C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5cccc6ccccc56 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C10 compound treatment 1086240.0 -101000.0 -1.68 1095640.0 -94000.0 -1.69 -2.3877 -1.0 3000766 BCB02_000042 O=c1oc2ccccc2cc1C#C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C11 compound treatment 1224440.0 37600.0 0.63 1228000.0 38300.0 0.69 0.9339 0.9989 3093840 BCB02_000043 OC(C1CCC=CC1)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C12 compound treatment 1236880.0 50100.0 0.84 1233600.0 43900.0 0.79 1.1524 0.9996 3000767 BCB02_000044 Cn1c2C3NC(C(=O)c2c4ccccc14)C(C)(C=C3)C(=O)OCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C13 compound treatment 1220080.0 33300.0 0.56 1213880.0 24200.0 0.44 0.7024 0.9927 3093841 BCB02_000045 CC(=O)n1cc(C(O)C2C=CC3C(N2n4cnnc4)C(=O)N(Cc5ccccc5)C3=O)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C14 compound treatment 1225360.0 38600.0 0.65 1224080.0 34400.0 0.62 0.8948 0.9998 3000768 BCB02_000046 [O-][N+](=O)c1ccccc1S(=O)(=O)N2C3CC=C(C2C(=O)c4c3[nH]c5ccccc45)C(=O)OCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C15 compound treatment 1212720.0 25900.0 0.43 1225080.0 35400.0 0.64 0.758 0.9823 3093842 BCB02_000047 CCCCC(CC)C(O)C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C16 compound treatment 1206520.0 19700.0 0.33 1197360.0 7710.0 0.14 0.3315 0.926 3093843 BCB02_000048 CCOC(=O)C1=CC[C@@H]2[C@H]1C(=O)N(C2=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C17 mock treatment 1213560.0 26800.0 0.45 1222320.0 32700.0 0.59 0.7328 0.9909 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C18 mock treatment 1195320.0 8520.0 0.14 1212840.0 23200.0 0.42 0.3962 0.8976 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C19 mock treatment 1188000.0 1200.0 0.02 1198000.0 8350.0 0.15 0.1205 0.7943 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C20 mock treatment 1202120.0 15300.0 0.26 1202000.0 12300.0 0.22 0.3385 0.9975 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C21 mock treatment 1186440.0 -363.0 -0.01 1191200.0 1550.0 0.03 0.0154 0.54 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C22 mock treatment 1186240.0 -563.0 -0.01 1177360.0 -12300.0 -0.22 -0.1633 -0.7365 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C23 mock treatment 1173680.0 -13100.0 -0.22 1167360.0 -22300.0 -0.4 -0.4393 -0.9596 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 C24 mock treatment 1187120.0 317.0 0.01 1184560.0 -5090.0 -0.09 -0.0611 -0.6652 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D01 compound treatment 1265960.0 79200.0 1.32 1264560.0 74900.0 1.35 1.891 1.0 3000769 BCB02_000049 CCCCC(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D02 compound treatment 1293080.0 106000.0 1.78 1289040.0 99400.0 1.79 2.5238 1.0 3093844 BCB02_000050 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](CC=C([C@@H]2c3ccccc3)C(=O)O)c4ccc(F)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D03 compound treatment 1257960.0 71200.0 1.19 1254920.0 65300.0 1.18 1.6735 1.0 3093845 BCB02_000051 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5c(F)cccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D04 compound treatment 1264560.0 77800.0 1.3 1264680.0 75000.0 1.35 1.8759 0.9998 3000770 BCB02_000052 Cc1ccc(cc1)S(=O)(=O)N2C[C@H]([C@@H](C[C@H]2c3ccccc3)Sc4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D05 compound treatment 1239200.0 52400.0 0.88 1228800.0 39100.0 0.71 1.1187 0.9942 3093846 BCB02_000053 Cc1cc(C)c(C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5)c(C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D06 compound treatment 1259800.0 73000.0 1.22 1274240.0 84600.0 1.52 1.9414 0.994 3000771 BCB02_000054 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D07 compound treatment 1248200.0 61400.0 1.03 1224920.0 35300.0 0.64 1.1758 0.9733 3092586 BCB02_000055 Cc1ccccc1C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D08 compound treatment 1244800.0 58000.0 0.97 1256360.0 66700.0 1.2 1.5361 0.9944 3092495 BCB02_000056 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(F)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D09 compound treatment 1224240.0 37400.0 0.63 1220040.0 30400.0 0.55 0.8301 0.9977 3000772 BCB02_000057 OC(C1CCC=CC1)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D10 compound treatment 1251280.0 64500.0 1.08 1248680.0 59000.0 1.06 1.515 1.0 3092496 BCB02_000058 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(OC)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D11 compound treatment 1235560.0 48800.0 0.82 1228920.0 39300.0 0.71 1.0772 0.9975 3092497 BCB02_000059 CC(=O)n1cc(C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D12 compound treatment 1243240.0 56400.0 0.94 1229640.0 40000.0 0.72 1.1772 0.9911 3000773 BCB02_000060 CCOC(=O)C1=C[C@H](N([C@H]1c2cccc(Cl)c2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D13 compound treatment 1184640.0 -2160.0 -0.04 1212240.0 22600.0 0.41 0.2621 0.6417 3092498 BCB02_000061 CCCCC(CC)C(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D14 compound treatment 1217280.0 30500.0 0.51 1228840.0 39200.0 0.71 0.8599 0.9873 3000774 BCB02_000062 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2Cl)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D15 compound treatment 1211040.0 24200.0 0.41 1202720.0 13100.0 0.24 0.4533 0.9665 3092499 BCB02_000063 CC(=CCC/C(=C/C(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)/C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D16 compound treatment 1215680.0 28900.0 0.48 1218960.0 29300.0 0.53 0.7151 0.999 3000775 BCB02_000064 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(C)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D17 mock treatment 1192400.0 5600.0 0.09 1201600.0 11900.0 0.22 0.2184 0.9305 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D18 mock treatment 1208720.0 21900.0 0.37 1207680.0 18000.0 0.32 0.489 0.9982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D19 mock treatment 1192480.0 5680.0 0.09 1185280.0 -4370.0 -0.08 0.0114 0.0928 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D20 mock treatment 1181960.0 -4840.0 -0.08 1186560.0 -3090.0 -0.06 -0.0967 -0.9833 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D21 mock treatment 1174160.0 -12600.0 -0.21 1180160.0 -9490.0 -0.17 -0.2706 -0.9944 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D22 mock treatment 1179000.0 -7800.0 -0.13 1180960.0 -8690.0 -0.16 -0.2031 -0.9959 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D23 mock treatment 1169240.0 -17600.0 -0.29 1169160.0 -20500.0 -0.37 -0.4689 -0.9936 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 D24 mock treatment 1190640.0 3840.0 0.06 1182680.0 -6970.0 -0.13 -0.0434 -0.3079 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E01 compound treatment 1246920.0 60100.0 1.01 1259840.0 70200.0 1.26 1.6055 0.9936 3092500 BCB02_000065 CCCCC(CC)C(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E02 compound treatment 1250720.0 63900.0 1.07 1262880.0 73200.0 1.32 1.6892 0.9946 3000776 BCB02_000066 CCOC(=O)C1=CC[C@@H]2[C@H]1C(=O)N(CC)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E03 compound treatment 1258520.0 71700.0 1.2 1250400.0 60700.0 1.09 1.6225 0.9989 3000847 BCB02_000067 CC1(C)[C@H]2C[C@@H]1C=C(C2)C(O)C3C=CC4C(N3n5cnnc5)C(=O)N(Cc6ccccc6)C4=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E04 compound treatment 1250640.0 63800.0 1.07 1240280.0 50600.0 0.91 1.4004 0.9969 3000848 BCB02_000068 CCOC(=O)[C@H]1[C@H](C[C@@H]2[C@H]1C(=O)N(CC)C2=O)Sc3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E05 compound treatment 1260840.0 74000.0 1.24 1251560.0 61900.0 1.12 1.6648 0.9986 3000849 BCB02_000069 OC(C1C=CC2C(N1n3cnnc3)C(=O)N(Cc4ccccc4)C2=O)c5ccc(Br)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E06 compound treatment 1255440.0 68600.0 1.15 1249160.0 59500.0 1.07 1.5703 0.9994 3000850 BCB02_000070 OC(=O)C1=CC[C@@H]2[C@H]1C(=O)N(C2=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E07 compound treatment 1189520.0 2720.0 0.05 1167320.0 -22300.0 -0.4 -0.2524 -0.6233 3000851 BCB02_000071 OC(/C=C/c1ccc(cc1)[N+](=O)[O-])C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E08 compound treatment 1246120.0 59300.0 0.99 1240680.0 51000.0 0.92 1.352 0.9993 3092501 BCB02_000072 OC(=O)[C@H]1[C@H](C[C@@H]2[C@H]1C(=O)N(C2=O)c3ccccc3)Sc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E09 compound treatment 1210800.0 24000.0 0.4 1192400.0 2750.0 0.05 0.3189 0.7883 3000852 BCB02_000073 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E10 compound treatment 1231520.0 44700.0 0.75 1239280.0 49600.0 0.89 1.1614 0.9961 3092502 BCB02_000074 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E11 compound treatment 1212920.0 26100.0 0.44 1222840.0 33200.0 0.6 0.7318 0.9881 3092503 BCB02_000075 COc1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E12 compound treatment 1231760.0 45000.0 0.75 1205280.0 15600.0 0.28 0.7311 0.9101 3000853 BCB02_000076 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E13 compound treatment 1164920.0 -21900.0 -0.37 1176920.0 -12700.0 -0.23 -0.4212 -0.9746 3092504 BCB02_000077 CN(C)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E14 compound treatment 1208680.0 21900.0 0.37 1221000.0 31300.0 0.56 0.6582 0.978 3000854 BCB02_000078 CCOC(=O)C1=CC[C@H](N([C@H]1c2cccc(OC)c2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E15 compound treatment 1206400.0 19600.0 0.33 1194560.0 4910.0 0.09 0.2944 0.8668 3092505 BCB02_000079 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3Nc5ccccc5F)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E16 compound treatment 1224360.0 37600.0 0.63 1226640.0 37000.0 0.67 0.9156 0.9996 3000855 BCB02_000080 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E17 mock treatment 1211000.0 24200.0 0.4 1200240.0 10600.0 0.19 0.4212 0.941 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E18 mock treatment 1220720.0 33900.0 0.57 1216520.0 26900.0 0.48 0.7436 0.9969 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E19 mock treatment 1202600.0 15800.0 0.26 1193840.0 4190.0 0.08 0.2403 0.874 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E20 mock treatment 1202000.0 15200.0 0.25 1206360.0 16700.0 0.3 0.3927 0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E21 mock treatment 1185720.0 -1080.0 -0.02 1186520.0 -3130.0 -0.06 -0.0527 -0.8894 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E22 mock treatment 1180160.0 -6640.0 -0.11 1182160.0 -7490.0 -0.14 -0.1741 -0.9953 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E23 mock treatment 1181640.0 -5160.0 -0.09 1182000.0 -7650.0 -0.14 -0.1586 -0.9746 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 E24 mock treatment 1188520.0 1720.0 0.03 1191240.0 1590.0 0.03 0.0405 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F01 compound treatment 1253840.0 67000.0 1.12 1248200.0 58500.0 1.05 1.5391 0.9995 3092506 BCB02_000081 OC(COCc1ccccc1)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F02 compound treatment 1276760.0 90000.0 1.51 1258800.0 69100.0 1.25 1.9454 0.9956 3092507 BCB02_000082 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(OC)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F03 compound treatment 1182080.0 -4720.0 -0.08 1140320.0 -49300.0 -0.89 -0.6844 -0.767 3000856 BCB02_000083 COc1ccc(NN2C3C(C=CC2C(O)c4ccccc4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F04 compound treatment 1263720.0 76900.0 1.29 1261360.0 71700.0 1.29 1.8237 1.0 3092508 BCB02_000084 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F05 compound treatment 1235600.0 48800.0 0.82 1227800.0 38100.0 0.69 1.0634 0.9963 3092509 BCB02_000085 CCCCC(O)C1C=CC2C(N1Nc3ccc(OC)cc3)C(=O)N(C4CCCCC4)C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F06 compound treatment 1247320.0 60500.0 1.01 1253360.0 63700.0 1.15 1.5277 0.9981 3000857 BCB02_000086 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(F)cc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F07 compound treatment 1231840.0 45000.0 0.75 1195920.0 6270.0 0.11 0.6128 0.8041 3092510 BCB02_000087 COc1ccc(NN2C3C(C=CC2C(O)c4ccc(F)cc4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F08 compound treatment 1242840.0 56000.0 0.94 1243120.0 53500.0 0.96 1.3443 0.9999 3000858 BCB02_000088 CCOC(=O)C1=C[C@H](N([C@H]1c2ccc(Cl)c(Cl)c2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F09 compound treatment 1208360.0 21600.0 0.36 1216480.0 26800.0 0.48 0.5968 0.9896 3092511 BCB02_000089 C/C=C/C(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F10 compound treatment 1240040.0 53200.0 0.89 1237680.0 48000.0 0.87 1.2418 0.9999 3000859 BCB02_000090 CCOC(=O)C1=C[C@H](N([C@H]1c2cccc(Cl)c2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F11 compound treatment 1220440.0 33600.0 0.56 1216440.0 26800.0 0.48 0.7393 0.9971 3092512 BCB02_000091 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F12 compound treatment 1246920.0 60100.0 1.01 1206600.0 16900.0 0.31 0.9273 0.882 3092513 BCB02_000092 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2Cl)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F13 compound treatment 1162400.0 -24400.0 -0.41 1174360.0 -15300.0 -0.28 -0.4836 -0.9817 3000860 BCB02_000093 CN(C)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F14 compound treatment 1232320.0 45500.0 0.76 1218640.0 29000.0 0.52 0.9079 0.983 3092514 BCB02_000094 CCOC(=O)C1=C[C@H](N([C@H]1c2cccc3ccccc23)S(=O)(=O)c4ccc(C)cc4)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F15 compound treatment 1180560.0 -6240.0 -0.1 1164280.0 -25400.0 -0.46 -0.3971 -0.8469 3092515 BCB02_000095 COc1cc(cc(OC)c1OC)C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F16 compound treatment 1217520.0 30700.0 0.51 1209120.0 19500.0 0.35 0.6115 0.9826 3000861 BCB02_000096 CCOC(=O)C1=C[C@@H](C(C)C)N([C@H]1c2ccc(cc2)C(F)(F)F)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F17 mock treatment 1186240.0 -563.0 -0.01 1192560.0 2910.0 0.05 0.0304 0.5706 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F18 mock treatment 1207640.0 20800.0 0.35 1213040.0 23400.0 0.42 0.5445 0.9956 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F19 mock treatment 1173520.0 -13300.0 -0.22 1190840.0 1190.0 0.02 -0.1421 -0.6362 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F20 mock treatment 1189720.0 2920.0 0.05 1187520.0 -2130.0 -0.04 0.0073 0.1179 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F21 mock treatment 1179440.0 -7360.0 -0.12 1182920.0 -6730.0 -0.12 -0.1729 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F22 mock treatment 1169960.0 -16800.0 -0.28 1175320.0 -14300.0 -0.26 -0.3819 -0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F23 mock treatment 1149520.0 -37300.0 -0.62 1162120.0 -27500.0 -0.5 -0.792 -0.9935 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 F24 mock treatment 1186960.0 157.0 0.0 1180800.0 -8850.0 -0.16 -0.1109 -0.6954 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G01 compound treatment 1273600.0 86800.0 1.45 1261160.0 71500.0 1.29 1.9381 0.9982 3092516 BCB02_000097 CC(C(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G02 compound treatment 1290880.0 104000.0 1.74 1288240.0 98600.0 1.78 2.4875 1.0 3000862 BCB02_000098 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2C)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G03 compound treatment 1262440.0 75600.0 1.27 1265480.0 75800.0 1.37 1.861 0.9993 3092587 BCB02_000099 CCCCCCCCCCC(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G04 compound treatment 1288200.0 101000.0 1.7 1281400.0 91700.0 1.65 2.3687 0.9999 3000863 BCB02_000100 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)C[Si](C)(C)C)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G05 compound treatment 1240760.0 54000.0 0.9 1251400.0 61700.0 1.11 1.4251 0.9946 3092588 BCB02_000101 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccc(F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G06 compound treatment 1256000.0 69200.0 1.16 1239080.0 49400.0 0.89 1.4485 0.9916 3092589 BCB02_000102 CCOC(=O)C1=CC[C@H](N([C@H]1/C=C/c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G07 compound treatment 1256600.0 69800.0 1.17 1218280.0 28600.0 0.52 1.1906 0.9325 3000864 BCB02_000103 COc1ccc(C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5)c6ccccc16 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G08 compound treatment 1247080.0 60300.0 1.01 1239560.0 49900.0 0.9 1.3491 0.9984 3092590 BCB02_000104 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)c4cccc(Cl)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G09 compound treatment 1244680.0 57900.0 0.97 1247200.0 57500.0 1.04 1.418 0.9994 3092591 BCB02_000105 COc1ccc(cc1OCc2ccccc2)C(O)C3C=CC4C(N3Nc5ccc(cc5)[N+](=O)[O-])C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G10 compound treatment 1246520.0 59700.0 1.0 1256000.0 66300.0 1.2 1.5519 0.996 3000865 BCB02_000106 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2I)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G11 compound treatment 1217400.0 30600.0 0.51 1212560.0 22900.0 0.41 0.6539 0.9943 3092592 BCB02_000107 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccccn5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G12 compound treatment 1216640.0 29800.0 0.5 1258120.0 68500.0 1.23 1.2253 0.9208 3000866 BCB02_000108 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G13 compound treatment 1210320.0 23500.0 0.39 1166160.0 -23500.0 -0.42 -0.021 -0.0364 3092593 BCB02_000109 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G14 compound treatment 1253440.0 66600.0 1.12 1250320.0 60700.0 1.09 1.5614 0.9999 3000867 BCB02_000110 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G15 compound treatment 1223000.0 36200.0 0.61 1221400.0 31700.0 0.57 0.8328 0.9996 3092594 BCB02_000111 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G16 compound treatment 1190880.0 4080.0 0.07 1194240.0 4590.0 0.08 0.1067 0.9955 3092595 BCB02_000112 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(SC)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(OCc5ccccc5)c(OC)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G17 mock treatment 1199840.0 13000.0 0.22 1198320.0 8670.0 0.16 0.2647 0.9865 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G18 mock treatment 1215680.0 28900.0 0.48 1187640.0 -2010.0 -0.04 0.316 0.6522 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G19 mock treatment 1200720.0 13900.0 0.23 1212240.0 22600.0 0.41 0.4524 0.9649 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G20 mock treatment 1193000.0 6200.0 0.1 1190160.0 506.0 0.01 0.0798 0.7663 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G21 mock treatment 1191640.0 4840.0 0.08 1198280.0 8630.0 0.16 0.1671 0.9538 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G22 mock treatment 1211240.0 24400.0 0.41 1203760.0 14100.0 0.25 0.4689 0.9738 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G23 mock treatment 1181680.0 -5120.0 -0.09 1191760.0 2110.0 0.04 -0.0338 -0.3604 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 G24 mock treatment 1185560.0 -1240.0 -0.02 1196120.0 6470.0 0.12 0.0677 0.5718 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H01 compound treatment 1275240.0 88400.0 1.48 1264800.0 75100.0 1.35 2.0038 0.999 3000868 BCB02_000113 CC(=CCC/C(=C/C(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)/C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H02 compound treatment 1287200.0 100000.0 1.68 1285760.0 96100.0 1.73 2.4124 0.9999 3092596 BCB02_000114 CCOC(=O)C1=C[C@@H](C(C)C)N([C@H]1c2ccc(cc2)C(C)C)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H03 compound treatment 1245600.0 58800.0 0.98 1251480.0 61800.0 1.11 1.4834 0.9981 3092597 BCB02_000115 OC(CCc1ccccc1)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H04 compound treatment 1259280.0 72500.0 1.21 1265560.0 75900.0 1.37 1.8247 0.9982 3000869 BCB02_000116 CCOC(=O)C1=C[C@@H](C(C)C)N([C@H]1c2ccccc2F)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H05 compound treatment 1236840.0 50000.0 0.84 1246400.0 56700.0 1.02 1.315 0.9951 3092598 BCB02_000117 COc1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccccc4F)C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H06 compound treatment 1275160.0 88400.0 1.48 1273880.0 84200.0 1.52 2.1186 0.9999 3000870 BCB02_000118 CCOC(=O)C1=C[C@@H](CC)N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H07 compound treatment 1210680.0 23900.0 0.4 1215840.0 26200.0 0.47 0.6161 0.9966 3000871 BCB02_000119 O=c1cccc(o1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H08 compound treatment 1261520.0 74700.0 1.25 1257600.0 67900.0 1.22 1.7498 0.9999 3092599 BCB02_000120 CCOC(=O)C1=CCN(C1c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H09 compound treatment 1194320.0 7520.0 0.13 1179960.0 -9690.0 -0.17 -0.0346 -0.1605 3000872 BCB02_000121 COc1cccc(c1)c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H10 compound treatment 1249520.0 62700.0 1.05 1242120.0 52500.0 0.95 1.4106 0.9986 3092600 BCB02_000122 CCC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccccc3)C(=O)OCC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H11 compound treatment 1146800.0 -40000.0 -0.67 1130200.0 -59500.0 -1.07 -1.2308 -0.9744 1984103 BCB02_000123 Cc1ccc(cc1)c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H12 compound treatment 1222400.0 35600.0 0.6 1215920.0 26300.0 0.47 0.7559 0.9935 3092601 BCB02_000124 CCOC(=O)C1=C[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H13 compound treatment 1219120.0 32300.0 0.54 1212400.0 22700.0 0.41 0.6722 0.9906 3000873 BCB02_000125 Clc1cccc(c1)c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H14 compound treatment 1226280.0 39500.0 0.66 1218760.0 29100.0 0.52 0.8379 0.9935 3000874 BCB02_000126 Cc1ccc(cc1)[C@@H]2N(CC=C2C(=O)O)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H15 compound treatment 1198680.0 11900.0 0.2 1201720.0 12100.0 0.22 0.2943 0.999 3000875 BCB02_000127 Clc1ccccc1c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H16 compound treatment 1212120.0 25300.0 0.42 1202800.0 13100.0 0.24 0.4671 0.9623 3092602 BCB02_000128 C[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H17 mock treatment 1206560.0 19800.0 0.33 1203160.0 13500.0 0.24 0.4059 0.9886 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H18 mock treatment 1222000.0 35200.0 0.59 1196600.0 6950.0 0.13 0.505 0.8386 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H19 mock treatment 1200200.0 13400.0 0.22 1198680.0 9030.0 0.16 0.2735 0.9876 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H20 mock treatment 1186800.0 -3.33 0.0 1196400.0 6750.0 0.12 0.0859 0.7068 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H21 mock treatment 1168440.0 -18400.0 -0.31 1184880.0 -4770.0 -0.09 -0.2781 -0.8715 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H22 mock treatment 1173160.0 -13600.0 -0.23 1182000.0 -7650.0 -0.14 -0.259 -0.9709 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H23 mock treatment 1162280.0 -24500.0 -0.41 1159960.0 -29700.0 -0.54 -0.6685 -0.9914 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 H24 mock treatment 1171920.0 -14900.0 -0.25 1167240.0 -22400.0 -0.4 -0.4617 -0.973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I01 compound treatment 1259880.0 73100.0 1.22 1255920.0 66300.0 1.19 1.709 0.9999 3092603 BCB02_000129 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5cccs5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I02 compound treatment 1295000.0 108000.0 1.81 1268000.0 78300.0 1.41 2.2784 0.9924 3000947 BCB02_000130 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(cc2)[N+](=O)[O-])S(=O)(=O)c3ccc(C)cc3)c4ccc(F)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I03 compound treatment 1260320.0 73500.0 1.23 1251920.0 62300.0 1.12 1.6632 0.9989 3000948 BCB02_000131 OC(C(c1ccccc1)c2ccccc2)C3C=CC4C(N3Nc5ccc(cc5)[N+](=O)[O-])C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I04 compound treatment 1278880.0 92100.0 1.54 1258240.0 68600.0 1.24 1.9633 0.994 3000949 BCB02_000132 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(cc2)[N+](=O)[O-])S(=O)(=O)c3ccc(C)cc3)c4cccc(Br)c4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I05 compound treatment 1242280.0 55500.0 0.93 1235400.0 45700.0 0.82 1.2393 0.9982 3000950 BCB02_000133 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5cccc6ccccc56 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I06 compound treatment 1240520.0 53700.0 0.9 1255040.0 65400.0 1.18 1.4687 0.9911 3000951 BCB02_000134 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I07 compound treatment 1250880.0 64100.0 1.07 1230680.0 41000.0 0.74 1.2809 0.9835 3092604 BCB02_000135 C/C=C/C(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I08 compound treatment 1260320.0 73500.0 1.23 1256120.0 66500.0 1.2 1.7167 0.9999 3000952 BCB02_000136 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3cccc4ccccc34 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I09 compound treatment 1238360.0 51600.0 0.86 1231000.0 41300.0 0.74 1.1368 0.9973 3092605 BCB02_000137 CCC(CC)C(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I10 compound treatment 1247360.0 60600.0 1.01 1242960.0 53300.0 0.96 1.3957 0.9996 3092606 BCB02_000138 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(F)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I11 compound treatment 1238440.0 51600.0 0.86 1234640.0 45000.0 0.81 1.1841 0.9995 3000953 BCB02_000139 CC(C)C(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I12 compound treatment 1218000.0 31200.0 0.52 1215040.0 25400.0 0.46 0.6926 0.9978 3092607 BCB02_000140 CCOC(=O)[C@@H]1N([C@@H](CC=C1C(=O)OCC)c2ccccc2)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I13 compound treatment 1218800.0 32000.0 0.54 1233040.0 43400.0 0.78 0.9314 0.983 3092678 BCB02_000141 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5cccc(O)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I14 compound treatment 1233120.0 46300.0 0.78 1232640.0 43000.0 0.77 1.0957 1.0 3000954 BCB02_000142 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(OC)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I15 compound treatment 1204960.0 18200.0 0.3 1211320.0 21700.0 0.39 0.4909 0.9923 3092679 BCB02_000143 OB(O)c1ccc(cc1)C(O)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I16 compound treatment 1203360.0 16600.0 0.28 1201520.0 11900.0 0.21 0.3471 0.9918 3000955 BCB02_000144 CCOC(=O)C1=CC[C@H](N([C@H]1C)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I17 mock treatment 1206400.0 19600.0 0.33 1219560.0 29900.0 0.54 0.6129 0.9717 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I18 mock treatment 1214000.0 27200.0 0.46 1202120.0 12500.0 0.22 0.4806 0.947 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I19 mock treatment 1201960.0 15200.0 0.25 1191920.0 2270.0 0.04 0.2082 0.8105 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I20 mock treatment 1200840.0 14000.0 0.23 1194840.0 5190.0 0.09 0.2322 0.9184 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I21 mock treatment 1191160.0 4360.0 0.07 1202880.0 13200.0 0.24 0.2201 0.883 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I22 mock treatment 1176240.0 -10600.0 -0.18 1197080.0 7430.0 0.13 -0.0304 -0.1371 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I23 mock treatment 1171360.0 -15400.0 -0.26 1176800.0 -12900.0 -0.23 -0.3465 -0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 I24 mock treatment 1160800.0 -26000.0 -0.44 1171160.0 -18500.0 -0.33 -0.5433 -0.9913 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J01 compound treatment 1282400.0 95600.0 1.6 1263800.0 74100.0 1.34 2.0758 0.996 3000956 BCB02_000145 CCCc1cccc(=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J02 compound treatment 1282160.0 95400.0 1.6 1280000.0 90300.0 1.63 2.2794 1.0 3092680 BCB02_000146 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J03 compound treatment 1260760.0 74000.0 1.24 1257120.0 67500.0 1.22 1.7347 1.0 3000957 BCB02_000147 Fc1ccc(cc1)c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J04 compound treatment 1260320.0 73500.0 1.23 1261560.0 71900.0 1.3 1.786 0.9997 3092681 BCB02_000148 CCC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J05 compound treatment 1261440.0 74600.0 1.25 1252040.0 62400.0 1.12 1.678 0.9986 3000958 BCB02_000149 O=c1cccc(o1)c2ccc(C#N)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J06 compound treatment 1276400.0 89600.0 1.5 1251560.0 61900.0 1.12 1.8489 0.9894 3000959 BCB02_000150 CC(C)[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J07 compound treatment 1228240.0 41400.0 0.69 1218160.0 28500.0 0.51 0.8535 0.9891 3092682 BCB02_000151 FC(F)(F)c1ccc(cc1)c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J08 compound treatment 1252160.0 65400.0 1.09 1245240.0 55600.0 1.0 1.4815 0.999 3092683 BCB02_000152 Cc1ccc(cc1)[C@@H]2N([C@@H](C=C2C(=O)O)C(C)(C)C)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J09 compound treatment 1243880.0 57100.0 0.96 1233800.0 44100.0 0.8 1.2378 0.9959 3000960 BCB02_000153 FC(F)(F)c1ccccc1c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J10 compound treatment 1230440.0 43600.0 0.73 1234920.0 45300.0 0.82 1.0931 0.9985 3092684 BCB02_000154 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccccc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J11 compound treatment 1106360.0 -80400.0 -1.35 1038520.0 -151000.0 -2.72 -2.8774 -0.9472 3000961 BCB02_000155 O=c1cccc(o1)c2ccc3ccccc3c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J12 compound treatment 1213240.0 26400.0 0.44 1206080.0 16400.0 0.3 0.5221 0.9809 3000962 BCB02_000156 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(C#N)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J13 compound treatment 1223200.0 36400.0 0.61 1187600.0 -2050.0 -0.04 0.4045 0.6629 3092685 BCB02_000157 O=c1cccc(o1)c2ccco2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J14 compound treatment 1235680.0 48900.0 0.82 1225960.0 36300.0 0.65 1.0409 0.9939 3092686 BCB02_000158 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(OC)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J15 compound treatment 1187000.0 197.0 0.0 1191840.0 2190.0 0.04 0.0302 0.7635 3000963 BCB02_000159 O=c1cccc(CCc2ccccc2)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J16 compound treatment 1211840.0 25000.0 0.42 1210040.0 20400.0 0.37 0.556 0.9978 3092687 BCB02_000160 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3cccc(Cl)c3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J17 mock treatment 1211240.0 24400.0 0.41 1212120.0 22500.0 0.4 0.5754 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J18 mock treatment 1201600.0 14800.0 0.25 1200320.0 10700.0 0.19 0.311 0.9921 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J19 mock treatment 1185360.0 -1440.0 -0.02 1190880.0 1230.0 0.02 -0.0015 -0.0446 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J20 mock treatment 1189200.0 2400.0 0.04 1204080.0 14400.0 0.26 0.2121 0.8067 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J21 mock treatment 1176040.0 -10800.0 -0.18 1177720.0 -11900.0 -0.22 -0.2794 -0.9961 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J22 mock treatment 1187880.0 1080.0 0.02 1191240.0 1590.0 0.03 0.0329 0.9753 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J23 mock treatment 1172920.0 -13900.0 -0.23 1181040.0 -8610.0 -0.16 -0.274 -0.9808 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 J24 mock treatment 1174760.0 -12000.0 -0.2 1192560.0 2910.0 0.05 -0.1055 -0.5066 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K01 compound treatment 1265360.0 78600.0 1.31 1257400.0 67700.0 1.22 1.7927 0.9993 3000964 BCB02_000161 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccc(C#N)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K02 compound treatment 1148040.0 -38800.0 -0.65 1163920.0 -25700.0 -0.46 -0.7865 -0.9864 3092688 BCB02_000162 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccncc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K03 compound treatment 1257440.0 70600.0 1.18 1248080.0 58400.0 1.05 1.5802 0.9983 3092689 BCB02_000163 CC(C(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K04 compound treatment 1272400.0 85600.0 1.43 1276760.0 87100.0 1.57 2.1226 0.999 3000965 BCB02_000164 CCOC(=O)C1=CC[C@H](N([C@H]1C=C(C)C)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K05 compound treatment 1250160.0 63400.0 1.06 1244400.0 54700.0 0.99 1.4472 0.9993 3092690 BCB02_000165 CC(CC(O)C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccc(C)o5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K06 compound treatment 1197720.0 10900.0 0.18 1161680.0 -28000.0 -0.5 -0.2272 -0.4238 3000966 BCB02_000166 CCOC(=O)C1=CC[C@H](N([C@H]1C#N)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K07 compound treatment 1236960.0 50200.0 0.84 1229480.0 39800.0 0.72 1.1009 0.997 3092691 BCB02_000167 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5cccs5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K08 compound treatment 1256280.0 69500.0 1.16 1247880.0 58200.0 1.05 1.5639 0.9987 3092692 BCB02_000168 CCOC(=O)C1=CC[C@H](N([C@H]1c2cccc(OC)c2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K09 compound treatment 1251080.0 64300.0 1.08 1236720.0 47100.0 0.85 1.3602 0.9931 3000967 BCB02_000169 OC(Cc1ccccc1)C2C=CC3C(N2Nc4ccc(cc4)[N+](=O)[O-])C(=O)N(C3=O)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K10 compound treatment 1247160.0 60400.0 1.01 1248880.0 59200.0 1.07 1.4688 0.9996 3092693 BCB02_000170 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(C#N)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K11 compound treatment 1203320.0 16500.0 0.28 1196200.0 6550.0 0.12 0.2788 0.9279 3000968 BCB02_000171 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccc(C#N)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K12 compound treatment 1212320.0 25500.0 0.43 1232600.0 42900.0 0.77 0.8491 0.9607 3092694 BCB02_000172 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(cc4)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K13 compound treatment 1198000.0 11200.0 0.19 1209200.0 19500.0 0.35 0.3815 0.9564 3092695 BCB02_000173 OC(C1C=CC2C(N1Nc3ccc(cc3)[N+](=O)[O-])C(=O)N(C2=O)c4ccccc4)c5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K14 compound treatment 1210320.0 23500.0 0.39 1188240.0 -1410.0 -0.03 0.2603 0.66 3000969 BCB02_000174 CCOC(=O)C1=CC[C@H](N([C@H]1C=C)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K15 compound treatment 1209080.0 22300.0 0.37 1191360.0 1710.0 0.03 0.2853 0.7628 3092696 BCB02_000175 CC1(C)[C@H]2C[C@@H]1C=C(C2)C(O)C3C=CC4C(N3Nc5ccc(cc5)[N+](=O)[O-])C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K16 compound treatment 1220200.0 33400.0 0.56 1215080.0 25400.0 0.46 0.7191 0.9951 3000970 BCB02_000176 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(cc2)[N+](=O)[O-])S(=O)(=O)c3ccc(C)cc3)c4ccc(cc4)N(CC)CC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K17 mock treatment 1214040.0 27200.0 0.46 1217760.0 28100.0 0.51 0.6804 0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K18 mock treatment 1203440.0 16600.0 0.28 1197880.0 8230.0 0.15 0.3017 0.9565 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K19 mock treatment 1222480.0 35700.0 0.6 1200920.0 11300.0 0.2 0.5657 0.8971 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K20 mock treatment 1213800.0 27000.0 0.45 1204400.0 14700.0 0.27 0.5073 0.968 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K21 mock treatment 1196800.0 10000.0 0.17 1199400.0 9750.0 0.18 0.2425 0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K22 mock treatment 1188880.0 2080.0 0.03 1189560.0 -93.9 0.0 0.0234 0.6719 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K23 mock treatment 1171440.0 -15400.0 -0.26 1182920.0 -6730.0 -0.12 -0.2676 -0.9413 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 K24 mock treatment 1169160.0 -17600.0 -0.3 1167320.0 -22300.0 -0.4 -0.4933 -0.9884 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L01 compound treatment 1254640.0 67800.0 1.14 1258200.0 68500.0 1.24 1.676 0.9991 3000971 BCB02_000177 [O-][N+](=O)c1ccc(cc1)c2cccc(=O)o2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L02 compound treatment 1220800.0 34000.0 0.57 1207640.0 18000.0 0.32 0.6314 0.9644 3092697 BCB02_000178 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])c3ccccc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L03 compound treatment 1243240.0 56400.0 0.94 1242840.0 53200.0 0.96 1.3454 1.0 3000972 BCB02_000179 O=c1cccc(/C=C/c2ccccc2)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L04 compound treatment 1238400.0 51600.0 0.86 1227280.0 37600.0 0.68 1.0899 0.9928 3092698 BCB02_000180 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccco3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L05 compound treatment 1256440.0 69600.0 1.17 1244520.0 54900.0 0.99 1.523 0.9966 3000973 BCB02_000181 O=c1cccc(o1)c2cccc3ccccc23 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L06 compound treatment 1253840.0 67000.0 1.12 1242080.0 52400.0 0.94 1.4612 0.9963 3092699 BCB02_000182 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3cccc4ccccc34)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L07 compound treatment 1234640.0 47800.0 0.8 1217720.0 28100.0 0.51 0.9236 0.9755 3000974 BCB02_000183 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(Cl)c2)c3cccc(Cl)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L08 compound treatment 1227840.0 41000.0 0.69 1225440.0 35800.0 0.64 0.9415 0.9995 3092700 BCB02_000184 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(Br)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L09 compound treatment 1243320.0 56500.0 0.95 1240160.0 50500.0 0.91 1.3122 0.9998 3092701 BCB02_000185 CCOC(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(c2)[N+](=O)[O-])c3cccc(c3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L10 compound treatment 1220240.0 33400.0 0.56 1216200.0 26500.0 0.48 0.7339 0.9969 3000975 BCB02_000186 CC[C@@H]1C=C([C@@H](N1S(=O)(=O)c2ccc(C)cc2)c3ccc(cc3)C(C)C)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L11 compound treatment 1227040.0 40200.0 0.67 1202000.0 12300.0 0.22 0.6334 0.8932 3092771 BCB02_000187 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccccn2)c3ccccn3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L12 compound treatment 1237640.0 50800.0 0.85 1235560.0 45900.0 0.83 1.1864 0.9999 3000976 BCB02_000188 Cc1ccc(cc1)S(=O)(=O)N2[C@@H](C=C([C@@H]2c3ccccc3)C(=O)O)C(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L13 compound treatment 1139960.0 -46800.0 -0.78 1096840.0 -92800.0 -1.67 -1.7368 -0.9404 3092772 BCB02_000189 COC(=O)c1cccc(c1)[C@@H]2C/C(=C\C(=O)OC(C)C)/O[C@@H](O2)c3cccc(c3)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L14 compound treatment 1213120.0 26300.0 0.44 1198680.0 9030.0 0.16 0.4264 0.9083 3092773 BCB02_000190 CC(C)[C@@H]1[C@@H](Sc2ccccc2)[C@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L15 compound treatment 1190600.0 3800.0 0.06 1172120.0 -17500.0 -0.32 -0.1785 -0.5538 3000977 BCB02_000191 CC(C)OC(=O)/C=C\1/C[C@H](O[C@H](O1)c2ccc(C#N)cc2)c3ccc(C#N)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L16 compound treatment 1207400.0 20600.0 0.34 1212440.0 22800.0 0.41 0.534 0.9962 3092774 BCB02_000192 CC[C@@H]1C(Sc2ccccc2)C([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L17 mock treatment 1202600.0 15800.0 0.26 1200560.0 10900.0 0.2 0.3259 0.9893 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L18 mock treatment 1216240.0 29400.0 0.49 1216320.0 26700.0 0.48 0.6881 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L19 mock treatment 1200200.0 13400.0 0.22 1199960.0 10300.0 0.19 0.2898 0.9956 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L20 mock treatment 1201120.0 14300.0 0.24 1204000.0 14300.0 0.26 0.3522 0.9993 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L21 mock treatment 1180600.0 -6200.0 -0.1 1184360.0 -5290.0 -0.1 -0.1408 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L22 mock treatment 1186440.0 -363.0 -0.01 1177080.0 -12600.0 -0.23 -0.1645 -0.7258 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L23 mock treatment 1177520.0 -9280.0 -0.16 1173680.0 -16000.0 -0.29 -0.3134 -0.9581 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 L24 mock treatment 1153320.0 -33500.0 -0.56 1165080.0 -24600.0 -0.44 -0.7093 -0.9932 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M01 compound treatment 1229600.0 42800.0 0.72 1220960.0 31300.0 0.56 0.9053 0.993 3000978 BCB02_000193 CC1(C)[C@H]2C[C@H]1C=C(C2)C(O)C3C=CC4C(N3Nc5ccccc5F)C(=O)N(C4=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M02 compound treatment 1066560.0 -120000.0 -2.01 1045080.0 -145000.0 -2.6 -3.2647 -0.9919 3001047 BCB02_000194 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(c(OC)c4)c5ccc(OCc6ccccc6)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M03 compound treatment 1252920.0 66100.0 1.11 1229480.0 39800.0 0.72 1.2898 0.978 3092775 BCB02_000195 COc1ccc(NN2C3C(C=CC2C(O)c4ccc(I)cc4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M04 compound treatment 1272880.0 86100.0 1.44 1261800.0 72100.0 1.3 1.9377 0.9987 3001048 BCB02_000196 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccccc2)S(=O)(=O)c3ccc(C)cc3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M05 compound treatment 1244760.0 58000.0 0.97 1209560.0 19900.0 0.36 0.9394 0.9085 3092776 BCB02_000197 COc1ccc(NN2C3C(C=CC2C(O)c4ccc(cc4)[N+](=O)[O-])C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M06 compound treatment 1276280.0 89500.0 1.5 1259760.0 70100.0 1.26 1.9519 0.9964 3001049 BCB02_000198 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M07 compound treatment 1252760.0 66000.0 1.1 1226600.0 36900.0 0.67 1.2512 0.9707 3092777 BCB02_000199 COc1ccc(NN2C3C(C=CC2C(O)c4ccc(OC)cc4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M08 compound treatment 1253520.0 66700.0 1.12 1242640.0 53000.0 0.95 1.4645 0.997 3092778 BCB02_000200 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(CC)cc2)S(=O)(=O)c3ccc(C)cc3)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M09 compound treatment 1223000.0 36200.0 0.61 1199760.0 10100.0 0.18 0.5571 0.8807 3001050 BCB02_000201 COc1ccc(NN2C3C(C=CC2C(O)c4ccc(cc4)N(C)C)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M10 compound treatment 1232800.0 46000.0 0.77 1225840.0 36200.0 0.65 1.0053 0.9966 3001168 BCB02_000202 CCOC(=O)C1=C(N([C@@H](CC1)c2ccccc2)S(=O)(=O)CC[Si](C)(C)C)C(=O)OCC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M11 compound treatment 1217720.0 30900.0 0.52 1206600.0 16900.0 0.31 0.5817 0.9683 3092779 BCB02_000203 COc1ccc(NN2C3C(C=CC2C(O)c4cc(OC)c(OC)c(OC)c4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M12 compound treatment 1223240.0 36400.0 0.61 1230600.0 40900.0 0.74 0.9528 0.9955 3092780 BCB02_000204 CCOC(=O)C1=CC[C@H](N([C@H]1c2ccc(OC)cc2)S(=O)(=O)c3ccc(C)cc3)c4cc(Cl)ccc4Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M13 compound treatment 1180760.0 -6040.0 -0.1 1164520.0 -25100.0 -0.45 -0.3917 -0.8442 3001169 BCB02_000205 COc1ccc(NN2C3C(C=CC2C(O)C4=CC[C@H](CC4)C(=C)C)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M14 compound treatment 1215240.0 28400.0 0.48 1231080.0 41400.0 0.75 0.8643 0.9764 3092781 BCB02_000206 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M15 compound treatment 1184000.0 -2800.0 -0.05 1164120.0 -25500.0 -0.46 -0.3585 -0.7752 3001170 BCB02_000207 COc1ccc(NN2C3C(C=CC2C(O)c4ccco4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M16 mock treatment 1199920.0 13100.0 0.22 1206920.0 17300.0 0.31 0.3752 0.9854 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M17 mock treatment 1208760.0 22000.0 0.37 1204160.0 14500.0 0.26 0.4446 0.9861 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M18 mock treatment 1222960.0 36200.0 0.61 1222200.0 32500.0 0.59 0.8425 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M19 mock treatment 1191200.0 4400.0 0.07 1189200.0 -454.0 -0.01 0.0462 0.6247 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M20 mock treatment 1191720.0 4920.0 0.08 1200400.0 10700.0 0.19 0.1951 0.9273 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M21 mock treatment 1177960.0 -8840.0 -0.15 1190040.0 386.0 0.01 -0.0997 -0.6731 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M22 mock treatment 1186400.0 -403.0 -0.01 1174920.0 -14700.0 -0.27 -0.1925 -0.7249 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M23 mock treatment 1177120.0 -9680.0 -0.16 1189760.0 106.0 0.0 -0.1132 -0.6987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 M24 mock treatment 1190160.0 3360.0 0.06 1193920.0 4270.0 0.08 0.0941 0.9881 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N01 compound treatment 1172160.0 -14600.0 -0.25 1165720.0 -23900.0 -0.43 -0.4782 -0.9641 3092782 BCB02_000208 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccc(cc2)C(F)(F)F)c3ccc(cc3)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N02 compound treatment 1257000.0 70200.0 1.17 1238720.0 49100.0 0.88 1.4558 0.9902 3092783 BCB02_000209 CCC[C@@H]1[C@@H](Sc2ccccc2)[C@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N03 compound treatment 1228680.0 41900.0 0.7 1228600.0 38900.0 0.7 0.9917 1.0 3001171 BCB02_000210 CC(C)OC(=O)/C=C\1/C[C@H](O[C@H](O1)c2ccc([Ac])cc2)c3ccc([Ac])cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N04 compound treatment 1239400.0 52600.0 0.88 1232240.0 42600.0 0.77 1.1649 0.9977 3092784 BCB02_000211 CCS[C@@H]1[C@@H](CC)N([C@H]([C@@H]1C(=O)O)c2ccc(C)cc2)S(=O)(=O)c3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N05 compound treatment 1168920.0 -17900.0 -0.3 1151920.0 -37700.0 -0.68 -0.6923 -0.9321 3001172 BCB02_000212 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccc([Ac])cc2)c3ccc([Ac])cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N06 compound treatment 1233280.0 46500.0 0.78 1231880.0 42200.0 0.76 1.0879 0.9999 3092785 BCB02_000213 CCOC1=C2C(N(CC2C3C(C1)C(=O)N(C3=O)c4ccccc4)S(=O)(=O)c5ccc(C)cc5)c6ccc(C)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N07 compound treatment 1159640.0 -27200.0 -0.45 1147040.0 -42600.0 -0.77 -0.8643 -0.9687 3092786 BCB02_000214 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(c2)C(F)(F)F)c3cccc(c3)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N08 compound treatment 1230600.0 43800.0 0.73 1234920.0 45300.0 0.82 1.0949 0.9986 3001173 BCB02_000215 CCOC1=C2C(N(CC2n3n(C1)c(=O)n(c4ccccc4)c3=O)S(=O)(=O)c5ccc(C)cc5)c6ccc(C)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N09 compound treatment 1224360.0 37600.0 0.63 1213440.0 23800.0 0.43 0.7474 0.9826 3092787 BCB02_000216 CC(C)OC(=O)/C=C\1/C[C@H](O[C@H](O1)c2cccc(c2)C(F)(F)F)c3cccc(c3)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N10 compound treatment 1221200.0 34400.0 0.58 1215120.0 25500.0 0.46 0.7315 0.9937 3001174 BCB02_000217 Cc1ccc(cc1)C2C3C(CN2S(=O)(=O)c4ccc(C)cc4)C5C(CC3=O)C(=O)N(C5=O)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N11 compound treatment 1217880.0 31100.0 0.52 1197240.0 7590.0 0.14 0.4644 0.8636 3092788 BCB02_000218 CC(C)OC(=O)/C=C/1\C[C@H](O[C@H](O1)c2ccccc2C(F)(F)F)c3ccccc3C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N12 compound treatment 1198240.0 11400.0 0.19 1188480.0 -1170.0 -0.02 0.1204 0.6252 3092789 BCB02_000219 CCN1C(=O)C2CC(=O)C3C(N(CC3C2C1=O)S(=O)(=O)c4ccc(C)cc4)c5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N13 compound treatment 1172920.0 -13900.0 -0.23 1175560.0 -14100.0 -0.25 -0.3438 -0.999 3001175 BCB02_000220 CON(C)C(=O)/C=C/1\C[C@H](O[C@H](O1)c2cccc(Cl)c2)c3cccc(Cl)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N14 compound treatment 1208000.0 21200.0 0.35 1208960.0 19300.0 0.35 0.4968 1.0 3092790 BCB02_000221 CC[C@@H]1[C@@H]2[C@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)CC5C2C(=O)N(CC)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N15 compound treatment 1202400.0 15600.0 0.26 1208080.0 18400.0 0.33 0.4193 0.9929 3001176 BCB02_000222 CC(C)OC(=O)CC(=O)CC(O)c1ccc(cc1)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N16 mock treatment 1196280.0 9480.0 0.16 1192880.0 3230.0 0.06 0.1532 0.9073 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N17 mock treatment 1181920.0 -4880.0 -0.08 1186240.0 -3410.0 -0.06 -0.1013 -0.9902 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N18 mock treatment 1182760.0 -4040.0 -0.07 1198480.0 8830.0 0.16 0.0646 0.3738 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N19 mock treatment 1183960.0 -2840.0 -0.05 1185320.0 -4330.0 -0.08 -0.0889 -0.9718 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N20 mock treatment 1183040.0 -3760.0 -0.06 1182200.0 -7450.0 -0.13 -0.1395 -0.9404 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N21 mock treatment 1145400.0 -41400.0 -0.69 1151120.0 -38500.0 -0.69 -0.9809 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N22 mock treatment 1171520.0 -15300.0 -0.26 1174480.0 -15200.0 -0.27 -0.3742 -0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N23 mock treatment 1152800.0 -34000.0 -0.57 1158920.0 -30700.0 -0.55 -0.7939 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 N24 mock treatment 1168880.0 -17900.0 -0.3 1172400.0 -17300.0 -0.31 -0.4319 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O01 compound treatment 1258800.0 72000.0 1.2 1257120.0 67500.0 1.22 1.7115 1.0 3092791 BCB02_000223 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccc(Br)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O02 compound treatment 1114200.0 -72600.0 -1.21 1132960.0 -56700.0 -1.02 -1.5814 -0.9963 3001177 BCB02_000224 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccco3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O03 compound treatment 1231840.0 45000.0 0.75 1239160.0 49500.0 0.89 1.1636 0.9965 3092792 BCB02_000225 COc1ccc(NN2C3C(C=CC2C(O)c4ccc(OC)c(OCc5ccccc5)c4)C(=O)N(C6CCCCC6)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O04 compound treatment 1191080.0 4280.0 0.07 1160360.0 -29300.0 -0.53 -0.3226 -0.6057 3001178 BCB02_000226 CCOC(=O)C1=CC[C@H](N([C@@H]1C#N)S(=O)(=O)c2ccc(C)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O05 compound treatment 1105800.0 -81000.0 -1.36 1049880.0 -140000.0 -2.52 -2.7393 -0.9578 3092860 BCB02_000227 COc1ccc(NN2C3C(C=CC2C(O)c4ccccn4)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O06 compound treatment 1243320.0 56500.0 0.95 1231440.0 41800.0 0.75 1.2011 0.9936 3001179 BCB02_000228 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)CC[Si](C)(C)C)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O07 compound treatment 1187360.0 557.0 0.01 1184920.0 -4730.0 -0.09 -0.0537 -0.6262 3092861 BCB02_000229 CCOc1cc(ccc1O)C(O)C2C=CC3C(N2Nc4ccc(OC)cc4)C(=O)N(C5CCCCC5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O08 compound treatment 1167800.0 -19000.0 -0.32 1129080.0 -60600.0 -1.09 -0.9966 -0.8767 3001245 BCB02_000230 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3cccn3C(=O)OC(C)(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O09 compound treatment 1208840.0 22000.0 0.37 1197440.0 7790.0 0.14 0.36 0.9123 3092862 BCB02_000231 COc1ccc(NN2C3C(C=CC2C(O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O10 compound treatment 1190160.0 3360.0 0.06 1195520.0 5870.0 0.11 0.1145 0.9563 3001246 BCB02_000232 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccc(C#N)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O11 compound treatment 1203960.0 17200.0 0.29 1196440.0 6790.0 0.12 0.2895 0.9276 3092863 BCB02_000233 Cc1ccc(NN2C3C(C=CC2C(O)c4c(F)cccc4Cl)C(=O)N(C5CCCCC5)C3=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O12 compound treatment 1084040.0 -103000.0 -1.72 1034360.0 -155000.0 -2.8 -3.1945 -0.9727 3001247 BCB02_000234 CCOC(=O)C1=CCC(NC1)c2cc3ccccc3[nH]2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O13 compound treatment 1210840.0 24000.0 0.4 1209760.0 20100.0 0.36 0.5406 0.9986 3092864 BCB02_000235 OC(C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O14 compound treatment 1188960.0 2160.0 0.04 1181520.0 -8130.0 -0.15 -0.0781 -0.5175 3001248 BCB02_000236 CCOC(=O)C1=CCC(N(C1)S(=O)(=O)c2ccccc2[N+](=O)[O-])c3cc4ccccc4[nH]3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O15 compound treatment 1194360.0 7560.0 0.13 1199200.0 9550.0 0.17 0.211 0.9886 3092865 BCB02_000237 CCC(CC)C(O)C1C=CC2C(N1Nc3ccccc3F)C(=O)N(C2=O)c4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O16 mock treatment 1169840.0 -17000.0 -0.28 1170320.0 -19300.0 -0.35 -0.447 -0.9948 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O17 mock treatment 1199080.0 12300.0 0.21 1195440.0 5790.0 0.1 0.219 0.9505 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O18 mock treatment 1201520.0 14700.0 0.25 1191080.0 1430.0 0.03 0.1923 0.7767 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O19 mock treatment 1169400.0 -17400.0 -0.29 1171160.0 -18500.0 -0.33 -0.4415 -0.9977 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O20 mock treatment 1168960.0 -17800.0 -0.3 1164440.0 -25200.0 -0.45 -0.5324 -0.9793 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O21 mock treatment 1175960.0 -10800.0 -0.18 1175800.0 -13900.0 -0.25 -0.3048 -0.9877 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O22 mock treatment 1166720.0 -20100.0 -0.34 1169960.0 -19700.0 -0.35 -0.4886 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O23 mock treatment 1152680.0 -34100.0 -0.57 1161600.0 -28100.0 -0.51 -0.7612 -0.9981 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 O24 mock treatment 1172960.0 -13800.0 -0.23 1179480.0 -10200.0 -0.18 -0.2934 -0.9933 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P01 compound treatment 1266200.0 79400.0 1.33 1265000.0 75300.0 1.36 1.8994 0.9999 3001249 BCB02_000238 CC(C)OC(=O)CC(=O)CC(O)c1cccc(c1)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P02 compound treatment 1250320.0 63500.0 1.06 1245480.0 55800.0 1.01 1.4628 0.9996 3092866 BCB02_000239 CC[C@@H]1[C@H]2[C@@H]([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)CC5C2C(=O)N(CC)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P03 compound treatment 1249000.0 62200.0 1.04 1226080.0 36400.0 0.66 1.2001 0.9753 3001250 BCB02_000240 CC(C)OC(=O)CC(=O)CC(O)c1cccc(C#N)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P04 compound treatment 1241760.0 55000.0 0.92 1236240.0 46600.0 0.84 1.2438 0.999 3092867 BCB02_000241 CCOC(=O)C1=CC[C@H](N([C@H]1CC)S(=O)(=O)c2ccc(C)cc2)c3ccc(OC)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P05 compound treatment 1228600.0 41800.0 0.7 1221640.0 32000.0 0.58 0.9021 0.9954 3001251 BCB02_000242 CC(C)OC(=O)CC(=O)CC(O)c1ccc(C#N)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P06 compound treatment 1212520.0 25700.0 0.43 1213960.0 24300.0 0.44 0.614 1.0 3092868 BCB02_000243 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P07 compound treatment 1224440.0 37600.0 0.63 1211480.0 21800.0 0.39 0.7234 0.9743 3001252 BCB02_000244 COC(=O)C1=CCC(CC1)(C=C)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P08 compound treatment 1068200.0 -119000.0 -1.98 1083960.0 -106000.0 -1.9 -2.75 -0.9998 3092869 BCB02_000245 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3cccc(Cl)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P09 compound treatment 1218680.0 31900.0 0.53 1214920.0 25300.0 0.46 0.6991 0.9969 3001253 BCB02_000246 COC(=O)/C=C(/CC(O)c1cccc(Cl)c1)\OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P10 compound treatment 1214080.0 27300.0 0.46 1204720.0 15100.0 0.27 0.5147 0.9692 3092870 BCB02_000247 CCOC(=O)C1=CC[C@H](N(C1)S(=O)(=O)c2ccc(C)cc2)c3ccccc3C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P11 compound treatment 1208000.0 21200.0 0.35 1198560.0 8910.0 0.16 0.3643 0.9357 3001254 BCB02_000248 OC(C/C(=C/C(=O)OCCF)/OCCF)c1cccc(Cl)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P12 compound treatment 1217640.0 30800.0 0.52 1207600.0 17900.0 0.32 0.5935 0.9746 3092871 BCB02_000249 CCOC(=O)C1=CC[C@H](N([C@H]1c2cccc(Br)c2)S(=O)(=O)c3ccc(C)cc3)c4ccc(OCC=C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P13 compound treatment 1183320.0 -3480.0 -0.06 1182320.0 -7330.0 -0.13 -0.1347 -0.9324 3001255 BCB02_000250 CCO/C(=C\C(=O)OC)/CC(O)c1cccc(Cl)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P14 compound treatment 1179960.0 -6840.0 -0.11 1195640.0 5990.0 0.11 -0.0047 -0.03 3092774 BCB02_000251 CC[C@@H]1C(Sc2ccccc2)C([C@@H](N1S(=O)(=O)c3ccc(C)cc3)c4ccc(C)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P15 compound treatment 1188200.0 1400.0 0.02 1194640.0 4990.0 0.09 0.08 0.8624 3092872 BCB02_000252 FCCOC(=O)C1=CCC(O1)c2cccc(Cl)c2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P16 mock treatment 1187880.0 1080.0 0.02 1176880.0 -12800.0 -0.23 -0.15 -0.6498 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P17 mock treatment 1192200.0 5400.0 0.09 1180920.0 -8730.0 -0.16 -0.0474 -0.2613 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P18 mock treatment 1167000.0 -19800.0 -0.33 1162120.0 -27500.0 -0.5 -0.5851 -0.9808 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P19 mock treatment 1166400.0 -20400.0 -0.34 1163320.0 -26300.0 -0.47 -0.5769 -0.987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P20 mock treatment 1166920.0 -19900.0 -0.33 1161960.0 -27700.0 -0.5 -0.5881 -0.9806 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P21 mock treatment 1151400.0 -35400.0 -0.59 1154520.0 -35100.0 -0.63 -0.8665 -0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P22 mock treatment 1173880.0 -12900.0 -0.22 1178560.0 -11100.0 -0.2 -0.2943 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P23 mock treatment 1162240.0 -24600.0 -0.41 1173920.0 -15700.0 -0.28 -0.4911 -0.9835 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2088 P24 mock treatment 1191040.0 4240.0 0.07 1192640.0 2990.0 0.05 0.0882 0.9907 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A01 compound treatment 1093760.0 -102000.0 -1.71 1084480.0 -114000.0 -2.06 -2.6626 -0.9957 3186889 PK04_093001 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A02 compound treatment 1144400.0 -51400.0 -0.86 1143160.0 -55500.0 -1.0 -1.3158 -0.9972 3067555 PK04_093002 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A03 compound treatment 1136560.0 -59200.0 -0.99 1134120.0 -64600.0 -1.16 -1.5238 -0.9968 3186890 PK04_093003 CN(C)C(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A04 compound treatment 742880.0 -453000.0 -7.58 739560.0 -459000.0 -8.27 -11.2089 -0.999 3186891 PK04_093004 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A05 compound treatment 763000.0 -433000.0 -7.24 760400.0 -438000.0 -7.9 -10.7054 -0.9991 3067558 PK04_093005 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A06 compound treatment 732120.0 -464000.0 -7.76 733680.0 -465000.0 -8.38 -11.4112 -0.9993 3186892 PK04_093006 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A07 compound treatment 803880.0 -392000.0 -6.56 802440.0 -396000.0 -7.14 -9.686 -0.9991 3067559 PK04_093007 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A08 compound treatment 843360.0 -352000.0 -5.9 841120.0 -358000.0 -6.44 -8.7261 -0.999 3186893 PK04_093008 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A09 compound treatment 1165880.0 -29900.0 -0.5 1160200.0 -38500.0 -0.69 -0.8445 -0.9872 3186894 PK04_093009 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A10 compound treatment 721200.0 -475000.0 -7.94 724040.0 -475000.0 -8.55 -11.6632 -0.9993 3067560 PK04_093010 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A11 compound treatment 1042840.0 -153000.0 -2.56 1047240.0 -151000.0 -2.73 -3.7396 -0.9995 3186895 PK04_093011 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A12 compound treatment 1034400.0 -161000.0 -2.7 1045640.0 -153000.0 -2.76 -3.8599 -0.9999 3186896 PK04_093012 NC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A13 mock treatment 1195400.0 -397.0 -0.01 1191960.0 -6740.0 -0.12 -0.0906 -0.7446 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A14 mock treatment 1165760.0 -30000.0 -0.5 1166920.0 -31800.0 -0.57 -0.7603 -0.9979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A15 compound treatment 900840.0 -295000.0 -4.94 938360.0 -260000.0 -4.69 -6.8071 -0.9997 3067562 PK04_093013 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A16 compound treatment 1136160.0 -59600.0 -1.0 1146800.0 -51900.0 -0.94 -1.3669 -0.9995 3186897 PK04_093014 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A17 compound treatment 1137680.0 -58100.0 -0.97 1146480.0 -52200.0 -0.94 -1.353 -0.9999 3067564 PK04_093015 NC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A18 compound treatment 765600.0 -430000.0 -7.2 783240.0 -415000.0 -7.49 -10.3836 -0.9998 3186898 PK04_093016 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A19 compound treatment 1024720.0 -171000.0 -2.86 1049040.0 -150000.0 -2.7 -3.9311 -0.9996 3186899 PK04_093017 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A20 compound treatment 1093480.0 -102000.0 -1.71 1097640.0 -101000.0 -1.82 -2.4983 -0.9995 3067604 PK04_093018 COCCCNC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A21 compound treatment 1152360.0 -43400.0 -0.73 1148000.0 -50700.0 -0.91 -1.16 -0.9936 3186900 PK04_093019 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A22 compound treatment 1137560.0 -58200.0 -0.97 1140720.0 -58000.0 -1.04 -1.4278 -0.9994 3067607 PK04_093020 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A23 compound treatment 1132600.0 -63200.0 -1.06 1142320.0 -56400.0 -1.02 -1.4661 -0.9998 3186901 PK04_093021 NC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 A24 compound treatment 1055680.0 -140000.0 -2.34 1027680.0 -171000.0 -3.08 -3.8369 -0.9909 3186902 PK04_093022 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B01 compound treatment 1001400.0 -194000.0 -3.25 995440.0 -203000.0 -3.66 -4.8899 -0.9983 3067612 PK04_093023 COC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B02 compound treatment 1186040.0 -9760.0 -0.16 1205240.0 6540.0 0.12 -0.0322 -0.1598 3186903 PK04_093024 NC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B03 compound treatment 628800.0 -567000.0 -9.49 641480.0 -557000.0 -10.04 -13.8084 -0.9996 3067614 PK04_093025 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B04 compound treatment 1215640.0 19800.0 0.33 1212200.0 13500.0 0.24 0.4068 0.9883 3186904 PK04_093026 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B05 compound treatment 989680.0 -206000.0 -3.45 888920.0 -310000.0 -5.58 -6.3857 -0.9732 3186905 PK04_093027 COC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B06 compound treatment 1165480.0 -30300.0 -0.51 1144160.0 -54500.0 -0.98 -1.0536 -0.9527 3068180 PK04_093028 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B07 compound treatment 416720.0 -779000.0 -13.04 416720.0 -782000.0 -14.09 -19.1814 -0.9992 3186906 PK04_093029 COC(=O)[C@H]1N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B08 compound treatment 1075320.0 -120000.0 -2.02 1046480.0 -152000.0 -2.74 -3.365 -0.9885 3186992 PK04_093030 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B09 compound treatment 749720.0 -446000.0 -7.46 753240.0 -445000.0 -8.03 -10.9537 -0.9993 3068181 PK04_093031 COC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B10 compound treatment 787840.0 -408000.0 -6.83 790160.0 -409000.0 -7.36 -10.0323 -0.9993 3186993 PK04_093032 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B11 compound treatment 1142160.0 -53600.0 -0.9 1144600.0 -54100.0 -0.97 -1.324 -0.9992 3068182 PK04_093033 COC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B12 compound treatment 1158840.0 -37000.0 -0.62 1166800.0 -31900.0 -0.57 -0.8438 -0.9993 3186994 PK04_093034 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B13 mock treatment 1147080.0 -48700.0 -0.82 1160880.0 -37800.0 -0.68 -1.0583 -0.996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B14 mock treatment 1201080.0 5280.0 0.09 1215840.0 17100.0 0.31 0.2808 0.8744 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B15 compound treatment 630080.0 -566000.0 -9.47 631720.0 -567000.0 -10.22 -13.9176 -0.9993 3068183 PK04_093035 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B16 compound treatment 1186720.0 -9080.0 -0.15 1179320.0 -19400.0 -0.35 -0.3544 -0.9305 3186995 PK04_093036 NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B17 compound treatment 1138320.0 -57500.0 -0.96 1139120.0 -59600.0 -1.07 -1.4392 -0.9985 3186996 PK04_093037 COC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B18 compound treatment 1148400.0 -47400.0 -0.79 1165360.0 -33300.0 -0.6 -0.9856 -0.9906 3068184 PK04_093038 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B19 compound treatment 979240.0 -217000.0 -3.62 990280.0 -208000.0 -3.76 -5.2179 -0.9998 3186997 PK04_093039 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B20 compound treatment 734600.0 -461000.0 -7.72 765560.0 -433000.0 -7.8 -10.9757 -1.0 3186998 PK04_093040 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B21 compound treatment 998280.0 -198000.0 -3.31 936520.0 -262000.0 -4.72 -5.6775 -0.9848 3068185 PK04_093041 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B22 compound treatment 1082440.0 -113000.0 -1.9 1092160.0 -107000.0 -1.92 -2.6987 -1.0 3186999 PK04_093042 CN(C)C(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B23 compound treatment 1111440.0 -84400.0 -1.41 1135720.0 -63000.0 -1.13 -1.8006 -0.9941 3068186 PK04_093043 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 B24 compound treatment 757800.0 -438000.0 -7.33 836560.0 -362000.0 -6.52 -9.7966 -0.9983 3187000 PK04_093044 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C01 compound treatment 919800.0 -276000.0 -4.62 948920.0 -250000.0 -4.5 -6.4482 -0.9999 3187001 PK04_093045 CN(C)C(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C02 compound treatment 1221760.0 26000.0 0.43 1205680.0 6980.0 0.13 0.3961 0.8758 3068187 PK04_093046 CN(C)C(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C03 compound treatment 694320.0 -501000.0 -8.39 723680.0 -475000.0 -8.56 -11.9859 -1.0 3187002 PK04_093047 COCCCNC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C04 compound treatment 1174960.0 -20800.0 -0.35 1172520.0 -26200.0 -0.47 -0.5801 -0.9889 3068188 PK04_093048 NC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C05 compound treatment 646160.0 -550000.0 -9.2 651080.0 -548000.0 -9.87 -13.4807 -0.9994 3187003 PK04_093049 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C06 compound treatment 1187640.0 -8160.0 -0.14 1179160.0 -19500.0 -0.35 -0.3455 -0.9149 3187004 PK04_093050 CN(C)C(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C07 compound treatment 1068880.0 -127000.0 -2.12 1006560.0 -192000.0 -3.46 -3.9497 -0.9725 3068189 PK04_093051 NC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C08 compound treatment 1191120.0 -4680.0 -0.08 1189800.0 -8900.0 -0.16 -0.1688 -0.9456 3187005 PK04_093052 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C09 compound treatment 774240.0 -422000.0 -7.05 739480.0 -459000.0 -8.27 -10.8389 -0.9969 3187006 PK04_093053 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C10 compound treatment 1126520.0 -69300.0 -1.16 1092760.0 -106000.0 -1.91 -2.1695 -0.9714 3068190 PK04_093054 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C11 mock treatment 1212000.0 16200.0 0.27 1216520.0 17800.0 0.32 0.4187 0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C12 mock treatment 1178320.0 -17500.0 -0.29 1182280.0 -16400.0 -0.3 -0.416 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C13 compound treatment 995960.0 -200000.0 -3.34 1007880.0 -191000.0 -3.44 -4.7958 -0.9999 3187007 PK04_093055 COC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C14 compound treatment 1098280.0 -97500.0 -1.63 1153720.0 -45000.0 -0.81 -1.727 -0.9478 3068191 PK04_093056 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C15 mock treatment 1185040.0 -10800.0 -0.18 1196680.0 -2020.0 -0.04 -0.1531 -0.8334 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C16 mock treatment 1154600.0 -41200.0 -0.69 1165000.0 -33700.0 -0.61 -0.9169 -0.998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C17 compound treatment 1107080.0 -88700.0 -1.48 1105680.0 -93000.0 -1.68 -2.2349 -0.9982 3187008 PK04_093057 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C18 compound treatment 810720.0 -385000.0 -6.44 913280.0 -285000.0 -5.14 -8.193 -0.9937 3068193 PK04_093058 COCCCNC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C19 compound treatment 961400.0 -234000.0 -3.92 984080.0 -215000.0 -3.87 -5.508 -1.0 3187009 PK04_093059 COC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C20 compound treatment 1031320.0 -164000.0 -2.75 1092840.0 -106000.0 -1.91 -3.295 -0.9839 3187010 PK04_093060 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C21 compound treatment 982560.0 -213000.0 -3.57 976000.0 -223000.0 -4.01 -5.3605 -0.9983 3068197 PK04_093061 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C22 compound treatment 1125440.0 -70400.0 -1.18 1138840.0 -59900.0 -1.08 -1.5952 -0.999 3187011 PK04_093062 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C23 compound treatment 1142040.0 -53800.0 -0.9 1139080.0 -59600.0 -1.07 -1.3957 -0.9961 3068199 PK04_093063 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 C24 compound treatment 1101760.0 -94000.0 -1.57 1078000.0 -121000.0 -2.17 -2.6505 -0.9874 3187012 PK04_093064 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)N3CCCCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D01 compound treatment 1157880.0 -37900.0 -0.63 1161240.0 -37500.0 -0.67 -0.926 -0.9995 3187091 PK04_093065 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D02 compound treatment 1171840.0 -24000.0 -0.4 1165800.0 -32900.0 -0.59 -0.7027 -0.9819 3068202 PK04_093066 CN(C)C(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D03 compound treatment 1130640.0 -65200.0 -1.09 1136520.0 -62200.0 -1.12 -1.5632 -0.9999 3187092 PK04_093067 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D04 compound treatment 1226280.0 30500.0 0.51 1226240.0 27500.0 0.5 0.7115 0.9999 3187093 PK04_093068 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D05 compound treatment 1127400.0 -68400.0 -1.14 1110440.0 -88300.0 -1.59 -1.9338 -0.987 3068220 PK04_093069 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D06 compound treatment 1065240.0 -131000.0 -2.18 1073920.0 -125000.0 -2.25 -3.1346 -0.9999 3187094 PK04_093070 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D07 compound treatment 312880.0 -883000.0 -14.78 321920.0 -877000.0 -15.8 -21.6179 -0.9994 3068223 PK04_093071 COC(=O)[C@H]1COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D08 compound treatment 974360.0 -221000.0 -3.71 966280.0 -232000.0 -4.19 -5.5814 -0.9981 3187095 PK04_093072 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D09 compound treatment 1120560.0 -75200.0 -1.26 1109560.0 -89100.0 -1.61 -2.026 -0.9927 3068225 PK04_093073 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D10 compound treatment 1169960.0 -25800.0 -0.43 1166360.0 -32300.0 -0.58 -0.7178 -0.9892 3187096 PK04_093074 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D11 mock treatment 1209080.0 13300.0 0.22 1224640.0 25900.0 0.47 0.4876 0.9423 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D12 mock treatment 1215200.0 19400.0 0.32 1211920.0 13200.0 0.24 0.398 0.9884 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D13 compound treatment 841640.0 -354000.0 -5.93 955640.0 -243000.0 -4.38 -7.2874 -0.9889 3187097 PK04_093075 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D14 compound treatment 830600.0 -365000.0 -6.11 840920.0 -358000.0 -6.45 -8.8796 -0.9996 3068228 PK04_093076 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D15 mock treatment 1167320.0 -28500.0 -0.48 1186600.0 -12100.0 -0.22 -0.4912 -0.9372 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D16 mock treatment 1194640.0 -1160.0 -0.02 1188480.0 -10200.0 -0.18 -0.1439 -0.7771 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D17 compound treatment 1123920.0 -71900.0 -1.2 1117680.0 -81000.0 -1.46 -1.8828 -0.9954 3187098 PK04_093077 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D18 compound treatment 883720.0 -312000.0 -5.22 946200.0 -253000.0 -4.55 -6.9098 -0.9976 3187099 PK04_093078 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D19 compound treatment 656560.0 -539000.0 -9.02 724760.0 -474000.0 -8.54 -12.4189 -0.9996 3068229 PK04_093079 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D20 compound treatment 833480.0 -362000.0 -6.06 858280.0 -340000.0 -6.13 -8.6244 -1.0 3187100 PK04_093080 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D21 compound treatment 1077280.0 -119000.0 -1.98 1091600.0 -107000.0 -1.93 -2.7669 -0.9999 3068232 PK04_093081 COC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D22 compound treatment 1140240.0 -55600.0 -0.93 1147280.0 -51400.0 -0.93 -1.3125 -1.0 3187101 PK04_093082 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D23 compound treatment 1008480.0 -187000.0 -3.13 1016440.0 -182000.0 -3.28 -4.5386 -0.9997 3187102 PK04_093083 COC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 D24 compound treatment 1132920.0 -62900.0 -1.05 1149200.0 -49500.0 -0.89 -1.3747 -0.9966 3068234 PK04_093084 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E01 mock treatment 1227440.0 31600.0 0.53 1222880.0 24200.0 0.44 0.6825 0.9953 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E02 mock treatment 1250320.0 54500.0 0.91 1223880.0 25200.0 0.45 0.9659 0.948 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E03 compound treatment 884160.0 -312000.0 -5.22 852160.0 -347000.0 -6.24 -8.1026 -0.996 3187103 PK04_093085 COC(=O)[C@H]1N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E04 compound treatment 1155960.0 -39800.0 -0.67 1130360.0 -68300.0 -1.23 -1.3421 -0.9585 3187104 PK04_093086 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E05 compound treatment 1214200.0 18400.0 0.31 1211680.0 13000.0 0.23 0.3831 0.9908 3068237 PK04_093087 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E06 compound treatment 1200120.0 4320.0 0.07 1226440.0 27700.0 0.5 0.4045 0.8011 3187105 PK04_093088 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E07 compound treatment 1190800.0 -5000.0 -0.08 1185160.0 -13500.0 -0.24 -0.2317 -0.8982 3068240 PK04_093089 COC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E08 compound treatment 1203800.0 8000.0 0.13 1205680.0 6980.0 0.13 0.1836 0.9995 3187106 PK04_093090 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E09 mock treatment 1222560.0 26800.0 0.45 1206800.0 8100.0 0.15 0.4198 0.8913 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E10 mock treatment 1219200.0 23400.0 0.39 1219200.0 20500.0 0.37 0.5381 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E11 compound treatment 1126360.0 -69400.0 -1.16 1111680.0 -87000.0 -1.57 -1.9303 -0.9891 3068242 PK04_093091 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E12 compound treatment 803840.0 -392000.0 -6.56 789280.0 -409000.0 -7.38 -9.8542 -0.9983 3187107 PK04_093092 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E13 compound treatment 1066360.0 -129000.0 -2.17 1107320.0 -91400.0 -1.65 -2.6959 -0.9908 3068264 PK04_093093 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E14 compound treatment 1186920.0 -8880.0 -0.15 1174320.0 -24400.0 -0.44 -0.4157 -0.8964 3187108 PK04_093094 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E15 compound treatment 745200.0 -451000.0 -7.54 828280.0 -370000.0 -6.67 -10.0512 -0.9981 3187109 PK04_093095 COC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E16 compound treatment 832720.0 -363000.0 -6.08 851120.0 -348000.0 -6.26 -8.7246 -0.9999 3068267 PK04_093096 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E17 mock treatment 1180080.0 -15700.0 -0.26 1180440.0 -18300.0 -0.33 -0.4187 -0.9938 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E18 mock treatment 1187160.0 -8640.0 -0.14 1182960.0 -15700.0 -0.28 -0.3028 -0.9511 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E19 compound treatment 1040480.0 -155000.0 -2.6 1056440.0 -142000.0 -2.56 -3.6503 -1.0 3187110 PK04_093097 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E20 compound treatment 1120720.0 -75100.0 -1.26 1116200.0 -82500.0 -1.49 -1.9395 -0.9965 3187111 PK04_093098 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E21 compound treatment 865160.0 -331000.0 -5.53 763040.0 -436000.0 -7.85 -9.4628 -0.9853 3068269 PK04_093099 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E22 compound treatment 1131720.0 -64100.0 -1.07 1136480.0 -62200.0 -1.12 -1.551 -0.9998 3187184 PK04_093100 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E23 compound treatment 1131840.0 -64000.0 -1.07 1157240.0 -41500.0 -0.75 -1.2851 -0.9845 3068272 PK04_093101 COC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 E24 compound treatment 1138520.0 -57300.0 -0.96 1158480.0 -40200.0 -0.72 -1.1902 -0.9905 3187185 PK04_093102 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F01 mock treatment 1174600.0 -21200.0 -0.35 1187520.0 -11200.0 -0.2 -0.3933 -0.9641 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F02 mock treatment 1243040.0 47200.0 0.79 1240320.0 41600.0 0.75 1.0892 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F03 compound treatment 913600.0 -282000.0 -4.72 956840.0 -242000.0 -4.36 -6.4206 -0.9992 3068274 PK04_093103 COC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F04 compound treatment 1148680.0 -47100.0 -0.79 1136080.0 -62600.0 -1.13 -1.3554 -0.9846 3187186 PK04_093104 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F05 compound treatment 1205440.0 9640.0 0.16 1219880.0 21200.0 0.38 0.3839 0.9267 3068276 PK04_093105 COC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F06 compound treatment 1056280.0 -140000.0 -2.33 1061520.0 -137000.0 -2.47 -3.3986 -0.9996 3187187 PK04_093106 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F07 compound treatment 1175160.0 -20600.0 -0.35 1184200.0 -14500.0 -0.26 -0.429 -0.9905 3187188 PK04_093107 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F08 compound treatment 1104840.0 -91000.0 -1.52 1072200.0 -127000.0 -2.28 -2.688 -0.9807 3068278 PK04_093108 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F09 mock treatment 1195960.0 163.0 0.0 1201200.0 2500.0 0.04 0.0337 0.7486 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F10 mock treatment 1216520.0 20700.0 0.35 1205280.0 6580.0 0.12 0.329 0.8978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F11 compound treatment 1162440.0 -33400.0 -0.56 1170040.0 -28700.0 -0.52 -0.7599 -0.9992 3187189 PK04_093109 COC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F12 compound treatment 1178440.0 -17400.0 -0.29 1177960.0 -20700.0 -0.37 -0.4697 -0.9922 3068280 PK04_093110 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F13 compound treatment 1175160.0 -20600.0 -0.35 1138040.0 -60700.0 -1.09 -1.0171 -0.8873 3187190 PK04_093111 COC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F14 compound treatment 1098400.0 -97400.0 -1.63 1097680.0 -101000.0 -1.82 -2.4396 -0.9985 3187191 PK04_093112 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F15 compound treatment 1170560.0 -25200.0 -0.42 1176040.0 -22700.0 -0.41 -0.5874 -0.9999 3068282 PK04_093113 COC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F16 compound treatment 1162120.0 -33700.0 -0.56 1161200.0 -37500.0 -0.68 -0.8763 -0.9959 3187192 PK04_093114 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F17 mock treatment 1158680.0 -37100.0 -0.62 1162440.0 -36300.0 -0.65 -0.9012 -0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F18 mock treatment 1159360.0 -36400.0 -0.61 1164160.0 -34500.0 -0.62 -0.8712 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F19 compound treatment 1075320.0 -120000.0 -2.02 1076360.0 -122000.0 -2.2 -2.9843 -0.999 3187193 PK04_093115 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F20 compound treatment 1026600.0 -169000.0 -2.83 1019960.0 -179000.0 -3.22 -4.2793 -0.9979 3068312 PK04_093116 NC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F21 compound treatment 1064000.0 -132000.0 -2.21 1061960.0 -137000.0 -2.46 -3.3017 -0.9985 3068314 PK04_093117 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F22 compound treatment 1017520.0 -178000.0 -2.98 999360.0 -199000.0 -3.59 -4.6492 -0.9957 3187194 PK04_093118 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F23 compound treatment 1093520.0 -102000.0 -1.71 1126960.0 -71700.0 -1.29 -2.1243 -0.9904 3187195 PK04_093119 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 F24 compound treatment 1105760.0 -90000.0 -1.51 1125760.0 -72900.0 -1.31 -1.9947 -0.9977 3068317 PK04_093120 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G01 compound treatment 649760.0 -546000.0 -9.14 653600.0 -545000.0 -9.82 -13.406 -0.9994 3187196 PK04_093121 COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G02 compound treatment 1170600.0 -25200.0 -0.42 1198560.0 -143.0 0.0 -0.3 -0.7114 3068319 PK04_093122 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)N3CCCCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G03 mock treatment 1244880.0 49100.0 0.82 1253120.0 54400.0 0.98 1.2741 0.9961 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G04 mock treatment 1256440.0 60600.0 1.01 1265440.0 66700.0 1.2 1.5678 0.9964 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G05 compound treatment 1147800.0 -48000.0 -0.8 1166960.0 -31700.0 -0.57 -0.9724 -0.9861 3187197 PK04_093123 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G06 compound treatment 1233160.0 37400.0 0.63 1225400.0 26700.0 0.48 0.7822 0.9916 3187198 PK04_093124 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G07 compound treatment 1211960.0 16200.0 0.27 1216200.0 17500.0 0.32 0.4142 0.9971 3068323 PK04_093125 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G08 compound treatment 1198760.0 2960.0 0.05 1195360.0 -3340.0 -0.06 -0.0075 -0.0965 3187199 PK04_093126 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G09 compound treatment 699040.0 -497000.0 -8.31 648800.0 -550000.0 -9.91 -12.884 -0.9962 3068325 PK04_093127 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G10 compound treatment 1193880.0 -1920.0 -0.03 1169800.0 -28900.0 -0.52 -0.3909 -0.7492 3187200 PK04_093128 COCCCNC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G11 compound treatment 1006200.0 -190000.0 -3.17 948880.0 -250000.0 -4.5 -5.4263 -0.9853 3187201 PK04_093129 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G12 compound treatment 1016640.0 -179000.0 -3.0 914320.0 -284000.0 -5.12 -5.743 -0.9674 3068327 PK04_093130 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G13 compound treatment 1142200.0 -53600.0 -0.9 1137000.0 -61700.0 -1.11 -1.4203 -0.9943 3187202 PK04_093131 COC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G14 compound treatment 1024000.0 -172000.0 -2.87 1018760.0 -180000.0 -3.24 -4.3254 -0.9982 3187203 PK04_093132 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G15 compound treatment 923240.0 -273000.0 -4.56 930800.0 -268000.0 -4.83 -6.6383 -0.9996 3068330 PK04_093133 COC(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G16 compound treatment 1162160.0 -33600.0 -0.56 1162680.0 -36000.0 -0.65 -0.857 -0.9975 3068332 PK04_093134 NC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G17 compound treatment 1139640.0 -56200.0 -0.94 1134240.0 -64500.0 -1.16 -1.4858 -0.9945 3187278 PK04_093135 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G18 compound treatment 1172520.0 -23300.0 -0.39 1179920.0 -18800.0 -0.34 -0.5147 -0.9975 3187279 PK04_093136 COCCCNC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G19 mock treatment 1186640.0 -9160.0 -0.15 1198960.0 257.0 0.0 -0.1051 -0.6854 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G20 mock treatment 1174920.0 -20900.0 -0.35 1177680.0 -21000.0 -0.38 -0.5149 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G21 compound treatment 1128200.0 -67600.0 -1.13 1114560.0 -84100.0 -1.52 -1.8719 -0.9896 3187280 PK04_093137 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G22 compound treatment 1128280.0 -67500.0 -1.13 1112320.0 -86400.0 -1.56 -1.8995 -0.9876 3068361 PK04_093138 COCCCNC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G23 compound treatment 1149040.0 -46800.0 -0.78 1159520.0 -39200.0 -0.71 -1.0525 -0.9987 3187281 PK04_093139 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 G24 compound treatment 1106120.0 -89700.0 -1.5 1131200.0 -67500.0 -1.22 -1.9212 -0.9946 3187282 PK04_093140 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H01 compound treatment 690400.0 -505000.0 -8.46 698120.0 -501000.0 -9.02 -12.3579 -0.9995 3068365 PK04_093141 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H02 compound treatment 1205600.0 9800.0 0.16 1212680.0 14000.0 0.25 0.2941 0.9784 3187283 PK04_093142 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H03 mock treatment 1251160.0 55400.0 0.93 1237360.0 38700.0 0.7 1.1476 0.9901 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H04 mock treatment 1242160.0 46400.0 0.78 1230800.0 32100.0 0.58 0.9575 0.9895 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H05 compound treatment 1193000.0 -2800.0 -0.05 1203080.0 4380.0 0.08 0.0227 0.2472 3068368 PK04_093143 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H06 compound treatment 1132960.0 -62800.0 -1.05 1162520.0 -36200.0 -0.65 -1.2045 -0.9736 3187284 PK04_093144 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H07 compound treatment 1141440.0 -54400.0 -0.91 1147640.0 -51100.0 -0.92 -1.2938 -1.0 3187285 PK04_093145 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(CC=C)C1=O)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H08 compound treatment 853440.0 -342000.0 -5.73 820240.0 -378000.0 -6.82 -8.8728 -0.9963 3068370 PK04_093146 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H09 compound treatment 970480.0 -225000.0 -3.77 975200.0 -224000.0 -4.03 -5.5136 -0.9995 3187286 PK04_093147 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H10 compound treatment 1202040.0 6240.0 0.1 1186000.0 -12700.0 -0.23 -0.088 -0.3496 3187287 PK04_093148 CN(C)C(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H11 compound treatment 1156520.0 -39300.0 -0.66 1165800.0 -32900.0 -0.59 -0.884 -0.9987 3068373 PK04_093149 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H12 compound treatment 1207720.0 11900.0 0.2 1170480.0 -28200.0 -0.51 -0.2185 -0.4 3187288 PK04_093150 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCc3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H13 compound treatment 1000240.0 -196000.0 -3.27 1020600.0 -178000.0 -3.21 -4.5831 -1.0 3187289 PK04_093151 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3N(CC=C)C1=O)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H14 compound treatment 1034640.0 -161000.0 -2.7 1013360.0 -185000.0 -3.34 -4.2683 -0.9944 3068375 PK04_093152 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H15 compound treatment 1069440.0 -126000.0 -2.11 1056120.0 -143000.0 -2.57 -3.3117 -0.9953 3187290 PK04_093153 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H16 compound treatment 1148400.0 -47400.0 -0.79 1143520.0 -55200.0 -0.99 -1.2639 -0.9937 3187291 PK04_093154 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H17 compound treatment 1053040.0 -143000.0 -2.39 1034280.0 -164000.0 -2.96 -3.784 -0.9943 3068378 PK04_093155 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H18 compound treatment 1183360.0 -12400.0 -0.21 1167760.0 -30900.0 -0.56 -0.5414 -0.9098 3187292 PK04_093156 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H19 mock treatment 1161000.0 -34800.0 -0.58 1161240.0 -37500.0 -0.67 -0.889 -0.9973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H20 mock treatment 1147240.0 -48600.0 -0.81 1151880.0 -46800.0 -0.84 -1.1711 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H21 compound treatment 866720.0 -329000.0 -5.51 834720.0 -364000.0 -6.56 -8.5312 -0.9962 3187293 PK04_093157 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H22 compound treatment 1028120.0 -168000.0 -2.81 967320.0 -231000.0 -4.17 -4.932 -0.9814 3068380 PK04_093158 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H23 compound treatment 1125200.0 -70600.0 -1.18 1127520.0 -71200.0 -1.28 -1.7423 -0.9992 3068402 PK04_093159 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 H24 compound treatment 1130960.0 -64800.0 -1.09 1139720.0 -59000.0 -1.06 -1.5187 -0.9999 3187294 PK04_093160 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I01 compound treatment 1172680.0 -23100.0 -0.39 1173640.0 -25100.0 -0.45 -0.5929 -0.997 3068406 PK04_093161 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I02 compound treatment 989360.0 -206000.0 -3.45 996400.0 -202000.0 -3.64 -5.0201 -0.9996 3187295 PK04_093162 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I03 compound treatment 1196960.0 1160.0 0.02 1191240.0 -7460.0 -0.13 -0.0813 -0.5985 3068409 PK04_093163 COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I04 compound treatment 1230760.0 35000.0 0.59 1244320.0 45600.0 0.82 0.9949 0.9861 3187296 PK04_093164 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I05 mock treatment 1252880.0 57100.0 0.96 1249280.0 50600.0 0.91 1.3198 0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I06 mock treatment 1238680.0 42900.0 0.72 1234720.0 36000.0 0.65 0.9663 0.9987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I07 compound treatment 1203720.0 7920.0 0.13 1214840.0 16100.0 0.29 0.2993 0.9368 3187297 PK04_093165 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I08 compound treatment 1135280.0 -60500.0 -1.01 1114560.0 -84100.0 -1.52 -1.7881 -0.9808 3068413 PK04_093166 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I09 compound treatment 1046680.0 -149000.0 -2.5 1007040.0 -192000.0 -3.45 -4.2063 -0.9873 3187298 PK04_093167 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I10 compound treatment 1173440.0 -22400.0 -0.37 1213480.0 14800.0 0.27 -0.0763 -0.1661 3187366 PK04_093168 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I11 compound treatment 718200.0 -478000.0 -7.99 691280.0 -507000.0 -9.14 -12.1161 -0.9978 3068416 PK04_093169 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I12 compound treatment 645360.0 -550000.0 -9.21 532720.0 -666000.0 -12.0 -14.9981 -0.9915 3187367 PK04_093170 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I13 compound treatment 1168400.0 -27400.0 -0.46 1182080.0 -16600.0 -0.3 -0.536 -0.9787 3068419 PK04_093171 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I14 compound treatment 798840.0 -397000.0 -6.64 828680.0 -370000.0 -6.67 -9.4114 -1.0 3187368 PK04_093172 CN(C)C(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I15 compound treatment 865920.0 -330000.0 -5.52 844320.0 -354000.0 -6.38 -8.4183 -0.9974 3068421 PK04_093173 COC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I16 compound treatment 1158360.0 -37400.0 -0.63 1152160.0 -46500.0 -0.84 -1.036 -0.9897 3187369 PK04_093174 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I17 compound treatment 1183560.0 -12200.0 -0.2 1186040.0 -12700.0 -0.23 -0.3061 -0.9985 3068423 PK04_093175 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I18 compound treatment 1150520.0 -45300.0 -0.76 1149640.0 -49100.0 -0.88 -1.1608 -0.9971 3187370 PK04_093176 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I19 compound treatment 93680.0 -1100000.0 -18.44 99440.0 -1100000.0 -19.81 -27.0462 -0.9994 3187371 PK04_093177 COC(=O)[C@H]1N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I20 compound treatment 728600.0 -467000.0 -7.82 628880.0 -570000.0 -10.27 -12.788 -0.991 3068425 PK04_093178 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I21 mock treatment 1149360.0 -46400.0 -0.78 1169960.0 -28700.0 -0.52 -0.9157 -0.9805 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I22 mock treatment 1163480.0 -32300.0 -0.54 1174560.0 -24100.0 -0.43 -0.69 -0.9942 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I23 compound treatment 711960.0 -484000.0 -8.1 686520.0 -512000.0 -9.23 -12.2505 -0.9979 3187372 PK04_093179 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 I24 compound treatment 1134960.0 -60800.0 -1.02 1144480.0 -54200.0 -0.98 -1.4107 -0.9998 3068456 PK04_093180 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J01 compound treatment 949800.0 -246000.0 -4.12 982600.0 -216000.0 -3.89 -5.6641 -0.9996 3187373 PK04_093181 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3N(CC=C)C1=O)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J02 compound treatment 815840.0 -380000.0 -6.36 813240.0 -385000.0 -6.94 -9.4069 -0.999 3187374 PK04_093182 CN(C)C(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J03 compound treatment 1133560.0 -62200.0 -1.04 1140520.0 -58200.0 -1.05 -1.4777 -1.0 3068460 PK04_093183 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J04 compound treatment 1249240.0 53400.0 0.89 1229800.0 31100.0 0.56 1.0286 0.9746 3187375 PK04_093184 COCCCNC(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J05 mock treatment 1228120.0 32300.0 0.54 1242320.0 43600.0 0.79 0.9382 0.9834 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J06 mock treatment 1224400.0 28600.0 0.48 1237920.0 39200.0 0.71 0.8381 0.982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J07 compound treatment 1235640.0 39800.0 0.67 1218160.0 19500.0 0.35 0.7194 0.9549 3187376 PK04_093185 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J08 compound treatment 1147560.0 -48200.0 -0.81 1124560.0 -74100.0 -1.34 -1.5154 -0.9709 3068463 PK04_093186 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J09 compound treatment 1140160.0 -55600.0 -0.93 1122200.0 -76500.0 -1.38 -1.633 -0.9818 3187377 PK04_093187 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J10 compound treatment 1196480.0 683.0 0.01 1188920.0 -9780.0 -0.18 -0.1166 -0.6599 3068465 PK04_093188 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J11 compound treatment 1188320.0 -7480.0 -0.13 1185920.0 -12800.0 -0.23 -0.2513 -0.9589 3187378 PK04_093189 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(Cc5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J12 compound treatment 1192480.0 -3320.0 -0.06 1198000.0 -703.0 -0.01 -0.0482 -0.8467 3068467 PK04_093190 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J13 compound treatment 1188120.0 -7680.0 -0.13 1150040.0 -48700.0 -0.88 -0.7108 -0.8022 3187379 PK04_093191 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(Cc5ccccc5)C3=O)[C@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J14 compound treatment 1060840.0 -135000.0 -2.26 1067600.0 -131000.0 -2.36 -3.2672 -0.9997 3187380 PK04_093192 COCCCNC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J15 compound treatment 1144120.0 -51700.0 -0.86 1132640.0 -66100.0 -1.19 -1.4531 -0.9877 3068470 PK04_093193 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J16 compound treatment 843120.0 -353000.0 -5.9 770600.0 -428000.0 -7.71 -9.6273 -0.9913 3187381 PK04_093194 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J17 compound treatment 1157320.0 -38500.0 -0.64 1161480.0 -37200.0 -0.67 -0.9295 -0.9998 3187382 PK04_093195 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J18 compound treatment 1183040.0 -12800.0 -0.21 1163200.0 -35500.0 -0.64 -0.6033 -0.8946 3068473 PK04_093196 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J19 compound treatment 1118200.0 -77600.0 -1.3 1107600.0 -91100.0 -1.64 -2.0789 -0.9933 3187383 PK04_093197 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J20 compound treatment 1117360.0 -78400.0 -1.31 1138880.0 -59800.0 -1.08 -1.6903 -0.9952 3068475 PK04_093198 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J21 mock treatment 1155920.0 -39900.0 -0.67 1167640.0 -31100.0 -0.56 -0.8676 -0.9962 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J22 mock treatment 1160600.0 -35200.0 -0.59 1164800.0 -33900.0 -0.61 -0.8484 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J23 compound treatment 1110600.0 -85200.0 -1.43 1144400.0 -54300.0 -0.98 -1.7 -0.9831 3187384 PK04_093199 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 J24 compound treatment 772960.0 -423000.0 -7.08 937000.0 -262000.0 -4.72 -8.3376 -0.9805 3068477 PK04_093200 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K01 compound treatment 1211760.0 16000.0 0.27 1221280.0 22600.0 0.41 0.4765 0.9792 3187385 PK04_093201 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K02 compound treatment 1237680.0 41900.0 0.7 1221120.0 22400.0 0.4 0.7812 0.9657 3187386 PK04_093202 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K03 compound treatment 573560.0 -622000.0 -10.41 590040.0 -609000.0 -10.97 -15.1174 -0.9997 3187447 PK04_093203 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K04 compound treatment 1149880.0 -45900.0 -0.77 1168240.0 -30500.0 -0.55 -0.9314 -0.9864 3068500 PK04_093204 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K05 compound treatment 1164240.0 -31600.0 -0.53 1189720.0 -8980.0 -0.16 -0.4879 -0.8833 3187448 PK04_093205 COC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K06 compound treatment 1216560.0 20800.0 0.35 1200600.0 1900.0 0.03 0.2699 0.7729 3187449 PK04_093206 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K07 mock treatment 1241720.0 45900.0 0.77 1213880.0 15200.0 0.27 0.7368 0.9032 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K08 mock treatment 1232680.0 36900.0 0.62 1229400.0 30700.0 0.55 0.8275 0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K09 compound treatment 777960.0 -418000.0 -6.99 764520.0 -434000.0 -7.82 -10.4758 -0.9984 3068503 PK04_093207 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K10 compound treatment 1205040.0 9240.0 0.15 1183640.0 -15100.0 -0.27 -0.0825 -0.2642 3187450 PK04_093208 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K11 compound treatment 1186520.0 -9280.0 -0.16 1185160.0 -13500.0 -0.24 -0.2823 -0.9762 3068506 PK04_093209 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K12 compound treatment 884720.0 -311000.0 -5.21 775400.0 -423000.0 -7.63 -9.0739 -0.9827 3187451 PK04_093210 CN(C)C(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K13 compound treatment 1001440.0 -194000.0 -3.25 884080.0 -315000.0 -5.67 -6.3082 -0.9652 3187452 PK04_093211 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K14 compound treatment 1170840.0 -25000.0 -0.42 1148240.0 -50500.0 -0.91 -0.9382 -0.9377 3068509 PK04_093212 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K15 mock treatment 1191160.0 -4640.0 -0.08 1195840.0 -2860.0 -0.05 -0.0913 -0.9803 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K16 mock treatment 1204520.0 8720.0 0.15 1200800.0 2100.0 0.04 0.1299 0.8617 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K17 compound treatment 1182480.0 -13300.0 -0.22 1172040.0 -26700.0 -0.48 -0.4973 -0.939 3187453 PK04_093213 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K18 compound treatment 1079840.0 -116000.0 -1.94 1066200.0 -133000.0 -2.39 -3.0602 -0.9947 3187454 PK04_093214 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K19 compound treatment 1034640.0 -161000.0 -2.7 1088440.0 -110000.0 -1.99 -3.3117 -0.9887 3068511 PK04_093215 COC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K20 compound treatment 899160.0 -297000.0 -4.96 863560.0 -335000.0 -6.04 -7.7799 -0.9953 3187455 PK04_093216 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K21 compound treatment 1142280.0 -53500.0 -0.9 1160240.0 -38500.0 -0.69 -1.1233 -0.992 3068513 PK04_093217 COC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K22 compound treatment 1014760.0 -181000.0 -3.03 1028040.0 -171000.0 -3.07 -4.3165 -1.0 3187456 PK04_093218 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K23 mock treatment 1155640.0 -40200.0 -0.67 1175560.0 -23100.0 -0.42 -0.77 -0.9737 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 K24 mock treatment 1145640.0 -50200.0 -0.84 1153920.0 -44800.0 -0.81 -1.1641 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L01 compound treatment 709440.0 -486000.0 -8.14 703080.0 -496000.0 -8.93 -12.0694 -0.9989 3187457 PK04_093219 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L02 compound treatment 992880.0 -203000.0 -3.4 979040.0 -220000.0 -3.96 -5.1997 -0.9971 3068516 PK04_093220 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L03 compound treatment 1137880.0 -57900.0 -0.97 1141120.0 -57600.0 -1.04 -1.419 -0.9994 3187458 PK04_093221 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L04 compound treatment 703320.0 -492000.0 -8.24 719840.0 -479000.0 -8.63 -11.9283 -0.9997 3187459 PK04_093222 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L05 compound treatment 1154560.0 -41200.0 -0.69 1167200.0 -31500.0 -0.57 -0.8893 -0.9953 3068518 PK04_093223 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L06 compound treatment 1086080.0 -110000.0 -1.84 1135720.0 -63000.0 -1.13 -2.1007 -0.9733 3187460 PK04_093224 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L07 mock treatment 1222680.0 26900.0 0.45 1208400.0 9700.0 0.17 0.4417 0.9151 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L08 mock treatment 1219000.0 23200.0 0.39 1218000.0 19300.0 0.35 0.5204 0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L09 compound treatment 1179240.0 -16600.0 -0.28 1179560.0 -19100.0 -0.34 -0.4398 -0.9941 3068520 PK04_093225 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(CC=C)C1=O)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L10 compound treatment 1196400.0 603.0 0.01 1194720.0 -3980.0 -0.07 -0.0436 -0.6017 3187461 PK04_093226 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L11 compound treatment 1036760.0 -159000.0 -2.66 1027200.0 -172000.0 -3.09 -4.0669 -0.9972 3187462 PK04_093227 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L12 compound treatment 1190720.0 -5080.0 -0.08 1198360.0 -343.0 -0.01 -0.0644 -0.7566 3187463 PK04_093228 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L13 compound treatment 1145160.0 -50600.0 -0.85 1109480.0 -89200.0 -1.61 -1.7359 -0.9553 3068543 PK04_093229 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(Cc5ccccc5)C3=O)[C@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L14 compound treatment 1074880.0 -121000.0 -2.02 1014760.0 -184000.0 -3.31 -3.7743 -0.972 3187464 PK04_093230 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L15 mock treatment 1186400.0 -9400.0 -0.16 1193520.0 -5180.0 -0.09 -0.1772 -0.969 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L16 mock treatment 1183520.0 -12300.0 -0.21 1191720.0 -6980.0 -0.13 -0.2342 -0.9723 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L17 compound treatment 1137800.0 -58000.0 -0.97 1124400.0 -74300.0 -1.34 -1.6329 -0.9875 3068545 PK04_093231 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L18 compound treatment 1090680.0 -105000.0 -1.76 1049240.0 -149000.0 -2.69 -3.148 -0.9787 3187465 PK04_093232 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L19 compound treatment 1099320.0 -96500.0 -1.61 1101120.0 -97600.0 -1.76 -2.3848 -0.9991 3187466 PK04_093233 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L20 compound treatment 1153360.0 -42400.0 -0.71 1159440.0 -39300.0 -0.71 -1.0024 -1.0 3068547 PK04_093234 NC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L21 compound treatment 1119440.0 -76400.0 -1.28 1119840.0 -78900.0 -1.42 -1.9083 -0.9986 3187467 PK04_093235 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L22 compound treatment 1139280.0 -56500.0 -0.95 1153080.0 -45600.0 -0.82 -1.25 -0.9976 3068549 PK04_093236 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L23 mock treatment 1128360.0 -67400.0 -1.13 1176680.0 -22000.0 -0.4 -1.0786 -0.9016 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 L24 mock treatment 1154320.0 -41500.0 -0.69 1147440.0 -51300.0 -0.92 -1.1439 -0.9901 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M01 compound treatment 1227880.0 32100.0 0.54 1233960.0 35300.0 0.64 0.8288 0.9965 3187528 PK04_093237 COC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M02 compound treatment 1227160.0 31400.0 0.52 1212600.0 13900.0 0.25 0.5482 0.9427 3187529 PK04_093238 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M03 compound treatment 1243960.0 48200.0 0.81 1245240.0 46500.0 0.84 1.1628 0.9998 3068551 PK04_093239 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M04 compound treatment 826480.0 -369000.0 -6.18 708360.0 -490000.0 -8.83 -10.6172 -0.9847 3187530 PK04_093240 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M05 compound treatment 1222840.0 27000.0 0.45 1234720.0 36000.0 0.65 0.7789 0.9845 3068553 PK04_093241 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M06 compound treatment 1080560.0 -115000.0 -1.93 1140800.0 -57900.0 -1.04 -2.1013 -0.9584 3187531 PK04_093242 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M07 compound treatment 1194440.0 -1360.0 -0.02 1199840.0 1140.0 0.02 -0.0016 -0.0514 3187532 PK04_093243 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M08 compound treatment 1125560.0 -70200.0 -1.18 1137880.0 -60800.0 -1.1 -1.606 -0.9994 3068555 PK04_093244 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M09 mock treatment 1227480.0 31700.0 0.53 1237800.0 39100.0 0.7 0.873 0.9902 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M10 mock treatment 1216080.0 20300.0 0.34 1219320.0 20600.0 0.37 0.5027 0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M11 compound treatment 1160000.0 -35800.0 -0.6 1161840.0 -36900.0 -0.66 -0.8932 -0.9987 3187533 PK04_093245 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M12 compound treatment 975000.0 -221000.0 -3.69 930480.0 -268000.0 -4.83 -6.0299 -0.9912 3187534 PK04_093246 COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M13 mock treatment 1196480.0 683.0 0.01 1186960.0 -11700.0 -0.21 -0.1415 -0.6679 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M14 mock treatment 1197080.0 1280.0 0.02 1206640.0 7940.0 0.14 0.1163 0.8043 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M15 compound treatment 1047840.0 -148000.0 -2.48 1029560.0 -169000.0 -3.05 -3.9057 -0.9947 3068558 PK04_093247 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M16 compound treatment 1171480.0 -24300.0 -0.41 1145760.0 -52900.0 -0.95 -0.9622 -0.9279 3187535 PK04_093248 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M17 compound treatment 998160.0 -198000.0 -3.31 973440.0 -225000.0 -4.06 -5.2085 -0.9948 3068560 PK04_093249 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M18 compound treatment 673640.0 -522000.0 -8.74 673600.0 -525000.0 -9.46 -12.8686 -0.9992 3187536 PK04_093250 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M19 compound treatment 1140880.0 -54900.0 -0.92 1136400.0 -62300.0 -1.12 -1.4436 -0.9951 3187537 PK04_093251 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M20 compound treatment 1151600.0 -44200.0 -0.74 1156920.0 -41800.0 -0.75 -1.0553 -1.0 3068562 PK04_093252 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)N3CCOCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M21 compound treatment 1106160.0 -89600.0 -1.5 1109720.0 -89000.0 -1.6 -2.1943 -0.9994 3068586 PK04_093253 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M22 compound treatment 1110560.0 -85200.0 -1.43 1129680.0 -69000.0 -1.24 -1.888 -0.9977 3187538 PK04_093254 NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M23 compound treatment 1106240.0 -89600.0 -1.5 1108840.0 -89900.0 -1.62 -2.2046 -0.9993 3068589 PK04_093255 COC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 M24 compound treatment 660920.0 -535000.0 -8.95 703960.0 -495000.0 -8.91 -12.6323 -1.0 3187539 PK04_093256 NC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N01 compound treatment 892920.0 -303000.0 -5.07 894840.0 -304000.0 -5.47 -7.4552 -0.9993 3187540 PK04_093257 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3N(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N02 compound treatment 1245480.0 49700.0 0.83 1242640.0 43900.0 0.79 1.1477 0.9997 3187541 PK04_093258 CN(C)C(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N03 compound treatment 1167400.0 -28400.0 -0.48 1172640.0 -26100.0 -0.47 -0.6681 -1.0 3068594 PK04_093259 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(CC=C)C3=O)[C@@H](O2)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N04 compound treatment 1192160.0 -3640.0 -0.06 1188520.0 -10200.0 -0.18 -0.1728 -0.8938 3187542 PK04_093260 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N05 compound treatment 1198280.0 2480.0 0.04 1187960.0 -10700.0 -0.19 -0.1075 -0.5429 3068597 PK04_093261 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N06 compound treatment 1085760.0 -110000.0 -1.84 1067200.0 -132000.0 -2.37 -2.9774 -0.9922 3187543 PK04_093262 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N07 compound treatment 1122000.0 -73800.0 -1.23 1157840.0 -40900.0 -0.74 -1.3938 -0.9695 3187544 PK04_093263 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(CC=C)C3=O)[C@H](O2)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N08 compound treatment 884480.0 -311000.0 -5.21 968000.0 -231000.0 -4.16 -6.623 -0.9937 3068600 PK04_093264 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N09 mock treatment 1192680.0 -3120.0 -0.05 1203760.0 5060.0 0.09 0.0275 0.2623 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N10 mock treatment 1205920.0 10100.0 0.17 1209160.0 10500.0 0.19 0.253 0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N11 compound treatment 1146680.0 -49100.0 -0.82 1168480.0 -30200.0 -0.54 -0.9663 -0.98 3187545 PK04_093265 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N12 compound treatment 1172640.0 -23200.0 -0.39 1154160.0 -44500.0 -0.8 -0.8415 -0.9442 3187546 PK04_093266 COCCCNC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N13 mock treatment 1184320.0 -11500.0 -0.19 1186680.0 -12000.0 -0.22 -0.289 -0.9982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N14 mock treatment 1188520.0 -7280.0 -0.12 1175480.0 -23200.0 -0.42 -0.382 -0.8765 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N15 compound treatment 809920.0 -386000.0 -6.46 903800.0 -295000.0 -5.31 -8.3232 -0.9953 3068603 PK04_093267 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3N(CCS(=O)(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N16 compound treatment 1087000.0 -109000.0 -1.82 1102280.0 -96400.0 -1.74 -2.5158 -0.9997 3187547 PK04_093268 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N17 compound treatment 890240.0 -306000.0 -5.11 937360.0 -261000.0 -4.71 -6.9452 -0.9992 3068605 PK04_093269 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N18 compound treatment 1113760.0 -82000.0 -1.37 1125480.0 -73200.0 -1.32 -1.9036 -0.9998 3187548 PK04_093270 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N19 compound treatment 1127720.0 -68100.0 -1.14 1135040.0 -63700.0 -1.15 -1.6166 -1.0 3068607 PK04_093271 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N20 compound treatment 616600.0 -579000.0 -9.69 633000.0 -566000.0 -10.19 -14.0608 -0.9997 3186297 PK04_093272 NC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N21 compound treatment 1067680.0 -128000.0 -2.14 1109560.0 -89100.0 -1.61 -2.6517 -0.9899 3186298 PK04_093273 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(CC=C)C3=O)[C@@H](O2)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N22 compound treatment 1121320.0 -74500.0 -1.25 1137240.0 -61500.0 -1.11 -1.6643 -0.9983 3068610 PK04_093274 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N23 compound treatment 1117920.0 -77900.0 -1.3 1114160.0 -84500.0 -1.52 -1.9986 -0.997 3068635 PK04_093275 CC(=O)N1Cc2ccccc2C[C@]3(N=C(O[C@@H]3c4ccccc4)c5ccc(OCCCO)cc5)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 N24 compound treatment 1133640.0 -62200.0 -1.04 1131880.0 -66800.0 -1.2 -1.5868 -0.9973 3186299 PK04_093276 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O01 compound treatment 1224560.0 28800.0 0.48 1224400.0 25700.0 0.46 0.6677 0.9998 3068638 PK04_093277 COC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O02 compound treatment 1120720.0 -75100.0 -1.26 1134720.0 -64000.0 -1.15 -1.7035 -0.9991 3186300 PK04_093278 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O03 compound treatment 1103680.0 -92100.0 -1.54 1123000.0 -75700.0 -1.36 -2.0545 -0.9981 3068640 PK04_093279 COC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O04 compound treatment 682040.0 -514000.0 -8.6 847640.0 -351000.0 -6.33 -10.5519 -0.9886 3186301 PK04_093280 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O05 compound treatment 1177960.0 -17800.0 -0.3 1201880.0 3180.0 0.06 -0.1706 -0.5613 3068642 PK04_093281 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O06 compound treatment 1211080.0 15300.0 0.26 1205840.0 7140.0 0.13 0.2718 0.9494 3186302 PK04_093282 COCCCNC(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O07 compound treatment 1119880.0 -75900.0 -1.27 1107640.0 -91100.0 -1.64 -2.0585 -0.992 3186303 PK04_093283 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O08 compound treatment 647080.0 -549000.0 -9.18 793240.0 -405000.0 -7.31 -11.6587 -0.9936 3068645 PK04_093284 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O09 compound treatment 1120680.0 -75100.0 -1.26 1130600.0 -68100.0 -1.23 -1.7565 -0.9999 3186304 PK04_093285 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O10 compound treatment 1167440.0 -28400.0 -0.47 1159720.0 -39000.0 -0.7 -0.8322 -0.9818 3186305 PK04_093286 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O11 mock treatment 1186120.0 -9680.0 -0.16 1206080.0 7380.0 0.13 -0.0205 -0.098 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O12 mock treatment 1202840.0 7040.0 0.12 1181440.0 -17300.0 -0.31 -0.1366 -0.4107 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O13 compound treatment 852640.0 -343000.0 -5.74 881720.0 -317000.0 -5.71 -8.099 -1.0 3068648 PK04_093287 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O14 compound treatment 1161280.0 -34500.0 -0.58 1163960.0 -34700.0 -0.63 -0.8511 -0.9992 3186306 PK04_093288 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O15 compound treatment 766760.0 -429000.0 -7.18 864720.0 -334000.0 -6.02 -9.3318 -0.9961 3068650 PK04_093289 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O16 compound treatment 643840.0 -552000.0 -9.24 743080.0 -456000.0 -8.21 -12.336 -0.9983 3186307 PK04_093290 CN(C)C(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O17 compound treatment 631440.0 -564000.0 -9.44 639960.0 -559000.0 -10.07 -13.7965 -0.9995 3186308 PK04_093291 COC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O18 compound treatment 1127400.0 -68400.0 -1.14 1148040.0 -50700.0 -0.91 -1.4548 -0.9937 3068652 PK04_093292 COCCCNC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O19 compound treatment 1121920.0 -73900.0 -1.24 1156760.0 -41900.0 -0.76 -1.4086 -0.9721 3186309 PK04_093293 COC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O20 compound treatment 1149040.0 -46800.0 -0.78 1147320.0 -51400.0 -0.93 -1.2079 -0.9965 3068654 PK04_093294 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O21 compound treatment 977400.0 -218000.0 -3.65 1008400.0 -190000.0 -3.43 -5.0088 -0.9995 3186310 PK04_093295 COC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O22 compound treatment 1129680.0 -66100.0 -1.11 1129800.0 -68900.0 -1.24 -1.6602 -0.9984 3186311 PK04_093296 NC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O23 compound treatment 396320.0 -799000.0 -13.38 532520.0 -666000.0 -12.0 -17.9475 -0.9985 3068656 PK04_093297 COC(=O)[C@@H]1N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 O24 compound treatment 1143720.0 -52100.0 -0.87 1135920.0 -62800.0 -1.13 -1.4161 -0.9917 3186312 PK04_093298 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P01 compound treatment 1048920.0 -147000.0 -2.46 1043640.0 -155000.0 -2.79 -3.7135 -0.998 3186313 PK04_093299 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(CCS(=O)(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P02 compound treatment 1021240.0 -175000.0 -2.92 1018280.0 -180000.0 -3.25 -4.3642 -0.9986 3186314 PK04_093300 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P03 compound treatment 1090280.0 -106000.0 -1.77 1100480.0 -98200.0 -1.77 -2.5 -1.0 3067960 PK04_093301 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P04 compound treatment 1005760.0 -190000.0 -3.18 1065840.0 -133000.0 -2.39 -3.9414 -0.9902 3186315 PK04_093302 CN(C)C(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P05 compound treatment 820680.0 -375000.0 -6.28 836360.0 -362000.0 -6.53 -9.0551 -0.9998 3186316 PK04_093303 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P06 compound treatment 970880.0 -225000.0 -3.76 987040.0 -212000.0 -3.81 -5.3581 -1.0 3067963 PK04_093304 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P07 compound treatment 1045040.0 -151000.0 -2.52 1062120.0 -137000.0 -2.46 -3.524 -0.9999 3186317 PK04_093305 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P08 compound treatment 1160960.0 -34800.0 -0.58 1157880.0 -40800.0 -0.74 -0.9323 -0.9934 3186362 PK04_093306 COCCCNC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P09 compound treatment 1154760.0 -41000.0 -0.69 1158000.0 -40700.0 -0.73 -1.0042 -0.9995 3067965 PK04_093307 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(CCS(=O)(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P10 compound treatment 1168600.0 -27200.0 -0.46 1177720.0 -21000.0 -0.38 -0.5892 -0.9957 3186363 PK04_093308 COCCCNC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P11 mock treatment 1180520.0 -15300.0 -0.26 1179640.0 -19100.0 -0.34 -0.4236 -0.9894 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P12 mock treatment 1189000.0 -6800.0 -0.11 1196400.0 -2300.0 -0.04 -0.1098 -0.9066 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P13 compound treatment 714560.0 -481000.0 -8.05 743320.0 -455000.0 -8.2 -11.4961 -1.0 3186364 PK04_093309 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5N(CCS(=O)(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P14 compound treatment 1084840.0 -111000.0 -1.86 1077720.0 -121000.0 -2.18 -2.8543 -0.9968 3067968 PK04_093310 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P15 compound treatment 1093800.0 -102000.0 -1.71 1118720.0 -80000.0 -1.44 -2.2259 -0.9965 3186365 PK04_093311 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5N(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P16 compound treatment 1116200.0 -79600.0 -1.33 1121160.0 -77500.0 -1.4 -1.9298 -0.9997 3186366 PK04_093312 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P17 compound treatment 1097120.0 -98700.0 -1.65 1102120.0 -96600.0 -1.74 -2.3981 -0.9997 3067970 PK04_093313 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(CC=C)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P18 compound treatment 1134760.0 -61000.0 -1.02 1142400.0 -56300.0 -1.01 -1.4396 -1.0 3186367 PK04_093314 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P19 compound treatment 1120760.0 -75000.0 -1.26 1121600.0 -77100.0 -1.39 -1.8702 -0.9987 3067972 PK04_093315 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(CC=C)C3=O)[C@H](O2)c5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P20 compound treatment 1038960.0 -157000.0 -2.62 1065120.0 -134000.0 -2.41 -3.5577 -0.9991 3186368 PK04_093316 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P21 compound treatment 1103960.0 -91800.0 -1.54 1101560.0 -97100.0 -1.75 -2.3243 -0.9979 3067974 PK04_093317 CC(=O)N1Cc2ccccc2C[C@@]3(N=C(O[C@H]3c4ccccc4)c5ccc(OCCCO)cc5)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P22 compound treatment 1098680.0 -97100.0 -1.63 1126960.0 -71700.0 -1.29 -2.0632 -0.9936 3186369 PK04_093318 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P23 compound treatment 1098080.0 -97700.0 -1.64 1117360.0 -81300.0 -1.47 -2.1926 -0.9985 3067976 PK04_093319 CC(=O)N1Cc2ccccc2C[C@@]3(COC(=N3)c4ccc(OCCCO)cc4)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2093 P24 compound treatment 1125360.0 -70400.0 -1.18 1143200.0 -55500.0 -1.0 -1.5406 -0.9967 3186370 PK04_093320 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A01 compound treatment 1183680.0 4560.0 0.08 1191520.0 11700.0 0.21 0.2032 0.9052 3186371 PK04_094001 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A02 compound treatment 1030440.0 -149000.0 -2.49 951080.0 -229000.0 -4.12 -4.6734 -0.9708 3067979 PK04_094002 COCCCNC(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A03 compound treatment 887560.0 -292000.0 -4.88 865320.0 -314000.0 -5.67 -7.4567 -0.9972 3068002 PK04_094003 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A04 compound treatment 833480.0 -346000.0 -5.78 849240.0 -331000.0 -5.96 -8.3015 -0.9999 3186372 PK04_094004 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A05 compound treatment 1182320.0 3200.0 0.05 1189040.0 9240.0 0.17 0.1555 0.8895 3068007 PK04_094005 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A06 compound treatment 1207240.0 28100.0 0.47 1199360.0 19600.0 0.35 0.5818 0.9899 3186373 PK04_094006 CN(C)C(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A07 compound treatment 1178200.0 -925.0 -0.02 1180080.0 277.0 0.0 -0.0074 -0.4562 3186374 PK04_094007 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A08 compound treatment 980480.0 -199000.0 -3.32 990720.0 -189000.0 -3.41 -4.7595 -0.9999 3068010 PK04_094008 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A09 compound treatment 1137440.0 -41700.0 -0.7 1149960.0 -29800.0 -0.54 -0.8735 -0.9917 3186375 PK04_094009 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A10 compound treatment 942640.0 -236000.0 -3.96 935520.0 -244000.0 -4.4 -5.9105 -0.9986 3068013 PK04_094010 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A11 compound treatment 1077480.0 -102000.0 -1.7 1072920.0 -107000.0 -1.93 -2.5645 -0.9981 3186376 PK04_094011 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A12 compound treatment 1176320.0 -2810.0 -0.05 1170720.0 -9080.0 -0.16 -0.1489 -0.8747 3186377 PK04_094012 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A13 mock treatment 1206840.0 27700.0 0.46 1201240.0 21400.0 0.39 0.6011 0.9959 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A14 mock treatment 1185360.0 6240.0 0.1 1186280.0 6480.0 0.12 0.1563 0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A15 compound treatment 1159600.0 -19500.0 -0.33 1154440.0 -25400.0 -0.46 -0.5542 -0.9865 3068016 PK04_094013 CN(C)C(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A16 compound treatment 958000.0 -221000.0 -3.7 928840.0 -251000.0 -4.52 -5.8139 -0.995 3186378 PK04_094014 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A17 compound treatment 819040.0 -360000.0 -6.03 822720.0 -357000.0 -6.43 -8.8102 -0.9995 3068018 PK04_094015 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A18 compound treatment 1175160.0 -3970.0 -0.07 1162720.0 -17100.0 -0.31 -0.2646 -0.8402 3186379 PK04_094016 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A19 compound treatment 1156960.0 -22200.0 -0.37 1163560.0 -16200.0 -0.29 -0.4692 -0.9931 3186380 PK04_094017 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A20 compound treatment 1016360.0 -163000.0 -2.72 1001040.0 -179000.0 -3.22 -4.2035 -0.9965 3068020 PK04_094018 NC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A21 compound treatment 1177240.0 -1890.0 -0.03 1159920.0 -19900.0 -0.36 -0.2756 -0.7664 3186381 PK04_094019 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A22 compound treatment 1150840.0 -28300.0 -0.47 1127320.0 -52500.0 -0.95 -1.0033 -0.9488 3186437 PK04_094020 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A23 compound treatment 1132800.0 -46300.0 -0.78 1125440.0 -54400.0 -0.98 -1.2408 -0.9933 3068021 PK04_094021 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 A24 compound treatment 1147600.0 -31500.0 -0.53 1139360.0 -40400.0 -0.73 -0.8883 -0.9874 3186438 PK04_094022 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B01 compound treatment 1200320.0 21200.0 0.35 1202520.0 22700.0 0.41 0.5402 0.9975 3186439 PK04_094023 CCCN1C(=O)[C@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B02 compound treatment 1227280.0 48200.0 0.81 1225400.0 45600.0 0.82 1.1507 1.0 3089331 PK04_094024 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B03 compound treatment 1166320.0 -12800.0 -0.21 1181240.0 1440.0 0.03 -0.1332 -0.6172 3068022 PK04_094025 CCCN1C(=O)[C@]2(Cc3ccccc13)N=C(O[C@@H]2c4ccccc4)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B04 compound treatment 1217040.0 37900.0 0.63 1211000.0 31200.0 0.56 0.8461 0.9982 3089332 PK04_094026 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B05 compound treatment 1132520.0 -46600.0 -0.78 1154880.0 -24900.0 -0.45 -0.869 -0.9656 3186440 PK04_094027 CCCN1C(=O)[C@@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B06 compound treatment 1167600.0 -11500.0 -0.19 1200240.0 20400.0 0.37 0.124 0.2983 3000708 PK04_094028 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B07 compound treatment 1024280.0 -155000.0 -2.59 1004680.0 -175000.0 -3.16 -4.0634 -0.9952 3068023 PK04_094029 CN1C(=O)[C@]2(Cc3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B08 compound treatment 1183960.0 4840.0 0.08 1179640.0 -163.0 0.0 0.0551 0.681 3089333 PK04_094030 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B09 compound treatment 860200.0 -319000.0 -5.34 873200.0 -307000.0 -5.52 -7.68 -0.9999 3186441 PK04_094031 CN1C(=O)[C@@]2(CC=C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B10 compound treatment 1164920.0 -14200.0 -0.24 1173480.0 -6320.0 -0.11 -0.2486 -0.9433 3089654 PK04_094032 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B11 compound treatment 1051240.0 -128000.0 -2.14 1065000.0 -115000.0 -2.07 -2.9759 -0.9999 3186442 PK04_094033 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B12 compound treatment 1152920.0 -26200.0 -0.44 1158680.0 -21100.0 -0.38 -0.5792 -0.9975 3089334 PK04_094034 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B13 mock treatment 1201200.0 22100.0 0.37 1168880.0 -10900.0 -0.2 0.1221 0.2916 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B14 mock treatment 1191400.0 12300.0 0.21 1184560.0 4760.0 0.09 0.2059 0.9249 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B15 compound treatment 1170760.0 -8370.0 -0.14 1171720.0 -8080.0 -0.15 -0.202 -0.9998 3068024 PK04_094035 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B16 compound treatment 1168920.0 -10200.0 -0.17 1164080.0 -15700.0 -0.28 -0.3211 -0.9706 3000709 PK04_094036 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3)[C@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B17 compound treatment 1156600.0 -22500.0 -0.38 1141520.0 -38300.0 -0.69 -0.7543 -0.9596 3186443 PK04_094037 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B18 compound treatment 1156520.0 -22600.0 -0.38 1157920.0 -21900.0 -0.39 -0.5463 -0.9998 3089363 PK04_094038 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4)[C@H]1OC(=O)Nc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B19 compound treatment 1037600.0 -142000.0 -2.37 1008000.0 -172000.0 -3.1 -3.8635 -0.9913 3068025 PK04_094039 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5N(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B20 compound treatment 1153800.0 -25300.0 -0.42 1136720.0 -43100.0 -0.78 -0.8486 -0.9595 3089652 PK04_094040 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4)[C@H]1OC(=O)Nc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B21 compound treatment 1133560.0 -45600.0 -0.76 1108320.0 -71500.0 -1.29 -1.4499 -0.9687 3186444 PK04_094041 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B22 compound treatment 1147880.0 -31200.0 -0.52 1136360.0 -43400.0 -0.78 -0.9232 -0.9808 3089653 PK04_094042 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4)[C@H]1OC(=O)Nc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B23 compound treatment 1117240.0 -61900.0 -1.04 1096920.0 -82900.0 -1.49 -1.7882 -0.984 3186445 PK04_094043 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 B24 compound treatment 1115200.0 -63900.0 -1.07 1111400.0 -68400.0 -1.23 -1.6279 -0.9975 3089657 PK04_094044 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C01 compound treatment 1212360.0 33200.0 0.56 1198200.0 18400.0 0.33 0.6277 0.9694 3068026 PK04_094045 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C02 compound treatment 1181280.0 2160.0 0.04 1153720.0 -26100.0 -0.47 -0.3068 -0.6509 3068051 PK04_094046 CN(C)C(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C03 compound treatment 1193880.0 14800.0 0.25 1195520.0 15700.0 0.28 0.3748 0.9977 3068052 PK04_094047 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C04 compound treatment 1201040.0 21900.0 0.37 1203840.0 24000.0 0.43 0.5656 0.9966 3068053 PK04_094048 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)N3CCOCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C05 compound treatment 1127840.0 -51300.0 -0.86 1151320.0 -28500.0 -0.51 -0.9697 -0.9698 3068054 PK04_094049 COCCCNC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C06 compound treatment 1184000.0 4880.0 0.08 1188800.0 9000.0 0.16 0.1723 0.9495 3186446 PK04_094050 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C07 compound treatment 1125640.0 -53500.0 -0.9 1139600.0 -40200.0 -0.72 -1.1451 -0.9945 3068055 PK04_094051 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C08 compound treatment 1135200.0 -43900.0 -0.74 1133800.0 -46000.0 -0.83 -1.1059 -0.9982 3186447 PK04_094052 COCCCNC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C09 compound treatment 1163280.0 -15800.0 -0.27 1165080.0 -14700.0 -0.27 -0.3751 -1.0 3068056 PK04_094053 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C10 compound treatment 1115480.0 -63600.0 -1.07 1104720.0 -75100.0 -1.35 -1.7097 -0.993 3186448 PK04_094054 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C11 mock treatment 1178920.0 -205.0 0.0 1192960.0 13200.0 0.24 0.1652 0.6968 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C12 mock treatment 1182760.0 3640.0 0.06 1194120.0 14300.0 0.26 0.2254 0.8505 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C13 compound treatment 1163240.0 -15900.0 -0.27 1144520.0 -35300.0 -0.64 -0.6375 -0.9252 3186449 PK04_094055 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C14 compound treatment 1172040.0 -7090.0 -0.12 1167720.0 -12100.0 -0.22 -0.2378 -0.9592 3068057 PK04_094056 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C15 mock treatment 1179040.0 -85.0 0.0 1177200.0 -2600.0 -0.05 -0.0342 -0.7282 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C16 mock treatment 1180520.0 1400.0 0.02 1167280.0 -12500.0 -0.23 -0.143 -0.6306 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C17 compound treatment 1175680.0 -3450.0 -0.06 1183320.0 3520.0 0.06 0.004 0.0471 3186450 PK04_094057 NC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C18 compound treatment 1166800.0 -12300.0 -0.21 1162080.0 -17700.0 -0.32 -0.3716 -0.9776 3186451 PK04_094058 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C19 compound treatment 1110360.0 -68800.0 -1.15 1103920.0 -75900.0 -1.37 -1.7805 -0.9963 3068058 PK04_094059 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C20 compound treatment 1122560.0 -56600.0 -0.95 1122880.0 -56900.0 -1.03 -1.3945 -0.9992 3186452 PK04_094060 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C21 compound treatment 1022920.0 -156000.0 -2.61 868400.0 -311000.0 -5.61 -5.8157 -0.9396 3068059 PK04_094061 NC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C22 compound treatment 970640.0 -208000.0 -3.49 855040.0 -325000.0 -5.85 -6.6045 -0.9695 3186453 PK04_094062 NC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C23 compound treatment 1168280.0 -10800.0 -0.18 1156280.0 -23500.0 -0.42 -0.428 -0.9284 3186454 PK04_094063 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 C24 compound treatment 1165320.0 -13800.0 -0.23 1134840.0 -45000.0 -0.81 -0.7362 -0.8739 3068060 PK04_094064 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D01 compound treatment 1074080.0 -105000.0 -1.76 1071920.0 -108000.0 -1.94 -2.6175 -0.9987 3186455 PK04_094065 CN1C(=O)[C@@]2(CCC(=O)OC(C)(C)C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D02 compound treatment 887920.0 -291000.0 -4.87 874200.0 -306000.0 -5.51 -7.3393 -0.9981 3000713 PK04_094066 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D03 compound treatment 1078160.0 -101000.0 -1.69 1081040.0 -98800.0 -1.78 -2.453 -0.9997 3186456 PK04_094067 CCCN1C(=O)[C@@]2(CCC(=O)OC(C)(C)C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D04 compound treatment 966760.0 -212000.0 -3.55 965600.0 -214000.0 -3.86 -5.2419 -0.9992 3089658 PK04_094068 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D05 compound treatment 1002640.0 -176000.0 -2.95 1025880.0 -154000.0 -2.77 -4.0494 -0.9995 3068061 PK04_094069 CCCN1C(=O)[C@@]2(Cc3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D06 compound treatment 997080.0 -182000.0 -3.05 1013480.0 -166000.0 -3.0 -4.2731 -1.0 3089659 PK04_094070 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D07 compound treatment 1103280.0 -75800.0 -1.27 1128440.0 -51400.0 -0.93 -1.5519 -0.988 3186457 PK04_094071 CCCN1C(=O)[C@]2(CCC(=O)OC(C)(C)C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D08 compound treatment 862680.0 -316000.0 -5.3 858960.0 -321000.0 -5.78 -7.8321 -0.999 3089664 PK04_094072 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D09 compound treatment 1038800.0 -140000.0 -2.35 1022480.0 -157000.0 -2.83 -3.6648 -0.9956 3068062 PK04_094073 CCCN1C(=O)[C@@]2(CC=C)N=C(O[C@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D10 compound treatment 867120.0 -312000.0 -5.22 863560.0 -316000.0 -5.7 -7.721 -0.999 3000714 PK04_094074 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D11 mock treatment 1195120.0 16000.0 0.27 1180560.0 757.0 0.01 0.1989 0.7422 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D12 mock treatment 1194040.0 14900.0 0.25 1185000.0 5200.0 0.09 0.2427 0.9104 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D13 compound treatment 1144840.0 -34300.0 -0.57 1135040.0 -44800.0 -0.81 -0.976 -0.9861 3186504 PK04_094075 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4)[C@@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D14 compound treatment 972920.0 -206000.0 -3.45 964800.0 -215000.0 -3.87 -5.1792 -0.9983 3089660 PK04_094076 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D15 mock treatment 1168480.0 -10600.0 -0.18 1161360.0 -18400.0 -0.33 -0.3609 -0.9573 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D16 mock treatment 1165160.0 -14000.0 -0.23 1169120.0 -10700.0 -0.19 -0.3014 -0.9954 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D17 compound treatment 1095680.0 -83400.0 -1.4 1100120.0 -79700.0 -1.44 -2.0026 -0.9999 3186505 PK04_094077 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(Cc5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D18 compound treatment 940680.0 -238000.0 -3.99 975040.0 -205000.0 -3.69 -5.4302 -0.9992 3000715 PK04_094078 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@H]1OC(=O)Nc6ccc7OCOc7c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D19 compound treatment 1111360.0 -67800.0 -1.13 1092280.0 -87500.0 -1.58 -1.9169 -0.9869 3068063 PK04_094079 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D20 compound treatment 962640.0 -216000.0 -3.62 898480.0 -281000.0 -5.07 -6.1458 -0.9864 3089662 PK04_094080 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@H]1OC(=O)Nc6ccc7OCOc7c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D21 compound treatment 1097960.0 -81200.0 -1.36 1051000.0 -129000.0 -2.32 -2.6014 -0.9674 3186506 PK04_094081 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4N(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D22 compound treatment 913000.0 -266000.0 -4.45 889720.0 -290000.0 -5.23 -6.8448 -0.9968 3000716 PK04_094082 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@H]1OC(=O)Nc6ccc7OCOc7c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D23 compound treatment 1100440.0 -78700.0 -1.32 1084760.0 -95000.0 -1.71 -2.1419 -0.9916 3068064 PK04_094083 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3N(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 D24 compound treatment 1143480.0 -35600.0 -0.6 1145120.0 -34700.0 -0.62 -0.8637 -0.9997 3000811 PK04_094084 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E01 mock treatment 1228960.0 49800.0 0.83 1218280.0 38500.0 0.69 1.0799 0.9958 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E02 mock treatment 1224680.0 45600.0 0.76 1210560.0 30800.0 0.55 0.9309 0.9877 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E03 compound treatment 880400.0 -299000.0 -5.0 842080.0 -338000.0 -6.08 -7.8375 -0.9952 3186507 PK04_094085 CN(C)C(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E04 compound treatment 1183760.0 4640.0 0.08 1182880.0 3080.0 0.06 0.094 0.9864 3186508 PK04_094086 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E05 compound treatment 1192040.0 12900.0 0.22 1202160.0 22400.0 0.4 0.4377 0.9574 3068065 PK04_094087 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E06 compound treatment 756880.0 -422000.0 -7.07 766320.0 -413000.0 -7.45 -10.2643 -0.9997 3186509 PK04_094088 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E07 compound treatment 1156400.0 -22700.0 -0.38 1165880.0 -13900.0 -0.25 -0.4463 -0.9796 3068066 PK04_094089 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E08 compound treatment 939960.0 -239000.0 -4.0 936080.0 -244000.0 -4.39 -5.9351 -0.9989 3186510 PK04_094090 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3N=[N+]=[N-])C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E09 mock treatment 1197040.0 17900.0 0.3 1185040.0 5240.0 0.09 0.2787 0.8868 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E10 mock treatment 1198760.0 19600.0 0.33 1199880.0 20100.0 0.36 0.4881 0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E11 compound treatment 1138400.0 -40700.0 -0.68 1125520.0 -54300.0 -0.98 -1.1735 -0.9844 3186511 PK04_094091 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E12 compound treatment 1180280.0 1160.0 0.02 1180360.0 557.0 0.01 0.0208 0.9533 3068067 PK04_094092 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E13 compound treatment 1097040.0 -82100.0 -1.37 1116320.0 -63500.0 -1.14 -1.7801 -0.9959 3186512 PK04_094093 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E14 compound treatment 1121520.0 -57600.0 -0.96 1113120.0 -66700.0 -1.2 -1.5312 -0.994 3068068 PK04_094094 NC(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E15 compound treatment 1168880.0 -10200.0 -0.17 1155600.0 -24200.0 -0.44 -0.4296 -0.9168 3186513 PK04_094095 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E16 compound treatment 895960.0 -283000.0 -4.74 883680.0 -296000.0 -5.34 -7.1234 -0.9983 3068069 PK04_094096 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E17 mock treatment 1170960.0 -8170.0 -0.14 1166400.0 -13400.0 -0.24 -0.2674 -0.9636 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E18 mock treatment 1181280.0 2160.0 0.04 1181640.0 1840.0 0.03 0.0489 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E19 compound treatment 1026080.0 -153000.0 -2.56 1004640.0 -175000.0 -3.16 -4.0426 -0.9946 3186514 PK04_094097 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E20 compound treatment 1153120.0 -26000.0 -0.44 1141600.0 -38200.0 -0.69 -0.7944 -0.9755 3186515 PK04_094098 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E21 compound treatment 1104680.0 -74400.0 -1.25 1072360.0 -107000.0 -1.94 -2.2498 -0.9773 3068070 PK04_094099 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E22 compound treatment 956200.0 -223000.0 -3.73 877320.0 -302000.0 -5.45 -6.4916 -0.9829 3186516 PK04_094100 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E23 compound treatment 1143360.0 -35800.0 -0.6 1144640.0 -35200.0 -0.63 -0.8712 -0.9996 3068071 PK04_094101 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 E24 compound treatment 1012080.0 -167000.0 -2.8 994040.0 -186000.0 -3.35 -4.3433 -0.996 3186517 PK04_094102 COCCCNC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F01 mock treatment 1224760.0 45600.0 0.76 1222680.0 42900.0 0.77 1.0863 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F02 mock treatment 1225760.0 46600.0 0.78 1226800.0 47000.0 0.85 1.1506 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F03 compound treatment 1069840.0 -109000.0 -1.83 1061960.0 -118000.0 -2.12 -2.7945 -0.9972 3068072 PK04_094103 CN1C(=O)[C@]2(CCC(=O)OC(C)(C)C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F04 compound treatment 1208240.0 29100.0 0.49 1194520.0 14700.0 0.27 0.532 0.9591 3000813 PK04_094104 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]2OC(=O)Nc5ccccc5c6ccccc6)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F05 compound treatment 1015760.0 -163000.0 -2.73 1002640.0 -177000.0 -3.19 -4.1902 -0.997 3186518 PK04_094105 CN1C(=O)[C@]2(CC=C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F06 compound treatment 1195320.0 16200.0 0.27 1194000.0 14200.0 0.26 0.3725 0.9996 3000814 PK04_094106 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F07 compound treatment 1211000.0 31900.0 0.53 1208640.0 28800.0 0.52 0.7446 0.9999 3186519 PK04_094107 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4CN(C(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F08 compound treatment 1155880.0 -23200.0 -0.39 1157320.0 -22500.0 -0.41 -0.5615 -0.9998 3089667 PK04_094108 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F09 mock treatment 1186920.0 7800.0 0.13 1184720.0 4920.0 0.09 0.1549 0.9822 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F10 mock treatment 1196200.0 17100.0 0.29 1194000.0 14200.0 0.26 0.3829 0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F11 compound treatment 1165080.0 -14000.0 -0.24 1155640.0 -24200.0 -0.44 -0.474 -0.9581 3068073 PK04_094109 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(C(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F12 compound treatment 1169000.0 -10100.0 -0.17 1155680.0 -24100.0 -0.43 -0.4271 -0.9156 3089654 PK04_094110 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F13 compound treatment 1140480.0 -38600.0 -0.65 1125360.0 -54400.0 -0.98 -1.1509 -0.9796 3186520 PK04_094111 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(C(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F14 compound treatment 1163080.0 -16000.0 -0.27 1141320.0 -38500.0 -0.69 -0.6801 -0.9147 3089708 PK04_094112 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F15 compound treatment 1125600.0 -53500.0 -0.9 1125360.0 -54400.0 -0.98 -1.327 -0.999 3186521 PK04_094113 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4N(C(=O)c5ccccc5)C3=O)[C@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F16 compound treatment 1155160.0 -24000.0 -0.4 1143800.0 -36000.0 -0.65 -0.7423 -0.9733 3000817 PK04_094114 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F17 mock treatment 1149400.0 -29700.0 -0.5 1149800.0 -30000.0 -0.54 -0.734 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F18 mock treatment 1148280.0 -30800.0 -0.52 1148400.0 -31400.0 -0.57 -0.7651 -0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F19 compound treatment 1124680.0 -54400.0 -0.91 1118120.0 -61700.0 -1.11 -1.4301 -0.9951 3068074 PK04_094115 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(Cc6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F20 compound treatment 1132800.0 -46300.0 -0.78 1126960.0 -52800.0 -0.95 -1.2214 -0.9948 3089709 PK04_094116 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F21 compound treatment 1133600.0 -45500.0 -0.76 1123080.0 -56700.0 -1.02 -1.2614 -0.9895 3186522 PK04_094117 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F22 compound treatment 1125720.0 -53400.0 -0.89 1123560.0 -56200.0 -1.01 -1.3485 -0.998 3000821 PK04_094118 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F23 compound treatment 1113160.0 -66000.0 -1.1 1115880.0 -63900.0 -1.15 -1.595 -0.9998 3186523 PK04_094119 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 F24 compound treatment 1138520.0 -40600.0 -0.68 1137680.0 -42100.0 -0.76 -1.0171 -0.9985 3089711 PK04_094120 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@H]1OC(=O)Nc6ccccc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G01 compound treatment 937440.0 -242000.0 -4.04 936360.0 -243000.0 -4.39 -5.9614 -0.9992 3068075 PK04_094121 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G02 compound treatment 1211120.0 32000.0 0.54 1208920.0 29100.0 0.52 0.7496 0.9999 3186524 PK04_094122 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G03 mock treatment 1217640.0 38500.0 0.64 1207360.0 27600.0 0.5 0.8068 0.9917 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G04 mock treatment 1213880.0 34800.0 0.58 1216560.0 36800.0 0.66 0.8795 0.9979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G05 compound treatment 933640.0 -245000.0 -4.11 863560.0 -316000.0 -5.7 -6.9338 -0.9871 3186575 PK04_094123 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G06 compound treatment 1158960.0 -20200.0 -0.34 1144880.0 -34900.0 -0.63 -0.6835 -0.9573 3186576 PK04_094124 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G07 compound treatment 1223480.0 44400.0 0.74 1236640.0 56800.0 1.02 1.249 0.9875 3068110 PK04_094125 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G08 compound treatment 1187840.0 8720.0 0.15 1182840.0 3040.0 0.05 0.1418 0.9104 3186577 PK04_094126 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G09 compound treatment 1181320.0 2200.0 0.04 1169360.0 -10400.0 -0.19 -0.1071 -0.5585 3068111 PK04_094127 COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G10 compound treatment 1187760.0 8640.0 0.14 1188520.0 8720.0 0.16 0.2132 0.9991 3186578 PK04_094128 CN(C)C(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G11 compound treatment 1166200.0 -12900.0 -0.22 1150320.0 -29500.0 -0.53 -0.5286 -0.9216 3186579 PK04_094129 COCCCNC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G12 compound treatment 1183720.0 4600.0 0.08 1178160.0 -1640.0 -0.03 0.0334 0.4058 3068112 PK04_094130 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G13 compound treatment 1169760.0 -9370.0 -0.16 1125440.0 -54400.0 -0.98 -0.8034 -0.8099 3186580 PK04_094131 OCCCOc1ccc(cc1)C2=N[C@](CC=C)(CO2)C(=O)NCCN3CCOCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G14 compound treatment 915760.0 -263000.0 -4.41 826920.0 -353000.0 -6.36 -7.6122 -0.984 3186581 PK04_094132 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G15 compound treatment 796600.0 -383000.0 -6.4 759520.0 -420000.0 -7.57 -9.8809 -0.9965 3068113 PK04_094133 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G16 compound treatment 1165880.0 -13200.0 -0.22 1163840.0 -16000.0 -0.29 -0.3601 -0.9917 3186582 PK04_094134 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G17 compound treatment 1201640.0 22500.0 0.38 1206080.0 26300.0 0.47 0.6012 0.9936 3186583 PK04_094135 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G18 compound treatment 983800.0 -195000.0 -3.27 932840.0 -247000.0 -4.45 -5.4576 -0.9885 3068114 PK04_094136 NC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G19 mock treatment 1163320.0 -15800.0 -0.26 1153520.0 -26300.0 -0.47 -0.5219 -0.9621 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G20 mock treatment 1162320.0 -16800.0 -0.28 1170640.0 -9160.0 -0.17 -0.3156 -0.9678 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G21 compound treatment 1139440.0 -39700.0 -0.66 1159560.0 -20200.0 -0.36 -0.7275 -0.9602 3186584 PK04_094137 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G22 compound treatment 923520.0 -256000.0 -4.28 832680.0 -347000.0 -6.25 -7.447 -0.9828 3068115 PK04_094138 COCCCNC(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G23 compound treatment 1141040.0 -38100.0 -0.64 1126880.0 -52900.0 -0.95 -1.1249 -0.9808 3186585 PK04_094139 CN(C)C(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 G24 compound treatment 1160360.0 -18800.0 -0.31 1141200.0 -38600.0 -0.7 -0.7139 -0.9354 3186586 PK04_094140 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)NCc3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H01 compound treatment 1016200.0 -163000.0 -2.73 1008040.0 -172000.0 -3.09 -4.1162 -0.998 3068116 PK04_094141 CCCN1C(=O)[C@]2(Cc3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H02 compound treatment 1213120.0 34000.0 0.57 1204200.0 24400.0 0.44 0.7131 0.9919 3000914 PK04_094142 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H03 mock treatment 1214800.0 35700.0 0.6 1221400.0 41600.0 0.75 0.9521 0.9937 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H04 mock treatment 1217360.0 38200.0 0.64 1217320.0 37500.0 0.68 0.9304 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H05 compound treatment 1094040.0 -85100.0 -1.42 1083640.0 -96200.0 -1.73 -2.2319 -0.9953 3068117 PK04_094143 CCCN1C(=O)[C@]2(CC=C)N=C(O[C@@H]2c3ccccc13)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H06 compound treatment 1183320.0 4200.0 0.07 1194240.0 14400.0 0.26 0.2336 0.8669 3089723 PK04_094144 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H07 compound treatment 966760.0 -212000.0 -3.55 874000.0 -306000.0 -5.51 -6.4089 -0.9775 3186589 PK04_094145 CN1C(=O)[C@@]2(Cc3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H08 compound treatment 1180720.0 1600.0 0.03 1179160.0 -643.0 -0.01 0.0107 0.367 3089724 PK04_094146 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H09 compound treatment 1134360.0 -44800.0 -0.75 1128240.0 -51600.0 -0.93 -1.1866 -0.9943 3186590 PK04_094147 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4N(C(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H10 compound treatment 1176160.0 -2970.0 -0.05 1172520.0 -7280.0 -0.13 -0.1279 -0.9115 3000917 PK04_094148 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H11 compound treatment 1154680.0 -24400.0 -0.41 1142800.0 -37000.0 -0.67 -0.7607 -0.9725 3068119 PK04_094149 CC(C)(C)OC(=O)CC[C@]12N=C(O[C@@H]2c3ccccc3CN(C(=O)c4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H12 compound treatment 1172920.0 -6210.0 -0.1 1169840.0 -9960.0 -0.18 -0.2004 -0.9661 3089768 PK04_094150 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H13 compound treatment 1135560.0 -43600.0 -0.73 1123480.0 -56300.0 -1.01 -1.2331 -0.9868 3186593 PK04_094151 OCCCOc1ccc(cc1)C2=N[C@]3(CC=C)[C@H](O2)c4ccccc4CN(C(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H14 compound treatment 1151320.0 -27800.0 -0.47 1149080.0 -30700.0 -0.55 -0.7204 -0.9963 3089763 PK04_094152 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H15 compound treatment 1135480.0 -43600.0 -0.73 1141000.0 -38800.0 -0.7 -1.0108 -0.9998 3186594 PK04_094153 OCCCOc1ccc(cc1)C2=N[C@@]3(CCS(=O)(=O)c4ccccc4)[C@@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H16 compound treatment 1140960.0 -38200.0 -0.64 1148360.0 -31400.0 -0.57 -0.8522 -0.9982 3089764 PK04_094154 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3)[C@@H]1OC(=O)Nc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H17 compound treatment 1127400.0 -51700.0 -0.87 1125200.0 -54600.0 -0.98 -1.3077 -0.998 3068121 PK04_094155 OCCCOc1ccc(cc1)C2=N[C@@]3(CO2)Cc4ccccc4CN(C(=O)c5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H18 compound treatment 1137120.0 -42000.0 -0.7 1148280.0 -31500.0 -0.57 -0.8987 -0.9944 3000919 PK04_094156 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4)[C@@H]1OC(=O)Nc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H19 mock treatment 1141880.0 -37200.0 -0.62 1141240.0 -38600.0 -0.69 -0.932 -0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H20 mock treatment 1131120.0 -48000.0 -0.8 1123360.0 -56400.0 -1.02 -1.2871 -0.9932 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H21 compound treatment 1095880.0 -83200.0 -1.39 1084560.0 -95200.0 -1.72 -2.1985 -0.9946 3068122 PK04_094157 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3N(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H22 compound treatment 1137320.0 -41800.0 -0.7 1124280.0 -55500.0 -1.0 -1.2021 -0.9847 3089766 PK04_094158 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4)[C@@H]1OC(=O)Nc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H23 compound treatment 1111120.0 -68000.0 -1.14 1111880.0 -67900.0 -1.22 -1.6701 -0.9993 3068123 PK04_094159 OCCCOc1ccc(cc1)C2=N[C@@]3(CC=C)[C@@H](O2)c4ccccc4CN(Cc5ccccc5)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 H24 compound treatment 988520.0 -191000.0 -3.19 917320.0 -262000.0 -4.73 -5.5995 -0.9816 3089769 PK04_094160 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I01 compound treatment 1209120.0 30000.0 0.5 1202560.0 22800.0 0.41 0.6449 0.995 3186651 PK04_094161 COCCCNC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I02 compound treatment 1191920.0 12800.0 0.21 1202160.0 22400.0 0.4 0.4362 0.9563 3068124 PK04_094162 COCCCNC(=O)[C@@]1(CC=C)N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I03 compound treatment 1051520.0 -128000.0 -2.14 1044640.0 -135000.0 -2.44 -3.232 -0.9979 3186652 PK04_094163 NC(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I04 compound treatment 1177160.0 -1970.0 -0.03 1196120.0 16300.0 0.29 0.1846 0.6241 3068125 PK04_094164 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I05 mock treatment 1204320.0 25200.0 0.42 1213520.0 33700.0 0.61 0.7277 0.9841 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I06 mock treatment 1209880.0 30800.0 0.51 1214600.0 34800.0 0.63 0.8072 0.9952 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I07 compound treatment 1178680.0 -445.0 -0.01 1180840.0 1040.0 0.02 0.0079 0.395 3186653 PK04_094165 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I08 compound treatment 1197640.0 18500.0 0.31 1191680.0 11900.0 0.21 0.3704 0.9837 3068126 PK04_094166 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I09 compound treatment 1179040.0 -85.0 0.0 1169920.0 -9880.0 -0.18 -0.1269 -0.7127 3186654 PK04_094167 COCCCNC(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I10 compound treatment 1173800.0 -5330.0 -0.09 1164080.0 -15700.0 -0.28 -0.2633 -0.8867 3068572 PK04_094168 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I11 compound treatment 795040.0 -384000.0 -6.43 743640.0 -436000.0 -7.86 -10.1017 -0.995 3186655 PK04_094169 COCCCNC(=O)[C@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I12 compound treatment 1086720.0 -92400.0 -1.55 1078000.0 -102000.0 -1.83 -2.3904 -0.9964 3186656 PK04_094170 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I13 compound treatment 906680.0 -272000.0 -4.56 885680.0 -294000.0 -5.3 -6.971 -0.9972 3068573 PK04_094171 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I14 compound treatment 1162760.0 -16400.0 -0.27 1153800.0 -26000.0 -0.47 -0.5249 -0.9673 3186657 PK04_094172 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I15 compound treatment 1093080.0 -86000.0 -1.44 1095920.0 -83900.0 -1.51 -2.0869 -0.9997 3068574 PK04_094173 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I16 compound treatment 1135160.0 -44000.0 -0.74 1140320.0 -39500.0 -0.71 -1.0233 -0.9999 3186658 PK04_094174 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I17 compound treatment 936400.0 -243000.0 -4.06 856960.0 -323000.0 -5.82 -6.9852 -0.9846 3186659 PK04_094175 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I18 compound treatment 944640.0 -234000.0 -3.92 928000.0 -252000.0 -4.54 -5.9827 -0.9974 3068575 PK04_094176 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I19 compound treatment 1123800.0 -55300.0 -0.93 1120440.0 -59400.0 -1.07 -1.411 -0.9974 3186660 PK04_094177 CN(C)C(=O)[C@]1(CCC(=O)OC(C)(C)C)N=C(O[C@@H]1c2ccccc2)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I20 compound treatment 969800.0 -209000.0 -3.5 897560.0 -282000.0 -5.09 -6.0728 -0.9834 3068577 PK04_094178 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I21 mock treatment 1146640.0 -32500.0 -0.54 1144400.0 -35400.0 -0.64 -0.8354 -0.9968 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I22 mock treatment 1160120.0 -19000.0 -0.32 1152240.0 -27600.0 -0.5 -0.576 -0.9768 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I23 compound treatment 1133640.0 -45500.0 -0.76 1114640.0 -65200.0 -1.17 -1.3684 -0.978 3186661 PK04_094179 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 I24 compound treatment 1128720.0 -50400.0 -0.84 1136040.0 -43800.0 -0.79 -1.154 -0.9994 3186662 PK04_094180 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J01 compound treatment 1139840.0 -39300.0 -0.66 1145720.0 -34100.0 -0.61 -0.8991 -0.9994 3068611 PK04_094181 CN1C(=O)[C@@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J02 compound treatment 763080.0 -416000.0 -6.96 740960.0 -439000.0 -7.91 -10.514 -0.998 3089770 PK04_094182 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J03 compound treatment 1162080.0 -17000.0 -0.29 1168920.0 -10900.0 -0.2 -0.3403 -0.9833 3068612 PK04_094183 OCCCOc1ccc(cc1)C2=N[C@]3(CCS(=O)(=O)c4ccccc4)[C@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J04 compound treatment 1016960.0 -162000.0 -2.71 980560.0 -199000.0 -3.59 -4.4573 -0.9905 3001007 PK04_094184 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J05 mock treatment 1169920.0 -9210.0 -0.15 1164280.0 -15500.0 -0.28 -0.3067 -0.9605 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J06 mock treatment 1197080.0 18000.0 0.3 1207200.0 27400.0 0.49 0.5615 0.9717 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J07 compound treatment 1176000.0 -3130.0 -0.05 1139320.0 -40500.0 -0.73 -0.5527 -0.7559 3186665 PK04_094185 CC(C)(C)OC(=O)CC[C@@]12N=C(O[C@H]2c3ccccc3CN(Cc4ccccc4)C1=O)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J08 compound treatment 953880.0 -225000.0 -3.77 877200.0 -303000.0 -5.45 -6.5205 -0.9838 3089771 PK04_094186 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J09 compound treatment 1143120.0 -36000.0 -0.6 1123480.0 -56300.0 -1.01 -1.1436 -0.969 3186666 PK04_094187 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4N(C(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J10 compound treatment 861880.0 -317000.0 -5.31 765440.0 -414000.0 -7.47 -9.033 -0.986 3089776 PK04_094188 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccc4OCOc4c3)[C@H]2OC(=O)Nc5ccc6OCOc6c5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J11 compound treatment 1126600.0 -52500.0 -0.88 1098440.0 -81400.0 -1.47 -1.6581 -0.9701 3068615 PK04_094189 CCCN1C(=O)[C@]2(COC(=N2)c3ccc(OCCCO)cc3)Cc4ccccc14 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J12 compound treatment 500120.0 -679000.0 -11.36 449560.0 -730000.0 -13.16 -17.3381 -0.9973 3001011 PK04_094190 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J13 compound treatment 1126480.0 -52600.0 -0.88 1130040.0 -49800.0 -0.9 -1.2569 -1.0 3068616 PK04_094191 OCCCOc1ccc(cc1)C2=N[C@]3(Cc4ccccc4)[C@H](O2)c5ccccc5CN(C(=O)c6ccccc6)C3=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J14 compound treatment 906640.0 -272000.0 -4.56 894280.0 -286000.0 -5.14 -6.8619 -0.9982 3089772 PK04_094192 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccc4OCOc4c3)[C@@H]1OC(=O)Nc5ccc6OCOc6c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J15 compound treatment 1136240.0 -42900.0 -0.72 1118080.0 -61700.0 -1.11 -1.2938 -0.9775 3068617 PK04_094193 OCCCOc1ccc(cc1)C2=N[C@@]3(Cc4ccccc4CN(C(=O)c5ccccc5)C3=O)[C@@H](O2)c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J16 compound treatment 807200.0 -372000.0 -6.22 765920.0 -414000.0 -7.46 -9.6739 -0.996 3089773 PK04_094194 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@@H]1OC(=O)Nc6ccc7OCOc7c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J17 compound treatment 1120320.0 -58800.0 -0.98 1096520.0 -83300.0 -1.5 -1.7569 -0.9791 3186732 PK04_094195 CN1C(=O)[C@]2(CCS(=O)(=O)c3ccccc3)N=C(O[C@@H]2c4ccccc14)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J18 compound treatment 881600.0 -298000.0 -4.98 834080.0 -346000.0 -6.23 -7.9252 -0.9938 3089774 PK04_094196 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@@H]1OC(=O)Nc6ccc7OCOc7c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J19 compound treatment 1072320.0 -107000.0 -1.79 1023800.0 -156000.0 -2.81 -3.2513 -0.9761 3186733 PK04_094197 CCCN1C(=O)[C@@]2(Cc3ccccc13)N=C(O[C@H]2c4ccccc4)c5ccc(OCCCO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J20 compound treatment 1015840.0 -163000.0 -2.73 926800.0 -253000.0 -4.56 -5.1554 -0.97 3089775 PK04_094198 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccc5OCOc5c4)[C@@H]1OC(=O)Nc6ccc7OCOc7c6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J21 mock treatment 1110360.0 -68800.0 -1.15 1087000.0 -92800.0 -1.67 -1.996 -0.9834 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J22 mock treatment 1148480.0 -30600.0 -0.51 1152120.0 -27700.0 -0.5 -0.7153 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J23 compound treatment 972960.0 -206000.0 -3.45 793520.0 -386000.0 -6.96 -7.3608 -0.9476 3068619 PK04_094199 COC(=O)C1ON(C(=N1)c2ccc(OCCCO)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 J24 compound treatment 1126160.0 -53000.0 -0.89 1131680.0 -48100.0 -0.87 -1.2398 -0.9999 3089828 PK04_094200 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K01 compound treatment 1206920.0 27800.0 0.47 1193600.0 13800.0 0.25 0.5047 0.9569 3068620 PK04_094201 COCCCNC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K02 compound treatment 1201720.0 22600.0 0.38 1197880.0 18100.0 0.33 0.4977 0.9972 3186736 PK04_094202 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K03 compound treatment 1198080.0 19000.0 0.32 1190560.0 10800.0 0.19 0.3613 0.9721 3186737 PK04_094203 CN(C)C(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K04 compound treatment 1152480.0 -26600.0 -0.45 1152800.0 -27000.0 -0.49 -0.6593 -0.9991 3068660 PK04_094204 CN(C)C(=O)[C@@]1(CCC(=O)OC(C)(C)C)N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K05 compound treatment 790360.0 -389000.0 -6.51 765840.0 -414000.0 -7.46 -9.8742 -0.9977 3186738 PK04_094205 OCCCOc1ccc(cc1)C2=N[C@@](CCS(=O)(=O)c3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K06 compound treatment 1207520.0 28400.0 0.48 1211080.0 31300.0 0.56 0.7345 0.9964 3068661 PK04_094206 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)(CO2)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K07 mock treatment 1211120.0 32000.0 0.54 1197600.0 17800.0 0.32 0.6053 0.9699 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K08 mock treatment 1189080.0 9960.0 0.17 1198840.0 19000.0 0.34 0.3603 0.945 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K09 compound treatment 1179360.0 235.0 0.0 1184880.0 5080.0 0.09 0.0675 0.7368 3186739 PK04_094207 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K10 compound treatment 1172160.0 -6970.0 -0.12 1174160.0 -5640.0 -0.1 -0.1543 -0.9977 3186740 PK04_094208 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K11 compound treatment 1159080.0 -20000.0 -0.34 1153680.0 -26100.0 -0.47 -0.57 -0.9862 3068664 PK04_094209 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K12 compound treatment 1153720.0 -25400.0 -0.43 1142080.0 -37700.0 -0.68 -0.7812 -0.9745 3186741 PK04_094210 COCCCNC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K13 compound treatment 768480.0 -411000.0 -6.87 700960.0 -479000.0 -8.63 -10.9597 -0.9936 3068666 PK04_094211 CN(C)C(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K14 compound treatment 1172840.0 -6290.0 -0.11 1172400.0 -7400.0 -0.13 -0.1687 -0.9931 3186742 PK04_094212 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K15 mock treatment 1178160.0 -965.0 -0.02 1178800.0 -1000.0 -0.02 -0.0242 -0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K16 mock treatment 1172320.0 -6810.0 -0.11 1181360.0 1560.0 0.03 -0.0607 -0.5175 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K17 compound treatment 1082760.0 -96400.0 -1.61 1047640.0 -132000.0 -2.38 -2.8241 -0.982 3186743 PK04_094213 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K18 compound treatment 1037200.0 -142000.0 -2.38 991680.0 -188000.0 -3.39 -4.0761 -0.9849 3068667 PK04_094214 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K19 compound treatment 848440.0 -331000.0 -5.53 762800.0 -417000.0 -7.51 -9.2257 -0.9887 3186744 PK04_094215 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K20 compound treatment 1158680.0 -20400.0 -0.34 1147120.0 -32700.0 -0.59 -0.6583 -0.9666 3186745 PK04_094216 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K21 compound treatment 1143000.0 -36100.0 -0.6 1138640.0 -41200.0 -0.74 -0.9519 -0.9949 3068668 PK04_094217 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K22 compound treatment 1153200.0 -25900.0 -0.43 1141560.0 -38200.0 -0.69 -0.794 -0.9751 3186746 PK04_094218 CN(C)C(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K23 mock treatment 1139840.0 -39300.0 -0.66 1154160.0 -25600.0 -0.46 -0.7916 -0.9851 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 K24 mock treatment 1131400.0 -47700.0 -0.8 1142320.0 -37500.0 -0.68 -1.0423 -0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L01 compound treatment 1113160.0 -66000.0 -1.1 1127520.0 -52300.0 -0.94 -1.4467 -0.9969 3068669 PK04_094219 CCOC(=O)N1C(N=C(N1C(=O)OCC)c2ccc(OCCCO)cc2)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L02 compound treatment 1220280.0 41200.0 0.69 1227080.0 47300.0 0.85 1.0893 0.9944 3001020 PK04_094220 CCc1cccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3c4ccccc4)[C@H]2OC(=O)Nc5ccccc5c6ccccc6)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L03 compound treatment 760720.0 -418000.0 -7.0 748160.0 -432000.0 -7.78 -10.4502 -0.9986 3068670 PK04_094221 COCCCNC(=O)C1ON(C(=N1)c2ccc(OCCCO)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L04 compound treatment 1224280.0 45200.0 0.76 1210320.0 30500.0 0.55 0.9231 0.9878 3089829 PK04_094222 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L05 compound treatment 857920.0 -321000.0 -5.38 862800.0 -317000.0 -5.71 -7.8395 -0.9995 3186813 PK04_094223 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L06 compound treatment 1188240.0 9120.0 0.15 1180880.0 1080.0 0.02 0.1216 0.7907 3001022 PK04_094224 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L07 mock treatment 1192240.0 13100.0 0.22 1194200.0 14400.0 0.26 0.3386 0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L08 mock treatment 1185600.0 6480.0 0.11 1196840.0 17000.0 0.31 0.2937 0.9022 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L09 compound treatment 1129560.0 -49600.0 -0.83 1097320.0 -82500.0 -1.49 -1.6374 -0.9621 3067926 PK04_094225 COC(=O)[C@]1(CO)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L10 compound treatment 1186760.0 7640.0 0.13 1188200.0 8400.0 0.15 0.1973 0.9965 3089768 PK04_094226 CCOC(=O)c1ccc(NC(=O)O[C@@H]2[C@@H](CO)O[C@H](OC)[C@@H](OC(=O)Nc3ccccc3)[C@H]2OC(=O)Nc4ccccc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L11 compound treatment 1155640.0 -23500.0 -0.39 1148520.0 -31300.0 -0.56 -0.6765 -0.9845 3186815 PK04_094227 COC(=O)[C@]1(CO)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L12 compound treatment 1204680.0 25600.0 0.43 1218680.0 38900.0 0.7 0.7977 0.972 3089830 PK04_094228 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(cc2)C(F)(F)F)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L13 compound treatment 818120.0 -361000.0 -6.04 659960.0 -520000.0 -9.37 -10.8947 -0.9775 3067927 PK04_094229 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L14 compound treatment 1160400.0 -18700.0 -0.31 1171280.0 -8520.0 -0.15 -0.3302 -0.9461 3089831 PK04_094230 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2c(C)cccc2OC)[C@H](OC(=O)Nc3ccccc3c4ccccc4)[C@@H]1OC(=O)Nc5ccccc5c6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L15 mock treatment 1151000.0 -28100.0 -0.47 1150520.0 -29300.0 -0.53 -0.7059 -0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L16 mock treatment 1156080.0 -23000.0 -0.39 1160120.0 -19700.0 -0.35 -0.5235 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L17 compound treatment 880440.0 -299000.0 -5.0 759360.0 -420000.0 -7.58 -8.8909 -0.9796 3067928 PK04_094231 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L18 compound treatment 1156600.0 -22500.0 -0.38 1162640.0 -17200.0 -0.31 -0.4852 -0.9952 3001180 PK04_094232 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@@H]1OC(=O)Nc6ccccc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L19 compound treatment 895880.0 -283000.0 -4.74 802760.0 -377000.0 -6.79 -8.1552 -0.9845 3067929 PK04_094233 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L20 compound treatment 1148040.0 -31100.0 -0.52 1141320.0 -38500.0 -0.69 -0.8581 -0.99 3001092 PK04_094234 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2c3ccccc3)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@@H]1OC(=O)Nc6ccccc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L21 compound treatment 825720.0 -353000.0 -5.91 673040.0 -507000.0 -9.13 -10.6381 -0.9779 3067930 PK04_094235 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L22 compound treatment 1150400.0 -28700.0 -0.48 1152320.0 -27500.0 -0.5 -0.69 -0.9999 3001093 PK04_094236 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Oc3ccccc3)cc2)[C@H](OC(=O)Nc4ccccc4c5ccccc5)[C@@H]1OC(=O)Nc6ccccc6c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L23 mock treatment 1103840.0 -75300.0 -1.26 1094400.0 -85400.0 -1.54 -1.9789 -0.9951 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 L24 mock treatment 1149400.0 -29700.0 -0.5 1145400.0 -34400.0 -0.62 -0.79 -0.9941 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M01 compound treatment 1201080.0 22000.0 0.37 1190840.0 11000.0 0.2 0.4004 0.9584 3067931 PK04_094237 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M02 compound treatment 1026280.0 -153000.0 -2.56 1033880.0 -146000.0 -2.63 -3.6677 -0.9999 3186821 PK04_094238 COCCCNC(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M03 compound treatment 1217000.0 37900.0 0.63 1211800.0 32000.0 0.58 0.8558 0.9989 3067933 PK04_094239 NC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M04 compound treatment 1213280.0 34200.0 0.57 1223840.0 44000.0 0.79 0.9652 0.987 3186822 PK04_094240 CC(C)(C)OC(=O)CC[C@@]1(COC(=N1)c2ccc(OCCCO)cc2)C(=O)NCCN3CCOCC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M05 compound treatment 1198240.0 19100.0 0.32 1197480.0 17700.0 0.32 0.4514 1.0 3067934 PK04_094241 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)(CO2)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M06 compound treatment 879840.0 -299000.0 -5.01 804280.0 -376000.0 -6.77 -8.3257 -0.989 3186823 PK04_094242 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M07 compound treatment 974320.0 -205000.0 -3.43 973400.0 -206000.0 -3.72 -5.0531 -0.9992 3186824 PK04_094243 CN(C)C(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M08 compound treatment 1047400.0 -132000.0 -2.2 1046080.0 -134000.0 -2.41 -3.2624 -0.999 3186825 PK04_094244 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M09 mock treatment 1203000.0 23900.0 0.4 1208600.0 28800.0 0.52 0.6494 0.9917 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M10 mock treatment 1181800.0 2680.0 0.04 1186360.0 6560.0 0.12 0.1152 0.9118 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M11 compound treatment 1173600.0 -5530.0 -0.09 1156520.0 -23300.0 -0.42 -0.362 -0.8427 3067981 PK04_094245 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M12 compound treatment 1176600.0 -2530.0 -0.04 1167360.0 -12400.0 -0.22 -0.1884 -0.8258 3186826 PK04_094246 NC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M13 mock treatment 1187000.0 7880.0 0.13 1180640.0 837.0 0.02 0.1038 0.7829 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M14 mock treatment 1185320.0 6200.0 0.1 1177840.0 -1960.0 -0.04 0.0483 0.4409 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M15 compound treatment 1002680.0 -176000.0 -2.95 938960.0 -241000.0 -4.34 -5.1563 -0.9824 3067982 PK04_094247 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M16 compound treatment 988160.0 -191000.0 -3.2 940160.0 -240000.0 -4.32 -5.3128 -0.989 3186827 PK04_094248 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M17 compound treatment 1151640.0 -27500.0 -0.46 1150280.0 -29500.0 -0.53 -0.7014 -0.9974 3067983 PK04_094249 CN(C)C(=O)[C@]1(Cc2ccccc2)N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M18 compound treatment 1138200.0 -40900.0 -0.68 1130360.0 -49400.0 -0.89 -1.1142 -0.9916 3186828 PK04_094250 NC(=O)[C@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@@H]1c3ccccc3CN=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M19 compound treatment 1151240.0 -27900.0 -0.47 1139760.0 -40000.0 -0.72 -0.8401 -0.9778 3186829 PK04_094251 CN(C)C(=O)[C@]1(CC=C)N=C(O[C@@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M20 compound treatment 872560.0 -307000.0 -5.13 825520.0 -354000.0 -6.38 -8.1412 -0.9941 3067984 PK04_094252 NC(=O)[C@@]1(Cc2ccccc2)N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M21 compound treatment 1123360.0 -55800.0 -0.93 1120560.0 -59200.0 -1.07 -1.4146 -0.9978 3186907 PK04_094253 OCCCOc1ccc(cc1)C2=N[C@](CCS(=O)(=O)c3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M22 compound treatment 1134680.0 -44400.0 -0.74 1125600.0 -54200.0 -0.98 -1.2165 -0.991 3067985 PK04_094254 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M23 compound treatment 1089160.0 -90000.0 -1.51 1081880.0 -97900.0 -1.76 -2.3121 -0.9969 3186908 PK04_094255 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 M24 compound treatment 1029440.0 -150000.0 -2.5 1029440.0 -150000.0 -2.71 -3.6869 -0.9992 3186909 PK04_094256 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N01 compound treatment 692440.0 -487000.0 -8.14 687920.0 -492000.0 -8.86 -12.0256 -0.9991 3067986 PK04_094257 OCCCOc1ccc(cc1)C2=NC(ON2c3ccccc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N02 compound treatment 1215000.0 35900.0 0.6 1206880.0 27100.0 0.49 0.7695 0.9947 3186910 PK04_094258 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N03 compound treatment 585600.0 -594000.0 -9.93 560160.0 -620000.0 -11.16 -14.9176 -0.9983 3067987 PK04_094259 CN(C)C(=O)C1ON(C(=N1)c2ccc(OCCCO)cc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N04 compound treatment 1191760.0 12600.0 0.21 1190840.0 11000.0 0.2 0.2901 0.9995 3186911 PK04_094260 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N05 compound treatment 618160.0 -561000.0 -9.39 621560.0 -558000.0 -10.06 -13.75 -0.9994 3414052 PK04_094261 COC(=O)[C@@H]1N=C(O[C@@H]1C)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N06 compound treatment 1174440.0 -4690.0 -0.08 1195120.0 15300.0 0.28 0.1397 0.4869 3186912 PK04_094262 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N07 compound treatment 1191560.0 12400.0 0.21 1196120.0 16300.0 0.29 0.355 0.9857 3186913 PK04_094263 OCC(NS(=O)(=O)c1ccc(Br)cc1)C=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N08 compound treatment 1166280.0 -12800.0 -0.21 1169480.0 -10300.0 -0.19 -0.2835 -0.9974 1952953 PK04_094264 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N09 mock treatment 1179040.0 -85.0 0.0 1182680.0 2880.0 0.05 0.0356 0.6874 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N10 mock treatment 1163960.0 -15200.0 -0.25 1177200.0 -2600.0 -0.05 -0.2126 -0.8238 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N11 compound treatment 1180520.0 1400.0 0.02 1166840.0 -13000.0 -0.23 -0.1486 -0.6333 3068027 PK04_094265 CC(=O)OC[C@H](C=C)N(C(=O)OC(C)(C)C)S(=O)(=O)c1ccc(Br)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N12 compound treatment 1167360.0 -11800.0 -0.2 1154960.0 -24800.0 -0.45 -0.4557 -0.932 3186914 PK04_094266 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2cccc(F)c2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N13 mock treatment 1169960.0 -9170.0 -0.15 1155920.0 -23900.0 -0.43 -0.4127 -0.9035 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N14 mock treatment 1166120.0 -13000.0 -0.22 1156040.0 -23800.0 -0.43 -0.4566 -0.9508 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N15 compound treatment 1148440.0 -30700.0 -0.51 1143680.0 -36100.0 -0.65 -0.8233 -0.9931 3068028 PK04_094267 CC(=O)OC[C@@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N16 compound treatment 1142560.0 -36600.0 -0.61 1135920.0 -43900.0 -0.79 -0.9918 -0.992 3186915 PK04_094268 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N17 compound treatment 1158240.0 -20900.0 -0.35 1159720.0 -20100.0 -0.36 -0.503 -0.9998 3068029 PK04_094269 CC(=O)OC[C@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N18 compound treatment 1137720.0 -41400.0 -0.69 1138640.0 -41200.0 -0.74 -1.0144 -0.9994 1952947 PK04_094270 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@@H]4OC(=O)[C@@H](Cc5ccccc5)C/C=C/C[C@H](Cc6ccccc6)C(=O)O[C@@H]14 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N19 compound treatment 1143920.0 -35200.0 -0.59 1143640.0 -36200.0 -0.65 -0.8773 -0.9987 3068030 PK04_094271 OC[C@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N20 compound treatment 1122800.0 -56300.0 -0.94 1123640.0 -56200.0 -1.01 -1.382 -0.9994 3186916 PK04_094272 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(Br)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N21 compound treatment 1121800.0 -57300.0 -0.96 1109560.0 -70200.0 -1.27 -1.5732 -0.9907 3068031 PK04_094273 CC(=O)OC[C@@H](C=C)N(C(=O)OC(C)(C)C)S(=O)(=O)c1ccc(Br)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N22 compound treatment 1112080.0 -67000.0 -1.12 1124400.0 -55400.0 -1.0 -1.4992 -0.9983 1952944 PK04_094274 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(C#N)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccccc4)C/C=C/C[C@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N23 compound treatment 1145600.0 -33500.0 -0.56 1117520.0 -62300.0 -1.12 -1.1902 -0.9487 3186917 PK04_094275 CC(=O)OC[C@H](C=C)N(Cc1ccc(cc1)[N+](=O)[O-])S(=O)(=O)c2ccc(Br)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 N24 compound treatment 1139120.0 -40000.0 -0.67 1122320.0 -57500.0 -1.04 -1.2057 -0.9777 3413982 PK04_094276 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O01 compound treatment 904800.0 -274000.0 -4.59 920600.0 -259000.0 -4.67 -6.5484 -1.0 3068032 PK04_094277 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4N=[N+]=[N-])C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O02 compound treatment 1196760.0 17600.0 0.3 1201560.0 21800.0 0.39 0.4859 0.9902 3186919 PK04_094278 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3)([C@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O03 compound treatment 1192720.0 13600.0 0.23 1192480.0 12700.0 0.23 0.3224 1.0 3068033 PK04_094279 NC(=O)[C@@]1(CC=C)COC(=N1)c2ccc(OCCCO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O04 compound treatment 1162920.0 -16200.0 -0.27 1185680.0 5880.0 0.11 -0.1169 -0.4015 3186920 PK04_094280 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O05 compound treatment 1188800.0 9680.0 0.16 1177880.0 -1920.0 -0.03 0.09 0.5435 3068035 PK04_094281 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3CN=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O06 compound treatment 1009080.0 -170000.0 -2.85 1046360.0 -133000.0 -2.4 -3.7122 -0.9965 3186921 PK04_094282 CN(C)C(=O)[C@@]1(Cc2ccccc2N=[N+]=[N-])COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O07 compound treatment 1137320.0 -41800.0 -0.7 1134080.0 -45700.0 -0.82 -1.0772 -0.9967 3186922 PK04_094283 CN(C)C(=O)[C@]1(Cc2ccccc2N=[N+]=[N-])N=C(O[C@@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O08 compound treatment 1061760.0 -117000.0 -1.96 1078160.0 -102000.0 -1.83 -2.6837 -0.9994 3068037 PK04_094284 CN(C)C(=O)[C@@]1(Cc2ccccc2)COC(=N1)c3ccc(OCCCO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O09 compound treatment 1158280.0 -20800.0 -0.35 1149440.0 -30400.0 -0.55 -0.6335 -0.9764 3186923 PK04_094285 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3)([C@@H](O2)c4ccccc4CN=[N+]=[N-])C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O10 compound treatment 1094760.0 -84400.0 -1.41 1102080.0 -77700.0 -1.4 -1.9885 -1.0 3068038 PK04_094286 OCCCOc1ccc(cc1)C2=N[C@@](Cc3ccccc3N=[N+]=[N-])([C@@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O11 mock treatment 1171600.0 -7530.0 -0.13 1179160.0 -643.0 -0.01 -0.0972 -0.7689 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O12 mock treatment 1189200.0 10100.0 0.17 1173240.0 -6560.0 -0.12 0.0356 0.1729 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O13 compound treatment 1099160.0 -80000.0 -1.34 1098000.0 -81800.0 -1.47 -1.9884 -0.9988 3186924 PK04_094287 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2)c3ccc(OCCCO)cc3)C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O14 compound treatment 1093880.0 -85200.0 -1.43 1093240.0 -86600.0 -1.56 -2.1115 -0.999 3186925 PK04_094288 CC(C)(C)OC(=O)CC[C@@]1(N=C(O[C@H]1c2ccccc2CN=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O15 compound treatment 778360.0 -401000.0 -6.71 726760.0 -453000.0 -8.16 -10.5141 -0.9952 3187013 PK04_094289 CC(C)(C)OC(=O)CC[C@]1(N=C(O[C@@H]1c2ccccc2N=[N+]=[N-])c3ccc(OCCCO)cc3)C(=O)N 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O16 compound treatment 1125760.0 -53400.0 -0.89 1114720.0 -65100.0 -1.17 -1.4606 -0.991 3068077 PK04_094290 OCCCOc1ccc(cc1)C2=N[C@@](CC=C)([C@@H](O2)c3ccccc3CN=[N+]=[N-])C(=O)N4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O17 compound treatment 1083480.0 -95600.0 -1.6 1077040.0 -103000.0 -1.85 -2.441 -0.9974 3187014 PK04_094291 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)NCC(O)CO 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O18 compound treatment 1091720.0 -87400.0 -1.46 1070160.0 -110000.0 -1.98 -2.4311 -0.9891 3187015 PK04_094292 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O19 compound treatment 1059720.0 -119000.0 -2.0 1061960.0 -118000.0 -2.12 -2.9143 -0.9995 3068081 PK04_094293 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])(CO2)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O20 compound treatment 1119120.0 -60000.0 -1.0 1101000.0 -78800.0 -1.42 -1.714 -0.9856 3187016 PK04_094294 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3CN=[N+]=[N-])(CO2)C(=O)N4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O21 compound treatment 1104560.0 -74600.0 -1.25 1108880.0 -70900.0 -1.28 -1.7859 -0.9999 3187017 PK04_094295 COCCCNC(=O)[C@@]1(CCS(=O)(=O)c2ccccc2)N=C(O[C@H]1c3ccccc3)c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O22 compound treatment 979720.0 -199000.0 -3.34 982400.0 -197000.0 -3.56 -4.8745 -0.9995 3068083 PK04_094296 COCCCNC(=O)[C@@]1(Cc2ccccc2CN=[N+]=[N-])N=C(O[C@H]1c3ccccc3N=[N+]=[N-])c4ccc(OCCCO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O23 compound treatment 1057720.0 -121000.0 -2.03 1058440.0 -121000.0 -2.19 -2.9828 -0.9993 3187018 PK04_094297 OCCCOc1ccc(cc1)C2=N[C@](Cc3ccccc3N=[N+]=[N-])([C@H](O2)c4ccccc4)C(=O)N5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 O24 compound treatment 1138280.0 -40800.0 -0.68 1135160.0 -44600.0 -0.8 -1.0521 -0.9967 3068084 PK04_094298 OCCCOc1ccc(cc1)C2=N[C@](CC=C)([C@H](O2)c3ccccc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P01 compound treatment 1198280.0 19200.0 0.32 1188280.0 8480.0 0.15 0.3347 0.9425 3187019 PK04_094299 CC(=O)OC[C@H](C=C)N(Cc1ccccc1[N+](=O)[O-])S(=O)(=O)c2ccc(Br)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P02 compound treatment 1206880.0 27800.0 0.46 1205720.0 25900.0 0.47 0.6586 1.0 3413984 PK04_094300 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P03 compound treatment 1189920.0 10800.0 0.18 1197720.0 17900.0 0.32 0.356 0.9624 3068086 PK04_094301 COc1ccc(CN([C@H](CO)C=C)S(=O)(=O)c2ccc(Br)cc2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P04 compound treatment 1186720.0 7600.0 0.13 1182400.0 2600.0 0.05 0.123 0.9078 3413986 PK04_094302 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P05 compound treatment 1195640.0 16500.0 0.28 1185760.0 5960.0 0.11 0.2713 0.9151 3068087 PK04_094303 COc1cc(CN([C@@H](COC(=O)C)C=C)S(=O)(=O)c2ccc(Br)cc2)ccc1OC(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P06 compound treatment 1158840.0 -20300.0 -0.34 1150240.0 -29600.0 -0.53 -0.6167 -0.9763 1952975 PK04_094304 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P07 compound treatment 1183560.0 4440.0 0.07 1170800.0 -9000.0 -0.16 -0.0622 -0.3488 3068088 PK04_094305 OCCCNS(=O)(=O)c1ccc(Br)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P08 compound treatment 1113280.0 -65800.0 -1.1 1129400.0 -50400.0 -0.91 -1.4213 -0.9954 3413993 PK04_094306 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@H](Cc4ccccc4)C/C=C/C[C@@H](Cc5ccccc5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P09 compound treatment 1186040.0 6920.0 0.12 1177920.0 -1880.0 -0.03 0.0578 0.4796 3068089 PK04_094307 CC[Si](CC)(CC)OC[C@@H](C=C)N(Cc1ccc(OC(=O)C)c(OC)c1)S(=O)(=O)c2ccc(Br)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P10 compound treatment 1102880.0 -76200.0 -1.28 1093920.0 -85900.0 -1.55 -1.9964 -0.9954 1952969 PK04_094308 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc3OCOc3c2)[C@@H]4OC(=O)[C@H](Cc5ccccc5)C/C=C/C[C@@H](Cc6ccccc6)C(=O)O[C@@H]14 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P11 mock treatment 1163240.0 -15900.0 -0.27 1147800.0 -32000.0 -0.58 -0.5957 -0.9382 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P12 mock treatment 1172720.0 -6410.0 -0.11 1165640.0 -14200.0 -0.26 -0.2562 -0.9258 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P13 compound treatment 1155200.0 -23900.0 -0.4 1143680.0 -36100.0 -0.65 -0.7433 -0.9728 3068090 PK04_094309 COc1cc(CO)ccc1OC(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P14 compound treatment 1146280.0 -32800.0 -0.55 1135080.0 -44700.0 -0.81 -0.9584 -0.9826 3068091 PK04_094310 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P15 compound treatment 974120.0 -205000.0 -3.43 957680.0 -222000.0 -4.0 -5.2557 -0.9971 3187025 PK04_094311 COc1ccc(CN(C2=CC[C@@]3(C(=O)N)C(=O)C(=C(Cl)C(=O)[C@]3(C2)C#N)Cl)S(=O)(=O)c4ccc(Br)cc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P16 compound treatment 1125560.0 -53600.0 -0.9 1129120.0 -50700.0 -0.91 -1.2795 -1.0 3187026 PK04_094312 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2ccc(Br)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P17 compound treatment 1144760.0 -34400.0 -0.58 1129760.0 -50000.0 -0.9 -1.0442 -0.9764 3068092 PK04_094313 CC(C)(C)OC(=O)N1[C@H](COC1(C)C)C=C(Br)Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P18 compound treatment 1122280.0 -56800.0 -0.95 1129680.0 -50100.0 -0.9 -1.3112 -0.9997 3187027 PK04_094314 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)c2c(OC)cccc2OC)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P19 compound treatment 1140160.0 -39000.0 -0.65 1121760.0 -58000.0 -1.05 -1.2006 -0.9742 1003211 PK04_094315 CNS(=O)(=O)c1ccc(C)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P20 compound treatment 1093400.0 -85700.0 -1.43 1104600.0 -75200.0 -1.35 -1.9725 -0.9996 3187028 PK04_094316 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccccc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P21 compound treatment 1121480.0 -57600.0 -0.96 1113680.0 -66100.0 -1.19 -1.5245 -0.9945 3068127 PK04_094317 COc1cc(COC(=O)C)ccc1OC(=O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P22 compound treatment 1085040.0 -94100.0 -1.57 1074240.0 -106000.0 -1.9 -2.4582 -0.9956 3187029 PK04_094318 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)Nc2ccc(OC)cc2)[C@@H]3OC(=O)[C@@H](Cc4ccc5ccccc5c4)C/C=C/C[C@H](Cc6ccc7ccccc7c6)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P23 compound treatment 1127960.0 -51200.0 -0.86 1131120.0 -48700.0 -0.88 -1.2257 -0.9999 3068129 PK04_094319 OC[C@@H](NS(=O)(=O)c1ccc(Br)cc1)C=C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2094 P24 compound treatment 1141680.0 -37400.0 -0.63 1130640.0 -49200.0 -0.89 -1.0694 -0.9856 3413981 PK04_094320 CO[C@H]1O[C@H](CO)[C@@H](OC(=O)CCc2ccccc2)[C@@H]3OC(=O)[C@H](Cc4cccc(Br)c4)C/C=C/C[C@@H](Cc5cccc(Br)c5)C(=O)O[C@@H]13 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A01 compound treatment 1220080.0 38200.0 0.64 1228120.0 42800.0 0.77 0.9967 0.9957 3067957 PK04_095001 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NC4CC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A02 compound treatment 1251280.0 69400.0 1.16 1232960.0 47600.0 0.86 1.4275 0.9889 3187176 PK04_095002 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2OC)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A03 compound treatment 1234880.0 53000.0 0.89 1241440.0 56100.0 1.01 1.3415 0.9979 3067577 PK04_095003 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCc6ccccc6)c7ccc(cc7)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A04 compound treatment 1234800.0 52900.0 0.89 1223080.0 37700.0 0.68 1.1066 0.9915 3187436 PK04_095004 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A05 compound treatment 1220440.0 38600.0 0.65 1199880.0 14500.0 0.26 0.6411 0.921 3186425 PK04_095005 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc6I)c7ccc(cc7)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A06 compound treatment 1232280.0 50400.0 0.84 1220600.0 35200.0 0.63 1.0452 0.9902 3187069 PK04_095006 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A07 compound treatment 1205200.0 23300.0 0.39 1204280.0 18900.0 0.34 0.5169 0.9977 3187427 PK04_095007 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A08 compound treatment 1203040.0 21200.0 0.35 1197920.0 12600.0 0.23 0.4103 0.9766 3187515 PK04_095008 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc6)c7ccc(cc7)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A09 compound treatment 1204520.0 22600.0 0.38 1196400.0 11000.0 0.2 0.4084 0.9547 3187425 PK04_095009 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A10 compound treatment 1195440.0 13600.0 0.23 1198640.0 13300.0 0.24 0.3295 0.9996 3068592 PK04_095010 CCCNC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A11 compound treatment 1195120.0 13200.0 0.22 1195080.0 9720.0 0.18 0.2804 0.9932 3187517 PK04_095011 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A12 compound treatment 1207840.0 26000.0 0.43 1195600.0 10200.0 0.18 0.4375 0.9272 3187344 PK04_095012 COCCCNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A13 mock treatment 1201400.0 19500.0 0.33 1190400.0 5040.0 0.09 0.2951 0.8706 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A14 mock treatment 1199160.0 17300.0 0.29 1208360.0 23000.0 0.41 0.4974 0.9845 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A15 compound treatment 1178680.0 -3210.0 -0.05 1189400.0 4040.0 0.07 0.0135 0.1491 3186552 PK04_095013 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A16 compound treatment 1190080.0 8190.0 0.14 1176680.0 -8680.0 -0.16 -0.0137 -0.0658 3187439 PK04_095014 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A17 compound treatment 1169720.0 -12200.0 -0.2 1163440.0 -21900.0 -0.4 -0.4233 -0.9525 3187073 PK04_095015 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A18 compound treatment 1189280.0 7390.0 0.12 1171920.0 -13400.0 -0.24 -0.0838 -0.3081 3187272 PK04_095016 COCCCNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A19 compound treatment 1174400.0 -7490.0 -0.13 1172400.0 -13000.0 -0.23 -0.2538 -0.9574 3187508 PK04_095017 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NC3CC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A20 compound treatment 1169000.0 -12900.0 -0.22 1155160.0 -30200.0 -0.54 -0.5373 -0.9179 3186432 PK04_095018 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(Cc5ccccc5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A21 compound treatment 1159960.0 -21900.0 -0.37 1137600.0 -47800.0 -0.86 -0.868 -0.9278 3068646 PK04_095019 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A22 compound treatment 1183320.0 1430.0 0.02 1156760.0 -28600.0 -0.52 -0.3475 -0.6735 3068651 PK04_095020 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A23 compound treatment 1157200.0 -24700.0 -0.41 1148880.0 -36500.0 -0.66 -0.7569 -0.9749 3187585 PK04_095021 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 A24 compound treatment 1168360.0 -13500.0 -0.23 1155280.0 -30100.0 -0.54 -0.5433 -0.925 3187430 PK04_095022 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B01 compound treatment 1176280.0 -5610.0 -0.09 1158320.0 -27000.0 -0.49 -0.4109 -0.828 3187519 PK04_095023 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)O)c4ccc(cc4)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B02 compound treatment 1251280.0 69400.0 1.16 1244680.0 59300.0 1.07 1.5768 0.9991 3186885 PK04_095024 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B03 compound treatment 1247880.0 66000.0 1.1 1239520.0 54200.0 0.98 1.4709 0.9981 3187435 PK04_095025 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B04 compound treatment 1231800.0 49900.0 0.84 1213560.0 28200.0 0.51 0.9498 0.9716 3186491 PK04_095026 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B05 compound treatment 1224320.0 42400.0 0.71 1231000.0 45600.0 0.82 1.0835 0.9973 3068539 PK04_095027 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4cc(F)cc(c4)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B06 compound treatment 1225280.0 43400.0 0.73 1234120.0 48800.0 0.88 1.1346 0.9955 3186559 PK04_095028 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B07 compound treatment 1198560.0 16700.0 0.28 1202160.0 16800.0 0.3 0.4113 0.9992 3068561 PK04_095029 CCCNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B08 compound treatment 1213920.0 32000.0 0.54 1218120.0 32800.0 0.59 0.7964 0.9988 3068322 PK04_095030 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B09 compound treatment 1197760.0 15900.0 0.27 1200920.0 15600.0 0.28 0.386 0.9996 3187432 PK04_095031 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B10 compound treatment 1198400.0 16500.0 0.28 1197240.0 11900.0 0.21 0.3467 0.992 3068145 PK04_095032 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCC(F)(F)F)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B11 compound treatment 1215280.0 33400.0 0.56 1199200.0 13800.0 0.25 0.5714 0.9338 3187265 PK04_095033 CC(C)N1[C@H]([C@H](C(=O)NCCCN(C)C)c2ccccc2C1=O)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B12 compound treatment 1206320.0 24400.0 0.41 1206520.0 21200.0 0.38 0.5587 0.9994 3186629 PK04_095034 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B13 mock treatment 1194520.0 12600.0 0.21 1189800.0 4440.0 0.08 0.206 0.9115 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B14 mock treatment 1186120.0 4230.0 0.07 1197480.0 12100.0 0.22 0.2045 0.8909 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B15 compound treatment 1171080.0 -10800.0 -0.18 1170040.0 -15300.0 -0.28 -0.3231 -0.979 3187269 PK04_095035 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C3CCCCC3)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B16 compound treatment 1169760.0 -12100.0 -0.2 1163160.0 -22200.0 -0.4 -0.4264 -0.9505 3186887 PK04_095036 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B17 compound treatment 1174160.0 -7730.0 -0.13 1167240.0 -18100.0 -0.33 -0.3223 -0.9178 3068417 PK04_095037 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B18 compound treatment 1174880.0 -7010.0 -0.12 1182160.0 -3200.0 -0.06 -0.1237 -0.9467 3067610 PK04_095038 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(C7CC7)c2c1)c8ccc(cc8)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B19 compound treatment 1140320.0 -41600.0 -0.7 1149640.0 -35700.0 -0.64 -0.947 -0.9992 3068639 PK04_095039 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3cc(F)cc(c3)C(F)(F)F)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B20 compound treatment 1145640.0 -36200.0 -0.61 1140640.0 -44700.0 -0.81 -0.9987 -0.9902 3068006 PK04_095040 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B21 compound treatment 1143800.0 -38100.0 -0.64 1134360.0 -51000.0 -0.92 -1.1005 -0.984 3068601 PK04_095041 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NCc4ccccc4)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B22 compound treatment 1152960.0 -28900.0 -0.48 1147680.0 -37700.0 -0.68 -0.8224 -0.9862 3068203 PK04_095042 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5Cl)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B23 compound treatment 1160120.0 -21800.0 -0.36 1152280.0 -33100.0 -0.6 -0.6791 -0.9721 3187355 PK04_095043 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NCC(F)(F)F)c4ccccc4C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 B24 compound treatment 1173080.0 -8810.0 -0.15 1172000.0 -13400.0 -0.24 -0.2745 -0.9722 3068156 PK04_095044 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C01 compound treatment 1218760.0 36900.0 0.62 1210720.0 25400.0 0.46 0.7594 0.9891 3187590 PK04_095045 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C02 compound treatment 1238520.0 56600.0 0.95 1230840.0 45500.0 0.82 1.2495 0.9974 3187180 PK04_095046 CC(C)NC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C03 compound treatment 1224520.0 42600.0 0.71 1220200.0 34800.0 0.63 0.9483 0.998 3186493 PK04_095047 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C04 compound treatment 1125040.0 -56800.0 -0.95 1123360.0 -62000.0 -1.12 -1.4626 -0.9968 3186427 PK04_095048 CN(C)CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C05 compound treatment 1214880.0 33000.0 0.55 1210120.0 24800.0 0.45 0.7058 0.9944 3187172 PK04_095049 COc1ccccc1CN2[C@H]([C@H](C(=O)NCCN3CCOCC3)c4ccccc4C2=O)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C06 compound treatment 1208280.0 26400.0 0.44 1214280.0 28900.0 0.52 0.6807 0.9966 3187080 PK04_095050 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C07 compound treatment 1187960.0 6070.0 0.1 1185400.0 35.6 0.0 0.0723 0.7116 3186988 PK04_095051 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C08 compound treatment 1191920.0 10000.0 0.17 1202840.0 17500.0 0.31 0.3414 0.9567 3068011 PK04_095052 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C09 compound treatment 1185720.0 3830.0 0.06 1187800.0 2440.0 0.04 0.0764 0.9828 3068498 PK04_095053 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C10 compound treatment 1186240.0 4350.0 0.07 1190920.0 5560.0 0.1 0.1223 0.9878 3186550 PK04_095054 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C11 mock treatment 1184440.0 2550.0 0.04 1184360.0 -1000.0 -0.02 0.0174 0.3754 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C12 mock treatment 1201880.0 20000.0 0.33 1183760.0 -1600.0 -0.03 0.2161 0.6436 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C13 compound treatment 1171920.0 -9970.0 -0.17 1177440.0 -7920.0 -0.14 -0.2189 -0.997 3187361 PK04_095055 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C14 compound treatment 1178760.0 -3130.0 -0.05 1169200.0 -16200.0 -0.29 -0.2429 -0.821 3068504 PK04_095056 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccc(OC(F)(F)F)cc3)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C15 mock treatment 1185320.0 3430.0 0.06 1167920.0 -17400.0 -0.31 -0.1816 -0.5684 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C16 mock treatment 1176320.0 -5570.0 -0.09 1173800.0 -11600.0 -0.21 -0.2132 -0.9341 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C17 compound treatment 1175240.0 -6650.0 -0.11 1169040.0 -16300.0 -0.29 -0.2866 -0.9115 3067969 PK04_095057 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCCCN(C)C)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C18 compound treatment 1160240.0 -21600.0 -0.36 1156120.0 -29200.0 -0.53 -0.6287 -0.9833 3187359 PK04_095058 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(Cc3ccc(OC(F)(F)F)cc3)C(=O)c4ccccc42)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C19 compound treatment 1151120.0 -30800.0 -0.51 1155000.0 -30400.0 -0.55 -0.7509 -0.9995 3187087 PK04_095059 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C20 compound treatment 1162080.0 -19800.0 -0.33 1164440.0 -20900.0 -0.38 -0.5009 -0.9979 3187443 PK04_095060 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C21 compound treatment 1147600.0 -34300.0 -0.57 1147920.0 -37400.0 -0.67 -0.8828 -0.9968 3067571 PK04_095061 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C22 compound treatment 1153480.0 -28400.0 -0.48 1161360.0 -24000.0 -0.43 -0.642 -0.9989 3187181 PK04_095062 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NCC(F)(F)F)c3ccccc3C2=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C23 compound treatment 1148400.0 -33500.0 -0.56 1142760.0 -42600.0 -0.77 -0.939 -0.988 3187509 PK04_095063 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C(C)C)[C@@H]2c3ccc(CO)cc3)c4ccc(cc4)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 C24 compound treatment 1151160.0 -30700.0 -0.51 1155240.0 -30100.0 -0.54 -0.7474 -0.9996 3068474 PK04_095064 CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D01 compound treatment 1233840.0 52000.0 0.87 1243480.0 58100.0 1.05 1.3552 0.9957 3068587 PK04_095065 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(CC3(CC4CC5CC(C4)C3)C5)C(=O)c6ccccc26)c7ccc(CO)cc7)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D02 compound treatment 1244720.0 62800.0 1.05 1244480.0 59100.0 1.07 1.4967 1.0 3068318 PK04_095066 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D03 compound treatment 1220200.0 38300.0 0.64 1223720.0 38400.0 0.69 0.942 0.9993 3187363 PK04_095067 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D04 compound treatment 1224600.0 42700.0 0.71 1220960.0 35600.0 0.64 0.9589 0.9985 3186486 PK04_095068 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(CCN7CCOCC7)c2c1)c8ccc(cc8)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D05 compound treatment 1221240.0 39400.0 0.66 1215560.0 30200.0 0.54 0.8504 0.9955 3187179 PK04_095069 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C(=O)c3ccccc23)c4ccc(C)cn4)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D06 compound treatment 1203920.0 22000.0 0.37 1200480.0 15100.0 0.27 0.4533 0.9889 3187522 PK04_095070 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D07 compound treatment 1202040.0 20200.0 0.34 1190880.0 5520.0 0.1 0.3088 0.8781 3068515 PK04_095071 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NC3CC3)c4ccccc4C2=O)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D08 compound treatment 1205280.0 23400.0 0.39 1206400.0 21000.0 0.38 0.5448 0.9999 3186872 PK04_095072 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D09 compound treatment 1192960.0 11100.0 0.19 1186040.0 676.0 0.01 0.1396 0.7519 3068609 PK04_095073 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D10 compound treatment 1189560.0 7670.0 0.13 1204000.0 18600.0 0.34 0.3282 0.913 3186795 PK04_095074 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D11 mock treatment 1196480.0 14600.0 0.24 1190800.0 5440.0 0.1 0.2419 0.9195 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D12 mock treatment 1190280.0 8390.0 0.14 1181520.0 -3840.0 -0.07 0.0503 0.3215 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D13 compound treatment 1167080.0 -14800.0 -0.25 1190280.0 4920.0 0.09 -0.1126 -0.4278 3067964 PK04_095075 CCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D14 compound treatment 1167720.0 -14200.0 -0.24 1172120.0 -13200.0 -0.24 -0.3364 -1.0 3068230 PK04_095076 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D15 mock treatment 1164240.0 -17600.0 -0.3 1167360.0 -18000.0 -0.32 -0.4382 -0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D16 mock treatment 1167480.0 -14400.0 -0.24 1167640.0 -17700.0 -0.32 -0.3963 -0.9904 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D17 compound treatment 1138000.0 -43900.0 -0.73 1142880.0 -42500.0 -0.77 -1.0606 -0.9998 3068595 PK04_095077 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCc3ccccc3)c4ccccc4C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D18 compound treatment 1154320.0 -27600.0 -0.46 1150800.0 -34600.0 -0.62 -0.7665 -0.9891 3186982 PK04_095078 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D19 compound treatment 1143080.0 -38800.0 -0.65 1144720.0 -40600.0 -0.73 -0.977 -0.9982 3187440 PK04_095079 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D20 compound treatment 1136560.0 -45300.0 -0.76 1141200.0 -44200.0 -0.8 -1.099 -0.9997 3068415 PK04_095080 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D21 compound treatment 1135840.0 -46000.0 -0.77 1136200.0 -49200.0 -0.89 -1.1712 -0.9976 3068596 PK04_095081 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCC(F)(F)F)c3ccccc3C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D22 compound treatment 1142480.0 -39400.0 -0.66 1146240.0 -39100.0 -0.7 -0.9647 -0.9994 3186713 PK04_095082 CC(C)CNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D23 compound treatment 1132240.0 -49600.0 -0.83 1135480.0 -49900.0 -0.9 -1.223 -0.9992 3187357 PK04_095083 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 D24 compound treatment 1143400.0 -38500.0 -0.64 1156000.0 -29400.0 -0.53 -0.8295 -0.9952 3068270 PK04_095084 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCCN6CCOCC6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E01 mock treatment 1234680.0 52800.0 0.88 1225480.0 40100.0 0.72 1.1358 0.995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E02 mock treatment 1232640.0 50800.0 0.85 1238280.0 52900.0 0.95 1.2747 0.9983 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E03 compound treatment 1220240.0 38400.0 0.64 1216520.0 31200.0 0.56 0.8508 0.9978 3068636 PK04_095085 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E04 compound treatment 1207520.0 25600.0 0.43 1211480.0 26100.0 0.47 0.636 0.9989 3186556 PK04_095086 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E05 compound treatment 1211920.0 30000.0 0.5 1206960.0 21600.0 0.39 0.6305 0.992 3187587 PK04_095087 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E06 compound treatment 1203800.0 21900.0 0.37 1202840.0 17500.0 0.31 0.4819 0.9971 3186428 PK04_095088 COCCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E07 compound treatment 1198240.0 16400.0 0.27 1194600.0 9240.0 0.17 0.3112 0.9716 3187266 PK04_095089 CCCNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E08 compound treatment 1198320.0 16400.0 0.28 1211320.0 26000.0 0.47 0.5251 0.968 3187351 PK04_095090 CC(C)CNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E09 mock treatment 1189200.0 7310.0 0.12 1195840.0 10500.0 0.19 0.22 0.978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E10 mock treatment 1200920.0 19000.0 0.32 1215560.0 30200.0 0.54 0.6099 0.9675 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E11 compound treatment 1183720.0 1830.0 0.03 1181480.0 -3880.0 -0.07 -0.0278 -0.3636 3068004 PK04_095091 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E12 compound treatment 1185400.0 3510.0 0.06 1178280.0 -7080.0 -0.13 -0.0487 -0.3464 3186500 PK04_095092 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E13 compound treatment 1159440.0 -22400.0 -0.38 1185440.0 75.6 0.0 -0.2646 -0.7045 3187346 PK04_095093 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCCN3CCOCC3)c4ccccc4C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E14 compound treatment 1191720.0 9830.0 0.16 1186240.0 876.0 0.02 0.1275 0.7714 3187262 PK04_095094 CC(C)N1[C@H]([C@H](C(=O)NCCN2CCOCC2)c3ccccc3C1=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E15 compound treatment 1170160.0 -11700.0 -0.2 1171320.0 -14000.0 -0.25 -0.3177 -0.9921 3067574 PK04_095095 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NC6CC6)c7ccc(cc7)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E16 compound treatment 1180160.0 -1730.0 -0.03 1160560.0 -24800.0 -0.45 -0.3364 -0.7512 3187350 PK04_095096 COCCCNC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E17 mock treatment 1157880.0 -24000.0 -0.4 1166120.0 -19200.0 -0.35 -0.5292 -0.9973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E18 mock treatment 1161600.0 -20300.0 -0.34 1180920.0 -4440.0 -0.08 -0.2967 -0.8506 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E19 compound treatment 1137760.0 -44100.0 -0.74 1154160.0 -31200.0 -0.56 -0.9197 -0.9909 3068657 PK04_095097 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E20 compound treatment 1149160.0 -32700.0 -0.55 1144200.0 -41200.0 -0.74 -0.9117 -0.9889 3068140 PK04_095098 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E21 compound treatment 1151240.0 -30600.0 -0.51 1154880.0 -30500.0 -0.55 -0.751 -0.9994 3186562 PK04_095099 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E22 compound treatment 1154720.0 -27200.0 -0.45 1144680.0 -40700.0 -0.73 -0.8398 -0.9736 3187591 PK04_095100 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E23 compound treatment 1146520.0 -35400.0 -0.59 1148680.0 -36700.0 -0.66 -0.8859 -0.9985 3187263 PK04_095101 CC(C)N1[C@H]([C@H](C(=O)NCc2ccccc2)c3ccccc3C1=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 E24 compound treatment 1154840.0 -27000.0 -0.45 1160640.0 -24700.0 -0.45 -0.635 -1.0 3068517 PK04_095102 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NCc3ccccc3)c4ccccc4C2=O)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F01 mock treatment 1245520.0 63600.0 1.06 1239800.0 54400.0 0.98 1.4465 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F02 mock treatment 1237480.0 55600.0 0.93 1242840.0 57500.0 1.04 1.3901 0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F03 compound treatment 1222640.0 40800.0 0.68 1219080.0 33700.0 0.61 0.9118 0.9983 3187079 PK04_095103 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F04 compound treatment 1197960.0 16100.0 0.27 1204720.0 19400.0 0.35 0.4368 0.9918 3068331 PK04_095104 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F05 compound treatment 1214080.0 32200.0 0.54 1212960.0 27600.0 0.5 0.7325 0.9992 3068563 PK04_095105 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2CC5(CC6CC7CC(C6)C5)C7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F06 compound treatment 1206560.0 24700.0 0.41 1204840.0 19500.0 0.35 0.5401 0.9967 3186879 PK04_095106 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NCCN6CCOCC6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F07 compound treatment 1194560.0 12700.0 0.21 1196000.0 10600.0 0.19 0.2855 0.9987 3187523 PK04_095107 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F08 compound treatment 1197080.0 15200.0 0.25 1204960.0 19600.0 0.35 0.4294 0.987 3186563 PK04_095108 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F09 mock treatment 1203200.0 21300.0 0.36 1203120.0 17800.0 0.32 0.4784 0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F10 mock treatment 1191560.0 9670.0 0.16 1199920.0 14600.0 0.26 0.2999 0.9731 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F11 compound treatment 1186880.0 4990.0 0.08 1189400.0 4040.0 0.07 0.1105 0.9976 3187257 PK04_095109 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2C5Cc6ccccc6C5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F12 compound treatment 1184280.0 2390.0 0.04 1173640.0 -11700.0 -0.21 -0.121 -0.563 3068241 PK04_095110 CCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F13 compound treatment 1142840.0 -39000.0 -0.65 1174240.0 -11100.0 -0.2 -0.6038 -0.8834 3068554 PK04_095111 COCCCNC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F14 compound treatment 1174120.0 -7770.0 -0.13 1159320.0 -26000.0 -0.47 -0.4237 -0.8702 3068362 PK04_095112 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C(C)C)[C@@H]2c3ccc(CO)cc3)Sc4ccc(C)cc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F15 compound treatment 1165800.0 -16100.0 -0.27 1165200.0 -20200.0 -0.36 -0.4472 -0.9891 3186423 PK04_095113 CC(C)CNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F16 compound treatment 1121520.0 -60400.0 -1.01 1099280.0 -86100.0 -1.55 -1.811 -0.9784 3068012 PK04_095114 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)O)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F17 mock treatment 1139920.0 -42000.0 -0.7 1151240.0 -34100.0 -0.61 -0.9313 -0.9978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F18 mock treatment 1149960.0 -31900.0 -0.53 1157520.0 -27800.0 -0.5 -0.7325 -0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F19 compound treatment 1126600.0 -55300.0 -0.93 1136480.0 -48900.0 -0.88 -1.277 -0.9997 3067568 PK04_095115 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F20 compound treatment 1143200.0 -38700.0 -0.65 1142360.0 -43000.0 -0.77 -1.0057 -0.996 3068266 PK04_095116 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F21 compound treatment 1126600.0 -55300.0 -0.93 1142600.0 -42800.0 -0.77 -1.199 -0.9959 3186419 PK04_095117 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCc4ccccc4)c5ccc(cc5)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F22 compound treatment 1123160.0 -58700.0 -0.98 1137480.0 -47900.0 -0.86 -1.305 -0.9979 3187524 PK04_095118 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F23 compound treatment 1132440.0 -49400.0 -0.83 1116720.0 -68600.0 -1.24 -1.4596 -0.9809 3068017 PK04_095119 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)O)c4ccccc4C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 F24 compound treatment 1138280.0 -43600.0 -0.73 1140560.0 -44800.0 -0.81 -1.0868 -0.9987 3186554 PK04_095120 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G01 compound treatment 1238200.0 56300.0 0.94 1239040.0 53700.0 0.97 1.3502 0.9999 3186418 PK04_095121 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCCN4CCOCC4)c5ccc(cc5)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G02 compound treatment 1234880.0 53000.0 0.89 1247360.0 62000.0 1.12 1.4169 0.9935 3067966 PK04_095122 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCCN3CCOCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G03 mock treatment 1231320.0 49400.0 0.83 1231880.0 46500.0 0.84 1.1776 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G04 mock treatment 1220560.0 38700.0 0.65 1222560.0 37200.0 0.67 0.9315 0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G05 compound treatment 1215520.0 33600.0 0.56 1222680.0 37300.0 0.67 0.8734 0.9961 3068153 PK04_095123 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NC6CC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G06 compound treatment 1203920.0 22000.0 0.37 1205880.0 20500.0 0.37 0.5221 1.0 3187356 PK04_095124 COCCCNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G07 compound treatment 1200760.0 18900.0 0.32 1187920.0 2560.0 0.05 0.2559 0.8017 3187173 PK04_095125 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3OC)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G08 compound treatment 1203000.0 21100.0 0.35 1208480.0 23100.0 0.42 0.5443 0.9967 3068514 PK04_095126 CCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G09 compound treatment 1201080.0 19200.0 0.32 1200000.0 14600.0 0.26 0.4136 0.9952 3187442 PK04_095127 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G10 compound treatment 1197240.0 15400.0 0.26 1203520.0 18200.0 0.33 0.413 0.9929 3068420 PK04_095128 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G11 compound treatment 1184480.0 2590.0 0.04 1197240.0 11900.0 0.21 0.182 0.8336 3187434 PK04_095129 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G12 compound treatment 1159520.0 -22400.0 -0.37 1172840.0 -12500.0 -0.23 -0.4242 -0.9707 3186416 PK04_095130 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G13 compound treatment 1186280.0 4390.0 0.07 1177680.0 -7680.0 -0.14 -0.0459 -0.2928 3068507 PK04_095131 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G14 compound treatment 1181560.0 -326.0 -0.01 1175960.0 -9400.0 -0.17 -0.1237 -0.7295 3187162 PK04_095132 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5cc(F)cc(c5)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G15 compound treatment 1174240.0 -7650.0 -0.13 1180200.0 -5160.0 -0.09 -0.1563 -0.9878 3068602 PK04_095133 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G16 compound treatment 1184080.0 2190.0 0.04 1180360.0 -5000.0 -0.09 -0.0378 -0.3883 3187426 PK04_095134 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G17 compound treatment 1150800.0 -31100.0 -0.52 1158320.0 -27000.0 -0.49 -0.7124 -0.9995 3067567 PK04_095135 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G18 compound treatment 1167200.0 -14700.0 -0.25 1159800.0 -25600.0 -0.46 -0.4995 -0.9567 3187525 PK04_095136 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G19 mock treatment 1151720.0 -30200.0 -0.5 1149920.0 -35400.0 -0.64 -0.8085 -0.9932 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G20 mock treatment 1150000.0 -31900.0 -0.53 1155000.0 -30400.0 -0.55 -0.7642 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G21 compound treatment 1152000.0 -29900.0 -0.5 1148120.0 -37200.0 -0.67 -0.8281 -0.9895 3187167 PK04_095137 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccc(OC(F)(F)F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G22 compound treatment 1151240.0 -30600.0 -0.51 1167840.0 -17500.0 -0.32 -0.5859 -0.9729 3187174 PK04_095138 COc1ccccc1CN2[C@H]([C@H](C(=O)NC(C)C)c3ccccc3C2=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G23 compound treatment 1148840.0 -33000.0 -0.55 1156560.0 -28800.0 -0.52 -0.758 -0.9995 3068478 PK04_095139 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 G24 compound treatment 1133840.0 -48000.0 -0.8 1151080.0 -34300.0 -0.62 -1.0053 -0.9915 3068471 PK04_095140 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H01 compound treatment 1235440.0 53600.0 0.9 1236840.0 51500.0 0.93 1.2895 0.9999 3068149 PK04_095141 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H02 compound treatment 1237400.0 55500.0 0.93 1229720.0 44400.0 0.8 1.222 0.9972 3068236 PK04_095142 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H03 mock treatment 1230080.0 48200.0 0.81 1221400.0 36000.0 0.65 1.0294 0.9942 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H04 mock treatment 1208560.0 26700.0 0.45 1223680.0 38300.0 0.69 0.8038 0.9777 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H05 compound treatment 1211160.0 29300.0 0.49 1212000.0 26600.0 0.48 0.6857 0.9999 3187083 PK04_095143 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H06 compound treatment 1204400.0 22500.0 0.38 1216800.0 31400.0 0.57 0.6669 0.9804 3068265 PK04_095144 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H07 compound treatment 1202000.0 20100.0 0.34 1204880.0 19500.0 0.35 0.4866 0.9998 3068458 PK04_095145 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H08 compound treatment 1208720.0 26800.0 0.45 1216480.0 31100.0 0.56 0.7139 0.994 3068401 PK04_095146 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H09 compound treatment 1198160.0 16300.0 0.27 1210960.0 25600.0 0.46 0.5187 0.9684 3187071 PK04_095147 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H10 compound treatment 1193320.0 11400.0 0.19 1194960.0 9600.0 0.17 0.2575 0.9987 3068139 PK04_095148 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H11 compound treatment 1185640.0 3750.0 0.06 1188120.0 2760.0 0.05 0.0795 0.9932 3187589 PK04_095149 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H12 compound treatment 1169160.0 -12700.0 -0.21 1156240.0 -29100.0 -0.52 -0.5216 -0.9211 3186627 PK04_095150 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4OC)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H13 compound treatment 1175640.0 -6250.0 -0.1 1178560.0 -6800.0 -0.12 -0.1606 -0.9969 3187261 PK04_095151 CC(C)N1[C@H]([C@H](C(=O)NC2CC2)c3ccccc3C1=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H14 compound treatment 1174200.0 -7690.0 -0.13 1168680.0 -16700.0 -0.3 -0.3035 -0.9283 3186980 PK04_095152 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H15 compound treatment 1163440.0 -18400.0 -0.31 1170480.0 -14900.0 -0.27 -0.4079 -0.9975 3187166 PK04_095153 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccc(OC(F)(F)F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H16 compound treatment 1134640.0 -47200.0 -0.79 1160400.0 -25000.0 -0.45 -0.8771 -0.9643 3186978 PK04_095154 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H17 compound treatment 1158360.0 -23500.0 -0.39 1163120.0 -22200.0 -0.4 -0.5618 -1.0 3187349 PK04_095155 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NCCCN(C)C)c3ccccc3C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H18 compound treatment 1155200.0 -26700.0 -0.45 1164240.0 -21100.0 -0.38 -0.5849 -0.9968 3068412 PK04_095156 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H19 mock treatment 1141520.0 -40400.0 -0.68 1155840.0 -29500.0 -0.53 -0.8538 -0.993 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H20 mock treatment 1137360.0 -44500.0 -0.75 1143480.0 -41900.0 -0.75 -1.0605 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H21 compound treatment 1137120.0 -44800.0 -0.75 1149640.0 -35700.0 -0.64 -0.9849 -0.9971 3187512 PK04_095157 COCCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H22 compound treatment 1141920.0 -40000.0 -0.67 1155920.0 -29400.0 -0.53 -0.848 -0.9934 3186806 PK04_095158 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H23 compound treatment 1110160.0 -71700.0 -1.2 1134480.0 -50900.0 -0.92 -1.497 -0.9912 3068599 PK04_095159 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NC4CC4)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 H24 compound treatment 1130840.0 -51000.0 -0.85 1132160.0 -53200.0 -0.96 -1.2819 -0.9983 3187586 PK04_095160 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I01 compound treatment 1233520.0 51600.0 0.86 1225200.0 39800.0 0.72 1.1185 0.9957 3187165 PK04_095161 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccc(OC(F)(F)F)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I02 compound treatment 1235440.0 53600.0 0.9 1242160.0 56800.0 1.02 1.3573 0.9978 3068418 PK04_095162 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I03 compound treatment 1229320.0 47400.0 0.79 1226840.0 41500.0 0.75 1.0897 0.9995 3187178 PK04_095163 Cc1ccc(nc1)N2[C@H]([C@H](C(=O)NCCN3CCOCC3)c4ccccc4C2=O)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I04 compound treatment 1224160.0 42300.0 0.71 1225040.0 39700.0 0.71 1.0057 1.0 3068019 PK04_095164 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I05 mock treatment 1216560.0 34700.0 0.58 1237160.0 51800.0 0.93 1.0702 0.9739 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I06 mock treatment 1211920.0 30000.0 0.5 1228280.0 42900.0 0.77 0.9021 0.9782 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I07 compound treatment 1204760.0 22900.0 0.38 1216840.0 31500.0 0.57 0.6717 0.9817 3068542 PK04_095165 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C3Cc4ccccc4C3)C(=O)c5ccccc25)c6ccc(CO)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I08 compound treatment 1207400.0 25500.0 0.43 1215880.0 30500.0 0.55 0.6907 0.9922 3187345 PK04_095166 CC(C)CNC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I09 compound treatment 1206360.0 24500.0 0.41 1201400.0 16000.0 0.29 0.4939 0.9854 3067971 PK04_095167 CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I10 compound treatment 1199200.0 17300.0 0.29 1203280.0 17900.0 0.32 0.4331 0.9985 3068641 PK04_095168 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I11 compound treatment 1202680.0 20800.0 0.35 1195200.0 9840.0 0.18 0.3714 0.951 3187358 PK04_095169 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I12 compound treatment 1165600.0 -16300.0 -0.27 1173760.0 -11600.0 -0.21 -0.3406 -0.9914 3068653 PK04_095170 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I13 compound treatment 1186720.0 4830.0 0.08 1178960.0 -6400.0 -0.12 -0.0244 -0.1731 3067962 PK04_095171 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I14 compound treatment 1182440.0 554.0 0.01 1178160.0 -7200.0 -0.13 -0.0852 -0.655 3068606 PK04_095172 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I15 compound treatment 1173320.0 -8570.0 -0.14 1178920.0 -6440.0 -0.12 -0.1835 -0.9945 3068476 PK04_095173 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5cc(F)cc(c5)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I16 compound treatment 1175960.0 -5930.0 -0.1 1172520.0 -12800.0 -0.23 -0.2338 -0.9285 3186417 PK04_095174 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NC4CC4)c5ccc(cc5)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I17 compound treatment 1173160.0 -8730.0 -0.15 1170480.0 -14900.0 -0.27 -0.2929 -0.9592 3187268 PK04_095175 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2C5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I18 compound treatment 1178480.0 -3410.0 -0.06 1173680.0 -11700.0 -0.21 -0.1892 -0.8673 3187264 PK04_095176 CC(C)N1[C@H]([C@H](C(=O)NCC(F)(F)F)c2ccccc2C1=O)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I19 compound treatment 1145640.0 -36200.0 -0.61 1158360.0 -27000.0 -0.49 -0.7729 -0.994 3186499 PK04_095177 COCCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3OC)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I20 compound treatment 1154880.0 -27000.0 -0.45 1148920.0 -36400.0 -0.66 -0.7839 -0.9834 3068422 PK04_095178 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I21 mock treatment 1156000.0 -25900.0 -0.43 1160280.0 -25100.0 -0.45 -0.6259 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I22 mock treatment 1155960.0 -25900.0 -0.43 1167440.0 -17900.0 -0.32 -0.5351 -0.9894 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I23 compound treatment 1142400.0 -39500.0 -0.66 1151640.0 -33700.0 -0.61 -0.8969 -0.9991 3068550 PK04_095179 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(C(C)C)C(=O)c3ccccc23)c4ccc(CO)cc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 I24 compound treatment 1137760.0 -44100.0 -0.74 1144440.0 -40900.0 -0.74 -1.0435 -1.0 3187258 PK04_095180 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2C4Cc5ccccc5C4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J01 compound treatment 1237120.0 55200.0 0.92 1233720.0 48400.0 0.87 1.2696 0.9996 3187273 PK04_095181 CC(C)CNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J02 compound treatment 1235480.0 53600.0 0.9 1237760.0 52400.0 0.94 1.3017 0.9997 3186630 PK04_095182 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J03 compound treatment 1234080.0 52200.0 0.87 1226120.0 40800.0 0.73 1.1368 0.9963 3187353 PK04_095183 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(C(=O)c3ccccc32)c4ccc(C)cn4)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J04 compound treatment 1216480.0 34600.0 0.58 1222520.0 37200.0 0.67 0.8827 0.9974 3187588 PK04_095184 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)O)c3ccccc3C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J05 mock treatment 1211480.0 29600.0 0.5 1219160.0 33800.0 0.61 0.7807 0.9947 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J06 mock treatment 1209080.0 27200.0 0.46 1218560.0 33200.0 0.6 0.7447 0.9909 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J07 compound treatment 1212680.0 30800.0 0.52 1203080.0 17700.0 0.32 0.5901 0.9735 3186420 PK04_095185 OCc1ccc([C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c4ccc(cc4)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J08 compound treatment 1203200.0 21300.0 0.36 1209000.0 23600.0 0.43 0.5533 0.9961 3186722 PK04_095186 COCCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J09 compound treatment 1201000.0 19100.0 0.32 1195480.0 10100.0 0.18 0.355 0.9644 3186426 PK04_095187 CC(C)NC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J10 compound treatment 1195520.0 13600.0 0.23 1204640.0 19300.0 0.35 0.4069 0.9792 3186639 PK04_095188 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J11 compound treatment 1196120.0 14200.0 0.24 1188000.0 2640.0 0.05 0.202 0.8317 3187270 PK04_095189 CC(C)NC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J12 compound treatment 1154920.0 -27000.0 -0.45 1157440.0 -27900.0 -0.5 -0.6749 -0.9985 3067980 PK04_095190 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J13 compound treatment 1160480.0 -21400.0 -0.36 1134040.0 -51300.0 -0.92 -0.9072 -0.9148 3186421 PK04_095191 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J14 compound treatment 1178480.0 -3410.0 -0.06 1183160.0 -2200.0 -0.04 -0.0684 -0.9844 3068150 PK04_095192 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J15 compound treatment 1141080.0 -40800.0 -0.68 1167240.0 -18100.0 -0.33 -0.7138 -0.943 3068598 PK04_095193 CCCNC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J16 compound treatment 1185200.0 3310.0 0.06 1179880.0 -5480.0 -0.1 -0.0307 -0.2706 3068324 PK04_095194 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J17 compound treatment 1142440.0 -39400.0 -0.66 1144440.0 -40900.0 -0.74 -0.9882 -0.9985 3067973 PK04_095195 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCCN6CCOCC6)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J18 compound treatment 1159000.0 -22900.0 -0.38 1157440.0 -27900.0 -0.5 -0.6266 -0.9909 3068414 PK04_095196 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J19 compound treatment 1152880.0 -29000.0 -0.49 1153840.0 -31500.0 -0.57 -0.7449 -0.9969 3187085 PK04_095197 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J20 compound treatment 1152760.0 -29100.0 -0.49 1150440.0 -34900.0 -0.63 -0.7896 -0.992 3186884 PK04_095198 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J21 mock treatment 1133760.0 -48100.0 -0.81 1148000.0 -37400.0 -0.67 -1.0455 -0.996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J22 mock treatment 1148200.0 -33700.0 -0.56 1147880.0 -37500.0 -0.68 -0.8762 -0.996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J23 compound treatment 1135560.0 -46300.0 -0.78 1129600.0 -55800.0 -1.0 -1.2586 -0.9918 3187082 PK04_095199 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 J24 compound treatment 1143720.0 -38200.0 -0.64 1149960.0 -35400.0 -0.64 -0.9027 -1.0 3068227 PK04_095200 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K01 compound treatment 1226200.0 44300.0 0.74 1232280.0 46900.0 0.85 1.1221 0.9979 3187514 PK04_095201 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NC6CC6)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K02 compound treatment 1234000.0 52100.0 0.87 1243760.0 58400.0 1.05 1.3606 0.9957 3187168 PK04_095202 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccc(OC(F)(F)F)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K03 compound treatment 1221880.0 40000.0 0.67 1225560.0 40200.0 0.72 0.9853 0.9992 3068143 PK04_095203 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NC5CC5)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K04 compound treatment 1206920.0 25000.0 0.42 1218360.0 33000.0 0.59 0.7166 0.9853 3187275 PK04_095204 CN(C)CCCNC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K05 compound treatment 1214880.0 33000.0 0.55 1223520.0 38200.0 0.69 0.8765 0.9941 3187271 PK04_095205 CN(C)CCCNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K06 compound treatment 1226920.0 45000.0 0.75 1217040.0 31700.0 0.57 0.9364 0.9906 3186561 PK04_095206 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K07 mock treatment 1209720.0 27800.0 0.47 1212840.0 27500.0 0.5 0.6794 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K08 mock treatment 1206760.0 24900.0 0.42 1206640.0 21300.0 0.38 0.5654 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K09 compound treatment 1215880.0 34000.0 0.57 1214600.0 29200.0 0.53 0.7747 0.9993 3068519 PK04_095207 CN(C)CCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K10 compound treatment 1204720.0 22800.0 0.38 1200320.0 15000.0 0.27 0.4607 0.9854 3068466 PK04_095208 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccccc4C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K11 compound treatment 1187640.0 5750.0 0.1 1183440.0 -1920.0 -0.03 0.0436 0.4257 3068556 PK04_095209 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2C5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K12 compound treatment 1142160.0 -39700.0 -0.66 1154040.0 -31300.0 -0.56 -0.8692 -0.9967 3067978 PK04_095210 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)O)c6ccc(cc6)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K13 compound treatment 1159920.0 -22000.0 -0.37 1155040.0 -30300.0 -0.55 -0.6463 -0.9814 3068499 PK04_095211 COCCCNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K14 compound treatment 1135960.0 -45900.0 -0.77 1171880.0 -13500.0 -0.24 -0.7152 -0.8874 3068588 PK04_095212 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2CC5(CC6CC7CC(C6)C5)C7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K15 mock treatment 1186960.0 5070.0 0.08 1179640.0 -5720.0 -0.1 -0.0129 -0.0965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K16 mock treatment 1176400.0 -5490.0 -0.09 1179520.0 -5840.0 -0.11 -0.1394 -0.9977 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K17 compound treatment 1154360.0 -27500.0 -0.46 1166200.0 -19200.0 -0.35 -0.5699 -0.9899 3068009 PK04_095213 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K18 compound treatment 1159040.0 -22800.0 -0.38 1156040.0 -29300.0 -0.53 -0.6439 -0.9874 3186498 PK04_095214 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCCCN(C)C)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K19 compound treatment 1157280.0 -24600.0 -0.41 1163880.0 -21500.0 -0.39 -0.5649 -0.9995 3068472 PK04_095215 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccccc4Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K20 compound treatment 1154200.0 -27700.0 -0.46 1155040.0 -30300.0 -0.55 -0.7139 -0.9966 3187259 PK04_095216 COCCCNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K21 compound treatment 1155520.0 -26400.0 -0.44 1156760.0 -28600.0 -0.52 -0.6764 -0.997 3187078 PK04_095217 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccccc5C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K22 compound treatment 1157240.0 -24600.0 -0.41 1156560.0 -28800.0 -0.52 -0.6586 -0.9935 3068508 PK04_095218 COc1ccccc1CN2[C@H]([C@H](C(=O)NC3CC3)c4ccccc4C2=O)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K23 mock treatment 1143680.0 -38200.0 -0.64 1156280.0 -29100.0 -0.52 -0.8226 -0.9951 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 K24 mock treatment 1134640.0 -47200.0 -0.79 1135600.0 -49800.0 -0.9 -1.1931 -0.998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L01 compound treatment 1209040.0 27200.0 0.45 1217480.0 32100.0 0.58 0.7305 0.9928 3187175 PK04_095219 COc1ccccc1CN2[C@H]([C@H](C(=O)NCCCN(C)C)c3ccccc3C2=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L02 compound treatment 1234280.0 52400.0 0.88 1223440.0 38100.0 0.69 1.1051 0.9926 3186714 PK04_095220 CC(C)NC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L03 compound treatment 1225240.0 43400.0 0.73 1222200.0 36800.0 0.66 0.9823 0.999 3067967 PK04_095221 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCc3ccccc3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L04 compound treatment 1213040.0 31200.0 0.52 1218520.0 33200.0 0.6 0.7911 0.9977 3186429 PK04_095222 CC(C)CN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L05 compound treatment 1215360.0 33500.0 0.56 1206040.0 20700.0 0.37 0.6595 0.9804 3068540 PK04_095223 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2C5Cc6ccccc6C5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L06 compound treatment 1212280.0 30400.0 0.51 1208440.0 23100.0 0.42 0.6536 0.995 3186551 PK04_095224 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L07 mock treatment 1224800.0 42900.0 0.72 1201720.0 16400.0 0.29 0.7162 0.9226 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L08 mock treatment 1187800.0 5910.0 0.1 1197360.0 12000.0 0.22 0.2228 0.9373 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L09 compound treatment 1202880.0 21000.0 0.35 1188800.0 3440.0 0.06 0.2922 0.8191 3187518 PK04_095225 CN(C)CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L10 compound treatment 1180320.0 -1570.0 -0.03 1189760.0 4400.0 0.08 0.0375 0.4491 3068144 PK04_095226 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCc5ccccc5)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L11 compound treatment 1181160.0 -726.0 -0.01 1186320.0 956.0 0.02 0.0036 0.1699 3187076 PK04_095227 COCCCNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L12 compound treatment 1188600.0 6710.0 0.11 1192120.0 6760.0 0.12 0.1655 0.9992 3068313 PK04_095228 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L13 compound treatment 1135680.0 -46200.0 -0.77 1134920.0 -50400.0 -0.91 -1.1894 -0.9968 3187347 PK04_095229 COc1ccc(CCNC(=O)[C@]2(C)[C@@H](N(C(C)C)C(=O)c3ccccc32)c4ccc(CO)cc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L14 compound treatment 1171400.0 -10500.0 -0.18 1167640.0 -17700.0 -0.32 -0.3499 -0.9602 3068194 PK04_095230 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CC(C)C)C4=O)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L15 mock treatment 1160640.0 -21200.0 -0.36 1166200.0 -19200.0 -0.35 -0.4956 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L16 mock treatment 1151720.0 -30200.0 -0.5 1169120.0 -16200.0 -0.29 -0.5639 -0.9664 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L17 compound treatment 1144960.0 -36900.0 -0.62 1149200.0 -36200.0 -0.65 -0.8977 -0.9996 3068510 PK04_095231 COc1ccccc1CN2[C@H]([C@H](C(=O)NCc3ccccc3)c4ccccc4C2=O)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L18 compound treatment 1159000.0 -22900.0 -0.38 1172360.0 -13000.0 -0.23 -0.4365 -0.9722 3068263 PK04_095232 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C(C)C)[C@@H]2c3ccc(CO)cc3I)Sc4ccc(C)cc4)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L19 compound treatment 1149400.0 -32500.0 -0.54 1150360.0 -35000.0 -0.63 -0.8304 -0.9973 3067958 PK04_095233 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCCN4CCOCC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L20 compound treatment 1144680.0 -37200.0 -0.62 1149040.0 -36300.0 -0.65 -0.903 -0.9997 3068403 PK04_095234 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L21 compound treatment 1137040.0 -44800.0 -0.75 1138400.0 -47000.0 -0.85 -1.129 -0.9982 3187163 PK04_095235 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3cc(F)cc(c3)C(F)(F)F)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L22 compound treatment 1137240.0 -44600.0 -0.75 1148160.0 -37200.0 -0.67 -1.0023 -0.9985 3186433 PK04_095236 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(CC(F)(F)F)c2c1)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L23 mock treatment 1142560.0 -39300.0 -0.66 1146800.0 -38600.0 -0.69 -0.9567 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 L24 mock treatment 1133400.0 -48500.0 -0.81 1151360.0 -34000.0 -0.61 -1.007 -0.9904 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M01 compound treatment 1229640.0 47800.0 0.8 1233520.0 48200.0 0.87 1.1786 0.9992 3187444 PK04_095237 CC(C)CNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M02 compound treatment 1236240.0 54400.0 0.91 1239720.0 54400.0 0.98 1.3357 0.9993 3068593 PK04_095238 CC(C)N1[C@@H](c2ccc(CO)cc2)[C@@](C)(C(=O)NC3CC3)c4ccccc4C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M03 compound treatment 1241960.0 60100.0 1.01 1243880.0 58500.0 1.05 1.4564 0.9997 3187441 PK04_095239 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M04 compound treatment 1230680.0 48800.0 0.82 1230840.0 45500.0 0.82 1.1567 1.0 3068649 PK04_095240 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M05 compound treatment 1208760.0 26900.0 0.45 1207960.0 22600.0 0.41 0.6059 0.9988 3068152 PK04_095241 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M06 compound treatment 1218080.0 36200.0 0.61 1219000.0 33600.0 0.61 0.8568 1.0 3068655 PK04_095242 C[C@]1([C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M07 compound treatment 1218080.0 36200.0 0.61 1229360.0 44000.0 0.79 0.9888 0.9912 3068005 PK04_095243 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M08 compound treatment 1207120.0 25200.0 0.42 1212560.0 27200.0 0.49 0.6451 0.9973 3187084 PK04_095244 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5ccccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M09 mock treatment 1209280.0 27400.0 0.46 1204600.0 19200.0 0.35 0.5692 0.9905 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M10 mock treatment 1191720.0 9830.0 0.16 1195040.0 9680.0 0.17 0.2396 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M11 compound treatment 1180440.0 -1450.0 -0.02 1178840.0 -6520.0 -0.12 -0.1002 -0.8352 3186422 PK04_095245 CCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5I)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M12 compound treatment 1194760.0 12900.0 0.22 1202560.0 17200.0 0.31 0.3714 0.9842 3068142 PK04_095246 CN(C)CCCNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(C3CCCCC3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M13 mock treatment 1148720.0 -33200.0 -0.56 1149840.0 -35500.0 -0.64 -0.845 -0.9975 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M14 mock treatment 1181480.0 -406.0 -0.01 1175040.0 -10300.0 -0.19 -0.1363 -0.7325 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M15 compound treatment 1164800.0 -17100.0 -0.29 1166640.0 -18700.0 -0.34 -0.4407 -0.9966 3068557 PK04_095247 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2C5CCCCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M16 compound treatment 1164240.0 -17600.0 -0.3 1166280.0 -19100.0 -0.34 -0.4519 -0.9971 3187170 PK04_095248 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2OC)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M17 compound treatment 1146120.0 -35800.0 -0.6 1160960.0 -24400.0 -0.44 -0.7341 -0.9885 3187431 PK04_095249 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M18 compound treatment 1166840.0 -15000.0 -0.25 1170120.0 -15200.0 -0.27 -0.3723 -0.9991 3187074 PK04_095250 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2Cc5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M19 compound treatment 1155800.0 -26100.0 -0.44 1148080.0 -37300.0 -0.67 -0.7837 -0.9782 3068552 PK04_095251 CC(C)NC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M20 compound treatment 1138200.0 -43700.0 -0.73 1146520.0 -38800.0 -0.7 -1.0118 -0.9998 3068014 PK04_095252 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)O)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M21 compound treatment 1136840.0 -45000.0 -0.75 1142680.0 -42700.0 -0.77 -1.0768 -1.0 3187086 PK04_095253 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M22 compound treatment 1144960.0 -36900.0 -0.62 1135680.0 -49700.0 -0.9 -1.0699 -0.9836 3187428 PK04_095254 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NC5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M23 compound treatment 1125560.0 -56300.0 -0.94 1148840.0 -36500.0 -0.66 -1.1318 -0.9846 3187081 PK04_095255 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 M24 compound treatment 1133240.0 -48600.0 -0.81 1127000.0 -58400.0 -1.05 -1.3192 -0.992 3068003 PK04_095256 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N01 compound treatment 1229080.0 47200.0 0.79 1210800.0 25400.0 0.46 0.8825 0.9665 3187360 PK04_095257 C[C@]1([C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N02 compound treatment 1220160.0 38300.0 0.64 1229040.0 43700.0 0.79 1.0093 0.9948 3068231 PK04_095258 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N03 compound treatment 1209280.0 27400.0 0.46 1212320.0 27000.0 0.49 0.6676 0.9996 3068544 PK04_095259 CC(C)NC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N04 compound treatment 1180240.0 -1650.0 -0.03 1174200.0 -11200.0 -0.2 -0.1617 -0.7965 3187527 PK04_095260 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)O)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N05 compound treatment 1200560.0 18700.0 0.31 1200000.0 14600.0 0.26 0.4074 0.9964 3187260 PK04_095261 CCCNC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N06 compound treatment 1198320.0 16400.0 0.28 1197760.0 12400.0 0.22 0.3524 0.9947 3186724 PK04_095262 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N07 compound treatment 1202320.0 20400.0 0.34 1188640.0 3280.0 0.06 0.2835 0.8171 3068501 PK04_095263 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N08 compound treatment 1176640.0 -5250.0 -0.09 1187280.0 1920.0 0.03 -0.0377 -0.3994 3186871 PK04_095264 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N09 mock treatment 1182440.0 554.0 0.01 1185880.0 516.0 0.01 0.0131 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N10 mock treatment 1181720.0 -166.0 0.0 1185960.0 596.0 0.01 0.0056 0.507 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N11 compound treatment 1167560.0 -14300.0 -0.24 1170200.0 -15200.0 -0.27 -0.3627 -0.9979 3187070 PK04_095265 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N12 compound treatment 1156080.0 -25800.0 -0.43 1159920.0 -25400.0 -0.46 -0.6295 -0.9996 3186804 PK04_095266 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N13 mock treatment 1151600.0 -30300.0 -0.51 1152160.0 -33200.0 -0.6 -0.7814 -0.9966 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N14 mock treatment 1167320.0 -14600.0 -0.24 1176880.0 -8480.0 -0.15 -0.2805 -0.9747 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N15 compound treatment 1128040.0 -53800.0 -0.9 1116920.0 -68400.0 -1.23 -1.5092 -0.9881 3186424 PK04_095267 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCCN6CCOCC6)c7ccc(cc7)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N16 compound treatment 1153520.0 -28400.0 -0.47 1159400.0 -26000.0 -0.47 -0.6664 -1.0 3068226 PK04_095268 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N17 compound treatment 1131960.0 -49900.0 -0.84 1140520.0 -44800.0 -0.81 -1.1621 -0.9999 3068455 PK04_095269 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N18 compound treatment 1150480.0 -31400.0 -0.53 1159520.0 -25800.0 -0.47 -0.7009 -0.9982 3068137 PK04_095270 CN(C)CCCN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N19 compound treatment 1132400.0 -49500.0 -0.83 1139320.0 -46000.0 -0.83 -1.1722 -1.0 3068647 PK04_095271 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N20 compound treatment 1110520.0 -71400.0 -1.19 1125120.0 -60200.0 -1.09 -1.612 -0.9989 3186492 PK04_095272 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N21 compound treatment 1112280.0 -69600.0 -1.16 1113200.0 -72200.0 -1.3 -1.743 -0.9985 3067959 PK04_095273 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N22 compound treatment 1130560.0 -51300.0 -0.86 1152040.0 -33300.0 -0.6 -1.0319 -0.9847 3187526 PK04_095274 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)O)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N23 compound treatment 1116160.0 -65700.0 -1.1 1125560.0 -59800.0 -1.08 -1.5397 -0.9999 3068468 PK04_095275 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 N24 compound treatment 1126760.0 -55100.0 -0.92 1147680.0 -37700.0 -0.68 -1.1324 -0.9886 3068222 PK04_095276 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O01 compound treatment 1222480.0 40600.0 0.68 1217680.0 32300.0 0.58 0.8921 0.9971 3068590 PK04_095277 CC(C)NC(=O)[C@H]1[C@@H](N(CC2(CC3CC4CC(C3)C2)C4)C(=O)c5ccccc15)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O02 compound treatment 1188480.0 6590.0 0.11 1193640.0 8280.0 0.15 0.1835 0.989 3067977 PK04_095278 COCCCNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O03 compound treatment 1209280.0 27400.0 0.46 1223200.0 37800.0 0.68 0.8062 0.9814 3068512 PK04_095279 COc1ccccc1CN2[C@H]([C@H](C(=O)NCC(F)(F)F)c3ccccc3C2=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O04 compound treatment 1225720.0 43800.0 0.73 1227440.0 42100.0 0.76 1.0547 0.9999 3068637 PK04_095280 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O05 compound treatment 1218120.0 36200.0 0.61 1217600.0 32200.0 0.58 0.8394 0.9998 3068459 PK04_095281 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2Cc4cc(cc(c4)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O06 compound treatment 1191560.0 9670.0 0.16 1190960.0 5600.0 0.1 0.1858 0.974 3187520 PK04_095282 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O07 compound treatment 1178680.0 -3210.0 -0.05 1189680.0 4320.0 0.08 0.017 0.1804 3186989 PK04_095283 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O08 compound treatment 1200840.0 19000.0 0.32 1213640.0 28300.0 0.51 0.5845 0.974 3187364 PK04_095284 C[C@]1([C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCc5ccccc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O09 compound treatment 1177720.0 -4170.0 -0.07 1176200.0 -9160.0 -0.17 -0.1661 -0.9265 3068604 PK04_095285 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O10 compound treatment 1172240.0 -9650.0 -0.16 1181880.0 -3480.0 -0.06 -0.1585 -0.9153 3187362 PK04_095286 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O11 mock treatment 1158640.0 -23200.0 -0.39 1166840.0 -18500.0 -0.33 -0.5111 -0.9971 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O12 mock treatment 1180000.0 -1890.0 -0.03 1179560.0 -5800.0 -0.1 -0.0963 -0.8813 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O13 compound treatment 1181840.0 -46.3 0.0 1180840.0 -4520.0 -0.08 -0.0582 -0.7138 3068644 PK04_095287 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O14 compound treatment 1155400.0 -26500.0 -0.44 1151480.0 -33900.0 -0.61 -0.7451 -0.9876 3068464 PK04_095288 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5ccccc5C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O15 compound treatment 1152560.0 -29300.0 -0.49 1153240.0 -32100.0 -0.58 -0.7563 -0.9966 3187516 PK04_095289 OCc1ccc(cc1)[C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCc6ccccc6)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O16 compound treatment 1139240.0 -42600.0 -0.71 1136440.0 -48900.0 -0.88 -1.1279 -0.9945 3187164 PK04_095290 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5cc(F)cc(c5)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O17 compound treatment 1155200.0 -26700.0 -0.45 1158120.0 -27200.0 -0.49 -0.6629 -0.9989 3187177 PK04_095291 CC(C)CNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O18 compound treatment 1150440.0 -31400.0 -0.53 1149800.0 -35600.0 -0.64 -0.8252 -0.9952 3068546 PK04_095292 CN(C)CCCNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O19 compound treatment 1141400.0 -40500.0 -0.68 1156840.0 -28500.0 -0.51 -0.8425 -0.9907 3187256 PK04_095293 CC(C)CNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O20 compound treatment 1129760.0 -52100.0 -0.87 1134400.0 -51000.0 -0.92 -1.2661 -0.9997 3187088 PK04_095294 COCCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2Cl)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O21 compound treatment 1132600.0 -49300.0 -0.82 1135600.0 -49800.0 -0.9 -1.2172 -0.9991 3186494 PK04_095295 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCC(C)C)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O22 compound treatment 1124120.0 -57800.0 -0.97 1130320.0 -55000.0 -0.99 -1.3848 -0.9999 3187161 PK04_095296 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O23 compound treatment 1118760.0 -63100.0 -1.06 1113320.0 -72000.0 -1.3 -1.6648 -0.9948 3187267 PK04_095297 CC(C)CNC(=O)[C@H]1[C@@H](N(C2CCCCC2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 O24 compound treatment 1125720.0 -56200.0 -0.94 1139800.0 -45600.0 -0.82 -1.2451 -0.9977 3068502 PK04_095298 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P01 compound treatment 1220360.0 38500.0 0.64 1225920.0 40600.0 0.73 0.9719 0.998 3068591 PK04_095299 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2CC4(CC5CC6CC(C5)C4)C6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P02 compound treatment 1204120.0 22200.0 0.37 1209320.0 24000.0 0.43 0.5683 0.9973 3187521 PK04_095300 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P03 compound treatment 1209760.0 27900.0 0.47 1205120.0 19800.0 0.36 0.5815 0.9911 3186990 PK04_095301 COc1ccc(CCNC(=O)[C@H]2[C@@H](N(Cc3ccccc3)C(=O)c4ccccc24)c5ccc(CO)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P04 compound treatment 1196480.0 14600.0 0.24 1192400.0 7040.0 0.13 0.2623 0.9534 3186985 PK04_095302 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P05 compound treatment 1173120.0 -8770.0 -0.15 1173800.0 -11600.0 -0.21 -0.2511 -0.9853 3067579 PK04_095303 OCc1ccc([C@H]2N(CC3(CC4CC5CC(C4)C3)C5)C(=O)C[C@@]2(C(=O)NCC(F)(F)F)c6ccc(cc6)[N+](=O)[O-])c(I)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P06 compound treatment 1170880.0 -11000.0 -0.18 1189160.0 3800.0 0.07 -0.0819 -0.4168 3186975 PK04_095304 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P07 compound treatment 1166920.0 -15000.0 -0.25 1183040.0 -2320.0 -0.04 -0.2067 -0.814 3068548 PK04_095305 CC(C)CNC(=O)[C@H]1[C@@H](N(C(C)C)C(=O)c2ccccc12)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P08 compound treatment 1151600.0 -30300.0 -0.51 1162600.0 -22800.0 -0.41 -0.6484 -0.9945 3067563 PK04_095306 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(CCN5CCOCC5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P09 compound treatment 1169000.0 -12900.0 -0.22 1178680.0 -6680.0 -0.12 -0.2376 -0.9621 3067961 PK04_095307 OCc1ccc(cc1)[C@H]2N(C3CCCCC3)C(=O)C[C@@]2(C(=O)NCc4ccccc4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P10 compound treatment 1162640.0 -19200.0 -0.32 1168480.0 -16900.0 -0.3 -0.4429 -0.9996 3068015 PK04_095308 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P11 mock treatment 1155240.0 -26600.0 -0.45 1156920.0 -28400.0 -0.51 -0.6777 -0.9976 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P12 mock treatment 1167200.0 -14700.0 -0.25 1181160.0 -4200.0 -0.08 -0.2273 -0.884 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P13 compound treatment 1137200.0 -44700.0 -0.75 1150040.0 -35300.0 -0.64 -0.9788 -0.9968 3187510 PK04_095309 CC(C)NC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P14 compound treatment 1137040.0 -44800.0 -0.75 1143960.0 -41400.0 -0.75 -1.0582 -1.0 3186495 PK04_095310 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NCCN5CCOCC5)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P15 compound treatment 1143760.0 -38100.0 -0.64 1135280.0 -50100.0 -0.9 -1.0892 -0.9856 3187437 PK04_095311 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P16 compound treatment 1138200.0 -43700.0 -0.73 1141280.0 -44100.0 -0.79 -1.0786 -0.9991 3186625 PK04_095312 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(C(C)C)C4=O)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P17 compound treatment 1135680.0 -46200.0 -0.77 1137120.0 -48200.0 -0.87 -1.1614 -0.9983 3068541 PK04_095313 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCCN3CCOCC3)c4ccccc4C(=O)N2C5Cc6ccccc6C5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P18 compound treatment 1134320.0 -47600.0 -0.8 1129160.0 -56200.0 -1.01 -1.2789 -0.9929 3186878 PK04_095314 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NC6CC6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P19 compound treatment 1116600.0 -65300.0 -1.09 1119640.0 -65700.0 -1.18 -1.6099 -0.9992 3187513 PK04_095315 CC(C)CNC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P20 compound treatment 1131720.0 -50200.0 -0.84 1133320.0 -52000.0 -0.94 -1.2567 -0.9985 3068271 PK04_095316 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCc6ccccc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P21 compound treatment 1090200.0 -91700.0 -1.53 1093000.0 -92400.0 -1.66 -2.2617 -0.9992 3068008 PK04_095317 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P22 compound treatment 1126760.0 -55100.0 -0.92 1134640.0 -50700.0 -0.91 -1.2985 -1.0 3068262 PK04_095318 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P23 compound treatment 1128000.0 -53900.0 -0.9 1122480.0 -62900.0 -1.13 -1.4388 -0.9936 3068469 PK04_095319 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccccc5Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2095 P24 compound treatment 1148480.0 -33400.0 -0.56 1150560.0 -34800.0 -0.63 -0.8387 -0.9984 3186794 PK04_095320 CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A01 compound treatment 1228560.0 49100.0 0.82 1201320.0 46700.0 0.84 1.1765 0.9999 3186490 PK04_096001 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A02 compound treatment 1231600.0 52100.0 0.87 1192000.0 37400.0 0.67 1.0937 0.9919 3186641 PK04_096002 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A03 compound treatment 1221800.0 42300.0 0.71 1216680.0 62100.0 1.12 1.2922 0.9757 3068261 PK04_096003 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NC4CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A04 compound treatment 1223920.0 44500.0 0.74 1203000.0 48400.0 0.87 1.143 0.9969 3186971 PK04_096004 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A05 compound treatment 1214520.0 35100.0 0.59 1194600.0 40000.0 0.72 0.9247 0.9948 3186883 PK04_096005 COCCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A06 compound treatment 1234080.0 54600.0 0.91 1209720.0 55100.0 0.99 1.3488 0.9991 3068309 PK04_096006 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A07 compound treatment 1211040.0 31600.0 0.53 1188440.0 33900.0 0.61 0.8051 0.9974 3186716 PK04_096007 COCCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2I)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A08 compound treatment 1196240.0 16800.0 0.28 1180520.0 25900.0 0.47 0.529 0.9703 3068367 PK04_096008 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)Sc6ccc(C)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A09 compound treatment 1198600.0 19100.0 0.32 1185480.0 30900.0 0.56 0.6202 0.9655 3068224 PK04_096009 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A10 compound treatment 1201000.0 21500.0 0.36 1185000.0 30400.0 0.55 0.6424 0.9793 3186633 PK04_096010 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5C(F)(F)F)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A11 compound treatment 1199320.0 19900.0 0.33 1176840.0 22300.0 0.4 0.5186 0.9956 3186986 PK04_096011 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A12 compound treatment 1203080.0 23600.0 0.4 1191160.0 36600.0 0.66 0.7455 0.9701 3186640 PK04_096012 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A13 mock treatment 1190840.0 11400.0 0.19 1180920.0 26300.0 0.47 0.4702 0.9195 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A14 mock treatment 1195320.0 15900.0 0.27 1186040.0 31500.0 0.57 0.5885 0.9402 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A15 compound treatment 1183000.0 3540.0 0.06 1165960.0 11400.0 0.21 0.1869 0.8754 3186881 PK04_096013 CC(C)NC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A16 compound treatment 1187720.0 8260.0 0.14 1167480.0 12900.0 0.23 0.2621 0.9691 3186790 PK04_096014 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A17 compound treatment 1176080.0 -3380.0 -0.06 1159360.0 4780.0 0.09 0.0209 0.2027 3186485 PK04_096015 CC(C)CN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A18 compound treatment 1192640.0 13200.0 0.22 1173760.0 19200.0 0.35 0.4003 0.9764 3186802 PK04_096016 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A19 compound treatment 1165040.0 -14400.0 -0.24 1144640.0 -9940.0 -0.18 -0.2973 -0.9892 3068405 PK04_096017 CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A20 compound treatment 1172960.0 -6500.0 -0.11 1154120.0 -456.0 -0.01 -0.0828 -0.7584 3068141 PK04_096018 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A21 compound treatment 1160960.0 -18500.0 -0.31 1142160.0 -12400.0 -0.22 -0.3771 -0.9873 3186624 PK04_096019 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5OC)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A22 compound treatment 1161520.0 -17900.0 -0.3 1149440.0 -5140.0 -0.09 -0.2778 -0.884 3068200 PK04_096020 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CCCN(C)C)C4=O)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A23 compound treatment 1169320.0 -10100.0 -0.17 1147960.0 -6620.0 -0.12 -0.2043 -0.985 3068358 PK04_096021 CC(C)CNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 A24 compound treatment 1174640.0 -4820.0 -0.08 1154120.0 -456.0 -0.01 -0.0629 -0.7751 3068371 PK04_096022 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B01 compound treatment 1241840.0 62400.0 1.04 1220800.0 66200.0 1.19 1.5818 0.9978 3187511 PK04_096023 CC(C)N1[C@H](c2ccc(CO)cc2)[C@](CC1=O)(C(=O)NCC(F)(F)F)c3ccc(cc3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B02 compound treatment 1223840.0 44400.0 0.74 1203160.0 48600.0 0.88 1.1441 0.9967 3187030 PK04_096024 OCCCc1cc[n+](Cc2cccc(OC(F)(F)F)c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B03 compound treatment 1224000.0 44500.0 0.75 1203440.0 48900.0 0.88 1.1495 0.9966 3187169 PK04_096025 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B04 compound treatment 1230320.0 50900.0 0.85 1213120.0 58500.0 1.05 1.3476 0.9943 3068853 PK04_096026 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B05 compound treatment 1218960.0 39500.0 0.66 1207160.0 52600.0 0.95 1.1373 0.9845 3068457 PK04_096027 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCc3ccccc3)c4ccccc4C(=O)N2Cc5cc(cc(c5)C(F)(F)F)C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B06 compound treatment 1201160.0 21700.0 0.36 1180800.0 26200.0 0.47 0.5908 0.9915 3068854 PK04_096028 C[n+]1ccc2ccc(O)cc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B07 compound treatment 1212960.0 33500.0 0.56 1198200.0 43600.0 0.79 0.9521 0.9863 3187352 PK04_096029 Cc1ccc(nc1)N2[C@@H](c3ccc(CO)cc3)[C@@](C)(C(=O)NCCN4CCOCC4)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B08 compound treatment 1207360.0 27900.0 0.47 1192040.0 37500.0 0.67 0.8074 0.9838 3187112 PK04_096030 COc1cc2CC[N+](=Cc2cc1O)Cc3cc4OCOc4cc3Br 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B09 compound treatment 1202440.0 23000.0 0.38 1167880.0 13300.0 0.24 0.4414 0.9741 3068505 PK04_096031 CC(C)NC(=O)[C@H]1[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B10 compound treatment 1190480.0 11000.0 0.18 1163680.0 9100.0 0.16 0.2463 0.9983 3068855 PK04_096032 C[n+]1ccc(CCCO)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B11 compound treatment 1201440.0 22000.0 0.37 1190520.0 35900.0 0.65 0.718 0.9641 3068374 PK04_096033 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B12 compound treatment 1179320.0 -144.0 0.0 1160320.0 5740.0 0.1 0.0715 0.6905 3187113 PK04_096034 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(C=C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B13 mock treatment 1190880.0 11400.0 0.19 1166080.0 11500.0 0.21 0.2816 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B14 mock treatment 1198160.0 18700.0 0.31 1175280.0 20700.0 0.37 0.485 0.9962 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B15 compound treatment 1188240.0 8780.0 0.15 1161760.0 7180.0 0.13 0.1954 0.998 3187255 PK04_096035 COCCCNC(=O)[C@H]1[C@@H](N(C(=O)c2ccccc12)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B16 compound treatment 1169760.0 -9700.0 -0.16 1145880.0 -8700.0 -0.16 -0.2256 -0.9998 3068856 PK04_096036 Oc1ccc2cc[n+](Cc3sc4ccccc4c3Cl)cc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B17 compound treatment 1167080.0 -12400.0 -0.21 1151720.0 -2860.0 -0.05 -0.1829 -0.8567 3068608 PK04_096037 CC(C)NC(=O)[C@]1(C)[C@@H](N(Cc2ccc(OC(F)(F)F)cc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B18 compound treatment 1177520.0 -1940.0 -0.03 1149720.0 -4860.0 -0.09 -0.0849 -0.9092 3187114 PK04_096038 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(C5CC5)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B19 compound treatment 1149480.0 -30000.0 -0.5 1116840.0 -37700.0 -0.68 -0.8356 -0.9888 3187171 PK04_096039 COc1ccccc1CN2[C@H]([C@H](C(=O)NCC(C)C)c3ccccc3C2=O)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B20 compound treatment 1141480.0 -38000.0 -0.64 1121720.0 -32900.0 -0.59 -0.8681 -0.9994 3068857 PK04_096040 OCCCc1cc[n+](Cc2ccc(o2)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B21 compound treatment 1134840.0 -44600.0 -0.75 1119480.0 -35100.0 -0.63 -0.9752 -0.9966 3068424 PK04_096041 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B22 compound treatment 1161160.0 -18300.0 -0.31 1132440.0 -22100.0 -0.4 -0.4986 -0.9915 3187115 PK04_096042 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B23 compound treatment 1146280.0 -33200.0 -0.56 1120200.0 -34400.0 -0.62 -0.8306 -0.9985 3187072 PK04_096043 CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 B24 compound treatment 1147360.0 -32100.0 -0.54 1119840.0 -34700.0 -0.63 -0.8224 -0.9971 3187116 PK04_096044 COC(=O)C1=CN(C)C(C=C(C=C1C(=O)OC)c2ccc(CO)cc2)c3cccs3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C01 compound treatment 1215160.0 35700.0 0.6 1187880.0 33300.0 0.6 0.8467 1.0 3068218 PK04_096045 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C02 compound treatment 1228080.0 48600.0 0.81 1196520.0 41900.0 0.76 1.1096 0.9993 3186566 PK04_096046 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C03 compound treatment 1196880.0 17400.0 0.29 1170280.0 15700.0 0.28 0.4062 0.9999 3186549 PK04_096047 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C04 compound treatment 1214280.0 34800.0 0.58 1187440.0 32900.0 0.59 0.8307 1.0 3186726 PK04_096048 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C05 compound treatment 1202680.0 23200.0 0.39 1181840.0 27300.0 0.49 0.6221 0.9933 3186792 PK04_096049 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C06 compound treatment 1194160.0 14700.0 0.25 1183480.0 28900.0 0.52 0.5421 0.9413 3186987 PK04_096050 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C07 compound treatment 1189000.0 9540.0 0.16 1167080.0 12500.0 0.23 0.2721 0.9857 3068275 PK04_096051 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C08 compound treatment 1193240.0 13800.0 0.23 1163480.0 8900.0 0.16 0.2765 0.9843 3186560 PK04_096052 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C09 compound treatment 1166400.0 -13100.0 -0.22 1162680.0 8100.0 0.15 -0.0513 -0.1953 3068147 PK04_096053 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C10 compound treatment 1189400.0 9940.0 0.17 1154040.0 -536.0 -0.01 0.1107 0.6649 3186976 PK04_096054 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C11 mock treatment 1190200.0 10700.0 0.18 1168280.0 13700.0 0.25 0.3016 0.9878 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C12 mock treatment 1195000.0 15500.0 0.26 1168520.0 13900.0 0.25 0.3615 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C13 compound treatment 1147880.0 -31600.0 -0.53 1122280.0 -32300.0 -0.58 -0.7852 -0.9988 3186974 PK04_096055 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C14 compound treatment 1174040.0 -5420.0 -0.09 1150440.0 -4140.0 -0.07 -0.1169 -0.9952 3186876 PK04_096056 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCCN(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C15 mock treatment 1163680.0 -15800.0 -0.26 1140480.0 -14100.0 -0.25 -0.3664 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C16 mock treatment 1178320.0 -1140.0 -0.02 1143920.0 -10700.0 -0.19 -0.1493 -0.7738 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C17 compound treatment 1186400.0 6940.0 0.12 1148160.0 -6420.0 -0.12 3.0E-4 0.002 3186553 PK04_096057 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C18 compound treatment 1171960.0 -7500.0 -0.13 1137880.0 -16700.0 -0.3 -0.3015 -0.9249 3186634 PK04_096058 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C19 compound treatment 1148960.0 -30500.0 -0.51 1132200.0 -22400.0 -0.4 -0.646 -0.9932 3186638 PK04_096059 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(Cc5ccccc5)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C20 compound treatment 1159040.0 -20400.0 -0.34 1134600.0 -20000.0 -0.36 -0.4962 -0.9997 3068219 PK04_096060 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C21 compound treatment 1142480.0 -37000.0 -0.62 1126640.0 -27900.0 -0.5 -0.7935 -0.9947 3068151 PK04_096061 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C22 compound treatment 1151000.0 -28500.0 -0.48 1131040.0 -23500.0 -0.42 -0.6367 -0.9983 3068158 PK04_096062 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CC(F)(F)F)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C23 compound treatment 1157240.0 -22200.0 -0.37 1135760.0 -18800.0 -0.34 -0.5027 -0.9989 3186800 PK04_096063 COCCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 C24 compound treatment 1162360.0 -17100.0 -0.29 1141560.0 -13000.0 -0.23 -0.3682 -0.9951 3068376 PK04_096064 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D01 compound treatment 1226400.0 46900.0 0.79 1206560.0 52000.0 0.94 1.2177 0.9962 3068407 PK04_096065 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D02 compound treatment 1216520.0 37100.0 0.62 1195160.0 40600.0 0.73 0.9555 0.9966 3187117 PK04_096066 CN1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5ccc(CN6CCCC6)cc5)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D03 compound treatment 1209400.0 29900.0 0.5 1181720.0 27100.0 0.49 0.7001 0.9999 3187274 PK04_096067 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2CC5(CC6CC7CC(C6)C5)C7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D04 compound treatment 1199080.0 19600.0 0.33 1172000.0 17400.0 0.31 0.4541 0.9998 3068858 PK04_096068 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(C=C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D05 compound treatment 1199040.0 19600.0 0.33 1173240.0 18700.0 0.34 0.4694 0.9999 3187075 PK04_096069 CN(C)CCCNC(=O)[C@H]1[C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D06 compound treatment 1201320.0 21900.0 0.37 1180880.0 26300.0 0.47 0.5937 0.9918 3187118 PK04_096070 OCCCC1=CC(N(Cc2cc3OCOc3cc2Br)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C1)c6ccc(CN7CCCC7)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D07 compound treatment 1185800.0 6340.0 0.11 1163520.0 8940.0 0.16 0.1889 0.9794 3068634 PK04_096071 CC(C)CNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D08 compound treatment 1169760.0 -9700.0 -0.16 1147240.0 -7340.0 -0.13 -0.2083 -0.9948 3068859 PK04_096072 OCc1ccc(cc1)c2cc[n+](Cc3ccc(o3)[N+](=O)[O-])cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D09 compound treatment 1192320.0 12900.0 0.22 1169760.0 15200.0 0.27 0.3456 0.9929 3067975 PK04_096073 CC(C)NC(=O)[C@]1(CC(=O)N(CC2(CC3CC4CC(C3)C2)C4)[C@@H]1c5ccc(CO)cc5)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D10 compound treatment 1184480.0 5020.0 0.08 1149080.0 -5500.0 -0.1 -0.0107 -0.0821 3068860 PK04_096074 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D11 mock treatment 1177240.0 -2220.0 -0.04 1162040.0 7460.0 0.13 0.0688 0.4929 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D12 mock treatment 1189080.0 9620.0 0.16 1159240.0 4660.0 0.08 0.1732 0.9541 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D13 compound treatment 1151400.0 -28100.0 -0.47 1141960.0 -12600.0 -0.23 -0.4928 -0.9445 3187429 PK04_096075 C[C@]1([C@@H](N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4)C(=O)NCCN5CCOCC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D14 compound treatment 1152600.0 -26900.0 -0.45 1142000.0 -12600.0 -0.23 -0.4781 -0.9497 3187119 PK04_096076 CN1C(=O)C2C(C3C(C4CC4)N(Cc5cccc(OC(F)(F)F)c5)C2C=C3CCCO)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D15 mock treatment 1162200.0 -17300.0 -0.29 1138880.0 -15700.0 -0.28 -0.4043 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D16 mock treatment 1168720.0 -10700.0 -0.18 1149800.0 -4780.0 -0.09 -0.188 -0.9431 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D17 compound treatment 1157960.0 -21500.0 -0.36 1121040.0 -33500.0 -0.6 -0.6817 -0.9693 3187348 PK04_096077 CC(C)NC(=O)[C@]1(C)[C@@H](N(C(C)C)C(=O)c2ccccc21)c3ccc(CO)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D18 compound treatment 1134960.0 -44500.0 -0.74 1123360.0 -31200.0 -0.56 -0.9243 -0.9904 3068861 PK04_096078 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C4CC4)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D19 compound treatment 1134400.0 -45100.0 -0.75 1117360.0 -37200.0 -0.67 -1.0074 -0.9983 3187354 PK04_096079 CC(C)NC(=O)[C@]1(C)[C@@H](N(C(=O)c2ccccc21)c3ccc(C)cn3)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D20 compound treatment 1134640.0 -44800.0 -0.75 1105040.0 -49500.0 -0.89 -1.1615 -0.9963 3187120 PK04_096080 OCc1ccc(cc1)c2cc[n+](Cc3sc4ccccc4c3Cl)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D21 compound treatment 1136320.0 -43100.0 -0.72 1102280.0 -52300.0 -0.94 -1.1768 -0.9914 3187433 PK04_096081 CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D22 compound treatment 1137360.0 -42100.0 -0.7 1110760.0 -43800.0 -0.79 -1.0564 -0.9984 3068862 PK04_096082 COc1cc2CCN(C)C(C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D23 compound treatment 1142880.0 -36600.0 -0.61 1114400.0 -40200.0 -0.72 -0.9447 -0.9965 3068462 PK04_096083 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NC3CC3)c4ccccc4C(=O)N2Cc5ccccc5C(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 D24 compound treatment 1113480.0 -66000.0 -1.1 1094120.0 -60500.0 -1.09 -1.551 -1.0 3187121 PK04_096084 COC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(C=C1C(=O)OC)c4ccc(CO)cc4)C5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E01 mock treatment 1218040.0 38600.0 0.65 1187200.0 32600.0 0.59 0.8721 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E02 mock treatment 1228720.0 49300.0 0.82 1193360.0 38800.0 0.7 1.077 0.9966 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E03 compound treatment 1220240.0 40800.0 0.68 1181600.0 27000.0 0.49 0.8268 0.9863 3186708 PK04_096085 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E04 compound treatment 1205560.0 26100.0 0.44 1175120.0 20500.0 0.37 0.5705 0.9966 3186710 PK04_096086 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E05 compound treatment 1202240.0 22800.0 0.38 1175120.0 20500.0 0.37 0.5312 0.9999 3186888 PK04_096087 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E06 compound treatment 1203680.0 24200.0 0.41 1161760.0 7180.0 0.13 0.3781 0.8887 3186565 PK04_096088 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(Cc7ccccc7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E07 compound treatment 1184360.0 4900.0 0.08 1159920.0 5340.0 0.1 0.126 0.9968 3186983 PK04_096089 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E08 compound treatment 1192240.0 12800.0 0.21 1165360.0 10800.0 0.19 0.2886 0.9989 3067581 PK04_096090 CCCN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E09 mock treatment 1191640.0 12200.0 0.2 1162880.0 8300.0 0.15 0.2499 0.9885 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E10 mock treatment 1192720.0 13300.0 0.22 1162800.0 8220.0 0.15 0.2616 0.9807 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E11 compound treatment 1174760.0 -4700.0 -0.08 1154000.0 -576.0 -0.01 -0.063 -0.7935 3186717 PK04_096091 CC(C)CNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E12 compound treatment 1174520.0 -4940.0 -0.08 1144120.0 -10500.0 -0.19 -0.1917 -0.9317 3068221 PK04_096092 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E13 compound treatment 1170120.0 -9340.0 -0.16 1145840.0 -8740.0 -0.16 -0.2219 -1.0 3068273 PK04_096093 CN(C)CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E14 compound treatment 1188960.0 9500.0 0.16 1142080.0 -12500.0 -0.23 -0.0468 -0.1699 3068377 PK04_096094 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E15 compound treatment 1168720.0 -10700.0 -0.18 1135320.0 -19300.0 -0.35 -0.3725 -0.9532 3068408 PK04_096095 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E16 compound treatment 1178560.0 -904.0 -0.02 1154000.0 -576.0 -0.01 -0.018 -0.9832 3186635 PK04_096096 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E17 mock treatment 1169880.0 -9580.0 -0.16 1141920.0 -12700.0 -0.23 -0.2746 -0.9852 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E18 mock treatment 1176840.0 -2620.0 -0.04 1144320.0 -10300.0 -0.18 -0.1617 -0.8514 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E19 compound treatment 1150040.0 -29400.0 -0.49 1124680.0 -29900.0 -0.54 -0.7291 -0.999 3186791 PK04_096097 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E20 compound treatment 1158200.0 -21300.0 -0.36 1133520.0 -21100.0 -0.38 -0.5199 -0.9995 3068233 PK04_096098 CC(C)N1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E21 compound treatment 1148680.0 -30800.0 -0.52 1127920.0 -26700.0 -0.48 -0.7039 -0.9994 3186719 PK04_096099 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)Sc6ccc(C)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E22 compound treatment 1162480.0 -17000.0 -0.28 1127720.0 -26900.0 -0.48 -0.5431 -0.9678 3186789 PK04_096100 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E23 compound treatment 1148840.0 -30600.0 -0.51 1127560.0 -27000.0 -0.49 -0.7066 -0.9997 3186803 PK04_096101 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 E24 compound treatment 1119840.0 -59600.0 -1.0 1101280.0 -53300.0 -0.96 -1.3845 -0.9998 3186711 PK04_096102 CN(C)CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F01 mock treatment 1223360.0 43900.0 0.73 1204120.0 49500.0 0.89 1.1506 0.9953 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F02 mock treatment 1230960.0 51500.0 0.86 1203800.0 49200.0 0.89 1.2365 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F03 compound treatment 1202040.0 22600.0 0.38 1175120.0 20500.0 0.37 0.5289 0.9999 3068521 PK04_096103 CCCNC(=O)[C@H]1[C@@H](N(C2Cc3ccccc3C2)C(=O)c4ccccc14)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F04 compound treatment 1192560.0 13100.0 0.22 1157840.0 3260.0 0.06 0.1965 0.8662 3187122 PK04_096104 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)c4ccc(CN5CCCC5)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F05 compound treatment 1195520.0 16100.0 0.27 1177000.0 22400.0 0.4 0.4757 0.9804 3068461 PK04_096105 CCCNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F06 compound treatment 1227720.0 48300.0 0.81 1199080.0 44500.0 0.8 1.138 1.0 3068863 PK04_096106 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(c5ccc(CN6CCCC6)cc5)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F07 compound treatment 1189640.0 10200.0 0.17 1170680.0 16100.0 0.29 0.3256 0.9678 3187077 PK04_096107 CC(C)CNC(=O)[C@H]1[C@@H](N(Cc2ccccc2C(F)(F)F)C(=O)c3ccccc13)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F08 compound treatment 1187000.0 7540.0 0.13 1139200.0 -15400.0 -0.28 -0.1067 -0.3506 3187123 PK04_096108 CN/1C(C=C(CCCO)C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CN5CCCC5)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F09 mock treatment 1189040.0 9580.0 0.16 1163320.0 8740.0 0.16 0.2247 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F10 mock treatment 1188560.0 9100.0 0.15 1155600.0 1020.0 0.02 0.1207 0.787 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F11 compound treatment 1169760.0 -9700.0 -0.16 1158160.0 3580.0 0.06 -0.0692 -0.3958 3187438 PK04_096109 CN(C)CCCNC(=O)[C@]1(C)[C@@H](N(Cc2ccccc2)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F12 compound treatment 1136320.0 -43100.0 -0.72 1121960.0 -32600.0 -0.59 -0.9261 -0.9948 3187124 PK04_096110 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(C=C1C(=O)OC)c3ccc(CO)cc3)c4cccs4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F13 compound treatment 1172560.0 -6900.0 -0.12 1150960.0 -3620.0 -0.07 -0.1278 -0.9633 3068559 PK04_096111 OCc1ccc(cc1)[C@H]2[C@H](C(=O)NCC(F)(F)F)c3ccccc3C(=O)N2C4CCCCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F14 compound treatment 1146200.0 -33300.0 -0.56 1132600.0 -22000.0 -0.4 -0.6736 -0.9861 3068864 PK04_096112 COC(=O)C1=CN(C)C(C=C(CCCO)C=C1C(=O)OC)c2cccs2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F15 compound treatment 1155800.0 -23700.0 -0.4 1132600.0 -22000.0 -0.4 -0.56 -1.0 3186801 PK04_096113 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F16 compound treatment 1139840.0 -39600.0 -0.66 1116000.0 -38600.0 -0.7 -0.9603 -0.9997 3187125 PK04_096114 COC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(CCCO)C=C1C(=O)OC)C4CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F17 mock treatment 1140920.0 -38500.0 -0.65 1121600.0 -33000.0 -0.59 -0.8762 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F18 mock treatment 1152000.0 -27500.0 -0.46 1131320.0 -23300.0 -0.42 -0.6213 -0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F19 compound treatment 1120400.0 -59100.0 -0.99 1109240.0 -45300.0 -0.82 -1.2765 -0.9955 3186718 PK04_096115 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NC6CC6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F20 compound treatment 1120960.0 -58500.0 -0.98 1099920.0 -54700.0 -0.98 -1.3886 -1.0 3068865 PK04_096116 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)c4cccs4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F21 compound treatment 1133680.0 -45800.0 -0.77 1110320.0 -44300.0 -0.8 -1.1056 -0.9998 3067569 PK04_096117 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)c4ccc(cc4)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F22 compound treatment 1118640.0 -60800.0 -1.02 1085160.0 -69400.0 -1.25 -1.6041 -0.9948 3187126 PK04_096118 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(C=C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F23 compound treatment 1137120.0 -42300.0 -0.71 1104840.0 -49700.0 -0.9 -1.1347 -0.9932 3068643 PK04_096119 COCCCNC(=O)[C@]1(C)[C@@H](N(Cc2cc(F)cc(c2)C(F)(F)F)C(=O)c3ccccc31)c4ccc(CO)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 F24 compound treatment 1122080.0 -57400.0 -0.96 1087960.0 -66600.0 -1.2 -1.5277 -0.9939 3187127 PK04_096120 CN/1C(C=C(C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CO)cc4)c5cccs5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G01 compound treatment 1233960.0 54500.0 0.91 1198440.0 43900.0 0.79 1.2037 0.9975 3186434 PK04_096121 CN(C)CCCN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G02 compound treatment 1228000.0 48500.0 0.81 1195720.0 41100.0 0.74 1.0985 0.999 3067602 PK04_096122 CC(C)N1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G03 mock treatment 1209000.0 29500.0 0.49 1173840.0 19300.0 0.35 0.5949 0.985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G04 mock treatment 1224200.0 44700.0 0.75 1193960.0 39400.0 0.71 1.0311 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G05 compound treatment 1211040.0 31600.0 0.53 1175880.0 21300.0 0.38 0.6451 0.9877 3068238 PK04_096123 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G06 compound treatment 1219040.0 39600.0 0.66 1174120.0 19500.0 0.35 0.7173 0.9563 3068315 PK04_096124 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G07 compound treatment 1196520.0 17100.0 0.29 1172000.0 17400.0 0.31 0.4238 0.9989 3186805 PK04_096125 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G08 compound treatment 1188360.0 8900.0 0.15 1164800.0 10200.0 0.18 0.2355 0.9944 3186712 PK04_096126 COCCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G09 compound treatment 1199040.0 19600.0 0.33 1176840.0 22300.0 0.4 0.5153 0.9949 3068360 PK04_096127 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCN4CCOCC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G10 compound treatment 1194120.0 14700.0 0.25 1164480.0 9900.0 0.18 0.2996 0.9878 3186431 PK04_096128 COc1ccc(CCN2C(=O)[C@]3(CC(=O)N([C@@H]3c4ccc(CO)cc24)C5CCCCC5)c6ccc(cc6)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G11 compound treatment 1173160.0 -6300.0 -0.11 1154320.0 -256.0 0.0 -0.0779 -0.7373 3186642 PK04_096129 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2I)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G12 compound treatment 1175000.0 -4460.0 -0.07 1157200.0 2620.0 0.05 -0.0194 -0.2194 3068326 PK04_096130 CCCNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G13 compound treatment 1163160.0 -16300.0 -0.27 1140960.0 -13600.0 -0.25 -0.3664 -0.9986 3186484 PK04_096131 CCCN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G14 compound treatment 1163640.0 -15800.0 -0.26 1152160.0 -2420.0 -0.04 -0.218 -0.8124 3068146 PK04_096132 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G15 compound treatment 1171720.0 -7740.0 -0.13 1132000.0 -22600.0 -0.41 -0.3793 -0.8884 3068195 PK04_096133 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(C6CC6)C4=O)c7ccccc7C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G16 compound treatment 1176080.0 -3380.0 -0.06 1149720.0 -4860.0 -0.09 -0.1019 -0.9778 3068279 PK04_096134 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G17 compound treatment 1169960.0 -9500.0 -0.16 1153560.0 -1020.0 -0.02 -0.1254 -0.7833 3068328 PK04_096135 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G18 compound treatment 1147840.0 -31600.0 -0.53 1143600.0 -11000.0 -0.2 -0.514 -0.9099 3068311 PK04_096136 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G19 mock treatment 1152360.0 -27100.0 -0.45 1129920.0 -24700.0 -0.44 -0.6348 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G20 mock treatment 1160000.0 -19500.0 -0.33 1133600.0 -21000.0 -0.38 -0.4976 -0.9973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G21 compound treatment 1138360.0 -41100.0 -0.69 1121080.0 -33500.0 -0.6 -0.9131 -0.9979 3068284 PK04_096137 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G22 compound treatment 1160200.0 -19300.0 -0.32 1125960.0 -28600.0 -0.52 -0.5925 -0.9744 3186501 PK04_096138 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G23 compound treatment 1137200.0 -42300.0 -0.71 1118760.0 -35800.0 -0.65 -0.9564 -0.999 3186555 PK04_096139 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 G24 compound treatment 1144520.0 -34900.0 -0.58 1120200.0 -34400.0 -0.62 -0.8514 -0.9996 3186877 PK04_096140 CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H01 compound treatment 1230440.0 51000.0 0.85 1206600.0 52000.0 0.94 1.266 0.9989 3186629 PK04_096141 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H02 compound treatment 1189640.0 10200.0 0.17 1155120.0 544.0 0.01 0.1273 0.7466 3068866 PK04_096142 OCc1ccc(cc1)c2cc[n+](Cc3cc4OCOc4cc3Br)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H03 mock treatment 1215600.0 36100.0 0.6 1190640.0 36100.0 0.65 0.8871 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H04 mock treatment 1213120.0 33700.0 0.56 1186360.0 31800.0 0.57 0.8032 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H05 compound treatment 1190360.0 10900.0 0.18 1168200.0 13600.0 0.25 0.3025 0.9893 3186432 PK04_096143 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(Cc5ccccc5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H06 compound treatment 1189040.0 9580.0 0.16 1160920.0 6340.0 0.11 0.1941 0.9863 3068867 PK04_096144 OCc1ccc(cc1)c2cc[n+](Cc3cccc(OC(F)(F)F)c3)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H07 compound treatment 1191000.0 11500.0 0.19 1165680.0 11100.0 0.2 0.278 0.9998 3187128 PK04_096145 CC(C)CN1C(=O)[C@]2(CC(=O)N(CC3C4CC5CC(C4)CC3C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H08 compound treatment 1195560.0 16100.0 0.27 1178880.0 24300.0 0.44 0.5001 0.9728 3068868 PK04_096146 COc1cc2CC[N+](=Cc2cc1O)Cc3sc4ccccc4c3Cl 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H09 compound treatment 1177120.0 -2340.0 -0.04 1145120.0 -9460.0 -0.17 -0.1482 -0.8477 3186637 PK04_096147 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H10 compound treatment 1183040.0 3580.0 0.06 1165960.0 11400.0 0.21 0.1873 0.8769 3187129 PK04_096148 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(C4CC4)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H11 compound treatment 1172400.0 -7060.0 -0.12 1157120.0 2540.0 0.05 -0.0512 -0.4037 3187130 PK04_096149 CC1(C)OB(OC1(C)C)/C=C\CC(OC(=O)c2ccncc2)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H12 compound treatment 1176920.0 -2540.0 -0.04 1134320.0 -20300.0 -0.36 -0.2882 -0.7843 3187131 PK04_096150 C[n+]1ccc(cc1)c2ccc(CO)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H13 compound treatment 1153600.0 -25900.0 -0.43 1143000.0 -11600.0 -0.21 -0.4535 -0.944 3068898 PK04_096151 COC(=O)c1ccc(OC)c(/C=C\CC(OC(=O)C)c2ccccc2)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H14 compound treatment 1102680.0 -76800.0 -1.28 1109920.0 -44700.0 -0.8 -1.4775 -0.9746 3187132 PK04_096152 CN1C(=O)C2C(C3C(N(Cc4cc5OCOc5cc4Br)C2C=C3CCCO)c6cccs6)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H15 compound treatment 1156120.0 -23300.0 -0.39 1132480.0 -22100.0 -0.4 -0.5577 -1.0 3187133 PK04_096153 COC(=O)c1ccc(OC)c(/C=C\CC(CCc2ccccc2)OC(=O)C)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H16 compound treatment 1125680.0 -53800.0 -0.9 1096120.0 -58500.0 -1.05 -1.3812 -0.9969 3187134 PK04_096154 OCc1ccc(cc1)C2=CC(N(Cc3cccc(OC(F)(F)F)c3)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C2)c6cccs6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H17 compound treatment 1150320.0 -29100.0 -0.49 1110040.0 -44500.0 -0.8 -0.9123 -0.9715 3068899 PK04_096155 COC(=O)c1ccc(OC)c(/C=C\CC(CCc2ccccc2)OC(=O)c3ccncc3)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H18 compound treatment 1153960.0 -25500.0 -0.43 1131760.0 -22800.0 -0.41 -0.5925 -0.9998 3068900 PK04_096156 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(C5CC5)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H19 mock treatment 1149560.0 -29900.0 -0.5 1116360.0 -38200.0 -0.69 -0.8407 -0.9877 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H20 mock treatment 1140920.0 -38500.0 -0.65 1094440.0 -60100.0 -1.08 -1.2222 -0.9693 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H21 compound treatment 1098040.0 -81400.0 -1.36 1062680.0 -91900.0 -1.66 -2.1343 -0.9953 3187204 PK04_096157 CC(C)(C)OC(=O)COc1cccc(c1)C(=O)CCN2CCOCC2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H22 compound treatment 1143840.0 -35600.0 -0.6 1116760.0 -37800.0 -0.68 -0.9033 -0.9978 3187205 PK04_096158 OCCCc1cc[n+](Cc2cc3OCOc3cc2Br)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H23 compound treatment 1066480.0 -113000.0 -1.89 1052600.0 -102000.0 -1.84 -2.6361 -0.9999 3068901 PK04_096159 COc1ccc(/C=C/C(=O)c2cccc(OCC(=O)OC(C)(C)C)c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 H24 compound treatment 1128120.0 -51300.0 -0.86 1105240.0 -49300.0 -0.89 -1.2361 -0.9999 3187206 PK04_096160 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(CCCO)C=C1C(=O)OC)C4CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I01 compound treatment 1240600.0 61100.0 1.02 1200920.0 46300.0 0.83 1.3139 0.9949 3186796 PK04_096161 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I02 compound treatment 1227960.0 48500.0 0.81 1191920.0 37300.0 0.67 1.0496 0.9957 3186628 PK04_096162 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4Cl)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I03 compound treatment 1218080.0 38600.0 0.65 1189920.0 35300.0 0.64 0.9072 1.0 3186882 PK04_096163 CN(C)CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I04 compound treatment 1211240.0 31800.0 0.53 1177160.0 22600.0 0.41 0.6637 0.9913 3186797 PK04_096164 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I05 mock treatment 1206760.0 27300.0 0.46 1181400.0 26800.0 0.48 0.6647 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I06 mock treatment 1203320.0 23900.0 0.4 1168640.0 14100.0 0.25 0.4615 0.9759 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I07 compound treatment 1189000.0 9540.0 0.16 1167480.0 12900.0 0.23 0.2772 0.9831 3186430 PK04_096165 OCc1ccc2[C@H]3N(C4CCCCC4)C(=O)C[C@@]3(C(=O)N(C5CC5)c2c1)c6ccc(cc6)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I08 compound treatment 1196640.0 17200.0 0.29 1163440.0 8860.0 0.16 0.3162 0.9615 3186557 PK04_096166 CC(C)CNC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I09 compound treatment 1162840.0 -16600.0 -0.28 1165400.0 10800.0 0.2 -0.0588 -0.1731 3186558 PK04_096167 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I10 compound treatment 1176400.0 -3060.0 -0.05 1157760.0 3180.0 0.06 0.0043 0.056 3068320 PK04_096168 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I11 compound treatment 1187120.0 7660.0 0.13 1149640.0 -4940.0 -0.09 0.0277 0.1777 3068364 PK04_096169 COCCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I12 compound treatment 1177600.0 -1860.0 -0.03 1144800.0 -9780.0 -0.18 -0.1466 -0.8196 3186489 PK04_096170 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCCN6CCOCC6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I13 compound treatment 1169360.0 -10100.0 -0.17 1138280.0 -16300.0 -0.29 -0.3272 -0.9656 3186807 PK04_096171 CC(C)CNC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I14 compound treatment 1177640.0 -1820.0 -0.03 1142080.0 -12500.0 -0.23 -0.1808 -0.7957 3068281 PK04_096172 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I15 compound treatment 1167120.0 -12300.0 -0.21 1139680.0 -14900.0 -0.27 -0.3358 -0.9916 3186567 PK04_096173 CN(C)CCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I16 compound treatment 1164440.0 -15000.0 -0.25 1132400.0 -22200.0 -0.4 -0.4603 -0.9751 3068410 PK04_096174 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I17 compound treatment 1161280.0 -18200.0 -0.3 1138400.0 -16200.0 -0.29 -0.4213 -0.9998 3186973 PK04_096175 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I18 compound treatment 1165440.0 -14000.0 -0.23 1122280.0 -32300.0 -0.58 -0.5774 -0.9203 3068148 PK04_096176 CC(C)NC(=O)[C@]1(Cc2ccccc2I)[C@@H](N(Cc3ccccc3Cl)C(=O)c4ccccc41)c5ccc(CO)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I19 compound treatment 1159840.0 -19600.0 -0.33 1118600.0 -36000.0 -0.65 -0.6906 -0.9503 3068239 PK04_096177 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I20 compound treatment 1152760.0 -26700.0 -0.45 1119200.0 -35400.0 -0.64 -0.7667 -0.9849 3068268 PK04_096178 CCCNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I21 mock treatment 1150040.0 -29400.0 -0.49 1122880.0 -31700.0 -0.57 -0.752 -0.9973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I22 mock treatment 1157600.0 -21900.0 -0.37 1128960.0 -25600.0 -0.46 -0.5851 -0.9934 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I23 compound treatment 1116440.0 -63000.0 -1.05 1124760.0 -29800.0 -0.54 -1.1256 -0.951 3186564 PK04_096179 OCc1ccc(cc1)[C@@H]2N(C3CCCCC3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 I24 compound treatment 1139400.0 -40100.0 -0.67 1115840.0 -38700.0 -0.7 -0.9676 -0.9998 3068366 PK04_096180 CC(C)CNC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J01 compound treatment 1200400.0 20900.0 0.35 1183640.0 29100.0 0.52 0.618 0.9809 1230870 PK04_096181 Oc1cccc(c1)C(=O)CCN2CCOCC2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J02 compound treatment 1182640.0 3180.0 0.05 1166480.0 11900.0 0.21 0.1892 0.8564 3187207 PK04_096182 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OC)C3CC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J03 compound treatment 1194680.0 15200.0 0.25 1162040.0 7460.0 0.13 0.2751 0.9555 3068902 PK04_096183 COc1ccc(CC[C@H](O)c2cccc(OCC(=O)OC(C)(C)C)c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J04 compound treatment 1192120.0 12700.0 0.21 1192480.0 37900.0 0.68 0.6327 0.8848 3187208 PK04_096184 CN1C(=O)C2C(C3C(N(Cc4cccc(OC(F)(F)F)c4)C2C=C3CCCO)c5cccs5)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J05 mock treatment 1201440.0 22000.0 0.37 1170840.0 16300.0 0.29 0.4672 0.9937 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J06 mock treatment 1196960.0 17500.0 0.29 1165120.0 10500.0 0.19 0.3414 0.9781 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J07 compound treatment 1203680.0 24200.0 0.41 1188400.0 33800.0 0.61 0.7175 0.9804 3187209 PK04_096185 CCCN1C(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@H](N2C1=O)c5cccc(O)c5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J08 compound treatment 1187040.0 7580.0 0.13 1142000.0 -12600.0 -0.23 -0.0706 -0.2718 3068903 PK04_096186 OCc1ccc(cc1)C2=CC(C3CC3)N(Cc4cc5OCOc5cc4Br)/C(=N\P(=O)(Oc6ccccc6)Oc7ccccc7)/C2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J09 compound treatment 1198800.0 19300.0 0.32 1174280.0 19700.0 0.36 0.4798 0.9989 1032549 PK04_096187 CCOC(=O)C1CCCCN1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J10 compound treatment 1185640.0 6180.0 0.1 1144640.0 -9940.0 -0.18 -0.0535 -0.2588 3187210 PK04_096188 COc1cc2CCN(C)C(C=C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J11 compound treatment 1189480.0 10000.0 0.17 1147600.0 -6980.0 -0.13 0.0296 0.1415 3187211 PK04_096189 CCOC(=O)[C@@H]1CCCCN1C(=O)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J12 compound treatment 1150960.0 -28500.0 -0.48 1129320.0 -25300.0 -0.46 -0.6591 -0.9997 3187212 PK04_096190 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(c4ccc(CN5CCCC5)cc4)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J13 compound treatment 1149320.0 -30100.0 -0.5 1108720.0 -45900.0 -0.83 -0.9409 -0.972 3068904 PK04_096191 [O-][N+](=O)c1cc(Br)ccc1C(=O)NCc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J14 compound treatment 1149560.0 -29900.0 -0.5 1126840.0 -27700.0 -0.5 -0.7072 -1.0 3068905 PK04_096192 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(C=C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J15 compound treatment 1163720.0 -15700.0 -0.26 1122720.0 -31900.0 -0.57 -0.5921 -0.9376 3187213 PK04_096193 CC(=O)Nc1cc(Br)ccc1C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J16 compound treatment 1167880.0 -11600.0 -0.19 1132360.0 -22200.0 -0.4 -0.4201 -0.9446 3187214 PK04_096194 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(c5cccs5)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J17 compound treatment 1148760.0 -30700.0 -0.51 1132040.0 -22500.0 -0.41 -0.6504 -0.9932 3068906 PK04_096195 CC(=O)Nc1cc(Br)ccc1C(=O)NCc2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J18 compound treatment 1154920.0 -24500.0 -0.41 1125800.0 -28800.0 -0.52 -0.657 -0.9933 3187215 PK04_096196 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(c5cccs5)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J19 compound treatment 811080.0 -368000.0 -6.16 751320.0 -403000.0 -7.27 -9.4966 -0.9967 3068907 PK04_096197 Brc1ccc2c(=O)oc(nc2c1)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J20 compound treatment 1131520.0 -47900.0 -0.8 1091440.0 -63100.0 -1.14 -1.3717 -0.9854 3187216 PK04_096198 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(c4ccc(CN5CCCC5)cc4)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J21 mock treatment 1136600.0 -42900.0 -0.72 1109360.0 -45200.0 -0.81 -1.0833 -0.998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J22 mock treatment 1150760.0 -28700.0 -0.48 1126920.0 -27700.0 -0.5 -0.692 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J23 compound treatment 1145880.0 -33600.0 -0.56 1099280.0 -55300.0 -1.0 -1.1019 -0.9633 3068908 PK04_096199 Nc1cc(Br)ccc1C(=O)O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 J24 compound treatment 1104840.0 -74600.0 -1.25 1067240.0 -87300.0 -1.57 -1.9957 -0.9934 3068910 PK04_096200 Oc1ccc2cc[n+](Cc3ccc(o3)[N+](=O)[O-])cc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K01 compound treatment 1217440.0 38000.0 0.64 1188680.0 34100.0 0.61 0.8839 0.9999 3068198 PK04_096201 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(Cc6ccccc6)C4=O)c7ccccc7C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K02 compound treatment 1223400.0 43900.0 0.74 1196080.0 41500.0 0.75 1.0487 1.0 3186870 PK04_096202 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K03 compound treatment 1217680.0 38200.0 0.64 1187800.0 33200.0 0.6 0.8755 0.9995 3068155 PK04_096203 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K04 compound treatment 1210880.0 31400.0 0.53 1190240.0 35700.0 0.64 0.8261 0.995 3186875 PK04_096204 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCC(F)(F)F 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K05 compound treatment 1212640.0 33200.0 0.56 1198280.0 43700.0 0.79 0.9494 0.9854 3068359 PK04_096205 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NC4CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K06 compound treatment 1221480.0 42000.0 0.7 1191080.0 36500.0 0.66 0.9622 0.9994 3186626 PK04_096206 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CC(F)(F)F)C4=O)c6ccccc6C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K07 mock treatment 1207520.0 28100.0 0.47 1185920.0 31300.0 0.56 0.7313 0.9958 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K08 mock treatment 1199200.0 19700.0 0.33 1175720.0 21100.0 0.38 0.5029 0.9975 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K09 compound treatment 1188440.0 8980.0 0.15 1180720.0 26100.0 0.47 0.4393 0.8885 3186869 PK04_096207 COc1ccc(CCNC(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K10 compound treatment 1188760.0 9300.0 0.16 1172680.0 18100.0 0.33 0.3406 0.9426 3068235 PK04_096208 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K11 compound treatment 1175680.0 -3780.0 -0.06 1136840.0 -17700.0 -0.32 -0.2707 -0.8311 3186487 PK04_096209 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(Cc7ccccc7)c2c1)c8ccc(cc8)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K12 compound treatment 1170760.0 -8700.0 -0.15 1146240.0 -8340.0 -0.15 -0.2092 -0.9999 3068411 PK04_096210 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K13 compound treatment 1175720.0 -3740.0 -0.06 1142080.0 -12500.0 -0.23 -0.2035 -0.8708 3068329 PK04_096211 CC(C)NC(=O)[C@]1(CC(=O)N([C@@H]1c2ccc(CO)cc2)C3CCCCC3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K14 compound treatment 1165600.0 -13900.0 -0.23 1143720.0 -10900.0 -0.2 -0.3024 -0.9964 3067608 PK04_096212 COCCCN1C(=O)[C@]2(CC(=O)N([C@@H]2c3ccc(CO)cc13)C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K15 mock treatment 1170320.0 -9140.0 -0.15 1147360.0 -7220.0 -0.13 -0.2001 -0.9967 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K16 mock treatment 1184880.0 5420.0 0.09 1156320.0 1740.0 0.03 0.0863 0.8997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K17 compound treatment 1164280.0 -15200.0 -0.25 1151240.0 -3340.0 -0.06 -0.2222 -0.8509 3186979 PK04_096213 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K18 compound treatment 1167320.0 -12100.0 -0.2 1145520.0 -9060.0 -0.16 -0.2591 -0.9941 3186636 PK04_096214 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K19 compound treatment 1151920.0 -27500.0 -0.46 1136560.0 -18000.0 -0.32 -0.5555 -0.9853 3186793 PK04_096215 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K20 compound treatment 1164200.0 -15300.0 -0.26 1142160.0 -12400.0 -0.22 -0.3388 -0.9978 3186637 PK04_096216 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K21 compound treatment 1144000.0 -35500.0 -0.59 1129760.0 -24800.0 -0.45 -0.7358 -0.9903 3067613 PK04_096217 COc1ccc(CCN2C(=O)[C@]3(CC(=O)N(CC4(CC5CC6CC(C5)C4)C6)[C@@H]3c7ccc(CO)cc27)c8ccc(cc8)[N+](=O)[O-])cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K22 compound treatment 1144880.0 -34600.0 -0.58 1135240.0 -19300.0 -0.35 -0.6556 -0.9705 3186873 PK04_096218 CCCNC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K23 mock treatment 1158440.0 -21000.0 -0.35 1139720.0 -14900.0 -0.27 -0.438 -0.9909 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 K24 mock treatment 1142400.0 -37100.0 -0.62 1119120.0 -35500.0 -0.64 -0.8903 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L01 compound treatment 1233800.0 54300.0 0.91 1195440.0 40900.0 0.74 1.1636 0.9945 3068940 PK04_096219 Cc1nc2cc(Br)ccc2c(=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L02 compound treatment 1113240.0 -66200.0 -1.11 1108360.0 -46200.0 -0.83 -1.3724 -0.9901 3187217 PK04_096220 COc1cc2CCN(Cc3cc4OCOc4cc3Br)C(c5ccc(CN6CCCC6)cc5)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L03 compound treatment 1207400.0 27900.0 0.47 1181400.0 26800.0 0.48 0.6723 0.9999 3068941 PK04_096221 CC(C)c1nc2cc(Br)ccc2c(=O)o1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L04 compound treatment 1229720.0 50300.0 0.84 1216960.0 62400.0 1.12 1.3895 0.9898 3068942 PK04_096222 COc1cc2CCN(Cc3sc4ccccc4c3Cl)C(C)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L05 compound treatment 1411200.0 232000.0 3.88 1441800.0 287000.0 5.17 6.4014 0.9899 3187218 PK04_096223 Cc1nc2cc(Br)ccc2c(=O)n1Cc3cccc(O)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L06 compound treatment 1179760.0 296.0 0.0 1165760.0 11200.0 0.2 0.146 0.7243 3068943 PK04_096224 COc1cc2CCN(C)C(c3cccs3)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L07 mock treatment 1201400.0 21900.0 0.37 1176840.0 22300.0 0.4 0.5432 0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L08 mock treatment 1193200.0 13700.0 0.23 1169680.0 15100.0 0.27 0.355 0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L09 compound treatment 1183880.0 4420.0 0.07 1146040.0 -8540.0 -0.15 -0.0565 -0.3311 3187219 PK04_096225 Oc1cccc(CNC(=O)c2ccc(Br)cc2NC(=O)c3ccccc3)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L10 compound treatment 1143760.0 -35700.0 -0.6 1123600.0 -31000.0 -0.56 -0.8171 -0.9994 3187220 PK04_096226 COC(=O)C1=CN(Cc2cc3OCOc3cc2Br)C(C=C(C=C1C(=O)OC)c4ccc(CO)cc4)C5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L11 compound treatment 1168120.0 -11300.0 -0.19 1143720.0 -10900.0 -0.2 -0.2725 -0.9999 3068944 PK04_096227 Oc1cccc(Cn2c(nc3cc(Br)ccc3c2=O)c4ccccc4)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L12 compound treatment 1157800.0 -21700.0 -0.36 1138800.0 -15800.0 -0.28 -0.4573 -0.9928 3187221 PK04_096228 CN1C(=O)C2C(C3C(N(Cc4cc5OCOc5cc4Br)C2C=C3CCCO)c6ccc(CN7CCCC7)cc6)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L13 compound treatment 945960.0 -234000.0 -3.91 911200.0 -243000.0 -4.38 -5.8637 -0.9983 1980253 PK04_096229 Cc1c(NC(=O)/C(=C/C=C/c2ccccc2)/C#N)c(=O)n(c3ccccc3)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L14 compound treatment 1124120.0 -55300.0 -0.93 1095520.0 -59100.0 -1.06 -1.4073 -0.9976 3068945 PK04_096230 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OC)c3cccs3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L15 mock treatment 1157920.0 -21500.0 -0.36 1126040.0 -28500.0 -0.51 -0.6185 -0.9849 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L16 mock treatment 1155640.0 -23800.0 -0.4 1137880.0 -16700.0 -0.3 -0.4946 -0.9904 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L17 compound treatment 993920.0 -186000.0 -3.1 962600.0 -192000.0 -3.46 -4.6414 -0.9985 3187222 PK04_096231 Cc1c(NC(=O)/C(=C/C=C/c2ccccc2[N+](=O)[O-])/C#N)c(=O)n(c3ccccc3)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L18 compound treatment 1139520.0 -39900.0 -0.67 1106840.0 -47700.0 -0.86 -1.0808 -0.9922 3187223 PK04_096232 OCCCC1=CC(N(Cc2cc3OCOc3cc2Br)/C(=N\P(=O)(Oc4ccccc4)Oc5ccccc5)/C1)c6cccs6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L19 compound treatment 973040.0 -206000.0 -3.45 954640.0 -200000.0 -3.6 -4.9898 -0.9998 3068946 PK04_096233 Cc1c(NC(=O)/C(=C/C=C/c2ccc(cc2)[N+](=O)[O-])/C#N)c(=O)n(c3ccccc3)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L20 compound treatment 1090960.0 -88500.0 -1.48 1080800.0 -73800.0 -1.33 -1.9872 -0.9985 3187224 PK04_096234 OCCCC1=CC(N(Cc2cccc(OC(F)(F)F)c2)/C(=N\P(=O)(Oc3ccccc3)Oc4ccccc4)/C1)c5cccs5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L21 compound treatment 1016880.0 -163000.0 -2.72 992040.0 -163000.0 -2.93 -3.9946 -0.9993 3068947 PK04_096235 CN(C)c1ccc(/C=C/C=C(\C#N)/C(=O)Nc2c(C)n(C)n(c3ccccc3)c2=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L22 compound treatment 1143360.0 -36100.0 -0.6 1119640.0 -34900.0 -0.63 -0.8723 -0.9998 3187225 PK04_096236 COc1cc2CCN(C)C(C3CC3)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L23 mock treatment 1130360.0 -49100.0 -0.82 1115920.0 -38700.0 -0.7 -1.0735 -0.9966 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 L24 mock treatment 1150000.0 -29500.0 -0.49 1128040.0 -26500.0 -0.48 -0.6867 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M01 compound treatment 1215160.0 35700.0 0.6 1194440.0 39900.0 0.72 0.9303 0.9958 3186502 PK04_096237 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M02 compound treatment 1233240.0 53800.0 0.9 1210920.0 56300.0 1.02 1.3542 0.9982 3186497 PK04_096238 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@@](Cc4ccccc4I)(C(=O)NC(C)C)c5ccccc5C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M03 compound treatment 1228160.0 48700.0 0.81 1198800.0 44200.0 0.8 1.1396 0.9999 3068404 PK04_096239 COCCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M04 compound treatment 1225520.0 46100.0 0.77 1195320.0 40700.0 0.73 1.0641 0.9997 3186643 PK04_096240 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M05 compound treatment 1206400.0 26900.0 0.45 1185920.0 31300.0 0.56 0.7181 0.9938 3186723 PK04_096241 CCCNC(=O)[C@]1(CC(=O)N(Cc2ccccc2Cl)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M06 compound treatment 1208560.0 29100.0 0.49 1186280.0 31700.0 0.57 0.7482 0.9968 3186868 PK04_096242 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3)C4CCCCC4)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M07 compound treatment 1213520.0 34100.0 0.57 1187200.0 32600.0 0.59 0.8186 0.9999 3186798 PK04_096243 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M08 compound treatment 1210560.0 31100.0 0.52 1190680.0 36100.0 0.65 0.8279 0.9939 3186799 PK04_096244 CN(C)CCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3I)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M09 mock treatment 1191040.0 11600.0 0.19 1166760.0 12200.0 0.22 0.2922 0.9981 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M10 mock treatment 1196960.0 17500.0 0.29 1159680.0 5100.0 0.09 0.2721 0.8865 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M11 compound treatment 1185320.0 5860.0 0.1 1161120.0 6540.0 0.12 0.1527 0.9958 3186496 PK04_096245 COc1ccc(CCNC(=O)[C@]2(Cc3ccccc3I)[C@@H](N(Cc4ccccc4OC)C(=O)c5ccccc52)c6ccc(CO)cc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M12 compound treatment 1177760.0 -1700.0 -0.03 1173360.0 18800.0 0.34 0.2191 0.6452 3068379 PK04_096246 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M13 mock treatment 1150880.0 -28600.0 -0.48 1155720.0 1140.0 0.02 -0.3237 -0.676 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M14 mock treatment 1181360.0 1900.0 0.03 1164080.0 9500.0 0.17 0.1435 0.8241 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M15 compound treatment 1165040.0 -14400.0 -0.24 1142720.0 -11900.0 -0.21 -0.3217 -0.9981 3186488 PK04_096247 CC(C)N1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M16 compound treatment 1170720.0 -8740.0 -0.15 1145280.0 -9300.0 -0.17 -0.2219 -0.9977 3186886 PK04_096248 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M17 compound treatment 1155040.0 -24400.0 -0.41 1129400.0 -25200.0 -0.45 -0.6098 -0.9986 3068154 PK04_096249 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3)C(=O)c4ccccc4[C@]2(Cc5ccccc5I)C(=O)NCc6ccccc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M18 compound treatment 1157160.0 -22300.0 -0.37 1149440.0 -5140.0 -0.09 -0.3294 -0.8565 3068369 PK04_096250 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M19 compound treatment 1164080.0 -15400.0 -0.26 1146160.0 -8420.0 -0.15 -0.2893 -0.9681 3186727 PK04_096251 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M20 compound treatment 1148720.0 -30700.0 -0.51 1124080.0 -30500.0 -0.55 -0.7523 -0.9995 3186984 PK04_096252 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M21 compound treatment 1127760.0 -51700.0 -0.87 1121640.0 -32900.0 -0.59 -1.0314 -0.9831 3068372 PK04_096253 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M22 compound treatment 1146000.0 -33500.0 -0.56 1128560.0 -26000.0 -0.47 -0.7274 -0.9961 3186721 PK04_096254 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5I)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M23 compound treatment 1165600.0 -13900.0 -0.23 1131280.0 -23300.0 -0.42 -0.4608 -0.9609 3068316 PK04_096255 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 M24 compound treatment 1132280.0 -47200.0 -0.79 1108000.0 -46600.0 -0.84 -1.1517 -0.9995 3068283 PK04_096256 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N01 compound treatment 1192480.0 13000.0 0.22 1185760.0 31200.0 0.56 0.5513 0.9149 1694663 PK04_096257 Cc1c(NC(=O)CC#N)c(=O)n(c2ccccc2)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N02 compound treatment 1185920.0 6460.0 0.11 1175840.0 21300.0 0.38 0.3473 0.8725 3187226 PK04_096258 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C)C=C(CCCO)C=C1C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N03 compound treatment 1201720.0 22300.0 0.37 1189000.0 34400.0 0.62 0.7019 0.9702 3068949 PK04_096259 Cc1ccccc1/C=C/C=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N04 compound treatment 1171120.0 -8340.0 -0.14 1145960.0 -8620.0 -0.16 -0.2085 -0.9986 3187227 PK04_096260 COC(=O)C1=CN(C)C(C=C(CCCO)C=C1C(=O)OC)c2ccc(CN3CCCC3)cc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N05 compound treatment 1202840.0 23400.0 0.39 1195640.0 41100.0 0.74 0.7998 0.9556 3068950 PK04_096261 CCOc1ccc(cc1)N2C(SCC2=O)c3cccc(c3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N06 compound treatment 1161480.0 -18000.0 -0.3 1151200.0 -3380.0 -0.06 -0.2558 -0.8332 3187228 PK04_096262 Oc1ccc2cc[n+](Cc3cccc(OC(F)(F)F)c3)cc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N07 compound treatment 1188120.0 8660.0 0.14 1160160.0 5580.0 0.1 0.1736 0.9841 3068951 PK04_096263 [O-][N+](=O)c1cccc(c1)C2SCC(=O)N2c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N08 compound treatment 1157080.0 -22400.0 -0.37 1144760.0 -9820.0 -0.18 -0.3899 -0.9413 3187299 PK04_096264 CN1C(=O)C2C(C3C(N(C)C2C=C3CCCO)c4cccs4)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N09 mock treatment 1174720.0 -4740.0 -0.08 1152320.0 -2260.0 -0.04 -0.0849 -0.9517 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N10 mock treatment 1176440.0 -3020.0 -0.05 1153800.0 -776.0 -0.01 -0.0457 -0.8699 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N11 compound treatment 1123440.0 -56000.0 -0.94 1128720.0 -25900.0 -0.47 -0.9923 -0.9479 3068985 PK04_096265 Cc1cc(C)cc(c1)N2C(SCC2=O)c3cccc(c3)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N12 compound treatment 1135320.0 -44100.0 -0.74 1130320.0 -24300.0 -0.44 -0.8314 -0.9686 3187300 PK04_096266 COc1cc2CCN(C)C(c3ccc(CN4CCCC4)cc3)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N13 mock treatment 1151960.0 -27500.0 -0.46 1138080.0 -16500.0 -0.3 -0.5356 -0.9776 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N14 mock treatment 1151880.0 -27600.0 -0.46 1128040.0 -26500.0 -0.48 -0.6645 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N15 compound treatment 1144600.0 -34900.0 -0.58 1127640.0 -26900.0 -0.49 -0.7557 -0.9958 3068986 PK04_096267 COc1ccc(/C=C/C=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N16 compound treatment 1132760.0 -46700.0 -0.78 1123280.0 -31300.0 -0.56 -0.9514 -0.9872 3187301 PK04_096268 OCCCC1=CC(C2CC2)N(Cc3sc4ccccc4c3Cl)/C(=N\P(=O)(Oc5ccccc5)Oc6ccccc6)/C1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N17 compound treatment 1141080.0 -38400.0 -0.64 1115440.0 -39100.0 -0.71 -0.9528 -0.9989 3068987 PK04_096269 Cc1cccc(/C=C/C=O)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N18 compound treatment 1154360.0 -25100.0 -0.42 1128160.0 -26400.0 -0.48 -0.6336 -0.9981 3068988 PK04_096270 OCCCc1cc[n+](Cc2sc3ccccc3c2Cl)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N19 compound treatment 1128160.0 -51300.0 -0.86 1108640.0 -45900.0 -0.83 -1.1923 -0.9998 3068989 PK04_096271 Cc1ccc(/C=C/C=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N20 compound treatment 1104120.0 -75300.0 -1.26 1087280.0 -67300.0 -1.21 -1.7489 -0.9998 3187302 PK04_096272 CN1C(=O)C2C(C3C(C4CC4)N(Cc5sc6ccccc6c5Cl)C2C=C3c7ccc(CO)cc7)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N21 compound treatment 1115040.0 -64400.0 -1.08 1107440.0 -47100.0 -0.85 -1.3629 -0.993 3068990 PK04_096273 COc1cccc(/C=C/C=O)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N22 compound treatment 1131960.0 -47500.0 -0.79 1109920.0 -44700.0 -0.8 -1.131 -1.0 3068991 PK04_096274 Oc1ccc2cc[n+](Cc3cc4OCOc4cc3Br)cc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N23 compound treatment 1104200.0 -75300.0 -1.26 1051280.0 -103000.0 -1.86 -2.2066 -0.9819 3187303 PK04_096275 Clc1ccccc1/C=C/C=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 N24 compound treatment 1129000.0 -50500.0 -0.84 1108280.0 -46300.0 -0.83 -1.187 -1.0 3187304 PK04_096276 CN/1C(C=C(C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)c4ccc(CO)cc4)C5CC5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O01 compound treatment 1223600.0 44100.0 0.74 1200480.0 45900.0 0.83 1.1071 0.9984 3186631 PK04_096277 CC(C)CN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(Cc4ccccc4C(F)(F)F)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O02 compound treatment 1219880.0 40400.0 0.68 1202400.0 47800.0 0.86 1.0875 0.9928 3067615 PK04_096278 OCc1ccc2[C@H]3N(CC4(CC5CC6CC(C5)C4)C6)C(=O)C[C@@]3(C(=O)N(CC(F)(F)F)c2c1)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O03 compound treatment 1187880.0 8420.0 0.14 1163680.0 9100.0 0.16 0.2156 0.9971 3186715 PK04_096279 CC(C)N1[C@H](c2ccc(CO)cc2I)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCCCN(C)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O04 compound treatment 1206560.0 27100.0 0.45 1178560.0 24000.0 0.43 0.6262 0.9997 3068363 PK04_096280 CC(C)NC(=O)[C@]1(CC(=O)N(C(C)C)[C@@H]1c2ccc(CO)cc2)Sc3ccc(C)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O05 compound treatment 1210200.0 30700.0 0.51 1191960.0 37400.0 0.67 0.84 0.9911 3068310 PK04_096281 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3C(F)(F)F)[C@@H]2c4ccc(CO)cc4I)C(=O)NCC(F)(F)F)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O06 compound treatment 1210680.0 31200.0 0.52 1188480.0 33900.0 0.61 0.8013 0.997 3068196 PK04_096282 COc1ccccc1CN2[C@@H](c3ccc(CO)cc3)[C@]4(Cc5ccccc5N(CCN6CCOCC6)C4=O)c7ccccc7C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O07 compound treatment 1201480.0 22000.0 0.37 1187040.0 32500.0 0.58 0.6741 0.9752 3068277 PK04_096283 COc1ccc(CCNC(=O)[C@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)Sc5ccc(C)cc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O08 compound treatment 1197200.0 17700.0 0.3 1177920.0 23300.0 0.42 0.5073 0.9854 3186720 PK04_096284 CC(C)NC(=O)[C@]1(CC(=O)N(C2Cc3ccccc3C2)[C@@H]1c4ccc(CO)cc4I)Sc5ccc(C)cc5 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O09 compound treatment 1173240.0 -6220.0 -0.1 1151600.0 -2980.0 -0.05 -0.1116 -0.9524 3186632 PK04_096285 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3C(F)(F)F)C(=O)c4ccccc4[C@]52Cc6ccccc6N(CCN7CCOCC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O10 compound treatment 1158720.0 -20700.0 -0.35 1127640.0 -26900.0 -0.49 -0.5886 -0.9865 3068157 PK04_096286 COc1ccc(CCN2C(=O)[C@]3(Cc4ccccc24)[C@@H](N(C5CCCCC5)C(=O)c6ccccc63)c7ccc(CO)cc7)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O11 mock treatment 1174240.0 -5220.0 -0.09 1147320.0 -7260.0 -0.13 -0.1543 -0.9808 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O12 mock treatment 1190440.0 11000.0 0.18 1161600.0 7020.0 0.13 0.2194 0.9835 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O13 compound treatment 1156080.0 -23400.0 -0.39 1131920.0 -22700.0 -0.41 -0.5653 -0.9998 3186874 PK04_096287 CC(C)N1[C@H](c2ccc(CO)cc2)[C@@](CC1=O)(Sc3ccc(C)cc3)C(=O)NCc4ccccc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O14 compound treatment 1147760.0 -31700.0 -0.53 1117800.0 -36800.0 -0.66 -0.8437 -0.9939 3068138 PK04_096288 COCCCN1C(=O)[C@]2(CC(=O)N(CC3(CC4CC5CC(C4)C3)C5)[C@@H]2c6ccc(CO)cc16)c7ccc(cc7)[N+](=O)[O-] 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O15 compound treatment 1146520.0 -32900.0 -0.55 1137320.0 -17300.0 -0.31 -0.6097 -0.9633 3186972 PK04_096289 CC(C)CNC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O16 compound treatment 1158560.0 -20900.0 -0.35 1145520.0 -9060.0 -0.16 -0.3627 -0.9397 3186981 PK04_096290 COCCCNC(=O)[C@]1(CC(=O)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O17 compound treatment 1156720.0 -22700.0 -0.38 1142680.0 -11900.0 -0.21 -0.4207 -0.9631 3186709 PK04_096291 Cc1ccc(S[C@@]2(CC(=O)N([C@@H]2c3ccc(CO)cc3I)C4CCCCC4)C(=O)NCc5ccccc5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O18 compound treatment 1159040.0 -20400.0 -0.34 1139760.0 -14800.0 -0.27 -0.4304 -0.9925 3186725 PK04_096292 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3Cl)[C@@H]2c4ccc(CO)cc4I)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O19 compound treatment 1119120.0 -60300.0 -1.01 1099400.0 -55200.0 -0.99 -1.417 -1.0 3068321 PK04_096293 Cc1ccc(S[C@@]2(CC(=O)N(Cc3ccccc3)[C@@H]2c4ccc(CO)cc4I)C(=O)NC5CC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O20 compound treatment 1145480.0 -34000.0 -0.57 1108960.0 -45600.0 -0.82 -0.9833 -0.9838 3068192 PK04_096294 COCCCN1C(=O)[C@]2(Cc3ccccc13)[C@@H](N(C4CCCCC4)C(=O)c5ccccc52)c6ccc(CO)cc6 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O21 compound treatment 1121320.0 -58100.0 -0.97 1099520.0 -55100.0 -0.99 -1.3894 -1.0 3068201 PK04_096295 OCc1ccc(cc1)[C@@H]2N(Cc3ccccc3Cl)C(=O)c4ccccc4[C@]52Cc6ccccc6N(C7CC7)C5=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O22 compound treatment 1140680.0 -38800.0 -0.65 1124400.0 -30200.0 -0.54 -0.8434 -0.9961 3068381 PK04_096296 CC(C)NC(=O)[C@]1(CC(=O)N(Cc2ccccc2C(F)(F)F)[C@@H]1c3ccc(CO)cc3)Sc4ccc(C)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O23 compound treatment 1104920.0 -74500.0 -1.25 1089320.0 -65300.0 -1.18 -1.7135 -0.9996 3186880 PK04_096297 Cc1ccc(S[C@@]2(CC(=O)N(C3Cc4ccccc4C3)[C@@H]2c5ccc(CO)cc5)C(=O)NCc6ccccc6)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 O24 compound treatment 1157440.0 -22000.0 -0.37 1121480.0 -33100.0 -0.6 -0.6823 -0.9733 3186977 PK04_096298 Cc1ccc(S[C@@]2(CC(=O)N(Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[C@@H]2c4ccc(CO)cc4)C(=O)NCCN5CCOCC5)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P01 compound treatment 1135960.0 -43500.0 -0.73 1109320.0 -45300.0 -0.82 -1.0914 -0.9984 3068992 PK04_096299 Cc1c(NC(=O)/C(=C/c2cccc(c2)[N+](=O)[O-])/C#N)c(=O)n(c3ccccc3)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P02 compound treatment 1205400.0 25900.0 0.43 1187520.0 32900.0 0.59 0.7266 0.9882 3187305 PK04_096300 COC(=O)C1=CN(C)C(C=C(CCCO)C=C1C(=O)OC)C2CC2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P03 compound treatment 1182720.0 3260.0 0.05 1160120.0 5540.0 0.1 0.1092 0.9594 3187306 PK04_096301 COc1cccc(/C=C(\C#N)/C(=O)Nc2c(C)n(C)n(c3ccccc3)c2=O)c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P04 compound treatment 1155440.0 -24000.0 -0.4 1133240.0 -21300.0 -0.38 -0.5561 -0.9997 3068993 PK04_096302 COc1cc2CC[N+](=Cc2cc1O)C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P05 compound treatment 1133040.0 -46400.0 -0.78 1134480.0 -20100.0 -0.36 -0.8054 -0.9396 3068994 PK04_096303 Cc1c(NC(=O)/C(=C/c2ccccc2Cl)/C#N)c(=O)n(c3ccccc3)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P06 compound treatment 1150880.0 -28600.0 -0.48 1132560.0 -22000.0 -0.4 -0.6187 -0.9957 3187307 PK04_096304 COc1cc2CCN(Cc3cccc(OC(F)(F)F)c3)C(c4cccs4)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P07 compound treatment 1168080.0 -11400.0 -0.19 1141320.0 -13300.0 -0.24 -0.3036 -0.9937 3187308 PK04_096305 Cc1c(NC(=O)/C(=C/c2ccc(Cl)cc2)/C#N)c(=O)n(c3ccccc3)n1C 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P08 compound treatment 1163680.0 -15800.0 -0.26 1151680.0 -2900.0 -0.05 -0.2237 -0.8307 3068995 PK04_096306 CN1C(=O)C2C(C3C(C4CC4)N(C)C2C=C3CCCO)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P09 compound treatment 1160520.0 -18900.0 -0.32 1150720.0 -3860.0 -0.07 -0.2733 -0.8421 1972122 PK04_096307 Cc1cc(C)cc(c1)N2C(c3cccc(c3)[N+](=O)[O-])S(=O)(=O)CC2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P10 compound treatment 1146760.0 -32700.0 -0.55 1133840.0 -20700.0 -0.37 -0.6512 -0.9827 3187309 PK04_096308 CN/1C(C=C(CCCO)C\C1=N\P(=O)(Oc2ccccc2)Oc3ccccc3)C4CC4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P11 mock treatment 1158160.0 -21300.0 -0.36 1129280.0 -25300.0 -0.46 -0.5744 -0.9926 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P12 mock treatment 1165760.0 -13700.0 -0.23 1152680.0 -1900.0 -0.03 -0.1863 -0.8036 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P13 compound treatment 1150320.0 -29100.0 -0.49 1125800.0 -28800.0 -0.52 -0.7115 -0.9995 3068996 PK04_096309 Clc1ccc(/C=C/C=O)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P14 compound treatment 1136400.0 -43100.0 -0.72 1128080.0 -26500.0 -0.48 -0.8471 -0.98 3187310 PK04_096310 COc1cc2CC[N+](=Cc2cc1O)Cc3cccc(OC(F)(F)F)c3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P15 compound treatment 1138800.0 -40700.0 -0.68 1110640.0 -43900.0 -0.79 -1.0409 -0.9972 3068997 PK04_096311 O=C/C=C/c1ccc2OCOc2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P16 compound treatment 1050400.0 -129000.0 -2.16 1034520.0 -120000.0 -2.16 -3.0568 -1.0 3187311 PK04_096312 COC(=O)C1=CN(Cc2cccc(OC(F)(F)F)c2)C(C=C(CCCO)C=C1C(=O)OC)c3ccc(CN4CCCC4)cc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P17 compound treatment 1154360.0 -25100.0 -0.42 1183280.0 28700.0 0.52 0.0686 0.103 3068998 PK04_096313 O=C/C=C/c1ccc(cc1)c2ccccc2 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P18 compound treatment 1097120.0 -82300.0 -1.38 1082040.0 -72500.0 -1.31 -1.8985 -0.9996 3187312 PK04_096314 CN1C(=O)C2C(C3C(C4CC4)N(Cc5cc6OCOc6cc5Br)C2C=C3c7ccc(CO)cc7)C1=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P19 compound treatment 1016640.0 -163000.0 -2.72 1005280.0 -149000.0 -2.69 -3.8288 -1.0 3187313 PK04_096315 O=C/C=C/c1ccc(\C=C\c2ccccc2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P20 compound treatment 1094920.0 -84500.0 -1.41 1055440.0 -99100.0 -1.79 -2.2634 -0.9933 3187314 PK04_096316 COc1cc2CCN(Cc3ccc(o3)[N+](=O)[O-])C(c4cccs4)c2cc1O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P21 compound treatment 1112280.0 -67200.0 -1.12 1090840.0 -63700.0 -1.15 -1.607 -0.9999 3069028 PK04_096317 [O-][N+](=O)c1cccc(c1)C2N(C(=O)CS2(=O)=O)c3ccccc3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P22 compound treatment 1067720.0 -112000.0 -1.87 1038480.0 -116000.0 -2.09 -2.8014 -0.9984 3187315 PK04_096318 COC(=O)C1=CN(Cc2sc3ccccc3c2Cl)C(C=C(CCCO)C=C1C(=O)OC)c4ccc(CN5CCCC5)cc4 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P23 compound treatment 1147160.0 -32300.0 -0.54 1114760.0 -39800.0 -0.72 -0.8895 -0.9903 3069029 PK04_096319 CCOc1ccc(cc1)N2C(c3cccc(c3)[N+](=O)[O-])S(=O)(=O)/C(=C\C=C\c4ccccc4OC)/C2=O 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2096 P24 compound treatment 1109760.0 -69700.0 -1.17 1077680.0 -76900.0 -1.39 -1.8045 -0.9963 3187316 PK04_096320 COC(=O)C1=CN(C)C(C=C(C=C1C(=O)OC)c2ccc(CO)cc2)C3CC3 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A01 compound treatment 1128760.0 -39000.0 -0.65 1126640.0 -38500.0 -0.69 -0.9521 -0.9995 2141518 PK04_097001 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A02 compound treatment 1193120.0 25400.0 0.42 1184440.0 19300.0 0.35 0.5459 0.9951 2141905 PK04_097002 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A03 compound treatment 985280.0 -182000.0 -3.05 971600.0 -194000.0 -3.49 -4.6251 -0.9978 2141091 PK04_097003 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A04 compound treatment 1201520.0 33800.0 0.57 1184760.0 19600.0 0.35 0.6494 0.9745 2141692 PK04_097004 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A05 compound treatment 1150240.0 -17500.0 -0.29 1148600.0 -16500.0 -0.3 -0.4181 -1.0 2141533 PK04_097005 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A06 compound treatment 1201680.0 33900.0 0.57 1191840.0 26700.0 0.48 0.7415 0.9966 2141714 PK04_097006 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A07 compound treatment 1175000.0 7240.0 0.12 1179440.0 14300.0 0.26 0.2678 0.9409 2141463 PK04_097007 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A08 compound treatment 1115360.0 -52400.0 -0.88 1101240.0 -63900.0 -1.15 -1.4342 -0.991 2141076 PK04_097008 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A09 compound treatment 1137440.0 -30300.0 -0.51 1138120.0 -27000.0 -0.49 -0.7031 -0.9998 2141109 PK04_097009 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A10 compound treatment 1139720.0 -28000.0 -0.47 1154560.0 -10600.0 -0.19 -0.4667 -0.9214 2141546 PK04_097010 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A11 compound treatment 1169640.0 1880.0 0.03 1163080.0 -2070.0 -0.04 -0.0041 -0.0837 2141079 PK04_097011 OC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A12 compound treatment 1129360.0 -38400.0 -0.64 1121840.0 -43300.0 -0.78 -1.0061 -0.9953 2141141 PK04_097012 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A13 mock treatment 1189400.0 21600.0 0.36 1187080.0 21900.0 0.4 0.5355 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A14 mock treatment 1180920.0 13200.0 0.22 1185840.0 20700.0 0.37 0.4194 0.9685 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A15 compound treatment 1151680.0 -16100.0 -0.27 1161440.0 -3710.0 -0.07 -0.2375 -0.8567 2141882 PK04_097013 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A16 compound treatment 1155280.0 -12500.0 -0.21 1148000.0 -17100.0 -0.31 -0.3661 -0.9818 2141936 PK04_097014 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A17 compound treatment 1149520.0 -18200.0 -0.31 1153080.0 -12100.0 -0.22 -0.3696 -0.9862 2141372 PK04_097015 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A18 compound treatment 1102920.0 -64800.0 -1.09 1099640.0 -65500.0 -1.18 -1.6018 -0.9991 2141092 PK04_097016 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A19 compound treatment 1147480.0 -20300.0 -0.34 1141760.0 -23400.0 -0.42 -0.5379 -0.9942 2141344 PK04_097017 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A20 compound treatment 1118520.0 -49200.0 -0.82 1103360.0 -61800.0 -1.11 -1.3698 -0.989 2141115 PK04_097018 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A21 compound treatment 1118720.0 -49000.0 -0.82 1116880.0 -48300.0 -0.87 -1.1952 -0.9996 2141570 PK04_097019 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A22 compound treatment 1121400.0 -46400.0 -0.78 1112040.0 -53100.0 -0.96 -1.2252 -0.9946 2141549 PK04_097020 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A23 compound treatment 1147760.0 -20000.0 -0.33 1152840.0 -12300.0 -0.22 -0.3935 -0.98 2141876 PK04_097021 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 A24 compound treatment 1109440.0 -58300.0 -0.98 1097480.0 -67700.0 -1.22 -1.5522 -0.9939 2141753 PK04_097022 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B01 compound treatment 1219320.0 51600.0 0.86 1180840.0 15700.0 0.28 0.81 0.8921 2141940 PK04_097023 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccccc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B02 compound treatment 1219960.0 52200.0 0.87 1183360.0 18200.0 0.33 0.8497 0.9106 2142685 PK04_097024 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B03 compound treatment 1211800.0 44000.0 0.74 1195960.0 30800.0 0.56 0.9137 0.9902 2141335 PK04_097025 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B04 compound treatment 1211640.0 43900.0 0.73 1206640.0 41500.0 0.75 1.0479 1.0 2143933 PK04_097026 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B05 compound treatment 1214440.0 46700.0 0.78 1208160.0 43000.0 0.77 1.1004 1.0 2141445 PK04_097027 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B06 compound treatment 1204320.0 36600.0 0.61 1200520.0 35400.0 0.64 0.8833 0.9998 2144925 PK04_097028 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B07 compound treatment 1192640.0 24900.0 0.42 1193680.0 28500.0 0.51 0.6579 0.9945 2141881 PK04_097029 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccccc3OCCO)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B08 compound treatment 1190320.0 22600.0 0.38 1188920.0 23800.0 0.43 0.5698 0.998 2144289 PK04_097030 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCCO)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B09 compound treatment 1169720.0 1960.0 0.03 1175240.0 10100.0 0.18 0.1518 0.8215 2141150 PK04_097031 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B10 compound treatment 1165840.0 -1920.0 -0.03 1176480.0 11300.0 0.2 0.1217 0.5887 2144633 PK04_097032 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B11 compound treatment 1163120.0 -4640.0 -0.08 1166800.0 1650.0 0.03 -0.0338 -0.4072 2141161 PK04_097033 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B12 compound treatment 1196640.0 28900.0 0.48 1195840.0 30700.0 0.55 0.7328 0.9978 2144765 PK04_097034 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8ccccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B13 mock treatment 1184080.0 16300.0 0.27 1180040.0 14900.0 0.27 0.3829 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B14 mock treatment 1169840.0 2080.0 0.03 1190240.0 25100.0 0.45 0.3443 0.7594 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B15 compound treatment 1124760.0 -43000.0 -0.72 1146480.0 -18700.0 -0.34 -0.7466 -0.94 2141135 PK04_097035 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B16 compound treatment 1157000.0 -10800.0 -0.18 1166560.0 1410.0 0.03 -0.1093 -0.6013 2144753 PK04_097036 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B17 compound treatment 1113600.0 -54200.0 -0.91 1119920.0 -45200.0 -0.81 -1.2171 -0.9986 2141225 PK04_097037 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B18 compound treatment 1134720.0 -33000.0 -0.55 1132600.0 -32500.0 -0.59 -0.8056 -0.9996 2144045 PK04_097038 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B19 compound treatment 1112960.0 -54800.0 -0.92 1115280.0 -49900.0 -0.9 -1.2838 -0.9999 2141420 PK04_097039 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B20 compound treatment 1147400.0 -20400.0 -0.34 1136680.0 -28500.0 -0.51 -0.6036 -0.9802 2144377 PK04_097040 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B21 compound treatment 1981600.0 814000.0 13.62 1112280.0 -52900.0 -0.95 8.9567 0.656 2141808 PK04_097041 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B22 compound treatment 1126160.0 -41600.0 -0.7 1130000.0 -35100.0 -0.63 -0.94 -0.9989 2143265 PK04_097042 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCNC(=O)N)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B23 compound treatment 1124840.0 -42900.0 -0.72 1124080.0 -41100.0 -0.74 -1.0311 -0.9999 2141931 PK04_097043 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 B24 compound treatment 1150960.0 -16800.0 -0.28 1140800.0 -24300.0 -0.44 -0.509 -0.9769 2142705 PK04_097044 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C01 compound treatment 1163000.0 -4760.0 -0.08 1150360.0 -14800.0 -0.27 -0.2447 -0.8799 2141223 PK04_097045 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C02 compound treatment 1135840.0 -31900.0 -0.53 1153880.0 -11300.0 -0.2 -0.5213 -0.9122 2141108 PK04_097046 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C03 compound treatment 1189280.0 21500.0 0.36 1177520.0 12400.0 0.22 0.4123 0.9734 2141329 PK04_097047 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C04 compound treatment 1198320.0 30600.0 0.51 1183600.0 18500.0 0.33 0.5967 0.9782 2141703 PK04_097048 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C05 compound treatment 1075160.0 -92600.0 -1.55 1076160.0 -89000.0 -1.6 -2.2294 -0.9999 2065845 PK04_097049 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C06 compound treatment 1165120.0 -2640.0 -0.04 1152520.0 -12600.0 -0.23 -0.1921 -0.8288 2141782 PK04_097050 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C07 compound treatment 1027840.0 -140000.0 -2.34 1037640.0 -128000.0 -2.3 -3.2801 -1.0 2141574 PK04_097051 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C08 compound treatment 1159880.0 -7880.0 -0.13 1150240.0 -14900.0 -0.27 -0.2832 -0.9463 2141856 PK04_097052 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C09 compound treatment 1140560.0 -27200.0 -0.46 1138440.0 -26700.0 -0.48 -0.6621 -0.9996 2141751 PK04_097053 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C10 compound treatment 1163840.0 -3920.0 -0.07 1162320.0 -2830.0 -0.05 -0.0824 -0.9923 2141441 PK04_097054 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C11 mock treatment 1181640.0 13900.0 0.23 1170680.0 5530.0 0.1 0.2347 0.9286 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C12 mock treatment 1184280.0 16500.0 0.28 1175160.0 10000.0 0.18 0.3231 0.9786 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C13 compound treatment 1149040.0 -18700.0 -0.31 1131720.0 -33400.0 -0.6 -0.6474 -0.9536 2141937 PK04_097055 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C14 compound treatment 1146960.0 -20800.0 -0.35 1152120.0 -13000.0 -0.23 -0.4121 -0.9816 2141727 PK04_097056 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C15 mock treatment 1159280.0 -8480.0 -0.14 1158560.0 -6590.0 -0.12 -0.1843 -0.9961 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C16 mock treatment 1162160.0 -5600.0 -0.09 1157480.0 -7670.0 -0.14 -0.1639 -0.9821 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C17 compound treatment 1100520.0 -67200.0 -1.13 1105800.0 -59300.0 -1.07 -1.5517 -0.9997 2141078 PK04_097057 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C18 compound treatment 1145560.0 -22200.0 -0.37 1153680.0 -11500.0 -0.21 -0.4088 -0.9617 2141467 PK04_097058 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C19 compound treatment 1126160.0 -41600.0 -0.7 1135480.0 -29700.0 -0.53 -0.8702 -0.9915 2141339 PK04_097059 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C20 compound treatment 1127320.0 -40400.0 -0.68 1138280.0 -26900.0 -0.48 -0.8208 -0.9865 2141364 PK04_097060 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C21 compound treatment 1132440.0 -35300.0 -0.59 1127240.0 -37900.0 -0.68 -0.9009 -0.9974 2141370 PK04_097061 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C22 compound treatment 1111120.0 -56600.0 -0.95 1131440.0 -33700.0 -0.61 -1.0997 -0.9769 2141489 PK04_097062 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(O)cc5)[C@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C23 compound treatment 1123480.0 -44300.0 -0.74 1116800.0 -48300.0 -0.87 -1.1399 -0.9968 2141706 PK04_097063 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 C24 compound treatment 1129720.0 -38000.0 -0.64 1124400.0 -40700.0 -0.73 -0.9692 -0.9975 2141172 PK04_097064 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D01 compound treatment 1204000.0 36200.0 0.61 1214040.0 48900.0 0.88 1.0517 0.9834 2141788 PK04_097065 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D02 compound treatment 1224320.0 56600.0 0.95 1209520.0 44400.0 0.8 1.2346 0.9965 2143973 PK04_097066 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCCO)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D03 compound treatment 1162360.0 -5400.0 -0.09 1163040.0 -2110.0 -0.04 -0.0907 -0.926 2141854 PK04_097067 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D04 compound treatment 1107280.0 -60500.0 -1.01 1121960.0 -43200.0 -0.78 -1.2659 -0.9916 2141969 PK04_097068 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D05 compound treatment 1116840.0 -50900.0 -0.85 1132840.0 -32300.0 -0.58 -1.0141 -0.9827 2141087 PK04_097069 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D06 compound treatment 1040400.0 -127000.0 -2.13 1049160.0 -116000.0 -2.09 -2.9847 -1.0 2144657 PK04_097070 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9ccccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D07 compound treatment 1164200.0 -3560.0 -0.06 1176560.0 11400.0 0.21 0.1033 0.4825 2141768 PK04_097071 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D08 compound treatment 1172640.0 4880.0 0.08 1165000.0 -149.0 0.0 0.0559 0.6835 2144733 PK04_097072 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D09 compound treatment 1040240.0 -128000.0 -2.13 1064280.0 -101000.0 -1.82 -2.794 -0.9968 2141552 PK04_097073 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D10 compound treatment 1168960.0 1200.0 0.02 1167560.0 2410.0 0.04 0.0449 0.9388 2143885 PK04_097074 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#Cc8ccc(OC)cc8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D11 mock treatment 1177160.0 9400.0 0.16 1160840.0 -4310.0 -0.08 0.0564 0.3212 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D12 mock treatment 1159400.0 -8360.0 -0.14 1176520.0 11400.0 0.2 0.046 0.1853 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D13 compound treatment 1139640.0 -28100.0 -0.47 1124480.0 -40700.0 -0.73 -0.8508 -0.9771 2141513 PK04_097075 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D14 compound treatment 1096120.0 -71600.0 -1.2 1114040.0 -51100.0 -0.92 -1.4988 -0.9915 2144449 PK04_097076 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D15 mock treatment 1140720.0 -27000.0 -0.45 1150080.0 -15100.0 -0.27 -0.5119 -0.9702 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D16 mock treatment 1146480.0 -21300.0 -0.36 1148640.0 -16500.0 -0.3 -0.4621 -0.996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D17 compound treatment 1114560.0 -53200.0 -0.89 1115160.0 -50000.0 -0.9 -1.2664 -1.0 2141816 PK04_097077 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D18 compound treatment 1108840.0 -58900.0 -0.99 1123080.0 -42100.0 -0.76 -1.2331 -0.9916 2142085 PK04_097078 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D19 compound treatment 1110640.0 -57100.0 -0.96 1106040.0 -59100.0 -1.06 -1.4289 -0.9985 2141432 PK04_097079 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D20 compound treatment 1089960.0 -77800.0 -1.3 1099640.0 -65500.0 -1.18 -1.7552 -0.9988 2144825 PK04_097080 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D21 compound treatment 948960.0 -219000.0 -3.66 961760.0 -203000.0 -3.66 -5.1802 -1.0 2141123 PK04_097081 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)O)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D22 compound treatment 1111160.0 -56600.0 -0.95 1119840.0 -45300.0 -0.82 -1.247 -0.9973 2144893 PK04_097082 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D23 compound treatment 1108840.0 -58900.0 -0.99 1120280.0 -44900.0 -0.81 -1.2688 -0.9951 2141421 PK04_097083 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 D24 compound treatment 1116520.0 -51200.0 -0.86 1105280.0 -59900.0 -1.08 -1.369 -0.9935 2143085 PK04_097084 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E01 mock treatment 1208720.0 41000.0 0.69 1178000.0 12900.0 0.23 0.6484 0.8962 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E02 mock treatment 1197280.0 29500.0 0.49 1179200.0 14100.0 0.25 0.5284 0.9518 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E03 compound treatment 1192480.0 24700.0 0.41 1177920.0 12800.0 0.23 0.4552 0.9617 2141878 PK04_097085 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E04 compound treatment 1142840.0 -24900.0 -0.42 1153960.0 -11200.0 -0.2 -0.4374 -0.9444 2141520 PK04_097086 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E05 compound treatment 1188760.0 21000.0 0.35 1194320.0 29200.0 0.53 0.6202 0.9809 2141359 PK04_097087 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E06 compound treatment 1125680.0 -42100.0 -0.7 1134000.0 -31100.0 -0.56 -0.8947 -0.9937 2141507 PK04_097088 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E07 compound treatment 1114920.0 -52800.0 -0.88 1116320.0 -48800.0 -0.88 -1.2473 -1.0 2141863 PK04_097089 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccccc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E08 compound treatment 1162600.0 -5160.0 -0.09 1150040.0 -15100.0 -0.27 -0.2535 -0.8877 2141163 PK04_097090 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E09 mock treatment 1176440.0 8680.0 0.15 1175080.0 9930.0 0.18 0.2293 0.9947 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E10 mock treatment 1183800.0 16000.0 0.27 1164160.0 -989.0 -0.02 0.1772 0.6587 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E11 compound treatment 1160560.0 -7200.0 -0.12 1167960.0 2810.0 0.05 -0.0494 -0.3777 2141456 PK04_097091 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E12 compound treatment 1141800.0 -26000.0 -0.43 1131800.0 -33300.0 -0.6 -0.732 -0.9873 2141683 PK04_097092 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E13 compound treatment 1164400.0 -3360.0 -0.06 1148240.0 -16900.0 -0.3 -0.2552 -0.8236 2141357 PK04_097093 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@@H]([C@@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E14 compound treatment 1150760.0 -17000.0 -0.28 1166360.0 1210.0 0.02 -0.1857 -0.651 2141366 PK04_097094 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E15 compound treatment 1097680.0 -70100.0 -1.17 1097800.0 -67300.0 -1.21 -1.6873 -0.9999 2141575 PK04_097095 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E16 compound treatment 1137600.0 -30200.0 -0.5 1131600.0 -33500.0 -0.6 -0.7843 -0.996 2141485 PK04_097096 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E17 mock treatment 1145600.0 -22200.0 -0.37 1137840.0 -27300.0 -0.49 -0.6101 -0.9903 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E18 mock treatment 1151600.0 -16200.0 -0.27 1146360.0 -18800.0 -0.34 -0.4306 -0.9938 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E19 compound treatment 1119280.0 -48500.0 -0.81 1101000.0 -64100.0 -1.16 -1.3909 -0.985 2141377 PK04_097097 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E20 compound treatment 1117280.0 -50500.0 -0.84 1129320.0 -35800.0 -0.65 -1.0538 -0.9912 2141326 PK04_097098 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E21 compound treatment 1114600.0 -53200.0 -0.89 1108920.0 -56200.0 -1.01 -1.3454 -0.9979 2141702 PK04_097099 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E22 compound treatment 1135040.0 -32700.0 -0.55 1130000.0 -35100.0 -0.63 -0.835 -0.9974 2141417 PK04_097100 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E23 compound treatment 1077800.0 -90000.0 -1.51 1079720.0 -85400.0 -1.54 -2.1528 -0.9999 2141167 PK04_097101 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 E24 compound treatment 921760.0 -246000.0 -4.12 933880.0 -231000.0 -4.17 -5.8573 -1.0 2141113 PK04_097102 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F01 mock treatment 1227240.0 59500.0 1.0 1216560.0 51400.0 0.93 1.3588 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F02 mock treatment 1212040.0 44300.0 0.74 1211480.0 46300.0 0.83 1.1143 0.9982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F03 compound treatment 1170560.0 2800.0 0.05 1170240.0 5090.0 0.09 0.098 0.9515 2141216 PK04_097103 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F04 compound treatment 1178720.0 11000.0 0.18 1185080.0 19900.0 0.36 0.3836 0.9514 2142933 PK04_097104 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F05 compound treatment 1178040.0 10300.0 0.17 1176760.0 11600.0 0.21 0.2696 0.9953 2141355 PK04_097105 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F06 compound treatment 1152400.0 -15400.0 -0.26 1162120.0 -3030.0 -0.05 -0.2203 -0.8386 2142833 PK04_097106 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F07 compound treatment 1168920.0 1160.0 0.02 1176080.0 10900.0 0.2 0.153 0.7732 2141414 PK04_097107 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F08 compound treatment 1154440.0 -13300.0 -0.22 1136840.0 -28300.0 -0.51 -0.5182 -0.9311 2144249 PK04_097108 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F09 mock treatment 1176800.0 9040.0 0.15 1172920.0 7770.0 0.14 0.206 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F10 mock treatment 1173720.0 5960.0 0.1 1171240.0 6090.0 0.11 0.1482 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F11 compound treatment 1136960.0 -30800.0 -0.52 1130480.0 -34700.0 -0.62 -0.8061 -0.9954 2141568 PK04_097109 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F12 compound treatment 1127360.0 -40400.0 -0.68 1129880.0 -35300.0 -0.64 -0.9274 -0.9995 2142765 PK04_097110 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F13 compound treatment 1142120.0 -25600.0 -0.43 1156640.0 -8510.0 -0.15 -0.4118 -0.9038 2141348 PK04_097111 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F14 compound treatment 1135560.0 -32200.0 -0.54 1126960.0 -38200.0 -0.69 -0.8675 -0.9927 2142645 PK04_097112 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F15 compound treatment 1098320.0 -69400.0 -1.16 1105840.0 -59300.0 -1.07 -1.5773 -0.9991 2141505 PK04_097113 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F16 compound treatment 1131440.0 -36300.0 -0.61 1085440.0 -79700.0 -1.44 -1.4452 -0.9268 2142977 PK04_097114 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCNC(=O)N)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F17 mock treatment 1123200.0 -44600.0 -0.75 1128440.0 -36700.0 -0.66 -0.9949 -0.9982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F18 mock treatment 1139520.0 -28200.0 -0.47 1138320.0 -26800.0 -0.48 -0.6759 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F19 compound treatment 1049240.0 -119000.0 -1.98 1071320.0 -93800.0 -1.69 -2.5978 -0.9968 2141200 PK04_097115 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F20 compound treatment 1089400.0 -78400.0 -1.31 1098920.0 -66200.0 -1.19 -1.771 -0.9989 2142045 PK04_097116 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F21 compound treatment 1107920.0 -59800.0 -1.0 1118480.0 -46700.0 -0.84 -1.3026 -0.9962 2141938 PK04_097117 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F22 compound treatment 1109000.0 -58800.0 -0.98 1105040.0 -60100.0 -1.08 -1.4611 -0.9988 2144373 PK04_097118 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F23 compound treatment 1109080.0 -58700.0 -0.98 1106800.0 -58300.0 -1.05 -1.4377 -0.9994 2141419 PK04_097119 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 F24 compound treatment 1068840.0 -98900.0 -1.66 1058480.0 -107000.0 -1.92 -2.5295 -0.9972 2142769 PK04_097120 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G01 compound treatment 1140240.0 -27500.0 -0.46 1135800.0 -29300.0 -0.53 -0.6995 -0.9976 2141178 PK04_097121 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G02 compound treatment 1198200.0 30400.0 0.51 1195360.0 30200.0 0.54 0.7451 0.9995 2141487 PK04_097122 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G03 mock treatment 1204440.0 36700.0 0.61 1199160.0 34000.0 0.61 0.8674 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G04 mock treatment 1204680.0 36900.0 0.62 1204560.0 39400.0 0.71 0.939 0.9976 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G05 compound treatment 1099280.0 -68500.0 -1.15 1075240.0 -89900.0 -1.62 -1.9557 -0.9856 2141519 PK04_097123 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G06 compound treatment 1169840.0 2080.0 0.03 1165960.0 811.0 0.01 0.035 0.9255 2141537 PK04_097124 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G07 compound treatment 1168200.0 443.0 0.01 1173160.0 8010.0 0.14 0.1073 0.7424 2141722 PK04_097125 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G08 compound treatment 1141280.0 -26500.0 -0.44 1130920.0 -34200.0 -0.62 -0.7494 -0.9868 2141577 PK04_097126 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G09 compound treatment 1182520.0 14800.0 0.25 1186880.0 21700.0 0.39 0.4515 0.9753 2141458 PK04_097127 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G10 compound treatment 1166080.0 -1680.0 -0.03 1151400.0 -13700.0 -0.25 -0.195 -0.7822 2141190 PK04_097128 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G11 compound treatment 1154760.0 -13000.0 -0.22 1151240.0 -13900.0 -0.25 -0.331 -0.9975 2141333 PK04_097129 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G12 compound treatment 1021680.0 -146000.0 -2.44 1023400.0 -142000.0 -2.55 -3.5344 -0.9998 2141508 PK04_097130 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G13 compound treatment 1149160.0 -18600.0 -0.31 1146160.0 -19000.0 -0.34 -0.462 -0.9989 2141118 PK04_097131 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G14 compound treatment 1153680.0 -14100.0 -0.24 1164080.0 -1070.0 -0.02 -0.1802 -0.7624 2141927 PK04_097132 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G15 compound treatment 1121200.0 -46600.0 -0.78 1136000.0 -29100.0 -0.53 -0.9223 -0.9816 2141159 PK04_097133 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G16 compound treatment 1143440.0 -24300.0 -0.41 1146560.0 -18600.0 -0.33 -0.5246 -0.9953 2141713 PK04_097134 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G17 compound treatment 1135720.0 -32000.0 -0.54 1152640.0 -12500.0 -0.23 -0.5385 -0.9259 2141795 PK04_097135 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G18 compound treatment 1117160.0 -50600.0 -0.85 1117680.0 -47500.0 -0.86 -1.2035 -1.0 2141553 PK04_097136 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G19 mock treatment 1143920.0 -23800.0 -0.4 1144720.0 -20400.0 -0.37 -0.5423 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G20 mock treatment 1134520.0 -33200.0 -0.56 1144560.0 -20600.0 -0.37 -0.6556 -0.9806 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G21 compound treatment 1133240.0 -34500.0 -0.58 1134560.0 -30600.0 -0.55 -0.7982 -0.9997 2141819 PK04_097137 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G22 compound treatment 1090600.0 -77200.0 -1.29 1087440.0 -77700.0 -1.4 -1.903 -0.9992 2141516 PK04_097138 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G23 compound treatment 1125080.0 -42700.0 -0.71 1127560.0 -37600.0 -0.68 -0.9839 -0.9996 2141691 PK04_097139 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 G24 compound treatment 1099960.0 -67800.0 -1.13 1111000.0 -54100.0 -0.98 -1.4921 -0.9972 2141155 PK04_097140 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H01 compound treatment 1197600.0 29800.0 0.5 1193360.0 28200.0 0.51 0.7125 1.0 2141157 PK04_097141 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H02 compound treatment 1210920.0 43200.0 0.72 1206720.0 41600.0 0.75 1.0404 0.9998 2143037 PK04_097142 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCC(C(=O)OC)C(=O)OC)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H03 mock treatment 1198760.0 31000.0 0.52 1207240.0 42100.0 0.76 0.9031 0.9829 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H04 mock treatment 1195680.0 27900.0 0.47 1207160.0 42000.0 0.76 0.8656 0.9731 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H05 compound treatment 1183760.0 16000.0 0.27 1180800.0 15700.0 0.28 0.3888 0.9997 2141926 PK04_097143 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H06 compound treatment 1172760.0 5000.0 0.08 1163400.0 -1750.0 -0.03 0.0369 0.4127 2143177 PK04_097144 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H07 compound treatment 1175920.0 8160.0 0.14 1170960.0 5810.0 0.1 0.1706 0.9914 2141694 PK04_097145 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H08 compound treatment 1190800.0 23000.0 0.39 1168480.0 3330.0 0.06 0.3151 0.8074 2143025 PK04_097146 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H09 compound treatment 1147840.0 -19900.0 -0.33 1142880.0 -22300.0 -0.4 -0.5194 -0.9958 2141749 PK04_097147 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H10 compound treatment 1161760.0 -6000.0 -0.1 1170640.0 5490.0 0.1 -0.001 -0.0072 2143077 PK04_097148 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H11 compound treatment 887720.0 -280000.0 -4.69 907920.0 -257000.0 -4.63 -6.5908 -1.0 2141097 PK04_097149 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H12 compound treatment 1137880.0 -29900.0 -0.5 1148600.0 -16500.0 -0.3 -0.5644 -0.9695 2142913 PK04_097150 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#Cc9ccc(OC)cc9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H13 compound treatment 1133080.0 -34700.0 -0.58 1121760.0 -43400.0 -0.78 -0.9631 -0.9892 2141401 PK04_097151 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H14 compound treatment 1150720.0 -17000.0 -0.29 1144040.0 -21100.0 -0.38 -0.4705 -0.9899 2143093 PK04_097152 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H15 compound treatment 1127040.0 -40700.0 -0.68 1132680.0 -32500.0 -0.59 -0.8955 -0.9971 2141777 PK04_097153 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H16 compound treatment 1139200.0 -28600.0 -0.48 1131960.0 -33200.0 -0.6 -0.7608 -0.9938 2143865 PK04_097154 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H17 compound treatment 1108000.0 -59800.0 -1.0 1103200.0 -61900.0 -1.12 -1.4964 -0.9985 2141142 PK04_097155 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H18 compound treatment 1116920.0 -50800.0 -0.85 1128640.0 -36500.0 -0.66 -1.0667 -0.9919 2143925 PK04_097156 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCNC(=O)N)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H19 mock treatment 1135280.0 -32500.0 -0.54 1141520.0 -23600.0 -0.43 -0.6853 -0.9927 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H20 mock treatment 1132360.0 -35400.0 -0.59 1109400.0 -55700.0 -1.0 -1.1291 -0.9683 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H21 compound treatment 1117920.0 -49800.0 -0.83 1106720.0 -58400.0 -1.05 -1.3341 -0.9933 2141168 PK04_097157 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H22 compound treatment 1132640.0 -35100.0 -0.59 1115040.0 -50100.0 -0.9 -1.0539 -0.9784 2143057 PK04_097158 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H23 compound treatment 1108200.0 -59600.0 -1.0 1108160.0 -57000.0 -1.03 -1.4308 -0.9999 2141804 PK04_097159 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 H24 compound treatment 1094480.0 -73300.0 -1.23 1086640.0 -78500.0 -1.41 -1.8673 -0.9975 2142649 PK04_097160 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I01 compound treatment 1197400.0 29600.0 0.5 1201000.0 35900.0 0.65 0.8075 0.9915 2141890 PK04_097161 O[C@@H](CNC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I02 compound treatment 1215720.0 48000.0 0.8 1202280.0 37100.0 0.67 1.0406 0.9959 2141465 PK04_097162 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I03 compound treatment 1169720.0 1960.0 0.03 1168160.0 3010.0 0.05 0.0616 0.9711 2141772 PK04_097163 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I04 compound treatment 1190640.0 22900.0 0.38 1167600.0 2450.0 0.04 0.302 0.7835 2141343 PK04_097164 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I05 mock treatment 1214800.0 47000.0 0.79 1191880.0 26700.0 0.48 0.8972 0.9722 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I06 mock treatment 1188520.0 20800.0 0.35 1189800.0 24700.0 0.44 0.5597 0.9926 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I07 compound treatment 1188920.0 21200.0 0.35 1161000.0 -4150.0 -0.07 0.1976 0.5458 2141794 PK04_097165 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I08 compound treatment 1190080.0 22300.0 0.37 1182920.0 17800.0 0.32 0.4905 0.9971 2141922 PK04_097166 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I09 compound treatment 1167960.0 203.0 0.0 1163880.0 -1270.0 -0.02 -0.0138 -0.5958 2141780 PK04_097167 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I10 compound treatment 1183080.0 15300.0 0.26 1142400.0 -22700.0 -0.41 -0.1085 -0.2244 2141799 PK04_097168 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I11 compound treatment 1123320.0 -44400.0 -0.74 1124280.0 -40900.0 -0.74 -1.0465 -1.0 2141177 PK04_097169 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I12 compound treatment 1128080.0 -39700.0 -0.66 1142520.0 -22600.0 -0.41 -0.7578 -0.9726 2141747 PK04_097170 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I13 compound treatment 1136200.0 -31600.0 -0.53 1131840.0 -33300.0 -0.6 -0.7978 -0.998 2141423 PK04_097171 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I14 compound treatment 1143080.0 -24700.0 -0.41 1131880.0 -33300.0 -0.6 -0.7159 -0.9835 2141775 PK04_097172 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I15 compound treatment 1100880.0 -66900.0 -1.12 1084000.0 -81100.0 -1.46 -1.8252 -0.9913 2141538 PK04_097173 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I16 compound treatment 1044520.0 -123000.0 -2.06 1063560.0 -102000.0 -1.83 -2.7525 -0.9982 2065871 PK04_097174 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)O)[C@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I17 compound treatment 1129840.0 -37900.0 -0.63 1127760.0 -37400.0 -0.67 -0.925 -0.9996 2141729 PK04_097175 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I18 compound treatment 1135240.0 -32500.0 -0.54 1133040.0 -32100.0 -0.58 -0.7939 -0.9995 2141892 PK04_097176 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccccc54)[C@@H]([C@@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I19 compound treatment 1131120.0 -36600.0 -0.61 1132360.0 -32800.0 -0.59 -0.8513 -0.9998 2141687 PK04_097177 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I20 compound treatment 1132160.0 -35600.0 -0.6 1121280.0 -43900.0 -0.79 -0.9801 -0.9903 2141680 PK04_097178 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I21 mock treatment 1149440.0 -18300.0 -0.31 1129400.0 -35700.0 -0.64 -0.6722 -0.9424 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I22 mock treatment 1139960.0 -27800.0 -0.47 1137680.0 -27500.0 -0.49 -0.6789 -0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I23 compound treatment 1112120.0 -55600.0 -0.93 1112480.0 -52700.0 -0.95 -1.3294 -1.0 2141841 PK04_097179 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 I24 compound treatment 1127560.0 -40200.0 -0.67 1126480.0 -38700.0 -0.7 -0.9683 -0.9998 2141766 PK04_097180 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NCC=C)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J01 compound treatment 1210840.0 43100.0 0.72 1203600.0 38500.0 0.69 0.9997 0.9998 2141705 PK04_097181 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccccc3OCCO)[C@@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J02 compound treatment 1189520.0 21800.0 0.36 1186600.0 21500.0 0.39 0.5308 0.9996 2143397 PK04_097182 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9(O)CCCCCC9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J03 compound treatment 1189120.0 21400.0 0.36 1182200.0 17100.0 0.31 0.47 0.9972 2141179 PK04_097183 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J04 compound treatment 1204760.0 37000.0 0.62 1209800.0 44700.0 0.8 1.0067 0.9916 2144337 PK04_097184 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J05 mock treatment 1206840.0 39100.0 0.65 1179080.0 13900.0 0.25 0.6399 0.9135 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J06 mock treatment 1206920.0 39200.0 0.66 1193800.0 28700.0 0.52 0.8284 0.993 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J07 compound treatment 1177080.0 9320.0 0.16 1189160.0 24000.0 0.43 0.4162 0.9051 2141805 PK04_097185 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J08 compound treatment 1149560.0 -18200.0 -0.3 1149920.0 -15200.0 -0.27 -0.4094 -0.9986 2143365 PK04_097186 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J09 compound treatment 1145360.0 -22400.0 -0.37 1138120.0 -27000.0 -0.49 -0.6094 -0.9916 2141901 PK04_097187 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J10 compound treatment 1174440.0 6680.0 0.11 1169200.0 4050.0 0.07 0.1307 0.9786 2144881 PK04_097188 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8ccccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J11 compound treatment 1157480.0 -10300.0 -0.17 1151720.0 -13400.0 -0.24 -0.2927 -0.986 2141717 PK04_097189 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J12 compound treatment 1134160.0 -33600.0 -0.56 1115680.0 -49500.0 -0.89 -1.0278 -0.9753 2143405 PK04_097190 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J13 compound treatment 1100400.0 -67400.0 -1.13 1119200.0 -45900.0 -0.83 -1.3824 -0.9885 2141188 PK04_097191 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J14 compound treatment 1130200.0 -37600.0 -0.63 1129840.0 -35300.0 -0.64 -0.8943 -1.0 2142929 PK04_097192 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#Cc%10ccc(OC)cc%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J15 compound treatment 1114360.0 -53400.0 -0.89 1119720.0 -45400.0 -0.82 -1.2106 -0.999 2141365 PK04_097193 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J16 compound treatment 1127920.0 -39800.0 -0.67 1133200.0 -31900.0 -0.58 -0.8784 -0.9973 2144325 PK04_097194 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J17 compound treatment 1096160.0 -71600.0 -1.2 1104720.0 -60400.0 -1.09 -1.6171 -0.9989 2141221 PK04_097195 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(OCCO)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J18 compound treatment 1126320.0 -41400.0 -0.69 1105520.0 -59600.0 -1.07 -1.25 -0.9776 2143377 PK04_097196 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J19 compound treatment 1131360.0 -36400.0 -0.61 1130720.0 -34400.0 -0.62 -0.8693 -1.0 2141815 PK04_097197 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(O)cc3)[C@@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@H]([C@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J20 compound treatment 1142040.0 -25700.0 -0.43 1106840.0 -58300.0 -1.05 -1.0472 -0.9224 2142585 PK04_097198 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#Cc8ccc(OC)cc8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J21 mock treatment 1132120.0 -35600.0 -0.6 1128000.0 -37100.0 -0.67 -0.895 -0.9983 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J22 mock treatment 1140120.0 -27600.0 -0.46 1147440.0 -17700.0 -0.32 -0.5527 -0.9836 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J23 compound treatment 1103640.0 -64100.0 -1.07 1093800.0 -71300.0 -1.29 -1.6677 -0.996 2141186 PK04_097199 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 J24 compound treatment 1126560.0 -41200.0 -0.69 1087040.0 -78100.0 -1.41 -1.4826 -0.9461 2144237 PK04_097200 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CCNC(=O)N)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K01 compound treatment 1189480.0 21700.0 0.36 1177080.0 11900.0 0.21 0.409 0.9686 2141164 PK04_097201 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K02 compound treatment 1191000.0 23200.0 0.39 1203560.0 38400.0 0.69 0.7644 0.9629 2141443 PK04_097202 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K03 compound treatment 1176560.0 8800.0 0.15 1185080.0 19900.0 0.36 0.3581 0.9226 2141548 PK04_097203 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K04 compound treatment 1212440.0 44700.0 0.75 1187080.0 21900.0 0.4 0.8081 0.9556 2141351 PK04_097204 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K05 compound treatment 1196240.0 28500.0 0.48 1193320.0 28200.0 0.51 0.6959 0.9995 2141786 PK04_097205 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(O)cc5)[C@@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K06 compound treatment 1184240.0 16500.0 0.28 1182000.0 16900.0 0.3 0.4097 0.9989 2141746 PK04_097206 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K07 mock treatment 1194920.0 27200.0 0.45 1190120.0 25000.0 0.45 0.6395 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K08 mock treatment 1189720.0 22000.0 0.37 1189640.0 24500.0 0.44 0.5719 0.9959 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K09 compound treatment 1176280.0 8520.0 0.14 1173320.0 8170.0 0.15 0.2049 0.9999 2141350 PK04_097207 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K10 compound treatment 1162000.0 -5760.0 -0.1 1164280.0 -869.0 -0.02 -0.0792 -0.8114 2141331 PK04_097208 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccccc6OCCO)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K11 compound treatment 1162480.0 -5280.0 -0.09 1156080.0 -9070.0 -0.16 -0.178 -0.9583 2141806 PK04_097209 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K12 compound treatment 1165760.0 -2000.0 -0.03 1156520.0 -8630.0 -0.16 -0.1336 -0.8399 2141720 PK04_097210 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K13 compound treatment 972400.0 -195000.0 -3.27 1017160.0 -148000.0 -2.67 -4.1971 -0.9949 2141904 PK04_097211 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccccc76)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K14 compound treatment 1047360.0 -120000.0 -2.01 1069880.0 -95300.0 -1.72 -2.6384 -0.9968 2141222 PK04_097212 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K15 mock treatment 1159640.0 -8120.0 -0.14 1153880.0 -11300.0 -0.2 -0.2396 -0.9809 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K16 mock treatment 1153560.0 -14200.0 -0.24 1160800.0 -4350.0 -0.08 -0.2234 -0.893 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K17 compound treatment 1149200.0 -18600.0 -0.31 1153040.0 -12100.0 -0.22 -0.3739 -0.9851 2141773 PK04_097213 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K18 compound treatment 1126400.0 -41400.0 -0.69 1129200.0 -35900.0 -0.65 -0.9474 -0.9995 2141524 PK04_097214 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K19 compound treatment 1112600.0 -55200.0 -0.92 1127520.0 -37600.0 -0.68 -1.1321 -0.9885 2141218 PK04_097215 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K20 compound treatment 1097440.0 -70300.0 -1.18 1120360.0 -44800.0 -0.81 -1.4027 -0.9831 2141861 PK04_097216 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K21 compound treatment 1125280.0 -42500.0 -0.71 1111960.0 -53200.0 -0.96 -1.1803 -0.9892 2141117 PK04_097217 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K22 compound treatment 1130680.0 -37100.0 -0.62 1138480.0 -26700.0 -0.48 -0.7785 -0.992 2141354 PK04_097218 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CCCO)cc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K23 mock treatment 1146920.0 -20800.0 -0.35 1144400.0 -20700.0 -0.37 -0.5109 -0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 K24 mock treatment 1122000.0 -45800.0 -0.77 1131880.0 -33300.0 -0.6 -0.9653 -0.9927 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L01 compound treatment 1148240.0 -19500.0 -0.33 1154720.0 -10400.0 -0.19 -0.3638 -0.9655 2141684 PK04_097219 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L02 compound treatment 939960.0 -228000.0 -3.81 960960.0 -204000.0 -3.68 -5.2969 -0.9998 2143489 PK04_097220 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10=CCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L03 compound treatment 1195760.0 28000.0 0.47 1183680.0 18500.0 0.33 0.5674 0.9862 2141375 PK04_097221 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccccc3OCCO)[C@]14C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L04 compound treatment 1170760.0 3000.0 0.05 1181360.0 16200.0 0.29 0.2421 0.8168 2143313 PK04_097222 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L05 compound treatment 1220520.0 52800.0 0.88 1197720.0 32600.0 0.59 1.0393 0.9803 2141889 PK04_097223 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L06 compound treatment 1177440.0 9680.0 0.16 1184440.0 19300.0 0.35 0.3603 0.9397 2144793 PK04_097224 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L07 mock treatment 1187320.0 19600.0 0.33 1190040.0 24900.0 0.45 0.5486 0.988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L08 mock treatment 1178520.0 10800.0 0.18 1182680.0 17500.0 0.32 0.3507 0.9645 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L09 compound treatment 1176680.0 8920.0 0.15 1163520.0 -1630.0 -0.03 0.0848 0.5574 2141438 PK04_097225 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L10 compound treatment 1162880.0 -4880.0 -0.08 1155640.0 -9510.0 -0.17 -0.1789 -0.9425 2142993 PK04_097226 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L11 compound treatment 1137360.0 -30400.0 -0.51 1146640.0 -18500.0 -0.33 -0.5955 -0.979 2141185 PK04_097227 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L12 compound treatment 1127920.0 -39800.0 -0.67 1132440.0 -32700.0 -0.59 -0.8881 -0.9981 2144653 PK04_097228 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L13 compound treatment 1103240.0 -64500.0 -1.08 1138960.0 -26200.0 -0.47 -1.0971 -0.9311 2141893 PK04_097229 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L14 compound treatment 1120800.0 -47000.0 -0.79 1124560.0 -40600.0 -0.73 -1.0728 -0.9994 2143417 PK04_097230 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L15 mock treatment 1145560.0 -22200.0 -0.37 1143680.0 -21500.0 -0.39 -0.5362 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L16 mock treatment 1142320.0 -25400.0 -0.43 1141880.0 -23300.0 -0.42 -0.5975 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L17 compound treatment 1121000.0 -46800.0 -0.78 1129920.0 -35200.0 -0.63 -1.0021 -0.9946 2141152 PK04_097231 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L18 compound treatment 1116600.0 -51200.0 -0.86 1120960.0 -44200.0 -0.8 -1.1683 -0.9993 2143325 PK04_097232 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CCCO)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L19 compound treatment 1127000.0 -40800.0 -0.68 1141400.0 -23700.0 -0.43 -0.7849 -0.9748 2141709 PK04_097233 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CCCO)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L20 compound treatment 1121800.0 -46000.0 -0.77 1126400.0 -38700.0 -0.7 -1.0375 -0.9988 2142773 PK04_097234 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L21 compound treatment 1100440.0 -67300.0 -1.13 1100200.0 -64900.0 -1.17 -1.624 -0.9998 2141174 PK04_097235 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L22 compound treatment 1133280.0 -34500.0 -0.58 1124720.0 -40400.0 -0.73 -0.923 -0.9933 2142985 PK04_097236 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L23 mock treatment 1133200.0 -34600.0 -0.58 1129400.0 -35700.0 -0.64 -0.8644 -0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 L24 mock treatment 1129200.0 -38600.0 -0.65 1136720.0 -28400.0 -0.51 -0.8184 -0.9935 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M01 compound treatment 1180440.0 12700.0 0.21 1163440.0 -1710.0 -0.03 0.1283 0.5983 2141838 PK04_097237 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)Nc4nc5ccccc5s4)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M02 compound treatment 1131840.0 -35900.0 -0.6 1129640.0 -35500.0 -0.64 -0.8774 -0.9995 2141189 PK04_097238 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M03 compound treatment 1208760.0 41000.0 0.69 1208280.0 43100.0 0.78 1.0347 0.9981 2141724 PK04_097239 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M04 compound treatment 1163160.0 -4600.0 -0.08 1163960.0 -1190.0 -0.02 -0.0696 -0.8709 2141153 PK04_097240 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M05 compound treatment 1178720.0 11000.0 0.18 1183280.0 18100.0 0.33 0.3607 0.9628 2141436 PK04_097241 OCCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NCC=C)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M06 compound treatment 1205960.0 38200.0 0.64 1181200.0 16100.0 0.29 0.6565 0.9357 2141769 PK04_097242 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)NC[C@H](O)c9ccccc9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M07 compound treatment 1199440.0 31700.0 0.53 1193360.0 28200.0 0.51 0.7343 0.9998 2141771 PK04_097243 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(O)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M08 compound treatment 1170000.0 2240.0 0.04 1168840.0 3690.0 0.07 0.0736 0.9633 2141480 PK04_097244 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M09 mock treatment 1196440.0 28700.0 0.48 1180880.0 15700.0 0.28 0.5398 0.9684 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M10 mock treatment 1179680.0 11900.0 0.2 1178600.0 13500.0 0.24 0.3124 0.9953 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M11 compound treatment 1101520.0 -66200.0 -1.11 1117000.0 -48100.0 -0.87 -1.3972 -0.9926 2141571 PK04_097245 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M12 compound treatment 1175360.0 7600.0 0.13 1159040.0 -6110.0 -0.11 0.0121 0.0721 2141879 PK04_097246 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccccc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M13 mock treatment 1138400.0 -29400.0 -0.49 1158440.0 -6710.0 -0.12 -0.4329 -0.8556 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M14 mock treatment 1166560.0 -1200.0 -0.02 1163040.0 -2110.0 -0.04 -0.041 -0.9553 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M15 compound treatment 1131000.0 -36800.0 -0.62 1136040.0 -29100.0 -0.52 -0.8058 -0.9969 2141832 PK04_097247 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M16 compound treatment 1102360.0 -65400.0 -1.09 1130360.0 -34800.0 -0.63 -1.2171 -0.965 2141542 PK04_097248 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M17 compound treatment 1114160.0 -53600.0 -0.9 1114320.0 -50800.0 -0.92 -1.2818 -0.9999 2141399 PK04_097249 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M18 compound treatment 1108920.0 -58800.0 -0.98 1113960.0 -51200.0 -0.92 -1.3484 -0.9995 2141903 PK04_097250 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccccc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M19 compound treatment 1132400.0 -35400.0 -0.59 1147880.0 -17300.0 -0.31 -0.6384 -0.955 2141716 PK04_097251 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M20 compound treatment 1121800.0 -46000.0 -0.77 1117920.0 -47200.0 -0.85 -1.1455 -0.9987 2141203 PK04_097252 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccc(OCCO)cc5)[C@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M21 compound treatment 1063280.0 -104000.0 -1.75 1076160.0 -89000.0 -1.6 -2.37 -0.9991 2141110 PK04_097253 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M22 compound treatment 1127680.0 -40100.0 -0.67 1133520.0 -31600.0 -0.57 -0.8772 -0.9967 2141731 PK04_097254 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M23 compound treatment 1049000.0 -119000.0 -1.99 1051240.0 -114000.0 -2.05 -2.8565 -0.9999 2141095 PK04_097255 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CC6(O)CCCCCC6)cc54)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 M24 compound treatment 1113840.0 -53900.0 -0.9 1096440.0 -68700.0 -1.24 -1.5134 -0.9879 2141894 PK04_097256 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N01 compound treatment 1205800.0 38000.0 0.64 1200120.0 35000.0 0.63 0.8957 1.0 2141340 PK04_097257 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N02 compound treatment 1116080.0 -51700.0 -0.86 1118800.0 -46300.0 -0.84 -1.202 -0.9998 2142089 PK04_097258 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N03 compound treatment 1150280.0 -17500.0 -0.29 1158080.0 -7070.0 -0.13 -0.2969 -0.9306 2141511 PK04_097259 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccc(OCCO)cc6)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCc%10cc(OC)c(OC)cc%10C9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N04 compound treatment 1177720.0 9960.0 0.17 1184720.0 19600.0 0.35 0.3672 0.9415 2144305 PK04_097260 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCC(C(=O)OC)C(=O)OC)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N05 compound treatment 1154960.0 -12800.0 -0.21 1176600.0 11500.0 0.21 -0.0055 -0.0187 2141839 PK04_097261 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N06 compound treatment 1136520.0 -31200.0 -0.52 1126960.0 -38200.0 -0.69 -0.8562 -0.9908 2142057 PK04_097262 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N07 compound treatment 1126240.0 -41500.0 -0.69 1087040.0 -78100.0 -1.41 -1.4864 -0.9471 2141431 PK04_097263 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N08 compound treatment 1149760.0 -18000.0 -0.3 1138160.0 -27000.0 -0.49 -0.5568 -0.9735 2144369 PK04_097264 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CC%10(O)CCCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N09 mock treatment 1177760.0 10000.0 0.17 1167200.0 2050.0 0.04 0.1445 0.8429 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N10 mock treatment 1173960.0 6200.0 0.1 1157440.0 -7710.0 -0.14 -0.0248 -0.1431 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N11 compound treatment 1086120.0 -81600.0 -1.37 1082320.0 -82800.0 -1.49 -2.0213 -0.999 2141527 PK04_097265 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N12 compound treatment 1099280.0 -68500.0 -1.15 1106080.0 -59100.0 -1.06 -1.5628 -0.9993 2144009 PK04_097266 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N13 mock treatment 1159280.0 -8480.0 -0.14 1156720.0 -8430.0 -0.15 -0.2077 -0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N14 mock treatment 1138800.0 -29000.0 -0.48 1157880.0 -7270.0 -0.13 -0.4353 -0.8671 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N15 compound treatment 1096000.0 -71800.0 -1.2 1101960.0 -63200.0 -1.14 -1.6541 -0.9996 2141907 PK04_097267 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccccc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N16 compound treatment 1119800.0 -48000.0 -0.8 1125200.0 -39900.0 -0.72 -1.0764 -0.9985 2143157 PK04_097268 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NC[C@H](O)c7ccccc7)c8cc(C#CC9=CCCCC9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N17 compound treatment 1085080.0 -82700.0 -1.38 1093080.0 -72100.0 -1.3 -1.8965 -0.9995 2141544 PK04_097269 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N18 compound treatment 1157960.0 -9800.0 -0.16 1142280.0 -22900.0 -0.41 -0.4073 -0.9184 2144297 PK04_097270 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CCCO)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N19 compound treatment 1108920.0 -58800.0 -0.98 1111480.0 -53700.0 -0.97 -1.38 -1.0 2141483 PK04_097271 O[C@@H](CNC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N20 compound treatment 1067240.0 -101000.0 -1.68 1074040.0 -91100.0 -1.64 -2.3502 -0.9999 2142217 PK04_097272 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9cc(C#CC%10=CCCCC%10)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N21 compound treatment 1097760.0 -70000.0 -1.17 1106640.0 -58500.0 -1.05 -1.5737 -0.9986 2141887 PK04_097273 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NCC=C)[C@@]24C(=O)Nc5ccccc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N22 compound treatment 1125320.0 -42400.0 -0.71 1126800.0 -38300.0 -0.69 -0.9907 -0.9999 2143065 PK04_097274 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(O)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N23 compound treatment 1107400.0 -60400.0 -1.01 1093600.0 -71500.0 -1.29 -1.6258 -0.9927 2141817 PK04_097275 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCN(CC4)c5ncccn5)[C@]26C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)C(=O)O[C@@H]([C@@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 N24 compound treatment 1128080.0 -39700.0 -0.66 1123200.0 -41900.0 -0.76 -1.0039 -0.9979 2144333 PK04_097276 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O01 compound treatment 1180960.0 13200.0 0.22 1159680.0 -5470.0 -0.1 0.0866 0.3578 2141166 PK04_097277 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O02 compound treatment 1165240.0 -2520.0 -0.04 1178200.0 13100.0 0.24 0.1365 0.5713 2141900 PK04_097278 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O03 compound treatment 1197640.0 29900.0 0.5 1186720.0 21600.0 0.39 0.6284 0.9922 2141790 PK04_097279 OCCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(O)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O04 compound treatment 1209040.0 41300.0 0.69 1188040.0 22900.0 0.41 0.7801 0.9696 2141883 PK04_097280 OCCOc1ccccc1[C@@H]2N3[C@H]([C@H](C(=O)N4CCN(CC4)c5ncccn5)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O05 compound treatment 1201240.0 33500.0 0.56 1162560.0 -2590.0 -0.05 0.3632 0.646 2141427 PK04_097281 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O06 compound treatment 1104600.0 -63200.0 -1.06 1089320.0 -75800.0 -1.37 -1.7134 -0.992 2141093 PK04_097282 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)O)[C@@]24C(=O)Nc5ccc(C#CCCO)cc54)C(=O)O[C@H]([C@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O07 compound treatment 1151200.0 -16600.0 -0.28 1180320.0 15200.0 0.27 -0.0026 -0.0068 2141812 PK04_097283 Oc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)N4CCCCCCC4)[C@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@@H]([C@@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O08 compound treatment 1165200.0 -2560.0 -0.04 1150240.0 -14900.0 -0.27 -0.2202 -0.8096 2141430 PK04_097284 NC(=O)NCC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O09 compound treatment 1162960.0 -4800.0 -0.08 1163480.0 -1670.0 -0.03 -0.078 -0.9102 2141454 PK04_097285 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCN(CC8)c9ncccn9)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O10 compound treatment 1089240.0 -78500.0 -1.31 1080600.0 -84500.0 -1.52 -2.0063 -0.9973 2141529 PK04_097286 NC(=O)[C@@H]1[C@@H]2N([C@H](c3ccc(OCCO)cc3)[C@@]14C(=O)Nc5ccc(C#CCCO)cc54)[C@H]([C@H](OC2=O)c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O11 mock treatment 1158000.0 -9760.0 -0.16 1159480.0 -5670.0 -0.1 -0.1877 -0.9745 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O12 mock treatment 1165480.0 -2280.0 -0.04 1148280.0 -16900.0 -0.3 -0.2419 -0.7896 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O13 compound treatment 1161640.0 -6120.0 -0.1 1151840.0 -13300.0 -0.24 -0.2419 -0.928 2141368 PK04_097287 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCc9cc(OC)c(OC)cc9C8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O14 compound treatment 1141680.0 -26100.0 -0.44 1124080.0 -41100.0 -0.74 -0.8318 -0.9683 2141362 PK04_097288 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccccc5OCCO)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)NC[C@H](O)c8ccccc8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O15 compound treatment 1142440.0 -25300.0 -0.42 1142160.0 -23000.0 -0.41 -0.5925 -0.9999 2141460 PK04_097289 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7(O)CCCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O16 compound treatment 785000.0 -383000.0 -6.41 807520.0 -358000.0 -6.44 -9.0854 -1.0 2141860 PK04_097290 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccccc76)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O17 compound treatment 1119680.0 -48100.0 -0.8 1119760.0 -45400.0 -0.82 -1.1472 -1.0 2141175 PK04_097291 OCCOc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)NC[C@H](O)c4ccccc4)[C@@]25C(=O)Nc6ccc(C#CCCO)cc65)C(=O)O[C@H]([C@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O18 compound treatment 1112560.0 -55200.0 -0.92 1111360.0 -53800.0 -0.97 -1.3384 -0.9997 2141486 PK04_097292 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)Nc4nc5ccccc5s4)[C@@]26C(=O)Nc7ccc(C#CC8=CCCCC8)cc76)C(=O)O[C@H]([C@H]3c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O19 compound treatment 1010560.0 -157000.0 -2.63 1009560.0 -156000.0 -2.8 -3.8424 -0.9995 2141156 PK04_097293 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(OCCO)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)Nc9nc%10ccccc%10s9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O20 compound treatment 1114640.0 -53100.0 -0.89 1126720.0 -38400.0 -0.69 -1.1181 -0.9924 2141685 PK04_097294 COc1ccc(C#Cc2ccc3NC(=O)[C@]4([C@@H]([C@@H]5N([C@@H]4c6ccccc6OCCO)[C@H]([C@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCN(CC9)c%10ncccn%10)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O21 compound treatment 1043520.0 -124000.0 -2.08 1039640.0 -126000.0 -2.26 -3.0691 -0.9991 2141094 PK04_097295 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(OCCO)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O22 compound treatment 1120640.0 -47100.0 -0.79 1129000.0 -36100.0 -0.65 -1.0181 -0.9955 2141379 PK04_097296 COc1cc2CCN(Cc2cc1OC)C(=O)[C@H]3[C@H]4N([C@@H](c5ccccc5OCCO)[C@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@@H]([C@@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O23 compound treatment 1070200.0 -97600.0 -1.63 1061040.0 -104000.0 -1.88 -2.4808 -0.9976 2141397 PK04_097297 NC(=O)[C@H]1[C@H]2N([C@@H](c3ccccc3OCCO)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 O24 compound treatment 992920.0 -175000.0 -2.93 1011200.0 -154000.0 -2.77 -4.0302 -0.9996 2065842 PK04_097298 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P01 compound treatment 1192920.0 25200.0 0.42 501680.0 -663000.0 -11.95 -8.1549 -0.6818 2141898 PK04_097299 OCCOc1ccc(cc1)[C@H]2N3[C@@H]([C@@H](C(=O)NCC=C)[C@]24C(=O)Nc5ccccc54)C(=O)O[C@@H]([C@@H]3c6ccccc6)c7ccccc7 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P02 compound treatment 1168720.0 963.0 0.02 294840.0 -870000.0 -15.68 -11.0764 -0.7064 2143305 PK04_097300 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(OCCO)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CCCO)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P03 compound treatment 1137920.0 -29800.0 -0.5 610400.0 -555000.0 -10.0 -7.4206 -0.7415 2141555 PK04_097301 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccc(OCCO)cc5)[C@@]36C(=O)Nc7ccc(C#CC8(O)CCCCCC8)cc76)[C@H]([C@H](OC4=O)c9ccccc9)c%10ccccc%10 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P04 compound treatment 1178120.0 10400.0 0.17 718040.0 -447000.0 -8.06 -5.5736 -0.6917 2144945 PK04_097302 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCc8cc(OC)c(OC)cc8C7)c9ccccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P05 compound treatment 1165960.0 -1800.0 -0.03 306520.0 -859000.0 -15.47 -10.9603 -0.7085 2141923 PK04_097303 OCCOc1ccccc1[C@H]2N3[C@@H]([C@@H](C(=O)NC[C@H](O)c4ccccc4)[C@]25C(=O)Nc6ccccc65)C(=O)O[C@@H]([C@@H]3c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P06 compound treatment 1148480.0 -19300.0 -0.32 727520.0 -438000.0 -7.88 -5.8035 -0.7354 2144433 PK04_097304 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P07 compound treatment 1157240.0 -10500.0 -0.18 925000.0 -240000.0 -4.33 -3.184 -0.7353 2141482 PK04_097305 Oc1ccc(cc1)[C@@H]2N3[C@H]([C@H](C(=O)N4CCCCCCC4)[C@@]25C(=O)Nc6ccc(C#CC7=CCCCC7)cc65)C(=O)O[C@H]([C@H]3c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P08 compound treatment 1088800.0 -79000.0 -1.32 1027160.0 -138000.0 -2.49 -2.6923 -0.9562 2143929 PK04_097306 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccccc4OCCO)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCNC(=O)N)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P09 compound treatment 1150960.0 -16800.0 -0.28 1052200.0 -113000.0 -2.04 -1.6377 -0.7972 2141698 PK04_097307 COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H]3[C@@H]4N([C@H](c5ccccc5OCCO)[C@@]36C(=O)Nc7ccc(C#CCNC(=O)N)cc76)[C@H]([C@H](OC4=O)c8ccccc8)c9ccccc9 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P10 compound treatment 1153600.0 -14200.0 -0.24 1028880.0 -136000.0 -2.46 -1.9036 -0.7718 2142653 PK04_097308 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCN(CC7)c8ncccn8)c9cc(C#CCNC(=O)N)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P11 mock treatment 1148600.0 -19200.0 -0.32 1039880.0 -125000.0 -2.26 -1.8226 -0.7995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P12 mock treatment 1170960.0 3200.0 0.05 1073040.0 -92100.0 -1.66 -1.1356 -0.6839 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P13 compound treatment 1115360.0 -52400.0 -0.88 1057240.0 -108000.0 -1.94 -1.9948 -0.9353 2141449 PK04_097309 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)N8CCCCCCC8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P14 compound treatment 1126680.0 -41100.0 -0.69 1073880.0 -91300.0 -1.64 -1.6488 -0.9251 2144933 PK04_097310 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7ccccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P15 compound treatment 1116000.0 -51800.0 -0.87 1073520.0 -91600.0 -1.65 -1.7798 -0.9547 2141416 PK04_097311 COc1ccc(C#Cc2ccc3NC(=O)[C@@]4([C@H]([C@H]5N([C@H]4c6ccc(O)cc6)[C@@H]([C@@H](OC5=O)c7ccccc7)c8ccccc8)C(=O)N9CCCCCCC9)c3c2)cc1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P16 compound treatment 1104920.0 -62800.0 -1.05 1068200.0 -96900.0 -1.75 -1.9787 -0.9705 2144445 PK04_097312 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N)c7cc(C#CC8=CCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P17 compound treatment 1099360.0 -68400.0 -1.14 1100840.0 -64300.0 -1.16 -1.6287 -1.0 2141453 PK04_097313 COC(=O)C(CC#Cc1ccc2NC(=O)[C@@]3([C@H]([C@H]4N([C@H]3c5ccc(O)cc5)[C@@H]([C@@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P18 compound treatment 1108600.0 -59200.0 -0.99 1091400.0 -73700.0 -1.33 -1.6396 -0.9895 2142745 PK04_097314 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)NCC=C)c7cc(C#CC8(O)CCCCCC8)ccc17 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P19 compound treatment 973200.0 -195000.0 -3.26 980160.0 -185000.0 -3.33 -4.659 -0.9999 2141541 PK04_097315 COC(=O)C(CC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccc(OCCO)cc5)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)Nc8nc9ccccc9s8)c2c1)C(=O)OC 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P20 compound treatment 1057080.0 -111000.0 -1.85 1049880.0 -115000.0 -2.08 -2.7782 -0.9984 2142193 PK04_097316 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccc(OCCO)cc4)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CC9=CCCCC9)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P21 compound treatment 972080.0 -196000.0 -3.27 976680.0 -188000.0 -3.4 -4.7166 -0.9998 2141134 PK04_097317 NC(=O)NCC#Cc1ccc2NC(=O)[C@]3([C@@H]([C@@H]4N([C@@H]3c5ccccc5OCCO)[C@H]([C@H](OC4=O)c6ccccc6)c7ccccc7)C(=O)O)c2c1 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P22 compound treatment 1071920.0 -95800.0 -1.6 1052760.0 -112000.0 -2.02 -2.5659 -0.9933 2142729 PK04_097318 COCCOC(=O)N1C(=O)[C@@]2([C@H]([C@H]3N([C@H]2c4ccccc4OCCO)[C@@H]([C@@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)Nc7nc8ccccc8s7)c9cc(C#CCC(C(=O)OC)C(=O)OC)ccc19 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P23 compound treatment 1024360.0 -143000.0 -2.4 1023640.0 -142000.0 -2.55 -3.4997 -0.9995 2141121 PK04_097319 OC(=O)[C@H]1[C@H]2N([C@@H](c3ccc(O)cc3)[C@]14C(=O)Nc5ccc(C#CC6=CCCCC6)cc54)[C@@H]([C@@H](OC2=O)c7ccccc7)c8ccccc8 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.2097 P24 compound treatment 1129520.0 -38200.0 -0.64 1130960.0 -34200.0 -0.62 -0.888 -0.9998 2144273 PK04_097320 COCCOC(=O)N1C(=O)[C@]2([C@@H]([C@@H]3N([C@@H]2c4ccc(O)cc4)[C@H]([C@H](OC3=O)c5ccccc5)c6ccccc6)C(=O)N7CCCCCCC7)c8cc(C#CCCO)ccc18 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A01 mock treatment 1257200.0 47000.0 0.79 1258200.0 52800.0 0.95 1.2293 0.9955 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A02 mock treatment 1256400.0 46200.0 0.77 1252000.0 46600.0 0.84 1.1408 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A03 mock treatment 1262000.0 51800.0 0.87 1247480.0 42100.0 0.76 1.1495 0.9978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A04 mock treatment 1252880.0 42700.0 0.71 1253360.0 48000.0 0.86 1.1165 0.9955 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A05 mock treatment 1252000.0 41800.0 0.7 1238840.0 33500.0 0.6 0.9211 0.9973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A06 mock treatment 1249800.0 39600.0 0.66 1240120.0 34800.0 0.63 0.9114 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A07 mock treatment 1250160.0 40000.0 0.67 1242840.0 37500.0 0.68 0.9503 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A08 mock treatment 1232120.0 21900.0 0.37 1235360.0 30000.0 0.54 0.6415 0.9822 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A09 mock treatment 1245520.0 35300.0 0.59 1240440.0 35100.0 0.63 0.8648 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A10 mock treatment 1234160.0 24000.0 0.4 1221080.0 15700.0 0.28 0.4837 0.9855 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A11 mock treatment 1241280.0 31100.0 0.52 1229360.0 24000.0 0.43 0.6735 0.9958 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A12 mock treatment 1234040.0 23800.0 0.4 1236680.0 31300.0 0.56 0.6811 0.9856 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A13 mock treatment 1231240.0 21000.0 0.35 1229880.0 24500.0 0.44 0.5613 0.9937 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A14 mock treatment 1228520.0 18300.0 0.31 1228840.0 23500.0 0.42 0.5159 0.9875 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A15 mock treatment 1213840.0 3640.0 0.06 1224280.0 18900.0 0.34 0.2841 0.8204 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A16 mock treatment 1208000.0 -2200.0 -0.04 1211800.0 6440.0 0.12 0.0559 0.4598 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A17 mock treatment 1197880.0 -12300.0 -0.21 1214760.0 9400.0 0.17 -0.0261 -0.0978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A18 mock treatment 1202480.0 -7720.0 -0.13 1218000.0 12600.0 0.23 0.0696 0.2659 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A19 mock treatment 1206760.0 -3440.0 -0.06 1196680.0 -8680.0 -0.16 -0.1514 -0.9079 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A20 mock treatment 1196480.0 -13700.0 -0.23 1208280.0 2920.0 0.05 -0.1252 -0.5315 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A21 mock treatment 1194040.0 -16200.0 -0.27 1206560.0 1200.0 0.02 -0.176 -0.6487 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A22 mock treatment 1198480.0 -11700.0 -0.2 1190160.0 -15200.0 -0.27 -0.3324 -0.9866 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A23 mock treatment 1203320.0 -6880.0 -0.12 1197040.0 -8320.0 -0.15 -0.1875 -0.9915 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base A24 mock treatment 1181960.0 -28200.0 -0.47 1192240.0 -13100.0 -0.24 -0.5014 -0.9488 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B01 mock treatment 1270760.0 60600.0 1.01 1274520.0 69200.0 1.25 1.5977 0.9947 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B02 mock treatment 1271200.0 61000.0 1.02 1265120.0 59800.0 1.08 1.4831 0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B03 mock treatment 1262800.0 52600.0 0.88 1259160.0 53800.0 0.97 1.3078 0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B04 mock treatment 1259640.0 49400.0 0.83 1255800.0 50400.0 0.91 1.2276 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B05 mock treatment 1252680.0 42500.0 0.71 1244440.0 39100.0 0.7 1.0005 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B06 mock treatment 1261800.0 51600.0 0.86 1240240.0 34900.0 0.63 1.0549 0.9878 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B07 mock treatment 1244120.0 33900.0 0.57 1239600.0 34200.0 0.62 0.8375 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B08 mock treatment 1235320.0 25100.0 0.42 1233040.0 27700.0 0.5 0.6498 0.9964 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B09 mock treatment 1236720.0 26500.0 0.44 1229240.0 23900.0 0.43 0.618 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B10 mock treatment 1233320.0 23100.0 0.39 1243320.0 38000.0 0.68 0.7571 0.9636 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B11 mock treatment 1235120.0 24900.0 0.42 1234360.0 29000.0 0.52 0.6643 0.9938 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B12 mock treatment 1238120.0 27900.0 0.47 1229160.0 23800.0 0.43 0.6335 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B13 mock treatment 1223880.0 13700.0 0.23 1222680.0 17300.0 0.31 0.3825 0.9884 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B14 mock treatment 1219800.0 9600.0 0.16 1213720.0 8360.0 0.15 0.22 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B15 mock treatment 1209080.0 -1120.0 -0.02 1219240.0 13900.0 0.25 0.1635 0.6522 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B16 mock treatment 1191240.0 -19000.0 -0.32 1204440.0 -923.0 -0.02 -0.2361 -0.7431 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B17 mock treatment 1196720.0 -13500.0 -0.23 1202680.0 -2680.0 -0.05 -0.1937 -0.8396 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B18 mock treatment 1211040.0 838.0 0.01 1199960.0 -5400.0 -0.1 -0.0589 -0.5991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B19 mock treatment 1184200.0 -26000.0 -0.44 1185360.0 -20000.0 -0.36 -0.5625 -0.9956 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B20 mock treatment 1180600.0 -29600.0 -0.5 1186720.0 -18600.0 -0.34 -0.5878 -0.9821 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B21 mock treatment 1168280.0 -41900.0 -0.7 1188920.0 -16400.0 -0.3 -0.7056 -0.9265 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B22 mock treatment 1182440.0 -27800.0 -0.46 1181640.0 -23700.0 -0.43 -0.6307 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B23 mock treatment 1185480.0 -24700.0 -0.41 1184400.0 -21000.0 -0.38 -0.5596 -0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base B24 mock treatment 1194200.0 -16000.0 -0.27 1194480.0 -10900.0 -0.2 -0.328 -0.9883 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C01 mock treatment 1252440.0 42200.0 0.71 1246360.0 41000.0 0.74 1.0221 0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C02 mock treatment 1250920.0 40700.0 0.68 1239560.0 34200.0 0.62 0.9175 0.9987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C03 mock treatment 1247000.0 36800.0 0.62 1226560.0 21200.0 0.38 0.7055 0.9736 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C04 mock treatment 1241160.0 31000.0 0.52 1233800.0 28400.0 0.51 0.7286 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C05 mock treatment 1237120.0 26900.0 0.45 1218520.0 13200.0 0.24 0.4861 0.955 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C06 mock treatment 1236320.0 26100.0 0.44 1219760.0 14400.0 0.26 0.4925 0.969 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C07 mock treatment 1230880.0 20700.0 0.35 1209840.0 4480.0 0.08 0.3017 0.8492 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C08 mock treatment 1221360.0 11200.0 0.19 1212680.0 7320.0 0.13 0.2253 0.9855 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C09 mock treatment 1213880.0 3680.0 0.06 1208560.0 3200.0 0.06 0.0842 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C10 mock treatment 1200240.0 -9960.0 -0.17 1219720.0 14400.0 0.26 0.065 0.2113 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C11 mock treatment 1211440.0 1240.0 0.02 1227240.0 21900.0 0.39 0.2934 0.7432 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C12 mock treatment 1225160.0 15000.0 0.25 1215400.0 10000.0 0.18 0.3049 0.9873 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C13 mock treatment 1222400.0 12200.0 0.2 1209240.0 3880.0 0.07 0.1937 0.898 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C14 mock treatment 1203640.0 -6560.0 -0.11 1210080.0 4720.0 0.08 -0.0176 -0.1264 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C15 mock treatment 1209360.0 -842.0 -0.01 1203160.0 -2200.0 -0.04 -0.038 -0.903 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C16 mock treatment 1197320.0 -12900.0 -0.22 1191560.0 -13800.0 -0.25 -0.3283 -0.9975 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C17 mock treatment 1199160.0 -11000.0 -0.18 1203560.0 -1800.0 -0.03 -0.1536 -0.8189 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C18 mock treatment 1185880.0 -24300.0 -0.41 1186520.0 -18800.0 -0.34 -0.5279 -0.9959 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C19 mock treatment 1187800.0 -22400.0 -0.37 1188720.0 -16600.0 -0.3 -0.4771 -0.9939 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C20 mock treatment 1177520.0 -32700.0 -0.55 1180200.0 -25200.0 -0.45 -0.7073 -0.9957 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C21 mock treatment 1177720.0 -32500.0 -0.54 1175320.0 -30000.0 -0.54 -0.7671 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C22 mock treatment 1174320.0 -35900.0 -0.6 1168960.0 -36400.0 -0.66 -0.8884 -0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C23 mock treatment 1177360.0 -32800.0 -0.55 1185600.0 -19800.0 -0.36 -0.6404 -0.9779 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base C24 mock treatment 1187240.0 -23000.0 -0.38 1179880.0 -25500.0 -0.46 -0.5964 -0.9961 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D01 mock treatment 1261640.0 51400.0 0.86 1265120.0 59800.0 1.08 1.37 0.9939 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D02 mock treatment 1266560.0 56400.0 0.94 1245600.0 40200.0 0.72 1.1795 0.9916 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D03 mock treatment 1250720.0 40500.0 0.68 1239360.0 34000.0 0.61 0.9126 0.9987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D04 mock treatment 1246560.0 36400.0 0.61 1246640.0 41300.0 0.74 0.9561 0.995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D05 mock treatment 1248120.0 37900.0 0.63 1239040.0 33700.0 0.61 0.8777 0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D06 mock treatment 1232880.0 22700.0 0.38 1230440.0 25100.0 0.45 0.5878 0.9962 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D07 mock treatment 1231520.0 21300.0 0.36 1226720.0 21400.0 0.38 0.5243 0.9993 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D08 mock treatment 1223240.0 13000.0 0.22 1212160.0 6800.0 0.12 0.2409 0.9627 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D09 mock treatment 1212360.0 2160.0 0.04 1218160.0 12800.0 0.23 0.1886 0.808 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D10 mock treatment 1231200.0 21000.0 0.35 1231160.0 25800.0 0.46 0.5771 0.9905 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D11 mock treatment 1224520.0 14300.0 0.24 1211520.0 6160.0 0.11 0.2479 0.9388 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D12 mock treatment 1197440.0 -12800.0 -0.21 1214040.0 8680.0 0.16 -0.0405 -0.1529 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D13 mock treatment 1219640.0 9440.0 0.16 1189960.0 -15400.0 -0.28 -0.0846 -0.2648 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D14 mock treatment 1189160.0 -21000.0 -0.35 1200480.0 -4880.0 -0.09 -0.3112 -0.8574 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D15 mock treatment 1192800.0 -17400.0 -0.29 1193680.0 -11700.0 -0.21 -0.3548 -0.9873 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D16 mock treatment 1196440.0 -13800.0 -0.23 1180280.0 -25100.0 -0.45 -0.4824 -0.9511 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D17 mock treatment 1175200.0 -35000.0 -0.59 1182520.0 -22800.0 -0.41 -0.7052 -0.9851 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D18 mock treatment 1179600.0 -30600.0 -0.51 1192880.0 -12500.0 -0.22 -0.5212 -0.9318 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D19 mock treatment 1172960.0 -37200.0 -0.62 1173960.0 -31400.0 -0.57 -0.8408 -0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D20 mock treatment 1162400.0 -47800.0 -0.8 1168560.0 -36800.0 -0.66 -1.0345 -0.9957 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D21 mock treatment 1154040.0 -56200.0 -0.94 1163880.0 -41500.0 -0.75 -1.1931 -0.9936 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D22 mock treatment 1153320.0 -56900.0 -0.95 1161520.0 -43800.0 -0.79 -1.2317 -0.9957 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D23 mock treatment 1147160.0 -63000.0 -1.05 1169920.0 -35400.0 -0.64 -1.1975 -0.9711 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base D24 mock treatment 1171640.0 -38600.0 -0.65 1164800.0 -40600.0 -0.73 -0.9731 -0.9981 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E01 mock treatment 1260880.0 50700.0 0.85 1256600.0 51200.0 0.92 1.2524 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E02 mock treatment 1249080.0 38900.0 0.65 1236000.0 30600.0 0.55 0.8504 0.9967 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E03 mock treatment 1237400.0 27200.0 0.46 1224680.0 19300.0 0.35 0.5679 0.9912 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E04 mock treatment 1237360.0 27200.0 0.45 1228480.0 23100.0 0.42 0.6159 0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E05 mock treatment 1254120.0 43900.0 0.73 1228360.0 23000.0 0.41 0.8127 0.9632 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E06 mock treatment 1236760.0 26600.0 0.44 1204800.0 -563.0 -0.01 0.3071 0.6908 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E07 mock treatment 1220800.0 10600.0 0.18 1213400.0 8040.0 0.14 0.2278 0.9949 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E08 mock treatment 1232000.0 21800.0 0.36 1202280.0 -3080.0 -0.06 0.2187 0.5926 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E09 mock treatment 1218920.0 8720.0 0.15 1218520.0 13200.0 0.24 0.2708 0.9728 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E10 mock treatment 1221720.0 11500.0 0.19 1208960.0 3600.0 0.06 0.1821 0.8956 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E11 mock treatment 1226720.0 16500.0 0.28 1215800.0 10400.0 0.19 0.3284 0.9824 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E12 mock treatment 1211800.0 1600.0 0.03 1217560.0 12200.0 0.22 0.1743 0.7873 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E13 mock treatment 1190920.0 -19300.0 -0.32 1177840.0 -27500.0 -0.5 -0.5788 -0.9783 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E14 mock treatment 1209200.0 -1000.0 -0.02 1217680.0 12300.0 0.22 0.1451 0.6518 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E15 mock treatment 1208080.0 -2120.0 -0.04 1202720.0 -2640.0 -0.05 -0.0588 -0.9896 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E16 mock treatment 1195600.0 -14600.0 -0.24 1202200.0 -3160.0 -0.06 -0.2131 -0.8492 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E17 mock treatment 1179360.0 -30800.0 -0.52 1198400.0 -6960.0 -0.13 -0.4537 -0.8541 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E18 mock treatment 1202480.0 -7720.0 -0.13 1196160.0 -9200.0 -0.17 -0.2086 -0.9924 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E19 mock treatment 1177920.0 -32300.0 -0.54 1164120.0 -41200.0 -0.74 -0.9074 -0.9877 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E20 mock treatment 1165880.0 -44300.0 -0.74 1176600.0 -28800.0 -0.52 -0.8909 -0.9846 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E21 mock treatment 1179920.0 -30300.0 -0.51 1178280.0 -27100.0 -0.49 -0.7034 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E22 mock treatment 1184600.0 -25600.0 -0.43 1172520.0 -32800.0 -0.59 -0.7214 -0.9874 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E23 mock treatment 1186200.0 -24000.0 -0.4 1180080.0 -25300.0 -0.46 -0.6061 -0.998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base E24 mock treatment 1174440.0 -35800.0 -0.6 1167000.0 -38400.0 -0.69 -0.9119 -0.9974 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F01 mock treatment 1260680.0 50500.0 0.84 1252120.0 46800.0 0.84 1.193 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F02 mock treatment 1252040.0 41800.0 0.7 1244120.0 38800.0 0.7 0.9888 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F03 mock treatment 1244120.0 33900.0 0.57 1228360.0 23000.0 0.41 0.6943 0.988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F04 mock treatment 1236760.0 26600.0 0.44 1226560.0 21200.0 0.38 0.5843 0.9971 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F05 mock treatment 1236720.0 26500.0 0.44 1227520.0 22200.0 0.4 0.5961 0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F06 mock treatment 1229840.0 19600.0 0.33 1231760.0 26400.0 0.48 0.5687 0.9837 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F07 mock treatment 1226720.0 16500.0 0.28 1221960.0 16600.0 0.3 0.4069 0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F08 mock treatment 1232800.0 22600.0 0.38 1191800.0 -13600.0 -0.24 0.0946 0.2101 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F09 mock treatment 1214600.0 4400.0 0.07 1222160.0 16800.0 0.3 0.266 0.8542 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F10 mock treatment 1204840.0 -5360.0 -0.09 1206840.0 1480.0 0.03 -0.0446 -0.4769 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F11 mock treatment 1209520.0 -682.0 -0.01 1210960.0 5600.0 0.1 0.0632 0.6231 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F12 mock treatment 1214560.0 4360.0 0.07 1200120.0 -5240.0 -0.09 -0.0152 -0.1276 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F13 mock treatment 1187480.0 -22700.0 -0.38 1188080.0 -17300.0 -0.31 -0.4891 -0.9951 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F14 mock treatment 1204560.0 -5640.0 -0.09 1199440.0 -5920.0 -0.11 -0.1422 -0.9981 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F15 mock treatment 1197960.0 -12200.0 -0.2 1189600.0 -15800.0 -0.28 -0.3457 -0.9871 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F16 mock treatment 1179520.0 -30700.0 -0.51 1181280.0 -24100.0 -0.43 -0.6699 -0.9965 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F17 mock treatment 1166160.0 -44000.0 -0.74 1170360.0 -35000.0 -0.63 -0.9671 -0.997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F18 mock treatment 1174760.0 -35400.0 -0.59 1173600.0 -31800.0 -0.57 -0.8241 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F19 mock treatment 1163200.0 -47000.0 -0.79 1173240.0 -32100.0 -0.58 -0.9654 -0.9886 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F20 mock treatment 1152480.0 -57700.0 -0.97 1159840.0 -45500.0 -0.82 -1.263 -0.9967 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F21 mock treatment 1150560.0 -59600.0 -1.0 1167000.0 -38400.0 -0.69 -1.1945 -0.9839 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F22 mock treatment 1157360.0 -52800.0 -0.88 1156480.0 -48900.0 -0.88 -1.2481 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F23 mock treatment 1156040.0 -54200.0 -0.91 1158160.0 -47200.0 -0.85 -1.2423 -0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base F24 mock treatment 1165400.0 -44800.0 -0.75 1160240.0 -45100.0 -0.81 -1.105 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G01 mock treatment 1265480.0 55300.0 0.93 1246640.0 41300.0 0.74 1.18 0.9941 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G02 mock treatment 1269760.0 59600.0 1.0 1249200.0 43800.0 0.79 1.2632 0.9934 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G03 mock treatment 1256200.0 46000.0 0.77 1233880.0 28500.0 0.51 0.9076 0.9807 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G04 mock treatment 1251160.0 41000.0 0.69 1224920.0 19600.0 0.35 0.7338 0.9522 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G05 mock treatment 1239240.0 29000.0 0.49 1234320.0 29000.0 0.52 0.7125 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G06 mock treatment 1238800.0 28600.0 0.48 1227760.0 22400.0 0.4 0.6237 0.9964 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G07 mock treatment 1245480.0 35300.0 0.59 1226360.0 21000.0 0.38 0.6849 0.9769 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G08 mock treatment 1226480.0 16300.0 0.27 1222560.0 17200.0 0.31 0.4117 0.9979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G09 mock treatment 1228840.0 18600.0 0.31 1235000.0 29600.0 0.53 0.5981 0.9672 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G10 mock treatment 1226920.0 16700.0 0.28 1210960.0 5600.0 0.1 0.2691 0.905 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G11 mock treatment 1222960.0 12800.0 0.21 1199640.0 -5720.0 -0.1 0.0781 0.3292 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G12 mock treatment 1196120.0 -14100.0 -0.24 1222760.0 17400.0 0.31 0.055 0.1403 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G13 mock treatment 1220440.0 10200.0 0.17 1199880.0 -5480.0 -0.1 0.0513 0.2594 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G14 mock treatment 1231200.0 21000.0 0.35 1214120.0 8760.0 0.16 0.36 0.9347 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G15 mock treatment 1200320.0 -9880.0 -0.17 1209440.0 4080.0 0.07 -0.065 -0.3592 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G16 mock treatment 1206240.0 -3960.0 -0.07 1201480.0 -3880.0 -0.07 -0.0964 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G17 mock treatment 1184880.0 -25300.0 -0.42 1204200.0 -1160.0 -0.02 -0.3145 -0.7412 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G18 mock treatment 1185960.0 -24200.0 -0.41 1185040.0 -20300.0 -0.37 -0.5458 -0.9987 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G19 mock treatment 1184320.0 -25900.0 -0.43 1179840.0 -25500.0 -0.46 -0.6314 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G20 mock treatment 1188280.0 -21900.0 -0.37 1186040.0 -19300.0 -0.35 -0.5056 -0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G21 mock treatment 1180400.0 -29800.0 -0.5 1178040.0 -27300.0 -0.49 -0.7008 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G22 mock treatment 1179560.0 -30600.0 -0.51 1183120.0 -22200.0 -0.4 -0.646 -0.9926 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G23 mock treatment 1178440.0 -31800.0 -0.53 1175480.0 -29900.0 -0.54 -0.7566 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base G24 mock treatment 1173120.0 -37100.0 -0.62 1170600.0 -34800.0 -0.63 -0.8817 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H01 mock treatment 1265120.0 54900.0 0.92 1258320.0 53000.0 0.95 1.3245 0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H02 mock treatment 1259960.0 49800.0 0.83 1236240.0 30900.0 0.56 0.9822 0.9808 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H03 mock treatment 1234320.0 24100.0 0.4 1242840.0 37500.0 0.68 0.7628 0.9697 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H04 mock treatment 1245920.0 35700.0 0.6 1233160.0 27800.0 0.5 0.7768 0.9961 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H05 mock treatment 1241000.0 30800.0 0.52 1229680.0 24300.0 0.44 0.6742 0.9967 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H06 mock treatment 1248400.0 38200.0 0.64 1216160.0 10800.0 0.19 0.5896 0.8823 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H07 mock treatment 1235000.0 24800.0 0.41 1223200.0 17800.0 0.32 0.5207 0.992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H08 mock treatment 1243320.0 33100.0 0.55 1214040.0 8680.0 0.16 0.5024 0.8725 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H09 mock treatment 1224560.0 14400.0 0.24 1211760.0 6400.0 0.12 0.2514 0.9434 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H10 mock treatment 1213840.0 3640.0 0.06 1214040.0 8680.0 0.16 0.1536 0.9155 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H11 mock treatment 1217280.0 7080.0 0.12 1205000.0 -363.0 -0.01 0.0791 0.667 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H12 mock treatment 1187240.0 -23000.0 -0.38 1209680.0 4320.0 0.08 -0.2167 -0.5528 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H13 mock treatment 1206560.0 -3640.0 -0.06 1155080.0 -50300.0 -0.91 -0.6837 -0.753 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H14 mock treatment 1196240.0 -14000.0 -0.23 1194200.0 -11200.0 -0.2 -0.3074 -0.9972 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H15 mock treatment 1185080.0 -25100.0 -0.42 1194000.0 -11400.0 -0.2 -0.442 -0.9453 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H16 mock treatment 1185120.0 -25100.0 -0.42 1176440.0 -28900.0 -0.52 -0.6653 -0.9942 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H17 mock treatment 1174600.0 -35600.0 -0.6 1180160.0 -25200.0 -0.45 -0.7424 -0.991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H18 mock treatment 1181280.0 -28900.0 -0.48 1182920.0 -22400.0 -0.4 -0.6282 -0.996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H19 mock treatment 1178160.0 -32000.0 -0.54 1167400.0 -38000.0 -0.68 -0.8628 -0.9927 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H20 mock treatment 1173240.0 -37000.0 -0.62 1161760.0 -43600.0 -0.79 -0.9929 -0.993 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H21 mock treatment 1174040.0 -36200.0 -0.61 1172240.0 -33100.0 -0.6 -0.8499 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H22 mock treatment 1165320.0 -44900.0 -0.75 1155720.0 -49600.0 -0.89 -1.1636 -0.9962 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H23 mock treatment 1145960.0 -64200.0 -1.08 1163680.0 -41700.0 -0.75 -1.2912 -0.9846 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base H24 mock treatment 1166200.0 -44000.0 -0.74 1150840.0 -54500.0 -0.98 -1.2153 -0.9899 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I01 mock treatment 1256360.0 46200.0 0.77 1265040.0 59700.0 1.08 1.3065 0.9868 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I02 mock treatment 1253400.0 43200.0 0.72 1244720.0 39400.0 0.71 1.0126 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I03 mock treatment 1245720.0 35500.0 0.59 1266760.0 61400.0 1.11 1.2025 0.9576 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I04 mock treatment 1247920.0 37700.0 0.63 1238120.0 32800.0 0.59 0.8636 0.9994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I05 mock treatment 1249600.0 39400.0 0.66 1226600.0 21200.0 0.38 0.7368 0.9665 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I06 mock treatment 1234640.0 24400.0 0.41 1219800.0 14400.0 0.26 0.4731 0.9761 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I07 mock treatment 1238960.0 28800.0 0.48 1208320.0 2960.0 0.05 0.378 0.7806 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I08 mock treatment 1228280.0 18100.0 0.3 1222720.0 17400.0 0.31 0.435 0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I09 mock treatment 1230040.0 19800.0 0.33 1232480.0 27100.0 0.49 0.5802 0.9823 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I10 mock treatment 1223040.0 12800.0 0.21 1205760.0 397.0 0.01 0.157 0.7302 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I11 mock treatment 1233040.0 22800.0 0.38 1222360.0 17000.0 0.31 0.4868 0.994 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I12 mock treatment 1186440.0 -23800.0 -0.4 1213320.0 7960.0 0.14 -0.1798 -0.4254 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I13 mock treatment 1222080.0 11900.0 0.2 1189520.0 -15800.0 -0.29 -0.0613 -0.1762 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I14 mock treatment 1210280.0 77.8 0.0 1203440.0 -1920.0 -0.03 -0.0236 -0.6801 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I15 mock treatment 1203800.0 -6400.0 -0.11 1201840.0 -3520.0 -0.06 -0.1206 -0.9688 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I16 mock treatment 1190400.0 -19800.0 -0.33 1190280.0 -15100.0 -0.27 -0.4265 -0.9951 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I17 mock treatment 1206040.0 -4160.0 -0.07 1195080.0 -10300.0 -0.19 -0.1803 -0.9107 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I18 mock treatment 1174760.0 -35400.0 -0.59 1190320.0 -15000.0 -0.27 -0.611 -0.937 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I19 mock treatment 1193880.0 -16300.0 -0.27 1198720.0 -6640.0 -0.12 -0.2778 -0.9315 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I20 mock treatment 1183440.0 -26800.0 -0.45 1175280.0 -30100.0 -0.54 -0.6999 -0.9955 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I21 mock treatment 1189000.0 -21200.0 -0.35 1177280.0 -28100.0 -0.51 -0.6087 -0.9849 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I22 mock treatment 1180520.0 -29700.0 -0.5 1166000.0 -39400.0 -0.71 -0.8527 -0.9848 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I23 mock treatment 1173720.0 -36500.0 -0.61 1172680.0 -32700.0 -0.59 -0.8481 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base I24 mock treatment 1160600.0 -49600.0 -0.83 1157640.0 -47700.0 -0.86 -1.1949 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J01 mock treatment 1261960.0 51800.0 0.87 1260800.0 55400.0 1.0 1.3187 0.9975 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J02 mock treatment 1255040.0 44800.0 0.75 1247280.0 41900.0 0.76 1.0646 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J03 mock treatment 1255480.0 45300.0 0.76 1247760.0 42400.0 0.76 1.0759 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J04 mock treatment 1235800.0 25600.0 0.43 1249240.0 43900.0 0.79 0.8619 0.9586 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J05 mock treatment 1244960.0 34800.0 0.58 1225680.0 20300.0 0.37 0.6701 0.9751 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J06 mock treatment 1241760.0 31600.0 0.53 1218240.0 12900.0 0.23 0.5375 0.9318 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J07 mock treatment 1246240.0 36000.0 0.6 1239320.0 34000.0 0.61 0.8591 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J08 mock treatment 1214120.0 3920.0 0.07 1227200.0 21800.0 0.39 0.3246 0.8137 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J09 mock treatment 1221880.0 11700.0 0.2 1214720.0 9360.0 0.17 0.2574 0.9973 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J10 mock treatment 1226800.0 16600.0 0.28 1226560.0 21200.0 0.38 0.4665 0.9878 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J11 mock treatment 1225920.0 15700.0 0.26 1211640.0 6280.0 0.11 0.266 0.9289 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J12 mock treatment 1192840.0 -17400.0 -0.29 1202720.0 -2640.0 -0.05 -0.2391 -0.8122 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J13 mock treatment 1182480.0 -27700.0 -0.46 1168160.0 -37200.0 -0.67 -0.802 -0.9838 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J14 mock treatment 1196280.0 -13900.0 -0.23 1196040.0 -9320.0 -0.17 -0.2835 -0.9871 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J15 mock treatment 1186600.0 -23600.0 -0.39 1193080.0 -12300.0 -0.22 -0.4358 -0.9625 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J16 mock treatment 1196840.0 -13400.0 -0.22 1187440.0 -17900.0 -0.32 -0.3865 -0.9839 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J17 mock treatment 1198400.0 -11800.0 -0.2 1190320.0 -15000.0 -0.27 -0.3313 -0.9879 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J18 mock treatment 1187840.0 -22400.0 -0.37 1181640.0 -23700.0 -0.43 -0.5668 -0.9978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J19 mock treatment 1176440.0 -33800.0 -0.56 1174360.0 -31000.0 -0.56 -0.7945 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J20 mock treatment 1205480.0 -4720.0 -0.08 1154080.0 -51300.0 -0.92 -0.7092 -0.7648 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J21 mock treatment 1173520.0 -36700.0 -0.61 1176760.0 -28600.0 -0.52 -0.7985 -0.9962 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J22 mock treatment 1165160.0 -45000.0 -0.75 1166880.0 -38500.0 -0.69 -1.0233 -0.9991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J23 mock treatment 1183000.0 -27200.0 -0.46 1162280.0 -43100.0 -0.78 -0.8708 -0.9677 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base J24 mock treatment 1161960.0 -48200.0 -0.81 1137120.0 -68200.0 -1.23 -1.4403 -0.9792 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K01 mock treatment 1268760.0 58600.0 0.98 1247000.0 41600.0 0.75 1.2234 0.9913 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K02 mock treatment 1224000.0 13800.0 0.23 1257720.0 52400.0 0.94 0.8303 0.8549 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K03 mock treatment 1252720.0 42500.0 0.71 1225280.0 19900.0 0.36 0.7569 0.9498 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K04 mock treatment 1249440.0 39200.0 0.66 1241960.0 36600.0 0.66 0.9306 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K05 mock treatment 1238440.0 28200.0 0.47 1234000.0 28600.0 0.52 0.699 0.999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K06 mock treatment 1227160.0 17000.0 0.28 1238240.0 32900.0 0.59 0.6195 0.9432 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K07 mock treatment 1217360.0 7160.0 0.12 1242440.0 37100.0 0.67 0.5571 0.8208 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K08 mock treatment 1230040.0 19800.0 0.33 1212160.0 6800.0 0.12 0.3213 0.9081 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K09 mock treatment 1243400.0 33200.0 0.56 1226800.0 21400.0 0.39 0.6659 0.9842 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K10 mock treatment 1232000.0 21800.0 0.36 1210200.0 4840.0 0.09 0.3196 0.8521 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K11 mock treatment 1214560.0 4360.0 0.07 1215280.0 9920.0 0.18 0.1779 0.9219 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K12 mock treatment 1225800.0 15600.0 0.26 1214520.0 9160.0 0.16 0.3012 0.9755 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K13 mock treatment 1197080.0 -13100.0 -0.22 1186760.0 -18600.0 -0.34 -0.3923 -0.979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K14 mock treatment 1209960.0 -242.0 0.0 1209360.0 4000.0 0.07 0.0481 0.6663 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K15 mock treatment 1219800.0 9600.0 0.16 1204120.0 -1240.0 -0.02 0.0977 0.6027 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K16 mock treatment 1208120.0 -2080.0 -0.03 1202880.0 -2480.0 -0.04 -0.0563 -0.9924 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K17 mock treatment 1199360.0 -10800.0 -0.18 1210160.0 4800.0 0.09 -0.0672 -0.3343 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K18 mock treatment 1213200.0 3000.0 0.05 1208840.0 3480.0 0.06 0.0798 0.9939 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K19 mock treatment 1199760.0 -10400.0 -0.17 1202840.0 -2520.0 -0.05 -0.1557 -0.8624 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K20 mock treatment 1191280.0 -18900.0 -0.32 1190920.0 -14400.0 -0.26 -0.4079 -0.9952 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K21 mock treatment 1187880.0 -22300.0 -0.37 1183480.0 -21900.0 -0.39 -0.5429 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K22 mock treatment 1175200.0 -35000.0 -0.59 1185720.0 -19600.0 -0.35 -0.6644 -0.9709 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K23 mock treatment 1184680.0 -25500.0 -0.43 1186040.0 -19300.0 -0.35 -0.5482 -0.9949 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base K24 mock treatment 1155280.0 -54900.0 -0.92 1157280.0 -48100.0 -0.87 -1.2625 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L01 mock treatment 1244240.0 34000.0 0.57 1255800.0 50400.0 0.91 1.0453 0.9747 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L02 mock treatment 1246760.0 36600.0 0.61 1231400.0 26000.0 0.47 0.7643 0.9914 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L03 mock treatment 1245120.0 34900.0 0.58 1243120.0 37800.0 0.68 0.8942 0.9971 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L04 mock treatment 1243360.0 33200.0 0.55 1245760.0 40400.0 0.73 0.907 0.991 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L05 mock treatment 1241320.0 31100.0 0.52 1238400.0 33000.0 0.6 0.7891 0.9978 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L06 mock treatment 1238880.0 28700.0 0.48 1219520.0 14200.0 0.26 0.5197 0.9563 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L07 mock treatment 1228600.0 18400.0 0.31 1227600.0 22200.0 0.4 0.501 0.9915 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L08 mock treatment 1219480.0 9280.0 0.16 1209640.0 4280.0 0.08 0.1643 0.9477 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L09 mock treatment 1222840.0 12600.0 0.21 1220640.0 15300.0 0.28 0.3442 0.9915 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L10 mock treatment 1215000.0 4800.0 0.08 1205520.0 157.0 0.0 0.0588 0.7316 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L11 mock treatment 1201680.0 -8520.0 -0.14 1214000.0 8640.0 0.16 0.0092 0.0435 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L12 mock treatment 1207920.0 -2280.0 -0.04 1200880.0 -4480.0 -0.08 -0.0841 -0.9415 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L13 mock treatment 1169240.0 -41000.0 -0.69 1189280.0 -16100.0 -0.29 -0.6896 -0.9266 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L14 mock treatment 1204320.0 -5880.0 -0.1 1196040.0 -9320.0 -0.17 -0.1884 -0.9676 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L15 mock treatment 1202320.0 -7880.0 -0.13 1183440.0 -21900.0 -0.39 -0.3726 -0.8947 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L16 mock treatment 1197240.0 -13000.0 -0.22 1182480.0 -22900.0 -0.41 -0.4449 -0.955 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L17 mock treatment 1184320.0 -25900.0 -0.43 1178680.0 -26700.0 -0.48 -0.6462 -0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L18 mock treatment 1189360.0 -20800.0 -0.35 1187440.0 -17900.0 -0.32 -0.475 -0.9993 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L19 mock treatment 1180280.0 -29900.0 -0.5 1178520.0 -26800.0 -0.48 -0.6961 -0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L20 mock treatment 1175680.0 -34500.0 -0.58 1166720.0 -38600.0 -0.7 -0.9008 -0.9957 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L21 mock treatment 1180400.0 -29800.0 -0.5 1171640.0 -33700.0 -0.61 -0.7823 -0.9952 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L22 mock treatment 1172120.0 -38100.0 -0.64 1165800.0 -39600.0 -0.71 -0.9547 -0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L23 mock treatment 1187200.0 -23000.0 -0.38 1168160.0 -37200.0 -0.67 -0.7462 -0.9653 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base L24 mock treatment 1156360.0 -53800.0 -0.9 1158080.0 -47300.0 -0.85 -1.2395 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M01 mock treatment 1260280.0 50100.0 0.84 1250200.0 44800.0 0.81 1.1638 0.9998 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M02 mock treatment 1255800.0 45600.0 0.76 1262200.0 56800.0 1.02 1.2637 0.9895 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M03 mock treatment 1274000.0 63800.0 1.07 1263960.0 58600.0 1.06 1.5015 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M04 mock treatment 1259320.0 49100.0 0.82 1251760.0 46400.0 0.84 1.1723 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M05 mock treatment 1243640.0 33400.0 0.56 1241800.0 36400.0 0.66 0.8599 0.9968 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M06 mock treatment 1241560.0 31400.0 0.52 1234240.0 28900.0 0.52 0.739 1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M07 mock treatment 1254120.0 43900.0 0.73 1236240.0 30900.0 0.56 0.9131 0.9906 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M08 mock treatment 1242280.0 32100.0 0.54 1229960.0 24600.0 0.44 0.6929 0.9955 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M09 mock treatment 1237000.0 26800.0 0.45 1222360.0 17000.0 0.31 0.5336 0.9827 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M10 mock treatment 1225280.0 15100.0 0.25 1210040.0 4680.0 0.08 0.238 0.8947 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M11 mock treatment 1228760.0 18600.0 0.31 1203880.0 -1480.0 -0.03 0.2007 0.6439 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M12 mock treatment 1224240.0 14000.0 0.23 1203920.0 -1440.0 -0.03 0.1477 0.625 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M13 mock treatment 1191360.0 -18800.0 -0.32 1197720.0 -7640.0 -0.14 -0.3203 -0.931 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M14 mock treatment 1210440.0 238.0 0.0 1210000.0 4640.0 0.08 0.0619 0.74 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M15 mock treatment 1201560.0 -8640.0 -0.14 1203240.0 -2120.0 -0.04 -0.1293 -0.8644 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M16 mock treatment 1195400.0 -14800.0 -0.25 1193000.0 -12400.0 -0.22 -0.3327 -0.9986 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M17 mock treatment 1199080.0 -11100.0 -0.19 1192720.0 -12600.0 -0.23 -0.2927 -0.995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M18 mock treatment 1213360.0 3160.0 0.05 1194040.0 -11300.0 -0.2 -0.1069 -0.5072 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M19 mock treatment 1187640.0 -22600.0 -0.38 1186640.0 -18700.0 -0.34 -0.5055 -0.9984 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M20 mock treatment 1181520.0 -28700.0 -0.48 1172520.0 -32800.0 -0.59 -0.7578 -0.9946 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M21 mock treatment 1183440.0 -26800.0 -0.45 1166880.0 -38500.0 -0.69 -0.807 -0.9776 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M22 mock treatment 1181240.0 -29000.0 -0.48 1169920.0 -35400.0 -0.64 -0.7943 -0.9907 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M23 mock treatment 1186880.0 -23300.0 -0.39 1183440.0 -21900.0 -0.39 -0.5553 -1.0 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base M24 mock treatment 1180240.0 -30000.0 -0.5 1163920.0 -41400.0 -0.75 -0.8825 -0.9812 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N01 mock treatment 1252160.0 42000.0 0.7 1254360.0 49000.0 0.88 1.1207 0.9936 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N02 mock treatment 1242720.0 32500.0 0.54 1253560.0 48200.0 0.87 0.9988 0.9747 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N03 mock treatment 1236240.0 26000.0 0.44 1246920.0 41600.0 0.75 0.8375 0.9668 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N04 mock treatment 1225880.0 15700.0 0.26 1220920.0 15600.0 0.28 0.3837 0.9995 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N05 mock treatment 1227120.0 16900.0 0.28 1234440.0 29100.0 0.52 0.5706 0.9583 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N06 mock treatment 1225600.0 15400.0 0.26 1218320.0 13000.0 0.23 0.3473 0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N07 mock treatment 1225160.0 15000.0 0.25 1225280.0 19900.0 0.36 0.4307 0.9845 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N08 mock treatment 1225480.0 15300.0 0.26 1215640.0 10300.0 0.19 0.3117 0.9875 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N09 mock treatment 1219560.0 9360.0 0.16 1206800.0 1440.0 0.03 0.129 0.813 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N10 mock treatment 1216960.0 6760.0 0.11 1204960.0 -403.0 -0.01 0.0748 0.6603 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N11 mock treatment 1205360.0 -4840.0 -0.08 1202680.0 -2680.0 -0.05 -0.0915 -0.9695 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N12 mock treatment 1179520.0 -30700.0 -0.51 1200400.0 -4960.0 -0.09 -0.4263 -0.8179 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N13 mock treatment 1187320.0 -22900.0 -0.38 1200200.0 -5160.0 -0.09 -0.3365 -0.854 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N14 mock treatment 1195960.0 -14200.0 -0.24 1200520.0 -4840.0 -0.09 -0.2302 -0.9071 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N15 mock treatment 1200040.0 -10200.0 -0.17 1184000.0 -21400.0 -0.38 -0.3924 -0.9326 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N16 mock treatment 1185040.0 -25200.0 -0.42 1187320.0 -18000.0 -0.33 -0.5276 -0.9918 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N17 mock treatment 1182840.0 -27400.0 -0.46 1179360.0 -26000.0 -0.47 -0.6551 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N18 mock treatment 1191280.0 -18900.0 -0.32 1181440.0 -23900.0 -0.43 -0.5287 -0.9885 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N19 mock treatment 1170280.0 -39900.0 -0.67 1163920.0 -41400.0 -0.75 -1.0004 -0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N20 mock treatment 1169240.0 -41000.0 -0.69 1164240.0 -41100.0 -0.74 -1.0086 -0.9992 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N21 mock treatment 1154680.0 -55500.0 -0.93 1145400.0 -60000.0 -1.08 -1.4209 -0.9972 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N22 mock treatment 1165160.0 -45000.0 -0.75 1156520.0 -48800.0 -0.88 -1.1553 -0.997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N23 mock treatment 1154320.0 -55900.0 -0.94 1141320.0 -64000.0 -1.15 -1.4772 -0.9946 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base N24 mock treatment 1160680.0 -49500.0 -0.83 1163520.0 -41800.0 -0.75 -1.1191 -0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O01 mock treatment 1279520.0 69300.0 1.16 1264000.0 58600.0 1.06 1.5673 0.9989 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O02 mock treatment 1273760.0 63600.0 1.06 1257120.0 51800.0 0.93 1.4115 0.9979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O03 mock treatment 1237520.0 27300.0 0.46 1253920.0 48600.0 0.87 0.9419 0.9542 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O04 mock treatment 1251080.0 40900.0 0.68 1225440.0 20100.0 0.36 0.7395 0.9556 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O05 mock treatment 1254120.0 43900.0 0.73 1230440.0 25100.0 0.45 0.8392 0.9727 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O06 mock treatment 1235360.0 25200.0 0.42 1236720.0 31400.0 0.56 0.6972 0.9895 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O07 mock treatment 1224720.0 14500.0 0.24 1233200.0 27800.0 0.5 0.5264 0.9446 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O08 mock treatment 1230680.0 20500.0 0.34 1213760.0 8400.0 0.15 0.3493 0.9325 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O09 mock treatment 1215040.0 4840.0 0.08 1199200.0 -6160.0 -0.11 -0.0213 -0.1548 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O10 mock treatment 1183920.0 -26300.0 -0.44 1174880.0 -30500.0 -0.55 -0.6994 -0.9939 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O11 mock treatment 1213880.0 3680.0 0.06 1196000.0 -9360.0 -0.17 -0.0758 -0.4219 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O12 mock treatment 1197320.0 -12900.0 -0.22 1207960.0 2600.0 0.05 -0.1194 -0.541 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O13 mock treatment 1216480.0 6280.0 0.11 1190600.0 -14800.0 -0.27 -0.1138 -0.3979 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O14 mock treatment 1190760.0 -19400.0 -0.33 1167920.0 -37400.0 -0.67 -0.7071 -0.9441 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O15 mock treatment 1197000.0 -13200.0 -0.22 1198440.0 -6920.0 -0.12 -0.2444 -0.9634 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O16 mock treatment 1164480.0 -45700.0 -0.77 1171240.0 -34100.0 -0.61 -0.9758 -0.9941 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O17 mock treatment 1190400.0 -19800.0 -0.33 1187400.0 -18000.0 -0.32 -0.4632 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O18 mock treatment 1185080.0 -25100.0 -0.42 1180680.0 -24700.0 -0.44 -0.6117 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O19 mock treatment 1177400.0 -32800.0 -0.55 1157720.0 -47600.0 -0.86 -0.9951 -0.9767 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O20 mock treatment 1155840.0 -54400.0 -0.91 1166560.0 -38800.0 -0.7 -1.1376 -0.9915 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O21 mock treatment 1177320.0 -32900.0 -0.55 1180720.0 -24600.0 -0.44 -0.7031 -0.9943 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O22 mock treatment 1165480.0 -44700.0 -0.75 1161640.0 -43700.0 -0.79 -1.0862 -0.9997 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O23 mock treatment 1161600.0 -48600.0 -0.81 1155600.0 -49800.0 -0.9 -1.2091 -0.9988 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base O24 mock treatment 1174760.0 -35400.0 -0.59 1187520.0 -17800.0 -0.32 -0.6467 -0.9586 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P01 mock treatment 1262960.0 52800.0 0.88 1244000.0 38600.0 0.7 1.1165 0.9931 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P02 mock treatment 1232600.0 22400.0 0.37 1236080.0 30700.0 0.55 0.6564 0.982 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P03 mock treatment 1242720.0 32500.0 0.54 1222280.0 16900.0 0.3 0.6003 0.9625 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P04 mock treatment 1227520.0 17300.0 0.29 1219400.0 14000.0 0.25 0.3838 0.9977 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P05 mock treatment 1223480.0 13300.0 0.22 1224640.0 19300.0 0.35 0.4027 0.9767 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P06 mock treatment 1205200.0 -5000.0 -0.08 1193360.0 -12000.0 -0.22 -0.2121 -0.9147 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P07 mock treatment 1221200.0 11000.0 0.18 1201480.0 -3880.0 -0.07 0.0807 0.4097 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P08 mock treatment 1193680.0 -16500.0 -0.28 1205080.0 -283.0 -0.01 -0.1991 -0.72 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P09 mock treatment 1211440.0 1240.0 0.02 1213200.0 7840.0 0.14 0.1145 0.8023 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P10 mock treatment 1201640.0 -8560.0 -0.14 1181520.0 -23800.0 -0.43 -0.4051 -0.8945 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P11 mock treatment 1195760.0 -14400.0 -0.24 1179440.0 -25900.0 -0.47 -0.5012 -0.953 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P12 mock treatment 1199240.0 -11000.0 -0.18 1198200.0 -7160.0 -0.13 -0.221 -0.9852 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P13 mock treatment 1191080.0 -19100.0 -0.32 1192680.0 -12700.0 -0.23 -0.3879 -0.9864 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P14 mock treatment 1170880.0 -39300.0 -0.66 1166800.0 -38600.0 -0.69 -0.9566 -0.9996 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P15 mock treatment 1179080.0 -31100.0 -0.52 1161360.0 -44000.0 -0.79 -0.9289 -0.9792 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P16 mock treatment 1170200.0 -40000.0 -0.67 1162520.0 -42800.0 -0.77 -1.0192 -0.9975 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P17 mock treatment 1177200.0 -33000.0 -0.55 1179040.0 -26300.0 -0.47 -0.7259 -0.9971 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P18 mock treatment 1168680.0 -41500.0 -0.69 1155160.0 -50200.0 -0.9 -1.1309 -0.9915 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P19 mock treatment 1166200.0 -44000.0 -0.74 1163240.0 -42100.0 -0.76 -1.0573 -0.9999 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P20 mock treatment 1160200.0 -50000.0 -0.84 1138000.0 -67400.0 -1.21 -1.4499 -0.9835 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P21 mock treatment 1138240.0 -72000.0 -1.2 1158360.0 -47000.0 -0.85 -1.4504 -0.9852 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P22 mock treatment 1156960.0 -53200.0 -0.89 1136600.0 -68800.0 -1.24 -1.5061 -0.9869 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P23 mock treatment 1163160.0 -47000.0 -0.79 1156600.0 -48800.0 -0.88 -1.1779 -0.9985 1057.0001 SteadyGlo(1057.0001) LuciferaseInhibition2006 1057.0001.Base P24 mock treatment 1178600.0 -31600.0 -0.53 1168880.0 -36500.0 -0.66 -0.8387 -0.9942